JP2023518529A5 - - Google Patents

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Publication number
JP2023518529A5
JP2023518529A5 JP2022558331A JP2022558331A JP2023518529A5 JP 2023518529 A5 JP2023518529 A5 JP 2023518529A5 JP 2022558331 A JP2022558331 A JP 2022558331A JP 2022558331 A JP2022558331 A JP 2022558331A JP 2023518529 A5 JP2023518529 A5 JP 2023518529A5
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JP
Japan
Prior art keywords
optionally substituted
compound
solid dispersion
alkyl
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022558331A
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English (en)
Japanese (ja)
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JP2023518529A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CA2021/050385 external-priority patent/WO2021189141A1/en
Publication of JP2023518529A publication Critical patent/JP2023518529A/ja
Publication of JP2023518529A5 publication Critical patent/JP2023518529A5/ja
Pending legal-status Critical Current

Links

JP2022558331A 2020-03-24 2021-03-24 非晶質3,4-ジフェニル-4,5-ジヒドロ-1h-ピラゾール誘導体の固体分散体、それを含む組成物及びカンナビノイドcb1受容体阻害剤としてのその使用 Pending JP2023518529A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062993775P 2020-03-24 2020-03-24
US62/993,775 2020-03-24
PCT/CA2021/050385 WO2021189141A1 (en) 2020-03-24 2021-03-24 Solid dispersions of amorphous 3, 4-diphenyl-4, 5-dihydro- 1h-pyrazole derivatives, compositions comprising them and uses thereof as cannabinoid cb1 receptor inhibitors

Publications (2)

Publication Number Publication Date
JP2023518529A JP2023518529A (ja) 2023-05-01
JP2023518529A5 true JP2023518529A5 (https=) 2024-02-27

Family

ID=77890104

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022558331A Pending JP2023518529A (ja) 2020-03-24 2021-03-24 非晶質3,4-ジフェニル-4,5-ジヒドロ-1h-ピラゾール誘導体の固体分散体、それを含む組成物及びカンナビノイドcb1受容体阻害剤としてのその使用

Country Status (9)

Country Link
US (1) US20230174493A1 (https=)
EP (1) EP4126822A4 (https=)
JP (1) JP2023518529A (https=)
KR (1) KR20220156930A (https=)
CN (1) CN115335361A (https=)
AU (1) AU2021242808A1 (https=)
CA (1) CA3169753A1 (https=)
MX (1) MX2022011899A (https=)
WO (1) WO2021189141A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4482490A4 (en) * 2022-02-24 2025-08-20 Novo Nordisk As METHODS OF TREATING SUBJECTS WITH HYPERTRIGLYCERIDEMIA, ABDOMINAL OBESITY AND/OR ALTERED GLUCOSE
WO2025040089A1 (zh) * 2023-08-21 2025-02-27 德睿智药(苏州)新药研发有限公司 用于选择性调节大麻素cb1功能的新型杂环类化合物
WO2025103493A1 (zh) * 2023-11-16 2025-05-22 西藏海思科制药有限公司 一种大麻素受体1拮抗剂及其应用
WO2025257151A1 (en) 2024-06-10 2025-12-18 Institut National de la Santé et de la Recherche Médicale Methods and pharmaceutical composition for treating ciliopathies

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2083799A1 (en) * 2006-10-20 2009-08-05 Solvay Pharmaceuticals B.V. Micellar nanoparticles of chemical substances
CN104884057B (zh) * 2012-11-13 2019-08-20 美国政府(由卫生和人类服务部的部长所代表) 大麻素受体介导的化合物
CA2955510C (en) * 2014-07-25 2018-09-04 Allen-Vanguard Corporation System and method for ultra wideband radio frequency scanning and signal generation
WO2016196646A1 (en) * 2015-06-04 2016-12-08 The United States Of America, As Represented By The Secretary, Departmet Of Health & Human Services Cannabinoid receptor mediating compounds
US12286405B2 (en) * 2019-05-17 2025-04-29 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Scalable synthesis of dual-target inhibitor of cannabinoid-1 receptor and inducible nitric oxide synthase

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