JP2023519362A5 - - Google Patents

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Publication number
JP2023519362A5
JP2023519362A5 JP2022558347A JP2022558347A JP2023519362A5 JP 2023519362 A5 JP2023519362 A5 JP 2023519362A5 JP 2022558347 A JP2022558347 A JP 2022558347A JP 2022558347 A JP2022558347 A JP 2022558347A JP 2023519362 A5 JP2023519362 A5 JP 2023519362A5
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JP
Japan
Prior art keywords
methyl
amino
triazolo
pyrimidine
pyridyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022558347A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023519362A (ja
JP7675094B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/057806 external-priority patent/WO2021191378A1/en
Publication of JP2023519362A publication Critical patent/JP2023519362A/ja
Publication of JP2023519362A5 publication Critical patent/JP2023519362A5/ja
Application granted granted Critical
Publication of JP7675094B2 publication Critical patent/JP7675094B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022558347A 2020-03-26 2021-03-25 トリアゾロン化合物 Active JP7675094B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062994908P 2020-03-26 2020-03-26
US62/994,908 2020-03-26
PCT/EP2021/057806 WO2021191378A1 (en) 2020-03-26 2021-03-25 5-amino-8-(4-pyridyl)-[1,2,4]triazolo[4,3-c]pyrimidin-3-one compounds for use against cancer

Publications (3)

Publication Number Publication Date
JP2023519362A JP2023519362A (ja) 2023-05-10
JP2023519362A5 true JP2023519362A5 (https=) 2024-04-01
JP7675094B2 JP7675094B2 (ja) 2025-05-12

Family

ID=75339740

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022558347A Active JP7675094B2 (ja) 2020-03-26 2021-03-25 トリアゾロン化合物

Country Status (8)

Country Link
US (1) US20230271964A1 (https=)
EP (1) EP4126872A1 (https=)
JP (1) JP7675094B2 (https=)
KR (1) KR20230049579A (https=)
CN (1) CN115867282B (https=)
AU (1) AU2021240344A1 (https=)
CA (1) CA3176944A1 (https=)
WO (1) WO2021191378A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3243621A1 (en) * 2022-02-01 2023-08-10 Eli Lilly And Company METHODS FOR PREPARING SELECTIVE ESTROGEN RECEPTOR DEGRADING AGENTS
JP2025512384A (ja) 2022-04-13 2025-04-17 ギリアード サイエンシーズ, インコーポレイテッド Trop-2発現がんを治療するための併用療法
WO2025137640A1 (en) 2023-12-22 2025-06-26 Gilead Sciences, Inc. Azaspiro wrn inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7452892B2 (en) 2005-06-17 2008-11-18 Bristol-Myers Squibb Company Triazolopyrimidine cannabinoid receptor 1 antagonists
ATE457988T1 (de) 2006-06-26 2010-03-15 Schering Corp A2a-adenosin-rezeptor-antagonisten
JP2011513417A (ja) 2008-03-04 2011-04-28 シェーリング コーポレイション アデノシンA2a受容体アンタゴニストとして使用するための1,2,4−トリアゾロ[4,3−c]ピリミジン−3−オンおよびピラゾロ[4,3−e]−1,2,4−トリアゾロ[4,3−c]ピリミジン−3−オン化合物
AU2011306358B2 (en) 2010-09-24 2014-08-14 Impetis Biosciences Ltd. Fused tricyclic compounds as adenosine receptor antagonist
EP3277689B1 (en) 2015-04-03 2019-09-04 Incyte Corporation Heterocyclic compounds as lsd1 inhibitors
AU2018233367B2 (en) 2017-03-16 2021-08-12 Jiangsu Hengrui Medicine Co., Ltd. Heteroaryl[4,3-c]pyrimidine-5-amine derivative, preparation method therefor, and medical uses thereof

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