JP2022501370A5 - - Google Patents

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Publication number
JP2022501370A5
JP2022501370A5 JP2021515492A JP2021515492A JP2022501370A5 JP 2022501370 A5 JP2022501370 A5 JP 2022501370A5 JP 2021515492 A JP2021515492 A JP 2021515492A JP 2021515492 A JP2021515492 A JP 2021515492A JP 2022501370 A5 JP2022501370 A5 JP 2022501370A5
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JP
Japan
Prior art keywords
alkyl
compound
hydrogen
cycloalkyl
group
Prior art date
Application number
JP2021515492A
Other languages
English (en)
Japanese (ja)
Other versions
JP7433303B2 (ja
JP2022501370A (ja
JPWO2020058844A5 (https=
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Priority claimed from PCT/IB2019/057814 external-priority patent/WO2020058844A1/en
Publication of JP2022501370A publication Critical patent/JP2022501370A/ja
Publication of JPWO2020058844A5 publication Critical patent/JPWO2020058844A5/ja
Publication of JP2022501370A5 publication Critical patent/JP2022501370A5/ja
Application granted granted Critical
Publication of JP7433303B2 publication Critical patent/JP7433303B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021515492A 2018-09-20 2019-09-17 ヒト免疫不全ウイルス複製の阻害剤 Active JP7433303B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862733692P 2018-09-20 2018-09-20
US62/733,692 2018-09-20
PCT/IB2019/057814 WO2020058844A1 (en) 2018-09-20 2019-09-17 Inhibitors of human immunodeficiency virus replication

Publications (4)

Publication Number Publication Date
JP2022501370A JP2022501370A (ja) 2022-01-06
JPWO2020058844A5 JPWO2020058844A5 (https=) 2022-09-05
JP2022501370A5 true JP2022501370A5 (https=) 2022-09-05
JP7433303B2 JP7433303B2 (ja) 2024-02-19

Family

ID=68000004

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021515492A Active JP7433303B2 (ja) 2018-09-20 2019-09-17 ヒト免疫不全ウイルス複製の阻害剤

Country Status (4)

Country Link
US (1) US11919897B2 (https=)
EP (1) EP3853228A1 (https=)
JP (1) JP7433303B2 (https=)
WO (1) WO2020058844A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2021004593A (es) 2018-10-24 2021-06-15 Viiv Healthcare Uk No 5 Ltd Inhibidores de la replicacion del virus de la inmunodeficiencia humana.
US20210395262A1 (en) * 2018-10-24 2021-12-23 VIIV Healthcare UK (No.5) Limited Inhibitors of human immunodeficiency virus replication
EP3873607B1 (en) * 2018-10-29 2023-11-29 VIIV Healthcare UK (No.5) Limited Quinazolinyl-indazole derivatives and their use as inhibitors of human immunodeficiency virus replication
SG11202107145SA (en) 2019-01-25 2021-08-30 Univ Brown Compositions and methods for treating, preventing or reversing age-associated inflammation and disorders
TW202128648A (zh) * 2019-10-04 2021-08-01 英商Viiv醫療保健英國(No 5)有限公司 人類免疫不全病毒複製之抑制劑
TWI902729B (zh) 2019-11-28 2025-11-01 日商鹽野義製藥股份有限公司 以組合整合酶阻礙劑及抗hiv藥為特徵之hiv感染症的預防及治療用醫藥
KR20220151655A (ko) * 2020-03-06 2022-11-15 비브 헬스케어 유케이 (넘버5) 리미티드 인간 면역결핍 바이러스 복제의 억제제
CN115397424A (zh) * 2020-04-15 2022-11-25 Viiv保健英国第五有限公司 人类免疫缺陷病毒复制的抑制剂
US20250042926A1 (en) * 2023-05-31 2025-02-06 Gilead Sciences, Inc. Therapeutic compounds for hiv
AR132951A1 (es) 2023-06-15 2025-08-13 Viiv Healthcare Uk No 5 Ltd Métodos e intermedios para preparar compuestos
US12594276B2 (en) 2024-02-05 2026-04-07 Viiv Healthcare Uk (No. 5) Limited Inhibitors of human immunodeficiency virus replication

Family Cites Families (15)

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CA2612585A1 (en) 2005-06-27 2007-01-04 Amgen Inc. Anti-inflammatory aryl nitrile compounds
CN102464654B (zh) 2010-11-12 2016-01-13 上海泓博智源医药技术有限公司 抗病毒化合物
EP2729448B1 (en) 2011-07-06 2015-09-09 Gilead Sciences, Inc. Compounds for the treatment of hiv
CN102863512B (zh) 2011-07-07 2016-04-20 上海泓博智源医药技术有限公司 抗病毒化合物
CA2897268C (en) 2013-01-09 2018-12-04 Gilead Sciences, Inc. Therapeutic compounds for the treatment of viral infections
TW201443037A (zh) 2013-01-09 2014-11-16 Gilead Sciences Inc 治療用化合物
CA2896244C (en) 2013-01-09 2017-07-04 Gilead Sciences, Inc. 5-membered heteroaryls and their use as antiviral agents
TWI694071B (zh) 2013-03-01 2020-05-21 美商基利科學股份有限公司 治療反轉錄病毒科(Retroviridae)病毒感染之治療性化合物
WO2015130964A1 (en) 2014-02-28 2015-09-03 Gilead Sciences, Inc. Therapeutic compounds
WO2015130966A1 (en) 2014-02-28 2015-09-03 Gilead Sciences, Inc. Antiviral agents
PT3186239T (pt) 2014-08-29 2019-01-10 Gilead Sciences Inc Agentes antirretrovirais
KR20230011471A (ko) 2016-08-19 2023-01-20 길리애드 사이언시즈, 인코포레이티드 Hiv 바이러스 감염의 예방적 또는 치유적 치료에 유용한 치료 화합물
TW201906834A (zh) 2017-05-02 2019-02-16 英商Viiv醫療保健英國(No.5)有限公司 人類免疫不全病毒複製之抑制劑
US10836746B2 (en) 2018-02-15 2020-11-17 Gilead Sciences, Inc. Therapeutic compounds
WO2019161280A1 (en) 2018-02-16 2019-08-22 Gilead Sciences, Inc. Methods and intermediates for preparing a therapeutic compound useful in the treatment of retroviridae viral infection

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