JP2023538090A5 - - Google Patents

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Publication number
JP2023538090A5
JP2023538090A5 JP2023512197A JP2023512197A JP2023538090A5 JP 2023538090 A5 JP2023538090 A5 JP 2023538090A5 JP 2023512197 A JP2023512197 A JP 2023512197A JP 2023512197 A JP2023512197 A JP 2023512197A JP 2023538090 A5 JP2023538090 A5 JP 2023538090A5
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JP
Japan
Prior art keywords
lymphoma
disease
pharmaceutically acceptable
stereoisomer
pharmaceutical composition
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Application number
JP2023512197A
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English (en)
Japanese (ja)
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JP2023538090A (ja
JP7669063B2 (ja
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Publication date
Priority claimed from CN202010836243.4A external-priority patent/CN114075190A/zh
Application filed filed Critical
Publication of JP2023538090A publication Critical patent/JP2023538090A/ja
Publication of JP2023538090A5 publication Critical patent/JP2023538090A5/ja
Application granted granted Critical
Publication of JP7669063B2 publication Critical patent/JP7669063B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023512197A 2020-08-20 2021-08-19 Btk阻害剤としての架橋二環式化合物 Active JP7669063B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN202010836243.4A CN114075190A (zh) 2020-08-20 2020-08-20 杂环类btk抑制剂
CN202010836243.4 2020-08-20
PCT/CN2021/113538 WO2022037650A1 (en) 2020-08-20 2021-08-19 Bridged bicyclic compounds as btk inhibitors

Publications (3)

Publication Number Publication Date
JP2023538090A JP2023538090A (ja) 2023-09-06
JP2023538090A5 true JP2023538090A5 (https=) 2024-08-26
JP7669063B2 JP7669063B2 (ja) 2025-04-28

Family

ID=80282666

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2023512198A Pending JP2023538091A (ja) 2020-08-20 2021-08-19 Btk阻害剤としての複素環式化合物
JP2023512197A Active JP7669063B2 (ja) 2020-08-20 2021-08-19 Btk阻害剤としての架橋二環式化合物

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2023512198A Pending JP2023538091A (ja) 2020-08-20 2021-08-19 Btk阻害剤としての複素環式化合物

Country Status (5)

Country Link
US (1) US20230192691A1 (https=)
EP (1) EP4200283A4 (https=)
JP (2) JP2023538091A (https=)
CN (2) CN114075190A (https=)
WO (2) WO2022037650A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021180107A1 (en) * 2020-03-12 2021-09-16 Fochon Pharmaceuticals, Ltd. Compounds useful as kinase inhibitors
CN114075190A (zh) * 2020-08-20 2022-02-22 北京诺诚健华医药科技有限公司 杂环类btk抑制剂
CN114573586B (zh) * 2020-11-28 2023-11-03 杭州和正医药有限公司 一种抑制布鲁顿酪氨酸激酶活性的多环化合物、药物组合物及其应用
CN114634512B (zh) * 2020-12-16 2023-11-14 江苏恒瑞医药股份有限公司 作为布鲁顿酪氨酸激酶抑制剂的化合物、其制备方法和医药应用
JP2025508964A (ja) * 2022-03-03 2025-04-10 深▲チェン▼市塔吉瑞生物医薬有限公司 シクロアルキルまたはヘテロシクリルで置換されたヘテロアリール化合物、並びにその組成物及び使用
WO2025007863A1 (zh) * 2023-07-03 2025-01-09 深圳市塔吉瑞生物医药有限公司 1H-吡唑并[4,3-c]吡啶化合物及其组合物及用途

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2548877A1 (en) * 2011-07-19 2013-01-23 MSD Oss B.V. 4-(5-Membered fused pyridinyl)benzamides as BTK-inhibitors
WO2015132799A2 (en) * 2014-02-03 2015-09-11 Cadila Healthcare Limited Novel heterocyclic compounds
GB201410430D0 (en) * 2014-06-11 2014-07-23 Redx Pharma Ltd Compounds
WO2016019237A2 (en) * 2014-07-31 2016-02-04 Pharmacyclics Llc Inhibitors of bruton's tyrosine kinase
WO2016106623A1 (en) * 2014-12-31 2016-07-07 Merck Sharp & Dohme Corp. Benzamide imidazopyrazine btk inhibitors
WO2016106624A1 (en) * 2014-12-31 2016-07-07 Merck Sharp & Dohme Corp. Tertiary alcohol imidazopyrazine btk inhibitors
WO2016106652A1 (en) * 2014-12-31 2016-07-07 Merck Sharp & Dohme Corp. Biarylether imidazopyrazine btk inhibitors
JP7337502B2 (ja) * 2015-09-16 2023-09-04 ロクソ オンコロジー, インコーポレイテッド がんの治療のためのbtk阻害剤としてのピラゾロピリミジン誘導体
AU2017383236B2 (en) * 2016-12-21 2022-02-10 Acerta Pharma B.V. Imidazopyrazine inhibitors of Bruton's tyrosine kinase
WO2020015735A1 (zh) * 2018-07-20 2020-01-23 正大天晴药业集团股份有限公司 布鲁顿酪氨酸激酶抑制剂
CN110964016B (zh) * 2018-09-29 2021-05-28 南京药捷安康生物科技有限公司 氨基降茨烷衍生物及其制备方法与应用
CN113365631B (zh) * 2019-01-18 2024-08-30 杭州邦顺制药有限公司 布鲁顿酪氨酸激酶抑制剂
WO2021180107A1 (en) * 2020-03-12 2021-09-16 Fochon Pharmaceuticals, Ltd. Compounds useful as kinase inhibitors
AU2020436612A1 (en) * 2020-03-16 2022-09-01 Flash Therapeutics, Llc Compounds for treating or inhibiting recurrence of acute myeloid leukemia
CN114075190A (zh) * 2020-08-20 2022-02-22 北京诺诚健华医药科技有限公司 杂环类btk抑制剂

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