JP2022552401A5 - - Google Patents
Info
- Publication number
- JP2022552401A5 JP2022552401A5 JP2022522773A JP2022522773A JP2022552401A5 JP 2022552401 A5 JP2022552401 A5 JP 2022552401A5 JP 2022522773 A JP2022522773 A JP 2022522773A JP 2022522773 A JP2022522773 A JP 2022522773A JP 2022552401 A5 JP2022552401 A5 JP 2022552401A5
- Authority
- JP
- Japan
- Prior art keywords
- piperidine
- imidazole
- propan
- methylthio
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2019/111690 | 2019-10-17 | ||
| CN2019111690 | 2019-10-17 | ||
| PCT/EP2020/079009 WO2021074281A1 (en) | 2019-10-17 | 2020-10-15 | Substituted azacyles as trmp8 modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022552401A JP2022552401A (ja) | 2022-12-15 |
| JP2022552401A5 true JP2022552401A5 (https=) | 2023-10-24 |
| JP7778688B2 JP7778688B2 (ja) | 2025-12-02 |
Family
ID=72964655
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022522773A Active JP7778688B2 (ja) | 2019-10-17 | 2020-10-15 | Ｔｒｍｐ８モジュレーターとしての置換アザシル |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US12528801B2 (https=) |
| EP (1) | EP4045491A1 (https=) |
| JP (1) | JP7778688B2 (https=) |
| KR (1) | KR20220085798A (https=) |
| CN (1) | CN114555594B (https=) |
| BR (1) | BR112022005289A2 (https=) |
| CO (1) | CO2022004130A2 (https=) |
| IL (1) | IL292156B1 (https=) |
| MX (1) | MX2022003494A (https=) |
| WO (1) | WO2021074281A1 (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB202012170D0 (en) * | 2020-08-05 | 2020-09-16 | Givaudan Sa | Organic compounds |
| GB202013383D0 (en) * | 2020-08-26 | 2020-10-07 | Givaudan Sa | Process |
| WO2022170519A1 (en) | 2021-02-09 | 2022-08-18 | Givaudan Sa | Organic compounds |
| GB202102676D0 (en) | 2021-02-25 | 2021-04-14 | Givaudan Sa | Compositions |
| GB202103207D0 (en) | 2021-03-08 | 2021-04-21 | Givaudan Sa | Organic compounds |
| GB202105661D0 (en) | 2021-04-21 | 2021-06-02 | Givaudan Sa | Organic compounds |
| JP2024522284A (ja) | 2021-05-28 | 2024-06-13 | フィルメニッヒ インコーポレイテッド | 清涼効果を増強する組成物 |
| US20240358611A1 (en) | 2021-08-16 | 2024-10-31 | Symrise Ag | Compositions |
| EP4525821A1 (en) | 2022-07-07 | 2025-03-26 | Firmenich Incorporated | Compositions that enhance the cooling effect |
| WO2022207944A2 (en) | 2022-07-11 | 2022-10-06 | Symrise Ag | Novel mixtures and uses of (2e)-3-(1,3-benzodioxol-5-yl)-n-phenyl-n-(tetrahydro-3-furanyl)-2-propenamide |
| CN120129464A (zh) | 2022-10-27 | 2025-06-10 | 弗门尼舍有限公司 | 黄酮类化合物及其用途 |
| CN120417784A (zh) | 2022-12-22 | 2025-08-01 | 弗门尼舍有限公司 | 含烷基乳酸酯的天然甜味剂组合物及其用途 |
| EP4608172A1 (en) | 2022-12-22 | 2025-09-03 | Firmenich SA | Natural sweetener compositions and uses thereof |
| JP2026511252A (ja) | 2023-03-28 | 2026-04-10 | フイルメニツヒ ソシエテ アノニム | 味改変組成物およびその使用 |
| WO2025051340A1 (en) | 2023-09-04 | 2025-03-13 | Symrise Ag | Trpm8 modulators and related method for modulating trpm8 receptors |
| GB202315636D0 (en) | 2023-10-12 | 2023-11-29 | Givaudan Sa | Composition |
| WO2025132323A1 (en) | 2023-12-21 | 2025-06-26 | Dsm-Firmenich Ag | Compositions comprising a sunscreen active agent |
| WO2026052684A1 (en) | 2024-09-04 | 2026-03-12 | Givaudan Sa | Flavour compositions |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3988433A (en) | 1973-08-10 | 1976-10-26 | The Procter & Gamble Company | Oral compositions for preventing or removing stains from teeth |
| US4083955A (en) | 1975-04-02 | 1978-04-11 | The Procter & Gamble Company | Processes and compositions for remineralization of dental enamel |
