JP2023514280A5 - - Google Patents

Info

Publication number
JP2023514280A5
JP2023514280A5 JP2022549325A JP2022549325A JP2023514280A5 JP 2023514280 A5 JP2023514280 A5 JP 2023514280A5 JP 2022549325 A JP2022549325 A JP 2022549325A JP 2022549325 A JP2022549325 A JP 2022549325A JP 2023514280 A5 JP2023514280 A5 JP 2023514280A5
Authority
JP
Japan
Application number
JP2022549325A
Other languages
Japanese (ja)
Other versions
JPWO2021168313A5 (https=
JP2023514280A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/018863 external-priority patent/WO2021168313A1/en
Publication of JP2023514280A publication Critical patent/JP2023514280A/ja
Publication of JP2023514280A5 publication Critical patent/JP2023514280A5/ja
Publication of JPWO2021168313A5 publication Critical patent/JPWO2021168313A5/ja
Pending legal-status Critical Current

Links

JP2022549325A 2020-02-19 2021-02-19 setd2阻害剤、および関連する方法と使用(併用療法を含む) Pending JP2023514280A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062978692P 2020-02-19 2020-02-19
US62/978,692 2020-02-19
PCT/US2021/018863 WO2021168313A1 (en) 2020-02-19 2021-02-19 Setd2 inhibitors and related methods and uses, including combination therapies

Publications (3)

Publication Number Publication Date
JP2023514280A JP2023514280A (ja) 2023-04-05
JP2023514280A5 true JP2023514280A5 (https=) 2024-02-27
JPWO2021168313A5 JPWO2021168313A5 (https=) 2024-02-27

Family

ID=77391740

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022549325A Pending JP2023514280A (ja) 2020-02-19 2021-02-19 setd2阻害剤、および関連する方法と使用(併用療法を含む)

Country Status (11)

Country Link
US (1) US20230133671A1 (https=)
EP (1) EP4107157A4 (https=)
JP (1) JP2023514280A (https=)
KR (1) KR20220143116A (https=)
CN (2) CN121695288A (https=)
AU (1) AU2021224855A1 (https=)
BR (1) BR112022016573A2 (https=)
CA (1) CA3168069A1 (https=)
IL (1) IL295654A (https=)
MX (1) MX2022010171A (https=)
WO (1) WO2021168313A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2020530844A (ja) 2017-08-14 2020-10-29 エピザイム,インコーポレイティド Setd2を阻害することにより癌を処置する方法
CN111093660A (zh) * 2017-09-05 2020-05-01 Epizyme股份有限公司 用于治疗癌症的组合疗法
CN112585119A (zh) 2018-08-14 2021-03-30 Epizyme股份有限公司 经取代的吲哚及其使用方法
US20240299352A1 (en) * 2021-06-09 2024-09-12 Epizyme, Inc. Combination therapies with setd2 inhibitors
JP2024539726A (ja) * 2021-11-01 2024-10-29 エピザイム,インコーポレイティド N-((1r,3s)-3-(4-アセチルピペラジン-1-イル)シクロヘキシル)-4-フルオロ-7-メチル-1h-インドール-2-カルボキサミドの結晶形態

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4595766A (en) * 1984-10-26 1986-06-17 Ciba-Geigy Corporation Process for the preparation of an indoline carboxylic acid
US20100035862A1 (en) * 2008-06-25 2010-02-11 Abbott Laboratories Novel aza-cyclic indole-2-carboxamides and methods of use thereof
NZ725860A (en) * 2014-04-04 2019-08-30 Iomet Pharma Ltd Indole derivatives for use in medicine
WO2016040505A1 (en) * 2014-09-10 2016-03-17 Epizyme, Inc. Smyd inhibitors
CN112585119A (zh) * 2018-08-14 2021-03-30 Epizyme股份有限公司 经取代的吲哚及其使用方法
SG11202105325QA (en) * 2018-11-30 2021-06-29 Epizyme Inc Methods of treating whsc1-overexpressing cancers by inhibiting setd2

Similar Documents

Publication Publication Date Title
BR112023005462A2 (https=)
BR112023012656A2 (https=)
BR112021014123A2 (https=)
BR112023009656A2 (https=)
BR112022009896A2 (https=)
JP2023514280A5 (https=)
JP2023515576A5 (https=)
BR112021017747A2 (https=)
BR112022024743A2 (https=)
BR112022026905A2 (https=)
BR112023011738A2 (https=)
BR112023004146A2 (https=)
BR102021018859A2 (https=)
BR102021015500A2 (https=)
BR112023016292A2 (https=)
BR112023011610A2 (https=)
BR112023011539A2 (https=)
BR112023008976A2 (https=)
BR102021020147A2 (https=)
BR102021018926A2 (https=)
BR102021018167A2 (https=)
BR102021017576A2 (https=)
BR102021016837A2 (https=)
BR102021016551A2 (https=)
BR102021016375A2 (https=)