JP2018521956A5 - - Google Patents

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JP2018521956A5
JP2018521956A5 JP2017548194A JP2017548194A JP2018521956A5 JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5 JP 2017548194 A JP2017548194 A JP 2017548194A JP 2017548194 A JP2017548194 A JP 2017548194A JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5
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alkenyl
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JP7266365B2 (ja
JP2018521956A (ja
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Priority claimed from PCT/US2016/033923 external-priority patent/WO2016191424A2/en
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JP2017548194A 2015-05-26 2016-05-24 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 Active JP7266365B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562166240P 2015-05-26 2015-05-26
US62/166,240 2015-05-26
PCT/US2016/033923 WO2016191424A2 (en) 2015-05-26 2016-05-24 Novel heteroaromatic silicon-fluoride-acceptors useful for 18f labeling of molecules and biomolecules, and methods of preparing same

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JP2021017722A Division JP2021073293A (ja) 2015-05-26 2021-02-05 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法

Publications (3)

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JP2018521956A JP2018521956A (ja) 2018-08-09
JP2018521956A5 true JP2018521956A5 (enExample) 2019-06-27
JP7266365B2 JP7266365B2 (ja) 2023-04-28

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JP2017548194A Active JP7266365B2 (ja) 2015-05-26 2016-05-24 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法
JP2021017722A Withdrawn JP2021073293A (ja) 2015-05-26 2021-02-05 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法

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US (4) US10800797B2 (enExample)
EP (1) EP3303349B1 (enExample)
JP (2) JP7266365B2 (enExample)
CN (1) CN107667109B (enExample)
CA (1) CA2982269C (enExample)
WO (1) WO2016191424A2 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7266365B2 (ja) 2015-05-26 2023-04-28 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法
US11413360B2 (en) * 2017-07-28 2022-08-16 Technische Universität München Dual mode radiotracer and—therapeutics
WO2019055825A1 (en) 2017-09-15 2019-03-21 The Regents Of The University Of California INHIBITION OF AMINOACYLASE 3 (AA3) IN THE TREATMENT OF CANCER
EP3917581A1 (en) * 2019-01-30 2021-12-08 Technische Universität München Silicon-fluoride acceptor substituted radiopharmaceuticals and precursors thereof
WO2020220020A1 (en) * 2019-04-26 2020-10-29 The Regents Of The University Of California Silicon-fluoride heteroaromatic systems for applications in positron emission tomography (pet) molecular imaging
EP3976562A1 (en) * 2019-05-24 2022-04-06 Duke University 18 f-radiolabeled biomolecules
US20230202944A1 (en) * 2020-05-29 2023-06-29 Fuzionaire, Inc. Methods for Rapid Formation of Chemicals Including Positron Emission Tomography Biomarkers
CN119301134A (zh) * 2022-04-20 2025-01-10 富齐奥奈尔治疗诊断股份有限公司 治疗诊断用的氟化硅杂芳族系统及其方法

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US6972336B2 (en) * 2002-07-18 2005-12-06 Novartis Ag N-alkylation of indole derivatives
WO2008040441A2 (en) 2006-10-02 2008-04-10 Bayer Schering Pharma Aktiengesellschaft Silicon derivatives for pet imaging
WO2010075286A1 (en) * 2008-12-24 2010-07-01 University Of Washington MOLECULAR ACTIVATORS OF THE Wnt/β-CATENIN PATHWAY
AU2011349482A1 (en) * 2010-12-22 2013-07-25 Ge Healthcare Limited HER2 binding peptides labeled with aluminium-(18) fluoride complexed by NOTA
JP7266365B2 (ja) 2015-05-26 2023-04-28 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法

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