JP2022525759A5 - - Google Patents

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Publication number
JP2022525759A5
JP2022525759A5 JP2021555545A JP2021555545A JP2022525759A5 JP 2022525759 A5 JP2022525759 A5 JP 2022525759A5 JP 2021555545 A JP2021555545 A JP 2021555545A JP 2021555545 A JP2021555545 A JP 2021555545A JP 2022525759 A5 JP2022525759 A5 JP 2022525759A5
Authority
JP
Japan
Prior art keywords
powder
crystal morphology
ray diffraction
morphology
angles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021555545A
Other languages
English (en)
Japanese (ja)
Other versions
JP7738482B2 (ja
JP2022525759A (ja
Filing date
Publication date
Priority claimed from PCT/CN2019/081985 external-priority patent/WO2020206623A1/en
Application filed filed Critical
Publication of JP2022525759A publication Critical patent/JP2022525759A/ja
Publication of JP2022525759A5 publication Critical patent/JP2022525759A5/ja
Priority to JP2025144862A priority Critical patent/JP2026004294A/ja
Application granted granted Critical
Publication of JP7738482B2 publication Critical patent/JP7738482B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021555545A 2019-04-10 2020-04-10 ピリダジノンtrpc阻害剤の結晶形態 Active JP7738482B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025144862A JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2019/081985 2019-04-10
PCT/CN2019/081985 WO2020206623A1 (en) 2019-04-10 2019-04-10 Crystal forms
PCT/US2020/027689 WO2020210639A1 (en) 2019-04-10 2020-04-10 Crystal forms of a pyridazinone trpc inhibitor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025144862A Division JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Publications (3)

Publication Number Publication Date
JP2022525759A JP2022525759A (ja) 2022-05-19
JP2022525759A5 true JP2022525759A5 (cg-RX-API-DMAC7.html) 2023-07-07
JP7738482B2 JP7738482B2 (ja) 2025-09-12

Family

ID=70482847

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021555545A Active JP7738482B2 (ja) 2019-04-10 2020-04-10 ピリダジノンtrpc阻害剤の結晶形態
JP2025144862A Pending JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025144862A Pending JP2026004294A (ja) 2019-04-10 2025-09-01 ピリダジノンtrpc阻害剤の結晶形態

Country Status (10)

Country Link
US (1) US12655132B2 (cg-RX-API-DMAC7.html)
EP (1) EP3953352A1 (cg-RX-API-DMAC7.html)
JP (2) JP7738482B2 (cg-RX-API-DMAC7.html)
CN (2) CN114502552B (cg-RX-API-DMAC7.html)
AU (2) AU2020272030C1 (cg-RX-API-DMAC7.html)
BR (1) BR112021018221A2 (cg-RX-API-DMAC7.html)
CA (1) CA3136652A1 (cg-RX-API-DMAC7.html)
MA (1) MA55614A (cg-RX-API-DMAC7.html)
MX (2) MX2021012313A (cg-RX-API-DMAC7.html)
WO (2) WO2020206623A1 (cg-RX-API-DMAC7.html)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12435078B2 (en) 2017-09-18 2025-10-07 Gfb (Abc), Llc Pyridazinones and methods of use thereof
LT3852533T (lt) * 2018-09-18 2024-06-10 Gfb (Abc), Llc Piridazinonai ir jų naudojimo būdai
WO2020206623A1 (en) 2019-04-10 2020-10-15 Goldfinch Bio, Inc. Crystal forms
CA3136632A1 (en) 2019-04-11 2020-10-15 Goldfinch Bio, Inc. Spray-dried formulation of a pyridazinone trpc5 inhibitor
AU2020357178A1 (en) * 2019-10-04 2022-05-12 Gfb (Abc), Llc Biomarker-based treatment of focal segmental glomerulosclerosis and diabetic kidney disease
KR102873922B1 (ko) 2020-07-03 2025-10-20 우한 크리에이터나 사이언스 앤드 테크놀로지 컴퍼니, 리미티드 헤테로고리 화합물 및 이의 용도
JP7701559B2 (ja) * 2021-09-10 2025-07-01 メッドシャイン ディスカバリー インコーポレイテッド ハロゲン置換のピリダジノン系化合物及びその使用
EP4470540A4 (en) * 2022-01-27 2025-06-11 Wuhan Createrna Science and Technology Co.,Ltd. USE OF A HETEROCYCLIC COMPOUND
CN119546303A (zh) * 2022-08-05 2025-02-28 武汉朗来科技发展有限公司 包含杂环化合物的药物组合物及其制备方法和应用
WO2025250920A1 (en) 2024-05-31 2025-12-04 Gfb (Abc), Llc Pyridazinone phosphate compounds, pharmaceutical compositions, and medical uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP310798A0 (en) * 1998-04-22 1998-05-14 Soltec Research Pty Ltd Vehicle system for a composition comprising a piperidinopyrimidine derivative
US8633233B2 (en) * 2008-08-06 2014-01-21 Hydra Biosciences, Inc. Methods and compositions for treating anxiety
EP3180340B1 (en) * 2014-08-11 2018-10-10 Hydra Biosciences, Inc. Pyrido[2,3-d]pyrimidine-2,4(1h,3h)-dione derivatives
US12435078B2 (en) * 2017-09-18 2025-10-07 Gfb (Abc), Llc Pyridazinones and methods of use thereof
LT3852533T (lt) 2018-09-18 2024-06-10 Gfb (Abc), Llc Piridazinonai ir jų naudojimo būdai
WO2020206623A1 (en) 2019-04-10 2020-10-15 Goldfinch Bio, Inc. Crystal forms
KR102873922B1 (ko) 2020-07-03 2025-10-20 우한 크리에이터나 사이언스 앤드 테크놀로지 컴퍼니, 리미티드 헤테로고리 화합물 및 이의 용도

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