JP2016500088A - 即時放出および持続放出のための組成物 - Google Patents

即時放出および持続放出のための組成物 Download PDF

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Publication number
JP2016500088A
JP2016500088A JP2015543424A JP2015543424A JP2016500088A JP 2016500088 A JP2016500088 A JP 2016500088A JP 2015543424 A JP2015543424 A JP 2015543424A JP 2015543424 A JP2015543424 A JP 2015543424A JP 2016500088 A JP2016500088 A JP 2016500088A
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
active ingredient
tolterodine
controlled release
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2015543424A
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English (en)
Japanese (ja)
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JP2016500088A5 (enrdf_load_stackoverflow
Inventor
アフジャー,バリンダー
ヴァーマ,ラジャン
ヴィナヤクラオ バラブド,ウメシュ
ヴィナヤクラオ バラブド,ウメシュ
ハグステン,アルネ
ワナーバーガー,クリスティン
ブールグ,ランバブ
ヴィラスラオ サムワンシ,アモル
ヴィラスラオ サムワンシ,アモル
Original Assignee
フェリング ベスローテン フェンノートシャップ
フェリング ベスローテン フェンノートシャップ
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Application filed by フェリング ベスローテン フェンノートシャップ, フェリング ベスローテン フェンノートシャップ filed Critical フェリング ベスローテン フェンノートシャップ
Publication of JP2016500088A publication Critical patent/JP2016500088A/ja
Publication of JP2016500088A5 publication Critical patent/JP2016500088A5/ja
Pending legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • A61K38/095Oxytocins; Vasopressins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5089Processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • Physiology (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
JP2015543424A 2012-11-21 2013-11-21 即時放出および持続放出のための組成物 Pending JP2016500088A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN3575DE2012 2012-11-21
IN3575/DEL/2012 2012-11-21
IN3947/DEL/2012 2012-12-20
IN3947DE2012 2012-12-20
PCT/EP2013/074373 WO2014079922A1 (en) 2012-11-21 2013-11-21 Composition for immediate and extended release

Publications (2)

Publication Number Publication Date
JP2016500088A true JP2016500088A (ja) 2016-01-07
JP2016500088A5 JP2016500088A5 (enrdf_load_stackoverflow) 2016-11-17

Family

ID=49619947

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015543424A Pending JP2016500088A (ja) 2012-11-21 2013-11-21 即時放出および持続放出のための組成物

Country Status (18)

Country Link
EP (1) EP2922525A1 (enrdf_load_stackoverflow)
JP (1) JP2016500088A (enrdf_load_stackoverflow)
KR (1) KR20150085826A (enrdf_load_stackoverflow)
CN (1) CN104797240A (enrdf_load_stackoverflow)
AR (1) AR093585A1 (enrdf_load_stackoverflow)
AU (1) AU2013349682A1 (enrdf_load_stackoverflow)
BR (1) BR112015011430A2 (enrdf_load_stackoverflow)
CA (1) CA2891365A1 (enrdf_load_stackoverflow)
EA (1) EA201590805A1 (enrdf_load_stackoverflow)
HK (1) HK1213779A1 (enrdf_load_stackoverflow)
IL (1) IL238648A0 (enrdf_load_stackoverflow)
IN (1) IN2015DN03984A (enrdf_load_stackoverflow)
MX (1) MX2015006399A (enrdf_load_stackoverflow)
PH (1) PH12015501096A1 (enrdf_load_stackoverflow)
SG (2) SG10201703388TA (enrdf_load_stackoverflow)
TW (1) TW201422254A (enrdf_load_stackoverflow)
WO (1) WO2014079922A1 (enrdf_load_stackoverflow)
ZA (1) ZA201503603B (enrdf_load_stackoverflow)

