JP2022501370A5 - - Google Patents

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Publication number
JP2022501370A5
JP2022501370A5 JP2021515492A JP2021515492A JP2022501370A5 JP 2022501370 A5 JP2022501370 A5 JP 2022501370A5 JP 2021515492 A JP2021515492 A JP 2021515492A JP 2021515492 A JP2021515492 A JP 2021515492A JP 2022501370 A5 JP2022501370 A5 JP 2022501370A5
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JP
Japan
Prior art keywords
alkyl
compound
hydrogen
cycloalkyl
group
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021515492A
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English (en)
Japanese (ja)
Other versions
JP7433303B2 (ja
JP2022501370A (ja
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Application filed filed Critical
Priority claimed from PCT/IB2019/057814 external-priority patent/WO2020058844A1/en
Publication of JP2022501370A publication Critical patent/JP2022501370A/ja
Publication of JP2022501370A5 publication Critical patent/JP2022501370A5/ja
Application granted granted Critical
Publication of JP7433303B2 publication Critical patent/JP7433303B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021515492A 2018-09-20 2019-09-17 ヒト免疫不全ウイルス複製の阻害剤 Active JP7433303B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862733692P 2018-09-20 2018-09-20
US62/733,692 2018-09-20
PCT/IB2019/057814 WO2020058844A1 (en) 2018-09-20 2019-09-17 Inhibitors of human immunodeficiency virus replication

Publications (3)

Publication Number Publication Date
JP2022501370A JP2022501370A (ja) 2022-01-06
JP2022501370A5 true JP2022501370A5 (https=) 2022-09-05
JP7433303B2 JP7433303B2 (ja) 2024-02-19

Family

ID=68000004

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021515492A Active JP7433303B2 (ja) 2018-09-20 2019-09-17 ヒト免疫不全ウイルス複製の阻害剤

Country Status (4)

Country Link
US (1) US11919897B2 (https=)
EP (1) EP3853228A1 (https=)
JP (1) JP7433303B2 (https=)
WO (1) WO2020058844A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2971987T3 (es) * 2018-10-24 2024-06-10 Viiv Healthcare Uk No 5 Ltd Inhibidores de la replicación del virus de inmunodeficiencia humana
US11541055B2 (en) 2018-10-24 2023-01-03 VIIV Healthcare UK (No.5) Limited Inhibitors of human immunodeficiency virus replication
EP3873607B1 (en) * 2018-10-29 2023-11-29 VIIV Healthcare UK (No.5) Limited Quinazolinyl-indazole derivatives and their use as inhibitors of human immunodeficiency virus replication
EP3914604B1 (en) 2019-01-25 2026-03-04 Brown University Compositions comprising censavudine or elvucitabine for treating age-associated inflammation and disorders
TW202128648A (zh) * 2019-10-04 2021-08-01 英商Viiv醫療保健英國(No 5)有限公司 人類免疫不全病毒複製之抑制劑
EP4066839A4 (en) 2019-11-28 2023-12-27 Shionogi & Co., Ltd PROPHYLACTIC AND THERAPEUTIC MEDICINAL PRODUCT FOR HIV INFECTIOUS DISEASES, CHARACTERIZED BY CONTAINING THE COMBINATION OF INTEGRAS INHIBITORS AND ANTI-HIV AGENTS
KR20220151655A (ko) * 2020-03-06 2022-11-15 비브 헬스케어 유케이 (넘버5) 리미티드 인간 면역결핍 바이러스 복제의 억제제
BR112022020933A2 (pt) * 2020-04-15 2022-12-06 Viiv Healthcare Uk No 5 Ltd Inibidores de replicação do vírus da imunodeficiência humana
US20250042926A1 (en) * 2023-05-31 2025-02-06 Gilead Sciences, Inc. Therapeutic compounds for hiv
CN121335877A (zh) 2023-06-15 2026-01-13 Viiv保健英国第五有限公司 用于制备化合物的方法和中间体
TW202547514A (zh) 2024-02-05 2025-12-16 英商Viiv醫療保健英國(No 5)有限公司 人類免疫不全病毒複製之抑制劑

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008546843A (ja) * 2005-06-27 2008-12-25 アムゲン インコーポレイティッド 抗炎症性アリールニトリル化合物
CN102464654B (zh) 2010-11-12 2016-01-13 上海泓博智源医药技术有限公司 抗病毒化合物
AU2012278976B2 (en) 2011-07-06 2017-05-11 Gilead Sciences, Inc. Compounds for the treatment of HIV
CN102863512B (zh) 2011-07-07 2016-04-20 上海泓博智源医药技术有限公司 抗病毒化合物
ES2642265T3 (es) 2013-01-09 2017-11-16 Gilead Sciences, Inc. Compuestos terapéuticos para el tratamiento de infecciones virales
TW201443037A (zh) 2013-01-09 2014-11-16 Gilead Sciences Inc 治療用化合物
US9220710B2 (en) 2013-01-09 2015-12-29 Gilead Sciences, Inc. Therapeutic compounds
TWI694071B (zh) 2013-03-01 2020-05-21 美商基利科學股份有限公司 治療反轉錄病毒科(Retroviridae)病毒感染之治療性化合物
WO2015130966A1 (en) 2014-02-28 2015-09-03 Gilead Sciences, Inc. Antiviral agents
US10202353B2 (en) 2014-02-28 2019-02-12 Gilead Sciences, Inc. Therapeutic compounds
EP3186239B1 (en) 2014-08-29 2018-10-10 Gilead Sciences, Inc. Antiretroviral agents
CN119462611A (zh) 2016-08-19 2025-02-18 吉利德科学公司 用于预防性或治疗性治疗hiv病毒感染的治疗性化合物
TW201906834A (zh) 2017-05-02 2019-02-16 英商Viiv醫療保健英國(No.5)有限公司 人類免疫不全病毒複製之抑制劑
JP7083398B2 (ja) 2018-02-15 2022-06-10 ギリアード サイエンシーズ, インコーポレイテッド ピリジン誘導体およびhiv感染を処置するためのその使用
EP3752496B1 (en) 2018-02-16 2023-07-05 Gilead Sciences, Inc. Methods and intermediates for preparing a therapeutic compound useful in the treatment of retroviridae viral infection

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