JP2025508402A5 - - Google Patents

Info

Publication number
JP2025508402A5
JP2025508402A5 JP2024548368A JP2024548368A JP2025508402A5 JP 2025508402 A5 JP2025508402 A5 JP 2025508402A5 JP 2024548368 A JP2024548368 A JP 2024548368A JP 2024548368 A JP2024548368 A JP 2024548368A JP 2025508402 A5 JP2025508402 A5 JP 2025508402A5
Authority
JP
Japan
Prior art keywords
weight
amino
pharmaceutically acceptable
phase
azaspiro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024548368A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508402A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2023/051532 external-priority patent/WO2023156979A1/en
Publication of JP2025508402A publication Critical patent/JP2025508402A/ja
Publication of JP2025508402A5 publication Critical patent/JP2025508402A5/ja
Pending legal-status Critical Current

Links

JP2024548368A 2022-02-21 2023-02-20 医薬製剤 Pending JP2025508402A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN202211009181 2022-02-21
IN202211009181 2022-02-21
PCT/IB2023/051532 WO2023156979A1 (en) 2022-02-21 2023-02-20 Pharmaceutical formulation

Publications (2)

Publication Number Publication Date
JP2025508402A JP2025508402A (ja) 2025-03-26
JP2025508402A5 true JP2025508402A5 (https=) 2026-02-20

Family

ID=85476156

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024548368A Pending JP2025508402A (ja) 2022-02-21 2023-02-20 医薬製剤

Country Status (11)

Country Link
US (1) US20250161223A1 (https=)
EP (1) EP4482471A1 (https=)
JP (1) JP2025508402A (https=)
KR (1) KR20240150600A (https=)
CN (1) CN118715005A (https=)
AU (1) AU2023221615A1 (https=)
CA (1) CA3251234A1 (https=)
IL (1) IL314206A (https=)
MX (1) MX2024009967A (https=)
TW (1) TW202342040A (https=)
WO (1) WO2023156979A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4580606A1 (en) * 2022-08-31 2025-07-09 Astrazeneca AB Pharmaceutical formulation

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3517B1 (ar) 2014-01-17 2020-07-05 Novartis Ag ان-ازاسبيرو الكان حلقي كبديل مركبات اريل-ان مغايرة وتركيبات لتثبيط نشاط shp2
CA3048340A1 (en) 2017-01-10 2018-07-19 Novartis Ag Pharmaceutical combination comprising an alk inhibitor and a shp2 inhibitor
CN112867718B (zh) 2018-09-29 2025-03-04 诺华股份有限公司 用于抑制shp2活性的化合物和组合物的制造
IL305106B2 (en) 2018-09-29 2025-08-01 Novartis Ag Process of manufacture of a compound for inhibiting the activity of shp2
MX2021009562A (es) 2019-02-12 2021-09-08 Novartis Ag Combinacion farmaceutica que comprende tno155 y un inhibidor de pd-1.
US20220152026A1 (en) 2019-02-12 2022-05-19 Novartis Ag Pharmaceutical combination comprising tno155 and a krasg12c inhibitor
EP3923941B1 (en) 2019-02-12 2025-12-03 Novartis AG Pharmaceutical combination comprising tno155 and ribociclib
EP4110338A1 (en) 2020-02-28 2023-01-04 Novartis AG A triple pharmaceutical combination comprising dabrafenib, an erk inhibitor and a shp2 inhibitor

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