JP2025508473A5 - - Google Patents

Info

Publication number
JP2025508473A5
JP2025508473A5 JP2024550248A JP2024550248A JP2025508473A5 JP 2025508473 A5 JP2025508473 A5 JP 2025508473A5 JP 2024550248 A JP2024550248 A JP 2024550248A JP 2024550248 A JP2024550248 A JP 2024550248A JP 2025508473 A5 JP2025508473 A5 JP 2025508473A5
Authority
JP
Japan
Prior art keywords
carbonyl
amino
pyrazole
trifluoromethyl
piperazine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024550248A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508473A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/054499 external-priority patent/WO2023161316A1/en
Publication of JP2025508473A publication Critical patent/JP2025508473A/ja
Publication of JP2025508473A5 publication Critical patent/JP2025508473A5/ja
Pending legal-status Critical Current

Links

JP2024550248A 2022-02-25 2023-02-23 両性イオン性抗菌化合物 Pending JP2025508473A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22158739.7 2022-02-25
EP22158739 2022-02-25
PCT/EP2023/054499 WO2023161316A1 (en) 2022-02-25 2023-02-23 Zwitterionic antibacterial compounds

Publications (2)

Publication Number Publication Date
JP2025508473A JP2025508473A (ja) 2025-03-26
JP2025508473A5 true JP2025508473A5 (https=) 2026-03-03

Family

ID=80461664

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024550248A Pending JP2025508473A (ja) 2022-02-25 2023-02-23 両性イオン性抗菌化合物

Country Status (7)

Country Link
US (1) US20250179066A1 (https=)
EP (1) EP4482583B1 (https=)
JP (1) JP2025508473A (https=)
CN (1) CN118632842A (https=)
AR (1) AR128612A1 (https=)
TW (1) TW202402748A (https=)
WO (1) WO2023161316A1 (https=)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2016347456B2 (en) 2015-10-27 2018-12-13 F. Hoffmann-La Roche Ag Peptide macrocycles against acinetobacter baumannii
US11505573B2 (en) 2018-03-28 2022-11-22 Hoffmann-La Roche Inc. Peptide macrocycles against Acinetobacter baumannii
US11819532B2 (en) 2018-04-23 2023-11-21 Hoffmann-La Roche Inc. Peptide macrocycles against Acinetobacter baumannii
WO2020182648A1 (en) 2019-03-08 2020-09-17 F. Hoffmann-La Roche Ag Novel imidazole-pyrazole derivatives
CN114981259B (zh) * 2020-01-22 2024-06-18 豪夫迈·罗氏有限公司 新型杂环化合物

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