JP2016175923A - Pest control composition and use therefor - Google Patents

Abstract

PROBLEM TO BE SOLVED: To provide a pest control composition having excellent control effect on pests.SOLUTION: A pest control composition comprises a tetrazolinone compound represented by formula (1) and the like, and one or more component selected from group A, group B, group C, group D, group E and group F [in the formula (1), Ris C6-C16 aryl group or the like; Xis O or S; Ris H, alkyl or the like; Rand Rindependently represent H or the like; R-Rindependently represent C1-C12 alkyl group or the like; Ris C1-C6 alkyl group or the like; Yis O or S; Qis O, S or NR.] Group A: bactericidal agent; Group B: insecticide and miticide, Group C: herbicide, Group D: phytotoxicity reducing agent, Group E: plant growth regulator, and Group F: microbial material.SELECTED DRAWING: None

Description

  The present invention relates to pest control compositions and methods for controlling pests.

  Conventionally, many compounds are known as an active ingredient of pest control composition (for example, refer to patent documents 1 and non-patent documents 1).

International Publication No. 2013/162072

The Pesticide Manual-16th edition (BCPC) ISBN 978-1-901396-86-7

  An object of the present invention is to provide a pest control composition having an excellent control effect against pests.

The inventors of the present invention have studied to find a pest control composition having an excellent control activity against pests, and as a result, the following formulas (1), (2), (3), (4), and (5) (6), (7), (8), (9), (10), (11), (12), (13), (14), (15) (16), Formula (17), Formula (18), Formula (19), Formula (20), Formula (21), Formula (22) or Formula (23) (hereinafter referred to as “compound”) The composition containing the compound (hereinafter referred to as "the present compound") was found to exhibit excellent pesticidal activity against pests, and led to the present invention.
That is, the present invention is as follows.
[1] Group (I), Group (II), Group (III), Group (IV), Group (V), Group (VI), Group (VII), Group (VIII), Group (IX), Group ( X), group (XI), group (XII), group (XIII), group (XIV), group (XV), group (XVI), group (XVII), group (XVIII), group (XVIII), group (XIX), group (X) XX) a compound according to any one selected from the group consisting of group (XXI), group (XXII) and group (XXIII), and one or more components selected from the group consisting of group A to group F Pest control composition.
Group A: fungicide group B; insecticide, acaricide group C; herbicide group D; safener group E; plant growth regulator group F;

Group (I): Formula (1)
[In the formula,
R ¹ is one or more substituents may be a C6-C16 aryl group, one or more substituents may be a C7-C18 selected from the group P ¹ is selected from the group P ¹ C 2 -C 12 optionally having one or more substituents selected from the group P ¹ and the C ¹ -C 12 alkyl group optionally having one or more substituents selected from the group P ¹ alkenyl group, 1 or more substituents may be a C2-C12 alkynyl group, one or more substituents may be a C3-C12 selected from the group P ¹ is selected from the group P ¹ cycloalkyl groups, one or more substituents acyl group which may C2-C12 optionally having one or more good adamantyl group optionally having a substituent selected from the group P ¹ is selected from the group P ¹ of , A C3-C12 trialkylsilyl group, a hydrogen atom, or (Wherein the C6-C16 aryl group, the C7-C18 aralkyl group, the C1-C12 alkyl group, the C2-C12 alkenyl group, the C2-C12 alkynyl group, the C3-C12 alkenyl group) When the C12 cycloalkyl group, the C2 to C12 acyl group, and the adamantyl group have two or more substituents, the substituents may be the same or different from each other),
X ¹ represents a sulfur atom or an oxygen atom,
R ² represents a hydrogen atom, an alkyl group of C1-C12, haloalkyl of C1-C12, an alkenyl group of C2-C12, haloalkenyl of C2-C12, alkynyl group C2-C12, haloalkynyl group C2-C12 , A C 2 -C 12 alkoxycarbonyl group, a hydroxycarbonyl group, or a halogen atom,
R ⁴ and R ⁵ independently of each other represent a hydrogen atom, a halogen atom or a C1-C3 alkyl group,
Or R ⁴ and R ⁵ may be combined to form a C3-C6 cycloalkane ring together with the carbon atom to which they are attached,
R ⁶ , R ⁷ , R ⁸ and R ⁹ are, independently of one another, a C1-C12 alkyl group, a halogen atom, a C1-C12 haloalkyl group, a C3-C12 cycloalkyl group, a C3-C12 halocycloalkyl Group, C1-C12 alkoxy group, C1-C12 haloalkoxy group, C1-C12 alkylthio group, C1-C12 haloalkylthio group, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, C2 -C12 alkenyl group, C2-C12 haloalkenyl group, C2-C12 alkynyl group, C2-C12 haloalkynyl group, C3-C12 cycloalkyloxy group, C3-C12 halocycloalkyloxy group, C3-C12 C12 cycloalkylthio group, C2 to C12 alkenyloxy group, C2 to C12 alkynyl alkoxy Group, C2-C12 haloalkenyloxy group, C2-C12 haloalkynyloxy group, C2-C12 alkynylthio group, C2-C12 alkenylthio group, C2-C12 haloalkenylthio group, C2-C12 halo Alkynylthio group, C2-C12 acyl group, C2-C12 haloacyl group, C2-C12 acyloxy group, C2-C12 acylthio group, C2-C12 alkoxycarbonyl group, C3-C12 trialkylsilyl group, C5 Substituted with a -C14 trialkylsilylethynyl group, a C1-C12 alkylsulfonyl group, a C1-C12 haloalkylsulfonyl group, a C1-C12 alkylsulfinyl group, a C1-C12 haloalkylsulfinyl group, a C1-C12 alkyl group; Aminosulfonyl group which may be substituted, C1-C12 alkyl group Optionally substituted amino group, C1-C12 alkyl group optionally substituted aminocarbonyl group, a hydrogen atom, or represents a hydroxy group or a formyl group,
Alternatively, adjacent R ⁶ and R ⁷ , R ⁷ and R ⁸ , and R ⁸ and R ⁹ are combined to form a C4-C6 cycloalkene ring, a C5-C6 cycloalkene ring and a carbon atom to which they are bound. It may form an alkyldiene ring or a benzene ring,
R ¹⁰ is a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkoxyalkyl group, a C3-C6 cycloalkyl group or a C3 Represents a -C6 halocycloalkyl group,
Y ¹ represents an oxygen atom or a sulfur atom,
Q ¹ represents an oxygen atom, a sulfur atom, or an NR ¹¹ group,
R ¹¹ represents a hydrogen atom, a C1-C6 alkyl group, or a C1-C6 haloalkyl group.
Group P ¹ : halogen atom, C1-C12 alkyl group, C1-C12 haloalkyl group, C1-C12 alkoxy group, C1-C12 haloalkoxy group, C1-C12 alkylthio group, C1-C12 haloalkylthio group , Hydroxycarbonyl group, formyl group, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, C2-C12 alkenyl group, C2-C12 haloalkenyl group, C2-C12 alkynyl group, C2-C12 , A C3-C12 cycloalkyl group, a C3-C12 halocycloalkyl group, a C3-C12 cycloalkyloxy group, a C3-C12 halocycloalkyloxy group, a C3-C12 cycloalkylthio group, and C2 -C12 alkenyloxy group, C2-C12 alkynyloxy group, C2-C12 haloalkenyloxy group, C2-C12 haloalkynyloxy group, C2-C12 alkynylthio group, C2-C12 alkenylthio group, C2-C12 haloalkenylthio group, C2-C12 haloalkynylthio Group, C2-C12 acyl group, C2-C12 haloacyl group, C2-C12 acyloxy group, C2-C12 acylthio group, C2-C12 alkoxycarbonyl group, C6-C16 aryl group, C6-C16 haloaryl Groups, C6-C16 aryloxy groups, C6-C16 haloaryloxy groups, C6-C16 arylthio groups, C6-C16 haloarylthio groups, C7-C18 aralkyl groups, C7-C18 haloaralkyl groups, C7-C18 arylalkoxy group, C7-C18 haloarylalkoxy group, C3-C12 Trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C12 alkylsulfonyl group, C1-C12 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloarylsulfonyl group, C1 -C12 alkylsulfinyl group, C1-C12 haloalkylsulfinyl group, C6-C16 arylsulfinyl group, C6-C16 haloarylsulfinyl group, C2-C11 polyoxaalkyloxy group, C2-C5 oxacycloalkyloxy Optionally substituted with a C 1 -C 12 alkyl group and / or an aminocarbonyl group optionally substituted with a C 6 -C 12 aryl group, a C 1 -C 12 alkyl group and / or a C 6 -C 12 aryl group Aminosulfonyl group and C1-C1 A group consisting of an amino group which may be substituted by 2 alkyl groups. ]
A tetrazolinone compound represented by the formula:

Group (II): Formula (2)
[In the formula,
R ²⁴ and R ²⁵ each represent a hydrogen atom or a C1-C3 alkyl group;
R ²⁶ represents a C1-C4 alkyl group, a C3-C6 cycloalkyl group, a C1-C4 haloalkyl group, a C3-C6 halocycloalkyl group, a halogen atom, a cyano group, a nitro group, a C2-C4 alkenyl group, a C2-C4 halo group Alkenyl group, C2-C4 alkynyl group, C2-C4 haloalkynyl group, C1-C4 alkoxy group, C1-C4 haloalkoxy group, C1-C4 alkylthio group or C1-C4 haloalkylthio group;
R ²⁷ , R ²⁸ and R ²⁹ each represent a hydrogen atom or a halogen atom;
R ³⁰ represents a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C2-C3 alkynyl group, a C2-C3 haloalkynyl group, a C3-C5 cycloalkyl group or a C3 -C5 represents a halocycloalkyl group;
X ² represents an oxygen atom or a sulfur atom;
R ³³ represents a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a hydrogen atom, a C1 to C6 haloalkyl group, a C3 to C6 halocycloalkyl group, a C2 to C6 alkenyl group, a C2 to C6 haloalkenyl group, or a C2 to C6 An alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group or a C1-C6 alkylthio group;
Q ² is a phenyl group, a phenoxy group, a phenylthio group, a phenylamino group (however, the phenyl portion of the phenyl group, the phenoxy group, the phenylthio group and the phenylamino group together with the adjacent carbon atom is a 4- or 5-membered ring The ring may form one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom as a ring-constituting atom, and may be the same. The carbon atom may have an oxo group, a thioxo group or a C1-C3 alkoxyimino group, and the same sulfur atom may have one or two oxide groups, and the phenyl moiety and the corresponding ones ring may have one or more atoms or groups selected from the group P ^21, when atom or a group selected from the group P ²¹ is two or more, the original Or groups can be different from the same or different.),
5- or 6-membered heterocyclyl group, 5- or 6-membered heterocyclyloxy group, 5- or 6-membered heterocyclylthio group, 5- or 6-membered heterocyclylamino group (provided that the 5- or 6-membered heterocyclyl group, 5- or 6-membered heterocyclyloxy group, 5 And the 5- or 6-membered heterocyclyl moiety of the 5- or 6-membered heterocyclylamino group and the 5- or 6-membered heterocyclylamino group together with the adjacent carbon atom form a 4-, 5-, 6- or 7-membered ring The ring may contain one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom as a ring member atom, and the 5- or 6-membered heterocyclyl moiety and the ring Are oxo, thioxo or C1-C3 alkoxyimino on the same carbon atom May also be, may have one or two oxide groups to the same sulfur atom, it may have one or more atoms or groups selected from the group P ^21, selected from the group P ²¹ When there are two or more atoms or groups, the atoms or groups may be the same or different),
A C3-C6 cycloalkyl group, a C3-C6 cycloalkenyl group, provided that the C3-C6 cycloalkyl group and the C3-C6 cycloalkenyl group, together with the adjacent carbon atom, are a 4-, 5-, or 6-membered ring Or a 7-membered ring may be formed, and the ring may contain one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom as a ring constituting atom, and the same sulfur atom may be used. The ring, the C3-C6 cycloalkyl group and the C3-C6 cycloalkenyl group may have an oxo group, a thioxo group or a C1-C3 alkoxyimino on the same carbon atom. may have a group may have one or more atoms or groups selected from the group P ^21, when atom or a group selected from the group P ²¹ is two or more, The atoms or groups may be the same or different),
C 1 -C 4 alkyl group (provided that the C 1 -C 4 alkyl group may have an oxo group, a thioxo group or a C 1 -C 3 alkoxyimino group at the same carbon atom, and one or more selected from group P ²¹ And may have an atom or group, and when the atom or group selected from group P ²¹ is 2 or more, the atoms or groups may be the same or different from each other),
C2-C4 alkenyl or C2-C4 alkynyl group (provided that the C2-C4 alkenyl and C2-C4 alkynyl group may have one or more atoms or groups selected from the group ^{P 21,} the group P ^{When the} atom or group selected from ²¹ is 2 or more, the atom or group may be the same or different;
Alternatively, the substituent in Q ² and R ³³ may form a 5-, 6-, or 7-membered ring together with the carbon atom or nitrogen atom to which they are attached, and the ring is One or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom may be contained as a ring constituent atom, and one or more atoms or a group selected from group P ²⁴ may be contained as a substituent Preferably, when the atom or group selected from the group P ²⁴ is 2 or more, the atoms or groups may be the same or different.
Group P ^21: the group P ²³ atoms or optionally may be C1-C6 alkyl group optionally having a group selected from atoms or optionally may be C3-C6 cycloalkyl group having a group selected from the group P ^23,
A phenyl group (however, the phenyl group may form a 4-, 5-, 6-, or 7-membered ring together with the adjacent carbon atom, and the ring includes an oxygen atom, a sulfur atom and a nitrogen atom; The ring may contain one or more atoms selected from the group consisting of atoms, and may have an oxo group, a thioxo group or a C1-C3 alkoxyimino group on the same carbon atom, and the same sulfur It may have 1 or 2 of the oxide group in atom, also the phenyl group and the ring may have one or more atoms or groups selected from the group P ^22, from the group P ²² When two or more atoms or groups are selected, the atoms or groups may be the same or different),
5- or 6-membered heterocyclyl group (provided that the 5- or 6-membered heterocyclyl group may form a 4-, 5-, 6-, or 7-membered ring together with the adjacent carbon atom, and the ring is And one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom may be contained as a ring-constituting atom, and the 5- or 6-membered heterocyclyl group and the ring may have the same carbon atom oxo group, thioxo group, or may have a C1-C3 alkoxyimino group may have one or two oxide groups to the same sulfur atom, 1 or more atoms selected from the group P ²² Or when it has two or more atoms or groups selected from group P ²² , the atoms or groups may be the same or different),
C1-C6 haloalkoxy group, halogen atom, nitro group, C1-C6 alkoxy group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 alkenyloxy Group, C3-C6 haloalkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkynyloxy group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group Group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, cyano group, amino group, hydroxy group, mercapto group, pentafluorosulfanyl group, C3-C9 Trialkylsilyl group, C2-C6 alkyl Carbonyl group, C2-C6 alkoxycarbonyl group, C2-C8 alkylaminocarbonyl group and C2-C8 group consisting alkylcarbonylamino group.
Group P ^22: the group P ²³ atoms or optionally may be C1-C6 alkyl group optionally having a group selected from atoms or optionally may be C3-C6 cycloalkyl group having a group selected from the group P ^23,
C1-C6 alkoxy group, C1-C6 haloalkoxy group, halogen atom, nitro group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 alkenyloxy Group, C3-C6 haloalkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkynyloxy group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group Group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, cyano group, amino group, hydroxy group, mercapto group, pentafluorosulfanyl group, C3-C9 Trialkylsilyl group, C2-C6 alkyl Carbonyl group, C2-C6 alkoxycarbonyl group, C2-C8 alkylaminocarbonyl group and C2-C8 group consisting alkylcarbonylamino group.
Group P ²³ : Halogen atom, C3 to C6 cycloalkyl group, C3 to C6 halocycloalkyl group, C1 to C4 alkoxy group, C1 to C4 haloalkoxy group, C1 to C4 alkylthio group and C1 to C4 haloalkylthio group .
Group P ²⁴ : halogen atom, cyano group, nitro group, C1 to C4 alkyl group, C3 to C6 cycloalkyl group, C1 to C4 haloalkyl group, C3 to C6 halocycloalkyl group, C1 to C4 alkoxy group, C1 to C4 halo A group consisting of an alkoxy group, a C1-C4 alkylthio group and a C1-C4 haloalkylthio group. ]
A tetrazolinone compound represented by the formula:

Group (III): Formula (3)
[In the formula,
R ⁴¹ , R ⁴² , R ⁴³ and R ⁵¹ each independently represent a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, C2-C6 C6 alkynyl group, C2 to C6 haloalkynyl group, C1 to C6 alkoxy group, C1 to C6 haloalkoxy group, C1 to C8 alkylamino group, C1 to C8 haloalkylamino group, C1 to C6 alkylthio group, C1 to C6 haloalkylthio group , C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2 -C6 alkoxycarbonyl group, C2-C9 alkyl amide Carbonyl group,
A C1-C6 alkyl group optionally having a group selected from Group P ³¹ ;
Or a C3-C6 cycloalkyl group optionally having one or more groups selected from group P ³¹ ;
R ⁴⁴ and R ⁴⁵ each represent a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ⁴⁶ is a C1-C4 alkyl group which may have a halogen atom, a hydrogen atom, a halogen atom, a C1-C4 alkoxy group which may have a halogen atom, a C2-C4 alkenyl group, a C2-C4 halo Alkenyl group, C2-C4 alkynyl group, C2-C4 haloalkynyl group, C1-C4 alkylthio group, C1-C4 haloalkylthio group, C3-C6 cycloalkyl group or C3-C6 halocycloalkyl group, cyano group, nitro group, A C1-C4 alkylsulfinyl group, a C1-C4 alkylsulfonyl group, a C1-C4 haloalkylsulfinyl group, a C1-C4 haloalkylsulfonyl group, a C1-C6 alkylamino group or a C1-C6 haloalkylamino group;
R ⁴⁷ , R ⁴⁸ and R ⁴⁹ each independently represent a hydrogen atom, a halogen atom, a C 1 -C 3 alkyl group, a C 1 -C 3 haloalkyl group, a C 2 -C 3 alkenyl group, a C 2 -C 3 haloalkenyl group, a C 1 -C 3 alkoxy group, or C 1 -C3 represents a haloalkoxy group;
R ⁵⁰ represents a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C2-C3 alkynyl group, a C2-C3 haloalkynyl group, a C3-C5 cycloalkyl group, or Represents a C3-C5 halocycloalkyl group;
X ³ represents an oxygen atom or a sulfur atom;
R ⁵² is
A C1-C6 alkyl group optionally having a group selected from Group P ³¹ ;
A C3-C6 cycloalkyl group optionally having a group selected from Group P ³¹ ;
A phenyl group which may have a group selected from group P ³² ;
Hydrogen atom, halogen atom, cyano group, nitro group, amino group, C2 to C6 alkenyl group, C2 to C6 haloalkenyl group, C1 to C6 haloalkyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C1 to C6 Alkoxy group, C1-C6 haloalkoxy group, C3-C6 cycloalkenyl group, C3-C6 halocycloalkenyl group, C1-C8 alkylamino group, C3-C12 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 Represents an alkoxycarbonyl group, or a C2-C9 alkylaminocarbonyl group;
R ⁵³ represents a C 1 -C 8 alkyl group, a C 1 -C 8 haloalkyl group, a C 2 -C 8 alkenyl group, a C 2 -C 8 haloalkenyl group, a C 2 -C 6 alkynyl group, a C 2 -C 6 haloalkynyl group, a C 3 -C 6 cycloalkyl group, C 3 -C6 halocycloalkyl group, C3-C6 cycloalkenyl group, C3-C6 halocycloalkenyl group,
Or a benzyl group which may have a group selected from group P ³² .
Group P ³¹ : halogen atom, cyano group, C3 to C6 cycloalkyl group, C3 to C6 halocycloalkyl group, C1 to C4 alkoxy group, C1 to C4 haloalkoxy group, C1 to C4 alkylthio group and C1 to C4 haloalkylthio group A group consisting of
Group P ³² : halogen atom, cyano group, amino group, hydroxy group, thiol group, C1 to C6 alkyl group, C1 to C6 haloalkyl group, C3 to C6 cycloalkyl group, C3 to C6 halocycloalkyl group, C2 to C6 alkenyl Group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C8 alkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1- A group consisting of C6 alkylsulfinyl group, C1-C6 alkylsulfonyl group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, and C2-C9 alkylamino carbonyl group . ]
A tetrazolinone compound represented by the formula:

Group (IV): Formula (4)
[In the formula,
R ⁶¹ and R ⁶² each independently represent a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ⁶³ represents a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, Nitro group, cyano group,
An aminocarbonyl group which may have a C1-C6 alkyl group,
C2-C6 haloalkenyl group, C2-C6 haloalkynyl group, C3-C6 halocycloalkyl group, C1-C6 haloalkoxy group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl group Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, C2-C6 alkoxycarbonyl group, hydroxyl group, thio Group, an amino group which may have a C1-C6 alkyl group, a pentafluorosulfanyl group, a C3-C9 trialkylsilyl group, a C5-C14 trialkylsilylethynyl group, a C1-C4 alkylsulfonyl group, a C1-C4 group. A haloalkylsulfonyl group, a C1-C4 alkylsulfinyl group, a C1-C4 haloalkylsulfinyl group, a C2-C5 alkoxyalkyl group or a C2-C5 alkylthioalkyl group;
R ⁶⁴ , R ⁶⁵ and R ⁶⁶ each independently represent a hydrogen atom, a halogen atom, a C 1 -C 4 alkyl group, a C 1 -C 4 haloalkyl group, a C 3 -C 5 cycloalkyl group, a C 3 -C 5 halocycloalkyl group, C 1 -C 4 Represents an alkoxy group or a C1-C4 haloalkoxy group;
R ⁶⁷ represents a C1-C6 alkyl group, a hydrogen atom, a C1-C6 haloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkoxyalkyl group, a C3-C6 cycloalkyl group or a C3-C6 halo group Represents a cycloalkyl group;
A ⁴ is a halogen atom, one or more atoms which may have a group C6-C16 aryl group selected from the group P ^40, have one or more atoms or groups selected from the group P ⁴⁰ A good C3-C12 cycloalkyl group, a C2-C9 heterocyclyl group optionally having one or more atoms or groups selected from group P ^40, provided that the C2-C9 heterocyclyl group is a nitrogen atom as a ring-constituting atom, When containing one or more atoms selected from the group consisting of an oxygen atom and a sulfur atom and containing two or more atoms selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom, each of the atoms is at least one other 1 may be different identical or different and the atom. further, a carbon atom or a nitrogen atom constituting the ring of the C2-C9 heterocyclyl group is not bonded to Q ⁴ .) Or represents one or more atoms C3-C12 cycloalkenyl group having a group selected from the group ^{P 40} (provided that the C6-C16 aryl group, the C3-C12 cycloalkyl group, said C2 The —C 9 heterocyclyl group and the C 3 -C 12 cycloalkenyl group may have one or more atoms or groups selected from group P ^40, and when having two or more atoms or groups selected from group P, Each of the atoms or groups may be the same as or different from at least one other atom or group);
Q ⁴ represents a group Q 41, Q 42, Q 43, Q 44, Q 45, Q 46, Q 47, Q 48, Q 49, Q 50, Q 51 or Q 52 {# represents a binding site to A, and ● represents a binding site to an oxygen atom Represents
R ⁶⁸ , R ⁶⁹ , R ⁷⁰ and R ⁷¹ each independently represent a hydrogen atom, a halogen atom, a C1-C6 alkyl group optionally having one or more atoms or groups selected from group P ⁴¹ , group P C3-C6 cycloalkyl group optionally having one or more atoms or groups selected from ⁴¹ , C1-C6 alkoxy group, C1-C6 haloalkoxy group, cyano group, nitro group, amino group, hydroxy group, thiol Group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group,
An amino group which may have a C1-C6 alkyl group,
An amino group which may have a C1-C6 haloalkyl group,
C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C9 tri An alkylsilyl group, a C2-C6 alkylcarbonyl group, a C2-C6 alkoxycarbonyl group or an aminocarbonyl group which may have a C1-C6 alkyl group;
X ⁴ represents an oxygen atom or a sulfur atom.
Group P ⁴⁰ : halogen atom, C1 to C6 alkyl group, C1 to C6 haloalkyl group, C2 to C6 alkenyl group, C2 to C6 haloalkenyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C3 to C6 cycloalkyl Group, C3-C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl group Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, hydroxycarbonyl group, formyl group, C2-C6 alkoxycarbonyl group, nitro group, cyano group, Hydroxyl group, C6-C16 aryl group, C6-C16 haloaryl group, C6-C16 aryloxy group, C6-C16 haloaryloxy group, C6-C16 arylthio group, C6-C16 haloarylthio group, C7-C18 aralkyl group, C7-C18 haloaralkyl group, C7-C18 arylalkoxy group, C7-C18 haloarylalkoxy group, thiol group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C6 Alkyls Phonyl group, C1-C6 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloarylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C6-C16 arylsulfinyl group, C6-C16 halo Arylsulfinyl group,
An amino group which may have a C1-C6 alkyl group,
A group consisting of an aminosulfonyl group optionally having a C1-C6 alkyl group and / or a C6-C12 aryl group, and an aminocarbonyl group optionally having a C1-C6 alkyl group.
Group P ⁴¹ : halogen atom, cyano group, C3 to C6 cycloalkyl group, C3 to C6 halocycloalkyl group, C1 to C4 alkoxy group, C1 to C4 haloalkoxy group, C1 to C4 alkylthio group and C1 to C4 haloalkylthio group A group consisting of ]
A tetrazolinone compound represented by the formula:

Group (V): Formula (5)
[In the formula,
Q ⁵ represents a group of the following Q53, Q54, Q55, Q56 or Q57;
R ⁸¹ , R ⁸² , R ⁸³ and R ⁹¹ each independently represent a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, C2-C6 C6 alkynyl group, C2 to C6 haloalkynyl group, C1 to C6 alkoxy group, C1 to C6 haloalkoxy group, C1 to C8 alkylamino group, C1 to C8 haloalkylamino group, C1 to C6 alkylthio group, C1 to C6 haloalkylthio group , C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2 -C6 alkoxycarbonyl group, C2-C8 alkylamino Carbonyl group, a group of a C1-C6 may be an alkyl group or a group optionally may be C3-C6 cycloalkyl group having a selected from the group P ⁵¹ selected from the group P ^51;
R ⁸⁴ and R ⁸⁵ each represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ⁸⁶ represents a C1 to C4 alkyl group, a halogen atom, a C1 to C4 alkoxy group, a cyano group, a nitro group, a C1 to C4 haloalkyl group, a C2 to C4 alkenyl group, a C2 to C4 haloalkenyl group, or a C3 to C6 cycloalkyl group , C2-C4 alkynyl group, C2-C4 haloalkynyl group, C1-C4 haloalkoxy group, C1-C4 alkylthio group, C1-C4 alkylsulfinyl group, C1-C4 alkylsulfonyl group, C1-C4 haloalkylthio group, C1- C4 haloalkylsulfinyl group, C1-C4 haloalkylsulfonyl group, C1-C6 alkylamino group, C1-C6 haloalkylamino group, C3-C6 halocycloalkyl group or hydrogen atom;
R ⁸⁷ , R ⁸⁸ and R ⁸⁹ each represent a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group or a C1-C3 alkoxy group;
R ⁹⁰ represents a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C2-C3 alkynyl group, a C2-C3 haloalkynyl group, a C3-C5 cycloalkyl group or a C3 -C5 represents a halocycloalkyl group;
X ⁵ represents an oxygen atom or a sulfur atom;
A ⁵¹ and A ⁵³ each independently represent a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 alkenyl group; C6 haloalkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C8 alkylamino group, C1-C8 dialkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group Group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, C2-C8 alky It represents Le aminocarbonyl group, a group of a C1-C6 may be an alkyl group or a group optionally may be C3-C6 cycloalkyl group having a selected from the group P ⁵¹ selected from the group P ^51;
A ⁵² , Z ⁵¹ and Z ⁵⁴ each independently represent a hydrogen atom, an amino group, a C3-C6 alkenyl group, a C3-C6 haloalkenyl group, a C3-C6 alkynyl group, a C3-C6 haloalkynyl group, a C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C3-C6 cycloalkylsulfonyl group, C3-C6 halocycloalkylsulfonyl group, C2-C8 alkylaminosulfonyl group, C2-C8 haloalkyl An aminosulfonyl group, a C3-C9 trialkylsilyl group, a C2-C6 alkylcarbonyl group, a C2-C6 alkoxycarbonyl group, a C2-C8 alkylaminocarbonyl group, a C4-C7 cycloalkylmethyl group, a group selected from the group P ⁵¹ ; C1-C6 alkyl which may be possessed Or a group optionally may be C3-C6 cycloalkyl group having a selected from the group P ^51;
Z ⁵⁵ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C6 cycloalkyl group or a C1-C6 halocycloalkyl group;
Y ⁵¹ , Y ⁵² , Y ⁵³ , Z ⁵² and Z ⁵³ each represents a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, an aldehyde group, a C2-C6 alkenyl group, a C2-C6 group Haloalkenyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C1 to C6 alkoxy group, C1 to C6 haloalkoxy group, C3 to C6 alkenyloxy group, C3 to C6 haloalkenyloxy group, C3 to C6 alkynyloxy Group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C1-C8 alkylamino group, C1-C8 Haloalkylamino group, C 1 -C 6 alkylthio group, C 1 -C 6 haloalkylthio group, C 1 -C 6 alkylsul , C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C8 alkylaminosulfonyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2-C6 alkyl carbonyl Group, a C1-C6 alkyl group which may have a group selected from C2-C6 alkoxycarbonyl group, a C2-C8 alkylaminocarbonyl group, an aminocarbonyl group, and a group P ^51, or a group selected from a group P ⁵¹ Represents an optionally substituted C3-C6 cycloalkyl group;
Or Y ⁵¹ and Y ⁵² may form a 5-, 6-, or 7-membered saturated ring together with the carbon atom to which they are attached (provided that the saturated ring is And may contain an oxygen atom or a sulfur atom as a ring-constituting atom, and the saturated ring may have a group selected from group P ⁵¹ as a substituent);
Y ⁵² and Y ⁵³ may form a 5-, 6-, or 7-membered saturated ring together with the carbon atom to which they are attached (provided that the saturated ring has the ring configuration thereof And may contain an oxygen atom or a sulfur atom as the atom, and the saturated ring may have a group selected from group P ⁵¹ as a substituent);
Z ⁵¹ and Z ⁵² may form a 5-, 6- or 7-membered saturated ring together with the carbon atom or nitrogen atom to which they are attached (provided that the saturated ring is And may contain an oxygen atom, a nitrogen atom or a sulfur atom as a ring member atom, and the saturated ring may have a group selected from group P ⁵¹ as a substituent);
Z ⁵² and Z ⁵³ may form a 5-, 6-, or 7-membered saturated ring together with the carbon atom to which they are attached (provided that the saturated ring has the ring configuration The atom may contain an oxygen atom, a nitrogen atom or a sulfur atom, and the saturated ring may have a group selected from group P ⁵¹ as a substituent).
Group P ⁵¹ : halogen atom, cyano group, C3 to C6 cycloalkyl group, C3 to C6 halocycloalkyl group, C1 to C4 alkoxy group, C1 to C4 haloalkoxy group, C1 to C4 alkylthio group and C1 to C4 haloalkylthio group A group consisting of ]
A tetrazolinone compound represented by the formula:

Group (VI): Formula (6)
[Wherein, Q ⁶ represents a 6-membered aromatic heterocyclic group which may have one or more atoms or groups selected from group P ⁶¹ (however, hetero atoms constituting the heterocyclic group are A nitrogen atom, wherein the number of nitrogen atoms is 1, 2 or 3);
R ^{101, R 102, R 103} and ^{R 111} are each independently 1 or more atoms may be C1-C6 alkyl group optionally having a group selected from the group ^{P 62,} one or more selected from the group ^{P 62} C3-C6 cycloalkyl group which may have one or more atoms, or a halogen atom, a hydrogen atom, a C1-C6 alkoxy group which may have one or more halogen atoms, a cyano group, a nitro group, an amino group , A hydroxy group, a sulfanyl group, a C2-C6 alkenyl group optionally having one or more halogen atoms, a C2-C6 alkynyl group optionally having one or more halogen atoms, one or two C1-C8 groups An amino group which may have an alkyl group (provided that it may have a halogen atom), a C1-C6 alkylthio group which may have one or more halogen atoms, one or more C1-C6 alkylsulfinyl group which may have a halogen atom, C1-C6 alkylsulfonyl group which may have one or more halogen atoms, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2- C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, or aminocarbonyl group optionally having one or more C2-C8 alkyl;
Each of R ¹⁰⁴ and R ¹⁰⁵ independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ¹⁰⁶ is a C1-C6 alkyl group optionally having one or more halogen atoms, a C3-C6 cycloalkyl group optionally having one or more halogen atoms, a halogen atom, a hydrogen atom, one or more halogens A C2-C6 alkenyl group which may have an atom, a C1-C6 alkoxy group which may have one or more halogen atoms, a C1-C6 alkylthio group which may have one or more halogen atoms, C2-C6 alkynyl group optionally having one or more halogen atoms, nitro group, cyano group, aminocarbonyl group optionally having one or two C1-C6 alkyl groups, one or more halogen atoms C3-C6 cycloalkoxy group which may have, C3-C6 cycloalkylthio group which may have one or more halogen atoms, may have one or more halogen atoms C3-C6 alkenyloxy group, C3-C6 alkynyloxy group optionally having one or more halogen atoms, C3-C6 alkenylthio group optionally having one or more halogen atoms, one or more halogen atoms A C3-C6 alkynylthio group which may have one or more substituents, a C2-C6 alkylcarbonyl group which may have one or more halogen atoms, a C2-C6 alkylcarbonyloxy group, a C2-C6 alkylcarbonylthio group, a C2 -C6 alkoxycarbonyl group, hydroxy group, sulfanyl group, amino group optionally having 1 or 2 C1-C6 alkyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C5-C14 trialkylsilyl Ethynyl group, C1-C4 alkylsulfonyl group optionally having one or more halogen atoms, one or more It represents androgenic atom C1-C4 alkyl sulfates may have a sulfinyl group, C2-C5 alkoxyalkyl group, or C2-C5 alkylthioalkyl group;
R ¹⁰⁷ , R ¹⁰⁸ and R ¹⁰⁹ may each independently have a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms Represents a C2-C3 alkenyl group or a C1-C3 alkoxy group optionally having one or more halogen atoms;
R ¹¹⁰ has a C1-C3 alkyl group which may have one or more halogen atoms, a C2-C3 alkenyl group which may have one or more halogen atoms, one or more halogen atoms, A C2-C3 alkynyl group or a C3-C5 cycloalkyl group optionally having one or more halogen atoms;
X ⁶ represents an oxygen atom or a sulfur atom.
Group P ⁶¹ : C1-C6 alkyl group optionally having one or more halogen atoms, halogen atom, C2-C6 alkenyl group optionally having one or more halogen atoms, one or more halogen atoms C2-C6 alkynyl group which may be substituted, C3-C6 cycloalkyl group which may have one or more halogen atoms, C1-C6 alkoxy group which may have one or more halogen atoms, one or more Or C1-C6 alkylthio group which may have one or more halogen atoms, C3-C6 cycloalkyloxy group which may have one or more halogen atoms, C3-C6 which may have one or more halogen atoms C6 cycloalkylthio group, C3 to C6 alkenyloxy group optionally having one or more halogen atoms, C3 to C6 alkynyloxy group optionally having one or more halogen atoms, A C3-C6 alkenylthio group which may have one or more halogen atoms, a C3-C6 alkynylthio group which may have one or more halogen atoms, C2 which may have one or more halogen atoms -C6 alkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, hydroxycarbonyl group, formyl group, C2-C6 alkoxycarbonyl group, nitro group, cyano group, hydroxy group, one or more halogen atoms A C6-C16 aryl group optionally having one or more carbon atoms, a C6-C16 aryloxy group optionally having one or more halogen atoms, a C6-C16 arylthio group optionally having one or more halogen atoms, C7-C18 aralkyl group optionally having one or more halogen atoms, C optionally having one or more halogen atoms -C18 arylalkoxy group, sulfanyl group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C6 alkylsulfonyl group optionally having one or more halogen atoms, C6-C16 arylsulfonyl group optionally having one or more halogen atoms, C1-C6 alkylsulfinyl group optionally having one or more halogen atoms, optionally having one or more halogen atoms C6-C16 arylsulfinyl group, C1-C6 alkyl group and / or aminosulfonyl group optionally having C6-C12 aryl group, amino group, C1-C8 alkyl group having 1 or 2 An amino group (which may have a halogen atom), and one or two C 1 -C 6 al The group consisting of which may aminocarbonyl group optionally having Le group.
Group P ⁶² : halogen atom, cyano group, C3-C6 cycloalkyl group optionally having one or more halogen atoms, C1-C4 alkoxy group optionally having one or more halogen atoms, and one or more A group consisting of a C1-C4 alkylthio group which may have a halogen atom. ]
A tetrazolinone compound represented by the formula:

Group (VII): Formula (7)
[In the formula,
R ¹²¹ and R ¹²² each independently represent a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ¹²³ represents a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, Nitro group, cyano group, aminocarbonyl group optionally having C1 to C6 alkyl group, C2 to C6 haloalkenyl group, C2 to C6 haloalkynyl group, C3 to C6 halocycloalkyl group, C1 to C6 haloalkoxy group , C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 halo Alkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Lucinylthio, C3-C6 haloalkenylthio, C3-C6 haloalkynylthio, C2-C6 alkylcarbonyl, C2-C6 haloalkylcarbonyl, C2-C6 alkylcarbonyloxy, C2-C6 alkylcarbonylthio, C2 -C6 alkoxycarbonyl group, hydroxy group, sulfanyl group, amino group optionally having C1-C6 alkyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1 -C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C2-C5 alkoxyalkyl group, C2-C5 alkylthioalkyl group or hydrogen atom;
R ¹²⁴ , R ¹²⁵ and R ¹²⁶ are each independently a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group or a C1-C3 alkoxy group Represents
R ¹²⁷ represents a C1-C3 alkyl group optionally having one or more halogen atoms;
Q ⁷ is a divalent 5-membered aromatic heterocyclic group optionally having one or more atoms or groups selected from group P ^72, provided that the heterocyclic group is a nitrogen atom, an oxygen atom or a sulfur atom Containing one or more heteroatoms selected, the number of nitrogen atoms being 0, 1, 2, 3 or 4 and the number of oxygen atoms and sulfur atoms being 0 or 1);
X ⁷ represents an oxygen atom or a sulfur atom;
A ⁷ represents a 5-10 membered monocyclic or fused heterocyclic group optionally having one or more atoms or groups selected from group P ⁷¹ (provided that the heterocyclic group is nitrogen Containing one or more hetero atoms selected from the group consisting of atoms, oxygen atoms and sulfur atoms, the number of nitrogen atoms is 0, 1, 2, 3 or 4 and the number of oxygen atoms and sulfur atoms is 0, 1, 2 or 3).
Group P ⁷¹ : halogen atom, C1 to C6 alkyl group, C1 to C6 haloalkyl group, C2 to C6 alkenyl group, C2 to C6 haloalkenyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C3 to C6 cycloalkyl Group, C3-C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl group Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, hydroxycarbonyl group, formyl group, C2-C6 alkoxycarbonyl group, nitro group, cyano group, Hydroxy group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloarylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkyl A group consisting of an amino group which may have a group, an aminosulfonyl group which may have a C1-C6 alkyl group, and an aminocarbonyl group which may have a C1-C6 alkyl group.
Group P ⁷² : halogen atom, C1 to C4 alkyl group, C1 to C4 haloalkyl group, cyano group, C3 to C6 cycloalkyl group, C3 to C6 halocycloalkyl group, C1 to C4 alkoxy group, C1 to C4 haloalkoxy group, A group consisting of a C1-C4 alkylthio group and a C1-C4 haloalkylthio group. ]
And tetrazolinone compounds and salts thereof.

Group (VIII): Formula (8)
[In the formula,
R ¹³¹ may have one or more atoms or C6-C16 aryl group optionally having a group, one or more atoms or groups selected from the group ^{P 81} selected from the group ^{P 81} C1- C12 alkyl group, 1 or more atoms may be C3-C12 cycloalkyl group optionally having a group selected from the group P ^81, may have one or more atoms or groups selected from the group P ⁸¹ C2 -C12 alkenyl group, 1 or more atoms C3-C12 cycloalkenyl group having a group selected from the group P ^81, may have one or more atoms or groups selected from the group P ⁸¹ C2-C12 alkynyl group, a 1 or more atoms C2-C12 acyl group or a hydrogen atom has a group selected from the group ^{P 81} (provided that the C6-C16 ants Group, the C1-C12 alkyl group, the C3-C12 cycloalkyl group, said C2-C12 alkenyl group, the C3-C12 cycloalkenyl group, the C2-C12 alkynyl group or the C2-C12 acyl group, the group P ^When having two or more atoms or groups selected from ⁸¹ , the substituents may be the same or different);
R ¹³² and R ¹³³ each represent a hydrogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C12 alkoxycarbonyl group, a hydroxycarbonyl group or a halogen atom;
R ¹³⁴ and R ¹³⁵ each represent a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ¹³⁶ is a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, A nitro group, a cyano group, an aminocarbonyl group which may have a C1-C6 alkyl group,
C2-C6 haloalkenyl group, C2-C6 haloalkynyl group, C3-C6 halocycloalkyl group, C1-C6 haloalkoxy group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl group Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 acyl group, C2-C6 haloacyl group, C2-C6 acyloxy group, C2-C6 acylthio group, C2-C6 alkoxycarbonyl group , Hydroxyl group, thiol group, amino group, C -C6 alkylamino group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C4 alkylsulfonyl group, C1-C4 haloalkylsulfonyl group, C1-C4 alkylsulfinyl group , A C 1 -C 4 haloalkylsulfinyl group, a C 2 -C 5 alkoxyalkyl group or a C 2 -C 5 alkylthioalkyl group;
R ¹³⁷ , R ¹³⁸ and R ¹³⁹ each represent a hydrogen atom, a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C3-C5 cycloalkyl group, a C3-C5 halocycloalkyl group, a C1-C4 alkoxy group or a C1 -C4 represents a haloalkoxy group;
R ¹⁴⁰ is a C1 to C6 alkyl group, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C2 to C6 haloalkenyl group, a C2 to C6 alkoxyalkyl group, a C3 to C6 cycloalkyl group or a C3 to C6 halocycloalkyl group Represents
X ⁸ represents an oxygen atom or a sulfur atom.
Group P ⁸¹ : halogen atom, C1 to C6 alkyl group, C1 to C6 haloalkyl group, C2 to C6 alkenyl group, C2 to C6 haloalkenyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C3 to C6 cycloalkyl Group, C3-C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, 3-C6 haloalkynylthio group, C2-C6 acyl group, C2-C6 haloacyl group, C2-C6 acyloxy group, C2-C6 acylthio group, hydroxycarbonyl group, formyl group, C2-C6 alkoxycarbonyl group, nitro group, cyano Group, hydroxyl group, C6-C16 aryl group, C6-C16 haloaryl group, C6-C16 aryloxy group, C6-C16 haloaryloxy group, C6-C16 arylthio group, C6-C16 haloarylthio group, C7-C18 aralkyl Group, C7-C18 haloaralkyl group, C7-C18 arylalkoxy group, C7-C18 haloarylalkoxy group, thiol group, pentafluorosulfuranyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group , C1-C6 al Cyl sulfonyl group, C1-C6 haloalkyl sulfonyl group, C6-C16 aryl sulfonyl group, C6-C16 halo aryl sulfonyl group, C1-C6 alkyl sulfinyl group, C1-C6 halo alkyl sulfinyl group, C6-C16 aryl sulfinyl group, C6-C16 A group consisting of an aminosulfonyl group which may have a haloarylsulfinyl group, a C1-C6 alkyl group or a C6-C12 aryl group, and an aminocarbonyl group which may have a C1-C6 alkyl group. ]
A tetrazolinone compound represented by the formula:

Group (IX): Formula (9)
{In the ceremony,
A ⁹ represents a 5-membered aromatic complex group selected from group P ⁹² ;
Or R ¹⁵⁴ and R ¹⁵⁵ independently represent a hydrogen atom or an alkyl group having 1 to 3 carbon atoms, or
R ¹⁵⁴ and ¹⁵⁵ may be combined to form a C 3 -C 6 cycloalkane ring together with the carbon atom to which they are attached;
R ¹⁵⁶ is an alkyl group having 1 to 12 carbon atoms, a halogen atom, a haloalkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, a halocycloalkyl group having 3 to 12 carbon atoms, 12 alkoxy group, haloalkoxy group having 1 to 12 carbon atoms, alkylthio group having 1 to 12 carbon atoms, haloalkylthio group having 1 to 12 carbon atoms, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group An alkenyl group having 2 to 12 carbon atoms, a haloalkenyl group having 2 to 12 carbon atoms, an alkynyl group having 2 to 12 carbon atoms, a haloalkynyl group having 2 to 12 carbon atoms, a cycloalkyloxy group having 3 to 12 carbon atoms, C3-C12 halocycloalkyloxy group, C3-C12 cycloalkylthio group, C2-C12 alkenyloxy group, C2-C1 2 alkynyloxy group, haloalkenyl oxy group having 2 to 12 carbon atoms, haloalkynyl oxy group having 2 to 12 carbon atoms, alkynylthio group having 2 to 12 carbon atoms, alkenylthio group having 2 to 12 carbon atoms, 2-12 haloalkenylthio group, C2-C12 haloalkynylthio group, C2-C12 alkylcarbonyl group, C2-C12 haloalkylcarbonyl group, C2-C12 alkylcarbonyloxy group An alkylcarbonylthio group having 2 to 12 carbon atoms, an alkoxycarbonyl group having 2 to 12 carbon atoms, a trialkylsilyl group having 3 to 12 carbon atoms, a trialkylsilylethynyl group having 5 to 14 carbon atoms, 1 to 12 carbon atoms Alkylsulfonyl group, haloalkylsulfonyl group having 1 to 12 carbon atoms, alkylsulfinyl group having 1 to 12 carbon atoms, 1 carbon atom 12 haloalkylsulfinyl groups, aminosulfonyl groups optionally having alkyl groups having 1 to 12 carbon atoms, amino groups optionally having alkyl groups having 1 to 12 carbon atoms, alkyl having 1 to 12 carbon atoms Represents an aminocarbonyl group which may have a group, a hydroxycarbonyl group, or a formyl group;
R ¹⁵⁷ , R ¹⁵⁸ and R ¹⁵⁹ each independently represent a hydrogen atom, an alkyl group having 1 to 12 carbon atoms, a halogen atom, a haloalkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, carbon A halocycloalkyl group having 3 to 12 carbons, an alkoxy group having 1 to 12 carbons, a haloalkoxy group having 1 to 12 carbons, an alkylthio group having 1 to 12 carbons, a haloalkylthio group having 1 to 12 carbons, a nitro group , Cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, alkenyl group having 2 to 12 carbon atoms, haloalkenyl group having 2 to 12 carbon atoms, alkynyl group having 2 to 12 carbon atoms, halo having 2 to 12 carbon atoms Alkynyl group, cycloalkyl group having 3 to 12 carbon atoms, halocycloalkyloxy group having 3 to 12 carbon atoms, cycloalkylthio group having 3 to 12 carbon atoms, carbon number To 12 alkenyloxy groups, alkynyl groups having 2 to 12 carbon atoms, haloalkenyloxy groups having 2 to 12 carbon atoms, haloalkynyloxy groups having 2 to 12 carbon atoms, alkynylthio groups having 2 to 12 carbon atoms, carbon Alkenylthio group having 2 to 12 carbon atoms, a haloalkenylthio group having 2 to 12 carbon atoms, a haloalkynylthio group having 2 to 12 carbon atoms, an alkylcarbonyl group having 2 to 12 carbon atoms, a haloalkylcarbonyl group having 2 to 12 carbon atoms An alkylcarbonyloxy group having 2 to 12 carbon atoms, an alkylcarbonylthio group having 2 to 12 carbon atoms, an alkoxycarbonyl group having 2 to 12 carbon atoms, a trialkylsilyl group having 3 to 12 carbon atoms, and 5 to 14 carbon atoms Trialkylsilylethynyl group, alkylsulfonyl group having 1 to 12 carbon atoms, haloalkylsulfonyl group having 1 to 12 carbon atoms, 1 carbon atom To 12 alkylsulfinyl group, haloalkylsulfinyl group having 1 to 12 carbon atoms, aminosulfonyl group which may have alkyl group having 1 to 12 carbon atoms, and alkyl group having 1 to 12 carbon atoms A good amino group, an aminocarbonyl group optionally having an alkyl group having 1 to 12 carbon atoms, a hydroxycarbonyl group, or a formyl group;
R ¹⁶⁰ represents an alkyl group of 1 to 3 carbon atoms or a haloalkyl group of 1 to 3 carbon atoms;
Y ⁹ represents an oxygen atom or a sulfur atom;
Q ⁹ represents an oxygen atom, a sulfur atom, or an NR ¹⁷² group;
R ¹⁷² represents a hydrogen atom, an alkyl group having 1 to 6 carbon atoms, or a haloalkyl group having 1 to 6 carbon atoms.
Group P ⁹² : a group consisting of the following structural formulas E1 to E36.
[Wherein, # represents a bonding position with Q ⁹ ;
R ¹⁶¹ represents a hydrogen atom, an alkyl group having 1 to 6 carbon atoms, a haloalkyl group having 1 to 6 carbon atoms, an alkenyl group having 2 to 6 carbon atoms, a haloalkenyl group having 2 to 6 carbon atoms, or 2 to 6 carbon atoms An alkynyl group, a haloalkynyl group having 2 to 6 carbon atoms;
R ¹⁵⁰ , R ¹⁵² and R ¹⁵³ each represents a hydrogen atom, a halogen atom, an alkyl group having 1 to 6 carbon atoms, a haloalkyl group having 1 to 6 carbon atoms, an alkenyl group having 2 to 6 carbon atoms, 2 to 6 carbon atoms A haloalkenyl group, an alkynyl group having 2 to 6 carbon atoms, a haloalkynyl group having 2 to 6 carbon atoms, an alkoxycarbonyl group having 2 to 6 carbon atoms, a hydroxycarbonyl group, or a cyano group;
R ¹⁵¹ is one or more atoms or aryl group which may having 6 to 16 carbon atoms which may have a group selected from the group P ^91, have one or more atoms or groups selected from the group P ⁹¹ Good aralkyl group having 7 to 18 carbon atoms, one or more atoms selected from group P ⁹¹ or a cycloalkyl group having 3 to 12 carbon atoms optionally having a group, one or more atoms selected from group P ⁹¹ or Adamantyl group which may have a group or a hydrogen atom (provided that the aryl group having 6 to 16 carbon atoms, the aralkyl group having 7 to 18 carbon atoms, the cycloalkyl group having 3 to 12 carbon atoms, and When the adamantyl group has two or more substituents, the substituents may be the same or different).
Group P ⁹¹ : halogen atom, alkyl group having 1 to 12 carbon atoms, haloalkyl group having 1 to 12 carbon atoms, alkoxy group having 1 to 12 carbon atoms, haloalkoxy group having 1 to 12 carbon atoms, or 1 to 12 carbon atoms Alkylthio group, haloalkylthio group having 1 to 12 carbon atoms, hydroxycarbonyl group, formyl group, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, alkenyl group having 2 to 12 carbon atoms, 2 to 2 carbon atoms 12, a haloalkenyl group, an alkynyl group having 2 to 12 carbon atoms, a haloalkynyl group having 2 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, a halocycloalkyl group having 3 to 12 carbon atoms, 3 to 3 carbon atoms 12 cycloalkyloxy groups, C3-C12 halocycloalkyloxy groups, C3-C12 cycloalkylthio groups, C2-C1 Alkenyloxy group, alkynyloxy group having 2 to 12 carbon atoms, haloalkenyloxy group having 2 to 12 carbon atoms, haloalkynyloxy group having 2 to 12 carbon atoms, alkynylthio group having 2 to 12 carbon atoms, 2 carbon atoms Alkenylthio group, haloalkenylthio group having 2 to 12 carbon atoms, haloalkynylthio group having 2 to 12 carbon atoms, alkylcarbonyl group having 2 to 12 carbon atoms, haloalkylcarbonyl group having 2 to 12 carbon atoms, carbon An alkylcarbonyloxy group having 2 to 12 carbon atoms, an alkylcarbonylthio group having 2 to 12 carbon atoms, an alkoxycarbonyl group having 2 to 12 carbon atoms, an aryl group having 6 to 16 carbon atoms, a haloaryl group having 6 to 16 carbon atoms, carbon An aryloxy group having 6 to 16 carbon atoms, a haloaryloxy group having 6 to 16 carbon atoms, an arylthio group having 6 to 16 carbon atoms, 6 to 16 carbon atoms Haloarylthio group, aralkyl group having 7 to 18 carbon atoms, haloaralkyl group having 7 to 18 carbon atoms, arylalkoxy group having 7 to 18 carbon atoms, haloarylalkoxy group having 7 to 18 carbon atoms, 3 to 3 carbon atoms 12 trialkylsilyl groups, C5-14 trialkylsilylethynyl groups, C1-12 alkylsulfonyl groups, C1-12 haloalkylsulfonyl groups, C6-16 arylsulfonyl groups, carbon Haloarylsulfonyl group having 6 to 16 carbon atoms, alkylsulfinyl group having 1 to 12 carbon atoms, haloalkylsulfinyl group having 1 to 12 carbon atoms, arylsulfinyl group having 6 to 16 carbon atoms, haloarylsulfinyl group having 6 to 16 carbon atoms , A polyoxaalkyloxy group having 2 to 11 carbon atoms, an oxacycloalkyloxy group having 2 to 5 carbon atoms, It has an aminocarbonyl group which may have an alkyl group having a prime of 1 to 12 and / or an aryl group having a carbon number of 6 to 12, an alkyl group having a carbon number of 1 to 12, and / or an aryl group having a carbon number of 6 to 12 A group consisting of an aminosulfonyl group which may be substituted and an amino group which may have an alkyl group having 1 to 12 carbon atoms. ]}
A tetrazolinone compound represented by the formula:

