JP2024539385A5 - - Google Patents

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Publication number
JP2024539385A5
JP2024539385A5 JP2024526649A JP2024526649A JP2024539385A5 JP 2024539385 A5 JP2024539385 A5 JP 2024539385A5 JP 2024526649 A JP2024526649 A JP 2024526649A JP 2024526649 A JP2024526649 A JP 2024526649A JP 2024539385 A5 JP2024539385 A5 JP 2024539385A5
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JP
Japan
Prior art keywords
compound
cancer
compounds
following
haloethylamine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024526649A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024539385A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2021/129077 external-priority patent/WO2023077452A1/zh
Publication of JP2024539385A publication Critical patent/JP2024539385A/ja
Publication of JP2024539385A5 publication Critical patent/JP2024539385A5/ja
Pending legal-status Critical Current

Links

JP2024526649A 2021-11-05 2021-11-05 Akr1c3活性化dnaアルキル化剤、およびその医学的応用 Pending JP2024539385A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/CN2021/129077 WO2023077452A1 (zh) 2021-11-05 2021-11-05 Akr1c3活化的dna烷化剂及其医药用途

Publications (2)

Publication Number Publication Date
JP2024539385A JP2024539385A (ja) 2024-10-28
JP2024539385A5 true JP2024539385A5 (cg-RX-API-DMAC7.html) 2024-11-13

Family

ID=86240506

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024526649A Pending JP2024539385A (ja) 2021-11-05 2021-11-05 Akr1c3活性化dnaアルキル化剤、およびその医学的応用

Country Status (7)

Country Link
US (1) US20260159536A1 (cg-RX-API-DMAC7.html)
EP (1) EP4428138A4 (cg-RX-API-DMAC7.html)
JP (1) JP2024539385A (cg-RX-API-DMAC7.html)
KR (1) KR20240110013A (cg-RX-API-DMAC7.html)
CN (1) CN118201940A (cg-RX-API-DMAC7.html)
TW (1) TW202320804A (cg-RX-API-DMAC7.html)
WO (1) WO2023077452A1 (cg-RX-API-DMAC7.html)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116120365A (zh) * 2021-11-12 2023-05-16 深圳艾欣达伟医药科技有限公司 一种氘代化合物及其制备方法和应用
CN121175032A (zh) 2023-05-11 2025-12-19 深圳艾欣达伟医药科技有限公司 一种注射液制剂、配伍药液及其制备方法
WO2025140580A1 (zh) * 2023-12-28 2025-07-03 深圳艾欣达伟医药科技有限公司 化合物晶型
WO2026130539A1 (zh) * 2024-12-20 2026-06-25 深圳艾欣达伟医药科技有限公司 Akr1c3酶活化的化合物与免疫检查点抑制剂联用治疗癌症、肿瘤患者的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016145092A1 (en) 2015-03-10 2016-09-15 Threshold Pharmaceuticals, Inc. Dna alkylating agents
WO2016161342A2 (en) * 2015-04-02 2016-10-06 Threshold Pharmaceuticals, Inc. Nitrobenzyl derivatives of anti-cancer agents
KR101985778B1 (ko) * 2015-11-16 2019-06-04 아센타위츠 파마슈티컬즈 리미티드 (r)- 및 (s)-1-(3-(3-n,n-다이메틸아미노카보닐)페녹시-4-나이트로페닐)-1-에틸-n,n'-비스(에틸렌)포스포르아미데이트, 조성물 및 이의 사용 방법 및 제조
CN118834240A (zh) * 2019-05-13 2024-10-25 深圳艾欣达伟医药科技有限公司 含氟化合物及抗癌医药用途
US20220387345A1 (en) * 2019-11-01 2022-12-08 Ascentawits Pharmaceuticals, Ltd. Anti-cancer compounds acting as non-pgp substrate
TWI837402B (zh) * 2019-12-20 2024-04-01 大陸商深圳艾欣達偉醫藥科技有限公司 含氟化合物、含氟化合物之製備方法及其抗癌醫藥用途

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