JP2020531486A5 - - Google Patents

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Publication number
JP2020531486A5
JP2020531486A5 JP2020510096A JP2020510096A JP2020531486A5 JP 2020531486 A5 JP2020531486 A5 JP 2020531486A5 JP 2020510096 A JP2020510096 A JP 2020510096A JP 2020510096 A JP2020510096 A JP 2020510096A JP 2020531486 A5 JP2020531486 A5 JP 2020531486A5
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JP
Japan
Prior art keywords
pyridyl
pyridine
oxo
trifluoromethyl
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020510096A
Other languages
English (en)
Japanese (ja)
Other versions
JP2020531486A (ja
JP7199737B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2018/072788 external-priority patent/WO2019038387A1/en
Publication of JP2020531486A publication Critical patent/JP2020531486A/ja
Publication of JP2020531486A5 publication Critical patent/JP2020531486A5/ja
Priority to JP2022198540A priority Critical patent/JP2023021276A/ja
Application granted granted Critical
Publication of JP7199737B2 publication Critical patent/JP7199737B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020510096A 2017-08-23 2018-08-23 ピリジルピリドン化合物 Active JP7199737B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022198540A JP2023021276A (ja) 2017-08-23 2022-12-13 ピリジルピリドン化合物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP17187544 2017-08-23
EP17187544.6 2017-08-23
PCT/EP2018/072788 WO2019038387A1 (en) 2017-08-23 2018-08-23 PYRIDYLPYRIDONE COMPOUNDS

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022198540A Division JP2023021276A (ja) 2017-08-23 2022-12-13 ピリジルピリドン化合物

Publications (3)

Publication Number Publication Date
JP2020531486A JP2020531486A (ja) 2020-11-05
JP2020531486A5 true JP2020531486A5 (https=) 2022-10-20
JP7199737B2 JP7199737B2 (ja) 2023-01-06

Family

ID=59686881

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020510096A Active JP7199737B2 (ja) 2017-08-23 2018-08-23 ピリジルピリドン化合物
JP2022198540A Pending JP2023021276A (ja) 2017-08-23 2022-12-13 ピリジルピリドン化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2022198540A Pending JP2023021276A (ja) 2017-08-23 2022-12-13 ピリジルピリドン化合物

Country Status (20)

Country Link
US (2) US11219618B2 (https=)
EP (2) EP4056556A1 (https=)
JP (2) JP7199737B2 (https=)
KR (1) KR102730718B1 (https=)
CN (3) CN111094244B (https=)
AU (2) AU2018320416B2 (https=)
CY (1) CY1125138T1 (https=)
DK (1) DK3672941T3 (https=)
ES (1) ES2910839T3 (https=)
HR (1) HRP20220571T1 (https=)
HU (1) HUE058977T2 (https=)
IL (3) IL302356A (https=)
LT (1) LT3672941T (https=)
PL (1) PL3672941T3 (https=)
PT (1) PT3672941T (https=)
RS (1) RS63161B1 (https=)
SI (1) SI3672941T1 (https=)
SM (1) SMT202200183T1 (https=)
TW (2) TW202308996A (https=)
WO (1) WO2019038387A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11919902B2 (en) 2017-12-22 2024-03-05 Hibercell, Inc. Aryl-bipyridine amine derivatives as phosphatidylinositol phosphate kinase inhibitors
CA3199999A1 (en) 2020-11-25 2022-06-02 Deciphera Pharmaceuticals, Llc Morpholino derivatives as vsp34 inhibitors for use in the treatment of a viral infection
US11801238B2 (en) 2020-11-25 2023-10-31 Deciphera Pharmaceuticals, Llc Anti-viral activity of VPS34 inhibitors
WO2023019259A1 (en) * 2021-08-13 2023-02-16 Deciphera Pharmaceuticals, Llc Combination therapy of vps34 inhibitors and sting agonist for use in the treatment of cancer

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4606161B2 (ja) * 2002-05-21 2011-01-05 アムジエン・インコーポレーテツド 置換複素環式化合物および使用方法
TW200908984A (en) * 2007-08-07 2009-03-01 Piramal Life Sciences Ltd Pyridyl derivatives, their preparation and use
WO2012085815A1 (en) 2010-12-21 2012-06-28 Novartis Ag Bi-heteroaryl compounds as vps34 inhibitors
DK2655375T3 (en) 2010-12-23 2015-03-09 Sanofi Sa PYRIMIDINON DERIVATIVES, PREPARATION AND PHARMACEUTICAL USE THEREOF
GB201120317D0 (en) 2011-11-24 2012-01-04 Queen Mary & Westfield College Screening method
DK2820009T3 (en) * 2012-03-01 2018-04-16 Array Biopharma Inc Serine / threonine kinase inhibitors
AU2012382373A1 (en) * 2012-06-12 2014-12-11 Abbvie Inc. Pyridinone and pyridazinone derivatives
FR2992314B1 (fr) 2012-06-22 2015-10-16 Sanofi Sa Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one et 1,2,3,4-tetrahydro-pyrimido{1,2-a}pyrimidin-6-one comportant une morpholine substituee, leur preparation et leur utilisation pharmaceutique
WO2015108881A1 (en) 2014-01-14 2015-07-23 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
WO2015108861A1 (en) 2014-01-14 2015-07-23 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
MA39823A (fr) 2014-04-03 2018-01-09 Janssen Pharmaceutica Nv Dérivés de pyridine macrocyclique
MA39822A (fr) 2014-04-03 2018-02-06 Janssen Pharmaceutica Nv Dérivés de pyrimidine bicycle
WO2016001789A1 (en) 2014-06-30 2016-01-07 Pfizer Inc. Pyrimidine derivatives as pi3k inhibitors for use in the treatment of cancer
TWI721104B (zh) * 2016-02-19 2021-03-11 瑞典商斯普林特生物科技公司 6‐芳基或6‐雜芳基‐4‐嗎啉‐4‐芳基‐吡啶‐2‐酮化合物
ES2821400T3 (es) 2016-02-19 2021-04-26 Sprint Bioscience Ab Compuestos de 6-heterociclil-4-morfolin-4-ilpiridin-2-ona útiles para el tratamiento del cáncer y la diabetes

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