JP2021513982A5 - - Google Patents
Info
- Publication number
- JP2021513982A5 JP2021513982A5 JP2020543562A JP2020543562A JP2021513982A5 JP 2021513982 A5 JP2021513982 A5 JP 2021513982A5 JP 2020543562 A JP2020543562 A JP 2020543562A JP 2020543562 A JP2020543562 A JP 2020543562A JP 2021513982 A5 JP2021513982 A5 JP 2021513982A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- heteroaryl
- compound
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023176793A JP2024009948A (ja) | 2018-02-16 | 2023-10-12 | Ｐ３００／ｃｂｐ ｈａｔ阻害剤及びそれらの使用の方法 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862631596P | 2018-02-16 | 2018-02-16 | |
| US62/631,596 | 2018-02-16 | ||
| US201862758885P | 2018-11-12 | 2018-11-12 | |
| US62/758,885 | 2018-11-12 | ||
| PCT/US2019/018158 WO2019161162A1 (en) | 2018-02-16 | 2019-02-15 | P300/cbp hat inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023176793A Division JP2024009948A (ja) | 2018-02-16 | 2023-10-12 | Ｐ３００／ｃｂｐ ｈａｔ阻害剤及びそれらの使用の方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021513982A JP2021513982A (ja) | 2021-06-03 |
| JP2021513982A5 true JP2021513982A5 (https=) | 2022-02-24 |
| JP7368365B2 JP7368365B2 (ja) | 2023-10-24 |
Family
ID=65685973
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020543562A Active JP7368365B2 (ja) | 2018-02-16 | 2019-02-15 | Ｐ３００／ｃｂｐ ｈａｔ阻害剤及びそれらの使用の方法 |
| JP2023176793A Pending JP2024009948A (ja) | 2018-02-16 | 2023-10-12 | Ｐ３００／ｃｂｐ ｈａｔ阻害剤及びそれらの使用の方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023176793A Pending JP2024009948A (ja) | 2018-02-16 | 2023-10-12 | Ｐ３００／ｃｂｐ ｈａｔ阻害剤及びそれらの使用の方法 |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US11274090B2 (https=) |
| EP (1) | EP3752497B1 (https=) |
| JP (2) | JP7368365B2 (https=) |
| CN (1) | CN112218857B (https=) |
| AU (1) | AU2019220662B2 (https=) |
| CA (1) | CA3091342A1 (https=) |
| DK (1) | DK3752497T3 (https=) |
| ES (1) | ES2989149T3 (https=) |
| FI (1) | FI3752497T3 (https=) |
| HR (1) | HRP20241225T1 (https=) |
| HU (1) | HUE068342T2 (https=) |
| LT (1) | LT3752497T (https=) |
| PL (1) | PL3752497T3 (https=) |
| PT (1) | PT3752497T (https=) |
| RS (1) | RS65966B1 (https=) |
| SI (1) | SI3752497T1 (https=) |
| SM (1) | SMT202400371T1 (https=) |
| TW (1) | TW202000658A (https=) |
| WO (1) | WO2019161162A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019161162A1 (en) * | 2018-02-16 | 2019-08-22 | Constellation Pharmaceuticals, Inc. | P300/cbp hat inhibitors |
| US11414384B2 (en) | 2018-02-16 | 2022-08-16 | Constellation Pharmaceuticals, Inc. | P300/CBP hat inhibitors |
| US20220135538A1 (en) * | 2019-02-27 | 2022-05-05 | Constellation Pharmaceuticals, Inc. | P300/cbp hat inhibitors and methods for their use |
| EP4003342A1 (en) * | 2019-07-29 | 2022-06-01 | Constellation Pharmaceuticals, Inc. | Compounds for use in treating neurological disorders |
| US20220372135A1 (en) | 2019-09-27 | 2022-11-24 | Disc Medicine, Inc. | Methods for treating myelofibrosis and related conditions |
| CN111358951B (zh) * | 2020-03-26 | 2022-06-24 | 上海交通大学医学院附属上海儿童医学中心 | 一种使成熟右心室心肌细胞转变为未成熟心肌细胞的方法 |
| KR20230012539A (ko) | 2020-05-13 | 2023-01-26 | 디스크 메디슨, 인크. | 골수섬유증을 치료하기 위한 항-헤모주벨린 (hjv) 항체 |
| US20240122941A1 (en) * | 2020-12-25 | 2024-04-18 | National Cancer Center | Therapy based on synthetic lethality in swi/snf complex-dysfunction cancer |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5153226A (en) | 1989-08-31 | 1992-10-06 | Warner-Lambert Company | Acat inhibitors for treating hypocholesterolemia |
| AU1615895A (en) * | 1994-03-31 | 1995-10-12 | Bristol-Myers Squibb Company | Imidazole-containing inhibitors of farnesyl protein transferase |
