JP2021514975A5 - - Google Patents

Info

Publication number
JP2021514975A5
JP2021514975A5 JP2020544823A JP2020544823A JP2021514975A5 JP 2021514975 A5 JP2021514975 A5 JP 2021514975A5 JP 2020544823 A JP2020544823 A JP 2020544823A JP 2020544823 A JP2020544823 A JP 2020544823A JP 2021514975 A5 JP2021514975 A5 JP 2021514975A5
Authority
JP
Japan
Prior art keywords
inhibitor
pharmaceutically acceptable
combination
acceptable salt
bromodomain
Prior art date
Application number
JP2020544823A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021514975A (ja
JPWO2019166928A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2019/051462 external-priority patent/WO2019166928A1/en
Publication of JP2021514975A publication Critical patent/JP2021514975A/ja
Publication of JP2021514975A5 publication Critical patent/JP2021514975A5/ja
Publication of JPWO2019166928A5 publication Critical patent/JPWO2019166928A5/ja
Pending legal-status Critical Current

Links

JP2020544823A 2018-02-27 2019-02-22 サイクリン依存性キナーゼ阻害剤およびbet−ブロモドメイン阻害剤の組合せ Pending JP2021514975A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862635916P 2018-02-27 2018-02-27
US62/635,916 2018-02-27
US201962796223P 2019-01-24 2019-01-24
US62/796,223 2019-01-24
PCT/IB2019/051462 WO2019166928A1 (en) 2018-02-27 2019-02-22 Combination of a cyclin dependent kinase inhibitor and a bet-bromodomain inhibitor

Publications (3)

Publication Number Publication Date
JP2021514975A JP2021514975A (ja) 2021-06-17
JP2021514975A5 true JP2021514975A5 (https=) 2022-03-02
JPWO2019166928A5 JPWO2019166928A5 (https=) 2022-03-02

Family

ID=65904498

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020544823A Pending JP2021514975A (ja) 2018-02-27 2019-02-22 サイクリン依存性キナーゼ阻害剤およびbet−ブロモドメイン阻害剤の組合せ

Country Status (5)

Country Link
US (1) US20200405809A1 (https=)
EP (1) EP3758753A1 (https=)
JP (1) JP2021514975A (https=)
CA (1) CA3092003A1 (https=)
WO (1) WO2019166928A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI841598B (zh) * 2018-09-13 2024-05-11 大陸商恒翼生物醫藥(上海)股份有限公司 用於治療雌激素受體陽性乳癌之組合療法
TW202126638A (zh) * 2019-09-30 2021-07-16 日商協和麒麟股份有限公司 Bet分解劑
CA3166741A1 (en) * 2020-01-09 2021-07-15 Astrazeneca Ab Combination therapy for treating cancer
JP7579564B2 (ja) 2020-10-28 2024-11-08 国立大学法人金沢大学 Rb1陽性癌の治療用医薬組成物及びキット
CN117100868A (zh) * 2023-10-10 2023-11-24 复旦大学 溶瘤单纯疱疹病毒oHSV联合NETosis抑制剂在制备抗肿瘤药物中的应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
WO2000035298A1 (en) 1996-11-27 2000-06-22 Wm. Wrigley Jr. Company Chewing gum containing medicament active agents
ES2251677T3 (es) 2002-01-22 2006-05-01 Warner-Lambert Company Llc 2-(piridin-2-ilamino)-pirido(2,3-d)pirimidin-7-onas.
ATE412650T1 (de) 2003-07-11 2008-11-15 Warner Lambert Co Isethionat salz eines selektiven cdk4 inhibitors
BRPI0716880A2 (pt) 2006-09-08 2013-10-15 Pfizer Prod Inc Síntese de 2-(piridin-2-ilamino)-pirido[2,3-d]pirimidin-7-onas
US9073878B2 (en) * 2012-11-21 2015-07-07 Zenith Epigenetics Corp. Cyclic amines as bromodomain inhibitors
SI2958916T1 (sl) 2013-02-21 2018-11-30 Pfizer Inc. Trdne oblike selektivnih zaviralcev CDK4/6
CA2929652A1 (en) * 2013-11-08 2015-05-14 Dana-Farber Cancer Institute, Inc. Combination therapy for cancer using bromodomain and extra-terminal (bet) protein inhibitors
EP3215135B1 (en) * 2014-11-07 2020-05-13 Tolero Pharmaceuticals, Inc. Methods to target transcriptional control at super-enhancer regions
MX376083B (es) 2015-06-04 2025-03-07 Pfizer Formas de dosificacion solidas de palbociclib.

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