JP2023541464A5 - - Google Patents

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Publication number
JP2023541464A5
JP2023541464A5 JP2023517408A JP2023517408A JP2023541464A5 JP 2023541464 A5 JP2023541464 A5 JP 2023541464A5 JP 2023517408 A JP2023517408 A JP 2023517408A JP 2023517408 A JP2023517408 A JP 2023517408A JP 2023541464 A5 JP2023541464 A5 JP 2023541464A5
Authority
JP
Japan
Prior art keywords
pyridine
amino
imidazo
methanone
fluorocyclopropyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023517408A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023541464A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/058378 external-priority patent/WO2022058890A1/en
Publication of JP2023541464A publication Critical patent/JP2023541464A/ja
Publication of JP2023541464A5 publication Critical patent/JP2023541464A5/ja
Pending legal-status Critical Current

Links

JP2023517408A 2020-09-15 2021-09-14 2-アミノ-3-カルボニルイミダゾピリジン及びピラゾロピリジン化合物 Pending JP2023541464A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063078372P 2020-09-15 2020-09-15
US63/078,372 2020-09-15
PCT/IB2021/058378 WO2022058890A1 (en) 2020-09-15 2021-09-14 2-amino-3-carbonyl imidazopyridine and pyrazolopyridine compounds

Publications (2)

Publication Number Publication Date
JP2023541464A JP2023541464A (ja) 2023-10-02
JP2023541464A5 true JP2023541464A5 (https=) 2024-02-07

Family

ID=80739409

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023517408A Pending JP2023541464A (ja) 2020-09-15 2021-09-14 2-アミノ-3-カルボニルイミダゾピリジン及びピラゾロピリジン化合物

Country Status (7)

Country Link
US (1) US11744824B2 (https=)
EP (1) EP4214207A4 (https=)
JP (1) JP2023541464A (https=)
KR (1) KR20230067669A (https=)
AU (1) AU2021342777A1 (https=)
CA (1) CA3192158A1 (https=)
WO (1) WO2022058890A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024140970A1 (zh) * 2022-12-30 2024-07-04 广州市联瑞制药有限公司 双环类化合物及其制备方法和应用
WO2025103406A1 (zh) * 2023-11-15 2025-05-22 南京明德新药研发有限公司 6并5杂芳基衍生物及其应用
TW202525805A (zh) * 2023-12-29 2025-07-01 大陸商廣州市聯瑞製藥有限公司 雙環類化合物及其製備方法和應用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4097483A (en) * 1974-11-01 1978-06-27 Kyorin Pharmaceutical Co., Ltd. Pyrazolo 1,5-a!pyridines
JPS5154583A (en) * 1974-11-01 1976-05-13 Kyorin Seiyaku Kk Shinkipirazoro * 1 55a * pirijinjudotaino seizoho
BRPI0610842A2 (pt) 2005-04-25 2010-07-27 Novartis Ag derivados de imidazo(1,2-a) piridina úteis como inibidores de peptìdeo desformilase (pdf)
PE20070978A1 (es) * 2006-02-14 2007-11-15 Novartis Ag COMPUESTOS HETEROCICLICOS COMO INHIBIDORES DE FOSFATIDILINOSITOL 3-QUINASAS (PI3Ks)
RU2008152776A (ru) 2006-06-06 2010-07-20 Эвиджен Инк. (Us) СОЕДИНЕНИЯ ЗАМЕЩЕННОГО ПИРАЗОЛО[1,5-a]ПИРИДИНА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ
JPWO2012102297A1 (ja) 2011-01-26 2014-06-30 杏林製薬株式会社 ピラゾロピリジン誘導体、またはその薬理学的に許容される塩
US20150158868A1 (en) 2013-12-06 2015-06-11 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
CN108084193A (zh) * 2017-12-19 2018-05-29 郭守东 一种brd4蛋白抑制剂
EP3849968B1 (en) * 2018-09-13 2022-12-21 Bristol-Myers Squibb Company 1h-indazole carboxamides as receptor-interacting protein kinase 1 inhibitors (ripk1)

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