JP2020536944A5 - - Google Patents

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Publication number
JP2020536944A5
JP2020536944A5 JP2020521319A JP2020521319A JP2020536944A5 JP 2020536944 A5 JP2020536944 A5 JP 2020536944A5 JP 2020521319 A JP2020521319 A JP 2020521319A JP 2020521319 A JP2020521319 A JP 2020521319A JP 2020536944 A5 JP2020536944 A5 JP 2020536944A5
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JP
Japan
Prior art keywords
cancer
crystal according
fluorobenzofuran
dioxolo
dione
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020521319A
Other languages
English (en)
Japanese (ja)
Other versions
JP2020536944A (ja
JP7776258B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2018/056083 external-priority patent/WO2019079299A1/en
Publication of JP2020536944A publication Critical patent/JP2020536944A/ja
Priority to JP2023151499A priority Critical patent/JP2024001040A/ja
Publication of JP2020536944A5 publication Critical patent/JP2020536944A5/ja
Application granted granted Critical
Publication of JP7776258B2 publication Critical patent/JP7776258B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020521319A 2017-10-16 2018-10-16 ３－（５－フルオロベンゾフラン－３－イル）－４－（５－メチル－５Ｈ－［１，３］ジオキソロ［４，５－ｆ］インドール－７－イル）ピロール－２，５－ジオンの固体形態 Active JP7776258B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023151499A JP2024001040A (ja) 2017-10-16 2023-09-19 ３－（５－フルオロベンゾフラン－３－イル）－４－（５－メチル－５Ｈ－［１，３］ジオキソロ［４，５－ｆ］インドール－７－イル）ピロール－２，５－ジオンの固体形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762572603P 2017-10-16 2017-10-16
US62/572,603 2017-10-16
PCT/US2018/056083 WO2019079299A1 (en) 2017-10-16 2018-10-16 SOLID FORMS OF 3- (5-FLUOROBENZOFURAN-3-YL) -4- (5-METHYL-5H- [1,3] DIOXOLO [4,5-F] INDOL-7-YL) PYRROLE-2,5-DIONE

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023151499A Division JP2024001040A (ja) 2017-10-16 2023-09-19 ３－（５－フルオロベンゾフラン－３－イル）－４－（５－メチル－５Ｈ－［１，３］ジオキソロ［４，５－ｆ］インドール－７－イル）ピロール－２，５－ジオンの固体形態

Publications (3)

Publication Number Publication Date
JP2020536944A JP2020536944A (ja) 2020-12-17
JP2020536944A5 true JP2020536944A5 (OSRAM) 2025-09-10
JP7776258B2 JP7776258B2 (ja) 2025-11-26

Family

ID=64110166

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020521319A Active JP7776258B2 (ja) 2017-10-16 2018-10-16 ３－（５－フルオロベンゾフラン－３－イル）－４－（５－メチル－５Ｈ－［１，３］ジオキソロ［４，５－ｆ］インドール－７－イル）ピロール－２，５－ジオンの固体形態
JP2023151499A Pending JP2024001040A (ja) 2017-10-16 2023-09-19 ３－（５－フルオロベンゾフラン－３－イル）－４－（５－メチル－５Ｈ－［１，３］ジオキソロ［４，５－ｆ］インドール－７－イル）ピロール－２，５－ジオンの固体形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023151499A Pending JP2024001040A (ja) 2017-10-16 2023-09-19 ３－（５－フルオロベンゾフラン－３－イル）－４－（５－メチル－５Ｈ－［１，３］ジオキソロ［４，５－ｆ］インドール－７－イル）ピロール－２，５－ジオンの固体形態

Country Status (16)

Country Link
US (3) US11407759B2 (OSRAM)
EP (2) EP4740944A2 (OSRAM)
JP (2) JP7776258B2 (OSRAM)
KR (1) KR102891811B1 (OSRAM)
CN (1) CN111315748B (OSRAM)
AU (1) AU2018352384B2 (OSRAM)
CA (1) CA3074037A1 (OSRAM)
DK (1) DK3697794T3 (OSRAM)
ES (1) ES3064009T3 (OSRAM)
FI (1) FI3697794T3 (OSRAM)
IL (1) IL273920B2 (OSRAM)
MX (1) MX2020003431A (OSRAM)
PL (1) PL3697794T3 (OSRAM)
PT (1) PT3697794T (OSRAM)
WO (1) WO2019079299A1 (OSRAM)
ZA (1) ZA202002740B (OSRAM)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2020003431A (es) * 2017-10-16 2020-07-29 Actuate Therapeutics Inc Formas solidas de 3-(5-fluorobenzofuran-3-il)-4-(5-metil-5h-[1,3]d ioxolo[4,5-f]indol-7-il)pirrol- 2,5-diona.
CN112437663A (zh) * 2018-05-17 2021-03-02 开动疗法公司 用β型糖原合酶激酶3抑制剂治疗特发性肺纤维化

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2446269T3 (es) 2006-12-19 2014-03-06 The Board Of Trustees Of The University Of Illinois 3-Benzofuranil-4-indolil-maleimidas como potentes inhibidores de GSK-3 para trastornos neurodegenerativos
FI3665176T3 (fi) 2017-08-11 2024-03-20 Actuate Therapeutics Inc 3-(5-fluoribentsofuran-3-yyli)-4-(5-metyyli-5h-[1,3]dioksolo[4,5-f]indol-7-yyli)pyrroli-2,5-dionin kiinteitä muotoja
MX2020003431A (es) * 2017-10-16 2020-07-29 Actuate Therapeutics Inc Formas solidas de 3-(5-fluorobenzofuran-3-il)-4-(5-metil-5h-[1,3]d ioxolo[4,5-f]indol-7-il)pirrol- 2,5-diona.

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