JP2023500483A5 - - Google Patents

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Publication number
JP2023500483A5
JP2023500483A5 JP2022525101A JP2022525101A JP2023500483A5 JP 2023500483 A5 JP2023500483 A5 JP 2023500483A5 JP 2022525101 A JP2022525101 A JP 2022525101A JP 2022525101 A JP2022525101 A JP 2022525101A JP 2023500483 A5 JP2023500483 A5 JP 2023500483A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound
pharmaceutical composition
compound described
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022525101A
Other languages
English (en)
Japanese (ja)
Other versions
JP7544815B2 (ja
JP2023500483A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/057996 external-priority patent/WO2021087136A1/en
Publication of JP2023500483A publication Critical patent/JP2023500483A/ja
Publication of JP2023500483A5 publication Critical patent/JP2023500483A5/ja
Priority to JP2024135814A priority Critical patent/JP7688769B2/ja
Application granted granted Critical
Publication of JP7544815B2 publication Critical patent/JP7544815B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022525101A 2019-10-30 2020-10-29 Cd73阻害剤 Active JP7544815B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024135814A JP7688769B2 (ja) 2019-10-30 2024-08-15 Cd73阻害剤

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201962928138P 2019-10-30 2019-10-30
US62/928,138 2019-10-30
US202062987806P 2020-03-10 2020-03-10
US62/987,806 2020-03-10
US202063088646P 2020-10-07 2020-10-07
US63/088,646 2020-10-07
PCT/US2020/057996 WO2021087136A1 (en) 2019-10-30 2020-10-29 Cd73 inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024135814A Division JP7688769B2 (ja) 2019-10-30 2024-08-15 Cd73阻害剤

Publications (3)

Publication Number Publication Date
JP2023500483A JP2023500483A (ja) 2023-01-06
JP2023500483A5 true JP2023500483A5 (https=) 2023-10-13
JP7544815B2 JP7544815B2 (ja) 2024-09-03

Family

ID=75686256

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022525101A Active JP7544815B2 (ja) 2019-10-30 2020-10-29 Cd73阻害剤
JP2024135814A Active JP7688769B2 (ja) 2019-10-30 2024-08-15 Cd73阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024135814A Active JP7688769B2 (ja) 2019-10-30 2024-08-15 Cd73阻害剤

Country Status (19)

Country Link
US (7) US12577272B2 (https=)
EP (2) EP4596048A3 (https=)
JP (2) JP7544815B2 (https=)
KR (2) KR102727229B1 (https=)
CN (2) CN114929721B (https=)
AU (1) AU2020375914B2 (https=)
CA (1) CA3159248C (https=)
DK (1) DK4051688T3 (https=)
ES (1) ES3034168T3 (https=)
FI (1) FI4051688T3 (https=)
HU (1) HUE072504T2 (https=)
IL (2) IL292570B2 (https=)
MX (1) MX2022005256A (https=)
PL (1) PL4051688T3 (https=)
PT (1) PT4051688T (https=)
SI (1) SI4051688T1 (https=)
TW (1) TWI830962B (https=)
WO (1) WO2021087136A1 (https=)
ZA (1) ZA202204941B (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018208980A1 (en) 2017-05-10 2018-11-15 Oric Pharmaceuticals, Inc. Cd73 inhibitors
US11377469B2 (en) 2017-11-03 2022-07-05 Oric Pharmaceuticals, Inc. CD73 inhibitors
IL304348B2 (en) 2018-04-30 2024-08-01 Oric Pharmaceuticals Inc CD73 inhibitors
JP7557522B2 (ja) 2019-07-16 2024-09-27 オリック ファーマシューティカルズ,インク. Cd73阻害剤
PL4051688T3 (pl) * 2019-10-30 2025-09-22 Oric Pharmaceuticals, Inc. Inhibitory cd73
JP2025512384A (ja) 2022-04-13 2025-04-17 ギリアード サイエンシーズ, インコーポレイテッド Trop-2発現がんを治療するための併用療法
CN120202181A (zh) * 2022-09-14 2025-06-24 欧瑞克制药公司 Cd73抑制剂的药物形式
WO2024076873A1 (en) * 2022-10-03 2024-04-11 Teon Therapeutics, Inc. Heterocyclic inhibitors of cd73 for treatment of disease
WO2024076872A1 (en) * 2022-10-03 2024-04-11 Teon Therapeutics, Inc. Heterocyclic inhibitors of cd73 for treatment of disease
WO2025111247A1 (en) * 2023-11-20 2025-05-30 Oric Pharmaceuticals, Inc. Treatment of refractory multiple myeloma
WO2025137640A1 (en) 2023-12-22 2025-06-26 Gilead Sciences, Inc. Azaspiro wrn inhibitors
WO2025233264A1 (en) 2024-05-07 2025-11-13 Innate Pharma Use of cd73 blocking agents in combination with anti-cd20 x cd3 t cell engagers

