JP2023145481A5 - - Google Patents

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Publication number
JP2023145481A5
JP2023145481A5 JP2023111632A JP2023111632A JP2023145481A5 JP 2023145481 A5 JP2023145481 A5 JP 2023145481A5 JP 2023111632 A JP2023111632 A JP 2023111632A JP 2023111632 A JP2023111632 A JP 2023111632A JP 2023145481 A5 JP2023145481 A5 JP 2023145481A5
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JP
Japan
Prior art keywords
compound
xrd
crystals
irradiated
light source
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2023111632A
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English (en)
Japanese (ja)
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JP2023145481A (ja
JP7773506B2 (ja
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Priority claimed from JP2020068458A external-priority patent/JP7352509B2/ja
Application filed filed Critical
Publication of JP2023145481A publication Critical patent/JP2023145481A/ja
Publication of JP2023145481A5 publication Critical patent/JP2023145481A5/ja
Application granted granted Critical
Publication of JP7773506B2 publication Critical patent/JP7773506B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2023111632A 2016-06-17 2023-07-06 ジフェニルメタン誘導体の製造方法 Active JP7773506B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
KR10-2016-0075910 2016-06-17
KR20160075910 2016-06-17
JP2020068458A JP7352509B2 (ja) 2016-06-17 2020-04-06 ジフェニルメタン誘導体の製造方法
JP2021102648A JP7669206B2 (ja) 2016-06-17 2021-06-21 ジフェニルメタン誘導体の製造方法

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2021102648A Division JP7669206B2 (ja) 2016-06-17 2021-06-21 ジフェニルメタン誘導体の製造方法

Publications (3)

Publication Number Publication Date
JP2023145481A JP2023145481A (ja) 2023-10-11
JP2023145481A5 true JP2023145481A5 (https=) 2025-09-26
JP7773506B2 JP7773506B2 (ja) 2025-11-19

Family

ID=60664449

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2018565754A Active JP6763978B2 (ja) 2016-06-17 2017-06-15 ジフェニルメタン誘導体の製造方法
JP2020068458A Active JP7352509B2 (ja) 2016-06-17 2020-04-06 ジフェニルメタン誘導体の製造方法
JP2021102648A Active JP7669206B2 (ja) 2016-06-17 2021-06-21 ジフェニルメタン誘導体の製造方法
JP2023111632A Active JP7773506B2 (ja) 2016-06-17 2023-07-06 ジフェニルメタン誘導体の製造方法

Family Applications Before (3)

Application Number Title Priority Date Filing Date
JP2018565754A Active JP6763978B2 (ja) 2016-06-17 2017-06-15 ジフェニルメタン誘導体の製造方法
JP2020068458A Active JP7352509B2 (ja) 2016-06-17 2020-04-06 ジフェニルメタン誘導体の製造方法
JP2021102648A Active JP7669206B2 (ja) 2016-06-17 2021-06-21 ジフェニルメタン誘導体の製造方法

Country Status (29)

Country Link
US (2) US10640496B2 (https=)
EP (2) EP3473621B1 (https=)
JP (4) JP6763978B2 (https=)
KR (2) KR102233229B1 (https=)
CN (2) CN113651803B (https=)
AU (1) AU2017285813B2 (https=)
CA (2) CA3026756C (https=)
CL (1) CL2018003645A1 (https=)
CO (1) CO2018014018A2 (https=)
DK (2) DK3663292T3 (https=)
DO (1) DOP2018000287A (https=)
EC (1) ECSP19000185A (https=)
ES (2) ES2898336T3 (https=)
HR (1) HRP20211670T8 (https=)
HU (1) HUE056428T2 (https=)
MA (2) MA44545B2 (https=)
MX (2) MX392177B (https=)
MY (1) MY203941A (https=)
NZ (1) NZ749398A (https=)
PE (2) PE20240590A1 (https=)
PH (1) PH12018550206A1 (https=)
PL (2) PL3663292T3 (https=)
PT (2) PT3663292T (https=)
RS (1) RS62550B1 (https=)
SA (2) SA521422474B1 (https=)
SG (2) SG10201911782RA (https=)
SI (1) SI3663292T1 (https=)
TN (1) TN2018000437A1 (https=)
WO (1) WO2017217792A1 (https=)

Families Citing this family (20)

