JP2023510212A5 - - Google Patents
Info
- Publication number
- JP2023510212A5 JP2023510212A5 JP2022540849A JP2022540849A JP2023510212A5 JP 2023510212 A5 JP2023510212 A5 JP 2023510212A5 JP 2022540849 A JP2022540849 A JP 2022540849A JP 2022540849 A JP2022540849 A JP 2022540849A JP 2023510212 A5 JP2023510212 A5 JP 2023510212A5
- Authority
- JP
- Japan
- Prior art keywords
- imidazo
- pyran
- tetrahydro
- phenoxyphenyl
- fluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2020070034 | 2020-01-02 | ||
| CNPCT/CN2020/070034 | 2020-01-02 | ||
| CNPCT/CN2020/134601 | 2020-12-08 | ||
| CN2020134601 | 2020-12-08 | ||
| PCT/CN2020/140517 WO2021136219A1 (en) | 2020-01-02 | 2020-12-29 | Btk inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023510212A JP2023510212A (ja) | 2023-03-13 |
| JP2023510212A5 true JP2023510212A5 (enExample) | 2024-01-10 |
| JP7649311B2 JP7649311B2 (ja) | 2025-03-19 |
Family
ID=76685855
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022540849A Active JP7649311B2 (ja) | 2020-01-02 | 2020-12-29 | Ｂｔｋ阻害薬 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US12624039B2 (enExample) |
| EP (1) | EP4087845A4 (enExample) |
| JP (1) | JP7649311B2 (enExample) |
| CN (2) | CN114945574B (enExample) |
| AU (1) | AU2020419422B2 (enExample) |
| BR (1) | BR112022013227A2 (enExample) |
| CA (1) | CA3163365A1 (enExample) |
| MX (1) | MX2022008148A (enExample) |
| TW (1) | TWI875911B (enExample) |
| WO (1) | WO2021136219A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2020436612A1 (en) * | 2020-03-16 | 2022-09-01 | Flash Therapeutics, Llc | Compounds for treating or inhibiting recurrence of acute myeloid leukemia |
| CN113943294A (zh) * | 2020-07-15 | 2022-01-18 | 成都海博为药业有限公司 | 一种作为btk抑制剂的化合物及其制备方法与用途 |
| CN115851606A (zh) * | 2022-12-19 | 2023-03-28 | 北京爱思益普生物科技股份有限公司 | Btk突变细胞株及其构建方法和应用 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008054827A2 (en) | 2006-11-03 | 2008-05-08 | Pharmacyclics, Inc. | Bruton's tyrosine kinase activity probe and method of using |
| ES2396613T3 (es) * | 2008-05-19 | 2013-02-22 | OSI Pharmaceuticals, LLC | Imidazopirazinas e imidazotriazinas sustituidas |
| US8940725B2 (en) | 2010-05-31 | 2015-01-27 | Ono Pharmaceutical Co., Ltd. | Purinone derivative |
| WO2012158795A1 (en) | 2011-05-17 | 2012-11-22 | Principia Biopharma Inc. | Pyrazolopyrimidine derivatives as tyrosine kinase inhibitors |
| CA2833867A1 (en) | 2013-11-21 | 2015-05-21 | Pharmascience Inc. | Protein kinase inhibitors |
| WO2016020901A1 (en) * | 2014-08-07 | 2016-02-11 | Acerta Pharma B.V. | Methods of treating cancers, immune and autoimmune diseases, and inflammatory diseases based on btk occupancy and btk resynthesis rate |
| WO2016106652A1 (en) * | 2014-12-31 | 2016-07-07 | Merck Sharp & Dohme Corp. | Biarylether imidazopyrazine btk inhibitors |
| US20180305350A1 (en) * | 2015-06-24 | 2018-10-25 | Principia Biopharma Inc. | Tyrosine kinase inhibitors |
| CN114605327B (zh) | 2015-12-16 | 2025-03-11 | 洛克索肿瘤学股份有限公司 | 可用作激酶抑制剂的化合物 |
| AU2015417922B2 (en) | 2015-12-23 | 2018-12-20 | Arqule, Inc. | Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereof |
| US10640512B2 (en) * | 2016-06-30 | 2020-05-05 | Hangzhou Sanyintai Pharmaceutical Technology Co., Ltd. | Imidazopyrazinamine phenyl derivative and use thereof |
| AU2017315343A1 (en) | 2016-08-24 | 2019-02-28 | Arqule, Inc. | Amino-pyrrolopyrimidinone compounds and methods of use thereof |
| CN111454268B (zh) | 2019-01-18 | 2023-09-08 | 明慧医药（上海）有限公司 | 作为布鲁顿酪氨酸激酶抑制剂的环状分子 |
| CA3126940A1 (en) | 2019-01-18 | 2020-07-23 | Xibin Liao | Bruton's tyrosine kinase inhibitors |
| CN113943294A (zh) | 2020-07-15 | 2022-01-18 | 成都海博为药业有限公司 | 一种作为btk抑制剂的化合物及其制备方法与用途 |
-
2020
- 2020-12-29 MX MX2022008148A patent/MX2022008148A/es unknown
- 2020-12-29 WO PCT/CN2020/140517 patent/WO2021136219A1/en not_active Ceased
- 2020-12-29 CN CN202080091669.XA patent/CN114945574B/zh active Active
- 2020-12-29 AU AU2020419422A patent/AU2020419422B2/en active Active
- 2020-12-29 EP EP20910897.6A patent/EP4087845A4/en active Pending
- 2020-12-29 BR BR112022013227A patent/BR112022013227A2/pt unknown
- 2020-12-29 TW TW109146658A patent/TWI875911B/zh active
- 2020-12-29 US US17/790,721 patent/US12624039B2/en active Active
- 2020-12-29 CA CA3163365A patent/CA3163365A1/en active Pending
- 2020-12-29 CN CN202510077904.2A patent/CN120118089A/zh active Pending
- 2020-12-29 JP JP2022540849A patent/JP7649311B2/ja active Active
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