JP2023538594A5 - - Google Patents

Info

Publication number
JP2023538594A5
JP2023538594A5 JP2023512073A JP2023512073A JP2023538594A5 JP 2023538594 A5 JP2023538594 A5 JP 2023538594A5 JP 2023512073 A JP2023512073 A JP 2023512073A JP 2023512073 A JP2023512073 A JP 2023512073A JP 2023538594 A5 JP2023538594 A5 JP 2023538594A5
Authority
JP
Japan
Prior art keywords
compound
hydrogen
formula
alkyl
diastereomer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023512073A
Other languages
English (en)
Japanese (ja)
Other versions
JP7851034B2 (ja
JP2023538594A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/046778 external-priority patent/WO2022040473A1/en
Publication of JP2023538594A publication Critical patent/JP2023538594A/ja
Publication of JP2023538594A5 publication Critical patent/JP2023538594A5/ja
Priority to JP2026062962A priority Critical patent/JP2026117077A/ja
Application granted granted Critical
Publication of JP7851034B2 publication Critical patent/JP7851034B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023512073A 2020-08-19 2021-08-19 選択されたプリンホスホルアミデートの立体選択的製造 Active JP7851034B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2026062962A JP2026117077A (ja) 2020-08-19 2026-04-07 選択されたプリンホスホルアミデートの立体選択的製造

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US202063067726P 2020-08-19 2020-08-19
US63/067,726 2020-08-19
US202063074302P 2020-09-03 2020-09-03
US63/074,302 2020-09-03
US202063094759P 2020-10-21 2020-10-21
US63/094,759 2020-10-21
US202063129306P 2020-12-22 2020-12-22
US63/129,306 2020-12-22
PCT/US2021/046778 WO2022040473A1 (en) 2020-08-19 2021-08-19 Stereoselective manufacture of selected purine phosphoramidates

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2026062962A Division JP2026117077A (ja) 2020-08-19 2026-04-07 選択されたプリンホスホルアミデートの立体選択的製造

Publications (3)

Publication Number Publication Date
JP2023538594A JP2023538594A (ja) 2023-09-08
JP2023538594A5 true JP2023538594A5 (cg-RX-API-DMAC7.html) 2024-08-27
JP7851034B2 JP7851034B2 (ja) 2026-04-24

Family

ID=80323295

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2023512073A Active JP7851034B2 (ja) 2020-08-19 2021-08-19 選択されたプリンホスホルアミデートの立体選択的製造
JP2026062962A Pending JP2026117077A (ja) 2020-08-19 2026-04-07 選択されたプリンホスホルアミデートの立体選択的製造

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2026062962A Pending JP2026117077A (ja) 2020-08-19 2026-04-07 選択されたプリンホスホルアミデートの立体選択的製造

Country Status (9)

Country Link
US (1) US20230331751A1 (cg-RX-API-DMAC7.html)
EP (1) EP4200309A4 (cg-RX-API-DMAC7.html)
JP (2) JP7851034B2 (cg-RX-API-DMAC7.html)
KR (1) KR20230053640A (cg-RX-API-DMAC7.html)
CN (1) CN115884977A (cg-RX-API-DMAC7.html)
AU (1) AU2021327241A1 (cg-RX-API-DMAC7.html)
CA (1) CA3173661A1 (cg-RX-API-DMAC7.html)
MX (1) MX2023002064A (cg-RX-API-DMAC7.html)
WO (1) WO2022040473A1 (cg-RX-API-DMAC7.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115477679A (zh) 2017-02-01 2022-12-16 阿堤亚制药公司 用于治疗丙型肝炎病毒的核苷酸半硫酸盐
US10874687B1 (en) 2020-02-27 2020-12-29 Atea Pharmaceuticals, Inc. Highly active compounds against COVID-19
AU2022291927A1 (en) 2021-06-17 2024-01-04 Atea Pharmaceuticals, Inc. Advantageous anti-hcv combination therapy
CN116462728B (zh) * 2021-12-15 2023-12-12 南京知和医药科技有限公司 一种抗病毒感染的嘌呤核苷衍生物及其药物组合物和用途
US12065404B2 (en) 2022-03-18 2024-08-20 Enveric Biosciences Canada Inc. C4-carboxylic acid-substituted tryptamine derivatives and methods of using
CN121628124B (zh) * 2026-02-05 2026-04-10 山东鲁源化工科技有限公司 一种高热稳定性聚磷酸酯阻燃剂及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2870169A1 (en) * 2012-07-03 2015-05-13 Bristol-Myers Squibb Company Process for preparing diastereomerically enriched phosphoramidate derivatives of nucleoside compounds for treatment of viral infections
FI3265102T3 (fi) * 2015-03-06 2025-10-31 Atea Pharmaceuticals Inc Beta-d-2'-deoksi-2'-alfa-fluori-2'-beta-c-substituoituja-2-modifioituja-n6-substituoituja puriininukleotideja hcv-hoitoa varten
PT3512863T (pt) * 2016-09-07 2022-03-09 Atea Pharmaceuticals Inc Nucleótidos de purina 2'-substituídos-n6-substituídos para tratamento de vírus de rna
US10874687B1 (en) * 2020-02-27 2020-12-29 Atea Pharmaceuticals, Inc. Highly active compounds against COVID-19
WO2021173713A1 (en) * 2020-02-27 2021-09-02 Atea Pharmaceuticals, Inc. Highly active compounds against covid-19