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JP2016525548A (ja) 2013-07-23 2016-08-25 アラーガン、インコーポレイテッドAllergan,I� Β−3アドレナリン受容体刺激薬と組み合わせたデスモプレシンを含む方法及び組成物
KR20150144209A (ko) * 2014-06-16 2015-12-24 훼링 비.브이. 안정화된 데스모프레신 또는 이의 약학적으로 허용가능한 염을 함유 약학 조성물
CN106999538A (zh) * 2014-11-20 2017-08-01 阿勒根公司 包含去氨加压素与α‑肾上腺素能受体拮抗剂组合的方法和组合物
WO2016114812A1 (en) * 2015-01-12 2016-07-21 Robert Niichel Layered sustained-release microbeads and methods of making the same
US20170042806A1 (en) 2015-04-29 2017-02-16 Dexcel Pharma Technologies Ltd. Orally disintegrating compositions
CN108135870A (zh) * 2015-09-01 2018-06-08 韦尔斯利医药有限公司 延缓、延迟和立即释放型制剂及其制造方法和用途
WO2017058428A1 (en) * 2015-09-30 2017-04-06 Wellesley Pharmaceuticals, Llc Composition for reducing the frequency of urination, method of making and use thereof
AU2016331879A1 (en) * 2015-09-30 2018-05-17 Wellesley Pharmaceuticals, Llc Composition for reducing the frequency of urination, method of making and use thereof
TW201726114A (zh) * 2015-11-23 2017-08-01 魏斯理製藥公司 降低排尿頻率之組成物、其製備方法、及其應用
CN108601782A (zh) * 2015-12-18 2018-09-28 韦尔斯利医药有限公司 用于缓解尿频的组合物,其制备方法和用途
KR20220100077A (ko) 2016-04-21 2022-07-14 발큐리아 에이비 암의 예비치료용 조성물 및 방법
US10076494B2 (en) 2016-06-16 2018-09-18 Dexcel Pharma Technologies Ltd. Stable orally disintegrating pharmaceutical compositions
KR20190104322A (ko) * 2017-01-11 2019-09-09 훼링 비.브이. 속붕해성 약학적 조성물
KR20190021180A (ko) * 2017-08-22 2019-03-05 아주대학교산학협력단 퇴행성 신경질환 치료용 복합 제형 조성물
US12389928B1 (en) * 2024-10-25 2025-08-19 Mccormick & Company, Inc. Flavor-changing product

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JP2003503341A (ja) * 1999-06-28 2003-01-28 サノフィ−サンテラボ 少なくとも一つの適時パルスを生ずる制御された放出用の医薬投与形態
JP2003517446A (ja) * 1998-11-11 2003-05-27 フアーマシア・アー・ベー 新規制御放出ビーズ、その製造方法、およびそれを含む多重ユニット製剤
JP2006502972A (ja) * 2002-05-07 2006-01-26 フェリング ベスローテン フェンノートシャップ デスモプレシンの口腔内分散性医薬製剤
WO2011120904A2 (en) * 2010-03-29 2011-10-06 Ferring B.V. A fast dissolving pharmaceutical composition
WO2011120903A2 (en) * 2010-03-29 2011-10-06 Ferring B.V. A fast dissolving pharmaceutical composition
US20120135050A1 (en) * 2010-07-08 2012-05-31 Wellesley Pharmaceuticals, Llc Extended-release formulation for reducing the frequency of urination and method of use thereof

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WO1998003184A1 (en) 1996-07-19 1998-01-29 Clarke-Garegg, Margaret, A. Levan derivatives, their preparation, composition and applications including medical and food applications
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JP2003503341A (ja) * 1999-06-28 2003-01-28 サノフィ−サンテラボ 少なくとも一つの適時パルスを生ずる制御された放出用の医薬投与形態
JP2006502972A (ja) * 2002-05-07 2006-01-26 フェリング ベスローテン フェンノートシャップ デスモプレシンの口腔内分散性医薬製剤
WO2011120904A2 (en) * 2010-03-29 2011-10-06 Ferring B.V. A fast dissolving pharmaceutical composition
WO2011120903A2 (en) * 2010-03-29 2011-10-06 Ferring B.V. A fast dissolving pharmaceutical composition
US20120135050A1 (en) * 2010-07-08 2012-05-31 Wellesley Pharmaceuticals, Llc Extended-release formulation for reducing the frequency of urination and method of use thereof

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Also Published As

Publication number Publication date
IL238648A0 (en) 2015-06-30
WO2014079922A1 (en) 2014-05-30
EA201590805A1 (ru) 2015-11-30
CN104797240A (zh) 2015-07-22
PH12015501096A1 (en) 2015-07-27
SG10201703388TA (en) 2017-05-30
IN2015DN03984A (enrdf_load_stackoverflow) 2015-10-02
CA2891365A1 (en) 2014-05-30
AU2013349682A1 (en) 2015-06-04
SG11201503913TA (en) 2015-06-29
EP2922525A1 (en) 2015-09-30
MX2015006399A (es) 2015-07-21
TW201422254A (zh) 2014-06-16
BR112015011430A2 (pt) 2017-07-11
KR20150085826A (ko) 2015-07-24
HK1213779A1 (zh) 2016-07-15
AR093585A1 (es) 2015-06-10
ZA201503603B (en) 2016-01-27

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