JP2022536655A5 - - Google Patents

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Publication number
JP2022536655A5
JP2022536655A5 JP2021573245A JP2021573245A JP2022536655A5 JP 2022536655 A5 JP2022536655 A5 JP 2022536655A5 JP 2021573245 A JP2021573245 A JP 2021573245A JP 2021573245 A JP2021573245 A JP 2021573245A JP 2022536655 A5 JP2022536655 A5 JP 2022536655A5
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JP
Japan
Prior art keywords
inventions described
inventions
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JP2021573245A
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English (en)
Japanese (ja)
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JP2022536655A (ja
JP7765972B2 (ja
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Priority claimed from PCT/US2020/037233 external-priority patent/WO2020252165A1/en
Publication of JP2022536655A publication Critical patent/JP2022536655A/ja
Publication of JP2022536655A5 publication Critical patent/JP2022536655A5/ja
Application granted granted Critical
Publication of JP7765972B2 publication Critical patent/JP7765972B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021573245A 2019-06-11 2020-06-11 キナゾリニル化合物及び使用方法 Active JP7765972B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2019090714 2019-06-11
CNPCT/CN2019/090714 2019-06-11
PCT/US2020/037233 WO2020252165A1 (en) 2019-06-11 2020-06-11 Quinazolinyl compounds and methods of use

Publications (3)

Publication Number Publication Date
JP2022536655A JP2022536655A (ja) 2022-08-18
JP2022536655A5 true JP2022536655A5 (https=) 2023-06-19
JP7765972B2 JP7765972B2 (ja) 2025-11-07

Family

ID=71409497

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021573245A Active JP7765972B2 (ja) 2019-06-11 2020-06-11 キナゾリニル化合物及び使用方法

Country Status (5)

Country Link
US (1) US20220249487A1 (https=)
EP (1) EP3983400B1 (https=)
JP (1) JP7765972B2 (https=)
CN (1) CN114302877A (https=)
WO (1) WO2020252165A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11840523B2 (en) * 2020-11-13 2023-12-12 The Regents Of The University Of California IRE1α inhibitors and uses thereof
IL302807A (en) 2020-11-18 2023-07-01 Deciphera Pharmaceuticals Llc Gcn2 and perk kinase inhibitors and methods of use thereof
PE20250609A1 (es) 2021-12-03 2025-02-26 Deciphera Pharmaceuticals Llc Inhibidores de gcn2 y perk quinasa y metodos de uso de los mismos
WO2024131893A1 (en) * 2022-12-22 2024-06-27 Shanghai Yi Zhong Xing Biotechnology Co., Ltd. IRE1α SMALL MOLECULE INHIBITORS

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3773919A (en) 1969-10-23 1973-11-20 Du Pont Polylactide-drug mixtures
US5543523A (en) 1994-11-15 1996-08-06 Regents Of The University Of Minnesota Method and intermediates for the synthesis of korupensamines
CA2564355C (en) 2004-05-07 2012-07-03 Amgen Inc. Protein kinase modulators and method of use
US20070054916A1 (en) * 2004-10-01 2007-03-08 Amgen Inc. Aryl nitrogen-containing bicyclic compounds and methods of use
US7868177B2 (en) 2006-02-24 2011-01-11 Amgen Inc. Multi-cyclic compounds and method of use
CN104230901A (zh) 2008-09-15 2014-12-24 加利福尼亚大学董事会 用于调节ire1、src和abl活性的方法和组合物
WO2016004254A1 (en) * 2014-07-01 2016-01-07 The Regents Of The University Of California Combined modulation of ire1
EP3548476A4 (en) * 2016-12-02 2020-05-20 Quentis Therapeutics, Inc. SMALL MOLECULAR IRE1 INHIBITORS
JP7126084B2 (ja) * 2017-06-01 2022-08-26 コーネル ユニバーシティー Ire1小分子阻害薬
WO2018222917A1 (en) * 2017-06-01 2018-12-06 Quentis Therapeutics, Inc. Ire1 small molecule inhibitors
US10392367B2 (en) * 2017-06-01 2019-08-27 Quentis Therapeutics, Inc. IRE1 small molecule inhibitors
WO2019094641A1 (en) * 2017-11-10 2019-05-16 Quentis Therapeutics, Inc. Ire1 small molecule inhibitors
US12071426B2 (en) * 2018-12-03 2024-08-27 Cornell University IRE1 small molecule inhibitors

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