JP2016540773A5 - - Google Patents

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Publication number
JP2016540773A5
JP2016540773A5 JP2016536710A JP2016536710A JP2016540773A5 JP 2016540773 A5 JP2016540773 A5 JP 2016540773A5 JP 2016536710 A JP2016536710 A JP 2016536710A JP 2016536710 A JP2016536710 A JP 2016536710A JP 2016540773 A5 JP2016540773 A5 JP 2016540773A5
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JP
Japan
Prior art keywords
composition
cancer
compound
pharmaceutically acceptable
acceptable salt
Prior art date
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Pending
Application number
JP2016536710A
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English (en)
Japanese (ja)
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JP2016540773A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2013/073482 external-priority patent/WO2015084384A1/en
Publication of JP2016540773A publication Critical patent/JP2016540773A/ja
Publication of JP2016540773A5 publication Critical patent/JP2016540773A5/ja
Pending legal-status Critical Current

Links

JP2016536710A 2013-12-06 2013-12-06 Atrキナーゼの阻害剤として有用な化合物 Pending JP2016540773A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2013/073482 WO2015084384A1 (en) 2013-12-06 2013-12-06 Compounds useful as inhibitors of atr kinase

Publications (2)

Publication Number Publication Date
JP2016540773A JP2016540773A (ja) 2016-12-28
JP2016540773A5 true JP2016540773A5 (enExample) 2017-02-09

Family

ID=49877037

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016536710A Pending JP2016540773A (ja) 2013-12-06 2013-12-06 Atrキナーゼの阻害剤として有用な化合物

Country Status (3)

Country Link
EP (1) EP3077393A1 (enExample)
JP (1) JP2016540773A (enExample)
WO (1) WO2015084384A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201516504D0 (en) * 2015-09-17 2015-11-04 Astrazeneca Ab Imadazo(4,5-c)quinolin-2-one Compounds and their use in treating cancer
HK1258570A1 (zh) 2015-09-30 2019-11-15 Vertex Pharmaceuticals Inc. 使用dna损伤剂及atr抑制剂的组合治疗癌症的方法
EP3461480A1 (en) 2017-09-27 2019-04-03 Onxeo Combination of a dna damage response cell cycle checkpoint inhibitors and belinostat for treating cancer
MX2021003263A (es) 2018-09-26 2021-05-12 Merck Patent Gmbh Combinacion de un antagonista de proteina de muerte programada 1 (pd-1), un inhibidor de ataxia telangiectasia y proteina relacionada con rad3 (atr) y un agente de platino para el tratamiento de cancer.
CN113164447A (zh) 2018-10-15 2021-07-23 默克专利股份公司 利用dna烷化剂和atr抑制剂的组合疗法
CA3195592A1 (en) 2020-10-16 2022-04-21 Xiaohui Liu Triheterocyclic derivative, and pharmaceutical composition and application thereof
CN115466258A (zh) * 2021-06-11 2022-12-13 成都苑东生物制药股份有限公司 Atr抑制剂及其用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0714665A2 (pt) * 2006-08-04 2012-03-13 Takeda Pharmaceutical Company Limited Composto, pró-droga, agente farmacêutico, e, método para a profilaxia ou tratamento do câncer
UA110324C2 (en) * 2009-07-02 2015-12-25 Genentech Inc Jak inhibitory compounds based on pyrazolo pyrimidine
US9018395B2 (en) * 2011-01-27 2015-04-28 Université de Montréal Pyrazolopyridine and pyrazolopyrimidine derivatives as melanocortin-4 receptor modulators

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