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WO2002048165A2 (en) 2000-12-15 2002-06-20 Pharmasset Ltd. Antiviral agents for treatment of flaviviridae infections
US20040229839A1 (en) 2003-05-14 2004-11-18 Biocryst Pharmaceuticals, Inc. Substituted nucleosides, preparation thereof and use as inhibitors of RNA viral polymerases
WO2005020885A2 (en) 2003-05-21 2005-03-10 Isis Pharmaceuticals, Inc. Compositions and methods for the treatment of severe acute respiratory syndrome (sars)
US20090029949A1 (en) 2006-05-25 2009-01-29 Parrill-Baker Abby L GPCR Ligands Identified by Computational Modeling
DE102007001370A1 (de) 2007-01-09 2008-07-10 Curevac Gmbh RNA-kodierte Antikörper
WO2009127230A1 (en) 2008-04-16 2009-10-22 Curevac Gmbh MODIFIED (m)RNA FOR SUPPRESSING OR AVOIDING AN IMMUNOSTIMULATORY RESPONSE AND IMMUNOSUPPRESSIVE COMPOSITION
US20090274686A1 (en) 2008-05-02 2009-11-05 Yat Sun Or Nucleoside phosphonate derivatives
MA39986A (fr) * 2014-04-25 2017-03-01 Vitae Pharmaceuticals Inc Dérivés de purine en tant qu'inhibiteurs de cd73 pour le traitement du cancer
CN104530166B (zh) 2014-12-04 2016-08-24 陕西汉江药业集团股份有限公司 选择性还原4,6-共轭双烯-3-酮甾体化合物的方法
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EP3510040A4 (en) * 2016-09-09 2020-06-03 Calithera Biosciences, Inc. EKTONUCLEOTIDASE INHIBITORS AND METHOD FOR USE THEREOF
EP3518934A4 (en) 2016-10-03 2020-06-24 Arcus Biosciences, Inc. Inhibitors of adenosine 5'-nucleotidase
WO2018094148A1 (en) 2016-11-18 2018-05-24 Arcus Biosciences, Inc. Inhibitors of cd73-mediated immunosuppression
KR102638592B1 (ko) 2016-12-22 2024-02-19 안텐진 테라퓨틱스 리미티드 엑토뉴클레오티다제 억제제 및 이의 용도
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WO2018208727A1 (en) * 2017-05-08 2018-11-15 Eternity Bioscience Inc. Nucleoside and nucleotide analogues as cd73 inhibitors and therapeutic uses thereof
WO2018208980A1 (en) * 2017-05-10 2018-11-15 Oric Pharmaceuticals, Inc. Cd73 inhibitors
US11377469B2 (en) 2017-11-03 2022-07-05 Oric Pharmaceuticals, Inc. CD73 inhibitors
CN111094317B (zh) 2017-12-29 2023-03-31 上海和誉生物医药科技有限公司 一种具有cd73抑制活性的膦酸衍生物、其制备方法和应用
IL304348B2 (en) 2018-04-30 2024-08-01 Oric Pharmaceuticals Inc CD73 inhibitors
WO2019232319A1 (en) 2018-05-31 2019-12-05 Peloton Therapeutics, Inc. Compositions and methods for inhibiting cd73
SG11202012001YA (en) 2018-06-21 2021-01-28 Calithera Biosciences Inc Ectonucleotidase inhibitors and methods of use thereof
WO2020046813A1 (en) 2018-08-27 2020-03-05 Arcus Biosciences, Inc. Cd73 inhibitors
WO2020257429A1 (en) 2019-06-20 2020-12-24 Calithera Biosciences, Inc. Ectonucleotidase inhibitors and methods of use thereof
JP7557522B2 (ja) 2019-07-16 2024-09-27 オリック ファーマシューティカルズ,インク. Cd73阻害剤
PL4051688T3 (pl) 2019-10-30 2025-09-22 Oric Pharmaceuticals, Inc. Inhibitory cd73

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