| CA2461094A1 (en) | 2001-09-25 | 2003-04-03 | Sony Corporation | P300 histone acetylase inhibitor |
| TW200306819A (en) * | 2002-01-25 | 2003-12-01 | Vertex Pharma | Indazole compounds useful as protein kinase inhibitors |
| US7244757B2 (en) * | 2004-04-01 | 2007-07-17 | Pfizer Inc | Pyrazole-amine compounds for the treatment of neurodegenerative disorders |
| CA2605110A1 (en) * | 2005-04-20 | 2006-11-02 | Merck & Co., Inc. | Benzothiophene derivatives |
| US8143259B2 (en) | 2008-08-19 | 2012-03-27 | Janssen Pharmaceutica, Nv | Cold menthol receptor antagonists |
| US8785468B2 (en) * | 2009-02-13 | 2014-07-22 | Amgen Inc. | Phenylalanine amide derivatives useful for treating insulin-related diseases and conditions |
| GB201116559D0 (en) | 2011-09-26 | 2011-11-09 | Univ Leuven Kath | Novel viral replication inhibitors |
| EP2791128A4 (en) | 2011-12-16 | 2015-04-22 | Olema Pharmaceuticals Inc | NOVEL BENZOPYRAN COMPOUNDS, COMPOSITIONS AND USES THEREOF |
| CN103172540B (zh) * | 2013-03-18 | 2015-07-01 | 潍坊博创国际生物医药研究院 | 苯甘氨酸类组蛋白去乙酰酶抑制剂及其制备方法和应用 |
| MX2016004570A (es) * | 2013-10-11 | 2016-09-08 | Genentech Inc | Uso de inhibidores del bromodominio de cbp/ep300 para la inmunoterapia del cáncer. |
| WO2016044777A1 (en) | 2014-09-18 | 2016-03-24 | Abbvie Inc. | Hat inhibitors and methods for their use |
| US20160235716A1 (en) | 2014-09-18 | 2016-08-18 | Abbvie Inc. | Spirocyclic hat inhibitors and methods for their use |
| WO2016044771A1 (en) | 2014-09-18 | 2016-03-24 | Abbvie Inc. | Hat inhibitors and methods for their use |
| CA2988421A1 (en) | 2015-06-01 | 2016-12-08 | The Scripps Research Institute | Small molecule analogs of the nemo binding peptide |
| EP3464270B1 (en) * | 2016-05-24 | 2022-02-23 | Genentech, Inc. | Heterocyclic inhibitors of cbp/ep300 and their use in the treatment of cancer |
| WO2019018855A1 (en) * | 2017-07-21 | 2019-01-24 | Kadmon Corporation, Llc | ALPHA PROPELLER PROTEIN KINASE INHIBITORS ("COILED-COIL") ASSOCIATED WITH RHO |
| CN108191748A (zh) * | 2018-01-24 | 2018-06-22 | 齐鲁师范学院 | 一种含芳杂环氨基肟类化合物、制备方法及其用途 |
| WO2019161162A1 (en) * | 2018-02-16 | 2019-08-22 | Constellation Pharmaceuticals, Inc. | P300/cbp hat inhibitors |
| US11414384B2 (en) | 2018-02-16 | 2022-08-16 | Constellation Pharmaceuticals, Inc. | P300/CBP hat inhibitors |
-
2019
- 2019-02-15 WO PCT/US2019/018158 patent/WO2019161162A1/en not_active Ceased
- 2019-02-15 HU HUE19709182A patent/HUE068342T2/hu unknown
- 2019-02-15 CN CN201980025884.7A patent/CN112218857B/zh active Active
- 2019-02-15 PT PT197091820T patent/PT3752497T/pt unknown
- 2019-02-15 TW TW108105099A patent/TW202000658A/zh unknown
- 2019-02-15 US US16/970,169 patent/US11274090B2/en active Active
- 2019-02-15 CA CA3091342A patent/CA3091342A1/en active Pending
- 2019-02-15 RS RS20241037A patent/RS65966B1/sr unknown
- 2019-02-15 DK DK19709182.0T patent/DK3752497T3/da active
- 2019-02-15 ES ES19709182T patent/ES2989149T3/es active Active
- 2019-02-15 SM SM20240371T patent/SMT202400371T1/it unknown
- 2019-02-15 SI SI201930823T patent/SI3752497T1/sl unknown
- 2019-02-15 JP JP2020543562A patent/JP7368365B2/ja active Active
- 2019-02-15 HR HRP20241225TT patent/HRP20241225T1/hr unknown
- 2019-02-15 AU AU2019220662A patent/AU2019220662B2/en active Active
- 2019-02-15 FI FIEP19709182.0T patent/FI3752497T3/fi active
- 2019-02-15 LT LTEPPCT/US2019/018158T patent/LT3752497T/lt unknown
- 2019-02-15 EP EP19709182.0A patent/EP3752497B1/en active Active
- 2019-02-15 PL PL19709182.0T patent/PL3752497T3/pl unknown
-
2023
- 2023-10-12 JP JP2023176793A patent/JP2024009948A/ja active Pending
-
2024
- 2024-08-29 US US18/818,774 patent/US20250230137A1/en active Pending
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