| US4528180A (en) | 1983-03-01 | 1985-07-09 | Schaeffer Hans A | Dental preparation, article and method for storage and delivery thereof |
| US4849213A (en) | 1983-03-01 | 1989-07-18 | Schaeffer Hans A | Dental preparation, article and method for storage and delivery therof |
| US5198220A (en) | 1989-11-17 | 1993-03-30 | The Procter & Gamble Company | Sustained release compositions for treating periodontal disease |
| US5145666A (en) | 1991-10-23 | 1992-09-08 | The Proctor & Gamble Co. | Methods of reducing plaque and gingivitis with reduced staining |
| US5213790A (en) | 1991-10-23 | 1993-05-25 | The Procter & Gamble Co. | Methods of reducing plaque and gingivitis with reduced staining |
| US5281410A (en) | 1991-10-23 | 1994-01-25 | The Proctor & Gamble Company | Methods of reducing plaque and gingivitis with reduced staining |
| US5242910A (en) | 1992-10-13 | 1993-09-07 | The Procter & Gamble Company | Sustained release compositions for treating periodontal disease |
| US5965537A (en) * | 1997-03-10 | 1999-10-12 | Basf Aktiengesellschaft | Dolastatin 15 derivatives with carbonyl and heterocyclic functionalities at the C-terminus |
| DE60128731T2 (de) * | 2000-10-30 | 2008-02-07 | Janssen Pharmaceutica N.V. | Tripeptidylpeptidase-hemmer |
| HUP0500920A2 (en) * | 2005-10-05 | 2007-07-30 | Richter Gedeon Nyrt | Oxadiazole derivatives, process for their preparation and their use |
| HUP0500921A2 (en) | 2005-10-05 | 2007-07-30 | Richter Gedeon Nyrt | Tetrazole derivatives, process for their preparation and their use |
| GB0704163D0 (en) | 2007-03-02 | 2007-04-11 | Quest Int Serv Bv | Compositions comprising a physiological coolant |
| US8143259B2 (en) * | 2008-08-19 | 2012-03-27 | Janssen Pharmaceutica, Nv | Cold menthol receptor antagonists |
| EP2346475B2 (en) | 2008-11-20 | 2023-04-19 | The Procter & Gamble Company | Personal care compositions providing enhanced cooling sensation |
| CN103201279A (zh) | 2010-11-05 | 2013-07-10 | 赛诺米克斯公司 | 作为trpm8的调节剂有用的化合物 |
| US20150216168A1 (en) | 2012-09-05 | 2015-08-06 | Bayer Cropscience Ag | Use of substituted 2-amidobenzimidazoles, 2-amidobenzoxazoles and 2-amidobenzothiazoles or salts thereof as active substances against abiotic plant stress |
| TWI674257B (zh) | 2014-03-14 | 2019-10-11 | 日商拉夸里亞創藥股份有限公司 | 作為ｔｒｐｍ８拮抗劑之氮雜螺衍生物 |
| AU2016281346B2 (en) * | 2015-06-23 | 2020-01-02 | Kissei Pharmaceutical Co., Ltd. | Pyrazole derivative, or pharmaceutically acceptable salt thereof |
| ES2967435T3 (es) | 2017-08-31 | 2024-04-30 | Basf Se | Uso de principios activos refrescantes fisiológicos y productos que contienen dichos principios activos |
| JP7487100B2 (ja) | 2017-12-21 | 2024-05-20 | フイルメニツヒ ソシエテ アノニム | 清涼および風味増強組成物 |
-
2020
- 2020-10-15 EP EP20793607.1A patent/EP4045491A1/en active Pending
- 2020-10-15 WO PCT/EP2020/079009 patent/WO2021074281A1/en not_active Ceased
- 2020-10-15 MX MX2022003494A patent/MX2022003494A/es unknown
- 2020-10-15 KR KR1020227016597A patent/KR20220085798A/ko active Pending
- 2020-10-15 US US17/769,198 patent/US12528801B2/en active Active
- 2020-10-15 JP JP2022522773A patent/JP7778688B2/ja active Active
- 2020-10-15 BR BR112022005289A patent/BR112022005289A2/pt unknown
- 2020-10-15 CN CN202080072667.6A patent/CN114555594B/zh active Active
-
2022
- 2022-03-31 CO CONC2022/0004130A patent/CO2022004130A2/es unknown
- 2022-04-11 IL IL292156A patent/IL292156B1/en unknown
-
2025
- 2025-12-15 US US19/419,870 patent/US20260103459A1/en active Pending
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