JP2017508816A5 - - Google Patents

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JP2017508816A5
JP2017508816A5 JP2017501113A JP2017501113A JP2017508816A5 JP 2017508816 A5 JP2017508816 A5 JP 2017508816A5 JP 2017501113 A JP2017501113 A JP 2017501113A JP 2017501113 A JP2017501113 A JP 2017501113A JP 2017508816 A5 JP2017508816 A5 JP 2017508816A5
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JP
Japan
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heterocyclyl
heteroaryl
alkyl
aralkyl
alkynyl
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JP2017501113A
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English (en)
Japanese (ja)
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JP2017508816A (ja
JP6568926B2 (ja
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Priority claimed from PCT/US2015/021475 external-priority patent/WO2015143161A1/en
Publication of JP2017508816A publication Critical patent/JP2017508816A/ja
Publication of JP2017508816A5 publication Critical patent/JP2017508816A5/ja
Application granted granted Critical
Publication of JP6568926B2 publication Critical patent/JP6568926B2/ja
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JP2017501113A 2014-03-20 2015-03-19 癌の治療のためのerbbチロシンキナーゼ阻害剤としてのベンゾイミダゾール誘導体 Active JP6568926B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461968243P 2014-03-20 2014-03-20
US61/968,243 2014-03-20
PCT/US2015/021475 WO2015143161A1 (en) 2014-03-20 2015-03-19 Benzimidazole derivatives as erbb tyrosine kinase inhibitors for the treatment of cancer

Publications (3)

Publication Number Publication Date
JP2017508816A JP2017508816A (ja) 2017-03-30
JP2017508816A5 true JP2017508816A5 (https=) 2018-05-17
JP6568926B2 JP6568926B2 (ja) 2019-08-28

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ID=52808184

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JP2017501113A Active JP6568926B2 (ja) 2014-03-20 2015-03-19 癌の治療のためのerbbチロシンキナーゼ阻害剤としてのベンゾイミダゾール誘導体

Country Status (9)

Country Link
US (4) US10202398B2 (https=)
EP (1) EP3119784B1 (https=)
JP (1) JP6568926B2 (https=)
KR (1) KR102409739B1 (https=)
CN (1) CN106661027B (https=)
AU (1) AU2015231215B2 (https=)
CA (1) CA2943231C (https=)
TW (1) TWI705967B (https=)
WO (1) WO2015143161A1 (https=)

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KR102409739B1 (ko) 2014-03-20 2022-06-17 카펠라 테라퓨틱스, 인크. 암 치료용의 erbb 티로신 키나제 억제제로서의 벤즈이미다졸 유도체
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CN116997549A (zh) * 2020-09-23 2023-11-03 蝎子疗法股份有限公司 用于治疗癌症的吡咯并[3,2-c]吡啶-4-酮衍生物
JP7805363B2 (ja) 2020-11-02 2026-01-23 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング EGFR阻害薬としての置換1H-ピラゾロ[4,3-c]及び誘導体
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