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Publication number Priority date Publication date Assignee Title
DE102011054773A1 (de) 2011-10-25 2013-04-25 Vb Autobatterie Gmbh & Co. Kgaa Anschlusspol für einen Akkumulator, Akkumulatorgehäuse und Maschine zur Herstellung eines Anschlusspols
EP3838894B1 (en) 2018-08-13 2024-03-13 Daewoong Pharmaceutical Co., Ltd. Method for producing intermediate useful for synethesis of sglt inhibitor
CN112341416A (zh) * 2019-08-09 2021-02-09 天津津艺医药科技发展有限责任公司 一种制备苯并含氧脂杂环衍生物的方法
EP4112612B1 (en) 2020-02-27 2025-10-22 Daewoong Pharmaceutical Co., Ltd. Intermediate useful for synthesis of sglt inhibitor and method for preparing sglt inhibitor using same
CN112094253B (zh) * 2020-09-10 2023-01-10 株式会社大熊制药 用于制备sglt抑制剂中间体的合成方法
PE20231373A1 (es) 2020-09-10 2023-09-07 Daewoong Pharmaceutical Co Ltd Metodo de sintesis para la preparacion de un intermedio de inhibidores de sglt
CN113200860B (zh) * 2021-04-29 2024-07-30 爱斯特(成都)生物制药股份有限公司 一种sglt2抑制剂中间体的制备方法
KR20230046784A (ko) * 2021-09-30 2023-04-06 주식회사 대웅제약 이나보글리플로진을 포함하는 약학 조성물
CN113801010A (zh) * 2021-11-18 2021-12-17 山东诚创蓝海医药科技有限公司 一种5-溴-2-氯苯甲酸的制备方法
CN113912487B (zh) * 2021-11-23 2024-05-28 山东研峰新材料科技有限公司 一种2,5-双卤代苯甲酸的合成方法
KR20230110001A (ko) * 2022-01-14 2023-07-21 주식회사 대웅제약 Ssglt 저해제의 합성에 유용한 중간체의 제조 방법
KR20240044194A (ko) 2022-09-28 2024-04-04 주식회사 대웅제약 이나보글리플로진의 신규한 공결정
KR20240044190A (ko) 2022-09-28 2024-04-04 주식회사 대웅제약 이나보글리플로진의 신규한 결정형 및 이의 제조방법
CN119968202A (zh) 2022-09-29 2025-05-09 株式会社大熊制药 用于预防或治疗心血管衰老疾病的包含依那格列净的药物组合物
WO2024076177A1 (ko) 2022-10-05 2024-04-11 주식회사 대웅제약 이나보글리플로진을 포함하는 신장애 및/또는 당뇨병 예방 또는 치료용 약학 조성물
CN120435283A (zh) 2022-12-21 2025-08-05 大熊治疗株式会社 包含依那格列净的滴眼剂形式的药物组合物
KR20240107660A (ko) 2022-12-30 2024-07-09 주식회사 대웅제약 이나보글리플로진 및 메트포르민을 포함하는 약학 조성물
KR102837941B1 (ko) * 2024-11-13 2025-07-25 대웅바이오(주) Inline quenching 공정을 도입한 연속반응 공정을 이용한 이나보글리플로진 합성방법
KR102853437B1 (ko) * 2024-11-13 2025-09-04 대웅바이오(주) 연속반응 공정을 이용한 이나보글리플로진 합성방법
KR102837948B1 (ko) * 2024-11-13 2025-07-25 대웅바이오(주) 분배 투입법을 도입한 연속반응 공정을 이용한 이나보글리플로진 합성방법

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US4966907A (en) * 1988-08-12 1990-10-30 Merck & Co., Inc. 6-substituted 5-hydroxy-2,3-dihydrobenzofurans as inhibitors of leukotriene biosynthesis
LT2896397T (lt) * 2003-08-01 2017-11-27 Mitsubishi Tanabe Pharma Corporation Nauji junginiai, turintys inhibitorinį aktyvumą prieš nuo natrio priklausomą gliukozės transporterį
AU2008279424B2 (en) 2007-07-26 2013-06-13 Lexicon Pharmaceuticals, Inc. Methods and compounds useful for the preparation of sodium glucose co-transporter 2 inhibitors
PE20110208A1 (es) 2008-07-30 2011-03-28 Ferrer Int Compuestos de 1,6-dihidro-2h-3-oxa-6-aza-as-indaceno
US8163704B2 (en) 2009-10-20 2012-04-24 Novartis Ag Glycoside derivatives and uses thereof
WO2012041898A1 (en) * 2010-09-29 2012-04-05 Celon Pharma Sp. Z O.O. Combination of sglt2 inhibitor and a sugar compound for the treatment of diabetes
WO2012165914A2 (en) * 2011-06-01 2012-12-06 Green Cross Corporation Novel diphenylmethane derivatives as sglt2 inhibitors
US9340521B2 (en) 2013-03-18 2016-05-17 Green Cross Corporation Method for dual inhibition of SGLT1 and SGLT2 using diphenylmethane derivatives
FR3017868A1 (fr) 2014-02-21 2015-08-28 Servier Lab Derives d'isoquinoleine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

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