JP2024516199A5 - - Google Patents

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Publication number
JP2024516199A5
JP2024516199A5 JP2023565369A JP2023565369A JP2024516199A5 JP 2024516199 A5 JP2024516199 A5 JP 2024516199A5 JP 2023565369 A JP2023565369 A JP 2023565369A JP 2023565369 A JP2023565369 A JP 2023565369A JP 2024516199 A5 JP2024516199 A5 JP 2024516199A5
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JP
Japan
Prior art keywords
formula
compound
reacting
hcl
item
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023565369A
Other languages
English (en)
Japanese (ja)
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JP2024516199A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/026208 external-priority patent/WO2022232060A1/en
Publication of JP2024516199A publication Critical patent/JP2024516199A/ja
Publication of JP2024516199A5 publication Critical patent/JP2024516199A5/ja
Pending legal-status Critical Current

Links

JP2023565369A 2021-04-26 2022-04-25 バルベナジンの合成方法 Pending JP2024516199A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163180043P 2021-04-26 2021-04-26
US63/180,043 2021-04-26
US202163286764P 2021-12-07 2021-12-07
US63/286,764 2021-12-07
PCT/US2022/026208 WO2022232060A1 (en) 2021-04-26 2022-04-25 Processes for the synthesis of valbenazine

Publications (2)

Publication Number Publication Date
JP2024516199A JP2024516199A (ja) 2024-04-12
JP2024516199A5 true JP2024516199A5 (enExample) 2025-05-08

Family

ID=81654703

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023565369A Pending JP2024516199A (ja) 2021-04-26 2022-04-25 バルベナジンの合成方法

Country Status (6)

Country Link
US (1) US20240239791A1 (enExample)
EP (1) EP4330255A1 (enExample)
JP (1) JP2024516199A (enExample)
CA (1) CA3215792A1 (enExample)
IL (1) IL307826A (enExample)
WO (1) WO2022232060A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2026050236A1 (en) 2024-08-27 2026-03-05 Neurocrine Biosciences, Inc. Muscarinic receptor agonist in combination with a vesicular monoamine transporter 2 inhibitor, for use in the treatment of a neurological or psychiatric disorder

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2081929T3 (da) 2006-11-08 2013-04-15 Neurocrine Biosciences Inc Substituerede 3-isobutyl-9,10-dimethoxy-1,3,4,6,7,11B-hexahydro-2H-pyrido[2,1-A]isoquinolin-2-ol-forbindelser og fremgangsmåder angående disse
IL284874B2 (en) 2015-10-30 2023-10-01 Neurocrine Biosciences Inc Valbenazine salts and polymorphs thereof
LT3394057T (lt) 2015-12-23 2022-06-27 Neurocrine Biosciences, Inc. Sintezės būdas, skirtas pagaminti (s)-(2r,3r,11br)-3-izobutil-9,10-dimetoksi-2,3,4,6,7,11b-heksahidro-1h-pirido[2,1-a]izochinolin-2-ilo 2-amino-3-metilbutanoato di(4-metilbenzensulfonatą)
RS66714B1 (sr) 2017-09-21 2025-05-30 Neurocrine Biosciences Inc Formulacija visoke doze valbenazina i sastavi, postupci i kompleti povezani sa njim
IL291221B2 (en) 2019-09-13 2026-05-01 Neurocrine Biosciences Inc Processes for the synthesis of valbenazine

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