Group (X): Formula (10)
[In the formula,
Each of R ¹⁸¹ and R ¹⁸² independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R ¹⁸³ has a C1-C6 alkyl group which may have one or more halogen atoms, a C1-C6 alkoxy group which may have one or more halogen atoms, and one or more halogen atoms, A C3-C6 cycloalkyl group, a halogen atom, a C2-C6 alkenyl group optionally having one or more halogen atoms, a cyano group, a C1-C6 alkylthio group optionally having one or more halogen atoms A C 2 -C 6 alkynyl group which may have one or more halogen atoms, a nitro group, an aminocarbonyl group which may have one or more C 1 -C 6 alkyl groups, one or more halogen atoms C3-C6 cycloalkyloxy group, C3-C6 cycloalkylthio group optionally having one or more halogen atoms, C optionally having one or more halogen atoms 3-C6 alkenyloxy group, C3-C6 alkynyloxy group optionally having one or more halogen atoms, C3-C6 alkenylthio group optionally having one or more halogen atoms, one or more halogen atoms Optionally substituted C3-C6 alkynylthio group, C2-C6 alkoxycarbonyl group, hydroxy group, sulfanyl group, C1-C8 alkylamino group optionally having one or more halogen atoms, pentafluorosulfanyl group , C3-C9 trialkylsilyl group, C1-C6 alkylsulfonyl group optionally having one or more halogen atoms, C1-C6 alkylsulfinyl group optionally having one or more halogen atoms, C2-C6 Alkyl carbonyl group, C2-C5 alkoxy alkyl group or C2-C5 alkyl thioalkyl group ;
R ¹⁸⁴ , R ¹⁸⁵ and R ¹⁸⁶ may each independently have a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms Represents a C1-C3 alkoxy group;
R ¹⁸⁷ represents a C1-C3 alkyl group which may have one or more halogen atoms;
Q ¹⁰ represents a divalent group selected from group P ¹⁰³ ,
A ¹⁰ may have one or more atoms or C6-C16 aryloxy group has a group, one or more atoms or groups selected from the group P ¹⁰² selected from the group P ¹⁰² C6 -C16 arylthio ^{group, R 195 O-N = C} (R 196) -, R 193 R 194 N-N = C (R 196) -, is selected from ^{R 193 R 194 N-CH =} N-, group P ¹⁰² 1 or more atoms be C7-C18 aralkyl group optionally having a group, 1 or more atoms be C7-C18 aralkyloxy group optionally having a group selected from the group P ^102, selected from the group P ¹⁰² C7-C16 aryloxyalkyl group which may have one or more atoms or groups, C7-C16 arylcarbonyl group optionally having one or more atoms or groups selected from group P ¹⁰² , group P one or more of the original selected from ¹⁰² Or optionally anilino group which may have a group, the heteroaryl in one or more atoms or groups which may have a C2-C9 heteroaryl group (wherein the heteroaryl group selected from the group P ¹⁰² The moiety represents a 5-, 6-, 5- and 5-membered ring, a 5- and 6-membered condensed ring, or a 6- and 6-membered ring), C 3 -C6 cycloalkyloxy group or C4-C10 cycloalkylalkoxy group is represented, and R ¹⁹³ and R ¹⁹⁴ are C 1 -C 3 alkyl group which may be the same or different and may have one or more halogen atoms;
R ¹⁹⁵ is a C1-C6 alkyl group which may have one or more halogen atoms, a C2-C6 alkenyl group which may have one or more halogen atoms, or one or more halogen atoms A good C2-C6 alkynyl group, a C3-C6 cycloalkyl group optionally having one or more halogen atoms, a C7-C18 aralkyl group optionally having one or more atoms or groups selected from group P ¹⁰¹ Or a phenyl group optionally having one or more atoms or groups selected from group P ¹⁰¹ ;
R ¹⁹⁶ is a C1-C6 alkyl group optionally having one or more halogen atoms, a hydrogen atom, a C3-C6 cycloalkyl group optionally having one or more halogen atoms, or one or more halogen atoms Represents a phenyl group which may be possessed;
X ¹⁰ represents an oxygen atom or a sulfur atom.
Group P ¹⁰¹ : halogen atom, cyano group, C1-C4 alkyl group optionally having one or more halogen atoms, C3-C6 cycloalkyl group optionally having one or more halogen atoms, one or more The group which consists of a C1-C4 alkoxy group which may have a halogen atom, and a C1-C4 alkylthio group which may have one or more halogen atoms.
Group P ¹⁰² : C1-C6 alkyl group optionally having one or more halogen atoms, halogen atom, cyano group, hydroxy group, C3-C6 cycloalkyl group optionally having one or more halogen atoms, C1 to C6 alkoxy group which may have one or more halogen atoms, C1 to C6 alkylthio group which may have one or more halogen atoms, C2-which may have one or more halogen atoms C6 alkenyl group, C2-C6 alkynyl group optionally having one or more halogen atoms, C1-C8 alkylamino group optionally having one or more halogen atoms, one or more halogen atoms C 1 -C 6 alkylsulfinyl group, C 1 -C 6 alkylsulfonyl group optionally having one or more halogen atoms, pentafluorosulfanyl group, C 2 C6 alkoxycarbonyl group, C2-C6 alkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylamino group, aminocarbonyl group optionally having one or more C1-C6 alkyl groups, and C3-C9 A group consisting of trialkylsilyl groups.
Group P ¹⁰³ : a group consisting of the group Q11 and the group Q12
(Wherein, R ¹⁸⁸ , R ¹⁸⁹ , R ¹⁹⁰ and R ¹⁹¹ each independently represent a hydrogen atom, a halogen atom, or a C1-C4 alkyl group optionally having one or more halogen atoms, and # is Represents a binding site to A ^10, and ● represents a binding site to an oxygen atom. ]
A tetrazolinone compound represented by the formula:

Group (XI): Formula (11)
[In the formula,
R ²⁰⁵ represents a C1-C3 alkyl group optionally having one or more halogen atoms;
E ⁴⁰ represents a divalent 5-membered heteroaryl group or a divalent 6-membered heteroaryl group;
Y ^{11 _{is, - (CH 2) n 11}} -G -, - G- (CH 2) n 11 -, - G- (CH 2) n 11 -G -, - G-CH 2 CH 2 -G-CH ₂ CH ₂ -G-, -CH ₂ -G-CH ₂ CH ₂ -G-, -G-CH ₂ CH ₂ -G-CH _2- , -CH = CH-, -CH = CH-G-,- _{G-CH = CH -, -} CH = CH-CH 2 -G -, - G-CH 2 -CH = CH -, - G-CH = CH-CH 2 -, - CH 2 -CH = CH-G- _{, -CH = CH-G-CH} 2 -, - CH 2 -G-CH = CH -, - CH = CH-CH 2 -G-CH 2 -, - CH 2 -G-CH 2 -CH = CH- _{, -CH = CH-G-CH} 2 CH 2 -, - CH 2 CH 2 -G-CH = CH -, - G-CH = CH-CH 2 CH 2 -, - CH 2 CH 2 -CH = CH G -, - CH = CH- G-CH = CH -, - C≡C -, - C≡C-CH 2 -G -, - G-CH 2 -C≡C -, - C≡C-CH 2 -G-CH ₂ -or -CH ₂ -G-CH ₂ -C≡C- (wherein the hydrogen atom of Y ¹¹ is one or more atoms selected from the group consisting of a halogen atom and a C1-C3 alkyl group) Or the group may be substituted, and when substituted by two or more atoms or groups, the atoms and groups may be the same or different; G represents an oxygen atom, a sulfur atom, or NR ^B ; R ^B represents a hydrogen atom or a C 1 -C 3 alkyl group, n ¹¹ represents an integer of 1 to 10. Q ¹³ is bonded to the left of Y ¹¹ and E ⁴⁰ is bonded to the right.
Q ¹³ is a divalent C 6 -C 10 aryl group (provided that the divalent C 6 -C 10 aryl group may have one or more atoms or groups selected from group P ¹¹² ) or divalent And the divalent 5-10 membered heterocyclic group may have one or more atoms or groups selected from Group P ¹¹² , and a nitrogen atom as a ring constituting atom And, when it contains one or more atoms selected from the group consisting of an oxygen atom and a sulfur atom and contains two or more atoms, the atoms may be the same or different).
X ¹¹ represents an oxygen atom or a sulfur atom;
A ¹¹ represents a C 6 -C 10 aryl group, an adamantyl group, a C 6 -C 10 aryloxy group, a C 6 -C 10 arylthio group, a C 6 -C 10 arylamino group, a C 3 -C 10 cycloalkyl group, a 5-10 membered heterocyclic group The 5- to 10-membered heterocyclic group contains one or more atoms selected from the group consisting of nitrogen atoms, oxygen atoms and sulfur atoms as ring-constituting atoms, and in the case of containing two or more atoms, the atoms are the same or A 5- to 10-membered heteroaryloxy group (wherein the 5- to 10-membered heteroaryloxy group is selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom as a ring-constituting atom) When containing one or more atoms and containing two or more atoms, the atoms may be the same or different from each other, a 5- to 10-membered heteroarylthio group (however, The 5-10 membered heteroarylthio group contains one or more atoms selected from the group consisting of nitrogen atoms, oxygen atoms and sulfur atoms as ring-constituting atoms, and in the case of containing two or more atoms, the atoms are A 5- to 10-membered heteroarylamino group (provided that the 5- to 10-membered heteroarylamino group is a ring constituent atom consisting of a nitrogen atom, an oxygen atom and a sulfur atom) When containing one or more atoms selected and containing two or more atoms, the atoms may be the same or different), a C6-C10 arylsulfonyl group, a C6-C10 arylsulfinyl group, or a group good -CH = NH optionally having 1 or 2 groups selected from P ¹¹³ (however, if the -CH = NH has two groups selected from the group P ^113, the base may be the same or (Wherein the C6-C10 aryl group, adamantyl group, C6-C10 aryloxy group, C6-C10 arylthio group, C6-C10 arylamino group, C3-C10 cycloalkyl group, 5-10 membered heterocyclic group, 5-10 membered heteroaryloxy group, 5-10 membered heteroarylthio group, 5-10 membered heteroarylamino group, C6-C10 arylsulfonyl group and C6-C10 arylsulfonyl group The group may have one or more atoms or groups selected from group P ^111, and in the case of having two or more atoms or groups, the atoms or groups may be the same or different).
Group P ¹¹¹ : halogen atom, C 1 -C 6 alkyl group, C 1 -C 6 haloalkyl group, C 2 -C 6 alkenyl group, C 2 -C 6 haloalkenyl group, C 2 -C 6 alkynyl group, C 2 -C 6 haloalkynyl group, C 3 -C 6 cycloalkyl Group, C3-C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3 C6 haloalkynyl thio group, C2 to C6 alkyl carbonyl group, C2 to C6 halo alkyl carbonyl group, C2 to C6 alkyl carbonyloxy group, C2 to C6 alkyl carbonyl thio group, hydroxy carbonyl group, formyl group, C2 to C6 alkoxy carbonyl group, It may have a nitro group, cyano group, hydroxyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkyl group A group consisting of an amino group, an aminosulfonyl group which may have a C1-C6 alkyl group, and an aminocarbonyl group which may have a C1-C6 alkyl group.
Group P ¹¹² : halogen atom, cyano group, C3-C6 cycloalkyl group, C3-C6 halocycloalkyl group, C1-C4 alkoxy group, C1-C4 haloalkoxy group, C1-C4 alkylthio group and C1-C4 haloalkylthio group A group consisting of
Group P ¹¹³ : a group consisting of a C 1 -C 6 alkyl group, a C 1 -C 6 haloalkyl group, a C 3 -C 6 cycloalkyl group, and a C 3 -C 6 halocycloalkyl group. ]
A tetrazolinone compound represented by the formula:

Group (XII): Formula (12)
[In the formula,
R ²¹¹ is a C 1 -C 6 alkyl group, a C 3 -C 6 cycloalkyl group, a halogen atom, a C 1 -C 6 haloalkyl group, a C 2 -C 6 alkenyl group, a C 1 -C 6 alkoxy group, a C 1 -C 6 alkylthio group, a C 2 -C 6 alkynyl group, Nitro group, cyano group, aminocarbonyl group optionally having C1 to C6 alkyl group, C2 to C6 haloalkenyl group, C2 to C6 haloalkynyl group, C3 to C6 halocycloalkyl group, C1 to C6 haloalkoxy group , C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 halo Alkenyloxy group, C 3 -C 6 haloalkynyloxy group, C 3 -C 6 al Kenylthio group, C3-C6 alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 C6 alkylcarbonylthio group, C2-C6 alkoxycarbonyl group, hydroxyl group, thiol group, amino group which may have C1-C6 alkyl group, pentafluorosulfuranyl group, C3-C9 trialkylsilyl group, C5 -C14 trialkylsilylethynyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C2-C6 alkoxyalkyl group or C2-C6 alkylthio alkyl It represents a group;
R ²¹² , R ²¹³ and R ²¹⁴ are the same or different hydrogen atom, halogen atom, C 1 -C 3 alkyl group, C 1 -C 3 haloalkyl group, C 2 -C 3 alkenyl group, C 2 -C 3 haloalkenyl group or C 1 -C 3 alkoxy group Represent;
R ²¹⁵ represents a C1-C3 alkyl group optionally having one or more halogen atoms;
Y ¹² is —C (R ^A1 R ^A2 ) —Z—, —C (R ^A1 R ^A2 ) C (R ^A3 R ^A4 ) —Z—, —C (R ^A1 R ^A2 ) —Z—C (R ^A3 R ^A4 )-, -Z-C (R ^A1 R ^A2 ) C (R ^A3 R ^A4 )-, -C (R ^A1 R ^A2 ) C (R ^A3 R ^A4 ) C (R ^A5 R ^A6 ) -Z-, -C (R ^A1 R ^A2 ) C (R ^A3 R ^A4 ) -ZC (R ^A5 R ^A6 )-,-C (R ^A1 R ^A2 ) -ZC (R ^A3 R ^A4 ) C (R ^A5 R ^{A6) -, - Z-C} (R A1 R A2) C (R A3 R A4) C (R A5 R A6) -, - C (R A1) = C (R A2) C (R A3 R A4) - Z-, -Z-C (R ^A1 R ^A2 ) C (R ^A3 ) = C (R ^A4 )-, -C≡C-C (R ^A1 R ^A2 ) -Z-, -Z-C (R ^A1 R ^{A2) -C≡C -, - Z-} C (R A1 R A2) C (R A3 R ^{4) -Z -, - C (} R A1) = C (R A2) -, - C (R A1) = C (R A2) C (R A3 R A4) -, - C (R A1) = C ( R ^A2 ) C (R ^A3 R ^A4 ) C (R ^A5 R ^A6 )-,-C (R ^A1 R ^A2 ) C (R ^A3 ) = C (R ^A4 ) C (R ^A5 R ^A6 )-,-C ( R ^A1 R ^A2 ) C (R ^A3 R ^A4 ) C (R ^A5 ) = C (R ^A6 )-,-C (R ^A1 ) = C (R ^A2 ) C (R ^A3 ) = C (R ^A4 )-, -C≡C-, -C≡C-C (R ^A1 R ^A2 )-, -C≡C-C (R ^A1 R ^A2 ) C (R ^A3 R ^A4 )-, -C (R ^A1 R ^A2 ) C (R ^A3 R ^A4 ) -C-C- or -C (R ^A1 R ^A2 ) -C≡C-C (R ^A3 R ^A4 )-(however, the left end of each is bonded to Q ¹⁴ , R ^A1 , R ^A2 , R ^A3 , R ^A4 , R ^A5 , and R ^{A 6} are each a hydrogen atom, a halogen atom or a C1-C3 alkyl group, Z is an oxygen atom, a sulfur atom or NR ^{C, R C} are each C1-C6 alkyl group, C1-C6 haloalkyl group, C3-C6 A cycloalkyl group, or a C3-C6 halocycloalkyl group.
Q ¹⁴ is a divalent C 3 -C 10 carbocyclic group or a divalent heterocyclic group (provided that the divalent heterocyclic group is selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom as a ring constituent atom) A single or fused ring containing one or more atoms, which may be the same or different, and in the case of fused rings, 5- and 5-membered rings, 5- and 6-membered rings, and 6 A ring formed by condensing a membered ring and a 6-membered ring.
X ¹² represents an oxygen atom or a sulfur atom;
A ¹² represents a C 6 -C 10 aryl group, a C 6 -C 10 aryloxy group, a C 6 -C 10 arylthio group, a C 6 -C 10 arylsulfonyl group, a C 6 -C 10 arylamino group, a hydrogen atom or a heterocyclic group In the case of containing one or more atoms selected from the group consisting of nitrogen atoms, oxygen atoms and sulfur atoms as ring constituent atoms, and containing two or more atoms selected from the group consisting of nitrogen atoms, oxygen atoms and sulfur atoms Or the atoms may be the same or different from each other) or R ^C2 —O—NNC (R ^C2 ) — (wherein R ^C2 represents a C1 to C6 alkyl group, a C1 to C6 haloalkyl group, or a C3 to C6, respectively). And a cycloalkyl group or a C3-C6 halocycloalkyl group. (However, a divalent C3-C10 carbon group Q, and divalent to heterocyclic groups, as well as C6-C10 aryl group A ^12, C6-C10 aryloxy group, C6-C10 arylthio group, C6-C10 aryl The amino group and the heterocyclic group may have one or more atoms or groups selected from group P ¹²¹ )
Group P ¹²¹ : halogen atom, C1 to C6 alkyl group, C1 to C6 haloalkyl group, C2 to C6 alkenyl group, C2 to C6 haloalkenyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C3 to C6 cycloalkyl Group, C3-C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C -C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, hydroxycarbonyl group, formyl group, C2-C6 alkoxycarbonyl group , Nitro group, cyano group, hydroxyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkyl group A group consisting of an amino group, an aminosulfonyl group which may have a C1-C6 alkyl group, and an aminocarbonyl group which may have a C1-C6 alkyl group. ]
A tetrazolinone compound represented by the formula:

Group (XIII): Formula (13)
[Wherein, X ¹³ represents CR ²²⁶ or a nitrogen atom,
R ²²¹ , R ²²² , R ²²³ , R ²²⁴ and R ²²⁶ are each independently a halogen atom, a hydrogen atom, a cyano group, a C1-C4 alkyl group optionally having one or more halogen atoms, or one or more A C1-C4 alkoxy group which may have one or more halogen atoms,
R ²²⁵ represents a halogen atom, a C1 to C4 alkyl group optionally having one or more halogen atoms, a C3 to C4 cycloalkyl group optionally having one or more halogen atoms, or one or more halogen atoms And a C1-C4 alkoxy group which may have ]
A tetrazolinone compound represented by the formula:

Group (XIV): Formula (14)
[Wherein, A ¹⁴ represents the following group A 15, A 16, A 17 or A 18;

R ²³¹ is a hydrogen atom, a halogen atom, a C1 to C4 alkyl group optionally having one or more halogen atoms, a C3 to C4 cycloalkyl group optionally having one or more halogen atoms, or one or more A C1-C4 alkoxy group which may have one or more halogen atoms,
R ²³² and R ²³³ each represent a hydrogen atom, a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, or a C1-C4 alkoxy group optionally having one or more halogen atoms Represents
E ⁵⁹ and E ⁶¹ each represents a hydrogen atom, a halogen atom, a C 1 -C 4 alkoxy group which may have one or more halogen atoms, or a C 1-C 4 alkyl group which may have one or more halogen atoms Represent
E ⁵³ , E ⁵⁸ and E ⁶⁰ each represent a hydrogen atom, a C 1 -C 4 alkyl group optionally having one or more halogen atoms, or a C 3-C 4 cycloalkyl group optionally having one or more halogen atoms Represents
E ⁵⁰ , E ⁵¹ , E ⁵² , E ⁵⁴ , E ⁵⁵ , E ⁵⁶ and E ⁵⁷ each independently represent a hydrogen atom, a halogen atom, a cyano group, an aldehyde group, C1-C4 optionally having one or more halogen atoms It represents an alkoxy group, a C1 to C4 alkyl group optionally having one or more halogen atoms, or a C3 to C4 cycloalkyl group optionally having one or more halogen atoms. ]
A tetrazolinone compound represented by the formula:

Group (XV): Formula (15)
[Wherein, R ²⁴¹ and R ²⁴² each independently have a hydrogen atom, a halogen atom, a C 1 -C 4 alkyl group which may have one or more halogen atoms, or one or more halogen atoms. Represents a good C1-C4 alkoxy group;
R ²⁴³ is a hydrogen atom, a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or one or more Represents a C1-C4 alkoxy group which may have a halogen atom;
R ²⁴⁴ represents a halogen atom, a C1 to C4 alkyl group optionally having one or more halogen atoms, a C1 to C4 alkoxy group optionally having one or more halogen atoms, or a cyano group;
n ¹⁵ represents an integer from 0 to 4 (provided that, when n ¹⁵ is 2 or more integer, each of R ²⁴⁴ may be the same or different and at least one other of R ^244.) ;
X ¹⁵ represents a nitrogen atom or CR ²⁴⁵ ;
R ²⁴⁵ represents a hydrogen atom, a halogen atom, a C1 to C4 alkyl group optionally having one or more halogen atoms, a C1 to C4 alkoxy group optionally having one or more halogen atoms, or a cyano group. ]
A tetrazolinone compound represented by the formula:

Group (XVI): Formula (16)
[Wherein, R ²⁵¹ and R ²⁵² each independently represent a halogen atom, a C 1 -C 4 alkyl group which may have one or more halogen atoms, or C 3-which may have one or more halogen atoms. C4 cycloalkyl group, C2 to C4 alkenyl group optionally having one or more halogen atoms, C2 to C4 alkynyl group optionally having one or more halogen atoms, one or more halogen atoms Represents a C1-C4 alkoxy group which may be substituted, a C1-C4 alkylthio group which may have one or more halogen atoms, a cyano group or a nitro group (provided that m ¹⁶ is an integer of 2 or more, two or more And R ²⁵¹ may be the same or different, and when n ¹⁶ is an integer of 2 or more, two or more R ²⁵² may be the same or different.);
m ¹⁶ and n ¹⁶ each independently represent an integer of 0 to 4;
Each of R ²⁵³ and R ²⁵⁴ independently represents a hydrogen atom or a C1-C3 alkyl group optionally having one or more halogen atoms;
Y ¹⁶ represents a formula ^{-OC (= X 16) Z 16} R 255 or ^{-SC (= X 16) Z 16} R 255;
R ²⁵⁵ represents a C1-C3 alkyl group which may have one or more halogen atoms;
Z ¹⁶ represents an oxygen atom, a sulfur atom, NR ²⁵⁸ or a direct bond;
R ²⁵⁸ represents a C1-C3 alkyl group optionally having one or more halogen atoms or a hydrogen atom;
Q ¹⁶ represents a pyrazolyl group optionally having one or more atoms or groups selected from group P ¹³¹ ;
W ¹⁶ and X ¹⁶ each independently represent an oxygen atom or a sulfur atom.
Group P ¹³¹ : halogen atom, C1-C6 alkyl group optionally having one or more halogen atoms, C2-C6 alkenyl group optionally having one or more halogen atoms, one or more halogen atoms C2-C6 alkynyl group which may be substituted, C3-C6 cycloalkyl group which may have one or more halogen atoms, C1-C6 alkoxy group which may have one or more halogen atoms, one or more C 1 -C 6 alkylthio group which may have one or more halogen atoms, C 3 -C 6 cycloalkyloxy group which may have one or more halogen atoms, C 3-which may have one or more halogen atoms C6 cycloalkylthio group, C3 to C6 alkenyloxy group optionally having one or more halogen atoms, C3 to C6 alkynyl optionally having one or more halogen atoms Oxy group, C3-C6 alkenylthio group optionally having one or more halogen atoms, C3-C6 alkynylthio group optionally having one or more halogen atoms, one or more halogen atoms C2 to C6 alkyl carbonyl group which may be substituted, C2 to C6 alkyl carbonyloxy group which may have one or more halogen atoms, C2 to C6 alkyl carbonyl thio group which may have one or more halogen atoms, A carboxy group, a formyl group, a C2-C6 alkoxycarbonyl group which may have one or more halogen atoms, a nitro group, a cyano group, and an amino group which may have a C1-C6 alkyl group (provided that the An alkyl group may have one or more halogen atoms); ]
An aromatic compound represented by

Group (XVII): Formula (17)
[Wherein, R ²⁶¹ represents a halogen atom or a C 1 -C 4 alkyl group which may have one or more halogen atoms;
R ²⁶³ represents a hydrogen atom or a C1-C4 alkyl group optionally having one or more halogen atoms;
R ²⁶⁷ is a C1-C3 alkyl group which may have one or more halogen atoms, a hydrogen atom, a halogen atom, a C1-C3 alkoxy group which may have one or more halogen atoms, one or more halogen atoms A C3-C4 cycloalkyl group optionally having one or more C2-C4 alkenyl groups optionally having one or more halogen atoms;
Z ¹⁷ represents a halogen atom, a C1-C3 alkoxy group or a C1-C3 alkyl group;
Z ¹⁸ represents a C1-C3 alkyl group optionally having one or more halogen atoms or a halogen atom;
Q ¹⁷ represents the following groups Q 18, Q 19 or Q 20;
R ²⁶⁵ represents a C1-C3 alkyl group optionally having one or more halogen atoms;
R ²⁷⁰ represents a hydrogen atom, a hydroxyl group or a methyl group;
R ²⁷¹ represents a hydrogen atom, a hydroxyl group, a methyl group or a methoxy group;
X ¹⁷ represents an oxygen atom or a sulfur atom;
X ¹⁸ represents an oxygen atom, a sulfur atom, NR ²⁷² or a direct bond;
R ²⁷² represents a C1-C3 alkyl group optionally having one or more halogen atoms, or a hydrogen atom. ]
An aromatic compound represented by

Group (XVIII): Formula (18)
[Wherein, R ²⁸¹ represents a halogen atom or a C 1 -C 4 alkyl group which may have one or more halogen atoms;
R ²⁸³ represents a hydrogen atom, a halogen atom or a C1-C4 alkyl group optionally having one or more halogen atoms;
R ²⁸⁷ is a C1-C3 alkyl group which may have one or more halogen atoms, a hydrogen atom, a halogen atom, a C1-C3 alkoxy group which may have one or more halogen atoms, or one or more halogen atoms Represents a C3-C4 cycloalkyl group which may have
A ¹⁸ represents the following groups A 19, A 20 or A 21;
Each of Z ¹⁹ and Z ²⁰ independently represents a halogen atom, a C 1 -C 3 alkyl group which may have one or more halogen atoms, or a C 1 -C 3 alkoxy group which may have one or more halogen atoms. Represent;
Q ²¹ represents the following groups Q ^22, Q 23 or Q 24;
R ²⁸⁵ represents a C1-C3 alkyl group optionally having one or more halogen atoms;
R ²⁹⁰ represents a hydrogen atom, a hydroxyl group or a methyl group;
R ²⁹¹ represents a hydrogen atom, a hydroxyl group, a methyl group or a methoxy group;
X ¹⁹ represents an oxygen atom or a sulfur atom;
X ²⁰ represents an oxygen atom, a sulfur atom, NR ²⁹² or a direct bond;
R ²⁹² represents a C1-C3 alkyl group optionally having one or more halogen atoms, or a hydrogen atom. ]
An aromatic compound represented by

Group (XIX): Formula (19)
[In the formula,
R ³⁰¹ represents a hydrogen atom or a C1-C3 alkyl group;
Each of R ³⁰² , R ³⁰³ , R ³⁰⁴ and R ³⁰⁵ independently has a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms. A C3-C4 cycloalkyl group which may be substituted or a C1-C3 alkoxy group which may have one or more halogen atoms;
Z ²¹ represents a C1-C3 alkyl group;
n ¹⁹ represents an integer of 1 to 4; ]
The carbamate compound shown by these.

Group (XX): Formula (20)
[In the formula,
R ³¹¹ represents a hydrogen atom or a C1-C3 alkyl group;
Each of R ³¹² , R ³¹³ , R ³¹⁴ and R ³¹⁵ independently has a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms A C3-C4 cycloalkyl group which may be substituted or a C1-C3 alkoxy group which may have one or more halogen atoms;
Z ²² represents a halogen atom;
Z ²³ represents a halogen atom or a C1-C3 alkyl group;
n ²⁰ represents an integer of 0 to 3; ]
The carbamate compound shown by these.

Group (XXI): Formula (21)
[In the formula,
R ³²¹ represents a hydrogen atom or a C1-C3 alkyl group;
Each of R ³²² , R ³²³ , R ³²⁴ and R ³²⁵ independently has a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms. A C3-C4 cycloalkyl group which may be substituted or a C1-C3 alkoxy group which may have one or more halogen atoms;
Z ²⁴ represents a C1-C3 alkyl group;
n ²¹ represents an integer of 1 to 3; ]
The carbamate compound shown by these.

Group (XXII): Formula (22)
[In the formula,
R ³³¹ represents a hydrogen atom or a C1-C3 alkyl group;
Each of R ³³² , R ³³³ , R ³³⁴ and R ³³⁵ independently has a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms. A C3-C4 cycloalkyl group which may be substituted or a C1-C3 alkoxy group which may have one or more halogen atoms;
Z ²⁵ represents a halogen atom;
Z ²⁶ represents a halogen atom or a C1-C3 alkyl group;
n ²² represents an integer of 0 to 2; ]
The carbamate compound shown by these.

Group (XXIII): Formula (23)
[Wherein, R ³⁴¹ represents a hydrogen atom or a C1-C3 alkyl group;
Each of R ³⁴² , R ³⁴³ , R ³⁴⁴ and R ³⁴⁵ independently has a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or one or more halogen atoms A C3-C4 cycloalkyl group which may be substituted or a C1-C3 alkoxy group which may have one or more halogen atoms;
Z ²⁷ represents a halogen atom, a C1-C3 alkyl group or a C1-C3 alkoxy group;
n ²³ represents an integer of 0 to 3; ]
The carbamate compound shown by these.
[2] Effective dose of [1] described group (I), group (II), group (III), group (IV), group (V), group (VI), group (VII), group (VIII) , Group (IX), Group (X), Group (XI), Group (XII), Group (XIII), Group (XIV), Group (XV), Group (XVI), Group (XVI), Group (XVII), Group (XVIII) , A group (XIX), a group (XX), a group (XXI), a group (XXII), and a group (XXIII), and the tetrazolinone compound according to any one of the group consisting of Or a method of controlling a pest comprising the step of applying one or more components selected from the group consisting of Group F to a plant or a soil for cultivating a plant.
[3] The pest control method according to [2], wherein the plant is a seed, a bulb or a seedling.
[4] The pest control method according to [2], wherein the plant is corn, soybean, cotton, wheat, barley, sugar beet, Brassica napus or rice.
[5] Effective dose of [1] described group (I), group (II), group (III), group (IV), group (V), group (VI), group (VII), group (VIII) , Group (IX), Group (X), Group (XI), Group (XII), Group (XIII), Group (XIV), Group (XV), Group (XVI), Group (XVI), Group (XVII), Group (XVIII) , A group (XIX), a group (XX), a group (XXI), a group (XXII), and a group (XXIII), and the tetrazolinone compound according to any one of the group consisting of And a method of controlling a pest comprising the step of applying one or more components selected from the group consisting of Group F to a pest or a habitat of the pest.
[6] Plant seeds or bulbs to which an effective amount of the pest control composition as described in [1] is attached.

  According to the present invention, pests can be controlled.

  The composition of the present invention contains the present compound and one or more components selected from the group consisting of Group A to Group F.

  First, the present compound will be described.

The substituents in the present specification will be described.
In the present specification,
The "optionally having one or more halogen atoms" means that, when having two or more halogen atoms, those halogen atoms may be the same as or different from each other.
In the present specification, for example, "C1-C3" means that the number of carbon atoms is 1 to 3.

  The halogen atom represents a fluorine atom, a chlorine atom, a bromine atom and an iodine atom.

In the present specification, Me represents methyl, Et represents ethyl, Pr represents propyl, i-Pr represents isopropyl, CF ₃ represents trifluoromethyl, and OCF ₃ represents trifluoromethoxy, CHF ₂ represents difluoromethyl, OCHF ₂ represents difluoromethoxy, OMe represents methoxy, OEt represents ethoxy, c-Pr represents cyclopropyl, NO ₂ represents a nitro group, F represents fluoro, Cl is chloro, Br is bromo, I is iodo, CN is cyano, SMe is methylthio, SEt is ethylthio, 2-Py is pyridin-2-yl, 3- 3- Py represents pyridin-3-yl, 4-Py represents pyridin-4-yl, 2-PYM represents pyridin-2-yl, S (O) Me represents methylsulfinyl, S (O) ) ₂ Me represents methyl sulfonyl, SCF ₃ is a trifluoromethylthio Table , S (O) CF ₃ represents a trifluoromethyl sulfinyl, S (O) ₂ CF ₃ represents a trifluoromethylsulfonyl, COOMe represents methoxycarbonyl, NO ₂ represents a nitro, NH ₂ represents an amino , NHMe represents methylamino, NMe ₂ represents dimethylamino, AC represents acetyl, ACNH represents acetylamino, N-AC-N-Me-N represents N-acetyl-N-methylamino, PYR represents pyrazole, 1-PYR represents pyrazole-1-yl group, 3-PYR represents pyrazole-3-yl group, 4-PYR represents pyrazole-3-yl group, TRI represents triazole 1-TRI represents 1,2,3-triazol-1-yl, 2-TRI represents 1,2,3-triazol-2-yl, TET represents tetrazole, THI represents thiophene, 2 -THI represents thiophen-2-yl, 3-THI represents thiophen-3-yl, FU R represents furan, 2-FUR represents furan-2-yl, 3-FUR represents furan-3-yl, THA represents thiazole, 2-THA represents thiazol-2-yl, 4- THA stands for thiazol-4-yl, 5-THA stands for thiazol-5-yl, OXA stands for oxazole, 2-OXA stands for oxazol-2-yl, 3-OXA stands for oxazol-3-yl 4-OXA represents oxazol-4-yl, IMI represents imidazole, PRL represents pyrrole, TDA represents tizadiazole, 1-Ph represents a benzene-1-yl group, and 2-QY represents quinoline -2-yl group, 3-QY represents quinolin-3-yl group, 6-QY represents quinolin-6-yl group, 7-QY represents quinolin-7-yl group, and diF represents difluoro , DiCl represents dichloro and diOMe dimethoxy.

  First, the synthesis method of the present compound will be described.

  The compound is an compound of WO 2013/162077, WO 2014/051165, WO 2014/051161, WO 2014/084223, WO 2014/104268, WO 2014/104382. And can be synthesized according to the methods described in WO 2014/104384 and the methods described.

  Moreover, this compound can also be manufactured according to the method as described in the following manufacturing method A-manufacturing method C, and the described method, for example.

(Manufacturing method A)
The present compound represented by the formula (4) can be produced by reacting the compound represented by the formula (41) with the compound represented by the formula (42) in the presence of a base.
[Wherein, R ⁶¹ , R ⁶² , R ⁶³ , R ⁶⁴ , R ⁶⁵ , R ⁶⁶ , R ⁶⁷ , X ⁴ , A ⁴ and Q ⁴ are as defined above, and Z ¹ is a chlorine atom, a bromine atom, etc. Represents a leaving group of ]

  The reaction is usually carried out in a solvent.

  Examples of the solvent used for the reaction include ethers such as tetrahydrofuran, 1,4-dioxane, ethylene glycol dimethyl ether and the like, nitriles such as acetonitrile, acid amides such as N, N-dimethylformamide, N-methylpyrrolidone and the like. These mixtures are mentioned.

  As a base used for the reaction, alkali metal carbonates such as sodium carbonate and potassium carbonate, alkali metal hydroxides such as sodium hydroxide and potassium hydroxide, alkali metal hydrides such as sodium hydride, sodium t-butoxide And alkali metal alkoxides such as potassium t-butoxide.

  In the reaction, the compound (42) is usually used in a proportion of 1 to 10 moles, and the base is usually used in a proportion of 0.5 to 5 moles, relative to 1 mole of the compound (41).

  The reaction temperature of the reaction is usually in the range of -20 to 150 ° C. The reaction time of the reaction is usually in the range of 0.1 to 24 hours.

  In the reaction, if necessary, sodium iodide, tetrabutylammonium iodide and the like may be added, and these compounds usually have a ratio of 0.001 to 1.2 moles relative to 1 mole of the compound (41) Used in

  After completion of the reaction, the reaction mixture can be extracted with an organic solvent, and the organic layer can be subjected to post-treatment procedures such as drying and concentration to isolate the compound (4). The isolated compound can also be further purified by chromatography, recrystallization and the like.

(Manufacturing method B)
The present compound represented by the formula (6) can be produced in the following three steps

(Step 1)
Compound (63) can be produced by reacting compound (61) with compound (62) in the presence of a base.
[Wherein, R ¹⁰¹ , R ¹⁰² , R ¹⁰³ , R ¹⁰⁴ , R ¹⁰⁵ , R ¹⁰⁶ , R ¹⁰⁷ , R ¹⁰⁸ , R ¹⁰⁹ , R ¹¹⁰ , R ¹¹⁰ , R ¹¹¹ and X ⁶ are as defined above, and Z ³ is Represents a chlorine atom, a bromine atom or an iodine atom, and the other symbols have the same meanings as described above. ]
The reaction can be carried out according to the reaction described in Production Method A.

(Step 2)
Compound (64) can be produced by reacting compound (63) with a borylation reagent in the presence of a catalyst and a base.
[Wherein, Z ² represents an alkoxyboranyl group, and the other symbols have the same meanings as described above. ]
The reaction is usually carried out in a solvent.

  Examples of the solvent used for the reaction include acid amides such as N, N-dimethylformamide, 1,3-dimethyl-2-imidazolidinone and N-methyl pyrrolidone, and sulfoxides such as dimethyl sulfoxide.

  Examples of borylation reagents used in the reaction include bis (pinacolato) diboron, pinacolborane and the like.

  Examples of the catalyst used in the reaction include palladium (II) acetate, dichlorobis (triphenylphosphine) palladium, tetrakistriphenylphosphinepalladium (0), bis (diphenylphosphane ferrocenyl) palladium (II) dichloride Be

  Examples of the base used for the reaction include alkali metal hydrogen carbonates such as potassium acetate and sodium acetate.

  In the reaction, the borylation reagent is usually used in a proportion of 1 to 10 moles, the base is usually in a proportion of 1 to 10 moles, and the catalyst is usually in a proportion of 0.0001 to 1 mole relative to 1 mole of the compound (B1).

  The reaction temperature of the reaction is usually in the range of 0 to 150 ° C. The reaction time of the reaction is usually in the range of 0.1 to 24 hours.

  After completion of the reaction, the reaction mixture can be extracted with an organic solvent, and the organic layer can be subjected to post-treatment procedures such as drying and concentration to isolate the compound (C1). Furthermore, purification may be performed by distillation, chromatography, recrystallization or the like.

(Step 3)
The present compound represented by the formula (6) can be produced by subjecting the compound represented by the formula (64) and the compound represented by the formula (65) to a coupling reaction in the presence of a base and a catalyst.
Wherein the symbols have the same meanings as described above. ]
The reaction is usually carried out in a solvent.

  Examples of the solvent used for the reaction include ethers such as tetrahydrofuran, 1,4-dioxane, ethylene glycol dimethyl ether and the like, acid amides such as N, N-dimethylformamide, N-methylpyrrolidone and the like, water and mixtures thereof. It can be mentioned.

  As the compound (65) used for the reaction, generally commercially available ones can be used.

  As a catalyst used for the reaction, palladium (II) acetate, dichlorobis (triphenylphosphine) palladium, tetrakistriphenylphosphine palladium (0), palladium (II) acetate / triscyclohexylphosphine, bis (diphenylphosphane ferrocenyl) And the like) palladium (II) dichloride and the like.

  Examples of the base used for the reaction include organic bases such as pyridine, alkali metal halides such as sodium fluoride, potassium fluoride and cesium fluoride, alkali metal phosphates such as tripotassium phosphate, sodium methoxide, sodium And alkali metal alkoxides such as ethoxide, sodium t-butoxide and potassium t-butoxide.

  In the reaction, the compound (65) is usually used at a ratio of 1 to 10 moles, the base is usually at a ratio of 1 to 10 moles, and the catalyst is usually at a ratio of 0.0001 to 1 mole per 1 mole of the compound (64). Be

  The reaction temperature of the reaction is usually in the range of 0 to 150 ° C. The reaction time of the reaction is usually in the range of 0.1 to 24 hours.

  After completion of the reaction, the reaction mixture is extracted with an organic solvent, and the organic layer is subjected to post-treatment procedures such as drying and concentration to isolate the compound (6). The isolated compound can also be further purified by chromatography, recrystallization and the like.

As an aspect of this compound in this invention composition, the compound which is shown below, for example is mentioned.
A tetrazolinone compound according to any of group (I).
A tetrazolinone compound according to any of group (II).
A tetrazolinone compound according to any of group (III).
A tetrazolinone compound according to any one of group (IV).
A tetrazolinone compound according to any one of group (V).
A tetrazolinone compound according to any of group (VI).
A tetrazolinone compound according to any of group (VII).
A tetrazolinone compound according to any one of group (VIII).
A tetrazolinone compound according to any one of group (IX).
A tetrazolinone compound according to any one of group (X).
A tetrazolinone compound according to any of group (XI).
A tetrazolinone compound according to any one of group (XII).
A tetrazolinone compound according to any of group (XIII).
The tetrazolinone compound as described in any of the group (XIV).
The tetrazolinone compound in any one of a group (XV).
An aromatic compound according to any one of the group (XVI).
An aromatic compound according to any one of group (XVII).
An aromatic compound according to any of group (XVIII).
The carbamate compound as described in any of the group (XIX).
The carbamate compound as described in any of the group (XX).
The carbamate compound as described in any of group (XXI).
The carbamate compound as described in any of the group (XXII).
The carbamate compound as described in any of the group (XXIII).

  The present invention will next be described in more detail by way of synthesis examples of the present compound, formulation examples of the present composition, test examples and the like, but the present invention is not limited to these examples.

  First, a synthesis example of the present compound is shown.

Synthesis example 1
1.18 g of 1-[(2-bromomethyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, 0.71 g of 4-phenyl-2-oxo-thiazole, 0.61 g of potassium carbonate and 20 mL of acetonitrile The mixture was stirred under heating reflux for 5 hours. The reaction mixture was allowed to cool, poured into water, and extracted with ethyl acetate. The organic layer was washed with water and saturated brine, dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The resulting residue is subjected to silica gel column chromatography to give 1- (2-{[(4-phenylthiazol-2-yl) oxy] methyl})-4-methyl-1,4-dihydrotetrazol-5-one Was obtained 0.08g.
¹ H-NMR (CDCl ₃ ) δ: 7.79-7.77 (2H, m), 7.74-7.72 (1H, m), 7.57-7.47 (3H, m), 7.39 (2H, t, J = 7.3 Hz), 7.30 (1 H, t, J = 7.3 Hz), 6. 85 (1 H, s), 5. 64 (2 H, s), 3. 64 (3 H, s).

Synthesis example 2
0.59 g of 1- (2-bromomethyl-3-chlorophenyl) -4-methyl-1,4-dihydrotetrazol-5-one, 0.38 g of 1-[(3-difluoromethyl) phenyl] ethanone oxime, potassium carbonate The mixture of 0.35 g and 10 mL of acetonitrile was stirred for 7 hours while heating to reflux. Cool to room temperature, filter the reaction mixture and concentrate the filtrate. The resulting residue is subjected to silica gel column chromatography to give 1- (3-chloro-2- {1-[[{[(3-difluoromethyl) phenyl] ethylidene} amino] oxy] methyl] phenyl] -4- Methyl-1,4-dihydrotetrazol-5-one was obtained.
¹ H-NMR (CDCl ₃ ) δ: 7.71 (1 H, s), 7.65 (1 H, d, J = 7.2 Hz), 7.60 (1 H, d, J = 7.2 Hz), 7.51-7.41 (3 H, m), 7.33 (1 H, d, J = 7.2 Hz), 6.67 (1 H, t, J = 56 Hz), 5.46 (2 H, s), 3.61 (3 H, s), 2.10 (3 H, s).

Synthesis example 3
1- [2- (2-bromopyridin-6-yloxymethyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one 0.27 g, 2-methyl-4- (1 A mixture of 0.16 g of -methoxyimino-propyl) phenol, 0.28 g of potassium carbonate and 10 mL of acetonitrile was stirred for 4 hours under heating to reflux. Cool to room temperature, filter the reaction mixture and concentrate the filtrate. The resulting residue is subjected to silica gel column chromatography to give 1- [2-({2-methyl-4-[(1-methoxyimino) propyl] phenoxy} methyl) phenyl] -4-methyl-1,4- 0.24 g of dihydrotetrazol-5-one was obtained.
¹ H-NMR (CDCl ₃ ) δ: 7.68 (1 H, d, J = 6.76 Hz), 7.55-7.48 (3 H, m), 7.46-7.46 (1 H, m), 7.35 (1 H, dd, J = 8.45, 2.41 Hz), 6.77 (1 H, d, J = 8.45 Hz), 5. 18 (2 H, s), 3. 95 (3 H, s), 3. 67 (3 H, s), 2. 69 (2 H, q, J = 7.57 Hz), 2.20 (3H, s), 1.10 (3H, t, J = 7.57 Hz).

