JP2024523313A - イソオキサゾリン殺害虫剤 - Google Patents

イソオキサゾリン殺害虫剤 Download PDF

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Publication number
JP2024523313A
JP2024523313A JP2023577341A JP2023577341A JP2024523313A JP 2024523313 A JP2024523313 A JP 2024523313A JP 2023577341 A JP2023577341 A JP 2023577341A JP 2023577341 A JP2023577341 A JP 2023577341A JP 2024523313 A JP2024523313 A JP 2024523313A
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JP
Japan
Prior art keywords
alkyl
cycloalkyl
group
halogen
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023577341A
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English (en)
Japanese (ja)
Other versions
JP2024523313A5 (enExample
Inventor
デュクレー，ピエール
ラジョー，デニーズ
トゥルバーグ，アンドレアス
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Elanco Animal Health GmbH
Original Assignee
Elanco Animal Health GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elanco Animal Health GmbH filed Critical Elanco Animal Health GmbH
Publication of JP2024523313A publication Critical patent/JP2024523313A/ja
Publication of JP2024523313A5 publication Critical patent/JP2024523313A5/ja
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/02—Acaricides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/04—Insecticides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Insects & Arthropods (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
JP2023577341A 2021-06-16 2022-06-15 イソオキサゾリン殺害虫剤 Pending JP2024523313A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163211478P 2021-06-16 2021-06-16
US63/211,478 2021-06-16
PCT/EP2022/066422 WO2022263573A1 (en) 2021-06-16 2022-06-15 Isoxazoline pesticides

Publications (2)

Publication Number Publication Date
JP2024523313A true JP2024523313A (ja) 2024-06-28
JP2024523313A5 JP2024523313A5 (enExample) 2025-06-17

Family

ID=82308417

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023577341A Pending JP2024523313A (ja) 2021-06-16 2022-06-15 イソオキサゾリン殺害虫剤

Country Status (10)

Country Link
US (1) US20240287005A1 (enExample)
EP (1) EP4355735A1 (enExample)
JP (1) JP2024523313A (enExample)
KR (1) KR20240044416A (enExample)
CN (1) CN117529473A (enExample)
AU (1) AU2022292908A1 (enExample)
BR (1) BR112023026357A2 (enExample)
CA (1) CA3223820A1 (enExample)
MX (1) MX2023015272A (enExample)
WO (1) WO2022263573A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12497370B2 (en) 2019-12-18 2025-12-16 Elanco Tiergesundheit Ag Isoxazoline derivatives
DK182016B1 (en) 2023-03-13 2025-05-28 Zoetis Services Llc Degradation of isoxazolines in ozonated sea water
WO2026006412A1 (en) * 2024-06-25 2026-01-02 Elanco Us Inc. Isooxazoline compounds as antiparasitic agents
WO2026006414A1 (en) * 2024-06-25 2026-01-02 Elanco Us Inc. Isoxazol-benzamide compounds as antiparasitic compounds

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005085216A1 (ja) * 2004-03-05 2005-09-15 Nissan Chemical Industries, Ltd. イソキサゾリン置換ベンズアミド化合物及び有害生物防除剤
JP2011517663A (ja) * 2008-03-14 2011-06-16 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト 殺虫性縮環式アリール化合物
JP2014508773A (ja) * 2011-03-10 2014-04-10 ゾエティス・エルエルシー 抗寄生虫薬としてのスピロ環式イソオキサゾリン誘導体
JP2023507117A (ja) * 2019-12-18 2023-02-21 エランコ・ティアゲゾンタイト・アーゲー 農薬としてのイソオキサゾリン誘導体

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI412322B (zh) 2005-12-30 2013-10-21 杜邦股份有限公司 控制無脊椎害蟲之異唑啉
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
BRPI0915665B1 (pt) 2008-07-09 2018-01-02 Basf Se Misturas pesticidas, métodos para proteger plantas do ataque ou infestação por insetos, acarídeos ou nematódeos, para controlar insetos, aracnídeos ou nematódeos, uso de uma mistura, e, composição pesticida ou parasiticida
AR074790A1 (es) 2008-12-19 2011-02-09 Novartis Ag Derivados de isooxazol sustituidos, composiciones farmaceuticas y para el control de parasitos que los comprenden y su uso en metodos para controlar parasitos en y sobre animales de sangre caliente.
AR088669A1 (es) 2011-11-21 2014-06-25 Lilly Co Eli Derivados de dihidrodibenzo[c][1,2]oxaborol y dihidroisoxazol utiles para el control de ectoparasitos
US20140343085A1 (en) 2011-11-29 2014-11-20 Novartis Ag Use of aryl derivatives for controlling ectoparasites

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005085216A1 (ja) * 2004-03-05 2005-09-15 Nissan Chemical Industries, Ltd. イソキサゾリン置換ベンズアミド化合物及び有害生物防除剤
JP2011517663A (ja) * 2008-03-14 2011-06-16 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト 殺虫性縮環式アリール化合物
JP2014508773A (ja) * 2011-03-10 2014-04-10 ゾエティス・エルエルシー 抗寄生虫薬としてのスピロ環式イソオキサゾリン誘導体
JP2023507117A (ja) * 2019-12-18 2023-02-21 エランコ・ティアゲゾンタイト・アーゲー 農薬としてのイソオキサゾリン誘導体

Also Published As

Publication number Publication date
BR112023026357A2 (pt) 2024-03-05
KR20240044416A (ko) 2024-04-04
EP4355735A1 (en) 2024-04-24
MX2023015272A (es) 2024-03-19
AU2022292908A1 (en) 2024-01-04
US20240287005A1 (en) 2024-08-29
CN117529473A (zh) 2024-02-06
CA3223820A1 (en) 2022-12-22
WO2022263573A1 (en) 2022-12-22

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