JP2023519361A5 - - Google Patents

Info

Publication number
JP2023519361A5
JP2023519361A5 JP2022558345A JP2022558345A JP2023519361A5 JP 2023519361 A5 JP2023519361 A5 JP 2023519361A5 JP 2022558345 A JP2022558345 A JP 2022558345A JP 2022558345 A JP2022558345 A JP 2022558345A JP 2023519361 A5 JP2023519361 A5 JP 2023519361A5
Authority
JP
Japan
Prior art keywords
pyridyl
amino
triazolo
pyrimidine
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022558345A
Other languages
English (en)
Japanese (ja)
Other versions
JP7774573B2 (ja
JP2023519361A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/057807 external-priority patent/WO2021191379A1/en
Publication of JP2023519361A publication Critical patent/JP2023519361A/ja
Publication of JP2023519361A5 publication Critical patent/JP2023519361A5/ja
Application granted granted Critical
Publication of JP7774573B2 publication Critical patent/JP7774573B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022558345A 2020-03-26 2021-03-25 トリアゾロン化合物 Active JP7774573B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062994970P 2020-03-26 2020-03-26
US62/994,970 2020-03-26
PCT/EP2021/057807 WO2021191379A1 (en) 2020-03-26 2021-03-25 5-amino-8-(4-pyridyl)-[1,2,4]triazolo[4,3-c]pyrimidin-3-one compounds for use against cancer

Publications (3)

Publication Number Publication Date
JP2023519361A JP2023519361A (ja) 2023-05-10
JP2023519361A5 true JP2023519361A5 (https=) 2024-04-01
JP7774573B2 JP7774573B2 (ja) 2025-11-21

Family

ID=75339741

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022558345A Active JP7774573B2 (ja) 2020-03-26 2021-03-25 トリアゾロン化合物

Country Status (8)

Country Link
US (1) US12528815B2 (https=)
EP (1) EP4126873A1 (https=)
JP (1) JP7774573B2 (https=)
KR (1) KR20230051118A (https=)
CN (1) CN115867280B (https=)
AU (1) AU2021243725A1 (https=)
CA (1) CA3177056A1 (https=)
WO (1) WO2021191379A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2025512384A (ja) 2022-04-13 2025-04-17 ギリアード サイエンシーズ, インコーポレイテッド Trop-2発現がんを治療するための併用療法
WO2025137640A1 (en) 2023-12-22 2025-06-26 Gilead Sciences, Inc. Azaspiro wrn inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7452892B2 (en) * 2005-06-17 2008-11-18 Bristol-Myers Squibb Company Triazolopyrimidine cannabinoid receptor 1 antagonists
ATE457988T1 (de) 2006-06-26 2010-03-15 Schering Corp A2a-adenosin-rezeptor-antagonisten
JP2011513417A (ja) * 2008-03-04 2011-04-28 シェーリング コーポレイション アデノシンA2a受容体アンタゴニストとして使用するための1,2,4−トリアゾロ[4,3−c]ピリミジン−3−オンおよびピラゾロ[4,3−e]−1,2,4−トリアゾロ[4,3−c]ピリミジン−3−オン化合物
AU2011306358B2 (en) 2010-09-24 2014-08-14 Impetis Biosciences Ltd. Fused tricyclic compounds as adenosine receptor antagonist
EP3277689B1 (en) 2015-04-03 2019-09-04 Incyte Corporation Heterocyclic compounds as lsd1 inhibitors
AU2018233367B2 (en) 2017-03-16 2021-08-12 Jiangsu Hengrui Medicine Co., Ltd. Heteroaryl[4,3-c]pyrimidine-5-amine derivative, preparation method therefor, and medical uses thereof

Similar Documents

Publication Publication Date Title
TWI868441B (zh) 非環氧氮呯化合物及其用途
JP2015511245A5 (https=)
ES2377849T3 (es) Compuestos amino-heterocíclicos
EP3630770B1 (en) Pyrazolo[3,4-b]pyrazine derivatives as shp2 phosphatase inhibitors
ES2420860T3 (es) Compuestos amino-heterocíclicos usados como inhibidores de la PDE9
JP2022500402A5 (https=)
RU2473549C2 (ru) Пиримидиновые соединения, композиции и способы применения
JP2025535367A (ja) 6-アザ部分を含むオキサゼピン化合物およびその使用
HRP20240994T1 (hr) Spoj inhibitora jak i njegova uporaba
JP2016538316A5 (https=)
JP2014506929A5 (https=)
RU2008110915A (ru) Новые диазаспироалканы и их применение для лечения заболеваний, опосредованных ccr8
JP2016500073A5 (https=)
JP2024123079A (ja) トリアゾロ-ピリミジン化合物およびそれらの使用
EP2920177A1 (en) Compounds and compositions for the treatment of parasitic diseases
JP2013522354A5 (https=)
RU2013120966A (ru) ФУРО[3,2-d]ПИРИМИДИНОВЫЕ СОЕДИНЕНИЯ
RU2017121278A (ru) Триазоло-пиразинильные производные, применимые в качестве растворимых активаторов гуанилатциклазы
JP2015522002A5 (https=)
JP2013523884A5 (https=)
JP2016515098A5 (https=)
TW201542520A (zh) 炔基醇及其使用方法
JP2016537384A5 (https=)
JP2017518326A5 (https=)
JP2023519361A5 (https=)