Synthesis example 4
0.40 g of 1- [2- (2-bromopyridine methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, 0.19 g of phenylboronic acid, tripotassium phosphate 0. A mixture of 68 g, 0.10 ml of water, 0.09 g of [1,1′-bis (diphenylphosphino) ferrocene] palladium (II) dichloride dichloromethane adduct and 5 mL of dioxane was stirred under heating reflux for 6 hours. After cooling, water was poured into the reaction solution and extracted with ethyl acetate. The organic layer was washed with water and saturated brine, dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The resulting residue is subjected to silica gel column chromatography to give 1-methyl-4- (3-methyl-2-{[(6-phenylpyridin-2-yl) oxy] methyl} phenyl) -1,4-dihydro 0.32 g of tetrazole-5-one was obtained.
1 H-NMR (CDCl 3) δ: 8.00-7.97 (2H, m), 7.59 (1H, dd, J = 8.0, 7.6 Hz), 7.48-7.44 (2H, m), 7.42-7.36 (3H, m), 7.33 (1H, d, J = 7.6 Hz), 7.26-7.22 (1H, m), 6.60 (1H, d, J = 8.0 Hz), 5.53 (2H, s), 3.49 (3H, s), 2.54 (3H, 5) s).

Synthesis example 5
0.28 g of 1-[(2-bromomethyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, 0.27 g of 2- (4-hydroxy-3-methylphenyl) -4-methylpyridine, A mixture of 0.20 g of potassium carbonate and 10 mL of acetonitrile was stirred for 5 hours while heating to reflux. Cool to room temperature, filter the reaction mixture and concentrate the filtrate. The resulting residue is subjected to silica gel column chromatography to give 1- {2- [2-methyl-4- (4-methylpyridin-2-yl) -phenoxymethyl] phenyl} -4-methyl-1,4- 0.27 g of dihydrotetrazol-5-one was obtained.
¹ H-NMR (CDCl ₃ ) δ: 2.25 (3 H, s), 2. 34 (3 H, s), 3.62 (3 H, s), 5. 20 (2 H, s), 6. 86 (1 H, d, J = 8.5 Hz) 6.95 (1 H, ddd, J = 5.0, 1.5, 0.7 Hz), 7.42-7.53 (4 H, m), 7.67-7.73 (2 H, m), 7.82 (1 H, dd, J = 1.5, 0.7 Hz), 8.48 ( 1 H, d, J = 5.0 Hz).

Synthesis example 6
A mixture of 0.28 g of 1- (2-bromomethyl-3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one, 0.17 g of p-hydroxybiphenyl, 0.28 g of potassium carbonate and 4 mL of acetonitrile The reaction mixture was stirred for 4 hours while heating under reflux. After cooling, water was poured into the reaction solution and extracted with ethyl acetate. The organic layer was washed with water and saturated brine, dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The resulting residue was subjected to silica gel column chromatography to give 1- {2-[(4-phenylphenoxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one 0. I got 30g.
¹ H-NMR (CDCl ₃ ) δ: 7.55 to 7.47 (4H, m), 7.42 to 7.37 (4H, m), 7.30 to 7.27 (2H, m), 6.96 to 6.92 (2H, m), 5.06 (2H, 2) s), 3.58 (3H, s), 2.49 (3H, s).

Synthesis example 7
0.44 g of 1- [2- (5-bromopyridin-2-yloxymethyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, 0.09 g of phenol, iodinated A mixture of 0.02 g copper, 0.06 g N-butylimidazole, 0.28 g potassium carbonate and 2 mL toluene was stirred at 120 ° C. for 16 hours. The reaction solution was poured into water and extracted with chloroform. The organic layer was washed with water and saturated brine, dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The resulting residue is subjected to silica gel column chromatography to give 1- [2-({[(5-phenoxypyridin-2-yl) oxy] methyl) -3-methylphenyl] -4-methyl-1,4- There were obtained 0.15 g of dihydrotetrazol-5-one.
¹ H-NMR (CDCl ₃ ) δ: 7.86 (1 H, d, J = 3.0 Hz), 7.43-7. 37 (2 H, m), 7. 35-7. 29 (2 H, m), 7. 28-7. 24 (2 H, m), 7.11 -7.05 (1H, m), 6.95-6.93 (2H, m), 6.66 (1H, d, J = 8.9 Hz), 5.35 (2H, s), 3.68 (3H, s), 2.56 (3H, s).

Synthesis example 8
1- (2-{[(1H-pyrazol-3-yl)] oxymethyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one 0.3 g, 1-methyl-indole A mixture of 0.21 g, 0.53 g iodine, 2 mL saturated aqueous ammonium formate and 2 mL acetonitrile was stirred at room temperature for 4 hours. The reaction mixture was poured into water and extracted with ethyl acetate. The organic layer was washed with water and saturated brine, dried over anhydrous sodium sulfate and concentrated under reduced pressure. The resulting residue is subjected to silica gel column chromatography to give 1- [3-methyl-2-({[1- (1-methylindol-2-yl) -1H-pyrazol-3-yl] oxy} methyl) 0.12 g of phenyl] -4-methyl-1,4-dihydro-tetrazol-5-one was obtained.
¹ H-NMR (CDCl ₃ ) δ: 7.62-7.60 (1H, m), 7.52 (1H, d, J = 2.1 Hz), 7.58-7.21 (5H, m), 7.15-7.11 (1H, m), 6.49 -6.48 (1H, m), 5.57 (1H, d, J = 2.1 Hz), 5.18 (2H, s), 3.49 (3H, s), 3.43 (3H, s), 2.39 (3H, s).

Synthesis example 9
1- (2-{[(4-bromo-2-methyl) phenoxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one 0.5 g, copper iodide (I A mixture of 0.05 g of cesium carbonate, 0.83 g of cesium carbonate, 0.17 g of pyrrole, and 2 ml of N, N-dimethylformamide was stirred at 120 ° C. for 40 hours. The reaction was diluted with ethyl acetate and washed with water. The organic layer is dried over anhydrous magnesium sulfate and then concentrated under reduced pressure, and the residue is chromatographed on silica gel to give 1- (3-methyl-2-{[2-methyl-4- (pyrrol-1-yl)]. 0.18 g of phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one was obtained.
¹ H-NMR (CDCl ₃ ) δ: 7.46-7.40 (2H, m), 7.30-7.25 (1H, m), 7.14-7.13 (2H, m), 6.98 (2H, t, J = 2.2 Hz), 6.86 (1H, d, J = 8.6 Hz), 6.31 (2H, t, J = 2.3 Hz), 5.05 (2H, s), 3.64 (3H, s), 2.52 (3H, s), 2.13 (3H, s) .

The present compounds produced according to the above synthesis examples are shown below.

1- {2-[({1- [2- (trichloroacetoxy) -1,1-dimethylethyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38-7.33 (2H, m), 7.24 (1 H, d, J = 2.5 Hz), 7.22 (1 H, dd, J = 6.3 , 2.9 Hz), 5.52 (1H, d, J = 2.5 Hz), 5.19 (2H, s), 4.44 (2H, s), 3.69 (3H, s), 2.52 (3H, s), 1.58 (6H, s) 1). [1- (2-[{[1- (2,6-dimethylpyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1). , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 (1 H, d, J = 8.0 Hz), 7.42-7.37 (2 H, m), 7.33 (1 H, d, J = 2.3 Hz), 7.26-7.24 (1H, m), 7.08 (1H, d, J = 8.0 Hz), 5.79 (1H, d, J = 2.5 Hz), 5.29 (2H, s), 3.59 (3H, s), 2.58 (3H, s), 2.55 (3H, s), 2.46 (3H, s). 1- {2-[({1- [6- (Cyclopropylmethoxy) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.30 (1 H, d, J = 2.5 Hz), 7.81 (1 H, dd, J = 8.9, 3.0 Hz), 7.56 (1 H, d , J = 2.5 Hz), 7.41-7.37 (2H, m), 7.26-7.24 (1 H, m), 6.83 (1 H, d, J = 8.9 Hz), 5.80 (1 H, d, J = 2.5 Hz), 5.32 (2H, s), 4.14 (2H, d, J = 7.1 Hz), 3.64 (3H, s), 2.56 (3H, s), 1.32-1.28 (1H, m), 0.64-0.62 (2H, m), 0.38-0.36 (2H, m) .; 1- {2-[({1- [3- (1,1-dimethylethoxy) -2-methoxypyridin-4-yl] -1H-pyrazol-3-yl} Oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.03 (1 H, d, J = 2.7 Hz), 7.90 ( 1H, d, J = 5. 5 Hz), 7.42-7.37 (2 H, m), 7. 28-7. 24 (1 H, m), 7.22 (1 H, d, J = 5.5 Hz), 5.81 (1 H, d, J = 2.5 Hz), 5.34 (2 H, 5 H) s), 3.98 (3H, s), 3.64 (3H, s), 2.55 (3H, s), 1.19 (9H, s) .; 1- [2-({[1- (2-acetoxy-1,1), 1. -Dimethylethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38 -7.33 (2H, m), 7.23-7.22 (2H, m), 5.51 (1H, d, J = 2.5 Hz), 5.20 (2H, s), 4.19 (2H, s), 3.69 (3H, s), 2.53 (3H, s), 1.99 (3H, s), 1.50 (6H, s) .; 1- [2-({[1- (2-methylpyridin-3-yl) -1H-pyrazol-3-yl] ] Oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.51 (1 H, dd, J = 4.8, 1.6 Hz) , 7.62 (1 H, dd, J = 7.8, 1.6 Hz), 7.41-7.38 (3 H, m), 7.25-7.23 (2 H, m), 5.82 (1H, d, J = 2.5 Hz), 5.31 (2H, s), 3.58 (3H, s), 2.55 (3H, s), 2.53 (3H, s) .; 1- {2- [ ({1- [5- (Difluoromethoxy) pyridin-2-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 8.26 (1 H, d, J = 2.9 Hz), 8. 20 (1 H, d, J = 2.7 Hz), 7. 77 (1 H, d, J = 9.1 Hz), 7.58 ( 1H, dd, J = 8.8, 2.7 Hz), 7.43-7.38 (2H, m), 7. 29-7. 25 (1 H, m), 6.53 (1 H, t, J = 72.7 Hz), 5. 85 (1 H, d, J = 2.7 Hz), 5.33 (2H, s), 3.66 (3H, s), 2.56 (3H, s) .; 1- [2-({[1- (3-butoxy-2-methoxypyridin-4-yl). -1H-Pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.26 (1 H, d , J = 2.7 Hz), 7.88 (1 H, d, J = 5.7 Hz), 7.42-7.39 (3H, m), 7.28-7.25 (1H, m), 5.84 (1H, d, J = 2.7 Hz), 5.33 (2H, s), 4.02 (3H, s), 3.93 (2H, t, J = 6.8 Hz), 3.64 (3 H, s), 2.56 (3 H, s), 1.74-1.67 (2 H, m), 1.44-1. 41 (2 H, m), 0.93 (3 H, t, J = 7.4 Hz). 1- (3-methyl-2-{[2-methyl-4- (1-propyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole-5 -ON, ¹ H-NMR (CDCl ₃ ) δ: 7.58 to 7.57 (1 H, m), 7.53 (1 H, dd, J = 8.2, 2.3 Hz), 7.43-7.38 (2 H, m), 7.36 (1 H, d) , J = 2.1 Hz), 7.27 (1 H, dd, J = 6.4, 2.1 Hz), 6.85 (1 H, d, J = 8.5 Hz), 6.43 (1 H, d, J = 2.3 Hz), 5.06 (2 H, s ), 4.10 (2H, q, J = 7.2 Hz), 3.61 (3H, s), 2.50 (3H, s), 2.12 (3H, s), 1.96-1.87 (2H, m), 0.94 (3H, t, J = 7.4 Hz) .; 1- [3-Methyl-2-({2,5-dimethyl-4- [1- (2,2-difluoroethyl) -5-methyl-1 H-pyrazol-3-yl]. Fenoki } Methyl) phenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.45-7.39 (2H, m), 7.31-7.27 (2H, m), 6.69 (1H, s), 6.31-6.01 (1H, m), 6.14 (1H, s), 5.04 (2H, s), 4.40 (2H, td, J = 13.2, 4.4 Hz), 3.64 (3H, s), 2.51 (3H, s), 2.41 (3H, s), 2.34 (3H, s), 2.06 (3H, s).

1- [2-({[1- (2-bromo-4-chlorophenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole- 5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.67 (1 H, d, J = 2.5 Hz), 7.63 (1 H, d, J = 2.5 Hz), 7.43-7.36 (4 H, m), 7.25 (1 H , m), 5.82 (1 H, d, J = 2.5 Hz), 5. 29 (2 H, s), 3.62 (3 H, s), 2.55 (3 H, s) .; 1- [2-({[1- (4) -Chloro-3-methoxyphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ δ: 7.65 (1H, d, J = 2.7 Hz), 7.39-7.33 (3H, m), 7.25 (2H, m), 6.99 (1H, dd, J = 8.6, 2.4 Hz), 5.81 (1H, d) , J = 2.7 Hz), 5.33 (2H, s), 3.97 (3H, s), 3.61 (3H, s), 2.56 (3H, s) .; 1- {2-[({1- [6-methoxy] -2- (trifluoromethyl) Pyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ : 7.74 (1H, d, J = 8.6 Hz), 7.38 (3H, m), 7.26 (1 H, s), 7.00 (1 H, d, J = 8.6 Hz), 5.81 (1 H, d, J = 2.5 Hz) , 5.26 (2H, s), 4.02 (3H, s), 3.62 (3H, s), 2.54 (3H, s) .; 1- {2-[({1- [1,1-dimethyl-2- (2)] Ethoxyimino) ethyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 (1H, s), 7.37-7.35 (2H, m), 7.25-7.20 (2H, m), 5.54 (1H, d, J = 2.3 Hz), 5.21 (2H, s), 4.10 (2H, q, J = 7.1 Hz), 3.68 (3 H, s), 2.53 (3 H, s), 1. 64 (6 H, s), 1.25 (3 H, t, J = 7.1 Hz). 1- [2-({[1-] (3-methoxypyridin-4-yl) -1H-pyra Lumpur-3-yl] oxy} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.36 (1H, s), 8.29 (1H, d, J = 5.3 Hz), 8.22 (1H, d, J = 2.7 Hz), 7.79 (1 H, d, J = 5.3 Hz), 7.43-7.38 (2H, m), 7.28-7.26 (1H , m), 5.84 (1H, d, J = 2.7 Hz), 5.34 (2H, s), 4.03 (3H, s), 3.64 (3H, s), 2.56 (3H, s). ({[1- (thiophen-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H- NMR (CDCl ₃ ) δ: 7.51 (1 H, d, J = 2.5 Hz), 7.41-7.37 (2 H, m), 7.24 (1 H, dd, J = 5.7, 3.7 Hz), 6.96 (1 H, dd, J = 4.8, 2.1 Hz), 6.91-6.89 (2 H, m), 5. 76 (1 H, d, J = 2.7 Hz), 5.31 (2 H, s), 3. 64 (3 H, s), 2.56 (3 H, s). 1 -[2-({[1- (5-methoxypyrazin-2-yl) -1H-pyrazol-3-yl] o Shi} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.55 (1H, d, J = 1.4 Hz), 8.12 ( 1H, d, J = 2.7 Hz), 7.95 (1 H, d, J = 1.4 Hz), 7.43-7.38 (2 H, m), 7.27-7.26 (1 H, m), 5.83 (1 H, d, J = 2.7 Hz) ), 5.35 (2H, s), 4.00 (3H, s), 3.68 (3H, s), 2.57 (3H, s) .; 1- [2-({[1- (6-propoxy-2-methylpyridine). -3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.48 (1 H, d, J = 8.7 Hz), 7.41-7.37 (2 H, m), 7.26-7.23 (2 H, m), 6.61 (1 H, d, J = 8.5 Hz), 5. 76 (1 H, d, J = 2.5 Hz), 5.27 (2H, s), 4.26 (2H, t, J = 6.6 Hz), 3.59 (3H, s), 2.55 (3H, s), 2.32 (3H, s), 1.82-1.79 (2H, 2) m), 1.03 (3 H, t, J = 7.4 Hz) .; 1- [3-ethyl-2-({2-methyl-4- [1- (2,2-di) Fluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.59-7.45 (5H, m), 7.30-7.27 (1H, m), 6.87 (1H, d, J = 8.4 Hz), 6.52 (1 H, d, J = 2.5 Hz), 6.14 (1 H, tt, J = 55.6, 4.4 Hz), 5.08 (2H, s), 4.48 (2H, td, J = 13.4, 4.5 Hz), 3.58 (3H, s), 2.85 (2H, q, J = 7.5 Hz), 2.11 (3H, s), 1.28 (3H) , t, J = 7.9 Hz) .; 1- [2-({[1- (5,6-dimethoxypyridin-2-yl) -1 H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl ¹ H-NMR (CDCl ₃ ) δ: 8.16 (1 H, d, J = 2.7 Hz), 7.42-7.38 (2 H, m), 7.27- 7.24 (2H, m), 7.16 (1 H, d, J = 8.4 Hz), 5. 78 (1 H, d, J = 2.7 Hz), 5.32 (2 H, s), 4.03 (3 H, s), 3. 90 (3 H, s) ), 3.65 (3H, s), 2.56 (3H, s) .;

1- [2-({[1- (4-chloro-3-trifluoromethylphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4- Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.88 (1 H, d, J = 2.7 Hz), 7. 69 (1 H, d, J = 2.7 Hz), 7. 66 (1 H, dd, J = 8.7) , 2.6 Hz), 7.53 (1 H, d, J = 8.6 Hz), 7.43-7.38 (2 H, m), 7. 27-7. 25 (1 H, m), 5. 87 (1 H, d, J = 2.7 Hz), 5. 34 (2 H) , s), 3.66 (3H, s), 2.57 (3H, s) .; 1- [2-({[1- (1-methylethyl) -1H-pyrazol-3-yl] oxy} methyl) -3. -Methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.34 (2H, m), 7.23 (1 H, dd, J = 6.1, 3.1 Hz), 7.13 (1H, d, J = 2.1 Hz), 5.51 (1H, d, J = 2.3 Hz), 5.20 (2H, s), 4.29-4.19 (1H, m), 3.68 (3H, s), 2.53 (3H, s), 1.40 (6H, d, J = 6.6 Hz). Le -2 - {[2,5-dimethyl-4- (1H-pyrazol-1-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydro-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.68 (1H, d, J = 1.8 Hz), 7.52 (1H, d, J = 2.3 Hz), 7.46-7.41 (2H, m), 7.34-7.27 (1H, m), 7.07 (1H , s), 6.72 (1H, s), 6.40 (1H, t, J = 2.0 Hz), 5.06 (2H, s), 3.66 (3H, s), 2.52 (3H, s), 2.15 (3H, s) , 2.07 (3H, s) .; 1- (3-ethyl-2-{[2-methyl-4- (5-chloro-1-methyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl)- 4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.51-7.43 (4 H, m), 7.28 (1 H, dd, J = 7.1, 2.1 Hz), 6.86 ( 1H, d, J = 8.5 Hz, 6.41 (1 H, s), 5.08 (2 H, s), 3. 87 (3 H, s), 3.58 (3 H, s), 2. 85 (2 H, q, J = 7.6 Hz), 2.10 (3H, s), 1.28 (3H, t, J = 7.6 Hz) .; 1- (2-{[2,5-dimethy] 4- (5-fluoro-pyrimidin-2-yl) phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.65 (2H, s ), 7.71 (1H, d, J = 7.0 Hz), 7.65 (1H, s), 7.56-7.48 (3H, m), 6.70 (1H, s), 5.21 (2H, s), 3.69 (3H, s) , 2.51 (3H, s), 2.19 (3H, s) .; 1- {2-[({1- [6- (methoxymethoxy) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) Methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.69-7.68 (1 H, m), 7.59 (1 H, dd, J = 9.7, 3.1 Hz), 7.43 (1 H, d, J = 2.5 Hz), 7.40-7.39 (2 H, m), 7.25-7.24 (1 H, m), 6.66 (1 H, d, J = 9.7 Hz), 5.79 (1H, d, J = 2.5 Hz), 5.39 (2H, s), 5.27 (2H, s), 3.67 (3H, s), 3.44 (3H, s), 2.55 (3H, s). 2-({[1- (1-methyl-1H-imidazol-2-yl) 1H- pyrazol-3-yl] oxy} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.80 (1H, d, J = 2.7 Hz), 7.43-7.37 (2H, m), 7.27-7.25 (1 H, m), 6.89 (1 H, d, J = 1.4 Hz), 6.80 (1 H, d, J = 1.4 Hz), 5.81 ( 1H, d, J = 2.7 Hz), 5.29 (2H, s), 3.76 (3H, s), 3.63 (3H, s), 2.53 (3H, s) .; 1- [2-({[1- (1) 6-Ethoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl 2) ₃ ) δ: 8.31 (1 H, d, J = 3.0 Hz), 7.80 (1 H, dd, J = 8.9, 2.7 Hz), 7.56 (1 H, d, J = 2.5 Hz), 7.42-7.37 (2 H, m) , 7.27-7.24 (1H, m), 6.79 (1H, d, J = 8.9 Hz), 5.80 (1H, d, J = 2.5 Hz), 5.32 (2H, s), 4.37 (2H, q, J = 7.1) Hz), 3.64 (3H, s), 2.56 (3H, s), 1.41 (3H, t, J = 7.1 Hz) .; 1- (3-methyl-2- { 2,5-Dimethyl-4- (4-methyl-4,5-dihydro-1,3-oxazol-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one ¹ H-NMR (CDCl ₃ ) δ: 7.57 (1 H, s), 7. 45-7. 39 (2 H, m), 7. 29-7. 26 (1 H, m), 6. 66 ( ¹ H, s), 5.0 6 (2 H, s), 4.45-4.31 (2H, m), 3.88 (1H, t, J = 7.3 Hz), 3.63 (3H, s), 2.55 (3H, s), 2.49 (3H, s), 2.04 (3H, s), 1.34 (3H, d, J = 6.4 Hz) .; 1- [3-Methyl-2-({2,5-dimethyl-4- [rel- (4R, 5R) -4,5-dimethyl-4,5-) Dihydro-1,3-oxazol-2-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.55 (1 H, s) , 7.45-7.39 (2H, m), 7.29-7.26 (1H, m), 6.65 (1H, s), 5.05 (2H, s), 4.26-4.20 (1H, m), 3.86-3. 79 (1H, m) , 3.63 (3H, s), 2.54 (3H, s), 2.49 (3H, s), 2.04 (3H, s), 1.39 (3H, d, J = 6.3 Hz), 1.31 (3 H, d, J = 6.8 Hz);

1- (3-Methyl-2-{[2-methyl-4- (4-cyano-5-fluoro-1-methyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.71-7.69 (1H, m), 7.67-7.64 (1H, m), 7.45-7.41 (2H, m), 7.30-7.28 (1H, m), 6.91 (1H, d, J = 8.4 Hz), 5.08 (2H, s), 3.81 (3H, s), 3.64 (3H, s), 2.51 (3H, s), 2.13 (3H, s) s) .; 1- (3-chloro-2-{[2,5-dimethyl-4- (5-fluoropyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole -5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.65 (2H, s), 7.63 (1H, dd, J = 7.9, 1.4 Hz), 7.61 (1H, s), 7.48 (1H, t, J = 8.0 Hz), 7.41 (1 H, dd, J = 7.9, 1.4 Hz), 6.75 (1 H, s), 5.37 (2 H, s), 3.62 (3 H, s), 2.53 (3 H, s), 2.03 (3 H) , s) .; 1- (3-ethyl-2-{[2- Chill-4- (5-fluoro-4-methyl-2-yl) phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.44 (1H, d, J = 1.4 Hz), 8.17 (1 H, dd, J = 8.5, 2.2 Hz), 8.13 (1 H, s), 7.51-7.44 (2 H, m), 7.29 (1 H, dd, J = 7.0, 2.0 Hz), 6.93 (1 H, d, J = 8.6 Hz), 5.13 (2 H, s), 3.58 (3 H, s), 2. 86 (2 H, q, J = 7.6 Hz), 2.57 (3 H, d, J = 2.5 Hz), 2.15 (3 H, s), 1. 29 (3 H, t, J = 7.6 Hz). 1- [2-({[1- (2-nitrophenyl) -1 H-pyrazol-3-yl] ] Oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.80 (1 H, d, J = 8.5 Hz), 7.63 (1H, t, J = 8.0 Hz), 7.52 (1 H, d, J = 8.0 Hz), 7.54 (1 H, d, J = 2.5 Hz), 7.45-7.37 (3 H, m), 7.24 (1 H, dd, J = 6.2, 3.2 Hz), 5.87 (1 H, d, J = 2.7 Hz), 5.21 (2 H, s), 3. 66 (3 H, s), 2.52 (3 H, s). 1- (3-Cyclopropyl-2-{[2-methyl-4- (5-chloro-1-methyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4- Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 to 7.41 (3 H, m), 7. 28-7. 26 (2 H, m), 6. 89 (1 H, d, J = 8.5 Hz), 6.41 (1 H , s), 5.28 (2H, s), 3.87 (3H, s), 3.60 (3H, s), 2.16-2.09 (1H, m), 2.10 (3H, s), 1.01-0.96 (2H, m), 0.78-0.74 (2H, m) .; 1- (3-methoxy-2-{[2-methyl-4- (5-fluoro-4-methylpyrimidin-2-yl) phenoxy] methyl} phenyl) -4- Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.41 (1 H, d, J = 1.4 Hz), 8.12 (1 H, dd, J = 8.6, 2.3 Hz), 8.08 (1H, s), 7.46 (1H, t, J = 8.3 Hz), 7.08 (2H, t, J = 7.2 Hz), 6.95 (1 H, d, J = 8.6 Hz), 5.34 (2H, s), 3.93 (3H, s), 3.58 (3H, s), 2.55 (3H, d, J = 2.5) Hz), 2.05 (3 H, s) .; 1- (3-ethyl-2-{[2,5-dimethyl-4- (3-methylbutanoyl) phenoxy] methyl} phenyl) -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.51-7.45 (2 H, m), 7. 40 ( ¹ H, s), 7. 29 ( ¹ H, d, J = 7.3 Hz), 6. 69 ( ¹ H , s), 5.09 (2H, s), 3.61 (3H, s), 3.44-3.33 (1H, m), 2.84 (2H, q, J = 7.6 Hz), 2.47 (3H, s), 2.06 (3H, s) s), 1.28 (3 H, t, J = 7.6 Hz), 1. 15 (6 H, d, J = 6.0 Hz) .; 1- (2-{[2-methyl-4- (5-fluoro-4-methyl pyrimidine) -2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.43 (1 H, d, J = 1.4 Hz), 8.15 -8.13 (2H, m), 7.73-7.71 (1H, m), 7.56-7.48 (3H, m), 6.88 (1H, d, J = 8.8 Hz), 5.23 (2H, s), 3.68 (3H, s) ), 2.56 (3H, d, J = 2.5 Hz), 2.26 (3H, s) .; 1- [3-Methyl-2-({2,5 Dimethyl-4-[(4S) -4-ethyl-4,5-dihydro-1,3-oxazol-2-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one ¹ H-NMR (CDCl ₃ ) δ: 7.56 (1 H, s), 7.44-7. 39 (2 H, m), 7. 29-7. 26 (1 H, m), 6. 66 (1 H, s), 5.05 (2 H, s), 4.40-4.36 (1H, m), 4.26-4.19 (1H, m), 4.00-3.96 (1H, m), 3.63 (3H, s), 2.55 (3H, s), 2.49 (3H, s), 2.04 (2. 3H, s), 1.77-1.70 (1H, m), 1.64-1.57 (4H, m), 0.99 (3H, t, J = 7.4 Hz) .; 1- [3- (trifluoromethoxy) -2- (2) {2-Methyl-4- [1- (2,2-difluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.61-7.56 (1 H, m), 7.53-7. 47 (4 H, m), 7. 45 (1 H, d, J = 2.3 Hz), 6.86 (1 H, d, J = 8.2 Hz) , 6.51 (1H, d, J = 2.5 Hz), 6.13 (1 H, tt, J = 55.6, 4.4 Hz), 5.30 (2H, s), 4.47 (2H, td, J = 13.4, 4.5 Hz), 3.57 (3H, s), 2.02 (3H, s).

1- {3-Methyl-2-[(4- (ethoxymethyl) -2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.27-7.25 (1H, m), 7.02 (1H, s), 6.65 (1H, s), 5.00 (2H, s), 4.39 (2H, s) , 3.65 (3H, s), 3.52 (2H, q, J = 6.9 Hz), 2.49 (3H, s), 2.31 (3H, s), 2.04 (3H, s), 1.23 (3H, t, J = 6.9) Hz) .; 1- [2-({[1- (adamantan-1-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38-7.35 (2 H, m), 7.23 (1 H, dd, J = 5.3, 2.5 Hz), 7.21 (1 H, d, J = 2.3 Hz) , 5.50 (1H, d, J = 2.3 Hz), 5.20 (2H, s), 3.67 (3H, s), 2.53 (3H, s), 2.19 (3H, s), 2.05 (6H, d, J = 3.0) Hz), 1.76-1.71 (6H, m) .; 1- [2-({[1- (5-fluoro-6-methyl). Pyridin-2-yl)-1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ : 8.25 (1H, d, J = 2.7 Hz), 7.56 (1H, dd, J = 8.8, 3.2 Hz), 7.40 (3H, m), 7.28-7.24 (1H, m), 5.81 (1H, d, J = 2.7 Hz), 5.32 (2 H, s), 3. 64 (3 H, s), 2.55 (3 H, s), 2. 48 (3 H, d, J = 2.9 Hz) .; 1- [3-cyclopropyl-2- (2) {2-Methyl-4- [5-fluoro-4- (difluoromethyl) -1-methyl-1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 7.46- 7. 38 (3 H, m), 7. 29-7. 27 (2 H, m), 6. 94 (1 H, d, J = 8.6 Hz), 6.62 (1 H, t, J = 54.3 Hz), 5.29 (2H, s), 3.79 (3H, s), 3.61 (3H, s), 2.16-2.09 (4H, m), 1.02-0.97 (2H, m), 0.79-0.75 (2H, m) ); 1- (3-cyclopropyl) -2-{[2-methyl-4- (5-fluoro-1,4-dimethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 7.45-7.37 (3 H, m), 7. 29-7. 27 (2 H, m), 6. 92 (1 H, d, J = 8.4 Hz), 5. 28 (2 H, s), 3.74 (3H, s), 3.61 (3H, s), 2.16-2.11 (4H, m), 2.09 (3H, s), 1.02-0.97 (2H, m), 0.78-0.74 (2H, m). (3-Methyl-2-{[2,5-dimethyl-4- (4,5-dihydro-1,3-oxazol-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.59 (1 H, s), 7. 45-7. 39 (2 H, m), 7. 29-7. 27 (1 H, m), 6. 67 ( ¹ H, s), 5.0 6 (5.0 H) 2H, s), 4.34 (2H, t, J = 9.3 Hz), 4.05 (2H, t, J = 9.3 Hz), 3.63 (3H, s), 2.56 (3H, s), 2.50 (3H, s), 2.05 (3H, s) .; 1- [3-methoxy-2-({2,5 -Dimethyl-4- [1- (2,2-difluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H- NMR (CDCl ₃ ) δ: 7.48-7.44 (2H, m), 7.26-7.23 (1H, m), 7.08 (2H, dd, J = 7.9, 6.1 Hz), 6.76 (1H, s), 6.37 (1H, 6) d, J = 2.3 Hz), 6.13 (1 H, tt, J = 55.6, 4.4 Hz), 5. 27 (2 H, s), 4. 47 (2 H, td, J = 13.4, 4.4 Hz), 3.94 (3 H, s), 3.60 (3H, s), 2.39 (3H, s), 1.98 (3H, s) .; 1- (3-methoxy-2-{[2,5-dimethyl-4- (cyclopropanecarbonyl) phenoxy] methyl} Phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.55 (1 H, s), 7.51-7. 45 (1 H, m), 7.12-7.06 (2 H, m), 6.73 (1H, s), 5.32 (2H, s), 3.95 (3H, s), 3.61 (3H, s), 2.47 (3H, s), 2.45-2.39 (1H, m), 1.99 (3H) , s), 1.19-1.15 (2H, m), 0.98-0.95 (2H, m). Sheet -2 - {[2-methyl-4- (5-fluoro-6-methyl-pyridin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydro-5-one, ¹ H -NMR (CDCl ₃ ) δ: 7.66-7.63 (2H, m), 7.49-7.41 (2H, m), 7.31 (1H, t, J = 8.7 Hz), 7.08 (2H, t, J = 8.0 Hz), 6.93 (1H, d, J = 8.2 Hz), 5.32 (2H, s), 3.94 (3H, s), 3.59 (3H, s), 2.56 (3H, d, J = 2.9 Hz), 2.05 (3H, s) 1- {3-Methyl-2-[(4-ethoxy-2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazole-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.23 (1H, m), 6.63 (1H, s), 6.60 (1H, s), 4.95 (2H, s), 3.95 (2H, q, J = 6.9 Hz), 3.64 (3H, s), 2.51 (3H, s), 2.17 (3H, s), 2.03 (3H, s), 1.38 (3H, t, J = 6.9 Hz);

1- [3-Methyl-2-({2,5-dimethyl-4-[(4R) -4- (1-methylethyl) -4,5-dihydro-1,3-oxazol-2-yl] phenoxy } Methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.55 (1 H, s), 7. 45-7. 39 (2 H, m), 7. 29-7. 26 (1H, m), 6.66 (1H, s), 5.05 (2H, s), 4.35-4.27 (1H, m), 4.15-4.04 (2H, m), 3.63 (3H, s), 2.56 (3H, s) ), 2.49 (3H, s), 2.04 (3H, s), 1.88-1.79 (1H, m), 1.02 (3H, d, J = 6.8 Hz), 0.93 (3 H, d, J = 6.8 Hz); 1- [2-({[1- (4-methoxypyridin-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole -5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.31 (1H, d, J = 2.7 Hz), 8.13 (1 H, d, J = 5.9 Hz), 7.43-7.38 (2H, m), 7.28 ( 1H, d, J = 2.3 Hz), 7.26-7.25 (1H, m ), 6.64 (1H, dd, J = 5.8, 2.4 Hz), 5.83 (1H, d, J = 2.7 Hz), 5.33 (2H, s), 3.95 (3H, s), 3.65 (3H, s), 2.56 (3H, s) .; 1- {3-methyl-2-[(4-methoxy-2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.24 (1H, m), 6.64 (1H, s), 6.60 (1H, s), 4.96 (2H, s), 3.76 ( 3H, s), 3.65 (3H, s), 2.51 (3H, s), 2.17 (3H, s), 2.05 (3H, s) .; 1- (3-methyl-2-{[2,5-dimethyl] -4- (propoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.72 (1 H, s), 7.46-7.40 ( 2H, m), 7.28 (1H, dd, J = 7.2, 2.0 Hz), 6.65 (1H, s), 5.07 (2H, s), 4.22 (2H, t, J = 6.7 Hz), 3.64 (3H, s) ), 2.58 (3H, s), 2.50 (3H, s), 2.06 (3H, s), 1.82-1. 73 (2H, m), 1.02 (3H, t, J = 7.4 Hz) .; 1-(3- Toxi-2-{[2,5-dimethyl-4- (1,5-dimethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one , ¹ H-NMR (CDCl ₃ ) δ: 7.48-7.44 (1H, m), 7.25 (1H, s), 7.09-7.06 (2H, m), 6.73 (1H, s), 6.09 (1H, d, J = 0.7 Hz), 5.26 (2H, s), 3.93 (3H, s), 3.80 (3H, s), 3.59 (3H, s), 2.39 (3H, s), 2.30 (3H, s), 1.96 (3H) 1- [2-({[1- (5-chloro-6-methoxypyridin-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4 -Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.21 (1 H, d, J = 2.7 Hz), 7.68 (1 H, d, J = 8.2 Hz), 7.42- 7.39 (2H, m), 7.28-7.25 (2H, m), 5.83 (1H, d, J = 2.7 Hz), 5.33 (2H, s), 4.03 (3H, s), 3.65 (3H, s), 2.56 (3H, s) .; 1- (2-{[(1-heptyl-1) - pyrazol-3-yl) oxy] methyl} -3-methylphenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.39-7.34 (2H, m ), 7.23 (1 H, dd, J = 6.5, 2.9 Hz), 7.08 (1 H, d, J = 2.3 Hz), 5. 50 (1 H, d, J = 2.3 Hz), 5. 19 (2 H, s), 3. 87 (2 H) , t, J = 7.2 Hz), 3.67 (3 H, s), 2.52 (3 H, s), 1. 78-1. 75 (2 H, m), 1.31-1. 20 (8 H, m), 0.88 (3 H, t, J = 7.0) Hz) .; 1- (3-Methyl-2-{[4- (1-methylethyl) -2,5-dimethylphenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one , ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.24 (1H, m), 6.63 (2H, d, J = 2.9 Hz), 4.95 (2H, s), 4.36- 4.30 (1H, m), 3.64 (3H, s), 2.51 (3H, s), 2.17 (3H, s), 2.03 (3H, s), 1.29 (6H, d, J = 6.1 Hz) .; 1-1 [2-({[1- (1-methylhexyl) -1H-pyrazol-3-yl] oxy} methyl) 3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.38-7.33 (2H, m), 7.22 (1H, dd, J = 6.2, 2.5 Hz), 7.09 (1 H, d, J = 2.1 Hz), 5. 49 (1 H, d, J = 2.1 Hz), 5. 19 (2 H, s), 4.03-4.00 (1 H, m), 3. 67 (3 H, s) , 2.53 (3 H, s), 1.84-1. 75 (1 H, m), 1. 68-1.52 (1 H, m), 1. 38 (3 H, d, J = 6.9 Hz), 1.28-1.07 (6 H, m), 0.85 (3 H , t, J = 6.9 Hz) .; 1- {2-[({1- [6- (difluoromethoxy) pyridin-3-yl] -1 H-pyrazol-3-yl} oxy) methyl] -3-methyl Phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.38 (1 H, d, J = 2.7 Hz), 7.96 (1 H, dd, J = 8.8, 2.9 Hz), 7.63 (1 H, d, J = 2.5 Hz), 7.45 (1 H, t, J = 72.3 Hz), 7.43-7.38 (2 H, m), 7.28-7. 25 (1 H, m), 6.98 (1 H, 1 H, m) d, J = 8.8 Hz), 5. 85 (1 H, d, J = 2.5 Hz), 5.32 (2 H, s), 3. 66 (3 H, s), 2.56 (3 H, s).

1- (2-{[(1-dodecyl-1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2 H, m), 7.23 (1 H, dd, J = 6.6, 2.7 Hz), 7.07 (1 H, d, J = 2.3 Hz), 5. 50 (1 H, d, J = 2.3 Hz), 5.19 (2H, s), 3.86 (2H, t, J = 7.2 Hz), 3.67 (3H, s), 2.52 (3H, s), 1.79-1.72 (2H, m), 1.25 (18H, s) ), 0.88 (3 H, t, J = 6.9 Hz) .; 1- [2-({[1- (2-butoxy-3-methoxypyridin-4-yl) -1 H-pyrazol-3-yl] oxy} Methyl) -3-Methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.24 (1 H, d, J = 2.7 Hz), 7.86 ( ¹ H, ¹ H, d, J = 5.7 Hz), 7.42-7.39 (3 H, m), 7. 27-7. 26 (1 H, m), 5. 85 (1 H, d, J = 2.7 Hz), 5.33 (2 H, s), 4. 39 (2 H, t) , J = 6.6 Hz), 3.82 (3H, s), 3.64 (3H, s), 2.56 (3H, s), 1.87-1.80 (2H, 2) m), 1.55-1.49 (2H, m), 1.00 (3H, t, J = 7.3 Hz) .; 1- [3-Methyl-2-({3,5-dimethyl-4-[(dimethylamino) carbonyl] ] Phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-7.38 (2H, m), 7.28-7.26 (1H, m) , 6.54 (2H, s), 4.97 (2H, s), 3.65 (3H, s), 3.13 (3H, s), 2.80 (3H, s), 2.48 (3H, s), 2.19 (6H, s). 1- (3-methyl-2-{[2,5-dimethyl-4- (1-ethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole; -5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-7.39 (3H, m), 7.32 (1H, s), 7.28-7.26 (1H, m), 6.70 (1H, s), 6.31 (1H) , d, J = 2.3 Hz), 5.04 (2H, s), 4.21 (2H, q, J = 7.3 Hz), 3.64 (3H, s), 2.51 (3H, s), 2.43 (3H, s), 2.07 (3H, s), 1.52 (3H, t, J = 7.4 Hz) .; 1-(3-cyclopropyl- - {[2,5-dimethyl-4- (3-methylbutanoyl) phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.47-7. 42 (1 H, m), 7. 40 (1 H, s), 7. 29-7. 25 (2 H, m), 6.72 (1 H, s), 5. 29 (2 H, s), 3.63 (3 H, s), 3.44-3. 35 ( 1H, m), 2.47 (3H, s), 2.15-2.08 (1H, m), 2.07 (3H, s), 1.15 (6H, d, J = 6.9 Hz), 1.03-0.98 (2H, m), 0.80 -0.75 (2H, m) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-methoxypyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.47 (2H, s), 7.56 (1H, s), 7.44-7.39 (2H, m), 7.29-7.26 (1H, m) 1), 6.72 (1H, s), 5.08 (2H, s), 3.95 (3H, s), 3.64 (3H, s), 2.51 (6H, bs), 2.09 (3H, s). (Piperidin-1-ylmethyl) -3-methylphenyl] -4-methyl-1, - _{^{dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.30-7.27 (2H, m), 7.18 (1H, dd, J = 6.3, 2.9 Hz), 3.71 (3H, s), 3.47 ( 2H, s), 2.44 (3H, s), 2.15 (4H, s), 1.34 (6H, s) .; 1- {2-[({1- [3- (trifluoromethyl) phenyl] -1H- Pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.83 (1 H, s), 7.74 -7.73 (2H, m), 7.53 (1H, t, J = 8.0 Hz), 7.44-7.40 (3H, m), 7.27-7.25 (1 H, m), 5.86 (1 H, d, J = 2.7 Hz), 5.35 (2H, s), 3.64 (3H, s), 2.57 (3H, s) .; 1- [3-methyl-2-({2-methyl-4- [5-fluoro-4- (difluoromethyl)] -1-Methyl-1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.45-7. 37 (4H, m), 7.31-7.27 (1H, m), 6.89 (1H, d, J = 8.4 Hz), 6.62 (1H, t, J = 54.4 Hz), 5.07 (2H, s), 3.79 (3H , s), 3.63 (3H, s), 2.51 (3H, s), 2.12 (3H, s) .; 1- {3-cyclopropyl-2-[(4-methoxy-2,5-dimethylphenoxy) methyl] ] Phenyl} -4-methyl-1,4-dihydrotetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.41 (1 H, t, J = 7.8 Hz), 7.24 (2 H, d, J = 7.8) Hz), 6.67 (1H, s), 6.60 (1H, s), 5.18 (2H, s), 3.76 (3H, s), 3.63 (3H, s), 2.19-2.12 (4H, m), 2.05 (3H) , s), 1.02-0.98 (2H, m), 0.78-0.74 (2H, m).

1- [3-Methyl-2-({2,5-dimethyl-4-[(4R) -4-ethyl-4,5-dihydro-1,3-oxazol-2-yl] phenoxy} methyl) phenyl] -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.56 (1 H, s), 7.44-7. 39 (2 H, m), 7. 29-7. 26 (1 H, m) , 6.66 (1H, s), 5.05 (2H, s), 4.40-4.36 (1H, m), 4.26-4.19 (1H, m), 4.00-3.96 (1H, m), 3.63 (3H, s), 2.55 (3H, s), 2.49 (3H, s), 2.04 (3H, s), 1.77-1.70 (1H, m), 1.64-1.57 (4H, m), 0.99 (3H, t, J = 7.4 Hz). 1- {2-[({1- [6- (2,2,2-trifluoroethoxy) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl}; -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.33 (1 H, dd, J = 2.8, 0.6 Hz), 7.88 (1 H, dd, J = 8.8, 2.7 Hz), 7.59 (1H, d, J = 2.5 Hz), 7.42-7.39 (2H, m), 7.26-7.25 (1 H, m), 6.93 (1 H, dd, J = 8.8, 0.7 Hz), 5.83 (1 H, d, J = 2.5 Hz), 5.32 (5 2H, s), 4.78 (2H, q, J = 8.5 Hz), 3.65 (3H, s), 2.56 (3H, s). 1- (3-methyl-2-{[2,5-dimethyl-4] -(3,4-Dimethyl-1H-pyrazol-1-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.45 7.38 (2H, m), 7.29-7.26 (2H, m), 7.07 (1H, s), 6.69 (1H, s), 5.04 (2H, s), 3.66 (3H, s), 2.51 (3H, s) , 2.23 (3H, s), 2.17 (3H, s), 2.07 (3H, s), 2.05 (3H, s) .; 1- {3-cyclopropyl-2- [2,5-dimethyl-4- (2) 5-chloro-1-methyl-1H-pyrazol-3-yl) phenoxymethyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (DMSO-D6) δ: 7.51 ( 1 H, t, J = 7.8 Hz), 7. 35 (1 H, dd, J = 7.8, 1.0 Hz), 7.28 (1H, d, J = 7.9 Hz), 7.25 (1H, s), 6.87 (1H, s), 6.60 (1H, s), 5.22 (2H, s), 3.82 (3H, s), 3.55 (3H) , s), 2.37 (3H, s), 2.23-2.16 (1H, m), 1.98 (3H, s), 1.03-0.98 (2H, m), 0.80-0.76 (2H, m) .; 1-[3 -Fluoro-2-({2-methyl-4- [5-fluoro-4- (difluoromethyl) -1-methyl-1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4 -Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.54-7.48 (1 H, m), 7. 38-7. 28 (4 H, m), 6. 91 (1 H, d, J = 9.1 Hz), 6.61 (6 1 H, t, J = 54.3 Hz), 5.31 (2 H, s), 3. 78 (3 H, s), 3. 60 (3 H, s), 2.03 (3 H, s) .; 1- [2-({[1- (1) 2-hydroxycyclohexyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.35 (2H, m), 7.24-7.22 (1 H, m), 7.19 (1 H, d, J = 2.5 Hz), 5.53 (1 H, d, J = 2.3 Hz), 5.25 (1 H, d, J = 12.2 Hz), 5.18 (1 H, d, J = 12.2) Hz), 3.70-3.63 (5H, m), 3.56 (1H, d, J = 1.8 Hz), 2.53 (3H, s), 2.13-2.07 (1H, m), 2.05-2.03 (1H, m), 1.82 -1.78 (2H, m), 1.73-1.65 (1H, m), 1.44-1.31 (3H, m) .; 1- [3-methoxy-2-({2,5-dimethyl-4-[(1,1) 1-Dimethylethoxy) carbonyl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 (1 H, s), 7.47 (1 H, t, J = 8.2 Hz), 7.10-7.06 (2 H, m), 6. 69 (1 H, s), 5. 30 (2 H, s), 3. 94 (3 H, s), 3. 60 (3 H, s), 2.52 (3 H, s) ), 1.95 (3H, s), 1.56 (9H, s) .; 1- {2-[({1- [1,1-dimethyl-2- (methoxyimino) ethyl] -1H-pyrazol-3-yl] } Oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one , ¹ H-NMR (CDCl ₃ ) δ: 7.49 (1H, s), 7.39-7.34 (2H, m), 7.23-7.21 (2H, m), 5.55 (1H, d, J = 2.5 Hz), 5.21 ( 2H, s), 3.85 (3H, s), 3.68 (3H, s), 2.53 (3H, s), 1.56 (6H, s) .; 1- [2-({[1- (2-ethoxy-3)] -Methoxypyridin-4-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ δ: 8.24 (1 H, d, J = 2.7 Hz), 7.87 (1 H, d, J = 5.7 Hz), 7.42-7.39 (3 H, m), 7.28-7. 25 (1 H, m), 5. 85 (1 H, d) , J = 2.7 Hz), 5.33 (2H, s), 4.47 (2H, q), 3.82 (3H, s), 3.64 (3H, s), 2.56 (3H, s), 1.46 (3H, t, J = 7.1 Hz) .; 1- [3-Methyl-2-({3,5-dimethyl-4-[(1-methylethoxy) carbonyl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazole -5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-7.38 (2H, m), 7.28-7.2 6 (1 H, m), 6.53 (2 H, s), 5. 30-5. 24 (1 H, m), 4.99 (2 H, s), 3. 64 (3 H, s), 2. 47 (3 H, s), 2. 30 (6 H, s) , 1.36 (6H, d, J = 6.4 Hz) .;

1- {3-Methyl-2-[({[1- (adamantan-1-yl) ethylidene] amino} oxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H -NMR (CDCl ₃ ) δ: 7.37-7.32 (2H, m), 7.21-7.17 (1H, m), 5.09 (2H, s), 3.70 (3H, s), 2.50 (3H, s), 1.98 (3H , s), 1.72-1.62 (12H, m), 1.60 (3H, s) .; 1- {2-[({1- [2- (1,1-dimethylethoxy) -3-methoxypyridine-4-]. Yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.21 (1 H , d, J = 2.7 Hz), 7.55 (1 H, d, J = 5.5 Hz), 7.42-7. 40 (2 H, m), 7.33 (1 H, d, J = 5.5 Hz), 7.26-7.25 (1 H, m) , 5.83 (1H, d, J = 2.7 Hz), 5.33 (2H, s), 3.80 (3H, s), 3.64 (3H, s), 2.56 (3H, s), 1.65 (9H, s) .; 1 -(3-methyl-2-{[2,5-di] Tyl-4- (4-ethyl-4-methyl-4,5-dihydro-1,3-oxazol-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one ¹ H-NMR (CDCl ₃ ) δ: 7.53 (1H, s), 7.44-7.39 (2H, m), 7.29-7.26 (1H, m), 6.65 (1H, s), 5.05 (2H, s), 4.12 (1H, d, J = 8.2 Hz), 3.94 (1H, d, J = 8.2 Hz), 3.63 (3H, s), 2.53 (3H, s), 2.49 (3H, s), 2.04 (3H, s) ), 1.73-1.60 (2H, m), 1.34 (3H, s), 0.92 (3H, t, J = 7.4 Hz). 1- {2-[({1- [4- (1,1-dimethyl). Ethyl) phenyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.64 (1H, d, J = 2.5 Hz), 7.48 (2H, d, J = 8.7 Hz), 7.43-7.38 (4H, m), 7.26-7.24 (1 H, m), 5.78 (1 H, d, J = 2.5) Hz), 5.33 (2H, s), 3.60 (3H, d, J = 0.7 Hz), 2.56 (3H, s), 34 (9 H, s) .; 1- [2-({[2- (3, 3-dimethyl-1-butynyl) thiazol-4-yl] oxy} methyl) -3- methylphenyl] -4- methyl- 1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-4.40 (2H, m), 7.26 (1 H, dd, J = 7.3, 1.8 Hz), 6.71 (1 H, s) , 5.45 (2H, s), 3.71 (3H, s), 2.51 (3H, s), 1.32 (9H, s) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (2) Isopropoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.69 (1 H, s), 7.42 (2 H, q, J = 7.7 Hz), 7.30-7.28 (1H, m), 6.64 (1H, s), 5.23-5.17 (1H, m), 5.07 (2H, s), 3.64 (3H, s), 2.57 (3H, s) , 2.49 (3H, s), 2.06 (3H, s), 1.35 (6H, d, J = 6.3 Hz) .; 1- [3- (trifluoromethyl) -2-({2-methyl-4- [ 1- (2,2-difluoroethyl) ) -1H-Pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.92 (1 H, dd, J = 6.8, 2.5 Hz), 7.71-7.63 (2 H, m), 7.54-7. 51 (2 H, m), 7.46 (1 H, d, J = 2.5 Hz), 6. 85 (1 H, d, J = 8.2 Hz), 6.52 ( 1H, d, J = 2.5 Hz, 6.14 (1 H, tt, J = 55.6, 4.4 Hz), 5.33 (2 H, s), 4.48 (2 H, td, J = 13.4, 4.4 Hz), 3.52 (3 H, s) ), 2.04 (3H, s) .; 1- [3-methyl-2-({2,5-dimethyl-4- [1- (2,2,2-trifluoroethyl) -1H-pyrazole-5-) [Il] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.65 (1 H, d, J = 1.8 Hz), 7.47-7. 2H, m), 7.29 (1H, dd, J = 6.8, 2.5 Hz), 6.91 (1H, s), 6.74 (1H, s), 6.22 (1 H, d, J = 1.8 Hz), 5.06 (2H, s) ), 4.49 (2H, q, J = 8.3 Hz), 3.67 (3H, s), 2.54 (3H, s), 2.09 (3H, s), 2.07 ( 3H, s) .; 1- (3-Cyclopropyl-2-{[2,5-dimethyl-4- (cyclopropanecarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole-5 -ON, ¹ H-NMR (CDCl ₃ ) δ: 7.58 (1 H, s), 7.47-7. 42 (1 H, m), 7.30-7.26 (2 H, m), 6.71 (1 H, s), 5. 30 (2 H, s) ), 3.63 (3H, s), 2.50 (3H, s), 2.47-2.40 (1H, m), 2.15-2.09 (1H, m), 2.08 (3H, s), 1.21-1.17 (2H, m), 1.03-0.95 (4H, m), 0.80-0.77 (2H, m) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (methoxycarbonyl) phenoxy] methyl} phenyl) -4 -Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.72 (1 H, s), 7. 45-7. 40 (2 H, m), 7. 28 (1 H, dd, J = 7.2, 2.0 Hz), 6.66 (1H, s), 5.08 (2H, s), 3.85 (3H, s), 3.63 (3H, s), 2.58 (3H, s), 2.50 (3H, s), 2.06 (3H, s) s).

