JP2021521132A5 - - Google Patents

Info

Publication number
JP2021521132A5
JP2021521132A5 JP2020555192A JP2020555192A JP2021521132A5 JP 2021521132 A5 JP2021521132 A5 JP 2021521132A5 JP 2020555192 A JP2020555192 A JP 2020555192A JP 2020555192 A JP2020555192 A JP 2020555192A JP 2021521132 A5 JP2021521132 A5 JP 2021521132A5
Authority
JP
Japan
Prior art keywords
compound according
amino
prevention
treatment
salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020555192A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021521132A (ja
JP7333336B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2019/058398 external-priority patent/WO2019197244A1/en
Publication of JP2021521132A publication Critical patent/JP2021521132A/ja
Publication of JP2021521132A5 publication Critical patent/JP2021521132A5/ja
Application granted granted Critical
Publication of JP7333336B2 publication Critical patent/JP7333336B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020555192A 2018-04-10 2019-04-03 置換オキソピリジン誘導体 Active JP7333336B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18166490.5 2018-04-10
EP18166490 2018-04-10
PCT/EP2019/058398 WO2019197244A1 (en) 2018-04-10 2019-04-03 A substituted oxopyridine derivative

Publications (3)

Publication Number Publication Date
JP2021521132A JP2021521132A (ja) 2021-08-26
JP2021521132A5 true JP2021521132A5 (https=) 2023-05-16
JP7333336B2 JP7333336B2 (ja) 2023-08-24

Family

ID=61965754

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020555192A Active JP7333336B2 (ja) 2018-04-10 2019-04-03 置換オキソピリジン誘導体

Country Status (17)

Country Link
US (1) US11884660B2 (https=)
EP (1) EP3774796B1 (https=)
JP (1) JP7333336B2 (https=)
KR (1) KR102858566B1 (https=)
CN (1) CN111902414B (https=)
AU (1) AU2019251699B2 (https=)
BR (1) BR112020018237A2 (https=)
CA (1) CA3096480A1 (https=)
DK (1) DK3774796T3 (https=)
ES (1) ES2922533T3 (https=)
IL (1) IL277811B2 (https=)
MX (1) MX2020010635A (https=)
PE (1) PE20210165A1 (https=)
SA (1) SA520420308B1 (https=)
SG (1) SG11202008352YA (https=)
WO (1) WO2019197244A1 (https=)
ZA (1) ZA202006963B (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116874469B (zh) * 2023-09-06 2023-11-10 成都施贝康生物医药科技有限公司 一种氧代吡啶类化合物、中间体及其制备方法和用途
CN116947818B (zh) * 2023-09-18 2023-12-19 成都施贝康生物医药科技有限公司 一种氧代吡啶类化合物、中间体及其制备方法和用途

