JP2025515926A5 - - Google Patents
Info
- Publication number
- JP2025515926A5 JP2025515926A5 JP2024568339A JP2024568339A JP2025515926A5 JP 2025515926 A5 JP2025515926 A5 JP 2025515926A5 JP 2024568339 A JP2024568339 A JP 2024568339A JP 2024568339 A JP2024568339 A JP 2024568339A JP 2025515926 A5 JP2025515926 A5 JP 2025515926A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- hydrogen
- pyridine
- formula
- membered ring
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202211018173.7A CN115353508B (zh) | 2022-08-24 | 2022-08-24 | 5-吡啶-1h-吲唑类化合物、药物组合物和应用 |
| CN202211018173.7 | 2022-08-24 | ||
| PCT/CN2022/133423 WO2024040768A1 (zh) | 2022-08-24 | 2022-11-22 | 5-吡啶-1h-吲唑类化合物、药物组合物和应用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025515926A JP2025515926A (ja) | 2025-05-20 |
| JP2025515926A5 true JP2025515926A5 (https=) | 2025-09-25 |
Family
ID=84003747
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024568339A Pending JP2025515926A (ja) | 2022-08-24 | 2022-11-22 | 5-ピリジン-1h-インダゾール系化合物、医薬組成物及び使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20260070889A1 (https=) |
| JP (1) | JP2025515926A (https=) |
| KR (1) | KR20250007528A (https=) |
| CN (1) | CN115353508B (https=) |
| AU (1) | AU2022475622A1 (https=) |
| CA (1) | CA3255205A1 (https=) |
| GB (1) | GB2632571A (https=) |
| WO (1) | WO2024040768A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN115353508B (zh) * | 2022-08-24 | 2023-07-21 | 中国药科大学 | 5-吡啶-1h-吲唑类化合物、药物组合物和应用 |
| CN115785071B (zh) * | 2023-01-09 | 2024-01-26 | 中国药科大学 | 3-乙炔基-5-(1h-1,2,3-三唑-4-基)-1h-吲唑类化合物及其应用 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030187026A1 (en) * | 2001-12-13 | 2003-10-02 | Qun Li | Kinase inhibitors |
| CN102595899A (zh) * | 2009-08-10 | 2012-07-18 | 埃皮瑟瑞克斯有限公司 | 作为wnt/b-联蛋白信号传导途径抑制剂的吲唑及其治疗用途 |
| CA2819373A1 (en) * | 2010-12-09 | 2012-06-14 | Amgen Inc. | Bicyclic compounds as pim inhibitors |
| PH12017500997A1 (en) * | 2012-04-04 | 2018-02-19 | Samumed Llc | Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof |
| WO2014137728A1 (en) * | 2013-03-04 | 2014-09-12 | Merck Sharp & Dohme Corp. | Compounds inhibiting leucine-rich repeat kinase enzyme activity |
| WO2014134772A1 (en) * | 2013-03-04 | 2014-09-12 | Merck Sharp & Dohme Corp. | Compounds inhibiting leucine-rich repeat kinase enzyme activity |
| CN106032359B (zh) * | 2015-03-09 | 2018-07-20 | 复旦大学 | 吲唑类化合物及其制备方法和用途 |
| MX380092B (es) * | 2015-11-06 | 2025-03-11 | Samumed Llc | Tratamiento de la osteoartritis. |
| CN105958990B (zh) * | 2016-05-24 | 2019-03-29 | 内蒙古包钢钢联股份有限公司 | 光电接近开关保护装置 |
| WO2019241540A1 (en) * | 2018-06-15 | 2019-12-19 | Samumed, Llc | Indazole containing macrocycles and therapeutic uses thereof |
| CA3118093A1 (en) * | 2018-09-28 | 2020-04-02 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Small molecule inhibitors of dyrk1/clk and uses thereof |
| US20230000842A1 (en) * | 2019-01-17 | 2023-01-05 | Samumed, Llc | Methods of treating cartilage disorders through inhibition of clk and dyrk |
| WO2022012058A1 (zh) * | 2020-07-16 | 2022-01-20 | 江苏凯迪恩医药科技有限公司 | 稠环化合物及其中间体、制备方法和应用 |
| CN115353508B (zh) * | 2022-08-24 | 2023-07-21 | 中国药科大学 | 5-吡啶-1h-吲唑类化合物、药物组合物和应用 |
-
2022
- 2022-08-24 CN CN202211018173.7A patent/CN115353508B/zh active Active
- 2022-11-22 AU AU2022475622A patent/AU2022475622A1/en active Pending
- 2022-11-22 KR KR1020247036196A patent/KR20250007528A/ko active Pending
- 2022-11-22 CA CA3255205A patent/CA3255205A1/en active Pending
- 2022-11-22 US US18/864,008 patent/US20260070889A1/en active Pending
- 2022-11-22 JP JP2024568339A patent/JP2025515926A/ja active Pending
- 2022-11-22 WO PCT/CN2022/133423 patent/WO2024040768A1/zh not_active Ceased
- 2022-11-22 GB GB2415076.5A patent/GB2632571A/en active Pending
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