1- (3-Methyl-2-{[4- (2,2-difluoroethoxy) -2,5-dimethylphenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.24 (1H, m), 6.63 (1H, s), 6.59 (1H, s), 6.05 (1H, tt, J = 55.3) , 4.1 Hz), 4.97 (2H, s), 4.15-4.07 (2H, m), 3.64 (3H, s), 2.51 (3H, s), 2.19 (3H, s), 2.03 (3H, s). 1- {3-Methyl-2-[(4- (methoxymethyl) -2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.44-7.38 (2H, m), 7.27-7.25 (1H, m), 7.02 (1H, s), 6.65 (1H, s), 5.00 (2H, s), 4.35 (2H, s) , 3.64 (3H, s), 3.36 (3H, s), 2.49 (3H, s), 2.30 (3H, s), 2.04 (3H, s). 3-Dimethyl-1-butynyl) -1H-pyrazol-3-yl] o Shi} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.41-7.38 (2H, m), 7.35 (1H, d , J = 2.7 Hz), 7.25 (1 H, dd, J = 6.9, 1.9 Hz), 5.66 (1 H, d, J = 2.5 Hz), 5.22 (2 H, s), 3.69 (3 H, s), 2.50 (3 H) , s), 1.32 (9 H, s) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (4,4-dimethyl-4,5-dihydro-1,3-oxazole) 2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.54 (1 H, s), 7.44-7. 39 (2 H, m ), 7.29-7.26 (1H, m), 6.65 (1H, s), 5.05 (2H, s), 4.03 (2H, s), 3.63 (3H, s), 2.52 (3H, s), 2.49 (3H, s) s), 2.03 (3H, s), 1.37 (6H, s) .; 1- {2-[({1- [2-chloro-4- (trifluoromethyl) phenyl] -1H-pyrazol-3-yl] } Oxy) methyl] -3- methyl Phenyl} _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.88 (1H, d, J = 2.5 Hz), 7.75 (2H, dd, J = 4.9, 3.3 Hz), 7.61 (1 H, dd, J = 8.5, 1.4 Hz), 7.43-7.38 (2 H, m), 7.27-7.26 (1 H, m), 5.88 (1 H, d, J = 2.7 Hz), 5.32 (5.31) 2H, s), 3.63 (3H, s), 2.56 (3H, s) .; 1- [2-({[1- (1,1-dimethyl-2-{[(1,1-dimethylethyl) amino] ] Carbonyloxy} ethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ : 7.38-7.33 (2H, m), 7.23-7.21 (2H, m), 5.50 (1H, d, J = 2.5 Hz), 5.21 (2H, s), 4.67 (1H, s), 4.16 (2H, s) ), 3.68 (3H, s), 2.53 (3H, s), 1.47 (6H, s), 1.29 (9H, s) .; 1- [2-({[1- (2-propoxy-3-methoxypyridine). -4-yl) -1H-pyrazol-3-yl Oxy} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.24 (1H, d, J = 2.7 Hz), 7.86 ( 1H, d, J = 5.5 Hz), 7.42-7.39 (3 H, m), 7.26-7.25 (1 H, m), 5. 85 (1 H, d, J = 2.7 Hz), 5.33 (2 H, s), 4. 36 (2 H) , t, J = 6.8 Hz), 3.83 (3H, s), 3.64 (3H, s), 2.56 (3H, s), 1.89-1.86 (2H, m), 1.07 (3H, t, J = 7.4 Hz) 1- [3-Methyl-2-({2,5-dimethyl-4-[(4S) -4- (1-methylethyl) -4,5-dihydro-1,3-oxazol-2-yl Phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.55 (1 H, s), 7.45-7.39 (2 H, m), 7.29 -7.26 (1H, m), 6.66 (1H, s), 5.05 (2H, s), 4.35-4.27 (1H, m), 4.15-4.04 (2H, m), 3.63 (3H, s), 2.56 (3H , s), 2.49 (3H, s), 2.04 (3H, s), 1.88-1.79 (1H, m), 1.02 (3H, d, J = 6.8 Hz), 0.93 (3H, d, J = 6.8) Hz) .; 1- (3-methoxy-2-{[2-methyl-4- (5-fluoropyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole-5. -ON, ¹ H-NMR (CDCl ₃ ) δ: 8.59 (2 H, s), 8. 14 (1 H, dd, J = 8.6, 2.2 Hz), 8.09 (1 H, s), 7.47 (1 H, t, J = 8.2 Hz), 7.09 (2H, t, J = 7.6 Hz), 6.97 (1H, d, J = 8.7 Hz), 5.35 (2H, s), 3.94 (3H, s), 3.59 (3H, s), 2.06 ( 3H, s) .; 1- {2-[({1- [6- (1-methylethoxy) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.31 (1 H, d, J = 2.7 Hz), 7. 78 (1 H, dd, J = 8.8, 2.9 Hz ), 7.55 (1H, d, J = 2.5 Hz), 7.42-7.37 (2H, m), 7.25 (1 H, dd, J = 6.1, 3.3 Hz), 6.74 (1 H, d, J = 8.9 Hz), 5.79 (1H, d, J = 2.5 Hz), 5.31-5.26 (3H, m), 3.64 (3H, s), 2.56 (3H, s), 1.36 (6H, d, J = 6.2 Hz);

1- (3-Cyclopropyl-2-{[4- (1-methylethyl) -2,5-dimethylphenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H -NMR (CDCl ₃ ) δ: 7.41 (1 H, t, J = 7.9 Hz), 7.25-7.23 (2 H, m), 6.65 (1 H, s), 6.63 (1 H, s), 5.17 (2 H, s), 4.34-4.30 (1H, m), 3.63 (3H, s), 2.17-2.12 (4H, m), 2.02 (3H, s), 1.29 (6H, d, J = 6.1 Hz), 1.02-0.97 (2H, s) m), 0.78-0.74 (2H, m) .; 1- [2-({[1- (6-fluoropyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methyl Phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.40 (1 H, s), 8.04-7.99 (1 H, m), 7. 65 (1 H, d, J = 2.5 Hz), 7.43-7.38 (2H, m), 7.27-7.26 (1 H, m), 7.01 (1 H, dd, J = 8.8, 3.4 Hz), 5.86 (1 H, d, J = 2.7 Hz), 5.33 (2H, s), 3.66 (3H, s), 2.56 (3H, s) .; 1- (3-methyl-2) {[2-methyl-4- (5-chloro-1-methyl -1H- pyrazole-3 -yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydro-5-one, ¹ H- NMR (CDCl ₃ ) δ: 7.52-7.41 (4 H, m), 7. 29-7. 27 (1 H, m), 6. 85 (1 H, d, J = 8.5 Hz), 6.41 (1 H, s), 5.06 (2 H, s) , 3.87 (3H, s), 3.62 (3H, s), 2.51 (3H, s), 2.12 (3H, s) .; 1- [3-methyl-2-({2,5-dimethyl-4-[{, (Dimethylamino) carbonyl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.45-7.39 (2H, m), 7.28-7.26 (1H, m), 6.91 (1H, s), 6.63 (1H, s), 5.01 (2H, s), 3.66 (3H, s), 3.11 (3H, s), 2.85 (3H, s), 2.50 (2.5) 3H, s), 2.24 (3H, s), 2.03 (3H, s). 1- (3-ethyl-2-{[2-methyl-4- (5-fluoro-1-methyl-1H-pyrazole-) 3-yl) fe Carboxymethyl] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.52-7.41 (4H, m), 7.30-7.27 (1H, m), 6.86 (1 H, d, J = 8.4 Hz), 5. 95 (1 H, d, J = 5.7 Hz), 5.07 (2 H, s), 3. 76 (3 H, d, J = 1.1 Hz), 3.58 (3 H, s), 2.85 (2H, q, J = 7.6 Hz), 2.10 (3H, s), 1.28 (3 H, t, J = 7.4 Hz) .; 1- [2-({[1- (2-fluoropyridine-3-). I) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.31 to 8.26 (1H, m), 8.03-8.01 (1H, m), 7. 92 (1H, t, J = 2.5 Hz), 7.43-7.26 (4H, m), 5. 88 (1 H, d, J = 2.7 Hz), 5.33 ( 2H, s), 3.65 (3H, s), 2.56 (3H, s) .; 1- {2-[({1- [4- (adamantan-1-yl) phenyl] -1H-pyrazol-3-yl] } Oxy) methyl] -3-methylphenyl} -4- _{^{Chill-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.43-7.38 (2H, m), 7.27-7.25 (3H, m), 6.83 (2H, dt, J = 9.6 , 2.7 Hz), 4.99 (2 H, s), 3.61 (3 H, s), 2. 49 (3 H, s), 2.08 (3 H, s), 1. 87 (6 H, d, J = 2.5 Hz), 1.80-1. 71 (6 H) , m) .; 1- [2-({[1- (3-propoxy-2-methoxypyridin-4-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4 -Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.26 (1 H, d, J = 2.7 Hz), 7.88 (1 H, d, J = 5.7 Hz), 7.42- 7.39 (3H, m), 7.26-7.26 (1H, m), 5.84 (1H, d, J = 2.7 Hz), 5.33 (2H, s), 4.03 (3H, s), 3.90 (2H, t, J = 6.9 Hz), 3.64 (3 H, s), 2.56 (3 H, s), 1. 76-1. 72 (2 H, m), 0.97 (3 H, t, J = 7.4 Hz) .; 1- (3-methoxy-2- { [2,5-Dimethyl-4- (ethoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1 _{^{4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.67 (1H, s), 7.49-7.45 (1H, m), 7.10-7.06 (2H, m), 6.71 (1H, s) , 5.31 (2H, s), 4.30 (2H, q, J = 7.1 Hz), 3.94 (3H, s), 3.60 (3H, s), 2.56 (3H, s), 1.96 (3H, s), 1.36 ( 3 H, t, J = 7.1 Hz) .; 1- [2-({[1- (2-formylphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl ^-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 10.09 (1 H, s), 7.99 (1 H, d, J = 7.8 Hz), 7.64 (1 H, t, J = 7.3) Hz), 7.56 (1 H, d, J = 2.7 Hz), 7.45-7.40 (4 H, m), 7.26-7.23 (1 H, m), 5. 90 (1 H, d, J = 2.5 Hz), 5.30 (2 H, s) ), 3.63 (3H, s), 2.54 (3H, s) .;

1- [3-Methyl-2-({2,5-dimethyl-4-[(1,1-dimethylethoxy) carbonyl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 7.63 (1 H, s), 7. 45-7. 39 (2 H, m), 7. 29-7. 27 (1 H, m), 6.62 ( ¹ H, s), 5.0 6 (2 H, s) , 3.64 (3H, s), 2.55 (3H, s), 2.49 (3H, s), 2.05 (3H, s), 1.57 (9H, s) .; 1- [2-({[1- (2-) Chloropyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.34 (1 H, dd, J = 4.5, 1.8 Hz), 7.96 (1 H, dd, J = 7.9, 1.8 Hz), 7.89 (1 H, d, J = 2.7 Hz), 7.43-7.36 (3 H, m) , 7.28-7.26 (1H, m), 5.88 (1H, d, J = 2.7 Hz), 5.31 (2H, s), 3.64 (3H, s), 2.56 (3H, s). {[1- (3-oxocyclohexyl) -1H- Pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.37-7.34 (2H, m) , 7.22 (1 H, dd, J = 6.6, 2.7 Hz), 7.11 (1 H, d, J = 2.3 Hz), 5.52 (1 H, d, J = 2.5 Hz), 5.19 (2 H, s), 4.28-4.21 ( 1H, m), 3.68 (3H, s), 2.88 (1H, dd, J = 14.3, 10.4 Hz), 2.71 (1H, dd, J = 14.4, 4.9 Hz), 2.53 (3H, s), 2.43-2.40 (2H, m), 2.17-2.12 (2H, m), 2.05-2.02 (1H, m), 1.74-1.62 (1H, m) .; 1- (3-methoxy-2-{[2,5-dimethyl] -4- (1-ethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46 ( 1H, t, J = 8.2 Hz), 7. 39 (1 H, d, J = 2.3 Hz), 7. 27 (1 H, s), 7.09-7.06 (2 H, m), 6. 75 (1 H, s), 6. 30 (1 H, d) , J = 2.3 Hz), 5.26 (2 H, s), 4. 20 (2 H, q, J = 7.3 Hz), 3. 93 (3 H, s), 3.59 (3 H, s), 2.41 (3 H, s), 1.9 7 (3H, s), 1.51 (3H, t, J = 7.4 Hz) .; 1- (3-ethyl-2-{[2,5-dimethyl-4- (5-fluoropyrimidin-2-yl) phenoxy] Methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.65 (2H, s), 7.62 (1H, s), 7.50 to 7.44 (2H) , m), 7.29 (1H, dd, J = 7.3, 2.1 Hz), 6.74 (1H, s), 5.10 (2H, s), 3.62 (3H, s), 2.85 (2H, q, J = 7.6 Hz) , 2.54 (3H, s), 2.08 (3H, s), 1.29 (3H, t, J = 7.4 Hz) .; 1- (3-Methyl-2-{[2-methyl-4- (pyridazine-3-). [Ill] phenoxy] methyl} phenyl) -4-methyl- ¹ , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 9.09 (1 H, dd, J = 4.8, 1.6 Hz), 7.90 ( 1H, d, J = 1.6 Hz), 7.87 (1 H, dd, J = 8.5, 2.3 Hz), 7.79 (1 H, dd, J = 8.5, 1.6 Hz), 7.49-7.42 (3 H, m), 7.29 (1 H , dd, J = 7.0, 2.4 Hz), 6.97 (1 H, d, J = 8.5 Hz), 5.12 (2 H, s), 3.63 (3 H, s), 2.52 (3 H) , s), 2.18 (3H, s) .; 1- [2-({[1- (2-methoxypyridin-4-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl ] ^1- H-NMR (CDCl ₃ ) δ: 8.14 (1 H, d, J = 5.9 Hz), 7.74 (1 H, d, J = 2.7 Hz) , 7.43-7.38 (2H, m), 7.27-7.25 (1H, m), 7.09 (1H, dd, J = 5.8, 1.9 Hz), 6.89 (1H, d, J = 1.8 Hz), 5.87 (1H, d) , J = 2.7 Hz), 5.34 (2H, s), 3.98 (3H, s), 3.66 (3H, s), 2.56 (3H, s) .; 1- [3-methyl-2- ({2-methyl {2 -4- [1- (2-methylpropyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ δ: 7.57-7.57 (1 H, m), 7.53 (1 H, dd, J = 8.5, 2.3 Hz), 7.44-7.39 (2 H, m), 7.34 (1 H, d, J = 2.3 Hz), 7.28-7.27 (1H, m), 6.85 (1H, d, J = 8.5 Hz), 6.43 (1 H, d, J = 2. 3 Hz), 5.06 (2H, s), 3.92 (2H, d, J = 7.3 Hz), 3.62 (3H, s), 2.50 (3H, s), 2.29-2.22 (1H, m), 2.12 (3H, s) s), 0.92 (6 H, d, J = 6.6 Hz) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-fluoro-6-methylpyridin-2-yl) phenoxy] Methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.45-7.40 (2H, m), 7.33 (1 H, t, J = 8.8 Hz ), 7.29-7.27 (1H, m), 7.15 (1H, dd, J = 8.4, 3.6 Hz), 7.12 (1H, s), 6.71 (1H, s), 5.05 (2H, s), 3.67 (3H, s) s), 2.56 (3H, d, J = 2.9 Hz), 2.51 (3H, s), 2.30 (3H, s), 2.08 (3H, s) .; 1- (3-methoxy-2-{[2, 2, 3] 5-Dimethyl-4- (propoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.68 (1 H, s), 7.47 (1H, t, J = 8.2 Hz), 7.10-7.06 (2H, m), 6.72 (1H, s), 5.31 (2H, s), 4.20 (2H, t, J = 6.6 Hz), 3.94 (3H, s), 3.60 (3H, s), 2.56 (3H, s), 1.96 (3H, s), 1.81-1. 72 (2H, m), 1.01 ( 3H, t, J = 7.4 Hz) .;

1- (2-{[(1-Hexyl-1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-6-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2 H, m), 7.23 (1 H, dd, J = 6.2, 3.1 Hz), 7.08 (1 H, d, J = 2.3 Hz), 5. 50 (1 H, d, J = 2.3 Hz), 5.19 (2H, s), 3.87 (2H, t, J = 7.2 Hz), 3.68 (3H, s), 2.53 (3H, s), 1.79-1.72 (2H, m), 1.30-1.2 (6H) , m), 0.88 (3 H, t, J = 6.9 Hz) .; 1- [2-[{[1- (thiazol-2-yl) -1 H-pyrazol-3-yl] oxy} methyl) -3-] Methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.07 (1 H, d, J = 2.7 Hz), 7.44 (1 H, d, J = 3.7 Hz), 7.43-7.38 (2 H, m), 7. 28-7. 25 (1 H, m), 7.00 (1 H, d, J = 3.7 Hz), 5. 85 (1 H, d, J = 2.7 Hz), 5.33 (2 H, s) ), 3.68 (3H, s), 2.57 (3H, s) .; 1- [2-({[1- (3-nitrophenyl)] ¹ ) ¹ H-NMR (CDCl ₃ ) δ: 8.39 (1H)-) ¹ H-Pyrazol-3-yl] oxy} methyl) 3-methylphenyl] 4-methyl- ¹ , 4-dihydrotetrazol-5-one , t, J = 2.2 Hz), 8.03 (1 H, d, J = 8.2 Hz), 7. 91 (1 H, d, J = 8.2 Hz), 7. 78 (1 H, d, J = 2.7 Hz), 7.58 (1 H, t , J = 8.2 Hz), 7.43-7.38 (2 H, m), 7. 30-7. 25 (1 H, m), 5. 90 (1 H, d, J = 2.5 Hz), 5. 36 (2 H, s), 3. 67 (3 H, s) , 2.58 (3H, s) .; 1- [2-({[1- (2-chloro-4-methylphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4 -Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.63 (1 H, d, J = 2.5 Hz), 7.43-7.38 (3 H, m), 7.27 (2 H, m ), 7.15 (1H, d, J = 8.7 Hz), 5.80 (1H, d, J = 2.5 Hz), 5.30 (2H, s), 3.62 (3H, s), 2.55 (3H, s), 2.37 (3H) , s) .; 1- (3-methoxy-2-{[2,5-dimethyl-4- (methoxy). Boniru) phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.68 (1H, s), 7.48 (1H, t, J = 8.3 Hz), 7.10-7.06 (2H, m), 6.72 (1H, s), 5.31 (2H, s), 3.94 (3H, s), 3.83 (3H, s), 3.60 (3H, s), 2.56 (3H) , s), 1.95 (3H, s) .; 1- (3-Cyclopropyl-2-{[2-methyl-4- (5-methoxy-1-methyl-1H-pyrazol-3-yl) phenoxy] methyl } Phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.47-7.41 (1 H, m), 7.29-7.27 (2H, m), 7.18-7.14 (2H, m), 6.93 (1H, d, J = 8.2 Hz), 5.64 (1H, s), 5.29 (2H, s), 3.90 (3H, s), 3.71 (3H, s), 3.63 (3H, s) s), 2.18-2.10 (1H, m), 2.12 (3H, s), 1.03-0.98 (2H, m), 0.80-0.76 (2H, m) .; 1-[2- ({[1-(1) -Methyl-1H-imidazol-5-yl) -1H-pyrazol-3-yl] o Xymethyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43 (1 H, s), 7.42-7. 37 (2 H, m) ), 7.31 (1 H, d, J = 2.5 Hz), 7.26-7.24 (1 H, m), 7.04 (1 H, s), 5. 78 (1 H, d, J = 2.5 Hz), 5. 29 (2 H, s), 3.59 (3H, s), 3.49 (3H, s), 2.54 (3H, s) .; 1- [3-methyl-2-({2,5-dimethyl-4- [1- (2-methylpropyl)- 1H-Pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-7.39 (2H, m), 7.36 (1H, d, J = 2.1 Hz), 7.30-7.27 (2H, m), 6.70 (1H, s), 6.29 (1H, d, J = 2.3 Hz), 5.04 (2H, s), 3.93 (2H, s) d, J = 7.3 Hz), 3.65 (3H, s), 2.51 (3H, s), 2.41 (3H, s), 2.29-2.23 (1H, m), 2.07 (3H, s), 0.93 (6H, d) , J = 6.6 Hz) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-chloro-6-methylpi) Lysyn-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.63 (1 H, d, J = 8.2 Hz), 7.45-7.40 (2H, m), 7.29-7.26 (1H, m), 7.14 (2H, t, J = 3.9 Hz), 6.71 (1H, s), 5.05 (2H, s), 3.67 (3H, s) , 2.66 (3H, s), 2.51 (3H, s), 2.32 (3H, s), 2.08 (3H, s) .; 1- [3-methyl-2-({2-methyl-4- [5-]. (Difluoromethyl) -3-methyl-1H-pyrazol-1-yl] phenoxy} methyl) phenyl)]-4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46-7.41 (2H, m), 7.29 (1H, dd, J = 7.1, 2.1 Hz), 7.23-7.18 (2H, m), 6.88 (1H, d, J = 8.7 Hz), 6.55 (1H, t, J = 53.8 Hz), 6.49 (1H, s), 5.08 (2H, s), 3.64 (3H, s), 2.51 (3H, s), 2.35 (3H, s), 2.12 (3H, s).

1- {2-[({1- [2- (trifluoromethyl) phenyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazole -5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.77 (1 H, d, J = 8.0 Hz), 7. 64 (1 H, t, J = 7.6 Hz), 7.52-7.48 (2 H, m), 7.43 ( 1H, d, J = 2.5 Hz), 7. 40-7. 38 (2 H, m), 7. 26-7. 25 (1 H, m), 5. 83 (1 H, d, J = 2.5 Hz), 5. 28 (2 H, s), 3.61 (3 H) , s), 2.54 (3H, s) .; 1- [2-({[1- (3,4,5-trifluorophenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methyl Phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 (1 H, d, J = 2.5 Hz), 7.43-7.38 (2 H, m), 7.26 -7.25 (1 H, m), 7.21-7.19 (2 H, m), 5. 85 (1 H, d, J = 2.7 Hz), 5.32 (2 H, s), 3.67 (3 H, s), 2.56 (3 H, s). 1- [2-({[1- (2,6-difluo); ) -1H- pyrazole-3 -yl] oxy} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.41-7.39 (3H, m), 7. 35-7. 28 (1 H, m), 7. 26-7. 24 (1 H, m), 7.0 4 (2 H, t, J = 8.6 Hz), 5. 86 (1 H, d, J = 2.5 Hz), 5. 28 ( 2H, s), 3.64 (3H, s), 2.54 (3H, s) .; 1- {2-[({1- [6- (1,1-dimethylethyl) pyridin-2-yl] -1H- Pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.45 (1 H, t, J = 7.8 Hz), 7.38 (2H, d, J = 4.8 Hz), 7.26-7.24 (1 H, m), 6.84 (1 H, d, J = 7.6 Hz), 6.43 (1 H, d, J = 8.0 Hz), 5.41 (2H, s), 3.62 (3H, s), 2.51 (3H, s), 1.29 (9H, s) .; 1- {2-[({1- [2, 3, 5, 6-tetrafluoro- 4- (trifluoromethyl) pheny ]-1H-pyrazol-3-yl} oxy) methyl] -3-methyl-phenyl} _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.53-7.52 ( 1H, m), 7.41-7. 37 (2H, m), 7.23 (1H, dd, J = 6.2, 2.8 Hz), 5.95 (1 H, d, J = 2.7 Hz), 5.32 (2H, s), 3.69 (3H , s), 2.55 (3H, s) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-methyl-4,5-dihydro-1,3-oxazole-2-) [Ill] phenoxy] methyl} phenyl) -4- methyl- ¹ , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.57 (1 H, s), 7. 45-7. 39 (2 H, m), 7.29-7.26 (1H, m), 6.66 (1H, s), 5.06 (2H, s), 4.81-4.72 (1H, m), 4.16-4.09 (1H, m), 3.63-3.58 (4H, m), 2.56 (3H, s), 2.49 (3H, s), 2.05 (3H, s), 1.40 (3H, d, J = 6.3 Hz) .; 1- (3-methyl-2-{[2,5-dimethyl] -4- (1-Cyclopropyl-1H-pyrazo) -5-yl) phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.46-7.41 (3H, m), 7.28 (1H , dd, J = 6.8, 2.5 Hz), 7.01 (1 H, s), 6. 75 (1 H, s), 6. 13 (1 H, d, J = 1.8 Hz), 5.06 (2 H, s), 3. 67 (3 H, s) , 3.34-3.28 (1H, m), 2.54 (3H, s), 2.16 (3H, s), 2.08 (3H, s), 1.15-1.11 (2H, m), 0.83 to 0.78 (2H, m). 1- (3-ethyl-2-{[2,5-dimethyl-4- (cyclopropanecarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 (1 H, s), 7.51-7. 44 (2 H, m), 7. 29 (1 H, dd, J = 7.3, 1.8 Hz), 6.68 (1 H, s), 5.09 (2 H, s), 3.61 (3H, s), 2.85 (2H, q, J = 7.6 Hz), 2.49 (3H, s), 2.47-2.40 (1H, m), 2.08 (3H, s), 1.26 (3H, t, J = 7.6 Hz), 1.21-1.17 (2H, m), 1.00-0.96 (2H, m) .; 1- [3-methyl-2-({2,5-dimethyl-4-[(meth) Shiimino) methyl] phenoxy} methyl) phenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.26 (1H, s), 7.48 (1H, s), 7.45-7.39 (2H, m), 7.28-7.27 (1H, m), 6.61 (1H, s), 5.04 (2H, s), 3.95 (3H, s), 3.64 (3H, s), 2.49 (3H, s) s), 2.36 (3H, s), 2.05 (3H, s) .; 1- (3-methyl-2-{[4- (1-methylpropoxy) -2,5-dimethylphenoxy] methyl} phenyl)- 4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.23 (1H, m), 6.63 (1H, s), 6.61 (1H, s), 4.95 (2H, s), 4.15-4.09 (1H, m), 3.64 (3H, s), 2.51 (3H, s), 2.17 (3H, s), 2.03 (3H, s) , 1.75-1.67 (1 H, m), 1.65-1. 56 (1 H, m), 1.24 (3 H, d, J = 6.1 Hz), 0.97 (3 H, t, J = 7.5 Hz) .;

1- (3-methyl-2-{[2,5-dimethyl-4- (3-methylbutanoyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H -NMR (CDCl ₃ ) δ: 7.46-7.38 (3H, m), 7.28 (1H, dd, J = 7.3, 2.1 Hz), 6.68 (1H, s), 5.07 (2H, s), 3.64 (3H, s) ), 3.43-3.34 (1H, m), 2.51 (3H, s), 2.46 (3H, s), 2.08 (3H, s), 1.15 (6H, d, J = 6.9 Hz) .; 1-(3- Methoxy-2-{[2,5-dimethyl-4- (5-fluoropyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.64 (2 H, s), 7.58 (1 H, s), 7. 47 (1 H, t, J = 8.2 Hz), 7.08 (2 H, dd, J = 8.2, 6.0 Hz), 6.79 (1 H, s), 5.31 (2H, s), 3.94 (3H, s), 3.60 (3H, s), 2.51 (3H, s), 2.00 (3H, s) .; 1- (2-{[(1-octyl). -1H-pyrazol-3-yl) oxy] methyl} -3-Methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2H, m), 7.23 (1 H, dd, J = 6.3 , 2.9 Hz), 7.08 (1 H, d, J = 2.3 Hz), 5. 50 (1 H, d, J = 2.3 Hz), 5.19 (2 H, s), 3.87 (2 H, t, J = 7.1 Hz), 3.67 (3 3H, s), 2.53 (3H, s), 1.79-1.72 (2H, m), 1.27 (10H, s), 0.88 (3H, t, J = 6.9 Hz) .; 1- [2-({[1 -(Thiazol-5-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.51 (1 H, s), 7. 76 (1 H, s), 7.53 (1 H, d, J = 2.7 Hz), 7.42-7.37 (2 H, m), 7.26-7.24 (1 H, m), 5.82 (1 H , d, J = 2.7 Hz), 5.30 (2H, s), 3.66 (3H, s), 2.56 (3H, s) .; 1- [2-({[1- (pyridin-3-yl) -1H] -Pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4 _{^{Dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.86 (1H, d, J = 2.7 Hz), 8.46 (1H, dd, J = 4.8, 1.4 Hz), 7.90 (1H, dq, J = 8.3, 1.4 Hz), 7.72 (1 H, d, J = 2.7 Hz), 7.42-7.38 (2 H, m), 7.36 (1 H, dd, J = 8.4, 4.8 Hz), 7.28-7.25 (1 H, m) , 5.87 (1H, d, J = 2.5 Hz), 5.35 (2H, s), 3.65 (3H, s), 2.57 (3H, s) .; 1- (3-methyl-2-{[3,5-] Dimethyl-4- (methoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-7.38 (2H, m), 7.28 -7.26 (1H, m), 6.53 (2H, s), 5.00 (2H, s), 3.88 (3H, s), 3.63 (3H, s), 2.47 (3H, s), 2.29 (6H, s). 1- (3-methoxy-2-{[2,5-dimethyl-4- (isopropoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H- NMR (CDCl ₃ ) δ: 7.65 (1 H, s), 7. 47 (1 H, t, J = 8.1 Hz), 7.10-7.06 (2H, m), 6.71 (1 H, s), 5.30 (2 H, s), 5.22-5. 15 (1 H, m), 3.94 (3 H, s), 3. 60 (3 H, s) ), 2.55 (3H, s), 1.96 (3H, s), 1.34 (6H, d, J = 6.4 Hz) .; 1- [3-Methyl-2-({2-methyl-4- [3- (3) Trifluoromethyl) -5-methyl-1H-pyrazol-1-yl] phenoxy} methyl) phenyl)]-4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.47-7.40 (2H, m), 7.29 (1H, dd, J = 7.1, 2.1 Hz), 7.19-7.15 (2H, m), 6.89 (1H, d, J = 8.5 Hz), 6.42 (1H, s) , 5.08 (2H, s), 3.65 (3H, s), 2.52 (3H, s), 2.30 (3H, s), 2.13 (3H, s). 5-Dimethyl-4- (ethoxycarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.72 (1 H, s), 7.45 -7.40 (2H, m), 7.28 (1 H, dd, J = 7.2, 2.0 Hz), 6.65 (1 H, s), 5. 07 (2H, s), 4.31 (2H, q, J = 7.1 Hz), 3.64 (3H, s), 2.58 (3H, s), 2.50 (3H, s), 2.06 (3H, s), 1.37 (3H) , t, J = 7.1 Hz) .; 1- (2-{[(1-butyl-1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydro Tetrazole-9-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2H, m), 7.23 (1 H, dd, J = 6.2, 3.1 Hz), 7.08 (1 H, d, J = 2.3 Hz) , 5.50 (1H, d, J = 2.3 Hz), 5.19 (2H, s), 3.88 (2H, t, J = 7.1 Hz), 3.68 (3H, s), 2.53 (3H, s), 1.78-1.71 ( 2H, m), 1.30-1. 26 (2H, m), 0.92 (3H, t, J = 7.5 Hz).

1- [2-({[1- (2-propoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole -5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.14 (1 H, d, J = 2.7 Hz), 8.07 (1 H, dd, J = 7.8, 1.7 Hz), 7.99 (1 H, dd, J = 4.8) , 1.8 Hz), 7.43-7.38 (2H, m), 7.28-7.25 (1 H, m), 6.99 (1 H, dd, J = 7.8, 4.9 Hz), 5.80 (1 H, d, J = 2.7 Hz), 5.31 (2H, s), 4.40 (2H, t, J = 6.7 Hz), 3.64 (3H, s), 2.55 (3H, s), 1. 88-1.84 (2H, m), 1.05 (3H, t, J = 7.5) Hz) .; 1- [3-Methyl-2-({2-methyl-4- [1- (2,2-difluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4- Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 to 7.51 (2H, m), 7.46 to 7.40 (3H, m), 7.31-7. 27 (1H, m), 6.86 (1H, d, J = 8.4 Hz), 6.52 (1H, d, J = 2) .5 Hz), 6.14 (1 H, tt, J = 55.7, 4.4 Hz), 5.07 (2 H, s), 4. 48 (2 H, td, J = 13.4, 4.5 Hz), 3.62 (3 H, s), 2.51 (3 H) , s), 2.13 (3H, s) .; 1- (3-methoxy-2-{[2,5-dimethyl-4- (3-methylbutanoyl) phenoxy] methyl} phenyl) -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 to 7.45 (1H, m), 7.36 (1H, s), 7.12 to 7.06 (2H, m), 6.74 (1H, s) ), 5.31 (2H, s), 3.95 (3H, s), 3.62 (3H, s), 3.42-3.33 (1H, m), 2.44 (3H, s), 1.98 (3H, s), 1.14 (6H, s). d, J = 6.9 Hz) .; 1- {2-[({1- [2- (Difluoromethyl) -6-methoxypyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3 -Methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.65 (1 H, d, J = 8.7 Hz), 7.42-7.39 (3 H, m) , 7.26-7.24 (1 H, m), 6.92 (1 H, d, J = 8.7 Hz), 5.82 (1 H, d, J = 2.5 Hz), 5.29 (2 H, s), 4.03 (3 H, s), 3.61 (3 H, s), 3. 35 (1 H, s), 2.55 (3 H, s). {[1- (6-Methoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.33 (1 H, d, J = 2.7 Hz), 7.81 (1 H, dd, J = 8.8, 2.9 Hz), 7.56 (1 H, d, J = 2.5 Hz), 7.42-7.37 (2H, m), 7. 27-7. 24 (1 H, m), 6.81 (1 H, d, J = 8.7 Hz), 5. 80 (1 H, d, J = 2.7 Hz), 5.32 (2 H, s), 3. 96 (3 H, 3) s), 3.64 (3H, s), 2.56 (3H, s) .; 1- [2-({[1- (2,2-dimethylpropyl) -1H-pyrazol-3-yl] oxy} methyl)- 3-Methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38-7.34 (2H, m), 7.23 (1 H, dd, J = 6.4, 2.7 Hz), 7.05 (1 H, d, J = 2.5 Hz), 5.51 (1 H, d, J = 2.3 Hz), 5. 19 (2 H, s) ), 3.67 (3H, s), 3.66 (2H, s), 2.52 (3H, s), 0.90 (9H, s) .; 1- {2-[({1- [2- (adamantan-1-yl]) ) Ethyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39- 7.34 (2H, m), 7.23 (1 H, dd, J = 6.1, 3.2 Hz), 7.08 (1 H, d, J = 2.5 Hz), 5.50 (1 H, d, J = 2.3 Hz), 5.18 (2 H, s ), 3.93-3.89 (2H, m), 3.68 (3H, s), 2.53 (3H, s), 1.96 (3H, s), 1.72 (3H, d, J = 12.0 Hz), 1.64 (3H, d, J = 12.2 Hz), 1.60-1. 56 (2H, m), 1.52 (6 H, d, J = 2.5 Hz). 1- [2-({[1- (furan-2-yl) -1 H-pyrazole-] 3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.57 (1 H, d, J = 2.5 Hz ), 7.40-7.39 (2H, m), 7.26-7.24 (1H, m), 7.20 (1H, dd, J = 2.1, 1.1 Hz), 6. 44 (1H, dd, J = 3.3, 1.9 Hz), 6.16 (1H, dd, J = 3.2, 0.9 Hz), 5.78 (1 H, d, J = 2.7 Hz), 5.29 (2H, s), 3.65 (3H , s), 2.54 (3H, s) .; 1- {2-[({1- [3- (1-methylethoxy) -2-methoxypyridin-4-yl] -1H-pyrazol-3-yl} Oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.28 (1 H, d, J = 2.7 Hz), 7.88 ( 1H, d, J = 5.7 Hz), 7.43-7.38 (2 H, m), 7. 37 (1 H, d, J = 5.5 Hz), 7.28-7. 25 (1 H, m), 5.82 (1 H, d, J = 2.7 Hz) ), 5.33 (2H, s), 4.54-4.41 (1H, m), 4.02 (3H, s), 3.64 (3H, s), 2.56 (3H, s), 1.20 (6H, d, J = 6.2 Hz) ; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-fluoro-1-methyl-1H-pyrazol-3-yl) phenyoxy] cymethyl} phenyl) -4-methyl-1 , 4-Dihydrotetrazol-5-one, ¹ H-NMR (CD Cl ₃ ) δ: 7.44-7.37 (2H, m), 7.30-7.27 (2H, m), 6.68 (1H, s), 5.83 (1H, d, J = 5.7 Hz), 5.04 (2H, s), 3.77 (3H, d, J = 1.1 Hz), 3.64 (3H, s), 2.51 (3H, s), 2.40 (3H, s), 2.06 (3H, s).

1- [2-({[1- (6-methoxy-2-methylpyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.48 (1 H, d, J = 8.5 Hz), 7.41-7. 37 (2 H, m), 7. 27-7. 23 (2 H, m), 6.63 (1H, d, J = 8.5 Hz), 5. 76 (1 H, d, J = 2.5 Hz), 5. 28 (2 H, s), 3. 95 (3 H, s), 3.59 (3 H, s), 2.55 (3 H, s) , 2.33 (3H, s) .; 1- {2-[({1- [2- (2,2,2-trifluoroethoxy) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) Methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.17 (1 H, dd, J = 7.9, 1.6 Hz), 8.06 1H, d, J = 2.7 Hz), 7. 98 (1 H, dd, J = 4.9, 1.7 Hz), 7.43-7.38 (2 H, m), 7.29-7.25 (1 H, m), 7.12 (1 H, dd, J = 7.9, 4.8 Hz), 5.84 (1 H, d, J = 2) .7 Hz), 5.32 (2H, s), 4.87 (2H, q, J = 8.4 Hz), 3.64 (3H, s), 2.55 (3H, s) .; 1- [3-Methyl-2-({{} 2,5-Dimethyl-4- [1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazole-5 ^-1 H-NMR (CDCl ₃ ) δ: 7.52 (1H, d, J = 2.0 Hz), 7.44-7.39 (2H, m), 7.30-7.27 (2H, m), 6.71 (1H, s), 6.44 (1H, dd, J = 2.4, 1.0 Hz), 5.05 (2H, s), 4.73 (2H, q, J = 8.2 Hz), 3.64 (3H, s), 2.51 (3H, s), 2.41 (3H) , s), 2.07 (3H, s) .; 1- (3-Methyl-2-{[2,5-dimethyl-4- (5-chloro-1-methyl-1H-pyrazol-3-yl) phenokil] Simethyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-7.39 (2H, m), 7.28-7.27 (2H, m), 6.69 ( 1H, s), 6.29 (1H, s), 5.04 (2H, s), 3.88 ( 3H, s), 3.64 (3H, s), 2.51 (3H, s), 2.40 (3H, s), 2.06 (3H, s) .; 1- (3-ethyl-2-{[2-methyl-4] -(5-Fluoropyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.61 (2H, s), 8.19 (1H, d, J = 8.2 Hz), 8.15 (1 H, s), 7.53-7.46 (2 H, m), 7.31 (1 H, dd, J = 7.0, 1.9 Hz), 6.95 (1 H, d, J = 8.7 Hz), 5.14 (2H, s), 3.60 (3H, s), 2.87 (2H, q, J = 7.5 Hz), 2.16 (3H, s), 1.30 (3 H, t, J = 7.7 Hz); 1- [2-({[1- (4-chloro-2-ethoxyphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole -5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.95 (1 H, d, J = 2.5 Hz), 7. 68 (1 H, d, J = 8.6 Hz), 7. 39 (2 H, m), 7. 25 (1 H, m), 7.00 (1 H, dd, J = 8.6, 2.3 Hz), 6.96 (1 H, d, J = 2.3 Hz), 5. 77 (1 H, d, J) J = 2.5 Hz), 5.30 (2 H, s), 4.13-4.06 (2 H, m), 3.62 (3 H, s), 2.55 (3 H, s), 1.44 (3 H, t, J = 6.9 Hz) .; 1 -[2-({[1- (2-bromo-6-methoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4 -Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.65 (1 H, d, J = 8.6 Hz), 7.55 (1 H, d, J = 2.5 Hz), 7.40-7. 39 (2 H, m) , 7.26-7.25 (1H, m) 6.78 (1H, d, J = 8.6 Hz), 5.81 (1H, d, J = 2.5 Hz), 5.28 (2H, s), 3.98 (3H, s), 3.63 (3H) , s), 2.55 (3H, s) .; 1- [2-({[1- (4-formylphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4- Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 9.98 (1 H, s), 7. 94 (2 H, d, J = 8.5 Hz), 7. 80 (1 H, d, J = 2.5 Hz), 7.73 (2H, d, J = 8.5 Hz), 7.43-7.39 (2H, m), 7.27-7.25 ( 1H, m), 5.91 (1H, d, J = 2.5 Hz), 5.36 (2H, s), 3.64 (3H, s), 2.57 (3H, s) .; 1- [2-({[1- (1) Tetrahydrofuran-2-ylmethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ 7.39-7.34 (2H, m), 7.23 (1H, dd, J = 6.5, 2.8 Hz), 7.20 (1 H, d, J = 2.3 Hz), 5.53 (1 H, d, J = 2.3 Hz), 5.19 (5 2H, s), 4.19-4.15 (1 H, m), 4.01 (1 H, dd, J = 14.3, 4.1 Hz), 3.91 (1 H, dd, J = 14.2, 6.2 Hz), 3.82-3. 78 (1 H, m) , 3.75-3.72 (1H, m), 3.68 (3H, s), 2.52 (3H, s), 1.90-1.91 (1 H, m), 1. 88-1. 78 (1 H, m), 1. 75-1. 71 (1 H, m) , 1.5-1 .55 (1 H, m) .; 1- [2-({[1- (pyridin-2-yl) -1 H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4- Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.34-8.32 (2H, m), 7.77-7.76 (2H, m), 7.43-7.38 (2H, m), 7.28-7.25 (1H, m), 7.10-7.08 (1H, m), 5.84 (1H, d, J = 2.7 Hz) , 5.34 (2H, s), 3.64 (3H, s), 2.56 (3H, s) .;

1- (3-Methyl-2-{[2,5-dimethyl-4- (5-chloro-1,4-dimethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-4.39 (2H, m), 7.30-7.27 (1H, m), 6.97 (1H, s), 6.71 (1H, s) ), 5.04 (2H, s), 3.84 (3H, s), 3.65 (3H, s), 2.51 (3H, s), 2.20 (3H, s), 2.05 (3H, s), 1.89 (3H, s) 1- (2-{[(1- {2- [2- (2-methoxyethoxy) ethoxy] ethyl} -1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl) -4- Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2H, m), 7.23 (1 H, dd, J = 6.3, 2.9 Hz), 7.21 (1 H, d, J = 2.3 Hz, 5. 50 (1 H, d, J = 2.3 Hz), 5. 18 (2 H, s), 4.06 (2 H, t, J = 5.3 Hz), 3. 75 (2 H, t, J = 5.3 Hz) , 3.68 (3H, s), 3.59-3.58 (4H, m), 3.54-3.5 2 (4H, m), 3.37 (3H, s), 2.53 (3H, s) .; 1- [2-({[1- (5-fluoro-6-methoxypyridin-2-yl) -1H-pyrazole] -3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.17 (1 H, d, J = 2.5) Hz), 7.43-7.39 (3H, m), 7.28-7. 23 (2H, m), 5.81 (1H, d, J = 2.7 Hz), 5.32 (2H, s), 4.04 (3H, s), 3.65 (3H) , s), 2.56 (3H, s) .; 1- [3-Methyl-2-({2,5-dimethyl-4- [1- (2,2-difluoroethyl) -1H-pyrazol-5-yl ] Phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.60 (1 H, d, J = 1.4 Hz), 7.46-7.41 (2 H) , m), 7.30-7.27 (1H, m), 6.92 (1H, s), 6.74 (1H, s), 6.19 (1H, d, J = 1.6 Hz), 6.14 (1 H, tt, J = 4.6, 55.6) Hz), 5.06 (2H, s), 4.21 (2H, td, J = 13. 1, 4.6 Hz), 3.67 (3H, s), 2.54 (3H, s), 2.09 (3H, s), 2.07 (3H, s). 1- [2-({[1- (3-cyanophenyl). ) -1H-Pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.88 (1 H, s), 7.78 (1H, d, J = 8.0 Hz), 7.70 (1H, d, J = 2.7 Hz), 7.53-7.46 (2H, m), 7.43-7.38 (2H, m), 7.28-7.26 (1H , m), 5.88 (1H, d, J = 2.7 Hz), 5.34 (2H, s), 3.67 (3H, s), 2.57 (3H, s) .; 1- {3-methoxy-2-[(2) 5-Dimethyl-4-ethanoylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 to 7.46 (2H, m), 7.11-7.06 (2H, m), 6.73 (1H, s), 5.32 (2H, s), 3.95 (3H, s), 3.62 (3H, s), 2.51 (3H, s), 2.51 (3H, s) , 1.98 (3H, s) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-fluoro) -4-Methylpyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.49 (1 H, s), 7.57 (1H, s), 7.45-7.40 (2H, m), 7.29-7. 27 (1H, m), 6.72 (1H, s), 5.08 (2H, s), 3.65 (3H, s), 2.57 (3H, d) , J = 2.5 Hz), 2.51 (6 H, bs), 2.10 (3 H, s). 1- [2-({[1- (5-methoxypyridin-3-yl) -1 H-pyrazol-3-yl]. ] Oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.42 (1 H, d, J = 1.1 Hz), 8.16 (1H, d, J = 2.1 Hz), 7.71 (1 H, d, J = 2.7 Hz), 7.47 (1 H, t, J = 2.4 Hz), 7.42-7.38 (2 H, m), 7.28-7.24 (1 H, m), 5.86 (1H, d, J = 2.5 Hz), 5.34 (2H, s), 3.94 (3H, s), 3.65 (3H, s), 2.57 (3H, s) .; 1-(3-ethyl) -2-{[2,5-dimethyl-4- (1,5-dimethyl-1H-pyrazo) -3-yl) phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.49-7.43 (2H, m), 7.28-7.26 (2H, m), 6.70 (1H, s), 6.10 (1H, s), 5.05 (2H, s), 3.81 (3H, s), 3.61 (3H, s), 2.85 (2H, q, J = 7.6) Hz), 2.42 (3H, s), 2.31 (3H, s), 2.05 (3H, s), 1.28 (3H, t, J = 7.1 Hz) .; 1- (3-methoxy-2-{[2-] Methyl-4- (5-fluoro-1,4-dimethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.47 (1 H, t, J = 8.4 Hz), 7. 37 (1 H, s), 7. 35-7. 33 (1 H, m), 7.09-7. 07 (2 H, m), 6. 91 (1 H, d, J = 8.4 Hz), 5.29 (2H, s), 3.93 (3H, s), 3.73 (3H, s), 3.59 (3H, s), 2.08 (3H, s), 2.03 (3H, s).

