JP2022541752A5 - - Google Patents

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Publication number
JP2022541752A5
JP2022541752A5 JP2022501191A JP2022501191A JP2022541752A5 JP 2022541752 A5 JP2022541752 A5 JP 2022541752A5 JP 2022501191 A JP2022501191 A JP 2022501191A JP 2022501191 A JP2022501191 A JP 2022501191A JP 2022541752 A5 JP2022541752 A5 JP 2022541752A5
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Japan
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cys
pro
phe
solvate
hydrate
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JP2022501191A
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English (en)
Japanese (ja)
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JP7801207B2 (ja
JP2022541752A (ja
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Priority claimed from EP19000325.1A external-priority patent/EP3763726A1/en
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Priority claimed from PCT/EP2020/069308 external-priority patent/WO2021005131A1/en
Publication of JP2022541752A publication Critical patent/JP2022541752A/ja
Publication of JP2022541752A5 publication Critical patent/JP2022541752A5/ja
Priority to JP2026000148A priority Critical patent/JP2026062901A/ja
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Publication of JP7801207B2 publication Critical patent/JP7801207B2/ja
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JP2022501191A 2019-07-08 2020-07-08 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用 Active JP7801207B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2026000148A JP2026062901A (ja) 2019-07-08 2026-01-05 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP19000325.1 2019-07-08
EP19000325.1A EP3763726A1 (en) 2019-07-08 2019-07-08 Compounds comprising a fibroblast activation protein ligand and use thereof
EP19198810.4 2019-09-20
EP19198810 2019-09-20
PCT/EP2020/069308 WO2021005131A1 (en) 2019-07-08 2020-07-08 Compounds comprising a fibroblast activation protein ligand and use thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2026000148A Division JP2026062901A (ja) 2019-07-08 2026-01-05 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用

Publications (3)

Publication Number Publication Date
JP2022541752A JP2022541752A (ja) 2022-09-27
JP2022541752A5 true JP2022541752A5 (https=) 2023-07-20
JP7801207B2 JP7801207B2 (ja) 2026-01-16

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ID=71409440

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JP2022501191A Active JP7801207B2 (ja) 2019-07-08 2020-07-08 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用
JP2026000148A Pending JP2026062901A (ja) 2019-07-08 2026-01-05 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用

Family Applications After (1)

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JP2026000148A Pending JP2026062901A (ja) 2019-07-08 2026-01-05 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用

Country Status (12)

Country Link
US (1) US20220315554A1 (https=)
EP (1) EP3997104A1 (https=)
JP (2) JP7801207B2 (https=)
KR (1) KR20220032078A (https=)
CN (3) CN114341158B (https=)
AU (1) AU2020309161A1 (https=)
BR (1) BR112022000144A2 (https=)
CA (1) CA3145872A1 (https=)
CL (1) CL2022000016A1 (https=)
IL (2) IL289673B2 (https=)
MX (1) MX2022000251A (https=)
WO (1) WO2021005131A1 (https=)

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WO2022115778A1 (en) * 2020-11-30 2022-06-02 Rayzebio, Inc. Radiopharmaceutical conjugate compositions and uses thereof
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WO2024198838A1 (zh) * 2023-03-27 2024-10-03 晶核生物医药科技(南京)有限公司 环状多肽类化合物及其应用
EP4692105A1 (en) * 2023-03-27 2026-02-11 Bivision Pharmaceuticals, Inc Cyclic polypeptide compound and use thereof
WO2024198836A1 (zh) * 2023-03-27 2024-10-03 晶核生物医药科技(南京)有限公司 环状多肽类化合物及其应用
CN118930606A (zh) * 2023-05-11 2024-11-12 成都纽瑞特医疗科技股份有限公司 靶向成纤维细胞活化蛋白的多肽放射性核素配合物及其应用
WO2025011611A1 (zh) * 2023-07-11 2025-01-16 江苏恒瑞医药股份有限公司 一种成纤维细胞活化蛋白配体及其用途
WO2025046043A1 (en) 2023-08-31 2025-03-06 Stichting Radboud Universitair Medisch Centrum Endometriosis tracer
WO2025082283A1 (zh) * 2023-10-16 2025-04-24 四川科伦博泰生物医药股份有限公司 环肽结构的配体化合物及其核素标记物、药物组合物及应用
US20250186630A1 (en) 2023-12-12 2025-06-12 Viewpoint Molecular Targeting, Inc. Fibroblast activation protein targeting peptides
WO2025163556A1 (en) 2024-02-01 2025-08-07 Novartis Ag Methods for treating cancer
WO2026008525A1 (en) * 2024-07-01 2026-01-08 Bayer Aktiengesellschaft Stable radionuclide-containing formulations
WO2026017046A1 (zh) * 2024-07-19 2026-01-22 晶核生物医药科技(南京)有限公司 一种环多肽、其制备方法和应用
WO2026021314A1 (zh) * 2024-07-22 2026-01-29 山东威智知科药业有限公司 Fap化合物及其用途
WO2026041109A1 (zh) * 2024-08-23 2026-02-26 苏州博锐创合医药有限公司 成纤维细胞活化蛋白抑制剂及其用途
CN120590466A (zh) * 2025-08-06 2025-09-05 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 一种靶向成纤维细胞活化蛋白的化合物及其应用

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EA202090776A1 (ru) 2017-10-23 2020-07-27 Дзе Джонс Хопкинс Юниверсити Визуализирующие и радиотерапевтические агенты, нацеленные на фибробласт-активирующий белок-альфа (fapalpha)
FI3997103T3 (fi) * 2019-07-08 2025-02-03 3B Pharmaceuticals Gmbh Fibroblastien aktivaatioproteiinin ligandia käsittäviä yhdisteitä ja niiden käyttö

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