Similar Documents

Publication Publication Date Title
JP2024503855A (ja) アミノピリミジン系fak阻害剤化合物を合成する方法
ES2641761T3 (es) Procedimientos para preparar inhibidores JAK y compuestos intermedios relacionados
CN101541818A (zh) 4’-叠氮基胞苷衍生物的制备方法
JP7851034B2 (ja) 選択されたプリンホスホルアミデートの立体選択的製造
ES2738211T3 (es) Procedimiento mejorado de preparación de profármacos a base de duocarmicina
WO2018104953A1 (en) Improved process for the preparation of 7-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]butoxy}-2oxo-3,4-dihydro-2h-quinolin-1-yl)methyl dodecanoate
JP2017057215A (ja) 4−アミノ−5−ビフェニル−4−イル−2−ヒドロキシメチル−2−メチル−ペンタン酸化合物を調製する方法
EP3411359B1 (en) Methods of preparing hydroxylamine derivatives useful in the preparation of anti-infective agents
EP1904489B1 (en) Process for the synthesis of triazoles
KR20100102107A (ko) β-뉴클레오시드의 새로운 합성 방법
TWI887245B (zh) 用於產生二氮雜螺內醯胺化合物之方法及中間物
EP3515915B1 (en) Process for preparing beta-lactamase inhibitor hydroxylurea intermediates
WO2011156355A1 (en) Production method of phenyl guanidine salts and their intermediates
KR102899410B1 (ko) 가교형 뉴클레오시드 중간체의 결정 및 그의 제조 방법, 그리고 가교형 뉴클레오시드 아미다이트의 제조 방법
CN113166184B (zh) 用于制备环状二核苷酸的方法
JP2023517735A (ja) オキシム中間体及び関連化合物を介した3’nヌクレオシドの合成
CN102924454B (zh) 恩替卡韦的合成方法
ES2314449T3 (es) Derivados de peptidil cetona heterociclicos y procedimiento de preparacion.
WO2017134607A1 (en) A process for the preparation of phosphatidylinositol 3-kinase inhibitor
JP4181233B2 (ja) ピロリジン−2,4−ジオン誘導体の製法
HK40120549A (en) Processes and intermediates for producing diazaspiro lactam compounds
KR20250121547A (ko) 핵산 합성용 링커, 및 담체, 그리고 그들의 제조방법
JP2022035954A (ja) N-Boc-ラクタム誘導体及びその製造方法、並びに、環状アミン誘導体の製造方法
JP6040250B2 (ja) 2−[(2e)−2−フルオロ−2−(3−ピペリジニリデン)エチル]−1h−イソインドール−1,3(2h)−ジオンを調製するための改良された方法
JPWO2009107692A1 (ja) 2’−水酸基が保護されたリボヌクレオシド誘導体およびその製造方法