1- [2-({[1- (2-Ethenyl-6-methoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.53 (1 H, d, J = 8.7 Hz), 7.40-7.38 (2 H, m), 7.28-7.25 (2 H, m), 6.71 (1H, d, J = 8.7 Hz), 6.61 (1 H, dd, J = 16.8, 10.4 Hz), 6.47 (1 H, dd, J = 16.8, 2.4 Hz), 5.78 (1 H, d, J = 2.5 Hz) , 5.47 (1H, dd, J = 10.4, 2.4 Hz), 5.29 (2H, s), 4.01 (3H, s), 3.60 (3H, s), 2.55 (3H, s) .; 1-(3-methyl) -2-{[3,6-dimethyl-5- (4,5-dihydro-1,3-oxazol-2-yl) pyridin-2-yl] oxymethyl} phenyl) -4-methyl-1,4- Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.76 (1 H, s), 7. 39-7. 35 (2 H, m), 7.25-7.2 2 (1 H, m), 5. 50 (2 H, s), 4. 35 (2H, t, J = 9.4 Hz), 4.05 ( 2H, t, J = 9.4 Hz), 3.66 (3H, s), 2.63 (3H, s), 2.58 (3H, s), 2.02 (3H, s) .; 1-(2- {[(4, 6) -Dimethoxypyrimidin-2-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.41-7.35 (2H, m), 7.26-7.24 (1H, m), 5.70 (1H, s), 5.40 (2H, s), 3.88 (6H, s), 3.67 (3H, s), 2.53 (3H, s). [2-({[1- (adamantan-1-ylmethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.37-7.33 (2 H, m), 7.22 (1 H, dd, J = 6.1, 3.2 Hz), 7.00 (1 H, d, J = 2.3 Hz), 5. 50 ( ¹ H, d , J = 2.3 Hz), 5.20 (2H, s), 3.67 (3H, s), 3.54 (2H, s), 2.53 (3H, s), 1.95 (3H, s), 1.68 (3H, d, J = 12.2 Hz), 1.57 (3 H, d, J = 11.3 Hz), 1. 44 (6 H, d, J = 2.5 Hz). 1- [2-({[1 (3 Etokishikishi-2-methoxy-4-yl)-1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.29 (1 H, d, J = 2.5 Hz), 7.88 (1 H, d, J = 5.7 Hz), 7.42-7.40 (3 H, m), 7.27-7. 25 (1 H, m) , 5.84 (1H, d, J = 2.7 Hz), 5.33 (2H, s), 4.04-4.00 (5H, m), 3.64 (3H, s), 2.56 (3H, s), 1.33 (3H, t, J = 7.1 Hz) .; 1- (3-ethyl-2-{[2-methyl-4- (5-fluoro-1,4-dimethyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4 -Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 to 7.36 (4H, m), 7.29 to 7.27 (1H, m), 6.89 (1H, d, J = 8.6 Hz), 5.08 (2H, s), 3.74 (3H, s), 3.59 (3H, s), 2.85 (2H, q, J = 7.6 Hz), 2.11 (3H, s), 2.09 (3H, s) , 1.28 (3H, t, J = 7.6 Hz) .; 1-(3- Chill -2 - {[4- (1-methoxyethyl) -2,5-dimethylphenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.44-7.39 (2H, m), 7.27-7.25 (1H, m), 7.10 (1H, s), 6.59 (1H, s), 5.00 (2H, s), 4.47 (1H, q, J = 6.4) Hz), 3.65 (3H, s), 3.21 (3H, s), 2.51 (3H, s), 2.28 (3H, s), 2.06 (3H, s), 1.37 (3H, d, J = 6.4 Hz). 1- (2-{[(1- {2-[(2-methylpropanoyl) oxy] -1,1-dimethylethyl} -1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl; ) -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38-7.33 (2H, m), 7.24-7.21 (2H, m), 5.50 (1H, d) , J = 2.3 Hz), 5.20 (2H, s), 4.17 (2H, s), 3.69 (3H, s), 2.52 (3H, s), 2.51-2.44 (1H, m), 1.51 (6H, s) , 1.08 (6 H, d, J = 7.1 Hz) .; 1- [2-({[1- (1-) Cyano-1-methylethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.36 (3 H, m), 7.24 (1 H, dd, J = 6.3, 2.9 Hz), 5. 64 (1 H, d, J = 2.5 Hz), 5.25 (2 H, s), 3. 69 (3 H, s) , 2.54 (3H, s), 1.88 (6H, s) .; 1- [2-({[1- (pyridin-4-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methyl] Phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.59 (2 H, dd, J = 4.7, 1.5 Hz), 7.80 (1 H, d, J = 2.7 Hz), 7.47 (2 H, dd, J = 4.6, 1.6 Hz), 7.43-7.37 (2 H, m), 7.29-7.25 (1 H, m), 5. 91 (1 H, d, J = 2.7 Hz), 5.36 (5 2H, s), 3.65 (3H, s), 2.57 (3H, s).

1- {2-[({1- [6- (1-methylethoxy) -2-methylpyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4 -Methyl-1,4-dihydrotetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46 (1 H, d, J = 8.4 Hz), 7.42-7.37 (2 H, m), 7.26-7.24 (2 H , m), 6.56 (1H, d, J = 8.6 Hz), 5.76 (1H, d, J = 2.5 Hz), 5.35-5.29 (1H, m), 5.27 (2H, s), 3.59 (3H, s) , 2.54 (3H, s), 2.31 (3H, s), 1.35 (6H, d, J = 6.1 Hz) .; 1- [3-cyclopropyl-2-({2-methyl-4- [1- (1) 2,2-Difluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 7.52 (2H, m), 7.47-1.41 (2H, m), 7.30-1.27 (2H, m), 6.91 (1H, d, J = 8.4 Hz), 6.52 (1 H, d, J = 2.3 Hz), 6.14 (1H, tt, J = 55.7, 4. 4 Hz), 5.29 (2H, s), 4.47 (2H, td, J = 13.4, 4.3 Hz), 3.60 (3H, s), 2.16-2.09 (1H, m), 2.12 (3H, s), 1.05- 0.97 (2H, m), 0.81-0.74 (2H, m) .; 1- [2-({[1- (3,4-difluoro-2-methoxyphenyl) -1H-pyrazol-3-yl] oxy} Methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.82 (1 H, d, J = 2.5 Hz), 7.39 (3 H, m), 7.26 (1H, m), 6.97 (1H, m), 5.80 (1H, d, J = 2.5 Hz), 5.31 (2H, s), 3.87 (3H, s), 3.62 (3H, s), 2.55 (3H, s) .; 1- [2-({[1- (2-cyanophenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.95 (1 H, d, J = 2.7 Hz), 7.72 (1 H, d, J = 7.8 Hz), 7.70-7.63 (2 H, m ), 7.43-7.38 (2H, m), 7.32 (1H, t, J = 7.3 Hz), 7.27-7.26 (1H, m), 5 .92 (1H, d, J = 2.7 Hz), 5.34 (2H, s), 3.66 (3H, s), 2.56 (3H, s) .; 1- (2-{[(1-ethyl-1H-pyrazole). -3-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-9-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2H, m), 7.23 (1 H, dd, J = 6.3, 2.7 Hz), 7. 10 (1 H, d, J = 2.0 Hz), 5.51 (1 H, d, J = 2.3 Hz), 5. 19 (2 H, s), 3. 95 (2 H, q , J = 7.3 Hz), 3.68 (3 H, s), 2.53 (3 H, s), 1. 39 (3 H, t, J = 7.4 Hz). 1- [2-({[1- (1-methyl-1H) -Pyrazole-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.76 (1 H, d, J = 2.5 Hz), 7.41-7.35 (2 H, m), 7.30 (1 H, d, J = 2.3 Hz), 7.24 (1 H, dd, J = 6.3, 3.1 Hz), 6.32 (1 H, d, J = 2.3 Hz), 5. 76 (1 H, d, J = 2.7 Hz), 5. 29 (2 H, s), 3. 86 (3 H, s), 3. 65 (3H, s), 2.54 (3H, s) .; 1- [3-fluoro-2-({2-methyl-4- [1- (2,2-difluoroethyl) -1H-pyrazol-3-yl Phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.54-7.48 (3 H, m), 7. 45 ( ¹ H, d, J = 2.5 Hz), 7.34-7.27 (2H, m), 6.88 (1 H, d, J = 8.4 Hz), 6.51 (1 H, d, J = 2.5 Hz), 6.13 (1 H, tt, J = 55.6, 4.4 Hz) , 5.30 (2H, s), 4.47 (2H, td, J = 13.5, 4.5 Hz), 3.59 (3H, s), 2.03 (3H, s) .; 1- {2-[({1- [2-] (Prop-1-yn-1-yl) -6-methoxypyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.99 (1 H, d, J = 2.7 Hz), 7.82 (1 H, d, J = 8.7 Hz), 7. 40-7. 39 (2 H, m), 7. 27 -7.25 (1H, m), 6.77 (1H, d, J = 8.7 Hz), 5.78 (1 H, d, J = 2.7 Hz), 5. 29 (2 H, s), 3. 97 (3 H, s), 3. 64 (3 H, s), 2.55 (3 H, s), 2.09 (3 H, s) 1- {3-Methyl-2-[(4-ethenyl-2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl 2; ₃ ) δ: 7.43-7.39 (2H, m), 7.27-7.26 (1H, m), 7.24 (1H, s), 6.85 (1H, dd, J = 17.4, 11.0 Hz), 6.61 (1H, s), 5.52 (1H, dd, J = 17.4, 1.4 Hz), 5.16 (1H, dd, J = 11.0, 1.4 Hz), 5.01 (2H, s), 3.64 (3H, s), 2.50 (3H, s), 2.31 (3H, s), 2.06 (3H, s) .; 1- {3-methyl-2-[(4-butoxy-2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.42-7.38 (2H, m), 7.26-7.23 (1H, m), 6.63 (1H, s), 6.59 (1H, s), 4.95 (4) 2H, s), 3.88 (2H, t, J = 6.3 Hz), 3.64 (3H, s), 2.51 (3H, s), 2.18 (3H, s), 2.04 (3H, s), 1.78-1.70 (2H) , m), 1.54-1.4 4 (2H, m), 0.97 (3H, t, J = 7.4 Hz) .;

1- [2-({[1- (1,1-dimethylpropyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole-5 -ON, ¹ H-NMR (CDCl ₃ ) δ: 7.37-7.33 (2 H, m), 7.24-4. 21 (1 H, m), 7. 19 (1 H, d, J = 2.3 Hz), 5. 47 (1 H, d, J = 2.3 Hz), 5.21 (2 H, s), 3. 67 (3 H, s), 2.53 (3 H, s), 1. 77 (2 H, q, J = 7.4 Hz), 1.43 (6 H, s), 0.59 (3 H, t) J = 7.3 Hz) .; 1- (3-Methyl-2-{[2,5-dimethyl-4- (5-methoxy-1-methyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46-7.41 (2H, m), 7.29-7.27 (1H, m), 6.94 (1H, s) , 6.72 (1H, s), 5.56 (1H, s), 5.05 (2H, s), 3.91 (3H, s), 3.67 (3H, s), 3.49 (3H, s), 2.53 (3H, s), 2.15 (3H, s), 2.07 (3H, s) .; 1- (3-methyl-2- { 2,5-dimethyl-4- (1,5-dimethyl--1H- pyrazole-3 -yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydro-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.44-7.39 (2H, m), 7.31-7.26 (2H, m), 6.68 (1H, s), 6.10 (1H, s), 5.04 (2H, s), 3.81 (3H, s) , 3.64 (3H, s), 2.51 (3H, s), 2.41 (3H, s), 2.30 (3H, s), 2.06 (3H, s) .; 1- [3-methyl-2-({2, 2, 3 5-Dimethyl-4- [1- (prop-2-en-1-yl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one , ¹ H-NMR (CDCl ₃ ) δ: 7.64 (1H, d, J = 2.3 Hz), 7.44-7.39 (2H, m), 7.30-7.26 (2H, m), 6.70 (1H, s), 6.38 (6) 1H, d, J = 2.5 Hz), 5.05 (2H, s), 4.98 (2H, d, J = 2.5 Hz), 3.64 (3H, s), 2.55-2.49 (1H, m), 2.51 (3H, s) ), 2.42 (3H, s), 2.07 (3H, s) .; 1- [3-methoxy-2-({2- Chill-4- [5-fluoro-4- (difluoromethyl) -1-methyl -1H- pyrazole-3 -yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydro-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.47 (1 H, t, J = 8.2 Hz), 7. 35-7. 32 (2 H, m), 7. 10-7. 07 (2 H, m), 6. 92 (1 H, d, J = 8.2 Hz) , 6.61 (1H, t, J = 54.3 Hz), 5.30 (2H, s), 3.94 (3H, s), 3.78 (3H, s), 3.60 (3H, s), 2.03 (3H, s) .; 1 -(3-Chloro-2-{[2,5-dimethyl-4- (cyclopropanecarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR ( CDCl ₃ ) δ: 7.63 (1 H, d, J = 8.0 Hz), 7.56 (1 H, s), 7.51-7.46 (1 H, m), 7.41 (1 H, d, J = 8.0 Hz), 6.69 (1 H, s) ), 5.35 (2H, s), 3.62 (3H, s), 2.48 (3H, s), 2.44-2.40 (1H, m), 2.03 (3H, s), 1.21-1.17 (2H, m), 1.00- 0.95 (2H, m) .; 1- (3-methyl-2-{[2-] Methyl-4- (5-fluoro-4-methylpyrimidin-2-yl) phenoxy} methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.44 (1 H, t, J = 1.5 Hz), 8. 16 (1 H, d, J = 8.9 Hz), 8.13 (1 H, s), 7.46-7.40 (2 H, m), 7. 29 (1 H, d, J = 6.6 Hz) ), 6.92 (1H, d, J = 8.5 Hz), 5.11 (2H, s), 3.63 (3H, s), 2.57 (3H, d, J = 2.3 Hz), 2.52 (3H, s), 2.16 (3H) , s) .; 1- (3-ethyl-2-{[2,5-dimethyl-4- (5-fluoro-4-methylpyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.48 (1 H, d, J = 1.6 Hz), 7.55 (1 H, s), 7.49-7.43 (2 H, m), 7.28 (7 1H, dd, J = 7.1, 2.2 Hz), 6.73 (1 H, s), 5.08 (2 H, s), 3.61 (3 H, s), 2. 84 (2 H, q, J = 7.6 Hz), 2.57 (3 H, d , J = 2.5 Hz), 2.51 (3 H, s), 2.07 (3 H, s), 1.27 (3 H, t, J = 7.6 Hz) .; 1-1 [2-({[1- (4-Chloro-2-fluorophenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole-5 -ON, ¹ H-NMR (CDCl ₃ ) δ: 7.81-7.77 (2H, m), 7.43-7.38 (2H, m), 7.26 (1H, m), 7.21 (2H, m), 5.84 (1H, d) , J = 2.7 Hz), 5.31 (2H, s), 3.65 (3H, s), 2.55 (3H, s) .; 1- (3-methyl-2-{[4- (2-methylpropoxy) -2]. 5-Dimethylphenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.23 (1H , m), 6.64 (1H, s), 6.58 (1H, s), 4.95 (2H, s), 3.65-3.64 (5H, m), 2.51 (3H, s), 2.19 (3H, s), 2.10- 2.02 (4H, m), 1.02 (6H, d, J = 6.6 Hz) .;

1- (3-Methyl-2-{[2,5-dimethyl-4- (4-ethyl-4,5-dihydro-1,3-oxazol-2-yl) phenoxy] methyl} phenyl) -4-methyl ^-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.56 (1 H, s), 7.44-7. 39 (2 H, m), 7. 29-7. 26 (1 H, m), 6. 66 (1 H , s), 5.05 (2H, s), 4.40-4.36 (1H, m), 4.26-4.19 (1H, m), 4.00-3.96 (1H, m), 3.63 (3H, s), 2.55 (3H, s) ), 2.49 (3H, s), 2.04 (3H, s), 1.77-1.70 (1H, m), 1.64-1.57 (4H, m), 0.99 (3H, t, J = 7.4 Hz). 3-Cyclopropyl-2-{[2,5-dimethyl-4- (4,4-dimethyl-4,5-dihydro-1,3-oxazol-2-yl) phenoxy] methyl} phenyl) -4-methyl ^-1 , 4-dihydrotetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.53 (1 H, s), 7.43 (1 H, t, J = 7.9 Hz), 7.28-7.26 (2 H, m), 6.69 (1H, s), 5.27 (2H, s), 4.03 (2H, s), 3.61 (3H, s), 2.53 (3H, s), 2.13-2.06 (1H, m), 2.02 (3H, s), 1.36 (6H, s), 1.01-0.96 (2H, s) m), 0.77-0.73 (2H, m) .; 1- (3-chloro-2-{[2-methyl-4- (5-fluoro-1,4-dimethyl-1H-pyrazol-3-yl) phenoxy] Methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.61 (1 H, dd, J = 8.0, 1.4 Hz), 7.47 (1 H, t , J = 8.0 Hz), 7.41-7.40 (2H, m), 7.37-7.35 (1 H, m), 6.88 (1 H, d, J = 8.6 Hz), 5.34 (2 H, s), 3.74 (3 H, s) , 3.59 (3H, s), 2.08 (3H, s), 2.06 (3H, s) .; 1- (3-methyl-2-{[2-methyl-4- (4-bromo-1-methyl-1H) -Pyrazol-5-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.51 (1 H, s), 7.47-7.42 ( 2H, m), 7.29 (1 H, dd, J = 6.9, 2.2 Hz), 7.18 (1 H, dd, J = 8.4, 2.3 Hz), 7.14 (1H, s), 6.95 (1H, d, J = 8.4 Hz), 5.09 (2H, s), 3.80 (3H, s), 3.65 (3H, s), 2.54 ( 3 H, s), 2.15 (3 H, s) .; 1- (3-Methyl-2-{[2,5-dimethyl-4- (3,5-difluoropyridin-2-yl) phenoxy] methyl} phenyl) -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.42 (1 H, d, J = 2.1 Hz), 7.45-7.40 (2 H, m), 7.29-7.25 (2H, m), 7.08 (1H, s), 6.75 (1H, s), 5.07 (2H, s), 3.65 (3H, s), 2.52 (3H, s), 2.20 (3H, s), 2.08 ( 3H, s) .; 1- {3-Methyl-2-[(4-ethyl-2,5-dimethylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H -NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.26-7.24 (1H, m), 6.88 (1H, s), 6.63 (1H, s), 4.98 (2H, s), 3.65 (3H) , s), 2.55-2.49 (5H, m), 2.26 (3H, s), 2.04 (3H, s), 1.15 (3H, t, J = 7.6 Hz) .; 1- (3-methoxy) -2-{[2,5-dimethyl-4- (4,5-dihydro-1,3-oxazol-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 7.54 (1H, s), 7.47 (1H, t, J = 8.3 Hz), 7.10-7.06 (2H, m), 6.72 (1H, s), 5.29 (2H , s), 4.33 (2H, t, J = 9.4 Hz), 4.07-4.02 (2H, m), 3.94 (3H, s), 3.59 (3H, s), 2.54 (3H, s), 1.94 (3H, s) s) .; 1- {2-[({1- [2- (triisopropylsilyl) ethynyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.41-7.37 (3 H, m), 7. 25 ( ¹ H, dd, J = 6.9, 2.3 Hz), 5.69 (1 H, d, J = 2.5 Hz), 5.25 (2H, s), 3.69 (3H, s), 2.51 (3H, s), 1.13-1.12 (21 H, m) .; 1- [2-({[1- (1, 1-) Dimethylethyl) -5-amino-1 H-Pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (DMSO-D6) δ: 7.47-7.44 (2H , m), 7.32-7.28 (1H, m), 4.98 (2H, s), 4.84 (2H, s), 4.70 (1H, s), 3.59 (3H, s), 2.46 (3H, s), 1.42 (1) 9 H, s) .; 1- [2-({[1- (1,1-dimethyl-2-propynyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl -1,4-dihydrotetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.55 (1 H, d, J = 2.5 Hz), 7.38-7.34 (2 H, m), 7.23 (1 H, dd, J = 6.5, 2.9 Hz), 5.53 (1 H, d, J = 2.5 Hz), 5.22 (2 H, s), 3. 67 (3 H, s), 2.55 (1 H, s), 2.53 (3 H, s), 1. 74 (6 H) , s) .;

1- {2-[({1- [2- (difluoromethoxy) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4 -Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.22 (1 H, d, J = 7.9 Hz), 8.05 (1 H, d, J = 2.7 Hz), 8.02 (1 H, d, J = 4.8 Hz), 7.76-7.39 (3H, m), 7.27-7.26 (1 H, m), 7.23 (1 H, dd, J = 7.9, 5.0 Hz), 5.86 (1 H, d, J = 2.5 Hz), 5.32 (5 2H, s), 3.65 (3H, s), 2.55 (3H, s) .; 1- [3-methyl-2-({2,5-dimethyl-4- [1- (2,2-difluoroethyl) -1H-Pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.47 (1 H, d, J = 2.3) Hz), 7.44-7.39 (2H, m), 7.31-7.27 (2H, m), 6.71 (1H, s), 6.39 (1H, d, J = 2.3 Hz), 6.14 (1 H, tt, J = 55.6, 4.4 Hz), 5.05 (2H, s), 4.48 ( 2H, td, J = 13.4, 4.4 Hz), 3.65 (3H, s), 2.51 (3H, s), 2.41 (3H, s), 2.07 (3H, s) .; 1-[2- ({[1 [ -(2-cyano-6-methoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.94 (1 H, d, J = 9.1 Hz), 7. 91 (1 H, d, J = 2.5 Hz), 7. 40 (2 H, m), 7. 26-7. 25 (1 H, m), 7.05 (1H, d, J = 9.1 Hz), 5.91 (1H, d, J = 2.5 Hz), 5.31 (2H, s), 3.99 (3H, s), 3.67 (3H, s), 2.55 (3H, s) 1- [3-Methyl-2-({2,5-dimethyl-4- [rel- (4R, 5S) -4,5-dimethyl-4,5-dihydro-1,3-oxazole-2). -Yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.54 (1 H, s), 7. 45-7. 39 (2 H, m) , 7.29-7.26 (1H, m), 6 .65 (1H, s), 5.05 (2H, s), 4.81-4.74 (1H, m), 4.34-4.27 (1H, m), 3.63 (3H, s), 2.54 (3H, s), 2.49 (3H) , s), 2.04 (3H, s), 1.33 (3H, d, J = 6.6 Hz), 1.22 (3 H, d, J = 7.0 Hz). 1- [2-({[1- (2-methoxy) -1,1-Dimethylethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ δ: 7.37-7.34 (2H, m), 7.24 (1 H, d, J = 2.3 Hz), 7.22 (1 H, dd, J = 6.2, 3.2 Hz), 5.50 (1 H, d, J = 2.5 Hz), 5.21 (2H, s), 3.67 (3H, s), 3.47 (2H, s), 3.17 (3H, s), 2.53 (3H, s), 1.46 (6H, s) .; 1- {2-[( {1- [4-Chloro-2- (trifluoromethyl) phenyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 7.74 (1 H, d, J = 2.3 Hz), 7.6 1 (1 H, dd, J = 8.5, 2.3 Hz), 7.48 (1 H, d, J = 8.5 Hz), 7.42-7.37 (3 H, m), 7.26-7.25 (1 H, m), 5.83 (1 H, d, J = 2.5 Hz), 5.27 (2H, s), 3.62 (3H, s), 2.53 (3H, s) .; 1- (2-{[(1-propyl-1H-pyrazol-3-yl) oxy] Methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-8-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39-7.34 (2H, m), 7.23 (1 H, dd, J = 6.3, 2.7 Hz), 7.09 (1 H, d, J = 2.3 Hz), 5.51 (1 H, d, J = 2.3 Hz), 5.19 (2 H, s), 3.84 (2 H, t, J = 7.0 Hz), 3.68 (3H, s), 2.53 (3H, s), 1.81-1.77 (2H, m), 0.87 (3H, t, J = 7.5 Hz) .; 1- [2-({[1- (5-methoxy) Pyridin-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ : 8.21 (1 H, d, J = 2.7 Hz), 8.02 (1 H, d, J = 2.9 Hz), 7. 70 (1 H, d, J = 9.1 Hz), 7.42-7 .38 (2H, m), 7.32 (1 H, dd, J = 8.9, 3.1 Hz), 7.26-7.25 (1 H, m), 5.81 (1 H, d, J = 2.5 Hz), 5.32 (2 H, s), 3.88 (3H, s), 3.64 (3H, s), 2.56 (3H, s) .; 1- [2-({[1- (2-methoxythiazol-5-yl) -1 H-pyrazol-3-yl] ] Oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.40-7.38 (3H, m), 7.24 (1H, 1H, dd, J = 6.5, 2.6 Hz), 7.01 (1 H, s), 5. 75 (1 H, d, J = 2.5 Hz), 5. 26 (2 H, s), 4.07 (3 H, s), 3. 67 (3 H, s), 2.54 (3H, s) .; 1- [3-Methyl-2-({2-methyl-4- [3- (difluoromethyl) -5-methyl-1H-pyrazol-1-yl] phenoxy} methyl) phenyl )]-4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46-7.41 (2H, m), 7.29 (1 H, dd, J = 7.2, 1.9 Hz) , 7.18-7.14 (2H, m), 6.89 (1 H, d, J = 8.2 Hz), 6.68 (1H, t, J = 55.2 Hz), 6.39 (1H, s), 5.08 (2H, s), 3.65 (3H, s), 2.52 (3H, s), 2.30 (3H, s), 2.13 (3H) , s) .;

1- [3-Methyl-2-({2,5-dimethyl-4- [1- (1-methylethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-4.39 (3 H, m), 7.31 (1 H, s), 7. 28-7. 27 (1 H, m), 6. 70 (1 H, s) , 6.30 (1H, d, J = 2.3 Hz), 5.04 (2H, s), 4.57-4.50 (1H, m), 3.65 (3H, s), 2.51 (3H, s), 2.43 (3H, s), 2.07 (3H, s), 1.54 (6H, d, J = 6.6 Hz) .; 1- {3-methyl-2-[(2,5-dimethyl-4-butanoylphenoxy) methyl] phenyl} -4- 4 Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.48 (1 H, s), 7.46-7.38 (2 H, m), 7. 28 (1 H, dd, J = 7.3, 2.1 Hz), 6.66 (1H, s), 5.07 (2H, s), 3.64 (3H, s), 2.83 (2H, t, J = 7.3 Hz), 2.51 (3H, s), 2.50 (3H, s), 2.08 (3 H, s), 1.73-1. 69 (2 H, m), 0.97 (3 H, t, J = 7.4 Hz) .; 1- {3-methyl- - [(2,5-dimethyl-4-acetoxy) methyl] phenyl} _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.53 (1H, s ), 7.46-7.39 (2H, m), 7.28 (1H, dd, J = 7.4, 1.9 Hz), 6.66 (1H, s), 5.08 (2H, s), 3.64 (3H, s), 2.54 (3H, 5) s), 2.53 (3H, s), 2.50 (3H, s), 2.08 (3H, s) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (5-ethyl pyrimidine)- 2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.63 (2H, s), 7.59 (1 H, s), 7.44-7.38 (2H, m), 7.28-7.26 (1H, m), 6.72 (1H, s), 5.08 (2H, s), 3.64 (3H, s), 2.67 (2H, q, J = 7.6 Hz) , 2.53 (3H, s), 2.51 (3H, s), 2.09 (3H, s), 1.31 (3H, t, J = 7.7 Hz). 1- (3-methoxy-2-{[2,5- Dimethyl-4- (5-fluoro-4-methylpyrimidin-2-yl) group Phenoxy] methyl} phenyl) _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 8.47 (1H, d, J = 1.6 Hz), 7.51 (1H, s) , 7.46 (1H, t, J = 8.2 Hz), 7.10-7.06 (2H, m), 6.77 (1H, s), 5.30 (2H, s), 3.94 (3H, s), 3.60 (3H, s), 2.56 (3 H, d, J = 2.5 Hz), 2.48 (3 H, s), 1.99 (3 H, s) .; 1- [2-({[1- (2,4-dichlorophenyl) -1 H-pyrazole-3] -Yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.70 (1 H, d, J = 2.5 Hz) , 7.50 (2H, m), 7.43-7.38 (2H, m), 7.33 (1H, dd, J = 8.6, 2.3 Hz), 7.26 (1 H, m), 5.83 (1 H, d, J = 2.5 Hz), 5.31 (2H, s), 3.63 (3H, s), 2.55 (3H, s) .; 1- [2-({[1- (2-chloro-6-methoxypyridin-3-yl) -1H-pyrazole] -3-yl] oxy} methyl) -3-methylphenyl]- - _{^{methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.76 (1H, d, J = 8.6 Hz), 7.62 (1H, d, J = 2.7 Hz), 7.41- 7.39 (2H, m), 7.25 (1 H, t, J = 4.1 Hz), 6.77 (1 H, d, J = 8.6 Hz), 5.81 (1 H, d, J = 2.7 Hz), 5.28 (2 H, s), 3.98 (3H, s), 3.64 (3H, s), 2.55 (3H, s) .; 1- [2-({[1- (4-methoxypyridin-3-yl) -1H-pyrazol-3-yl] ] Oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.83 (1 H, s), 8. 38 (1 H, d, J = 5.7 Hz), 7.84 (1 H, d, J = 2.5 Hz), 7. 40-7. 37 (2 H, m), 7. 27-7. 23 (1 H, m), 6. 92 (1 H, d, J = 5.7 Hz), 5. 80 (5 1H, d, J = 2.5 Hz), 5.34 (2H, s), 3.95 (3H, s), 3.65 (3H, s), 2.57 (3H, s) .; 1- [2-({[1- (1) 2-hydroxy-1,1-dimethylethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl ¹ H-NMR (CDCl ₃ ) δ: 7.40-7.35 (2H, m), 7.25-7.23 (2H, m), 5.53 (1H, d) , J = 2.5 Hz), 5.21 (2 H, s), 3.67-3.66 (5 H, m), 3.46 (1 H, t, J = 6.8 Hz), 2.53 (3 H, s), 1. 45 (6 H, s). 1- (2-{[(1- {1,1-dimethyl-2-[(1,1-dimethylethoxy) imino] ethyl} -1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl ) -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46 (1 H, s), 7.38-7.35 (2 H, m), 7.24-7. 22 (1 H, m) ), 7.19 (1H, d, J = 2.5 Hz), 5.53 (1H, d, J = 2.5 Hz), 5.21 (2H, s), 3.68 (3H, s), 2.53 (3H, s), 1.64 (6H) , s), 1.28 (9H, s) .;

1- [2-({[1- (furan-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CDCl ₃ ) δ: 7.68 (1 H, m), 7. 40-7. 38 (4 H, m), 7.2 4 (1 H, dd, J = 6.2, 3.0 Hz), 6.61 (1 H, m), 5.73 (1H, d, J = 2.5 Hz), 5.28 (2H, s), 3.65 (3H, s), 2.55 (3H, s) .; 1- [2-({[1- (2,3-dimethoxypyridine). -4-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.24 (1 H, d, J = 2.7 Hz), 7. 89 (1 H, d, J = 5.7 Hz), 7.43-7. 39 (3 H, m), 7. 26 (1 H, m), 5. 86 (1 H, d, J = 2.7 Hz) ), 5.34 (2H, s), 4.04 (3H, s), 3.80 (3H, s), 3.64 (3H, s), 2.56 (3H, s) .; 1- [2-({[1- (1) -Methyl-1H-pyrazol-5-yl) -1H- Razoru 3-yl] oxy} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.46 (1H, d, J = 2.1 Hz), 7.42-7.37 (2H, m), 7.36 (1H, d, J = 2.5 Hz), 7.26-7.24 (1H, m), 6.19 (1 H, d, J = 1.8 Hz), 5.81 (1H, 1H, m) d, J = 2.5 Hz), 5.31 (2H, s), 3.81 (3H, s), 3.59 (3H, s), 2.55 (3H, s) .; 1- (2-{[2-methyl-4-] (5-Fluoropyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.59 (2H, s), 8.16 -8.13 (2H, m), 7.72 (1 H, d, J = 7.3 Hz), 7.56-7.49 (3 H, m), 6.89 (1 H, d, J = 8.7 Hz), 5.24 (2 H, s), 3.67 (3 3H, s), 2.26 (3H, s) .; 1- (3-methoxy-2-{[2,5-dimethyl-4- (3,4-dimethyl-1H-pyrazol-1-yl) phenoxy] methyl } Phenyl) -4-methyl _{^{1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.47 (1H, t, J = 8.2 Hz), 7.20 (1H, s), 7.08 (2H, dd, J = 8.2, 4.5 Hz), 6.99 (1H, s), 6.74 (1H, s), 5.26 (2H, s), 3.94 (3H, s), 3.62 (3H, s), 2.25 (3H, s), 2.15 (3H, s) s), 2.05 (3H, s), 1.94 (3H, s) .; 1- [3-chloro-2-({2-methyl-4- [1- (2,2-difluoroethyl) -1H-pyrazole] -3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.62 (1 H, d, J = 8.0 Hz), 7.54 -7.39 (5H, m), 6.87 (1H, d, J = 8.2 Hz), 6.51 (1H, dd, J = 2.4, 1.3 Hz), 6.14 (1 H, tt, J = 56.0, 4.2 Hz), 5.35 ( 2H, s), 4.47 (2H, td, J = 13.3, 4.3 Hz), 3.59 (3H, s), 2.07 (3H, s) .; 1- {3-methoxy-2-[(2,5-dimethyl] -4-propanoylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetra _{^{Lumpur-5-, 1 H-NMR (CDCl 3}} ) δ: 7.50-7.44 (2H, m), 7.10-7.06 (2H, m), 6.73 (1H, s), 5.31 (2H, s), 3.95 (3H, s), 3.61 (3H, s), 2.87 (2H, q, J = 7.3 Hz), 2.50 (3H, s), 1.98 (3H, s), 1.16 (3H, t, J = 7.3 Hz) 1- [2-({[5- (2,6-dimethoxypyridin-3-yl) thiazol-2-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.60 (1 H, d, J = 8.2 Hz), 7. 40 (2 H, d, J = 7.5 Hz), 7.33 (1 H, s), 7.28-7.26 (1H, m), 6.32 (1H, d, J = 8.2 Hz), 5.47 (2H, s), 4.00 (3H, s), 3.91 (3H, s), 3.69 (3H, s), 2.53 (3H, s) s) .; 1- (3-methyl-2-{[2,5-dimethyl-4- (1-propyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4 -Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.37 (3H, m), 7.3 1 (1H, s), 7.29-7.26 (1H, m), 6.70 (1H, s), 6.30 (1H, d, J = 2.3 Hz), 5.05 (2H, s), 4.15-4.09 (2H, m) , 3.64 (3H, s), 2.51 (3H, s), 2.42 (3H, s), 2.07 (3H, s), 1.97-1.88 (2H, m), 0.94 (3H, t, J = 7.4 Hz). 1- [2-({[1- (4-chloro-2-methylphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro; Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.41-7.36 (2H, m), 7.31 (1H, m), 7.27 (1H, m), 7.25-7.22 (3H, m), 5.76 ( 1H, d, J = 2.5 Hz), 5.28 (2H, s), 3.57 (3H, s), 2.54 (3H, s), 2.24 (3H, s).

1- [2-({[1- (6-methoxy-pyridin-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.27 (1 H, d, J = 2.7 Hz), 7.65 (1 H, t, J = 7.9 Hz), 7.42-7.38 (2 H, m), 7.29 (1H, d, J = 7.8 Hz), 7.26-7.25 (1 H, m), 6.54 (1 H, d, J = 8.2 Hz), 5.81 (1 H, d, J = 2.5 Hz), 5.34 (2 H, s) , 3.94 (3H, s), 3.64 (3H, s), 2.56 (3H, s) .; 1- (3-Cyclopropyl-2-{[2,5-dimethyl-4- (1,5-dimethyl-) ¹ H-Pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.44-4.40 (1 H, m), 7.31 -7.27 (2H, m), 7.25-7.25 (1H, m), 6.73 (1H, s), 6.10 (1H, s), 5.26 (2H, s), 3.81 (3H, s), 3.62 (3H, s) ), 2.42 (3H, s), 2.31 (3H, s), 2.17-2.10 (1H, m), 2.05 (3H, s), 1.01-0.97 (2H, m), 0.78-0.74 (2H, m) .; 1- {3-cyclopropyl-2-[(2,5-dimethyl-4-propanoylphenoxy) methyl Phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 (1 H, s), 7.47-7.42 (1 H, m), 7.29-7.25 (2 H) , m), 6.71 (1H, s), 5.30 (2H, s), 3.62 (3H, s), 2.89 (2H, q, J = 7.3 Hz), 2.53 (3H, s), 2.15-2.08 (1H, 1) m), 2.07 (3H, s), 1.17 (3H, t, J = 7.3 Hz), 1.04-0.97 (2H, m), 0.80-0.74 (2H, m) .; 1-(3- {[2- Methyl-4- (5-chloro-1,4-dimethyl-1H-pyrazol-3-yl) phenoxy] methyl} pyridin-2-yl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.64 (1 H, d, J = 4.5 Hz), 8. 16 (1 H, d, J = 7.9 Hz), 7.53 (1 H, dd, J = 7.1, 5.3 Hz), 7.47 (1 H , s), 7.36 (1 H, d, J = 8.4 Hz), 6. 84 (1 H, d, J = 8.6 Hz), 5. 24 (2 H, s), 3.86 (3H, s), 3.72 (3H, s), 2.28 (3H, s), 2.14 (3H, s) .; 1- [3-ethyl-2-({2-methyl-4- [1- (2) , 2-Difluoroethyl) -1H-pyrazol-3-yl] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.55-7.44 (5H, m), 7.28 (1 H, dd, J = 7.1, 2.1 Hz), 6.88 (1 H, d, J = 8.2 Hz), 6.52 (1 H, d, J = 2.3 Hz), 6.14 (1 H, tt, J = 55.6, 4.5 Hz), 5.08 (2 H, s), 4. 48 (2 H, td, J = 13.4, 4.4 Hz), 3.58 (3 H, s), 2. 85 (2 H, q, J = 7.6 Hz), 2.12 (2. 3H, s), 1.28 (3H, t, J = 7.8 Hz) .; 1- (3-Methyl-2-{[2-methyl-4- (5-fluoro-1,4-dimethyl-1H-pyrazole-) 3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.36 (4H, m), 7.29-7.27 (1H , m), 6.88 (1 H, d, J = 8.4 Hz), 5.06 (2H, s), 3.74 (3H, s), 3.63 (3H, s), 2.51 (3H, s), 2.12 (3H, s), 2.09 (3H, s) .; 1- [2- ({[ 5- (Pyridin-2-yl) thiazol-2-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ : 8.49 (1H, m), 7.64 (1H, ddd, J = 8.6, 6.9, 1.1 Hz), 7.52 (2H, m), 7.42 (2H, m), 7.28 (1 H, dd, J = 7.4, 1.7 Hz , 7.11 (1H, ddd, J = 7.4, 4.9, 1.1 Hz), 5.51 (2H, s), 3.71 (3H, s), 2.55 (3H, s) .; 1- [2- ({[1- (2-fluoro-6-methoxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.10 (1H, dd, J = 9.7, 8.6 Hz), 7.72-7.70 (1H, m), 7.40-7.39 (2H, m), 7.26-7.25 (1H, m), 6.72 (1 H, d, J = 8.7 Hz), 5.82 (1 H, d, J = 2.5 Hz), 5. 29 (2 H, s), 3.94 (3H, s), 3.65 (3H, s), 2.55 (3H, s) .; 1- (3-methyl-2-{[4- (isopropoxymethyl) -2,5-dimethylphenoxy] methyl} phenyl ) -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.43-7.38 (2H, m), 7.27-7.25 (1H, m), 7.03 (1H, s) ), 6.64 (1H, s), 4.99 (2H, s), 4.37 (2H, s), 3.69-3.63 (4H, m), 2.49 (3H, s), 2.31 (3H, s), 2.03 (3H, s) s), 1.20 (6H, d, J = 6.1 Hz) .; 1- [2-({[1- (3-formylphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl ¹ H-NMR (CDCl ₃ ) δ: 10.08 (1 H, s), 8.06 (1 H, s), 7.87 (1 H, d, J = 8.2) Hz), 7.77 (1 H, d, J = 2.5 Hz), 7.71 (1 H, d, J = 7.6 Hz), 7.59 (1 H, t, J = 7.6 Hz), 7.42-7.40 (2 H, m), 7.28- 7.25 (1H, m), 5.87 (1H, d, J = 2.5 Hz), 5.35 (2H, s), 3.65 (3H, s), 2.57 (3H, s).