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7453002B2 (en) 2004-06-15 2008-11-18 Bristol-Myers Squibb Company Five-membered heterocycles useful as serine protease inhibitors
US7429604B2 (en) 2004-06-15 2008-09-30 Bristol Myers Squibb Company Six-membered heterocycles useful as serine protease inhibitors
GB0420722D0 (en) 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
US8163779B2 (en) 2006-12-20 2012-04-24 Takeda San Diego, Inc. Glucokinase activators
WO2014160592A2 (en) 2013-03-27 2014-10-02 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
TWI633089B (zh) 2013-03-28 2018-08-21 拜耳製藥股份有限公司 經取代的酮基吡啶衍生物
CA2918814C (en) 2013-07-23 2021-10-12 Bayer Pharma Aktiengesellschaft Substituted oxopyridine derivatives and use thereof as factor xia/plasma
EP3063150B1 (de) 2013-10-30 2017-11-22 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
CN105829298B (zh) 2014-02-14 2019-02-01 四川海思科制药有限公司 一种吡啶酮或嘧啶酮衍生物、及其制备方法和应用
US10077265B2 (en) 2014-09-24 2018-09-18 Bayer Pharma Aktiengesellschaft Substituted oxopyridine derivatives
US10414731B2 (en) 2014-09-24 2019-09-17 Bayer Pharma Aktiengesellschaft Substituted oxopyridine derivatives
EP3197889B1 (de) 2014-09-24 2018-08-01 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
EP3197891B1 (de) 2014-09-24 2018-11-21 Bayer Pharma Aktiengesellschaft Faktor xia hemmende pyridobenzazepin- und pyridobenzazocin-derivate
CN106687458B (zh) 2014-09-24 2020-10-27 拜耳制药股份公司 取代的氧代吡啶衍生物
EP3197872B1 (de) 2014-09-24 2019-01-30 Bayer Pharma Aktiengesellschaft (2h)-2-oxopyridine als faktor xia-inhibitoren zur behandlung von thrombotischen erkrankungen
CA2979937A1 (en) 2015-03-19 2016-09-22 Bayer Pharma Aktiengesellschaft Oxo-pyridine-derivatives as factor xia inhibitors for the treatment of thrombosis
JO3703B1 (ar) 2015-07-09 2021-01-31 Bayer Pharma AG مشتقات أوكسوبيريدين مستبدلة
EP3344618A1 (de) 2015-09-04 2018-07-11 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
BR112019003557A2 (pt) 2016-08-31 2019-05-21 Jiangsu Hengrui Medicine Co., Ltd. derivados de oxopicolinamida, método de preparação dos mesmos e uso farmacêutico dos mesmos

Similar Documents

Publication Publication Date Title
US11565994B2 (en) Inhibitors of histone lysine specific demethylase (LSD1) and histone deacetylases (HDACS)
JP6518683B2 (ja) 抗真菌化合物の調製方法
JP2021105028A (ja) ヘテロ環式化合物およびそれらの使用
WO2007007919A3 (en) Heterocyclic janus kinase 3 inhibitors
WO2007011833A3 (en) Spiropiperidine beta-secretase inhibitors for the treatment of alzheimer's disease
WO2008030412A3 (en) Spiropiperidine beta-secretase inhibitors for the treatment of alzheimer's disease
WO2006044497A3 (en) Spiropiperidine compounds useful as beta-secretase inhibitors for the treatment of alzhermer’s disease
NO20081482L (no) Delta- og epsilon-krystallformer for imatinibmesylat
JP2012144533A (ja) 転写因子調節化合物およびその使用法
WO2008002244A8 (en) Imidazol-pyrimidine derivatives for treatment of diseases related to glycogen synthase kinase (gsk3)
CN105085428B (zh) 芳杂环类衍生物及其在药物上的应用
WO2008054698A3 (en) Spiropiperidine beta-secretase inhibitors for the treatment of alzheimer's disease
JP2019089811A (ja) 抗真菌化合物の調製方法
JP2011502153A5 (https=)
TW200800957A (en) New compounds
JP2003516987A5 (https=)
CN114072404A (zh) Ret选择性抑制剂及其制备方法和用途
NO20091254L (no) Terapeutiske sammensetninger
WO2007056219A3 (en) [4-(6-halo-7-substituted-2,4-dioxo-1,4-dihydro-2h-quinazolin-3-yl)-phenyl]-5-chloro-thiophen-2-yl-sulfonylureas and forms and methods related thereto
EP2266969A3 (en) 6-(Pyridinyl)-4-pyrimidone derivatives as tau protein kinase 1 inhibitors
JP2021521132A5 (https=)
WO2019224774A1 (en) Heterocyclic amides as rip1 kinase inhibitors
WO2006078576A3 (en) Aminomethyl beta-secretase inhibitors for the treatment of alzheimer's disease
WO2010004221A3 (fr) Utilisation de derives d'indole comme activateurs de nurr-1, pour le traitement de la maladie de parkinson
WO2007058862A3 (en) Imidazolidinone compounds useful as beta-secretase inhibitors for the treatment of alzheimer's disease