JP2022516631A5 - - Google Patents

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Publication number
JP2022516631A5
JP2022516631A5 JP2021538743A JP2021538743A JP2022516631A5 JP 2022516631 A5 JP2022516631 A5 JP 2022516631A5 JP 2021538743 A JP2021538743 A JP 2021538743A JP 2021538743 A JP2021538743 A JP 2021538743A JP 2022516631 A5 JP2022516631 A5 JP 2022516631A5
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JP
Japan
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alkyl
independently
disease
substituted
optionally
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JP2021538743A
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English (en)
Japanese (ja)
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JP7566753B2 (ja
JP2022516631A (ja
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Priority claimed from PCT/US2020/012268 external-priority patent/WO2020142748A1/en
Publication of JP2022516631A publication Critical patent/JP2022516631A/ja
Publication of JP2022516631A5 publication Critical patent/JP2022516631A5/ja
Application granted granted Critical
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JP2021538743A 2019-01-03 2020-01-03 転写因子ebポリペプチドレベルを増加させるための方法および材料 Active JP7566753B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962788049P 2019-01-03 2019-01-03
US62/788,049 2019-01-03
US201962879374P 2019-07-26 2019-07-26
US62/879,374 2019-07-26
PCT/US2020/012268 WO2020142748A1 (en) 2019-01-03 2020-01-03 Methods and materials for increasing transcription factor eb polypeptide levels

Publications (3)

Publication Number Publication Date
JP2022516631A JP2022516631A (ja) 2022-03-01
JP2022516631A5 true JP2022516631A5 (enExample) 2023-01-06
JP7566753B2 JP7566753B2 (ja) 2024-10-15

Family

ID=71406977

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021538743A Active JP7566753B2 (ja) 2019-01-03 2020-01-03 転写因子ebポリペプチドレベルを増加させるための方法および材料

Country Status (12)

Country Link
US (2) US12286442B2 (enExample)
EP (1) EP3906033A4 (enExample)
JP (1) JP7566753B2 (enExample)
KR (1) KR102904932B1 (enExample)
CN (1) CN113316453B (enExample)
AU (1) AU2020204717B2 (enExample)
BR (1) BR112021012950A2 (enExample)
CA (1) CA3123902A1 (enExample)
IL (1) IL284403A (enExample)
MX (1) MX2021008152A (enExample)
SG (1) SG11202105685TA (enExample)
WO (1) WO2020142748A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022013684A1 (en) 2020-07-11 2022-01-20 Pfizer Inc. Antiviral heteroaryl ketone derivatives
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds
CZ309449B6 (cs) * 2020-12-24 2023-01-25 Ústav experimentální botaniky AV ČR, v. v. i. Chinazolinové deriváty jako selektivní inhibitory cyklooxygenázy-1
CN113248518B (zh) * 2021-06-21 2022-03-25 山东大学 嘧啶哌嗪类衍生物及其制备方法与应用
WO2025026988A1 (en) * 2023-07-28 2025-02-06 Theranexus Mutated tfeb for treating lysosomal disorders
CN119818678A (zh) * 2024-12-24 2025-04-15 广州医科大学附属妇女儿童医疗中心 Tfeb在制备变应性鼻炎的药物中的应用

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US5304121A (en) 1990-12-28 1994-04-19 Boston Scientific Corporation Drug delivery system making use of a hydrogel polymer coating
US5716981A (en) 1993-07-19 1998-02-10 Angiogenesis Technologies, Inc. Anti-angiogenic compositions and methods of use
US6099562A (en) 1996-06-13 2000-08-08 Schneider (Usa) Inc. Drug coating with topcoat
ES2266258T3 (es) 2000-09-15 2007-03-01 Vertex Pharmaceuticals Incorporated Compuestos de pirazol utiles como inhibidores de proteina cinasas.
JP2005503425A (ja) 2001-05-24 2005-02-03 アレックザ モレキュラー デリヴァリー コーポレイション 所定の吸入ルートによる薬剤エステルの送出
US20030158195A1 (en) * 2001-12-21 2003-08-21 Cywin Charles L. 1,6 naphthyridines useful as inhibitors of SYK kinase
WO2004037814A1 (en) * 2002-10-25 2004-05-06 Vertex Pharmaceuticals Incorporated Indazolinone compositions useful as kinase inhibitors
CL2004000409A1 (es) 2003-03-03 2005-01-07 Vertex Pharma Compuestos derivados de 2-(cilo sustituido)-1-(amino u oxi sustituido)-quinazolina, inhibidores de canales ionicos de sodio y calcio dependientes de voltaje; composicion farmaceutica; y uso del compuesto en el tratamiento de dolor agudo, cronico, neu
US7198926B2 (en) 2003-05-08 2007-04-03 E. I. Du Pont De Nemours And Company Preparation of (E)- and (Z)-2-methyl-2-butenoic acids
WO2004101512A2 (en) * 2003-05-13 2004-11-25 Smithkline Beecham Corporation Naphthyridine integrase inhibitors
US20090209536A1 (en) * 2007-06-17 2009-08-20 Kalypsys, Inc. Aminoquinazoline cannabinoid receptor modulators for treatment of disease
CN101917999A (zh) * 2007-11-07 2010-12-15 弗尔德里克斯制药股份有限公司 蛋白质运输的调节
WO2010015520A1 (de) 2008-08-05 2010-02-11 Boehringer Ingelheim International Gmbh Substituierte naphthyridine und ihre verwendung als arzneimittel
EP2313406B1 (de) * 2008-08-05 2015-02-25 Boehringer Ingelheim International GmbH 4-dimethylaminophenyl-substituierte napththyridine und ihre verwendung als arzneimittel
GB201007203D0 (en) * 2010-04-29 2010-06-16 Glaxo Group Ltd Novel compounds
GB201007347D0 (en) * 2010-04-30 2010-06-16 Karus Therapeutics Ltd Compounds
EP2922540A1 (en) 2012-11-20 2015-09-30 F. Hoffmann-La Roche AG Substituted 1,6-naphthyridines
US20170354666A1 (en) * 2014-11-19 2017-12-14 Rush University Medical Center Compositions and methods for treating lysosomal disorders
WO2018089499A1 (en) 2016-11-08 2018-05-17 Navitor Pharmaceuticals, Inc. PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF
WO2018089493A1 (en) 2016-11-08 2018-05-17 Navitor Pharmaceuticals, Inc. PYRROLE mTORC INHIBITORS AND USES THEREOF
WO2018089433A1 (en) * 2016-11-08 2018-05-17 Navitor Pharmaceuticals, Inc. PHENYL mTORC INHIBITORS AND USES THEREOF
WO2018191146A1 (en) 2017-04-10 2018-10-18 Navitor Pharmaceuticals, Inc. Heteroaryl rheb inhibitors and uses thereof

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