JP2022539342A5 - - Google Patents

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Publication number
JP2022539342A5
JP2022539342A5 JP2021576883A JP2021576883A JP2022539342A5 JP 2022539342 A5 JP2022539342 A5 JP 2022539342A5 JP 2021576883 A JP2021576883 A JP 2021576883A JP 2021576883 A JP2021576883 A JP 2021576883A JP 2022539342 A5 JP2022539342 A5 JP 2022539342A5
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JP
Japan
Prior art keywords
crystalline form
compound
approximately
solid crystalline
powder
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021576883A
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English (en)
Japanese (ja)
Other versions
JP7617043B2 (ja
JP2022539342A (ja
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Priority claimed from PCT/US2020/039163 external-priority patent/WO2020263847A1/en
Publication of JP2022539342A publication Critical patent/JP2022539342A/ja
Publication of JP2022539342A5 publication Critical patent/JP2022539342A5/ja
Priority to JP2025001914A priority Critical patent/JP2025069143A/ja
Application granted granted Critical
Publication of JP7617043B2 publication Critical patent/JP7617043B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021576883A 2019-06-24 2020-06-23 ｔｅｒｔ－ブチル（Ｓ）－２－（（２Ｓ，３Ｒ）－１－アミノ－３－ヒドロキシ－１－オキソブタン－２－イル）－１－オキソ－２，５－ジアザスピロ［３．４］オクタン－５－カルボキシレートの固体形態およびそれらを調製する方法 Active JP7617043B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025001914A JP2025069143A (ja) 2019-06-24 2025-01-06 ｔｅｒｔ－ブチル（Ｓ）－２－（（２Ｓ，３Ｒ）－１－アミノ－３－ヒドロキシ－１－オキソブタン－２－イル）－１－オキソ－２，５－ジアザスピロ［３．４］オクタン－５－カルボキシレートの固体形態およびそれらを調製する方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962865826P 2019-06-24 2019-06-24
US62/865,826 2019-06-24
PCT/US2020/039163 WO2020263847A1 (en) 2019-06-24 2020-06-23 Solid forms of tert-butyl (s)-2-((2s,3r) -1-amino-3-hydroxy-1-oxobu tan-2-yl)-1-oxo-2, 5-diazaspiro [3.4] octan e-5-carboxylate and methods of preparing them

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025001914A Division JP2025069143A (ja) 2019-06-24 2025-01-06 ｔｅｒｔ－ブチル（Ｓ）－２－（（２Ｓ，３Ｒ）－１－アミノ－３－ヒドロキシ－１－オキソブタン－２－イル）－１－オキソ－２，５－ジアザスピロ［３．４］オクタン－５－カルボキシレートの固体形態およびそれらを調製する方法

Publications (3)

Publication Number Publication Date
JP2022539342A JP2022539342A (ja) 2022-09-08
JP2022539342A5 true JP2022539342A5 (enExample) 2023-06-30
JP7617043B2 JP7617043B2 (ja) 2025-01-17

Family

ID=74060350

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021576883A Active JP7617043B2 (ja) 2019-06-24 2020-06-23 ｔｅｒｔ－ブチル（Ｓ）－２－（（２Ｓ，３Ｒ）－１－アミノ－３－ヒドロキシ－１－オキソブタン－２－イル）－１－オキソ－２，５－ジアザスピロ［３．４］オクタン－５－カルボキシレートの固体形態およびそれらを調製する方法
JP2025001914A Pending JP2025069143A (ja) 2019-06-24 2025-01-06 ｔｅｒｔ－ブチル（Ｓ）－２－（（２Ｓ，３Ｒ）－１－アミノ－３－ヒドロキシ－１－オキソブタン－２－イル）－１－オキソ－２，５－ジアザスピロ［３．４］オクタン－５－カルボキシレートの固体形態およびそれらを調製する方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025001914A Pending JP2025069143A (ja) 2019-06-24 2025-01-06 ｔｅｒｔ－ブチル（Ｓ）－２－（（２Ｓ，３Ｒ）－１－アミノ－３－ヒドロキシ－１－オキソブタン－２－イル）－１－オキソ－２，５－ジアザスピロ［３．４］オクタン－５－カルボキシレートの固体形態およびそれらを調製する方法

Country Status (11)

Country Link
US (1) US20220267341A1 (enExample)
EP (1) EP3986399A4 (enExample)
JP (2) JP7617043B2 (enExample)
CN (1) CN114364380A (enExample)
AU (1) AU2020304001B2 (enExample)
BR (1) BR112021026380A2 (enExample)
CA (1) CA3144600A1 (enExample)
IL (1) IL289198A (enExample)
MA (1) MA56550A (enExample)
MX (2) MX2022000069A (enExample)
WO (1) WO2020263847A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4484431A3 (en) * 2019-06-24 2025-03-26 Naurex Inc. Processes and intermediates for producing diazaspiro lactam compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0323204D0 (en) * 2003-10-03 2003-11-05 Novartis Ag Organic compounds
ES2416354T3 (es) * 2005-06-21 2013-07-31 Ajinomoto Co., Inc. Cristal de derivado de fenilalanina, método de producción del mismo y uso del mismo
BRPI0918868B8 (pt) * 2008-09-18 2021-05-25 Naurex Inc compostos moduladores do receptor de nmda e composições compreendendo os mesmos
US9758525B2 (en) * 2013-01-29 2017-09-12 Aptinyx Inc. Spiro-lactam NMDA receptor modulators and uses thereof
PE20151416A1 (es) * 2013-01-29 2015-10-10 Naurex Inc Moduladores de receptores nmda de espiro-lactama y sus usos
DK3436463T3 (da) * 2016-03-28 2021-08-30 Takeda Pharmaceuticals Co Krystalline former af 2-[(2s)-1-azabicyclo[2.2.2]oct-2-yl]-6-(3-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-on hemi-hydrat
PE20190174A1 (es) 2016-05-19 2019-02-01 Aptinyx Inc Moduladores del receptor espiro-lactama n-metil-d-aspartato y usos de los mismos
EP4484431A3 (en) * 2019-06-24 2025-03-26 Naurex Inc. Processes and intermediates for producing diazaspiro lactam compounds

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