1- [2-({[1- (2-methoxycyclohexyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one , ¹ H-NMR (CDCl ₃ ) δ: 7.36-7.33 (2H, m), 7.22 (1 H, dd, J = 6.1, 3.3 Hz), 7.14 (1 H, d, J = 2.3 Hz), 5.49 (1 H, 5 d, J = 2.3 Hz), 5. 24 (1 H, d, J = 12. 1 Hz), 5. 19 (1 H, d, J = 12. 1 Hz), 3. 67 (3 H, s), 3.58-3. 54 (1 H, m), 3.35 3.32 (1H, m), 2.89 (3H, s), 2.53 (3H, s), 2.17-2.14 (1H, m), 1.95-1.88 (2H, m), 1.81-1. 78 (2H, m), 1.42- 1.16 (3H, m) .; 1- (2-{[(1- {2-[(2,2-dimethylpropanoyl) oxy] -1,1-dimethylethyl} -1H-pyrazol-3-yl) Oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.37-7.33 (2H, m), 7.23-7.21 (2H , m), 5.50 (1 H, d, J = 2. 5 Hz), 5.19 (2H, s), 4.14 (2H, s), 3.69 (3H, s), 2.52 (3H, s), 1.51 (6H, s), 1.10 (9H, s). 2-{[(1-methyl-1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-8-one, ¹ H-NMR (CDCl ₃ δ: 7.40-7.35 (2H, m), 7.23 (1 H, dd, J = 6.5, 2.6 Hz), 7.06 (1 H, d, J = 2.3 Hz), 5.51 (1 H, d, J = 2.3 Hz), 5.18 (2H, s), 3.69 (3H, s), 3.68 (3H, s), 2.53 (3H, s) .; 1- [2-({[1- (1-methyl-1H-pyrazole-4-)] Yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.60 (1 H , s), 7.58 (1 H, s), 7. 40-7. 37 (3 H, m), 7.24 (1 H, dd, J = 6.5, 2.9 Hz), 5.71 (1 H, d, J = 2.5 Hz), 5.26 (2 H, 5 H) s), 3.92 (3H, s), 3.64 (3H, s), 2.54 (3H, s) .; 1- [2-({[1- (5-) Chloro-6-methylpyridin-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.29 (1 H, d, J = 2.7 Hz), 7.66 (1 H, d, J = 8.6 Hz), 7.54 (1 H, d, J = 8.6 Hz), 7.42-7.38 (2 H, m) , 7.28-7.24 (1 H, m), 5.82 (1 H, d, J = 2.7 Hz), 5.32 (2 H, s), 3. 65 (3 H, s), 2.57 (3 H, s), 2.55 (3 H, s). 1- {2-[({1- [2- (prop-2-en-1-yl) -6-methoxypyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3; -Methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 (1 H, d, J = 8.5 Hz), 7.40-7.38 (2 H, m) , 7.27-7.24 (2H, m), 6.65 (1H, d, J = 8.5 Hz), 6.06-5.96 (1H, m), 5. 76 (1 H, d, J = 2.5 Hz), 5.27 (2H, s), 5.00 (2H, dd, J = 19.5, 13.7 Hz), 3.96 (3H, s), 3.59 (3H, s) ), 3.38 (2H, d, J = 6.4 Hz), 2.55 (3H, s) .; 1- (3-methoxy-2-{[2,5-dimethyl-4- (1H-pyrazol-1-yl)]. Phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.67 (1 H, d, J = 1.6 Hz), 7.52-7.46 (2 H, m), 7.09 (2H, dd, J = 8.0, 6.4 Hz), 7.02 (1 H, s), 6.78 (1 H, s), 6.39 (1 H, t, J = 2.1 Hz), 5.29 (2 H, s), 3.95 (3H, s), 3.63 (3H, s), 2.13 (3H, s), 1.97 (3H, s) .; 1- {3-ethyl-2-[(2, 5-dimethyl-4-propanoyl] Phenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.52 to 7.43 (3 H, m), 7.28 (1 H, dd, J = 7.2 , 1.9 Hz), 6.68 (1 H, s), 5.09 (2 H, s), 3. 60 (3 H, s), 2. 89 (2 H, q, J = 7.6 Hz), 2. 84 (2 H, q, J = 7.6 Hz), 2.53 (3H, s), 2.06 (3H, s), 1.28 (3H, t, J = 7.6 Hz), 1.17 (3 H, t, J = 7.6 Hz) .; 1- [2- {[1- (2-methoxy-pyrimidin-4-yl)-1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.42 (1 H, d, J = 6.0 Hz), 8. 37 (1 H, d, J = 2.7 Hz), 7.43-7.39 (2 H, m), 7.26-7.26 (1 H, m) , 6.54 (1H, d, J = 5.7 Hz), 5.94 (1H, d, J = 2.7 Hz), 5.37 (2H, s), 4.05 (3H, s), 3.66 (3H, s), 2.54 (3H, s) s) .; 1- (3-methoxy-2-{[2,5-dimethyl-4- (1-methyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4-methyl-1,4 -Dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.46 (1 H, t, J = 8.2 Hz), 7. 35 (1 H, d, J = 2.1 Hz), 7.27 (1 H, s), 7.08 (2H, dd, J = 8.1, 4.7 Hz), 6.75 (1 H, s), 6.30 (1 H, d, J = 2.1 Hz), 5. 27 (2 H, s), 3. 93 (6 H, bs), 3.59 (3 H, s) s), 2.40 (3H, s), 1.97 (3H, s) .;

1- {2-[({1- [2- (trifluoromethyl) pyridin-3-yl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1, 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.92 (1 H, d, J = 2.5 Hz), 8.04 (1 H, dd, J = 8.6, 2.6 Hz), 7.79 (1 H, d , J = 2.7 Hz), 7.73 (1 H, d, J = 8.7 Hz), 7.42-7.39 (2 H, m), 7. 29-7. 25 (1 H, m), 5. 93 (1 H, d, J = 2.7 Hz), 5.36 (2H, s), 3.67 (3H, s), 2.57 (3H, s) .; 1- [2-({[1- (2-methoxypyrazin-3-yl) -1H-pyrazol-3-yl]; Oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.28 (1 H, d, J = 2.9 Hz), 8.11 ( 1H, d, J = 2.7 Hz), 7. 98 (1 H, d, J = 2.7 Hz), 7.43-7. 38 (2 H, m), 7. 26-7. 25 (1 H, m), 5. 93 (1 H, d, J = 2.7 Hz) ), 5.36 (2H, s), 4.11 (3H, s), 3.66 (3H, s), 2.5 3 (3 H, s) .; 1- [3-Methyl-2-({2-methyl-4- [4-bromo-1- (2,2-difluoroethyl) -1 H-pyrazol-3-yl] phenoxy } Methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.65 (1 H, d, J = 8.6 Hz), 7.59 (1 H, s), 7.55 (1H, s), 7.45-7.40 (2H, m), 7.30-7.27 (1H, m), 6.91 (1H, d, J = 8.4 Hz), 6.11 (1 H, tt, J = 55.5, 4.3 Hz) , 5.08 (2H, s), 4.45 (2H, td, J = 13.4, 4.3 Hz), 3.63 (3H, s), 2.51 (3H, s), 2.14 (3H, s) .; 1- {3-methyl -2-[(2,5-dimethyl-4-propanoylphenoxy) methyl] phenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.50 (1 H , s), 7.45-7.40 (2H, m), 7.28 (1H, dd, J = 7.1, 2.2 Hz), 6.66 (1H, s), 5.07 (2H, s), 3.64 (3H, s), 2.89 (2. 2H, q, J = 7.2 Hz), 2.52 (3H, s), 2.50 (3H, s), 2.08 (3H, s), 1.17 (3H, t, J = 7.2 Hz) .; 1- [2-({[1- (4-fluoro-2-methoxyphenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl ¹ H-NMR (CDCl ₃ ) δ: 7.76 (1 H, d, J = 2.5 Hz), 7.61 (1 H, m), 7. 38 (2 H, m), 7.25 (1H, m), 6.74 (2H, m), 5.75 (1H, d, J = 2.5 Hz), 5.29 (2H, s), 3.84 (3H, s), 3.61 (3H, s), 2.54 (3H, s) .; 1- (3-chloro-2-{[2-methyl-4- (5-fluoro-4-methylpyrimidin-2-yl) phenoxy] methyl} phenyl) -4-methyl- 1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.43 (1 H, d, J = 1.6 Hz), 8. 15 (1 H, dd, J = 8.6, 2.3 Hz), 8.11 (1 H , d, J = 1.4 Hz), 7.62 (1 H, dd, J = 7.9, 1.4 Hz), 7.48 (1 H, t, J = 8.0 Hz), 7.41 (1 H, dd, J = 7.9, 1.4 Hz), 6.92 (1H, d, J = 8.4 Hz), 5.39 (2H, s), 3.60 (3H, s), 2.56 ( 3H, d, J = 2.5 Hz), 2.10 (3H, s) .; 1- [2-({[1- (1,1-dimethyl-2-{[(prop-2-en-1-yl)]) Oxy] imino} ethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ : 7.55 (1H, s), 7.37-7.35 (2H, m), 7.24-7.20 (2H, m), 6.01-5.96 (1H, m), 5.54 (1H, d, J = 2.3 Hz), 5.33-5.21 (4H, m), 4.56 (2H, dt, J = 5.9, 1.3 Hz), 3.68 (3H, s), 2.53 (3H, s), 1.64 (6H, s) .; 1- [2- ({[ 1- (2-methoxypyrimidin-5-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H- NMR (CDCl ₃ ) δ: 8.72 (2 H, s), 7.58 (1 H, d, J = 2.5 Hz), 7.42-7.37 (2 H, m), 7.28-7.24 (1 H, m), 5.86 (1 H, d, 5) J = 2.7 Hz), 5.33 (2H, s), 4.05 (3H, s), 3.6 8 (3H, s), 2.57 (3H, s) .; 1- [3-Methyl-2-({2-methyl-4- [1- (2,2-difluoroethyl) -1H-pyrazole-5-) [Il] phenoxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 (1 H, d, J = 1.8 Hz), 7.47-7.42 ( 2H, m), 7.29 (1 H, dd, J = 6.8, 2.3 Hz), 7.18-7.13 (2 H, m), 6.91 (1 H, d, J = 8.4 Hz), 6.25 (1 H, d, J = 1.8 Hz ), 6.22 (1H, tt, J = 56.4 4.5 Hz), 5.08 (2H, s), 4.41 (2H, td, J = 13.0, 4.6 Hz), 3.65 (3H, s), 2.53 (3H, s), 2.13 (3H, s) .; 1- (3-methyl-2-{[2-methyl-4- (5-fluoro-1-methyl-1H-pyrazol-3-yl) phenoxy] methyl} phenyl) -4 -Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.51-7.50 (1 H, m), 7.47-7.45 (1 H, m), 7.43-7. 39 (2 H, m) , 7.29-7.26 (1H, m), 6.85 (1H, d, J = 8.5 H z), 5.95 (1 H, d, J = 5.7 Hz), 5.06 (2 H, s), 3. 76 (3 H, d, J = 1.4 Hz), 3.62 (3 H, s), 2.51 (3 H, s), 2.12 (2. 3H, s) .;

1- (3-Methyl-2-{[2,5-dimethyl-4- (cyclopropanecarbonyl) phenoxy] methyl} phenyl) -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.58 (1H, s), 7.47-7.38 (2H, m), 7.29 (1H, dd, J = 7.3, 2.1 Hz), 6.67 (1H, s), 5.08 (2H, s), 3.65 (3H, s), 2.51 (3H, s), 2.49 (3H, s), 2.46-2.39 (1H, m), 2.09 (3H, s), 1.22-1.16 (2H, m), 1.01-0.95 ( 2H, m) .; 1- {2-[({1- [2- (trifluoroacetoxy) -1,1-dimethylethyl] -1H-pyrazol-3-yl} oxy) methyl] -3-methylphenyl } -4-Methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38-7.33 (2H, m), 7.24-7.22 (2H, m), 5.53 (1H, d , J = 2.5 Hz), 5.18 (2H, s), 4.45 (2H, s), 3.68 (3H, s), 2.51 (3H, s), 1.55 (6H, s) .; 1-[2- ({ [1- (1,1-dimethylethyl) 1H- pyrazol-3-yl] thio} methyl) -3-methylphenyl] _{^{-4-methyl-1,4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.33 (1H, d, J = 2.3 Hz), 7.26-7.25 (2H, m), 7.18-7.13 (1 H, m), 5. 91 (1 H, d, J = 2.3 Hz), 4.15 (2 H, s), 3. 69 (3 H, s), 2.35 (3H, s), 1.54 (9H, s) .; 1- (3-chloro-2-{[2-methyl-4- (5-fluoropyrimidin-2-yl) phenoxy] methyl} phenyl) -4 -Methyl-1,4-dihydrotetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.60 (2H, s), 8.18-8.12 (2H, m), 7.62 (1 H, d, J = 8.0 Hz ), 7.48 (1 H, t, J = 8.0 Hz), 7.41 (1 H, d, J = 8.0 Hz), 6.94 (1 H, d, J = 8.7 Hz), 5. 39 (2 H, s), 3. 60 (3 H, s) ), 2.10 (3H, s) .; 1- [2-({[1- (3,4-difluorophenyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4- Methyl-1 _{^{4-dihydro-5-one, 1 H-NMR (CDCl 3}} ) δ: 7.60 (1H, d, J = 2.5 Hz), 7.46-7.38 (3H, m), 7.28-7.16 (3H, m), 5.82 (1H, d, J = 2.5 Hz), 5.32 (2H, s), 3.65 (3H, s), 2.56 (3H, s). 1- [2-({[1- (1-ethoxycarbonyl-1)] -Methylethyl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.38 -7.33 (2H, m), 7.29 (1 H, d, J = 2.5 Hz), 7.22 (1 H, dd, J = 6.3, 2.9 Hz), 5.57 (1 H, d, J = 2.5 Hz), 5.20 (2 H, 2 H, d s), 4.11 (2H, q, J = 7.1 Hz), 3.68 (3H, s), 2.51 (3H, s), 1. 73 (6H, s), 1.17 (3H, t, J = 7.1 Hz) .; 1 -[2-({[1- (tetrahydropyran-2-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole-5- On, ¹ H-NMR (CD Cl ₃ ) δ: 7.40-7.35 (2H, m), 7.33 (1H, d, J = 2.5 Hz), 7.23 (1 H, dd, J = 6.4, 2.7 Hz), 5.63 (1 H, d, J = 2.5 Hz ), 5.21 (2H, s), 5.14 (1H, dd, J = 9.6, 2.5 Hz), 4.07-4.03 (1H, m), 3.70-3.65 (4H, m), 2.51 (3H, s), 2.02- 1.91 (2H, m), 1.67-1.64 (2H, m), 1.59-1.48 (2H, m) .; 1- {3-methyl-2-[({[1- (3, 3-dimethylbutylidene-) 2-yl) amino] oxy} methyl) phenyl] -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.37-7.31 (2H, m), 7.21-7.17 (1H, m), 5.08 (2H, s), 3.70 (3H, s), 2.51 (3H, s), 1.65 (3H, s), 1.01 (9H, s) .; 1-(2- {[(( 1-Pentyl-1H-pyrazol-3-yl) oxy] methyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-7-one, ¹ H-NMR (CDCl ₃ ) δ: 7.39- 7.34 (2H, m), 7.23 (1 H, dd, J = 6.3, 2.9 Hz), 7.08 (1 H, d, J = 2.3 Hz), 5.50 (1 H, d, J = 2.3 Hz), 5.1 9 (2H, s), 3.87 (2H, t, J = 7.1 Hz), 3.68 (3H, s), 2.53 (3H, s), 1.80-1.73 (2H, m), 1.36-1.30 (2H, m) , 1.28-1. 19 (2H, m), 0.89 (3H, t, J = 7.2 Hz) .; 1- {3-methyl-2-[(piperidin-1-yloxy) methyl] phenyl} -4-methyl-1 , 4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.37-7.32 (2H, m), 7.20 (1 H, dd, J = 6.1, 3.1 Hz), 4.67 (2 H, s), 3.71 (3H, s), 3.11-3.09 (2H, m), 2.51 (3H, s), 2.28-2.26 (2H, m), 1.59-1.48 (5H, m), 1.08-1.06 (1H, m). ;

1- [2-({[1- (6-propyloxypyridin-3-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydro Tetrazole-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.31 (1 H, d, J = 2.7 Hz), 7. 80 (1 H, dd, J = 8.8, 2.9 Hz), 7.56 (1 H, d, J = 2.5 Hz), 7.42-7.37 (2 H, m), 7. 26 (1 H, m), 6. 79 (1 H, d, J = 8.9 Hz), 5. 80 (1 H, d, J = 2.7 Hz), 5.32 (2 H, s) , 4.26 (2H, t, J = 6.8 Hz), 3.64 (3 H, s), 2.56 (3 H, s), 1. 83-1. 79 (2 H, m), 1.04 (3 H, t, J = 7.4 Hz) .; 1 -[2-({[1- (2-methoxythiazol-4-yl) -1H-pyrazol-3-yl] oxy} methyl) -3-methylphenyl] -4-methyl-1,4-dihydrotetrazole- 5-one, ¹ H-NMR (CDCl ₃ ) δ: 7.88 (1 H, d, J = 2.7 Hz), 7.42-7. 37 (2 H, m), 7. 25 (1 H, dd, J = 7.2, 3.5 Hz), 6.50 (1H, s), 5.72 (1H, d, J = 2.7 Hz), 5.29 (2H, s), 4.09 (3H, s), 3.66 (3H, s), 2.55 (3H, s) .; 1- {2-[({1- [2- (1-methylethoxy) -3-methoxypyridin-4-yl] ] -1H-Pyrazol-3-yl} oxy) methyl] -3-methylphenyl} -4-methyl-1,4-dihydrotetrazol-5-one, ¹ H-NMR (CDCl ₃ ) δ: 8.23 (1 H, d, J = 2.9 Hz), 7. 86 (1 H, d, J = 5.7 Hz), 7.41-7. 40 (2 H, m), 7. 35 (1 H, d, J = 5.4 Hz), 7. 26-7. 25 (1 H, m), 5.84 (1H, d, J = 2.7 Hz), 5.43-5.37 (1H, m), 5.33 (2H, s), 3.80 (3H, s), 3.64 (3H, s), 2.56 (3H, s), 1.42 (6H, d, J = 6.3 Hz).

The present compounds AA1-BA1 to AA319-BA6365 can be obtained according to the method described above. The present compounds AA1-BA1 to AA319-BA6365 are compounds represented by the following formula (AABA).

[Wherein, each of X ^{111 to} X ¹¹⁷ represents a substituent corresponding to each of substituent numbers (MA 1) AA 1 to AA 3 19 shown below, and E ¹⁰¹ represents a substituent number shown below (MA 2) BA 1 to BA 6365 Each represents a corresponding substituent. ]
For example, the present compound AA1-BA1, in the compounds of formula (AABA), X ¹¹¹ ~X1 ¹⁷ substituents numbers MA1 (X ¹¹ is a sulfur atom, X ¹¹³ to X ¹¹⁶ is a hydrogen atom, X ¹¹² and X ¹¹⁷ Is an oxygen atom, and E ¹⁰¹ is a compound in which the substituent number (MA 2) is BA 1 (phenyl group), and is represented by the following formula.

[Substituent group number ^{(MA1); X 111, X} 112, X 113, X1 14, X 115, X 116, X 117], [AA1; S, O, H, H, H, H, O], [AA2 S, O, F, H, H, H, O, [AA 3; S, O, Cl, H, H, H, O], [AA 4; S, O, Br, H, H, H, O ], [AA5; S, O, I, H, H, H, O], [AA 6; S, O, Me, H, H, H, O], [AA 7; S, O, Et, H, H , H, O], [AA 8; S, O, Pr, H, H, H, O], [AA 9; S, O, i-Pr, H, H, H, O], [AA 10; S, O , CH = CH ₂ , H, H, H, O, [AA 11; S, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AA 12; S, O, C≡CH , H, H, H, O], [AA 13; S, O, C≡CCH ₃ , H, H, H, O], [AA 14; S, O, c-Pr, H, H, H, O] , [AA 15; S, O, OMe, H, H, H, O], [AA 16; S, O, OEt, H, H, H, O], [AA 17; S, O, Oi-Pr, H, H, H, O], [AA 18; S, O, S Me, H, H, H, O], [AA 19; S, O, SE t, H, H, H, O], [AA 20; S, O, _{CH 2 F, H, H,} H, O], [AA21; S, O, CHF 2, H, H, H, O], [AA22; S, O, CF 3, H, H, H, O] , [AA23; S, O, OCH 2 F, H, H, H, O], [AA24; S, O, OCHF 2, H, H, H, O], [AA25; S, O, OCF 3, H, H, H, O], [AA 26; S, O, SCH ₂ F, H, H, H, O], [AA 27; S, O, SCHF ₂ , H, H, H, O], [AA 28 S, O, SCF ₃ , H, H, H, O, [AA 29; S, O, CN, H, H, H, O], [AA 30; O, O, H, H, H, H, H, O], [AA 31; O, O, F, H, H, H, O], [AA 32; O, O, Cl, H, H, H, O], [AA 33; O, O, Br, H, H, H, O], [AA 34; O, O, I, H, H, H, O], [AA 35; O, O, Me, H, H, H, O], [AA 36; O, O, O, Et, H, H, H, O], [AA 37; O, O, Pr, H, H, H, O], [AA 38; O, O, i-Pr, H, H, H, O], [AA AA 39; O, O, CH = CH ₂ , H, H, H, O] , [AA40; O, O, C (CH 3) = CH 2, H, H, H, O], [AA41; O, O, C≡CH, H, H, H , O], [AA 42; O, O, C≡CCH ₃ , H, H, H, O], [AA 43; O, O, c-Pr, H, H, H, O], [AA 44; O, O, OMe, H, H, H, O], [AA 45; O, O, OEt, H, H, H, O], [AA 46; O, O, Oi-Pr, H, H, H, O] , [AA 47; O, O, SMe, H, H, H, O], [AA 48; O, O, SE t, H, H, H, O], [AA 49; O, O, CH ₂ F, H, H, H, O], [ AA50; O, O, CHF 2, H, H, H, O], [AA51; O, O, CF 3, H, H, H, O], [AA52; O, _{O, OCH 2 F, H,} H, H, O], [aA53; O, O, OCHF 2, H, H, H, O], [AA54; O, O, OCF 3, H, H, H, O], [AA 55; O, O, SCH ₂ F, H, H, H, O], [AA 56; O, O, SCHF ₂ , H, H, H, O], [AA 57; O, O, SCF ₃ , H, H, H, O], [AA 58; O, O, CN, H, H, H, O], [AA 59; S, S, H, H, H, H, O], [AA 60; S, S, F, H, H, H, O], [AA 61; S, S, Cl, H, H, H, O], [AA 62; S, S, Br, H, H, H, O] [AA 63; S, S, I, H, H, H, O], [AA 64; S, S, Me, H, H, H, O], [AA 65; S, S, Et, H, H, H H, O], [AA 66; S, S, Pr, H, H, H, O], [AA 67; S, S, i-Pr, H, H, H, O], [AA 68; S, S, S, _{CH = CH 2, H, H} , H, O], [AA69; S, S, C (CH 3) = CH 2, H, H, H, O], [AA70; S, S, C≡CH, H, H, H, O], [AA 71; S, S, C≡CCH ₃ , H, H, H, O], [AA 72; S, S, c-Pr, H, H, H, O], [AA 73; S, S, OMe, H, H, H, O], [AA 74; S, S, OEt, H, H, H, O], [AA 75; S, S, Oi-Pr, H, H , H, O], [AA 76; S, S, SMe, H, H, H, O], [AA 77; S, S, SE t, H, H, H, O], [AA 78; S, S, CH ₂ F, H, H, H, O], [AA 79; S, S, CHF ₂ , H, H, H, O], [ AA80; S, S, CF 3, H, H, H, O], [AA81; S, S, OCH 2 F, H, H, H, O], [AA82; S , S, OCHF ₂ , H, H, H, O], [AA 83; S, S, OCF ₃ , H, H, H, O], [AA 84; S, S, SCH ₂ F, H, H, H , O], [AA 85; S, S, SCHF ₂ , H, H, H, O], [AA 86; S, S, SCF ₃ , H, H, H, O], [AA 87; S, S, CN , H, H, H, O], [AA 88; O, S, H, H, H, H, O], [AA 89; O, S, F, H, H, H, O], [AA 90; O , S, Cl, H, H, H, O, [AA 91; O, S, Br, H, H, H, O], [AA 92; O, S, I, H, H, H, O], [AA 93; O, S, Me, H, H, H, O], [AA 94; O, S, Et, H, H, H, O], [AA 95; O, S, Pr, H, H, H , O], [AA96; O , S, i-Pr, H, H, H, O], [AA97; O, S, CH = CH 2, H, H, H, O], [AA98; O, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AA 99; O, S, C≡CH, H, H, H, O], [AA 100; O, S, C≡ CCH ₃ , H, H, H, O],

[AA 101; O, S, c-Pr, H, H, H, O], [AA 102; O, S, OMe, H, H, H, O], [AA 103; O, S, OE t, H, H , H, O], [AA 104; O, S, Oi-Pr, H, H, H, O], [AA 105; O, S, SMe, H, H, H, O], [AA 106; O, S , SEt, H, H, H, O], [AA 107; O, S, CH ₂ F, H, H, H, O], [AA 108; O, S, CHF ₂ , H, H, H, O] , [AA109; O, S, CF 3, H, H, H, O], [AA110; O, S, OCH 2 F, H, H, H, O], [AA111; O, S, OCHF 2, H, H, H, O] , [AA112; O, S, OCF 3, H, H, H, O], [AA113; O, S, SCH 2 F, H, H, H, O], [AA114 O, S, SCHF ₂ , H, H, H, O, [AA 115; O, S, SCF ₃ , H, H, H, O], [AA 116; O, S, CN, H, H, H , O], [AA117; S, O, H, H, H, H, S], [AA 118; S, O, F, H, H, H, S], [AA119; S, O, Cl, H , H, H, S], [AA 120; S, O, Br, H, H, S], [AA 121; S, O, I, H, H, H, S], [AA 122; S, O , Me, H, H, H, S], [AA 123; S, O, Et, H, H, H, S], [AA 124; S, O, Pr, H, H, H, S], [AA 125 S, O, i-Pr, H, H, H, S, [AA 126; S, O, CH = CH ₂ , H, H, H, S], [AA 127; S, O, C (CH _3; ) = CH ₂ , H, H, H, S], [AA 128; S, O, C≡CH, H, H, H, S], [AA 129; S, O, C≡ CCH ₃ , H, H, H H, S], [AA 130; S, O, c-Pr, H, H, H, S], [AA 131; S, O, OMe, H, H, H, S], [AA 132; S, O, OEt, H, H, H, S], [AA 133; S, O, Oi-Pr, H, H, H, S], [AA 134; S, O, SMe, H, H, H, S], [ AA 135; S, O, SEt, H, H, H, S], [AA 136; S, O, CH ₂ F, H, H, H, S], [AA 137; S, O, CHF ₂ , H, H , H, S], [AA138 ; S, O, CF 3, H, H, H, S], [AA139; S, O, OCH 2 F, H, H, H, S], [ AA 140; S, O, OCHF ₂ , H, H, H, S], [AA 141; S, O, OCF ₃ , H, H, H, S], [AA 142; S, O, SCH ₂ F, H, H, H, S], [ AA143; S, O, SCHF 2, H, H, H, S], [AA144; S, O, SCF 3, H, H, H, S], [AA145; S, O, CN, H, H, H, S], [AA 146; O, O, H, H, H, H, S], [AA 147; O, O, F, H, H, H, S], [AA AA 148; O, O, Cl, H, H, H, S], [AA 149; O, O, Br, H, H, H, S], [AA 150; O, O, I, H, H, H, S], [AA 151; O, O, Me, H, H, H, S], [AA 152; O, O, Et, H, H, H, S], [AA 153; O, O, Pr, H, S H, H, S], [ AA154; O, O, i-Pr, H, H, H, S], [AA155; O, O, CH = CH 2, H, H, H, S], [AA156 ; O, O, C (CH 3) = CH 2, H, H, H, S], [AA157; O, O, C≡CH, H, H, H, S], [AA158; O, O, C≡CCH ₃ , H, H, H, S], [AA 159; O, O, c-Pr, H, H, H, S], [AA 160; O, O, OMe, H, H, H, S ], [AA161; O, O, OEt, H, H, H, S], [AA 162; O, O, Oi-Pr, H, H, H, S], [AA 163; O, O, SMe, H , H, H, S], [AA 164; O, O, SE t, H, H, H, S], [AA 165; O, O, CH ₂ F, H, H, H, S], [AA 166; O _{, O, CHF 2, H,} H, H, S], [AA167; O, O, CF 3, H, H, H, S], [AA168; O, O, OCH 2 F, H, H, H , S], [AA169; O , O, OCHF 2, H, H, H, S], [AA170; O, O, OCF 3, H, H, H, S], [AA171; O, O, SCH ₂ F, H, H, H, S], [AA 172; O, O, SCHF ₂ , H, H, H, S], [AA 173; O, O, SCF ₃ , H, H, H, S], [AA 174; O, O, CN, H, H, H, S], [AA 175; S, S, H, H, H, H, S], [AA 176; S, S, F, H, H, H , S], [AA 177; S, S, Cl, H, H, H, S], [AA 178; S, S, Br, H, H, H, S], [AA 179 S, S, I, H, H, H, S], [AA 180; S, S, Me, H, H, H, S], [AA 181; S, S, Et, H, H, H, S ], [AA 182; S, S, Pr, H, H, H, S], [AA 183; S, S, i-Pr, H, H, H, S], [AA 184; S, S, CH = CH ₂ , H, H, H, S], [AA 185; S, S, C (CH ₃ ) = CH ₂ , H, H, H, S], [AA 186; S, S, C≡CH, H, H , H, S], [AA 187; S, S, C≡CCH ₃ , H, H, H, S], [AA 188; S, S, c-Pr, H, H, H, S], [AA 189; S, S, OMe, H, H, H, S], [AA 190; S, S, OEt, H, H, H, S], [AA 191; S, S, Oi-Pr, H, H, H, S], [AA 192; S, S, SMe, H, H, H, S], [AA 193; S, S, SE t, H, H, H, S], [AA 194; S, S, CH ₂ F, H, H, H, S] , [AA195; S, S, CHF 2, H, H, H, S], [AA196; S, S, CF 3, H, H, H, S], [AA197; _{S, S, OCH 2 F,} H, H, H, S], [AA198; S, S, OCHF 2, H, H, H, S], [AA199; S, S, OCF 3, H, H, H, S], [AA 200; S, S, SCH ₂ F, H, H, H, S],

[AA201; S, S, SCHF 2, H, H, H, S], [AA202; S, S, SCF 3, H, H, H, S], [AA203; S, S, CN, H, H , H, S], [AA 204; O, S, H, H, H, H, S], [AA 205; O, S, F, H, H, H, S], [AA 206; O, S, Cl , H, H, H, S], [AA 207; O, S, Br, H, H, S, [AA 208; O, S, I, H, H, H, S], [AA 209; , S, Me, H, H, H, S], [AA 210; O, S, Et, H, H, H, S], [AA 211; O, S, Pr, H, H, H, S], [AA212; O, S, i -Pr, H, H, H, S], [AA213; O, S, CH = CH 2, H, H, H, S], [AA214; O, S, C ( CH ₃ ) = CH ₂ , H, H, H, S, [AA 215; O, S, C≡CH, H, H, H, S], [AA 216; O, S, C≡CCH ₃ , H, H, H, S], [AA 217; O, S, c-Pr, H, H, H, S], [AA 218; O, S, OMe, H, H, H, S], [AA 219; O, S, OEt, H, H, H, S], [AA 220; O, S, Oi-Pr, H, H, H, S], [AA 221; O, S, SMe, H, H, H, S] , [AA 222; O, S, SEt, H, H, H, S], [AA 223; O, S, CH ₂ F, H, H, H, S], [AA 224; O, S, CHF ₂ , H , H, H, S], [AA225; O, S, CF 3, H, H, H, S], [AA226; O, S, OCH 2 F, H, H, H, S], [AA227; O, S, OCHF ₂ , H, H, H, S, [AA 228; O, S, OCF ₃ , H, H, H, S], [AA 229; O, S, SCH ₂ F, H, H, H, S], [AA 230; O, S, SCHF ₂ , H, H, H, S], [AA 231; O, S, SCF ₃ , H, H, H, S], [AA 232; O, S, CN, H, H, H, S], [AA 233; S, O, H, F, H, H, O], [AA 234; S, O, F, F, H, H, O], [AA 235; S, O, Cl, F, H, H, O], [AA 236; S, O, Br, F, H, H, O], [AA 237; S, O, I, F, H, H, O] [AA 238; S, O, Me, F, H, H, O], [AA 239: S, O, Et, F, H, H, O], [AA 240; S, O, Pr, F, H, H, O], [AA241; S, O, i-Pr, F, H, H, O], [AA242; S, O, CH = CH 2, F, H, H, O], [AA243; S, O , C (CH ₃ ) = CH ₂ , F, H, H, O], [AA 244; S, O, C≡CH, F, H, H, O], [AA 245; S, O, C≡CCH ₃ , F, H, H, O], [AA 246; S, O, c-Pr, F, H, H, O], [AA 247; S, O, OMe, F, H, H, O], [AA 248 S, O, OEt, F, H, H, O], [AA 249; S, O, Oi-Pr, F, H, H, O], [AA 250; S, O, SMe, F, H, H , O], [AA 251; S, O, SEt, F, H, H, O], [AA 252; S, O, CH ₂ F, F, H, H, O], [AA 253; S, O, CHF _{2, F, H, H,} O], [AA254; S, O, CF 3, F, H, H, O], [AA255; S, O, OCH 2 F, F, H, H, O], [AA256; S, O, OCHF 2, F, H, H, O], [AA257; S, O, OCF 3, F, H, H, O], [AA258; S, O, SCH 2 F, F , H, H, O], [AA 259; S, O, SCHF ₂ , F, H, H, O], [AA 260; S, O, SCF ₃ , F, H, H, O], [AA 261; , O, CN, F, H, H, O], [AA 262; S, O, H, H, F, H, O], [AA 263; S, O, F, H, F, H, O], [AA 264; S, O, Cl, H, F, H, O], [AA 265; S, O, Br, H, F, H, O], [AA 266; S, O, I, H, F, H , O], [AA 267; S, O, Me, H, F, H, O], [AA 268; S, O, Et, H, F, H, O], [AA 269; S, O, Pr, H , F, H, O], [AA270; S, O, i-Pr, H, F, H, O], [AA271; S, O, CH = CH 2, H, F, H, O], [ AA 272; S, O, C (CH ₃ ) = CH ₂ , H, F, H, O], [AA 273; S, O, C≡CH, H, F, H, O], [AA 274; S, O , C≡CCH ₃ , H, F, H, O], [AA 275; S, O, c-Pr, H, F, H, O], [AA 276; S, O, OMe, H, F, H, O], [AA 277; S, O, OEt, H, F, H, O], [AA 278; S, O, Oi-Pr, H, F, H, O], [AA 279; S, O, SMe, H, F, H, O], [AA 280; S, O, SE t, H, F, H, O], [AA 281; S, O, CH ₂ F, H, F, H, O], [AA282; S, O, CHF 2, H, F, H, O], [AA283; S, O, CF 3, H, F, H, O], [AA284; S, O, OCH 2 F, H, F, H, O], [AA285; S, O, OCHF 2, H, F, H, O], [AA286; S, O, OCF 3, H, F, H, O], [ AA 287; S, O, SCH ₂ F, H, F, H, O], [AA 288; S, O, SCHF ₂ , H, F, H, O], [AA 289; S, O, SCF ₃ , H, F, H, O], [AA 290; S, O, CN, H, F, H, O], [AA 291; S, O, H, H, H, F, O], [AA 292; S, O, F, H, H, F, O], [AA 293; S, O, Cl, H, H, F, O], [AA 294; S, O, Br, H, H, F, O], [AA 295; S, O, I, H, H, F, O], [AA 296; S, O, Me, H, H, F, O], [AA 297; S, O, Et, H, H, F, O] , [AA 298; S, O, Pr, H, H, F, O], [AA 299; S, O, i-Pr, H, H, F, O], [AA 300; S, O, CH = CH ₂ , H, H, F, O],

[AA301; S, O, C (CH 3) = CH 2, H, H, F, O], [AA302; S, O, C≡CH, H, H, F, O], [AA303; S, O, C≡CCH ₃ , H, H, F, O], [AA 304; S, O, c-Pr, H, H, F, O], [AA 305; S, O, OMe, H, H, F , O], [AA 306; S, O, OEt, H, H, F, O], [AA 307; S, O, Oi-Pr, H, H, F, O], [AA 308; S, O, SMe , H, H, F, O], [AA 309; S, O, SE t, H, H, F, O], [AA 310; S, O, CH ₂ F, H, H, F, O], [AA 311 _{; S, O, CHF 2,} H, H, F, O], [AA312; S, O, CF 3, H, H, F, O], [AA313; S, O, OCH 2 F, H, H , F, O], [AA314 ; S, O, OCHF 2, H, H, F, O], [AA315; S, O, OCF 3, H, H, F, O], [AA316; S, O , SCH ₂ F, H, H, F, O], [AA 317; S, O, SCHF ₂ , H, H, F, O], [AA 318; S, O, SCF ₃ , H, H, F, O ], [AA 319; S, O, CN, H, H, F, O] ,.

[Substituent group number ^{(MA2); E 101],} [BA1; phenyl], [BA2; 2-fluorophenyl], [BA3; 3- fluorophenyl], [BA4; 4-fluorophenyl], [BA5; 2, 4-difluorophenyl], [BA6; 2,4,6-trifluorophenyl], [BA7; 2,3,4,5,6-pentafluorophenyl], [BA8; 2,3-difluorophenyl], [BA BA9; 2-chlorophenyl], [BA10; 3-chlorophenyl], [BA11; 4-chlorophenyl], [BA12; 2,3-dichlorophenyl], [BA13; 2,4-dichlorophenyl], [BA14; Dichlorophenyl], [BA15; 2,6-dichlorophenyl], [BA16; 3,4-dichlorophenyl], [BA17; 3,5-dichlorophenyl], [BA18; 2,3,4-trichlorophenyl], [BA19; , 3,5-trichlorophenyl], [BA20; 2,3,6-trichlorophenyl], [BA21; 2,4,5-trichlorophenyl], [BA22; 2,4,6-trichlorophenyl], [BA23 3,4,5-Trichlorophenyl], [BA24; 2,3,4,6-tetrachlorophenyl], [BA25; 2,3,5,6-tetrachlorophenyl], [BA26; 5,6-Pentak Rophenyl], [BA27; 2-bromophenyl], [BA28; 3-bromophenyl], [BA29; 4-bromophenyl], [BA30; 2,4-dibromophenyl], [BA31; 2, 5-dibromophenyl ], [BA32; 2,6-dibromophenyl], [BA33; 2,4,6-tribromophenyl], [BA34; 2,3,4,5,6-pentabromophenyl], [BA35; Iodophenyl], [BA36; 3-iodophenyl], [BA37; 4-iodophenyl], [BA38; 2,4-diiodophenyl], [BA39; 2-chloro-3-fluorophenyl], [BA40; 2-chloro-4-fluorophenyl], [BA41; 2-chloro-5-fluorophenyl], [BA42; 2-chloro-6-fluorophenyl], [BA43; 2-chloro-3-bromophenyl], [BA43; 2-chloro-4-bromophenyl], [BA45; 2-chloro-5-bromophenyl], [BA46; 2-chloro-6-bromophenyl], [BA47; 2-bromo-3-chlorophenyl], [BA 48; 2-bromo-4-chlorophenyl], [BA 49; 2-bromo-5-chlorophenyl], [BA 50; 2-bromo-3-fluorophenyl], [BA 51; 2-bromo-4-fluo Phenyl], [BA 52; 2-bromo-5-fluorophenyl], [BA 53; 2-bromo-6-fluorophenyl], [BA 54; 2-fluoro-3-chlorophenyl], [BA 55; 2-fluoro-4- Chlorophenyl], [BA56; 2-fluoro-5-chlorophenyl], [BA57; 2-fluoro-4-bromophenyl], [BA58; 3-chloro-4-fluorophenyl], [BA59; 3-chloro-5- Fluorophenyl], [BA60; 3-chloro-4-bromophenyl], [BA61; 3-chloro-5-bromophenyl], [BA62; 3-fluoro-4-chlorophenyl], [BA63; 3-fluoro-4 -Bromophenyl], [BA64; 3-bromo-4-chlorophenyl], [BA65; 3-bromo-4-fluorophenyl], [BA66; 2,6-dichloro-4-bromophenyl], [BA67; 3-Difluoro-4-chlorophenyl], [BA 68; 2, 6-difluoro-4-chlorophenyl], [BA 69; 2, 5-difluoro-4-chlorophenyl], [BA 70; 3,5-difluoro-4-chlorophenyl] , [BA71; 2,3,5-trifluoro-4-chlorophenyl], [BA72; 2,3,6-trifluoro-4-chloro Phenyl], [BA73; 2,3,5,6-tetrafluoro-4-chlorophenyl], [BA74; 2-fluoro-4-bromophenyl], [BA75; 2,3-difluoro-4-bromophenyl], [BA 76; 2,6-difluoro-4-bromophenyl], [BA 77; 2, 5-difluoro-4-bromophenyl], [BA 78; 3,5-difluoro-4-bromophenyl], [BA 79; 3,5-Trifluoro-4-bromophenyl], [BA80; 2,3,6-trifluoro-4-bromophenyl], [BA81; 2,3,5,6-tetrafluoro-4-bromophenyl] [BA 82; 2-fluoro-4-iodophenyl], [BA 83; 3-fluoro-4-iodophenyl], [BA 84; 2,3-difluoro-4-iodophenyl], [BA 85; 2, 6-difluoro -4-iodophenyl], [BA86; 2,5-difluoro-4-iodophenyl], [BA87; 3,5-difluoro-4-iodophenyl], [BA88; 2,3,5-trifluoro-4 -Iodophenyl], [BA89; 2,3,6-trifluoro-4-iodophenyl], [BA90; 2,3,5,6-tetrafluoro-4-iodophenyl], [BA91; 2-methylphenyl ], [B A92; 3-methylphenyl], [BA93; 4-methylphenyl], [BA94; 2,3-dimethylphenyl], [BA95; 2,4-dimethylphenyl], [BA96; 2, 5-dimethylphenyl], [BA97; 2,6-dimethylphenyl], [BA98; 3,4-dimethylphenyl], [BA99; 3,5-dimethylphenyl], [BA100; 2,3,5-trimethylphenyl],

[BA101; 2,3,4-trimethylphenyl], [BA102; 2,3,6-trimethylphenyl], [BA103; 2,4,5-trimethylphenyl], [BA104; 2,4,6-trimethylphenyl ], [BA105; 3,4,5-trimethylphenyl], [BA106; 2,3,4,6-tetramethylphenyl], [BA107; 2,3,5,6-tetramethylphenyl], [BA108; 2,3,4,5,6-pentamethylphenyl], [BA109; 2-ethylphenyl], [BA110; 3-ethylphenyl], [BA111; 4-ethylphenyl], [BA112; 2,4-diethyl] Phenyl], [BA113; 2,6-diethylphenyl], [BA114; 3,5-diethylphenyl], [BA115; 2,4,6-triethylphenyl], [BA116; 2-propylphenyl], [BA117; 3-propylphenyl], [BA118; 4-propylphenyl], [BA119; 2-isopropylphenyl], [BA120; 3-isopropylphenyl], [BA121; 4-isopropylphenyl], [BA122; Phenyl], [BA123; 2,6-diisopropylphenyl], [BA124; 3,5-diisopropylphenyl], [BA125; 2-s-butylphenyl ], [BA126; 3-s-butylphenyl], [BA127; 4-s-butylphenyl], [BA128; 2-t-butylphenyl], [BA129; 3-t-butylphenyl], [BA130; 4] -t-Butylphenyl], [BA131; 2-butylphenyl], [BA132; 3-butylphenyl], [BA133; 4-butylphenyl], [BA134; 2-nonylphenyl], [BA135; 3-nonylphenyl ], [BA136; 4-nonylphenyl], [BA137; 2-methyl-4-t-butylphenyl], [BA138; 2-methyl-6-t-butylphenyl], [BA139; 2-methyl-4- Isopropylphenyl], [BA140; 2-methyl-5-isopropylphenyl], [BA141; 3-methyl-4-isopropylphenyl], [BA142; 2-cyclohexylphenyl], [BA143; 3-cyclohexylphenyl], [BA144 4-cyclohexylphenyl], [BA145; 2-cyclopropylphenyl], [BA146; 3-cyclopropylphenyl], [BA147; 4-cyclopropylphenyl], [BA148; 4-cyclobutylphenyl], [BA149; 2-Cyclopentylphenyl], [BA150; [N-yl], [BA151; 4-cyclopentylphenyl], [BA152; 2-chloro- (1,1'-biphenyl) -4-yl], [BA153; 2-bromo- (1,1'-biphenyl) -4 -Yl], [BA154; 2-hydroxyphenyl], [BA155; 3-hydroxyphenyl], [BA156; 4-hydroxyphenyl], [BA157; 2-methoxyphenyl], [BA158; 3-methoxyphenyl], [BA158; BA 159; 4-methoxyphenyl], [BA 160; 2-ethoxyphenyl], [BA 161; 3-ethoxyphenyl], [BA 162; 4-ethoxyphenyl], [BA 163; 2-propyloxyphenyl], [BA 164; Propyloxyphenyl], [BA165; 4-propyloxyphenyl], [BA166; 2-isopropyloxyphenyl], [BA167; 3-isopropyloxyphenyl], [BA168; 4-isopropyloxyphenyl], [BA169; Hexyloxyphenyl], [BA170; 3-hexyloxyphenyl], [BA171; 4-hexyloxyphenyl], [BA172; 2-benzyloxyphenyl], [BA173; 3-benzyloxyphenyl], [BA174; Ben Roxyphenyl], [BA175; 2,3-dimethoxyphenyl], [BA176; 2,4-dimethoxyphenyl], [BA177; 2,5-dimethoxyphenyl], [BA178; 2,6-dimethoxyphenyl], [ BA179; 3,4-dimethoxyphenyl], [BA180; 3,5-dimethoxyphenyl], [BA181; 2-t-butoxyphenyl], [BA182; 3-t-butoxyphenyl], [BA183; Butoxyphenyl], [BA184; 3- (3-chlorophenyl) phenyl], [BA185; 4- (4-chlorophenyl) phenyl], [BA186; 2-phenoxyphenyl], [BA187; 3-phenoxyphenyl], [BA188 4-phenoxyphenyl], [BA189; 2- (2-fluorophenoxy) phenyl], [BA190; 3- (3-chlorophenoxy) phenyl], [BA191; 4- (4-chlorophenoxy) phenyl], [BA BA192; 2,3,6-trimethyl-4-fluorophenyl], [BA193; 2,3,6-trimethyl-4-chlorophenyl], [BA194; 2,3,6-trimethyl-4-bromophenyl], [BA194; BA 195; 2,4-dimethyl-6-fluorophenyl], [BA 196; 2,4-dimethyl-6-chlorof Phenyl], [BA 197; 2,4-dimethyl-6-bromophenyl], [BA 198; 2-isopropyl-4-chloro-5-methylphenyl], [BA 199; 2-chloro-4-nitrophenyl], [BA 200 2-nitro-4-chlorophenyl],

[BA 201; 2-methoxy-5-nitrophenyl], [BA 202; 2,4-dichloro-5-nitrophenyl], [BA 203; 2,4-dichloro-6-nitrophenyl], [BA 204; 2, 6- Dichloro-4-nitrophenyl], [BA205; 2,6-dibromo-4-nitrophenyl], [BA206; 2,6-diiodo-4-nitrophenyl], [BA207; 2-methyl-5-isopropyl-4. -Chlorophenyl], [BA208; 2-methoxycarbonylphenyl], [BA209; 3-methoxycarbonylphenyl], [BA210; 4-methoxycarbonylphenyl], [BA211; 2-acetoxyphenyl], [BA212; 3-acetoxyphenyl ], [BA213; 4-acetoxyphenyl], [BA214; 2-methoxymethylphenyl], [BA215; 3-methoxymethylphenyl], [BA216; 4-methoxymethylphenyl], [BA217; (Biphenyl) -4-yl], [BA 218; (1,1′-biphenyl) -3-yl], [BA 219; (1,1′-biphenyl) -2-yl], [BA 220; Fluorophenyl) phenyl], [BA221; 2-methyl-5-bromophenyl], [BA222; 2-methyl-6-bromo 2-chloro-3-methylphenyl], [BA224; 2-chloro-4-methylphenyl], [BA225; 2-chloro-5-methylphenyl], [BA226; 2-fluoro-3 -Methylphenyl], [BA227; 2-fluoro-4-methylphenyl], [BA228; 2-fluoro-5-methylphenyl], [BA229; 2-bromo-3-methylphenyl], [BA230; 4-methylphenyl], [BA 231; 2-bromo-5-methylphenyl], [BA 232; 3-methyl-4-chlorophenyl], [BA 233; 3-methyl-5-chlorophenyl], [BA 234; 3-methyl -4-fluorophenyl], [BA235; 3-methyl-5-fluorophenyl], [BA236; 3-methyl-4-bromophenyl], [BA237; 3-methyl-5-bromophenyl], [BA238; 3 -Fluoro-4-methylphenyl], [BA239; 3-chloro-4-methylphenyl], [BA240; 3-bromo-4-methylphenyl], [BA241; 2-chloro-4,5-dimethylphenyl], [BA 242; 2-bromo-4, 5-dimethylphenyl], [BA 243; 2-chloro-3,5-dimethylphenyl], [BA 244; 2-bromo-3,5-dime 2, 2-Dibromo-4-methylphenyl], [BA246; 2,4-dichloro-6-methylphenyl], [BA 247; 2, 6-dichloro-4-methylphenyl], [BA248] 2,4-difluoro-6-methylphenyl], [BA 249; 2,4-dibromo-6-methylphenyl], [BA 250; 2,6-dimethyl-4-fluorophenyl], [BA 251; 2, 6- Dimethyl-4-chlorophenyl], [BA252; 2,6-dimethyl-4-bromophenyl], [BA253; 3,5-dimethyl-4-fluorophenyl], [BA254; 3,5-dimethyl-4-chlorophenyl] , [BA255; 3,5-dimethyl-4-bromophenyl], [BA256; 2,3-difluoro-4-methylphenyl], [BA257; 2,5-difluoro-4-methylphenyl], [BA258; 3 2, 5-difluoro-4-methylphenyl], [BA 259; 2, 6-difluoro-4-methylphenyl], [BA 260; 2, 3, 5-trifluoro-4-methylphenyl], [BA 261; , 6-trifluoro-4-methylphenyl], [BA262; 2,3,5,6-tetrafluoro-4-methylphenyl], [BA263; 2-fluoro-4-ethylphenyl], [BA 264; 3-fluoro-4-ethylphenyl], [BA 265; 2,3-difluoro-4-ethylphenyl], [BA 266; 2, 6-difluoro-4-ethylphenyl], [BA 267; 2, 5-difluoro -4-Ethylphenyl], [BA 268; 3,5-difluoro-4-ethylphenyl], [BA 269; 2,3,5-trifluoro-4-ethylphenyl], [BA 270; Fluoro-4-ethylphenyl], [BA 271; 2,3,5,6-tetrafluoro-4-ethylphenyl], [BA 272; 2-trifluoromethylphenyl], [BA 273; 3-trifluoromethylphenyl], [BA274; 4-trifluoromethylphenyl], [BA275; 4- (2,2,2-trifluoro-1-trifluoromethylethyl) phenyl], [BA276; 2-trifluoromethoxyphenyl], [BA277; 3-trifluoromethoxyphenyl], [BA 278; 4-trifluoromethoxyphenyl], [BA 279; 4- (2, 2-difluoroethoxy) phenyl], [BA 280; 4- (2, 2, 2- trifluoroethoxy) ) Phenyl], [BA 281; 2-nitrophenyl], [BA 282; [BA 283; 4-nitrophenyl], [BA 284; 2-cyanophenyl], [BA 285; 3-cyanophenyl], [BA 286; 4-cyanophenyl], [BA 287; 2-methyl-3-chlorophenyl] [BA 288; 2-methyl-4-chlorophenyl], [BA 289; 2-methyl-5-chlorophenyl], [BA 290; 2-methyl-6-chlorophenyl], [BA 291; 2-methyl-3-fluorophenyl], [BA292; 2-methyl-4-fluorophenyl], [BA293; 2-methyl-5-fluorophenyl], [BA294; 2-methyl-6-fluorophenyl], [BA295; 2-methyl-3-bromophenyl ], [BA 296; 2-methyl-4-bromophenyl], [BA 297; 2-methylthiophenyl], [BA 298; 3-methylthiophenyl], [BA 299; 4-methylthiophenyl], [BA 300; 2-methylsulfonylphenyl] ],

