JP2024521818A5 - - Google Patents
Info
- Publication number
- JP2024521818A5 JP2024521818A5 JP2023573154A JP2023573154A JP2024521818A5 JP 2024521818 A5 JP2024521818 A5 JP 2024521818A5 JP 2023573154 A JP2023573154 A JP 2023573154A JP 2023573154 A JP2023573154 A JP 2023573154A JP 2024521818 A5 JP2024521818 A5 JP 2024521818A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- ethyl
- amino
- pyridazine
- dione
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163193831P | 2021-05-27 | 2021-05-27 | |
| US63/193,831 | 2021-05-27 | ||
| US202163226980P | 2021-07-29 | 2021-07-29 | |
| US63/226,980 | 2021-07-29 | ||
| PCT/US2022/031133 WO2022251497A1 (en) | 2021-05-27 | 2022-05-26 | Heterocyclic compounds and methods of use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024521818A JP2024521818A (ja) | 2024-06-04 |
| JP2024521818A5 true JP2024521818A5 (enExample) | 2025-06-03 |
Family
ID=84229207
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023573154A Pending JP2024521818A (ja) | 2021-05-27 | 2022-05-26 | ヘテロ環式化合物およびその使用方法 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20240279221A1 (enExample) |
| EP (1) | EP4346815A4 (enExample) |
| JP (1) | JP2024521818A (enExample) |
| KR (1) | KR20240013792A (enExample) |
| WO (1) | WO2022251497A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2023116902A1 (zh) * | 2021-12-23 | 2023-06-29 | 北京望实智慧科技有限公司 | Sos1抑制剂 |
| EP4463454A1 (en) | 2022-01-14 | 2024-11-20 | Jazz Pharmaceuticals Ireland Limited | Novel amine-substituted phthalazines and derivatives as sos1 inhibitors |
| EP4472974A4 (en) * | 2022-02-04 | 2026-03-25 | Schroedinger Inc | HETEROCYCLIC COMPOUNDS AND METHODS OF USE |
| KR20260059498A (ko) * | 2024-10-23 | 2026-04-30 | 제일약품주식회사 | 바이사이클릭 헤테로사이클릴 화합물의 신규 염 및 이의 결정형 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2649029A1 (en) * | 2006-04-20 | 2007-11-01 | Glaxo Group Limited | 2-substituted 4-benzylphthalazinone derivatives as histamine h1 and h3 antagonists |
| WO2008074803A2 (en) * | 2006-12-20 | 2008-06-26 | Glaxo Group Limited | 4-benzyl-l ( 2h) -phthalazinones as h1 receptor antagonists |
| ES2724578T3 (es) * | 2013-04-18 | 2019-09-12 | Shanghai Fochon Pharmaceutical Co Ltd | Ciertos inhibidores de proteína quinasas |
| EP3189049B1 (en) * | 2014-09-05 | 2024-03-20 | Genentech, Inc. | Phthalazine derivatives of formula (i) as pcaf and gcn5 inhibitors for use in the treatment of cancer |
| PL3728254T3 (pl) * | 2017-12-21 | 2023-06-12 | Boehringer Ingelheim International Gmbh | Benzyloaminopodstawione pirydopirymidynony i pochodne jako inhibitory sos1 |
| WO2023116902A1 (zh) * | 2021-12-23 | 2023-06-29 | 北京望实智慧科技有限公司 | Sos1抑制剂 |
| CN118574830A (zh) * | 2022-01-28 | 2024-08-30 | 中山优理生物医药有限公司 | 一种哒嗪并吡啶酮类化合物、其药物组合物及应用 |
-
2022
- 2022-05-26 KR KR1020237044751A patent/KR20240013792A/ko active Pending
- 2022-05-26 US US18/564,291 patent/US20240279221A1/en active Pending
- 2022-05-26 WO PCT/US2022/031133 patent/WO2022251497A1/en not_active Ceased
- 2022-05-26 EP EP22812161.2A patent/EP4346815A4/en not_active Withdrawn
- 2022-05-26 JP JP2023573154A patent/JP2024521818A/ja active Pending
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