JP2025504382A5 - - Google Patents

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Publication number
JP2025504382A5
JP2025504382A5 JP2024540933A JP2024540933A JP2025504382A5 JP 2025504382 A5 JP2025504382 A5 JP 2025504382A5 JP 2024540933 A JP2024540933 A JP 2024540933A JP 2024540933 A JP2024540933 A JP 2024540933A JP 2025504382 A5 JP2025504382 A5 JP 2025504382A5
Authority
JP
Japan
Prior art keywords
azacycloundecine
methoxytetrahydro
oxazepine
pyrazino
decahydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2024540933A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025504382A (ja
JP7714811B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/060944 external-priority patent/WO2023141536A1/en
Publication of JP2025504382A publication Critical patent/JP2025504382A/ja
Publication of JP2025504382A5 publication Critical patent/JP2025504382A5/ja
Priority to JP2025118767A priority Critical patent/JP2025160251A/ja
Application granted granted Critical
Publication of JP7714811B2 publication Critical patent/JP7714811B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2024540933A 2022-01-21 2023-01-20 1,3,4,7-テトラヒドロ-2H-ピロロ[3’,2’:5,6]ピリド[2,3-B][1,4]オキサアゼピンBcl-2阻害剤 Active JP7714811B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025118767A JP2025160251A (ja) 2022-01-21 2025-07-15 1,3,4,7-テトラヒドロ-2H-ピロロ[3’,2’:5,6]ピリド[2,3-B][1,4]オキサアゼピンBcl-2阻害剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263267018P 2022-01-21 2022-01-21
US63/267,018 2022-01-21
PCT/US2023/060944 WO2023141536A1 (en) 2022-01-21 2023-01-20 1,3,4,7-tetrahydro-2h-pyrrolo [3',2':5,6] pyrido[2,3-b] [1,4] oxazepine bc1-2 inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025118767A Division JP2025160251A (ja) 2022-01-21 2025-07-15 1,3,4,7-テトラヒドロ-2H-ピロロ[3’,2’:5,6]ピリド[2,3-B][1,4]オキサアゼピンBcl-2阻害剤

Publications (3)

Publication Number Publication Date
JP2025504382A JP2025504382A (ja) 2025-02-12
JP2025504382A5 true JP2025504382A5 (https=) 2025-06-09
JP7714811B2 JP7714811B2 (ja) 2025-07-29

Family

ID=85382827

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2024540933A Active JP7714811B2 (ja) 2022-01-21 2023-01-20 1,3,4,7-テトラヒドロ-2H-ピロロ[3’,2’:5,6]ピリド[2,3-B][1,4]オキサアゼピンBcl-2阻害剤
JP2025118767A Pending JP2025160251A (ja) 2022-01-21 2025-07-15 1,3,4,7-テトラヒドロ-2H-ピロロ[3’,2’:5,6]ピリド[2,3-B][1,4]オキサアゼピンBcl-2阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025118767A Pending JP2025160251A (ja) 2022-01-21 2025-07-15 1,3,4,7-テトラヒドロ-2H-ピロロ[3’,2’:5,6]ピリド[2,3-B][1,4]オキサアゼピンBcl-2阻害剤

Country Status (13)

Country Link
US (3) US11964990B2 (https=)
EP (1) EP4466273A1 (https=)
JP (2) JP7714811B2 (https=)
KR (1) KR20240136972A (https=)
CN (1) CN119053610A (https=)
AR (1) AR128310A1 (https=)
AU (1) AU2023210279A1 (https=)
CA (1) CA3242074A1 (https=)
CO (1) CO2024009334A2 (https=)
IL (1) IL312709A (https=)
MX (1) MX2024008840A (https=)
TW (1) TW202340210A (https=)
WO (1) WO2023141536A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202340210A (zh) * 2022-01-21 2023-10-16 美商艾伯維有限公司 1,3,4,7-四氫-2H-吡咯并[3',2':5,6]吡啶并[2,3-b][1,4]氮呯Bcl-2抑制劑
CN117820134A (zh) * 2024-01-10 2024-04-05 山东盛安贝新材料有限公司南京分公司 一种顺式-3-甲氧基环丁胺盐酸盐的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111511748B (zh) 2017-08-23 2023-05-02 广州麓鹏制药有限公司 Bcl-2抑制剂
US11903950B2 (en) 2018-08-22 2024-02-20 Newave Pharmaceutical Inc. BCL-2 inhibitors
WO2020140005A2 (en) 2018-12-29 2020-07-02 Newave Pharmaceutical Inc. Bcl-2 inhibitors
US20220372042A1 (en) 2019-10-03 2022-11-24 Newave Pharmaceutical Inc. Condensed heterocycles as bcl-2 inhibitors
WO2021083135A1 (en) 2019-10-28 2021-05-06 Beigene, Ltd. Bcl-2 INHIBITORS
WO2021133817A1 (en) 2019-12-27 2021-07-01 Guangzhou Lupeng Pharmaceutical Company Ltd. 1h-pyrrolo[2,3-b]pyridine derivatives as bcl-2 inhibitors for the treatment of neoplastic and autoimmune diseases
JP7849296B2 (ja) 2020-02-24 2026-04-21 グアンジョウ・ルペン・ファーマシューティカル・カンパニー・リミテッド Bcl2阻害剤を含むホットメルト押出し固体分散体
TW202340210A (zh) * 2022-01-21 2023-10-16 美商艾伯維有限公司 1,3,4,7-四氫-2H-吡咯并[3',2':5,6]吡啶并[2,3-b][1,4]氮呯Bcl-2抑制劑

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