[BA301; 3-methylsulfonylphenyl], [BA302; 4-methylsulfonylphenyl], [BA303; 2-methylsulfinylphenyl], [BA304; 3-methylsulfinylphenyl], [BA305; 4-methylsulfinylphenyl], [BA306; 2-trifluoromethylthiophenyl], [BA307; 3-trifluoromethylthiophenyl], [BA308; 4-trifluoromethylthiophenyl], [BA309; 2-ethynylphenyl], [BA310; 3-ethynylphenyl] [BA311; 4-ethynylphenyl], [BA312; 2- (1-propynyl) phenyl], [BA313; 3- (1-propynyl) phenyl], [BA314; 4- (1-propynyl) phenyl], [BA BA315; 2-vinylphenyl], [BA316; 3-vinylphenyl], [BA317; 4-vinylphenyl], [BA318; 4- (2, 2- dichlorovinyl) phenyl], [BA 319; 2-Difluorovinyl) phenyl], [BA 320; cyclohexyl], [BA 321; 2-chlorocyclohexyl], [BA 322; 3-chlorocyclohexyl], [BA 323; 4-chlorocyclohexyl], [BA 32 4; 4, 4-dichlorocyclohexyl], [BA 325; 2-bromocyclohexyl], [BA 326; 3-bromocyclohexyl], [BA 327; 4-bromocyclohexyl], [BA 328; 4, 4-dibromocyclohexyl], [BA 329 2-iodocyclohexyl], [BA330; 3-iodocyclohexyl], [BA331; 4-iodocyclohexyl], [BA332; 2-fluorocyclohexyl], [BA333; 3-fluorocyclohexyl], [BA334; 4-fluorocyclohexyl ], [BA 335; 4, 4-difluorocyclohexyl], [BA 336; 4-methylcyclohexyl], [BA 337; 4-ethylcyclohexyl], [BA 338; 1-cyclohexenyl], [BA 339; 2-cyclohexenyl], [BA BA340; 3-cyclohexenyl], [BA341; 2-chloro-1-cyclohexenyl], [BA342; 3-chloro-1-cyclohexenyl], [BA343; 4-chloro-1-cyclohexenyl], [BA344; 5-chloro-1-cyclohexenyl], [BA 345; 6-chloro-1-cyclohexenyl], [BA 346; 1-chloro-2-cyclohexenyl], [BA 347; 2-chloro -2-cyclohexenyl], [BA 348; 3-chloro-2-cyclohexenyl], [BA 349; 4-chloro-2-cyclohexenyl], [BA 350; 5-chloro-2-cyclohexenyl], [BA 351; 6 -Chloro-2-cyclohexenyl], [BA352; 1-chloro-3-cyclohexenyl], [BA 353; 2-chloro-3-cyclohexenyl], [BA 354; 3-chloro-3-cyclohexenyl], [BA 355 4-chloro-3-cyclohexenyl], [BA 356; 5-chloro-3-cyclohexenyl], [BA 357; 6-chloro-3-cyclohexenyl], [BA 358; 4-bromo-1-cyclohexenyl], [BA 359; 4-bromo-2-cyclohexenyl], [BA 360; 4-bromo-3-cyclohexenyl], [BA 361; 4-methyl-1-cyclohexenyl], [BA 362; 4-methyl-2-cyclohexenyl ], [BA 363; 4-methyl-3-cyclohexenyl], [BA 364; 4-ethyl-1-cyclohexenyl], [BA 365; 4-ethyl-2-cyclohexenyl], [BA 366; Cyclohexenyl], [BA 367; trifluoromethyl], [BA 368; t-butyl], [BA 369; 4- (2- (2-meth) Xyethoxy) ethoxy) phenyl], [BA370; 4- (2-tetrahydropyranyloxy) phenyl], [BA 371; 4- (N, N-dimethylamino) sulfonyl) phenyl], [BA372; 1-naphthyl], [BA BA 373; 2-naphthyl], [BA 374; adamantan-1-yl], [BA 375; 3-methyladamantan-1-yl], [BA 376; 5-methyladamantan-1-yl], [BA 377; Dimethyladamantan-1-yl], [BA 378; 3,5-dimethyladamantan-1-yl], [BA 379; 3,5, 7-trimethyladamantan-1-yl], [BA 380; 5-methyladamantan-1-yl] [BA 381; 5,7-dimethyladamantan-1-yl], [BA 382; 3,5-dimethyladamantan-1-yl], [BA 383; 3,5, 7-trimethyladamantan-1-yl], [BA384; 2-Py], [BA 385; 3-F-2-Py], [BA 386; 4-Cl-3-F-2-Py], [BA 387; 5-Cl-3-F-2-Py ], [BA 388; 6-Cl-3-F-2-Py], [BA 389; 4-Me-3-F-2-Py], [BA 390; 5-Me-3-F-2-Py], [BA391; 6-Me-3 -F-2-Py], [BA392; 4-CF 3 -3-F-2-Py], [BA393; 5-CF 3 -3-F-2-Py], _{[BA394; 6-CF 3 -3} -F-2-Py], [BA395; 4-CN-3-F-2-Py], [BA396; 5-CN-3- F-2-Py !, [BA397; 6-CN-3-F-2-Py], [BA 398; 4-OMe-3-F-2-Py], [BA 399; 5-OMe-3-F- 2-Py], [BA 400; 6-OMe-3-F-2-Py], [BA 401; 4-F-2-Py], [BA 402; 3-Cl-4-F-2-Py], [BA BA403; 5-Cl-4-F-2-Py], [BA404; 6-Cl-4-F-2-Py], [BA405; 3-Me-4-F-2-Py], [BA406; 5-Me-4-F-2-Py !, [BA 407; 6-Me-4-F-2-Py], [BA 408; 3-CF ₃ -4-F-2-Py], [BA 409; _{-CF 3 -4-F-2-} Py], [BA410; 6-CF 3 -4-F-2-Py], [BA411; 3-CN-4-F-2-Py], [BA412; 5 -CN-4-F-2-Py], [BA413; 6-CN-4-F-2-Py], [BA414; 3-OMe-4-F-2-Py], [BA415; 5-OMe -4-F-2-Py !, [BA 416; 6-OMe-4-F-2-Py], [BA 417; 5-F-2-Py], [BA 418; 3-Cl-5-F-2 -Py], [BA419; 4-Cl-5-F-2-Py], [BA420; 6-Cl-5-F-2-Py], [BA421; 3-Me-5-F-2-Py ], [BA 422; 4-Me-5-F-2-Py], [BA 423; 6-Me-5-F-2-Py], [BA 424; 3-CF ₃ -5-F-2-Py] _{, [BA425; 4-CF 3} -5-F-2-Py], [BA426; 6-CF 3 -5-F-2-Py], [BA427; 3-CN-5-F-2-Py] , [BA428; 4-CN-5-F-2-Py], [BA429; 6-CN-5-F-2-Py], [BA 430; 3-OMe-5-F-2-Py], [BA 428; BA 431; 4-OMe-5-F-2-Py], [BA 432; 6-OMe-5-F-2-Py], [BA 433; 6-F-2-Py], [BA 434; 3-Cl- 6-F-2-Py, [BA 435; 4-Cl-6-F-2-Py], [BA 436; 5-Cl-6-F-2-Py], [BA 437; F-2-Py], [ BA438; 4-Me-6-F-2-Py], [BA439; 5-Me-6-F-2-Py], [BA440; 3-CF 3 -6-F -2-Py], [BA 441; 4- _{CF 3 -6-F-2-} Py], [BA442; 5-CF 3 -6-F-2-Py], [BA443; 3-CN-6-F-2-Py], [BA444; 4- CN-6-F-2-Py], [BA445; 5-CN-6-F-2-Py], [BA446; 3-OMe-6-F-2-Py], [BA 447; 4-OMe- 6-F-2-Py], [BA448; 5-OMe-6-F-2-Py], [BA449; 3-Cl-2-Py], [BA450; 4-Cl-3-Cl-2-] Py], [BA 451; 5-Cl-3-Cl-2-Py], [BA 452; 6-Cl-3-Cl-2-Py], [BA 453; 4-Me-3-Cl-2-Py] [BA 454; 5-Me-3-Cl-2-Py], [BA 455; 6-Me-3-Cl-2-Py], [BA 456; 4-CF ₃ -3-Cl-2-Py], _{[BA457; 5-CF 3 -3} -Cl-2-Py], [BA458; 6-CF 3 -3-Cl-2-Py], [BA459; 4-CN-3-Cl-2-Py], [BA 460; 5-CN-3-Cl-2-Py], [BA 461; 6-CN-3-Cl-2-Py], [BA 462; 4-OMe-3-Cl-2-Py], [BA 463] 5-OMe-3-Cl-2-Py !, [BA464; 6-OMe-3-Cl-2-Py], [BA465; 4-Cl-2-Py], [BA466; 3-Cl-4 -Cl-2-Py], [BA 467; 5-Cl-4-Cl-2-Py], [BA 468; 6-Cl-4-Cl-2-Py], [BA 469; 3-Me-4-Cl -2-Py], [BA 470; 5-Me-4-Cl-2-Py], [BA 471; 6-Me-4-Cl-2-Py], [BA 472; 3-CF ₃ -4-Cl- 2-Py], [BA473; 5-CF 3 -4-Cl-2-Py], [BA474; 6-CF 3 -4-Cl-2-Py], [BA475; 3-CN-4-Cl- 2-Py], [BA 476; 5-CN-4-Cl-2-Py], [BA 477; 6-CN-4-Cl-2-Py], [BA 478; 3-OMe-4-Cl-2- Py], [BA 479; 5-OMe-4-Cl-2-Py], [BA 480; 6-OMe-4-Cl-2-Py], [BA 481; 5-Cl-2-Py], [BA 482; 4-Cl-5-Cl-2-Py], [BA 483; 5-Cl-5-Cl-2-Py], [BA 484; 6-C l-5-Cl-2-Py],

[BA 485; 4-Me-5-Cl-2-Py], [BA 486; 5-Me-5-Cl-2-Py], [BA 487; 6-Me-5-Cl-2-Py], [BA 488] _{; 4-CF 3 -5-Cl} -2-Py], [BA489; 5-CF 3 -5-Cl-2-Py], [BA490; 6-CF 3 -5-Cl-2-Py], [ BA 491; 4-CN-5-Cl-2-Py], [BA 492; 3-CN-5-Cl-2-Py], [BA 493; 6-CN-5-Cl-2-Py], [BA 494; 4-OMe-5-Cl-2-Py, [BA 495; 5-OMe-5-Cl-2-Py], [BA 496; 6-OMe-5-Cl-2-Py], [BA 497; 6- Cl-2-Py !, [BA 498; 3-Cl-6-Cl-2-Py], [BA 499; 4-Cl-6-Cl-2-Py], [BA 500; 5-Cl-6-Cl- 2-Py], [BA501; 3-Me-6-Cl-2-Py], [BA502; 4-Me-6-Cl-2-Py], [BA 503; 5-Me-6-Cl-2- Py], [BA504; 3- CF 3 -6-Cl-2-Py], [BA505; 4-CF 3 -6-Cl-2-Py], [BA506; 5-CF 3 -6-Cl-2 -Py], [BA507; 3-CN-6-Cl-2-Py], [BA508; 4-CN-6-Cl-2-Py], [BA509; 5-CN-6-Cl-2-Py ], [BA510; 3-OMe-6-Cl-2-Py], [BA511; 4-OMe-6-Cl-2-Py], [BA512; 5-OMe-6-Cl-2-Py], [BA 513; 3-Br-2-Py], [BA 514; 4-Cl-3-Br-2-Py], [BA 515; 5-Cl-3-Br-2-Py], [BA 516; 6-Cl -3-Br-2-Py, [BA 517; 4-Me-3-Br-2-Py], [BA 518; 5-Me-3-Br-2-Py], [BA 519; 6-Me-3 -Br-2-Py], [ BA520; 4-CF 3 -3-Br-2-Py], [BA521; 5-CF 3 -3-Br-2-Py], [BA522; 6-CF 3 - 3-Br-2-Py], [BA523; 4-CN-3-Br-2-Py], [BA524; 5-CN-3-Br-2-Py], [BA525; 6-CN-3- Br-2-Py, [BA 526; 4-OMe-3-Br-2-Py], [BA 527; 5-O Me-3-Br-2-Py], [BA 528; 6-OMe-3-Br-2-Py], [BA 529; 4-Br-2-Py], [BA 530; 3-Cl-4-Br- 2-Py], [BA 531; 5-Cl-4-Br-2-Py], [BA 532; 6-Cl-4-Br-2-Py], [BA 533; 3-Me-4-Br-2- Py], [BA534; 5- Me-4-Br-2-Py], [BA535; 6-Me-4-Br-2-Py], [BA536; 3-CF 3 -4-Br-2-Py ], [BA 537; 5-CF ₃ 4-Br-2-Py], [BA 538; 6-CF ₃ 4-Br-2-Py], [BA 539; 3-CN-4-Br-2-Py] ], [BA540; 5-CN-4-Br-2-Py], [BA 541; 6-CN-4-Br-2-Py], [BA 542; 3-OMe-4-Br-2-Py], [BA543; 5-OMe-4-Br-2-Py], [BA544; 6-OMe-4-Br-2-Py], [BA545; 5-Br-2-Py], [BA546; -5-Br-2-Py, [BA547; 4-Cl-5-Br-2-Py], [BA 548; 6-Cl-5-Br-2-Py], [BA 549; 3-Me-5 -Br-2-Py, [BA550; 4-Me-5-Br-2-Py], [BA 551; 6-Me-5-Br-2-Py], [BA 552; 3-CF ₃ -5] Br-2-Py], [ BA553; 4-CF 3 -5-Br-2-Py], [BA554; 6-CF 3 -5-Br-2-Py], [BA555; 3-CN-5- Br-2-Py, [BA 556; 4-CN-5-Br-2-Py], [BA 557; 6-CN-5-Br-2-Py], [BA 558; 3-OMe-5-Br- 2-Py], [BA559; 4-OMe-5-Br-2-Py], [BA 560; 6-OMe-5-Br-2-Py], [BA 561; 6-Br-2-Py], BA 562; 3-Cl-6-Br-2-Py !, [BA 563; 4-Cl-6-Br-2-Py], [BA 564; 5-Cl-6-Br-2-Py], [BA 565; 3-Me-6-Br-2-Py], [BA566; 4-Me-6-Br-2-Py], [BA567; 5-Me-6-Br-2-Py], [BA568; 3- _{CF 3 -6-Br-2-} Py], [BA569; 4-CF 3 -6-Br-2-Py], [BA5 _{70; 5-CF 3 -6-} Br-2-Py], [BA571; 3-CN-6-Br-2-Py], [BA572; 4-CN-6-Br-2-Py], [BA573 5-CN-6-Br-2-Py !, [BA574; 3-OMe-6-Br-2-Py], [BA575; 4-OMe-6-Br-2-Py], [BA576; -OMe-6-Br-2-Py], [BA577; 3-I-2-Py], [BA 578; 4-Cl-3-I-2-Py], [BA 579; 5-Cl-3-I -2-Py !, [BA 580; 6-Cl-3-I-2-Py], [BA 581; 4-Me-3-I-2-Py], [BA 582; 5-Me-3-I-2 -Py], [BA583; 6- Me-3-I-2-Py], [BA584; 4-CF 3 -3-I-2-Py],

_{[BA585; 5-CF 3 -3} -I-2-Py], [BA586; 6-CF 3 -3-I-2-Py], [BA587; 4-CN-3-I-2-Py], [BA 588; 5-CN-3-I-2-Py], [BA 589; 6-CN-3-I-2-Py], [BA 590; 4-OMe-3-I-2-Py], [BA 591 5-OMe-3-I-2-Py !, [BA592; 6-OMe-3-I-2-Py], [BA593; 4-I-2-Py], [BA 594; 3-Cl-4 -I-2-Py, [BA 595; 5-Cl-4-I-2-Py], [BA 596; 6-Cl-4-I-2-Py], [BA 597; 3-Me-4-I -2-Py], [BA598; 5-Me-4-I-2-Py], [BA599; 6-Me-4-I-2-Py], [BA600; 3-CF ₃ -4-I- 2-Py], [BA601; 5-CF 3 -4-I-2-Py], [BA602; 6-CF 3 -4-I-2-Py], [BA603; 3-CN-4-I- 2-Py], [BA604; 5-CN-4-I-2-Py], [BA605; 6-CN-4-I-2-Py], [BA606; 3-OMe-4-I-2-] Py], [BA 607; 5-OMe-4-I-2-Py], [BA 608; 6-OMe-4-I-2-Py], [BA 609; 5-I-2-Py], [BA 610; 3-Cl-5-I-2-Py], [BA611; 4-Cl-5-I-2-Py], [BA612; 6-Cl-5-I-2-Py], [BA613; Me-5-I-2-Py, [BA 614; 4-Me-5-I-2-Py], [BA 615; 6-Me-5-I-2-Py], [BA 616; 3-CF ₃ -5-I-2-Py], [BA 617; 4-CF ₃ -5-I-2-Py], [BA 618; 6-CF ₃ -5-I-2-Py], [BA 619; 3-CN -5-I-2-Py, [BA620; 4-CN-5-I-2-Py], [BA 621; 6-CN-5-I-2-Py], [BA 622; 3-OMe-5 -I-2-Py, [BA 623; 4-OMe-5-I-2-Py], [BA 624; 6-OMe-5-I-2-Py], [BA 625; 6-I-2-Py [BA 626; 3-Cl-6-I-2-Py], [BA 627; 4-Cl-6-I-2-Py], [BA 628; 5-Cl-6-I-2-Py], [BA 629; 3-Me-6- I-2-Py], [BA630; 4-Me-6-I-2-Py], [BA631; 5-Me-6-I-2-Py], [BA632; 3-CF ₃ -6-I -2-Py], [BA633; 4-CF 3 -6-I-2-Py], [BA634; 5-CF 3 -6-I-2-Py], [BA635; 3-CN-6-I -2-Py, [BA 636; 4-CN-6-I-2-Py], [BA 637; 5-CN-6-I-2-Py], [BA 638; 3-OMe-6-I-2 -Py], [BA639; 4-OMe-6-I-2-Py], [BA640; 5-OMe-6-I-2-Py], [BA641; 3-Me-2-Py], [BA642] 4-Cl-3-Me-2-Py !, [BA643; 5-Cl-3-Me-2-Py], [BA 644; 6-Cl-3-Me-2-Py], [BA 645; -Me-3-Me-2-Py], [BA646; 5-Me-3-Me-2-Py], [BA647; 6-Me-3-Me-2-Py], [BA 648; 4-CF _{3 -3-Me-2-Py} ], [BA649; 5-CF 3 -3-Me-2-Py], [BA650; 6-CF 3 -3-Me-2-Py], [BA651; 4- CN-3-Me-2-Py !, [BA 652; 5-CN-3-Me-2-Py], [BA 653; 6-CN-3-Me-2-Py], [BA 654; 4-OMe- 3-Me-2-Py], [BA655; 5-OMe-3-Me-2-Py], [BA656; 6-OMe-3-Me-2-Py], [BA657; 4-Me-2- Py], [BA658; 3-Cl-4-Me-2-Py], [BA659; 5-Cl-4-Me-2-Py], [BA 660; 6-Cl-4-Me-2-Py] [BA 661; 3-Me-4-Me-2-Py], [BA 662; 5-Me-4-Me-2-Py], [BA 663; 6-Me-4-Me-2-Py], [BA 662; _{BA664; 3-CF 3 -4-} Me-2-Py], [BA665; 5-CF 3 -4-Me-2-Py], [BA666; 6-CF 3 -4-Me-2-Py], [BA 667; 3-CN-4-Me-2-Py], [BA 668; 5-CN-4-Me-2-Py], [BA 669; 6-CN-4-Me-2-Py], [BA 670] 3-OMe-4-Me-2-Py], [BA 671; 5-OMe-4-Me-2-Py], [BA 672; 6-OMe -4-Me-2-Py], [BA 673; 5-Me-2-Py], [BA 674; 3-Cl-5-Me-2-Py], [BA 675; 4-Cl-5-Me-2 -Py], [BA 676; 6-Cl-5-Me-2-Py], [BA 677; 3-Me-5-Me-2-Py], [BA 678; 4-Me-5-Me-2-Py ], [BA679; 6-Me -5-Me-2-Py], [BA680; 3-CF 3 -5-Me-2-Py], [BA681; 4-CF 3 -5-Me-2-Py ], [BA682; 6-CF 3 -5-Me-2-Py], [BA683; 3-CN-5-Me-2-Py], [BA684; 4-CN-5-Me-2-Py] ,

[BA 685; 6-CN-5-Me-2-Py], [BA 686; 3-OMe-5-Me-2-Py], [BA 687; 4-OMe-5-Me-2-Py], [BA 688] 6-OMe-5-Me-2-Py !, [BA 689; 6-Me-2-Py], [BA 690; 3-Cl-6-Me-2-Py], [BA 691; 4-Cl-6 -Me-2-Py], [BA692; 5-Cl-6-Me-2-Py], [BA693; 3-Me-6-Me-2-Py], [BA 694; 4-Me-6-Me -2-Py], [BA695; 5-Me-6-Me-2-Py], [BA696; 3-CF 3 -6-Me-2-Py], [BA697; 4-CF 3 -6-Me -2-Py !, [BA 698; 5-CF ₃ -6-Me-2-Py], [BA 699; 3-CN-6-Me-2-Py], [BA 700; 4-CN-6-Me- 2-Py], [BA 701; 5-CN-6-Me-2-Py], [BA 702; 3-OMe-6-Me-2-Py], [BA 703; 4-OMe-6-Me-2- 2 Py], [BA704; 5-OMe-6-Me-2-Py], [BA705; 3-OMe-2-Py], [BA706; 4-Cl-3-OMe-2-Py], [BA707; 5-Cl-3-OMe-2-Py, [BA 708; 6-Cl-3-OMe-2-Py], [BA 709; 4-Me-3-OMe-2-Py], [BA 710; Me-3-OMe-2- Py], [BA711; 6-Me-3-OMe-2-Py], [BA712; 4-CF 3 -3-OMe-2-Py], [BA713; 5-CF _{3 -3-OMe-2-Py} ], [BA714; 6-CF 3 -3-OMe-2-Py], [BA715; 4-CN-3-OMe-2-Py], [BA716; 5-CN -3-OMe-2-Py !, [BA717; 6-CN-3-OMe-2-Py], [BA718; 4-OMe-3-OMe-2-Py], [BA719; 5-OMe-3 6-OMe-2-Py !, [BA 720; 6-OMe-3-OMe-2-Py], [BA 721; 4-OMe-2-Py], [BA 722; 3-Cl-4-OMe-2-Py] ], [BA723; 5-Cl-4-OMe-2-Py], [BA724; 6-Cl-4-OMe-2-Py], [BA725; 3-Me-4-OMe-2-Py], [BA 726; 5-Me-4-OMe-2-Py], [BA727; 6-Me-4 -OMe-2-Py], [BA728; 3-CF 3 -4-OMe-2-Py], [BA729; 5-CF 3 -4-OMe-2-Py], _{[BA730; 6-CF 3 -4} -OMe-2-Py], [BA731; 3-CN-4-OMe-2-Py], [BA732; 5-CN-4-OMe-2-Py], [ BA733; 6-CN-4-OMe-2-Py], [BA734; 3-OMe-4-OMe-2-Py], [BA735; 5-OMe-4-OMe-2-Py], [BA736; 6-OMe-4-OMe-2-Py], [BA 737; 5-OMe-2-Py], [BA 738; 3-Cl-5-OMe-2-Py], [BA 739; 4-Cl-5- OMe-2-Py, [BA 740; 6-Cl-5-OMe-2-Py], [BA 741; 3-Me-5-OMe-2-Py], [BA 742; 4-Me-5-OMe- 2-Py], [BA743; 6-Me-5-OMe-2-Py], [BA744; 3-CF 3 -5-OMe-2-Py], [BA745; 4-CF 3 -5-OMe- 2-Py], [BA746; 6-CF 3 -5-OMe-2-Py], [BA747; 3-CN-5-OMe-2-Py], [BA748; 4-CN-5-OMe-2 -Py], [BA 749; 6-CN-5-OMe-2-Py], [BA 750; 3-OMe-5-OMe-2-Py], [BA 751; 4-OMe-5-OMe-2-Py ], [BA752; 6-OMe-5-OMe-2-Py], [BA753; 6-OMe-2-Py], [BA754; 3-Cl-6-OMe-2-Py], [BA755; 4] -Cl-6-OMe-2-Py], [BA756; 5-Cl-6-OMe-2-Py], [BA757; 3-Me-6-OMe-2-Py], [BA758; 4-Me -6-OMe-2-Py] , [BA759; 5-Me-6-OMe-2-Py], [BA760; 3-CF 3 -6-OMe-2-Py], [BA761; 4-CF 3 -6-OMe-2-Py] , [BA762; 5-CF 3 -6-OMe-2-Py], [BA763; 3-CN-6-OMe-2-Py], [BA764; 4-CN- 6-OMe-2-Py], [BA765; 5-CN-6-OMe-2-Py], [BA766; 3-OMe-6-OMe-2-Py], [BA767; 4-OMe-6- O Me-2-Py], [ BA768; 5-OMe-6-OMe-2-Py], [BA769; 3-CF 3 -2-Py], [BA770; 4-Cl-3-CF 3 -2- Py], [BA771; 5- Cl-3-CF 3 -2-Py], [BA772; 6-Cl-3-CF 3 -2-Py], [BA773; 4-Me-3-CF 3 -2 5-Py], [BA 774; 5-Me-3-CF ₃ -2-Py], [BA 775; 6-Me-3-CF ₃ -2-Py], [BA 776; 4-CF ₃ -3-CF ₃ -2-Py], [BA 777; 5-CF ₃ -3-CF ₃ -2-Py], [BA 778; 6-CF ₃ -3-CF ₃ -2-Py], [BA 779; 4-CN-3 _{-CF 3 -2-Py], [} BA780; 5-CN-3-CF 3 -2-Py], [BA781; 6-CN-3-CF 3 -2-Py], [BA782; 4-OMe- _{3-CF 3 -2-Py]} , [BA783; 5-OMe-3-CF 3 -2-Py], [BA784; 6-OMe-3-CF 3 -2-Py],

_{[BA785; 4-CF 3 -2} -Py], [BA786; 3-Cl-4-CF 3 -2-Py], [BA787; 5-Cl-4-CF 3 -2-Py], [BA788; _{6-Cl-4-CF 3} -2-Py], [BA789; 3-Me-4-CF 3 -2-Py], [BA790; 5-Me-4-CF 3 -2-Py], [BA791 ; 6-Me-4-CF 3 -2-Py], [BA792; 3-CF 3 -4-CF 3 -2-Py], [BA793; 5-CF 3 -4-CF 3 -2-Py] _{, [BA794; 6-CF 3} -4-CF 3 -2-Py], [BA795; 3-CN-4-CF 3 -2-Py], [BA796; 5-CN-4-CF 3 -2- Py], [BA797; 6- CN-4-CF 3 -2-Py], [BA798; 3-OMe-4-CF 3 -2-Py], [BA799; 5-OMe-4-CF 3 -2 -Py], [BA800; 6- OMe-4-CF 3 -2-Py], [BA801; 5-CF 3 -2-Py], [BA802; 3-Cl-5-CF 3 -2-Py] , [BA 803; 4-Cl-5-CF ₃ -2-Py], [BA 804; 6-Cl -5-CF ₃ -2-Py], [BA 805; 3-Me -5-CF ₃ -2-Py ], [BA806; 4-Me -5-CF 3 -2-Py], [BA807; 6-Me-5-CF 3 -2-Py], [BA808; 3-CF 3 -5-CF 3 -2 4-Py], [BA 809; 4-CF ₃ -5-CF ₃ -2-Py], [BA 810; 6-CF ₃ -5-CF ₃ -2-Py], [BA 811; 3-CN -5- CF _{3 -2-Py], [BA812} ; 4-CN-5-CF 3 -2-Py], [BA813; 6-CN-5-CF 3 -2-Py], [BA814; 3-OMe-5- CF ₃ -2-Py !, [BA 815; 4-OMe-5-CF ₃ -2-Py], [BA 816; 6-OMe -5-CF ₃ -2-Py], [BA 817; 6-CF _3- 2-Py], [BA818; 3-Cl-6-CF 3 -2-Py], [BA819; 4-Cl-6-CF 3 -2-Py], [BA820; 5-Cl-6-CF 3 -2-Py !, [BA 821; 3-Me-6-CF ₃ -2-Py], [BA 822; 4-Me-6-CF ₃ -2-Py], [BA 2 823; 5-Me-6- CF 3 -2-Py], [BA824; 3-CF 3 -6-CF 3 -2-Py], [BA825; 4-CF 3 -6-CF 3 -2-Py ], [BA826; 5-CF 3 -6-CF 3 -2-Py], [BA827; 3-CN-6-CF 3 -2-Py], [BA828; 4-CN-6-CF 3 -2 -Py], [BA829; 5- CN-6-CF 3 -2-Py], [BA830; 3-OMe-6-CF 3 -2-Py], [BA831; 4-OMe-6-CF 3 - 2-Py], [BA 832; 5-OMe-6-CF ₃ -2-Py], [BA 833; 3-OCF ₃ -2-Py], [BA 834; 4-Cl-3-OCF ₃ -2-Py ], [BA835; 5-Cl -3-OCF 3 -2-Py], [BA836; 6-Cl-3-OCF 3 -2-Py], [BA837; 4-Me-3-OCF 3 -2- Py], [BA838; 5- Me-3-OCF 3 -2-Py], [BA839; 6-Me-3-OCF 3 -2-Py], [BA840; 4-CF 3 -3-OCF 3 - 2-Py], [BA 841; 5-CF ₃ -3-OCF ₃ -2-Py], [BA 842; 6-CF ₃ -3-OCF ₃ -2-Py], [BA 843; OCF ₃ -2-Py !, [BA 844; 5-CN-3-OCF ₃ -2-Py], [BA 845; 6-CN -3-OCF ₃ -2-Py], [BA 846; 4-OMe-3] _{-OCF 3 -2-Py], [} BA847; 5-OMe-3-OCF 3 -2-Py], [BA848; 6-OMe-3-OCF 3 -2-Py], [BA849; 4-OCF 3 -2-Py], [BA850; 3-Cl-4-OCF 3 -2-Py], [BA851; 5-Cl-4-OCF 3 -2-Py], [BA852; 6-Cl-4-OCF _{3 -2-Py], [BA853} ; 3-Me-4-OCF 3 -2-Py], [BA854; 5-Me-4-OCF 3 -2-Py], [BA855; 6-Me-4- OCF ₃ -2-Py, [BA 856; 3-CF ₃ -4-OCF ₃ -2-Py], [BA 857; 5-CF ₃ -4-OCF ₃ -2-Py], [BA 858; 6-CF ₃ -4-OCF ₃ -2-Py, [BA 859; 3-CN -4-OCF _{3 -2-Py], [BA860} ; 5-CN-4-OCF 3 -2-Py], [BA861; 6-CN-4-OCF 3 -2-Py], [BA862; 3-OMe-4- _{OCF 3 -2-Py], [} BA863; 5-OMe-4-OCF 3 -2-Py], [BA864; 6-OMe-4-OCF 3 -2-Py], [BA865; 5-OCF 3 - 2-Py], [BA866; 3-Cl-5-OCF 3 -2-Py], [BA867; 4-Cl-5-OCF 3 -2-Py], [BA868; 6-Cl-5-OCF 3 -2-Py], [BA869; 3-Me-5-OCF 3 -2-Py], [BA870; 4-Me-5-OCF 3 -2-Py], [BA871; 6-Me-5-OCF _{3 -2-Py], [BA872} ; 3-CF 3 -5-OCF 3 -2-Py], [BA873; 4-CF 3 -5-OCF 3 -2-Py], [BA874; 6-CF 3 _{-5-OCF 3 -2-Py]} , [BA875; 3-CN-5-OCF 3 -2-Py], [BA876; 4-CN-5-OCF 3 -2-Py], [BA877; 6- _{CN-5-OCF 3 -2-} Py], [BA878; 3-OMe-5-OCF 3 -2-Py], [BA879; 4-OMe-5-OCF 3 -2-Py], [BA880; 6 _{-OMe-5-OCF 3 -2-} Py], [BA881; 6-OCF 3 -2-Py], [BA882; 3-Cl-6-OCF 3 -2-Py], [BA883; 4-Cl- _{6-OCF 3 -2-Py]} , [BA884; 5-Cl-6-OCF 3 -2-Py],

[BA885; 3-Me-6 -OCF 3 -2-Py], [BA886; 4-Me-6-OCF 3 -2-Py], [BA887; 5-Me-6-OCF 3 -2-Py] , [BA 888; 3-CF ₃ -6-OCF ₃ -2-Py], [BA 889; 4-CF ₃ -6-OCF ₃ -2-Py], [BA 890; 5-CF ₃ -6-OCF _3- 2-Py], [BA891; 3-CN-6-OCF 3 -2-Py], [BA892; 4-CN-6-OCF 3 -2-Py], [BA893; 5-CN-6-OCF 3 -2-Py], [BA 894; 3-OMe-6-OCF ₃ -2-Py], [BA 895; 4-OMe-6-OCF ₃ -2-Py], [BA 896; 5-OMe -6- OCF _{3 -2-Py], [BA897} ; 3-CHF 2 -2-Py], [BA898; 4-Cl-3-CHF 2 -2-Py], [BA899; 5-Cl-3-CHF 2 -2 -Py], [BA900; 6- Cl-3-CHF 2 -2-Py], [BA901; 4-Me-3-CHF 2 -2-Py], [BA902; 5-Me-3-CHF 2 - 2-Py], [BA903; 6-Me-3-CHF 2 -2-Py], [BA904; 4-CF 3 -3-CHF 2 -2-Py], [BA905; 5-CF 3 -3- _{CHF 2 -2-Py], [} BA906; 6-CF 3 -3-CHF 2 -2-Py], [BA907; 4-CN-3-CHF 2 -2-Py], [BA908; 5-CN- _{3-CHF 2 -2-Py]} , [BA909; 6-CN-3-CHF 2 -2-Py], [BA910; 4-OMe-3-CHF 2 -2-Py], [BA911; 5-OMe _{-3-CHF 2 -2-Py]} , [BA912; 6-OMe-3-CHF 2 -2-Py], [BA913; 4-CHF 2 -2-Py], [BA914; 3-Cl-4- _{CHF 2 -2-Py], [} BA915; 5-Cl-4-CHF 2 -2-Py], [BA916; 6-Cl-4-CHF 2 -2-Py], [BA917; 3-Me-4 _{-CHF 2 -2-Py], [} BA918; 5-Me-4-CHF 2 -2-Py], [BA919; 6-Me-4-CHF 2 -2-Py], [BA920; 3-CF 3 -4-CHF ₂ -2-Py], [BA 921; 5-CF ₃ -4-CHF ₂ -2-Py], [BA 922; 6-CF ₃ -4-CHF ₂ -2-Py], [BA 923; 3-CN-4-CHF ₂ -2-Py], [BA 924; _{5-CN-4-CHF 2} -2-Py], [BA925; 6-CN-4-CHF 2 -2-Py], [BA926; 3-OMe-4-CHF 2 -2-Py], [BA927 ; 5-OMe-4-CHF 2 -2-Py], [BA928; 6-OMe-4-CHF 2 -2-Py], [BA929; 5-CHF 2 -2-Py], [BA930; 3- _{Cl-5-CHF 2 -2-} Py], [BA931; 4-Cl-5-CHF 2 -2-Py], [BA932; 6-Cl-5-CHF 2 -2-Py], [BA933; 3 _{-Me-5-CHF 2 -2-} Py], [BA934; 4-Me-5-CHF 2 -2-Py], [BA935; 6-Me-5-CHF 2 -2-Py], [BA936; _{3-CF 3 -5-CHF 2} -2-Py], [BA937; 4-CF 3 -5-CHF 2 -2-Py], [BA938; 6-CF 3 -5-CHF 2 -2-Py] , [BA 939; 3-CN-5-CHF ₂ -2-Py], [BA 940; 4-CN -5-CHF ₂ -2-Py], [BA 941; 6-CN -5-CHF ₂ -2-Py ], [BA942; 3-OMe -5-CHF 2 -2-Py], [BA943; 4-OMe-5-CHF 2 -2-Py], [BA944; 6-OMe-5-CHF 2 -2- Py], [BA 945; 6-CHF ₂ -2-Py], [BA 946; 3-Cl-6-CHF ₂ -2-Py], [BA 947; 4-Cl -6-CHF ₂ -2-Py], [BA948; 5-Cl-6 -CHF 2 -2-Py], [BA949; 3-Me-6-CHF 2 -2-Py], [BA950; 4-Me-6-CHF 2 -2-Py] , [BA951; 5-Me- 6-CHF 2 -2-Py], [BA952; 3-CF 3 -6-CHF 2 -2-Py], [BA953; 4-CF 3 -6-CHF 2 -2 -Py], [BA954; 5- CF 3 -6-CHF 2 -2-Py], [BA955; 3-CN-6-CHF 2 -2-Py], [BA956; 4-CN-6-CHF 2 -2-Py], [BA 957; 5-CN-6-CHF ₂ -2-Py], [BA958; 3-OMe-6-CHF 2 -2-Py], [BA959; 4-OMe-6-CHF 2 -2-Py], [BA960; 5-OMe-6-CHF _{2 -2-Py], [BA961} ; 3-OCHF 2 -2-Py], [BA962; 4-Cl-3-OCHF 2 -2-Py], [BA963; 5-Cl-3-OCHF 2 -2 -Py], [BA964; 6- Cl-3-OCHF 2 -2-Py], [BA965; 4-Me-3-OCHF 2 -2-Py], [BA966; 5-Me-3-OCHF 2 - 2-Py], [BA967; 6-Me-3-OCHF ₂ -2-Py], [BA 968; 4-CF ₃ -3-OCHF ₂ -2-Py], [BA 969; 5-CF ₃ -3- _{OCHF 2 -2-Py], [} BA970; 6-CF 3 -3-OCHF 2 -2-Py], [BA971; 4-CN-3-OCHF 2 -2-Py], [BA972; 5-CN- 3-OCHF ₂ -2-Py], [BA 973; 6-CN -3-OCHF ₂ -2-Py], [BA 974; 4-OMe -3-OCHF ₂ -2-Py], [BA 975; _{-3-OCHF 2 -2-Py]} , [BA976; 6-OMe-3-OCHF 2 -2-Py], [BA977; 4-OCHF 2 -2-Py], [BA978; 3-Cl-4- _{OCHF 2 -2-Py], [} BA979; 5-Cl-4-OCHF 2 -2-Py], [BA980; 6-Cl-4-OCHF 2 -2-Py], [BA981; 3-Me-4 _{-OCHF 2 -2-Py], [} BA982; 5-Me-4-OCHF 2 -2-Py], [BA983; 6-Me-4-OCHF 2 -2-Py], [BA984; 3-CF 3 -4-OCHF ₂ -2-Py],

_{[BA985; 5-CF 3 -4} -OCHF 2 -2-Py], [BA986; 6-CF 3 -4-OCHF 2 -2-Py], [BA987; 3-CN-4-OCHF 2 -2- Py], [BA988; 5- CN-4-OCHF 2 -2-Py], [BA989; 6-CN-4-OCHF 2 -2-Py], [BA990; 3-OMe-4-OCHF 2 -2 -Py], [BA991; 5- OMe-4-OCHF 2 -2-Py], [BA992; 6-OMe-4-OCHF 2 -2-Py], [BA993; 5-OCHF 2 -2-Py] , [BA994; 3-Cl-5-OCHF ₂ -2-Py], [BA 995; 4-Cl -5-OCHF ₂ -2-Py], [BA 996; 6-Cl -5-OCHF ₂ -2-Py ], [BA997; 3-Me -5-OCHF 2 -2-Py], [BA998; 4-Me-5-OCHF 2 -2-Py], [BA999; 6-Me-5-OCHF 2 -2- Py], [BA1000; 3- CF 3 -5-OCHF 2 -2-Py], [BA1001; 4-CF 3 -5-OCHF 2 -2-Py], [BA1002; 6-CF 3 -5-OCHF _{2 -2-Py], [BA1003} ; 3-CN-5-OCHF 2 -2-Py], [BA1004; 4-CN-5-OCHF 2 -2-Py], [BA1005; 6-CN-5- OCHF ₂ -2-Py, [BA 1006; 3-OMe-5-OCHF ₂ -2-Py], [BA 1007; 4-OMe -5-OCHF ₂ -2-Py], [BA 1008; 6-OMe-5 _{-OCHF 2 -2-Py], [} BA1009; 6-OCHF 2 -2-Py], [BA1010; 3-Cl-6-OCHF 2 -2-Py], [BA1011; 4-Cl-6-OCHF 2 -2-Py], [BA1012; 5-Cl-6-OCHF 2 -2-Py], [BA1013; 3-Me-6-OCHF 2 -2-Py], [BA1014; 4-Me-6-OCHF ₂ -2-Py !, [BA 1015; 5-Me-6-OCHF ₂ -2-Py], [BA 1016; 3-CF ₃ -6-OCHF ₂ -2-Py], [BA 1017; 4-CF _3- 6-OCHF ₂ -2-Py], [BA 1018; 5-CF ₃ -6-OCHF ₂ -2-Py], [BA 10 19; 3] _{-CN-6-OCHF 2 -2-} Py], [BA1020; 4-CN-6-OCHF 2 -2-Py], [BA1021; 5-CN-6-OCHF 2 -2-Py], [BA1022; _{3-OMe-6-OCHF 2} -2-Py], [BA1023; 4-OMe-6-OCHF 2 -2-Py], [BA1024; 5-OMe-6-OCHF 2 -2-Py], [BA1025 3-Et-2-Py !, [BA1026; 4-Cl-3-Et-2-Py], [BA1027; 5-Cl-3-Et-2-Py], [BA1028; 6-Cl-3 -Et-2-Py], [BA1029; 4-Me-3-Et-2-Py], [BA1030; 5-Me-3-Et-2-Py], [BA1031; 6-Me-3-Et] -2-Py], [BA1032; 4-CF 3 -3-Et-2-Py], [BA1033; 5-CF 3 -3-Et-2-Py], [BA1034; 6-CF 3 -3- Et-2-Py, [BA1035; 4-CN-3-Et-2-Py], [BA1036; 5-CN-3-Et-2-Py], [BA1037; 6-CN-3-Et- 2-Py], [BA1038; 4-OMe-3-Et-2-Py], [BA1039; 5-OMe-3-Et-2-Py], [BA1040; 6-OMe-3-Et-2- Py], [BA1041; 4-Et-2-Py], [BA1042; 3-Cl-4-Et-2-Py], [BA1043; 5-Cl-4-Et-2-Py], [BA1044; 6-Cl-4-Et-2-Py], [BA 1045; 3-Me-4-Et-2-Py], [BA 1046; 5-Me-4-Et-2-Py], [BA 1047; 6- Me-4-Et-2- Py], [BA1048; 3-CF 3 -4-Et-2-Py], [BA1049; 5-CF 3 -4-Et-2-Py], [BA1050; 6- _{CF 3 -4-Et-2-} Py], [BA1051; 3-CN-4-Et-2-Py], [BA1052; 5-CN-4-Et-2-Py], [BA1053; 6-CN -4-Et-2-Py], [BA1054; 3-OMe-4-Et-2-Py], [BA1055; 5-OMe-4-Et-2-Py], [BA1056; 6-OMe-4 -Et-2-Py], [BA1057; 5-Et-2-Py], [BA1058; 3-Cl-5-Et-2-Py], [BA1059] 4-Cl-5-Et-2-Py !, [BA1060; 6-Cl-5-Et-2-Py], [BA1061; 3-Me-5-Et-2-Py], [BA1062; -Me-5-Et-2- Py], [BA1063; 6-Me-5-Et-2-Py], [BA1064; 3-CF 3 -5-Et-2-Py], [BA1065; 4- _{CF 3 -5-Et-2-} Py], [BA1066; 6-CF 3 -5-Et-2-Py], [BA1067; 3-CN-5-Et-2-Py], [BA1068; 4- CN-5-Et-2-Py], [BA1069; 6-CN-5-Et-2-Py], [BA 1070; 3-OMe-5-Et-2-Py], [BA1071; 4-OMe- 5-Et-2-Py], [BA1072; 6-OMe-5-Et-2-Py], [BA1073; 6-Et-2-Py], [BA1074; 3-Cl-6-Et-2- Py], [BA 1075; 4-Cl-6-Et-2-Py], [BA 1076; 5-Cl-6-Et-2-Py], [BA 1077; 3-Me-6-Et-2-Py] , [BA1078; 4-Me-6-Et-2-Py], [BA1079; 5-Me-6-Et-2-Py], [BA 1080; 3-CF ₃ -6-Et-2-Py], _{[BA1081; 4-CF 3 -6} -Et-2-Py], [BA1082; 5-CF 3 -6-Et-2-Py], [BA1083; 3-CN-6-Et-2-Py], [BA1084; 4-CN-6-Et-2-Py],

[BA1085; 5-CN-6-Et-2-Py], [BA1086; 3-OMe-6-Et-2-Py], [BA1087; 4-OMe-6-Et-2-Py], [BA1088 ; 5-OMe-6-Et -2-Py], [BA1089; 3-CH 2 CF 3 -2-Py], [BA1090; 4-Cl-3-CH 2 CF 3 -2-Py], [BA1091 ; 5-Cl-3-CH 2 CF 3 -2-Py], [BA1092; 6-Cl-3-CH 2 CF 3 -2-Py], [BA1093; 4-Me-3-CH 2 CF 3 - 2-Py], [BA1094; 5-Me-3-CH 2 CF 3 -2-Py], [BA1095; 6-Me-3-CH 2 CF 3 -2-Py], [BA1096; 4-CF 3 -3-CH ₂ CF ₃ -2-Py, [BA 1097; 5-CF ₃ -3-CH ₂ CF ₃ -2-Py], [BA 1098; 6-CF ₃ -3-CH ₂ CF ₃ -2- Py], [BA1099; 4- CN-3-CH 2 CF 3 -2-Py], [BA1100; 5-CN-3-CH 2 CF 3 -2-Py], [BA1101; 6-CN-3- _{CH 2 CF 3 -2-Py]} , [BA1102; 4-OMe-3-CH 2 CF 3 -2-Py], [BA1103; 5-OMe-3-CH 2 CF 3 -2-Py], [BA1104 ; 6-OMe-3-CH 2 CF 3 -2-Py], [BA1105; 4-CH 2 CF 3 -2-Py], [BA1106; 3-Cl-4-CH 2 CF 3 -2-Py] , [BA1107; 5-Cl- 4-CH 2 CF 3 -2-Py], [BA1108; 6-Cl-4-CH 2 CF 3 -2-Py], [BA1109; 3-Me-4-CH 2 _{CF 3 -2-Py], [} BA1110; 5-Me-4-CH 2 CF 3 -2-Py], [BA1111; 6-Me-4-CH 2 CF 3 -2-Py], [BA1112; 3 _{-CF 3 -4-CH 2 CF 3} -2-Py], [BA1113; 5-CF 3 -4-CH 2 CF 3 -2-Py], [BA1114; 6-CF 3 -4-CH 2 CF 3 -2-Py], [BA 1115; 3-CN-4-CH ₂ CF ₃ -2-Py], [BA 1116; 5-CN-4-CH ₂ CF _3- 2-Py], [BA1117; 6-CN-4-CH 2 CF 3 -2-Py], [BA1118; 3-OMe-4-CH 2 CF 3 -2-Py], [BA1119; 5-OMe- _{4-CH 2 CF 3 -2-} Py], [BA1120; 6-OMe-4-CH 2 CF 3 -2-Py], [BA1121; 5-CH 2 CF 3 -2-Py], [BA1122; 3 _{-Cl-5-CH 2 CF 3} -2-Py], [BA1123; 4-Cl-5-CH 2 CF 3 -2-Py], [BA1124; 6-Cl-5-CH 2 CF 3 -2- Py], [BA1125; 3- Me-5-CH 2 CF 3 -2-Py], [BA1126; 4-Me-5-CH 2 CF 3 -2-Py], [BA1127; 6-Me-5- _{CH 2 CF 3 -2-Py]} , [BA1128; 3-CF 3 -5-CH 2 CF 3 -2-Py], [BA1129; 4-CF 3 -5-CH 2 CF 3 -2-Py], _{[BA1130; 6-CF 3 -5} -CH 2 CF 3 -2-Py], [BA1131; 3-CN-5-CH 2 CF 3 -2-Py], [BA1132; 4-CN-5-CH 2 _{CF 3 -2-Py], [} BA1133; 6-CN-5-CH 2 CF 3 -2-Py], [BA1134; 3-OMe-5-CH 2 CF 3 -2-Py], [BA1135; 4 _{-OMe-5-CH 2 CF 3} -2-Py], [BA1136; 6-OMe-5-CH 2 CF 3 -2-Py], [BA1137; 6-CH 2 CF 3 -2-Py], [ BA1138; 3-Cl-6- CH 2 CF 3 -2-Py], [BA1139; 4-Cl-6-CH 2 CF 3 -2-Py], [BA1140; 5-Cl-6-CH 2 CF 3 -2-Py], [BA1141; 3-Me-6-CH 2 CF 3 -2-Py], [BA1142; 4-Me-6-CH 2 CF 3 -2-Py], [BA1143; 5-Me -6-CH ₂ CF ₃ -2-Py, [BA 1144; 3-CF ₃ -6-CH ₂ CF ₃ -2-Py], [BA 1145; 4-CF ₃ -6-CH ₂ CF ₃ -2- Py], [BA1146; 5- CF 3 -6-CH 2 CF 3 -2-Py], [BA1147; 3-CN-6-CH 2 _{CF 3 -2-Py], [} BA1148; 4-CN-6-CH 2 CF 3 -2-Py], [BA1149; 5-CN-6-CH 2 CF 3 -2-Py], [BA1150; 3 _{-OMe-6-CH 2 CF 3} -2-Py], [BA1151; 4-OMe-6-CH 2 CF 3 -2-Py], [BA1152; 5-OMe-6-CH 2 CF 3 -2- Py], [BA1153; 3-OEt-2-Py], [BA1154; 4-Cl-3-OEt-2-Py], [BA1155; 5-Cl-3-OEt-2-Py], [BA1156; 6-Cl-3-OEt-2-Py, [BA1157; 4-Me-3-OEt-2-Py], [BA1158; 5-Me-3-OEt-2-Py], [BA1159; 6- Me-3-OEt-2- Py], [BA1160; 4-CF 3 -3-OEt-2-Py], [BA1161; 5-CF 3 -3-OEt-2-Py], [BA1162; 6- _{CF 3 -3-OEt-2-} Py], [BA1163; 4-CN-3-OEt-2-Py], [BA1164; 5-CN-3-OEt-2-Py], [BA1165; 6-CN -3-OEt-2-Py, [BA1166; 4-OMe-3-OEt-2-Py], [BA1167; 5-OMe-3-OEt-2-Py], [BA1168; 6-OMe-3 -OEt-2-Py, [BA1169; 4-OEt-2-Py], [BA1170; 3-Cl-4-OEt-2-Py], [BA1171; 5-Cl-4-OEt-2-Py ], [BA1172; 6-Cl-4-OEt-2-Py], [BA1173; 3-Me-4-OEt-2-Py], [BA1174; 5-Me-4-OEt-2-Py], [BA1175; 6-Me-4 -OEt-2-Py], [BA1176; 3-CF 3 -4-OEt-2-Py], [BA1177; 5-CF 3 -4-OEt-2-Py], _{[BA1178; 6-CF 3 -4} -OEt-2-Py], [BA1179; 3-CN-4-OEt-2-Py], [BA1180; 5-CN-4-OEt-2-Py], [ BA1181; 6-CN-4-OEt-2-Py], [BA1182; 3-OMe-4-OEt-2-Py], [BA1183; 5-OMe-4-OEt-2-Py], [BA1184; 6-OMe-4-OEt-2-Py],

