JP2022500425A5 - - Google Patents

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Publication number
JP2022500425A5
JP2022500425A5 JP2021514019A JP2021514019A JP2022500425A5 JP 2022500425 A5 JP2022500425 A5 JP 2022500425A5 JP 2021514019 A JP2021514019 A JP 2021514019A JP 2021514019 A JP2021514019 A JP 2021514019A JP 2022500425 A5 JP2022500425 A5 JP 2022500425A5
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JP
Japan
Prior art keywords
compound
alkyl
hydrogen
salt according
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021514019A
Other languages
English (en)
Japanese (ja)
Other versions
JP7361766B2 (ja
JP2022500425A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2019/057710 external-priority patent/WO2020053811A1/en
Publication of JP2022500425A publication Critical patent/JP2022500425A/ja
Publication of JP2022500425A5 publication Critical patent/JP2022500425A5/ja
Application granted granted Critical
Publication of JP7361766B2 publication Critical patent/JP7361766B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021514019A 2018-09-14 2019-09-12 ヒト免疫不全ウイルス複製の阻害剤 Active JP7361766B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862731196P 2018-09-14 2018-09-14
US62/731,196 2018-09-14
US201862733259P 2018-09-19 2018-09-19
US62/733,259 2018-09-19
PCT/IB2019/057710 WO2020053811A1 (en) 2018-09-14 2019-09-12 Inhibitors of human immunodeficiency virus replication

Publications (3)

Publication Number Publication Date
JP2022500425A JP2022500425A (ja) 2022-01-04
JP2022500425A5 true JP2022500425A5 (https=) 2022-08-09
JP7361766B2 JP7361766B2 (ja) 2023-10-16

Family

ID=68240777

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021514019A Active JP7361766B2 (ja) 2018-09-14 2019-09-12 ヒト免疫不全ウイルス複製の阻害剤

Country Status (4)

Country Link
US (1) US20220089598A1 (https=)
EP (1) EP3849982A1 (https=)
JP (1) JP7361766B2 (https=)
WO (1) WO2020053811A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2971987T3 (es) * 2018-10-24 2024-06-10 Viiv Healthcare Uk No 5 Ltd Inhibidores de la replicación del virus de inmunodeficiencia humana
US11541055B2 (en) 2018-10-24 2023-01-03 VIIV Healthcare UK (No.5) Limited Inhibitors of human immunodeficiency virus replication
EP3873607B1 (en) * 2018-10-29 2023-11-29 VIIV Healthcare UK (No.5) Limited Quinazolinyl-indazole derivatives and their use as inhibitors of human immunodeficiency virus replication
EP3914604B1 (en) 2019-01-25 2026-03-04 Brown University Compositions comprising censavudine or elvucitabine for treating age-associated inflammation and disorders
TW202128648A (zh) * 2019-10-04 2021-08-01 英商Viiv醫療保健英國(No 5)有限公司 人類免疫不全病毒複製之抑制劑
US20220370451A1 (en) * 2019-10-08 2022-11-24 VIIV HEALTHCARE UK ( No. 5) LIMITED Inhibitors of human immunodeficiency virus replication
EP4066839A4 (en) 2019-11-28 2023-12-27 Shionogi & Co., Ltd PROPHYLACTIC AND THERAPEUTIC MEDICINAL PRODUCT FOR HIV INFECTIOUS DISEASES, CHARACTERIZED BY CONTAINING THE COMBINATION OF INTEGRAS INHIBITORS AND ANTI-HIV AGENTS
WO2024175044A2 (en) * 2023-02-23 2024-08-29 Ascletis Bioscience Co., Ltd. Inhibitors of human immunodeficiency virus replication, method of making and method of using thereof
US20250042926A1 (en) 2023-05-31 2025-02-06 Gilead Sciences, Inc. Therapeutic compounds for hiv
CN121335877A (zh) 2023-06-15 2026-01-13 Viiv保健英国第五有限公司 用于制备化合物的方法和中间体
TW202547514A (zh) 2024-02-05 2025-12-16 英商Viiv醫療保健英國(No 5)有限公司 人類免疫不全病毒複製之抑制劑

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102464654B (zh) 2010-11-12 2016-01-13 上海泓博智源医药技术有限公司 抗病毒化合物
AU2012278976B2 (en) 2011-07-06 2017-05-11 Gilead Sciences, Inc. Compounds for the treatment of HIV
CN102863512B (zh) 2011-07-07 2016-04-20 上海泓博智源医药技术有限公司 抗病毒化合物
ES2642265T3 (es) 2013-01-09 2017-11-16 Gilead Sciences, Inc. Compuestos terapéuticos para el tratamiento de infecciones virales
TW201443037A (zh) 2013-01-09 2014-11-16 Gilead Sciences Inc 治療用化合物
US9220710B2 (en) 2013-01-09 2015-12-29 Gilead Sciences, Inc. Therapeutic compounds
TWI694071B (zh) 2013-03-01 2020-05-21 美商基利科學股份有限公司 治療反轉錄病毒科(Retroviridae)病毒感染之治療性化合物
US10202353B2 (en) 2014-02-28 2019-02-12 Gilead Sciences, Inc. Therapeutic compounds
WO2015130966A1 (en) 2014-02-28 2015-09-03 Gilead Sciences, Inc. Antiviral agents
EP3186239B1 (en) 2014-08-29 2018-10-10 Gilead Sciences, Inc. Antiretroviral agents
CN119462611A (zh) 2016-08-19 2025-02-18 吉利德科学公司 用于预防性或治疗性治疗hiv病毒感染的治疗性化合物
TW201906834A (zh) 2017-05-02 2019-02-16 英商Viiv醫療保健英國(No.5)有限公司 人類免疫不全病毒複製之抑制劑
JP7083398B2 (ja) 2018-02-15 2022-06-10 ギリアード サイエンシーズ, インコーポレイテッド ピリジン誘導体およびhiv感染を処置するためのその使用
EP3752496B1 (en) 2018-02-16 2023-07-05 Gilead Sciences, Inc. Methods and intermediates for preparing a therapeutic compound useful in the treatment of retroviridae viral infection
EP3774775B8 (en) 2018-04-11 2023-11-15 VIIV Healthcare UK (No.5) Limited 4-oxo-3,4-dihydroquinazoline compounds as inhibitors of human immunodeficiency virus replication
EP3833436A1 (en) 2018-08-09 2021-06-16 VIIV Healthcare UK (No.5) Limited Inhibitors of human immunodeficiency virus replication

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