JP2023503898A5 - - Google Patents

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Publication number
JP2023503898A5
JP2023503898A5 JP2022529452A JP2022529452A JP2023503898A5 JP 2023503898 A5 JP2023503898 A5 JP 2023503898A5 JP 2022529452 A JP2022529452 A JP 2022529452A JP 2022529452 A JP2022529452 A JP 2022529452A JP 2023503898 A5 JP2023503898 A5 JP 2023503898A5
Authority
JP
Japan
Prior art keywords
alkyl
optionally substituted
group
aryl
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022529452A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023503898A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2020/061065 external-priority patent/WO2021100029A2/en
Publication of JP2023503898A publication Critical patent/JP2023503898A/ja
Publication of JP2023503898A5 publication Critical patent/JP2023503898A5/ja
Priority to JP2025202023A priority Critical patent/JP2026032104A/ja
Pending legal-status Critical Current

Links

JP2022529452A 2019-11-24 2020-11-24 フルベストラントのプロドラッグ Pending JP2023503898A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025202023A JP2026032104A (ja) 2019-11-24 2025-11-21 フルベストラントのプロドラッグ

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN201921047986 2019-11-24
IN201921047986 2019-11-24
IN202021029084 2020-07-08
IN202021029084 2020-07-08
PCT/IB2020/061065 WO2021100029A2 (en) 2019-11-24 2020-11-24 Prodrugs of fulvestrant

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025202023A Division JP2026032104A (ja) 2019-11-24 2025-11-21 フルベストラントのプロドラッグ

Publications (2)

Publication Number Publication Date
JP2023503898A JP2023503898A (ja) 2023-02-01
JP2023503898A5 true JP2023503898A5 (https=) 2023-12-18

Family

ID=75980095

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022529452A Pending JP2023503898A (ja) 2019-11-24 2020-11-24 フルベストラントのプロドラッグ
JP2025202023A Pending JP2026032104A (ja) 2019-11-24 2025-11-21 フルベストラントのプロドラッグ

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025202023A Pending JP2026032104A (ja) 2019-11-24 2025-11-21 フルベストラントのプロドラッグ

Country Status (7)

Country Link
US (1) US20230137764A1 (https=)
EP (1) EP4061376A4 (https=)
JP (2) JP2023503898A (https=)
CN (1) CN115151260A (https=)
AU (1) AU2020386864A1 (https=)
CA (1) CA3162182A1 (https=)
WO (1) WO2021100029A2 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4422636A4 (en) * 2021-10-29 2025-09-03 Kashiv Biosciences Llc INECTABLE PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF BREAST CANCER
WO2023103929A1 (zh) * 2021-12-06 2023-06-15 江苏亚虹医药科技股份有限公司 氟维司群衍生物及其制备方法和医药用途
EP4444318A4 (en) * 2021-12-06 2026-01-28 Amneal Pharmaceuticals Llc COMPOUNDS FOR CANCER TREATMENT
CN114716496B (zh) * 2022-04-29 2024-04-02 香港中文大学(深圳) 氟维司群衍生物及氟维司群衍生物制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2176208T3 (en) * 2007-07-30 2015-04-27 Zynerba Pharmaceuticals Inc Prodrugs of cannabidiol, compositions containing prodrugs of cannabidiol and methods of use thereof
US20140079636A1 (en) * 2012-04-16 2014-03-20 Dinesh U. Chimmanamada Targeted therapeutics
US20160060288A1 (en) * 2013-04-18 2016-03-03 Xi'anlibang Pharmaceutical Technology Co., Ltd. Ester derivatives of 7-alpha-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl)-estra-1,3,5(10)-triene-3,17beta-diol having anticancer activity and preparation method thereof
WO2014169456A1 (zh) * 2013-04-18 2014-10-23 西安力邦医药科技有限责任公司 7-α-[9-(4,4,5,5,5-五氟戊基亚硫酰基)壬基]-雌甾-1,3,5(10)-三烯-3,17β-二醇及其衍生物的用途
CN103421069A (zh) * 2013-05-23 2013-12-04 中国海洋大学 氟维司群磷酸酯衍生物及其制备方法和应用
EP3738594A1 (en) * 2013-09-10 2020-11-18 Madrigal Pharmaceuticals, Inc. Targeted therapeutics having an hsp90 ligand as binding moiety
WO2019050850A1 (en) * 2017-09-05 2019-03-14 Primetime Life Sciences, Llc BIGUANIDINE DERIVATIVES OF THERAPEUTIC AGENTS, AND PREPARATION METHODS AND METHODS OF USING SAME
JP7384903B2 (ja) * 2018-05-24 2023-11-21 ケーアイ ファーマシューティカルズ,リミテッド・ライアビリティ・カンパニー フルベストラントのプロドラッグ

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