JP2022539840A5 - - Google Patents

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Publication number
JP2022539840A5
JP2022539840A5 JP2022500764A JP2022500764A JP2022539840A5 JP 2022539840 A5 JP2022539840 A5 JP 2022539840A5 JP 2022500764 A JP2022500764 A JP 2022500764A JP 2022500764 A JP2022500764 A JP 2022500764A JP 2022539840 A5 JP2022539840 A5 JP 2022539840A5
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JP
Japan
Prior art keywords
cancer
pharmaceutically
veterinarily acceptable
use according
pyrazolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2022500764A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022539840A (ja
JP7536243B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2020/069459 external-priority patent/WO2021005183A1/en
Publication of JP2022539840A publication Critical patent/JP2022539840A/ja
Publication of JP2022539840A5 publication Critical patent/JP2022539840A5/ja
Application granted granted Critical
Publication of JP7536243B2 publication Critical patent/JP7536243B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022500764A 2019-07-10 2020-07-09 Mapキナーゼ相互作用セリン/スレオニン-プロテインキナーゼ1(mnk1)及びmapキナーゼ相互作用セリン/スレオニン-プロテインキナーゼ2(mnk2)の阻害剤、癌治療及び治療的組合せ Active JP7536243B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES201930643 2019-07-10
ESP201930643 2019-07-10
PCT/EP2020/069459 WO2021005183A1 (en) 2019-07-10 2020-07-09 Inhibitor of map kinase interacting serine/threonine kinase 1 (mnk1) and map kinase interacting serine/threonine kinase 2 (mnk2), cancer therapy and therapeutic combinations

Publications (3)

Publication Number Publication Date
JP2022539840A JP2022539840A (ja) 2022-09-13
JP2022539840A5 true JP2022539840A5 (https=) 2023-07-18
JP7536243B2 JP7536243B2 (ja) 2024-08-20

Family

ID=71607975

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022500764A Active JP7536243B2 (ja) 2019-07-10 2020-07-09 Mapキナーゼ相互作用セリン/スレオニン-プロテインキナーゼ1(mnk1)及びmapキナーゼ相互作用セリン/スレオニン-プロテインキナーゼ2(mnk2)の阻害剤、癌治療及び治療的組合せ

Country Status (5)

Country Link
US (1) US20220257571A1 (https=)
EP (1) EP3996710B1 (https=)
JP (1) JP7536243B2 (https=)
ES (1) ES3014017T3 (https=)
WO (1) WO2021005183A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11958832B1 (en) 2023-10-12 2024-04-16 King Faisal University 2-alkoxy[4,3:6,3-terpyridine]-3-carbonitriles as antimicrobial compounds
US11926611B1 (en) 2023-11-24 2024-03-12 King Faisal University 2-(2-ethoxyethoxy)-6-phenyl-4,4′-bipyridine-3-carbonitrile as an antimicrobial compound
US12071407B1 (en) 2023-12-05 2024-08-27 King Faisal University 6-(4-hydroxyphenyl)-2-(2-ethoxyethoxy)-4-(4-methoxyphenyl)nicotinonitrile as an antimicrobial compound
US11970451B1 (en) 2023-12-07 2024-04-30 King Faisal University 6-(3-hydroxyphenyl)-2-methoxy-4-(3-methylphenyl)nicotinonitrile as an antimicrobial compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2160780A1 (de) 1971-12-08 1973-06-14 Basf Ag Pyridino-pyrazole
US20100113415A1 (en) 2008-05-29 2010-05-06 Rajapakse Hemaka A Epha4 rtk inhibitors for treatment of neurological and neurodegenerative disorders and cancer
US8846673B2 (en) 2009-08-11 2014-09-30 Bristol-Myers Squibb Company Azaindazoles as kinase inhibitors and use thereof
JP2016527216A (ja) 2013-07-08 2016-09-08 バイエル・ファルマ・アクティエンゲゼルシャフト 置換ピラゾロピリジン
EP3285809B1 (en) * 2015-04-20 2019-09-11 eFFECTOR Therapeutics, Inc. Inhibitors of immune checkpoint modulators for use in treating cancer and infections

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