JP2025514712A5 - - Google Patents
Info
- Publication number
- JP2025514712A5 JP2025514712A5 JP2024560880A JP2024560880A JP2025514712A5 JP 2025514712 A5 JP2025514712 A5 JP 2025514712A5 JP 2024560880 A JP2024560880 A JP 2024560880A JP 2024560880 A JP2024560880 A JP 2024560880A JP 2025514712 A5 JP2025514712 A5 JP 2025514712A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- carboxamide
- quinoline
- oxo
- pyridine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE2250473-2 | 2022-04-19 | ||
| SE2250473 | 2022-04-19 | ||
| PCT/US2023/019121 WO2023205251A1 (en) | 2022-04-19 | 2023-04-19 | Compounds active towards bromodomains |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025514712A JP2025514712A (ja) | 2025-05-09 |
| JP2025514712A5 true JP2025514712A5 (cg-RX-API-DMAC7.html) | 2026-04-27 |
Family
ID=86331094
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024560880A Pending JP2025514712A (ja) | 2022-04-19 | 2023-04-19 | ブロモドメインに対して活性な化合物 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20250382308A1 (cg-RX-API-DMAC7.html) |
| EP (1) | EP4511119B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2025514712A (cg-RX-API-DMAC7.html) |
| CN (1) | CN119365455A (cg-RX-API-DMAC7.html) |
| AU (1) | AU2023255396A1 (cg-RX-API-DMAC7.html) |
| CA (1) | CA3255932A1 (cg-RX-API-DMAC7.html) |
| MX (1) | MX2024013002A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2023205251A1 (cg-RX-API-DMAC7.html) |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101910182B (zh) | 2007-12-28 | 2013-07-17 | 田边三菱制药株式会社 | 抗癌剂 |
| GB0919431D0 (en) | 2009-11-05 | 2009-12-23 | Glaxosmithkline Llc | Novel compounds |
| AU2010317096B2 (en) | 2009-11-05 | 2015-03-26 | Glaxosmithkline Llc | Benzodiazepine bromodomain inhibitor |
| GB0919423D0 (en) | 2009-11-05 | 2009-12-23 | Glaxosmithkline Llc | Novel compounds |
| CA2779355C (en) | 2009-11-05 | 2018-01-16 | Glaxosmithkline Llc | Benzodiazepine bromodomain inhibitor |
| GB0919426D0 (en) | 2009-11-05 | 2009-12-23 | Glaxosmithkline Llc | Novel compounds |
| GB0919434D0 (en) | 2009-11-05 | 2009-12-23 | Glaxosmithkline Llc | Novel compounds |
| ES2606958T3 (es) | 2010-05-14 | 2017-03-28 | Dana-Farber Cancer Institute, Inc. | Compuestos de tienotriazolodiazepina para tratar una neoplasia |
| EP2585465B1 (en) | 2010-06-22 | 2014-11-12 | GlaxoSmithKline LLC | Benzotriazolodiazepine compounds inhibitors of bromodomains |
| AR084070A1 (es) | 2010-12-02 | 2013-04-17 | Constellation Pharmaceuticals Inc | Inhibidores del bromodominio y usos de los mismos |
| WO2013027168A1 (en) | 2011-08-22 | 2013-02-28 | Pfizer Inc. | Novel heterocyclic compounds as bromodomain inhibitors |
| HK1211033A1 (en) | 2012-12-20 | 2016-05-13 | Bayer Pharma Aktiengesellschaft | Bet-protein-inhibiting dihydroquinoxalinones |
| JP2016504990A (ja) | 2012-12-20 | 2016-02-18 | バイエル ファーマ アクチエンゲゼルシャフト | Ｂｅｔタンパク質抑制性ジヒドロピリドピラジノン |
| SG10201900631TA (en) * | 2014-08-01 | 2019-02-27 | Nuevolution As | Compounds active towards bromodomains |
| EP3563851B1 (en) * | 2016-12-27 | 2021-04-21 | FUJIFILM Corporation | Antitumor agent and bromodomain inhibitor |
-
2023
- 2023-04-19 CA CA3255932A patent/CA3255932A1/en active Pending
- 2023-04-19 JP JP2024560880A patent/JP2025514712A/ja active Pending
- 2023-04-19 US US18/860,589 patent/US20250382308A1/en active Pending
- 2023-04-19 EP EP23723033.9A patent/EP4511119B1/en active Active
- 2023-04-19 CN CN202380043848.XA patent/CN119365455A/zh active Pending
- 2023-04-19 AU AU2023255396A patent/AU2023255396A1/en active Pending
- 2023-04-19 WO PCT/US2023/019121 patent/WO2023205251A1/en not_active Ceased
-
2024
- 2024-10-21 MX MX2024013002A patent/MX2024013002A/es unknown
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