[BA1185; 5-OEt-2-Py], [BA1186; 3-Cl-5-OEt-2-Py], [BA1187; 4-Cl-5-OEt-2-Py], [BA1188; 6-Cl -5-OEt-2-Py, [BA1189; 3-Me-5-OEt-2-Py], [BA1190; 4-Me-5-OEt-2-Py], [BA1191; 6-Me-5 -OEt-2-Py], [ BA1192; 3-CF 3 -5-OEt-2-Py], [BA1193; 4-CF 3 -5-OEt-2-Py], [BA1194; 6-CF 3 - 5-OEt-2-Py, [BA1195; 3-CN-5-OEt-2-Py], [BA1196; 4-CN-5-OEt-2-Py], [BA1197; 6-CN-5- OEt-2-Py], [BA1198; 3-OMe-5-OEt-2-Py], [BA1 199; 4-OMe-5-OEt-2-Py], [BA1200; 6-OMe-5-OEt- 2-Py], [BA1201; 6-OEt-2-Py], [BA1202; 3-Cl-6-OEt-2-Py], [BA1203; 4-Cl-6-OEt-2-Py], [BA 1203; BA 1204; 5-Cl-6-OEt-2-Py], [BA 1205; 3-Me-6-OEt-2-Py], [BA 1206; 4-Me-6-OEt-2-Py], [BA 1207; 5-Me-6-OEt- 2-Py], [BA1208; 3-CF 3 -6-OEt-2-Py], [BA1209; 4-CF 3 -6-OEt-2-Py], [BA1210; _{5-CF 3 -6-OEt-} 2-Py], [BA1211; 3-CN-6-OEt-2-Py], [BA1212; 4-CN-6-OEt-2-Py], [BA1213; 5 -CN-6-OEt-2-Py], [BA1214; 3-OMe-6-OEt-2-Py], [BA1215; 4-OMe-6-OEt-2-Py], [BA1216; 5-OMe -6-OEt-2-Py] , [BA1217; 3-OCH 2 CF 3 -2-Py], [BA1218; 4-Cl-3-OCH 2 CF 3 -2-Py], [BA1219; 5-Cl _{-3-OCH 2 CF 3 -2-} Py], [BA1220; 6-Cl-3-OCH 2 CF 3 -2-Py], [BA1221; 4-Me-3-OCH 2 CF 3 -2-Py] , [BA1222; 5-Me-3-OCH ₂ CF ₃ -2-Py], [BA1223; 6-Me-3-OCH 2 CF 3 -2-Py], [BA1224; 4-CF 3 -3-OCH 2 CF 3 -2-Py], [BA1225; 5- _{CF 3 -3-OCH 2 CF 3} -2-Py], [BA1226; 6-CF 3 -3-OCH 2 CF 3 -2-Py], [BA1227; 4-CN-3-OCH 2 CF 3 -2 -Py], [BA1228; 5- CN-3-OCH 2 CF 3 -2-Py], [BA1229; 6-CN-3-OCH 2 CF 3 -2-Py], [BA1230; 4-OMe-3 _{-OCH 2 CF 3 -2-Py]} , [BA1231; 5-OMe-3-OCH 2 CF 3 -2-Py], [BA1232; 6-OMe-3-OCH 2 CF 3 -2-Py], [ _{BA1233; 4-OCH 2 CF 3} -2-Py], [BA1234; 3-Cl-4-OCH 2 CF 3 -2-Py], [BA1235; 5-Cl-4-OCH 2 CF 3 -2-Py ], [BA1236; 6-Cl -4-OCH 2 CF 3 -2-Py], [BA1237; 3-Me-4-OCH 2 CF 3 -2-Py], [BA1238; 5-Me-4-OCH ₂ CF ₃ -2-Py, [BA 1239; 6-Me-4-OCH ₂ CF ₃ -2-Py], [BA 1240; 3-CF ₃ -4-OCH ₂ CF ₃ -2-Py], [BA 1241 _{; 5-CF 3 -4-OCH} 2 CF 3 -2-Py], [BA1242; 6-CF 3 -4-OCH 2 CF 3 -2-Py], [BA1243; 3-CN-4-OCH 2 CF _{3 -2-Py], [BA1244} ; 5-CN-4-OCH 2 CF 3 -2-Py], [BA1245; 6-CN-4-OCH 2 CF 3 -2-Py], [BA1246; 3- _{OMe-4-OCH 2 CF 3} -2-Py], [BA1247; 5-OMe-4-OCH 2 CF 3 -2-Py], [BA1248; 6-OMe-4-OCH 2 CF 3 -2-Py ], [BA1249; 5-OCH 2 CF 3 -2-Py], [BA1250; 3-Cl-5-OCH 2 CF 3 -2-Py], [BA1251; 4-Cl-5-OCH 2 CF 3 - 2-Py], [BA1252; 6-Cl-5-OCH 2 C _{F 3 -2-Py], [} BA1253; 3-Me-5-OCH 2 CF 3 -2-Py], [BA1254; 4-Me-5-OCH 2 CF 3 -2-Py], [BA1255; 6 _{-Me-5-OCH 2 CF 3} -2-Py], [BA1256; 3-CF 3 -5-OCH 2 CF 3 -2-Py], [BA1257; 4-CF 3 -5-OCH 2 CF 3 - 2-Py], [BA1258; 6-CF 3 -5-OCH 2 CF 3 -2-Py], [BA1259; 3-CN-5-OCH 2 CF 3 -2-Py], [BA1260; 4-CN _{-5-OCH 2 CF 3 -2-} Py], [BA1261; 6-CN-5-OCH 2 CF 3 -2-Py], [BA1262; 3-OMe-5-OCH 2 CF 3 -2-Py] , [BA1263; 4-OMe- 5-OCH 2 CF 3 -2-Py], [BA1264; 6-OMe-5-OCH 2 CF 3 -2-Py], [BA1265; 6-OCH 2 CF 3 -2 -Py], [BA1266; 3- Cl-6-OCH 2 CF 3 -2-Py], [BA1267; 4-Cl-6-OCH 2 CF 3 -2-Py], [BA1268; 5-Cl-6 _{-OCH 2 CF 3 -2-Py]} , [BA1269; 3-Me-6-OCH 2 CF 3 -2-Py], [BA1270; 4-Me-6-OCH 2 CF 3 -2-Py], [ BA1271; 5-Me-6- OCH 2 CF 3 -2-Py], [BA1272; 3-CF 3 -6-OCH 2 CF 3 -2-Py], [BA1273; 4-CF 3 -6-OCH 2 _{CF 3 -2-Py], [} BA1274; 5-CF 3 -6-OCH 2 CF 3 -2-Py], [BA1275; 3-CN-6-OCH 2 CF 3 -2-Py], [BA1276; _{4-CN-6-OCH 2} CF 3 -2-Py], [BA1277; 5-CN-6-OCH 2 CF 3 -2-Py], [BA1278; 3-OMe-6-OCH 2 CF 3 -2 -Py], [BA1279; 4- OMe-6-OCH 2 CF 3 -2-Py], [BA1280; 5-OMe-6-OCH 2 CF 3 -2-Py], [BA1281; 4-Cl-3 -Pr-2-Py], [BA1282; 5-Cl-3-Pr-2-Py ], [BA1283; 6-Cl-3-Pr-2-Py], [BA1284; 4-Me-3-Pr-2-Py],

[BA1285; 5-Me-3 -Pr-2-Py], [BA1286; 6-Me-3-Pr-2-Py], [BA1287; 4-CF 3 -3-Pr-2-Py], [ _{BA1288; 5-CF 3 -3-} Pr-2-Py], [BA1289; 6-CF 3 -3-Pr-2-Py], [BA1290; 4-CN-3-Pr-2-Py], [ BA1291; 5-CN-3-Pr-2-Py !, [BA1292; 6-CN-3-Pr-2-Py], [BA1293; 4-OMe-3-Pr-2-Py], [BA1294; 5-OMe-3-Pr-2-Py !, [BA1295; 6-OMe-3-Pr-2-Py], [BA1296; 4-Pr-2-Py], [BA1297; 3-Cl-4- Pr-2-Py, [BA1298; 5-Cl-4-Pr-2-Py], [BA1299; 6-Cl-4-Pr-2-Py], [BA1300; 3-Me-4-Pr- 2-Py], [BA1301; 5-Me-4-Pr-2-Py], [BA1302; 6-Me-4-Pr-2-Py], [BA1303; 3-CF ₃ -4-Pr-2 -Py], [BA1304; 5- CF 3 -4-Pr-2-Py], [BA1305; 6-CF 3 -4-Pr-2-Py], [BA1306; 3-CN-4-Pr-2 -Py], [BA1307; 5-CN-4-Pr-2-Py], [BA1308; 6-CN-4-Pr-2-Py], [BA1309; 3-OMe-4-Pr-2-Py ], [BA 1310; 5-OMe-4-Pr-2-Py], [BA 1311; 6-OMe-4-Pr-2-Py], [BA 1312; 5-Pr-2-Py], [BA 1313; 3] -Cl-5-Pr-2-Py], [BA 1314; 4-Cl-5-Pr-2-Py], [BA 1315; 6-Cl-5-Pr-2-Py], [BA 1316; 3-Me -5-Pr-2-Py, [BA1317; 4-Me-5-Pr-2-Py], [BA1318; 6-Me-5-Pr-2-Py], [BA1319; 3-CF _3- 5-Pr-2-Py] , [BA1320; 4-CF 3 -5-Pr-2-Py], [BA1321; 6-CF 3 -5-Pr-2-Py], [BA1322; 3-CN- 5-Pr-2-Py, [BA1323; 4-CN-5-Pr-2-Py], [BA1324; 6-CN-5-Pr-2-Py], [BA1325; 3-OMe-5- P r-2-Py], [BA1326; 4-OMe-5-Pr-2-Py], [BA1327; 6-OMe-5-Pr-2-Py], [BA1328; 6-Pr-2-Py] , [BA1329; 3-Cl-6-Pr-2-Py], [BA1330; 4-Cl-6-Pr-2-Py], [BA1331; 5-Cl-6-Pr-2-Py], [BA1331; BA1332; 3-Me-6-Pr-2-Py !, [BA1333; 4-Me-6-Pr-2-Py], [BA1334; 5-Me-6-Pr-2-Py], [BA1335; _{3-CF 3 -6-Pr-} 2-Py], [BA1336; 4-CF 3 -6-Pr-2-Py], [BA1337; 5-CF 3 -6-Pr-2-Py], [BA1338 3-CN-6-Pr-2-Py !, [BA1339; 4-CN-6-Pr-2-Py], [BA1340; 5-CN-6-Pr-2-Py], [BA1341; -OMe-6-Pr-2-Py], [BA1342; 4-OMe-6-Pr-2-Py], [BA1343; 5-OMe-6-Pr-2-Py], [BA1344; 3-OPr -2-Py !, [BA1345; 4-Cl-3-OPr-2-Py], [BA1346; 5-Cl-3-OPr-2-Py], [BA 1347; 6-Cl-3-OPr-2 -Py], [BA1348; 4-Me-3-OPr-2-Py], [BA1349; 5-Me-3-OPr-2-Py], [BA1350; 6-Me-3-OPr-2-Py ], [BA1351; 4-CF 3 -3-OPr-2-Py], [BA1352; 5-CF 3 -3-OPr-2-Py], [BA1353; 6-CF 3 -3-OPr-2- Py], [BA1354; 4-CN-3-OPr-2-Py], [BA1355; 5-CN-3-OPr-2-Py], [BA1356; 6-CN-3-OPr-2-Py] , [BA1357; 4-OMe-3-OPr-2-Py], [BA1358; 5-OMe-3-OPr-2-Py], [BA1359; 6-OMe-3-OPr-2-Py], [BA1357; BA1360; 4-OPr-2-Py], [BA1361; 3-Cl-4-OPr-2-Py], [BA1362; 5-Cl-4-OPr-2-Py], [BA1363; 6-Cl- 4-OPr-2-Py], [BA1364; 3-Me-4-OPr-2-Py], [BA1365; 5-Me-4-OPr-2-Py] , [BA1366; 6-Me- 4-OPr-2-Py], [BA1367; 3-CF 3 -4-OPr-2-Py], [BA1368; 5-CF 3 -4-OPr-2-Py] _{, [BA1369; 6-CF 3} -4-OPr-2-Py], [BA1370; 3-CN-4-OPr-2-Py], [BA1371; 5-CN-4-OPr-2-Py], [BA1372; 6-CN-4-OPr-2-Py], [BA1373; 3-OMe-4-OPr-2-Py], [BA1374; 5-OMe-4-OPr-2-Py], [BA1375] 6-OMe-4-OPr-2-Py !, [BA1376; 5-OPr-2-Py], [BA1377; 3-Cl-5-OPr-2-Py], [BA 1378; 4-Cl-5; -OPr-2-Py], [BA 1379; 6-Cl-5-OPr-2-Py], [BA 1380; 3-Me-5-OPr-2-Py], [BA 1381; 4-Me-5-OPr -2-Py], [BA1382; 6-Me-5-OPr-2-Py], [BA1383; 3-CF 3 -5-OPr-2-Py], [BA1384; 4-CF 3 -5-OPr -2-Py],

_{[BA1385; 6-CF 3 -5} -OPr-2-Py], [BA1386; 3-CN-5-OPr-2-Py], [BA1387; 4-CN-5-OPr-2-Py], [ BA1388; 6-CN-5-OPr-2-Py], [BA1389; 3-OMe-5-OPr-2-Py], [BA1390; 4-OMe-5-OPr-2-Py], [BA1391; 6-OMe-5-OPr-2-Py], [BA1392; 6-OPr-2-Py], [BA1393; 3-Cl-6-OPr-2-Py], [BA1394; 4-Cl-6- OPr-2-Py], [BA1395; 5-Cl-6-OPr-2-Py], [BA1396; 3-Me-6-OPr-2-Py], [BA1397; 4-Me-6-OPr- 2-Py], [BA1398; 5-Me-6-OPr-2-Py], [BA1399; 3-CF 3 -6-OPr-2-Py], [BA1400; 4-CF 3 -6-OPr- 2-Py], [BA1401; 5-CF 3 -6-OPr-2-Py], [BA1402; 3-CN-6-OPr-2-Py], [BA1403; 4-CN-6-OPr-2 -Py], [BA1404; 5-CN-6-OPr-2-Py], [BA1405; 3-OMe-6-OPr-2-Py], [BA1406; 4-OMe-6-OPr-2-Py ], [BA1407; 5-OMe-6-OPr-2-Py], [BA1408; 3-SMe-2-Py], [BA1409; 4-Cl-3-SMe-2-Py], [BA 1410; -Cl-3-SMe-2-Py !, [BA 1411; 6-Cl-3-SMe-2-Py], [BA 1412; 4-Me-3-SMe-2-Py], [BA 1413; 5-Me -3-SMe-2-Py !, [BA 1414; 6-Me-3-SMe-2-Py], [BA 1415; 4-CF ₃ -3-SMe-2-Py], [BA 1416; 5-CF ₃ -3-SMe-2-Py] , [BA1417; 6-CF 3 -3-SMe-2-Py], [BA1418; 4-CN-3-SMe-2-Py], [BA1419; 5-CN- 3-SMe-2-Py !, [BA1420; 6-CN-3-SMe-2-Py], [BA1421; 4-OMe-3-SMe-2-Py], [BA1422; 5-OMe-3- SMe-2-Py], [BA1423; 6-OMe-3-SMe-2-Py], [BA14] 24; 4-SMe-2-Py !, [BA1425; 3-Cl-4-SMe-2-Py], [BA1426; 5-Cl-4-SMe-2-Py], [BA1427; 6-Cl- 4-SMe-2-Py !, [BA1428; 3-Me-4-SMe-2-Py], [BA1429; 5-Me-4-SMe-2-Py], [BA1430; 6-Me-4- SMe-2-Py], [ BA1431; 3-CF 3 -4-SMe-2-Py], [BA1432; 5-CF 3 -4-SMe-2-Py], [BA1433; 6-CF 3 -4 -SMe-2-Py], [BA1434; 3-CN-4-SMe-2-Py], [BA1435; 5-CN-4-SMe-2-Py], [BA1436; 6-CN-4-SMe -2-Py !, [BA1437; 3-OMe-4-SMe-2-Py], [BA1438; 5-OMe-4-SMe-2-Py], [BA1439; 6-OMe-4-SMe-2 -Py], [BA1440; 5-SMe-2-Py], [BA1441; 3-Cl-5-SMe-2-Py], [BA1442; 4-Cl-5-SMe-2-Py], [BA1443] 6-Cl-5-SMe-2-Py !, [BA1444; 3-Me-5-SMe-2-Py], [BA1445; 4-Me-5-SMe-2-Py], [BA1446; -Me-5-SMe-2- Py], [BA1447; 3-CF 3 -5-SMe-2-Py], [BA1448; 4-CF 3 -5-SMe-2-Py], [BA1449; 6 _{-CF 3 -5-SMe-2-} Py], [BA1450; 3-CN-5-SMe-2-Py], [BA1451; 4-CN-5-SMe-2-Py], [BA1452; 6- CN-5-SMe-2-Py !, [BA1453; 3-OMe-5-SMe-2-Py], [BA1454; 4-OMe-5-SMe-2-Py], [BA1455; 6-OMe- 5-SMe-2-Py !, [BA1456; 6-SMe-2-Py], [BA1457; 3-Cl-6-SMe-2-Py], [BA1458; 4-Cl-6-SMe-2- Py], [BA1459; 5-Cl-6-SMe-2-Py], [BA1460; 3-Me-6-SMe-2-Py], [BA1461; 4-Me-6-SMe-2-Py] , [BA1462; 5-Me-6-SMe-2-Py], [BA1463; 3-CF ₃ -6-SMe -2-Py], [BA1464; 4-CF 3 -6-SMe-2-Py], [BA1465; 5-CF 3 -6-SMe-2-Py], [BA1466; 3-CN-6-SMe -2-Py !, [BA1467; 4-CN-6-SMe-2-Py], [BA1468; 5-CN-6-SMe-2-Py], [BA1469; 3-OMe-6-SMe-2 -Py], [BA1470; 4- OMe-6-SMe-2-Py], [BA1471; 5-OMe-6-SMe-2-Py], [BA1472; 3-SCF 3 -2-Py], [ BA1473; 4-Cl-3- SCF 3 -2-Py], [BA1474; 5-Cl-3-SCF 3 -2-Py], [BA1475; 6-Cl-3-SCF 3 -2-Py], [BA1476; 4-Me-3 -SCF 3 -2-Py], [BA1477; 5-Me-3-SCF 3 -2-Py], [BA1478; 6-Me-3-SCF 3 -2-Py] _{, [BA1479; 4-CF 3} -3-SCF 3 -2-Py], [BA1480; 5-CF 3 -3-SCF 3 -2-Py], [BA1481; 6-CF 3 -3-SCF 3 - 2-Py], [BA1482; 4-CN-3-SCF 3 -2-Py], [BA1483; 5-CN-3-SCF 3 -2-Py], [BA1484; 6-CN-3-SCF 3 -2-Py],

[BA1485; 4-OMe-3 -SCF 3 -2-Py], [BA1486; 5-OMe-3-SCF 3 -2-Py], [BA1487; 6-OMe-3-SCF 3 -2-Py] , [BA1488; 4-SCF ₃ -2-Py], [BA 1489; 3-Cl 4-SCF ₃ -2-Py], [BA 1490; 5-Cl 4-SCF ₃ -2-Py], [BA 14 1 ; 6-Cl-4-SCF 3 -2-Py], [BA1492; 3-Me-4-SCF 3 -2-Py], [BA1493; 5-Me-4-SCF 3 -2-Py], [ BA1494; 6-Me-4- SCF 3 -2-Py], [BA1495; 3-CF 3 -4-SCF 3 -2-Py], [BA1496; 5-CF 3 -4-SCF 3 -2-Py ], [BA1497; 6-CF 3 -4-SCF 3 -2-Py], [BA1498; 3-CN-4-SCF 3 -2-Py], [BA1499; 5-CN-4-SCF 3 -2 -Py], [BA1500; 6- CN-4-SCF 3 -2-Py], [BA1501; 3-OMe-4-SCF 3 -2-Py], [BA1502; 5-OMe-4-SCF 3 - 2-Py], [BA1503; 6-OMe-4-SCF ₃ -2-Py], [BA 1504; 5-SCF ₃ -2-Py], [BA 1505; 3-Cl-5-SCF ₃ -2-Py ], [BA1506; 4-Cl -5-SCF 3 -2-Py], [BA1507; 6-Cl-5-SCF 3 -2-Py], [BA1508; 3-Me-5-SCF 3 -2- Py], [BA 1509; 4-Me-5-SCF ₃ -2-Py], [BA 1510; 6-Me-5-SCF ₃ -2-Py], [BA 1511; 3-CF ₃ -5-SCF _3- 2-Py], [BA 1512; 4-CF ₃ -5-SCF ₃ -2-Py], [BA 1513; 6-CF ₃ -5-SCF ₃ 2-Py], [BA 1514; 3-CN-5- SCF ₃ -2-Py !, [BA 1515; 4-CN-5-SCF ₃ -2-Py], [BA 1516; 6-CN-5-SCF ₃ -2-Py], [BA 1517; 3-OMe-5] -SCF ₃ -2-Py, [BA1518; 4-OMe-5-SCF ₃ -2-Py], [BA 1519; 6-OMe-5-SCF ₃ -2-Py], [BA _{1520; 6-SCF 3 -2-} Py], [BA1521; 3-Cl-6-SCF 3 -2-Py], [BA1522; 4-Cl-6-SCF 3 -2-Py], [BA1523; 6 _{-Cl-6-SCF 3 -2-} Py], [BA1524; 3-Me-6-SCF 3 -2-Py], [BA1525; 4-Me-6-SCF 3 -2-Py], [BA1526; 6-Me-6-SCF ₃ -2-Py], [BA 1527; 3-CF ₃ -6-SCF ₃ -2-Py], [BA 1528; 4-CF ₃ -6-SCF ₃ -2-Py], _{[BA1529; 6-CF 3 -6} -SCF 3 -2-Py], [BA1530; 3-CN-6-SCF 3 -2-Py], [BA1531; 4-CN-6-SCF 3 -2-Py ], [BA1532; 6-CN -6-SCF 3 -2-Py], [BA1533; 3-OMe-6-SCF 3 -2-Py], [BA1534; 4-OMe-6-SCF 3 -2- Py], [BA1535; 6- OMe-6-SCF 3 -2-Py], [BA1536; 3-S (O) Me-2-Py], [BA1537; 4-Cl-3-S (O) Me -2-Py !, [BA1538; 5-Cl-3-S (O) Me-2-Py], [BA1539; 6-Cl-3-S (O) Me-2-Py], [BA1540; -Me-3-S (O) Me-2-Py], [BA1541; 5-Me-3-S (O) Me-2-Py], [BA1542; 6-Me-3-S (O) Me -2-Py], [BA1543; 4-CF 3 -3-S (O) Me-2-Py], [BA1544; 5-CF 3 -3-S (O) Me-2-Py], [BA1545 _{; 6-CF 3 -3-S} (O) Me-2-Py], [BA1546; 4-CN-3-S (O) Me-2-Py], [BA1547; 5-CN-3-S ( O) Me-2-Py], [BA1548; 6-CN-3-S (O) Me-2-Py], [BA1549; 4-OMe-3-S (O) Me-2-Py], [BA BA1550; 5-OMe-3-S (O) Me-2-Py], [BA1551; 6-OMe-3-S (O) Me-2-Py], [BA1552; 4-S (O) Me- 2-Py !, [BA1553; 3-Cl-4-S (O) Me-2-Py], [BA1554; 5-Cl-4-S (O) Me-2-Py], [BA1555; 6- Cl-4 -S (O) Me-2-Py], [BA1556; 3-Me-4-S (O) Me-2-Py], [BA1557; 5-Me-4-S (O) Me-2-Py ], [BA1558; 6-Me -4-S (O) Me-2-Py], [BA1559; 3-CF 3 -4-S (O) Me-2-Py], [BA1560; 5-CF 3 -4-S (O) Me- 2-Py], [BA1561; 6-CF 3 -4-S (O) Me-2-Py], [BA1562; 3-CN-4-S (O) Me- 2-Py], [BA1563; 5-CN-4-S (O) Me-2-Py], [BA1564; 6-CN-4-S (O) Me-2-Py], [BA1565; OMe-4-S (O) Me-2-Py], [BA1566; 5-OMe-4-S (O) Me-2-Py], [BA1567; 6-OMe-4-S (O) Me- 2-Py], [BA1568; 5-S (O) Me-2-Py], [BA1569; 3-Cl-5-S (O) Me-2-Py], [BA1570; 4-Cl-5- S (O) Me-2-Py], [BA1571; 6-Cl-5-S (O) Me-2-Py], [BA1572; 3-Me-5-S (O) Me-2-Py] , [BA1573; 4-Me- 5-S (O) Me-2-Py], [BA1574; 6-Me-5-S (O) Me-2-Py], [BA1575; 3-CF 3 -5 -S (O) Me-2- Py], [BA1576; 4-CF 3 -5-S (O) Me-2-Py], [BA1577; 6-CF 3 -5-S (O) Me-2 -Py], [BA1578; 3-CN-5-S (O) Me-2-Py], [BA1579; 4-CN-5-S (O) Me-2-Py], [BA1580; 6-CN -5-S (O) Me-2-Py], [BA1581; 3-OMe-5-S (O) Me-2-Py], [BA1582; 4-OMe-5-S (O) Me-2 -Py], [BA 1583; 6-OMe-5-S (O) Me-2-Py], [BA1584; 6-S (O) Me-2-Py],

[BA 1585; 3-Cl-6-S (O) Me-2-Py], [BA 1586; 4-Cl-6-S (O) Me-2-Py], [BA 1587; 5-Cl-6-S (O) Me-2-Py], [BA1588; 3-Me-6-S (O) Me-2-Py], [BA1589; 4-Me-6-S (O) Me-2-Py], [BA1590; 5-Me-6 -S (O) Me-2-Py], [BA1591; 3-CF 3 -6-S (O) Me-2-Py], [BA1592; 4-CF 3 -6 -S (O) Me-2- Py], [BA1593; 5-CF 3 -6-S (O) Me-2-Py], [BA1594; 3-CN-6-S (O) Me-2- Py], [BA1595; 4-CN-6-S (O) Me-2-Py], [BA1596; 5-CN-6-S (O) Me-2-Py], [BA1597; 3-OMe- 6-S (O) Me-2-Py], [BA 1598; 4-OMe-6-S (O) Me-2-Py], [BA1599; 5-OMe-6-S (O) Me-2- 2 Py], [BA1600; 3- S (O) CF 3 -2-Py], [BA1601; 4-Cl-3-S (O) CF 3 -2-Py], [BA1602; 5-Cl-3- _{S (O) CF 3 -2-} Py], [BA1603; 6-Cl-3-S (O) CF 3 -2-Py], [BA1604; 4-Me-3-S (O) CF 3 -2 -Py], [BA1605; 5- Me-3-S (O) CF 3 -2-Py], [BA1606; 6-Me-3-S (O) CF 3 -2-Py], [BA1607; 4 _{-CF 3 -3-S (O)} CF 3 -2-Py], [BA1608; 5-CF 3 -3-S (O) CF 3 -2-Py], [BA1609; 6-CF 3 -3- _{S (O) CF 3 -2-} Py], [BA1610; 4-CN-3-S (O) CF 3 -2-Py], [BA1611; 5-CN-3-S (O) CF 3 -2 -Py], [BA1612; 6- CN-3-S (O) CF 3 -2-Py], [BA1613; 4-OMe-3-S (O) CF 3 -2-Py], [BA1614; 5 -OMe-3-S (O) CF 3 -2-Py], [BA1615; 6-OMe-3-S (O) CF 3 -2-Py], [BA1616; 4-S (O) CF 3 - 2-Py], [BA1617; 3-Cl-4-S (O) CF 3 -2-Py], [BA1618; 5-Cl-4-S ( O) CF 3 -2-Py], [BA1619; 6-Cl-4-S (O) CF 3 -2-Py], [BA1620; 3-Me-4-S ( _{O) CF 3 -2-Py]} , [BA1621; 5-Me-4-S (O) CF 3 -2-Py], [BA1622; 6-Me-4-S (O) CF 3 -2-Py ], [BA1623; 3-CF 3 -4-S (O) CF 3 -2-Py], [BA1624; 5-CF 3 -4-S (O) CF 3 -2-Py], [BA1625; 6 _{-CF 3 -4-S (O)} CF 3 -2-Py], [BA1626; 3-CN-4-S (O) CF 3 -2-Py], [BA1627; 5-CN-4-S ( _{O) CF 3 -2-Py]} , [BA1628; 6-CN-4-S (O) CF 3 -2-Py], [BA1629; 3-OMe-4-S (O) CF 3 -2-Py ], [BA1630; 5-OMe -4-S (O) CF 3 -2-Py], [BA1631; 6-OMe-4-S (O) CF 3 -2-Py], [BA1632; 5-S _{(O) CF 3 -2-Py} ], [BA1633; 3-Cl-5-S (O) CF 3 -2-Py], [BA1634; 4-Cl-5-S (O) CF 3 -2- Py], [BA1635; 6- Cl-5-S (O) CF 3 -2-Py], [BA1636; 3-Me-5-S (O) CF 3 -2-Py], [BA1637; 4- Me-5-S (O) CF 3 -2-Py], [BA1638; 6-Me-5-S (O) CF 3 -2-Py], [BA1639; 3-CF 3 -5-S (O ) CF ₃ -2-Py !, [BA 1640; 4-CF ₃ -5-S (O) CF ₃ -2-Py], [BA 1641; 6-CF ₃ -5-S (O) CF ₃ -2-] Py], [BA1642; 3- CN-5-S (O) CF 3 -2-Py], [BA1643; 4-CN-5-S (O) CF 3 -2-Py], [BA1644; 6- CN-5-S (O) CF 3 -2-Py], [BA1645; 3-OMe-5-S (O) CF 3 -2-Py], [BA1646; 4-OMe-5-S (O) _{CF 3 -2-Py], [} BA1647; 6-OMe-5-S (O) CF 3 -2-Py], [BA1648; 6-S (O) CF 3 -2-Py], [BA1649; 3 -Cl-6-S (O) CF ₃ -2-Py], [B A1650; 4-Cl-6- S (O) CF 3 -2-Py], [BA1651; 5-Cl-6-S (O) CF 3 -2-Py], [BA1652; 3-Me-6- _{S (O) CF 3 -2-} Py], [BA1653; 4-Me-6-S (O) CF 3 -2-Py], [BA1654; 5-Me-6-S (O) CF 3 -2 -Py], [BA1655; 3- CF 3 -6-S (O) CF 3 -2-Py], [BA1656; 4-CF 3 -6-S (O) CF 3 -2-Py], [BA1657 _{; 5-CF 3 -6-S} (O) CF 3 -2-Py], [BA1658; 3-CN-6-S (O) CF 3 -2-Py], [BA1659; 4-CN-6- _{S (O) CF 3 -2-} Py], [BA1660; 5-CN-6-S (O) CF 3 -2-Py], [BA1661; 3-OMe-6-S (O) CF 3 -2 -Py], [BA1662; 4- OMe-6-S (O) CF 3 -2-Py], [BA1663; 5-OMe-6-S (O) CF 3 -2-Py], [BA1664; 3 _{-S (O) 2 Me-2} -Py], [BA1665; 4-Cl-3-S (O) 2 Me-2-Py], [BA1666; 5-Cl-3-S (O) 2 Me- 2-Py], [BA1667; 6-Cl-3-S (O) ₂ Me-2-Py], [BA1668; 4-Me-3-S (O) ₂ Me-2-Py], [BA1669; 5-Me-3-S ( O) 2 Me-2-Py], [BA1670; 6-Me-3-S (O) 2 Me-2-Py], [BA1671; 4-CF 3 -3-S _{(O) 2 Me-2-} Py], [BA1672; 5-CF 3 -3-S (O) 2 Me-2-Py], [BA1673; 6-CF 3 -3-S (O) 2 Me- 2-Py], [BA1674; 4-CN-3-S (O) ₂ Me-2-Py], [BA1675; 5-CN-3-S (O) ₂ Me-2-Py], [BA1676; 6-CN-3-S ( O) 2 Me-2-Py], [BA1677; 4-OMe-3-S (O) 2 Me-2-Py], [BA1678; 5-OMe-3-S ( O) ₂ Me-2-Py, [BA1679; 6-OMe-3-S (O) ₂ Me-2-Py], [BA 1680; 4-S (O) ₂ Me-2-Py], [BA1681 3-Cl-4-S (O) ₂ Me-2- Py], [BA1682; 5-Cl-4-S (O) ₂ Me-2-Py], [BA1683; 6-Cl-4-S (O) ₂ Me-2-Py], [BA1684; Me-4-S (O) ₂ Me-2-Py],

[BA1685; 5-Me-4 -S (O) 2 Me-2-Py], [BA1686; 6-Me-4-S (O) 2 Me-2-Py], [BA1687; 3-CF 3 - _{4-S (O) 2 Me} -2-Py], [BA1688; 5-CF 3 -4-S (O) 2 Me-2-Py], [BA1689; 6-CF 3 -4-S (O) ₂ Me-2-Py !, [BA 1690; 3-CN-4-S (O) ₂ Me-2-Py], [BA 1691; 5-CN-4-S (O) ₂ Me-2-Py], [BA1692; 6-CN-4 -S (O) 2 Me-2-Py], [BA1693; 3-OMe-4-S (O) 2 Me-2-Py], [BA1694; 5-OMe-4 _{-S (O) 2 Me-2} -Py], [BA1695; 6-OMe-4-S (O) 2 Me-2-Py], [BA1696; 5-S (O) 2 Me-2-Py] , [BA 1697; 3-Cl-5-S (O) ₂ Me-2-Py], [BA 1698; 4-Cl-5-S (O) ₂ Me-2-Py], [BA 1699; 6-Cl- _{5-S (O) 2 Me} -2-Py], [BA1700; 3-Me-5-S (O) 2 Me-2-Py], [BA1701; 4-Me-5-S (O) 2 Me -2-Py], [BA1702; 6-Me-5-S (O) ₂ Me-2-Py], [BA 1703; 3-CF ₃ -5-S (O) ₂ Me-2-Py], BA 1704; 4-CF ₃ -5-S (O) ₂ Me-2-Py], [BA 1705; 6-CF ₃ -5-S (O) ₂ Me-2-Py], [BA 1706; 3-CN- _{5-S (O) 2 Me} -2-Py], [BA1707; 4-CN-5-S (O) 2 Me-2-Py], [BA1708; 6-CN-5-S (O) 2 Me -2-Py], [BA 1709; 3-OMe-5-S (O) ₂ Me-2-Py], [BA 1710; 4-OMe-5-S (O) ₂ Me-2-Py], [BA 1711 ; 6-OMe-5-S (O) 2 Me-2-Py], [BA1712; 6-S (O) 2 Me-2-Py], [BA1713; 3-Cl-6-S (O) 2 Me-2-Py !, [BA1714; 4-Cl-6-S (O) ₂ Me-2-Py], [BA1715; 5-Cl-6-S (O) ₂ Me-2-Py], [BA1 14; BA1716; 3-Me-6-S (O) ₂ Me- 2-Py], [BA1717; 4-Me-6-S (O) ₂ Me-2-Py], [BA1718; 5-Me-6-S (O) ₂ Me-2-Py], [BA1719; _{3-CF 3 -6-S (} O) 2 Me-2-Py], [BA1720; 4-CF 3 -6-S (O) 2 Me-2-Py], [BA1721; 5-CF 3 -6 _{-S (O) 2 Me-2} -Py], [BA1722; 3-CN-6-S (O) 2 Me-2-Py], [BA1723; 4-CN-6-S (O) 2 Me- 2-Py], [BA1724; 5-CN-6-S (O) ₂ Me-2-Py], [BA1725; 3-OMe-6-S (O) ₂ Me-2-Py], [BA1726; 4-OMe-6-S ( O) 2 Me-2-Py], [BA1727; 5-OMe-6-S (O) 2 Me-2-Py], [BA1728; 3-S (O) 2 CF _{3 -2-Py], [BA1729} ; 4-Cl-3-S (O) 2 CF 3 -2-Py], [BA1730; 5-Cl-3-S (O) 2 CF 3 -2-Py] , [BA1731; 6-Cl- 3-S (O) 2 CF 3 -2-Py], [BA1732; 4-Me-3-S (O) 2 CF 3 -2-Py], [BA1733; 5- Me-3-S (O) 2 CF 3 -2-Py], [BA1734; 6-Me-3-S (O) 2 CF 3 -2-Py], [BA1735; 4-CF 3 -3-S _{(O) 2 CF 3 -2-} Py], [BA1736; 5-CF 3 -3-S (O) 2 CF 3 -2-Py], [BA1737; 6-CF 3 -3-S (O) 2 _{CF 3 -2-Py], [} BA1738; 4-CN-3-S (O) 2 CF 3 -2-Py], [BA1739; 5-CN-3-S (O) 2 CF 3 -2-Py ], [BA1740; 6-CN -3-S (O) 2 CF 3 -2-Py], [BA1741; 4-OMe-3-S (O) 2 CF 3 -2-Py], [BA1742; 5 -OMe-3-S (O) 2 CF 3 -2-Py], [BA1743; 6-OMe-3-S (O) 2 CF 3 -2-Py], [BA1744; 4-S (O) 2 _{CF 3 -2-Py], [} BA1745; 3-Cl-4-S (O) 2 CF 3 -2-Py], [BA1746; 5-Cl-4-S (O) 2 CF 3 -2-Py], [BA1747; 6-Cl-4-S (O) 2 CF 3 -2-Py], [BA1748; 3-Me-4-S (O) 2 CF 3 -2-Py], [BA1749; 5-Me-4 -S (O) 2 CF 3 -2-Py], [BA1750; 6-Me-4-S (O) 2 CF 3 -2-Py], [BA1751; 3-CF _{3 -4-S (O) 2} CF 3 -2-Py], [BA1752; 5-CF 3 -4-S (O) 2 CF 3 -2-Py], [BA1753; 6-CF 3 -4- _{S (O) 2 CF 3 -2} -Py], [BA1754; 3-CN-4-S (O) 2 CF 3 -2-Py], [BA1755; 5-CN-4-S (O) 2 CF _{3 -2-Py], [BA1756} ; 6-CN-4-S (O) 2 CF 3 -2-Py], [BA1757; 3-OMe-4-S (O) 2 CF 3 -2-Py] , [BA 1758; 5-OMe-4-S (O) ₂ CF ₃ -2-Py], [BA 1759; 6-OMe-4-S (O) ₂ CF ₃ -2-Py], [BA 1760; _{S (O) 2 CF 3 -2} -Py], [BA1761; 3-Cl-5-S (O) 2 CF 3 -2-Py], [BA1762; 4-Cl-5-S (O) 2 CF _{3 -2-Py], [BA1763} ; 6-Cl-5-S (O) 2 CF 3 -2-Py], [BA1764; 3-Me-5-S (O) 2 CF 3 -2-Py] , [BA1765; 4-Me- 5-S (O) 2 CF 3 -2-Py], [BA1766; 6-Me-5-S (O) 2 CF 3 -2-Py], [BA1767; 3- _{CF 3 -5-S (O)} 2 CF 3 -2-Py], [BA1768; 4-CF 3 -5-S (O) 2 CF 3 -2-Py], [BA1769; 6-CF 3 -5 _{-S (O) 2 CF 3 -2} -Py], [BA1770; 3-CN-5-S (O) 2 CF 3 -2-Py], [BA1771; 4-CN-5-S (O) 2 _{CF 3 -2-Py], [} BA1772; 6-CN-5-S (O) 2 CF 3 -2-Py], [BA1773; 3-OMe-5-S (O) 2 CF 3 -2-Py ], [BA1774; 4-OMe -5-S (O) 2 CF 3 -2-Py], [BA1775; 6-OMe-5-S (O) 2 _{CF 3 -2-Py], [} BA1776; 6-S (O) 2 CF 3 -2-Py], [BA1777; 3-Cl-6-S (O) 2 CF 3 -2-Py], [BA1778 ; 4-Cl-6-S (O) 2 CF 3 -2-Py], [BA1779; 5-Cl-6-S (O) 2 CF 3 -2-Py], [BA1780; 3-Me-6 _{-S (O) 2 CF 3 -2} -Py], [BA1781; 4-Me-6-S (O) 2 CF 3 -2-Py], [BA1782; 5-Me-6-S (O) 2 _{CF 3 -2-Py], [} BA1783; 3-CF 3 -6-S (O) 2 CF 3 -2-Py], [BA1784; 4-CF 3 -6-S (O) 2 CF 3 -2 -Py],

_{[BA1785; 5-CF 3 -6} -S (O) 2 CF 3 -2-Py], [BA1786; 3-CN-6-S (O) 2 CF 3 -2-Py], [BA1787; 4- CN-6-S (O) 2 CF 3 -2-Py], [BA1788; 5-CN-6-S (O) 2 CF 3 -2-Py], [BA1789; 3-OMe-6-S ( O) ₂ CF ₃ -2-Py, [BA 1790; 4-OMe-6-S (O) ₂ CF ₃ -2-Py], [BA 1791; 5-OMe-6-S (O) ₂ CF _3- 2-Py], [BA1792; 3-CN-2-Py], [BA1793; 4-Cl-3-CN-2-Py], [BA1794; 5-Cl-3-CN-2-Py], [BA1 794; BA 1795; 6-Cl-3-CN-2-Py], [BA1796; 4-Me-3-CN-2-Py], [BA1797; 5-Me-3-CN-2-Py], [BA 1798; 6-Me-3-CN- 2-Py], [BA1799; 4-CF 3 -3-CN-2-Py], [BA1800; 5-CF 3 -3-CN-2-Py], [BA1801; _{6-CF 3 -3-CN-} 2-Py], [BA1802; 4-CN-3-CN-2-Py], [BA1803; 5-CN-3-CN-2-Py], [BA1804; 6 -CN-3-CN-2-Py], [BA1805; 4-OMe-3-CN-2-Py], [BA1806; 5-OMe-3-CN-2-Py], [BA1807; 6-OMe -3-CN-2-Py !, [BA1808; 4-CN-2-Py], [BA1809; 3-Cl-4-CN-2-Py], [BA1810; 5-Cl-4-CN-2 -Py], [BA 1811; 6-Cl-4-CN-2-Py], [BA 1812; 3-Me-4-CN-2-Py], [BA 1813; 5-Me-4-CN-2-Py ], [BA1814; 6-Me -4-CN-2-Py], [BA1815; 3-CF 3 -4-CN-2-Py], [BA1816; 5-CF 3 -4-CN-2-Py ], [BA1817; 6-CF 3 -4-CN-2-Py], [BA1818; 3-CN-4-CN-2-Py], [BA1819; 5-CN-4-CN-2-Py] , [BA1820; 6-CN-4-CN-2-Py], [BA1821; 3-OMe-4-CN-2-Py], [BA1822; 5-OMe-4-CN-2-Py] , [BA1823; 6-OMe-4-CN-2-Py], [BA1824; 5-CN-2-Py], [BA1825; 3-Cl-5-CN-2-Py], [BA1826; Cl-5-CN-2-Py], [BA1827; 6-Cl-5-CN-2-Py], [BA1828; 3-Me-5-CN-2-Py], [BA1829; 4-Me- 5-CN-2-Py] , [BA1830; 6-Me-5-CN-2-Py], [BA1831; 3-CF 3 -5-CN-2-Py], [BA1832; 4-CF 3 - 5-CN-2-Py] , [BA1833; 6-CF 3 -5-CN-2-Py], [BA1834; 3-CN-5-CN-2-Py], [BA1835; 4-CN-5 -CN-2-Py], [BA1836; 6-CN-5-CN-2-Py], [BA1837; 3-OMe-5-CN-2-Py], [BA1838; 4-OMe-5-CN -2-Py], [BA1839; 6-OMe-5-CN-2-Py], [BA1840; 6-CN-2-Py], [BA1841; 3-Cl-6-CN-2-Py], [BA1842; 4-Cl-6-CN-2-Py], [BA1843; 5-Cl-6-CN-2-Py], [BA1844; 3-Me-6-CN-2-Py], [BA1845] ; 4-Me-6-CN -2-Py], [BA1846; 5-Me-6-CN-2-Py], [BA1847; 3-CF 3 -6-CN-2-Py], [BA1848; _{4-CF 3 -6-CN-} 2-Py], [BA1849; 5-CF 3 -6-CN-2-Py], [BA1850; 3-CN-6-CN-2-Py], [BA1851; 4-CN-6-CN-2-Py], [BA1852; 5-CN-6-CN-2-Py], [BA1853; 3-OMe-6-CN-2-Py], [BA1854; OMe-6-CN-2-Py !, [BA1855; 5-OMe-6-CN-2-Py], [BA1856; 3-COOMe-2-Py], [BA1857; 4-Cl-3-COOMe- 2-Py], [BA1858; 5-Cl-3-COOMe-2-Py], [BA1859; 6-Cl-3-COOMe-2-Py], [BA1860; 4-Me-3-COOMe-2-] Py], [BA1861; 5-Me-3-COOMe-2-Py], [BA1862; 6-Me-3-COOMe-2-Py], [BA1863; _{4-CF 3 -3-COOMe-} 2-Py], [BA1864; 5-CF 3 -3-COOMe-2-Py], [BA1865; 6-CF 3 -3-COOMe-2-Py], [BA1866 4-CN-3-COOMe-2-Py !, [BA1867; 5-CN-3-COOMe-2-Py], [BA1868; 6-CN-3-COOMe-2-Py], [BA1869; -OMe-3-COOMe-2-Py], [BA1870; 5-OMe-3-COOMe-2-Py], [BA1871; 6-OMe-3-COOMe-2-Py], [BA1872; -2-Py !, [BA1873; 3-Cl-4-COOMe-2-Py], [BA1874; 5-Cl-4-COOMe-2-Py], [BA1875; 6-Cl-4-COOMe-2 -Py], [BA1876; 3-Me-4-COOMe-2-Py], [BA1877; 5-Me-4-COOMe-2-Py], [BA1878; 6-Me-4-COOMe-2-Py] ], [BA1879; 3-CF 3 -4-COOMe-2-Py], [BA1880; 5-CF 3 -4-COOMe-2-Py], [BA1881; 6-CF 3 -4-COOMe-2- Py], [BA1882; 3-CN-4-COOMe-2-Py], [BA1883; 5-CN-4-COOMe-2-Py], [BA1884; 6-CN-4-COOMe-2-Py] ,

[BA1885; 3-OMe-4-COOMe-2-Py], [BA1886; 5-OMe-4-COOMe-2-Py], [BA1887; 6-OMe-4-COOMe-2-Py], [BA1888] 5-COOMe-2-Py !, [BA1889; 3-Cl-5-COOMe-2-Py], [BA1890; 4-Cl-5-COOMe-2-Py], [BA1891; 6-Cl-5; -COOMe-2-Py], [BA1892; 3-Me-5-COOMe-2-Py], [BA1893; 4-Me-5-COOMe-2-Py], [BA1894; 6-Me-5-COOMe -2-Py], [BA 1895; 3-CF ₃ -5-COOMe-2-Py], [BA 1896; 4-CF ₃ -5-COOMe-2-Py], [BA 1897; 6-CF ₃ -5-] COOMe-2-Py !, [BA1898; 3-CN-5-COOMe-2-Py], [BA1899; 4-CN-5-COOMe-2-Py], [BA1900; 6-CN-5-COOMe- 2-Py], [BA1901; 3-OMe-5-COOMe-2-Py], [BA1902; 4-OMe-5-COOMe-2-Py], [BA1903; 6-OMe-5-COOMe-2-] Py], [BA1904; 6-COOMe-2-Py], [BA1905; 3-Cl-6-COOMe-2-Py], [BA1906; 4-Cl-6-COOMe-2-Py], [BA1907; 5-Cl-6-COOMe-2-Py !, [BA1908; 3-Me-6-COOMe-2-Py], [BA1909; 4-Me-6-COOMe-2-Py], [BA1910; 5- Me-6-COOMe-2- Py], [BA1911; 3-CF 3 -6-COOMe-2-Py], [BA1912; 4-CF 3 -6-COOMe-2-Py], [BA1913; 5- _{CF 3 -6-COOMe-2-} Py], [BA1914; 3-CN-6-COOMe-2-Py], [BA1915; 4-CN-6-COOMe-2-Py], [BA1916; 5-CN -6-COOMe-2-Py !, [BA1917; 3-OMe-6-COOMe-2-Py], [BA1918; 4-OMe-6-COOMe-2-Py], [BA1919; 5-OMe-6 -COOMe-2-Py], [ BA1920; 4-Cl-3-NO 2 -2-Py], [BA1921; 5-C _{l-3-NO 2 -2-} Py], [BA1922; 6-Cl-3-NO 2 -2-Py], [BA1923; 4-Me-3-NO 2 -2-Py], [BA1924; 5 _{-Me-3-NO 2 -2-} Py], [BA1925; 6-Me-3-NO 2 -2-Py], [BA1926; 4-CF 3 -3-NO 2 -2-Py], [BA1927 _{; 5-CF 3 -3-NO} 2 -2-Py], [BA1928; 6-CF 3 -3-NO 2 -2-Py], [BA1929; 4-CN-3-NO 2 -2-Py] , [BA1930; 5-CN- 3-NO 2 -2-Py], [BA1931; 6-CN-3-NO 2 -2-Py], [BA1932; 4-OMe-3-NO 2 -2-Py ], [BA1933; 5-OMe -3-NO 2 -2-Py], [BA1934; 6-OMe-3-NO 2 -2-Py], [BA1935; 4-NO 2 -2-Py], [ BA1936; 3-Cl-4- NO 2 -2-Py], [BA1937; 5-Cl-4-NO 2 -2-Py], [BA1938; 6-Cl-4-NO 2 -2-Py], [BA1939; 3-Me-4 -NO 2 -2-Py], [BA1940; 5-Me-4-NO 2 -2-Py], [BA1941; 6-Me-4-NO 2 -2-Py] _{, [BA1942; 3-CF 3} -4-NO 2 -2-Py], [BA1943; 5-CF 3 -4-NO 2 -2-Py], [BA1944; 6-CF 3 -4-NO 2 - 2-Py], [BA1945; 3-CN-4-NO 2 -2-Py], [BA1946; 5-CN-4-NO 2 -2-Py], [BA1947; 6-CN-4-NO 2 -2-Py], [BA1948; 3-OMe-4-NO 2 -2-Py], [BA1949; 5-OMe-4-NO 2 -2-Py], [BA1950; 6-OMe-4-NO ₂ -2-Py], [BA1951; 5-NO ₂ -2-Py], [BA 1952; 3-Cl-5-NO ₂ -2-Py], [BA 1 965; 4-Cl-5-NO ₂ -2 -Py], [BA1954; 6- Cl-5-NO 2 -2-Py], [BA1955; 3-Me-5-NO 2 -2-Py], [BA1956; 4-Me-5-NO 2 - 2-Py], [BA 1957; 6-Me-5-NO ₂ -2-Py ], [BA1958; 3-CF 3 -5-NO 2 -2-Py], [BA1959; 4-CF 3 -5-NO 2 -2-Py], [BA1960; 6-CF 3 -5-NO 2 -2-Py], [BA1961; 3-CN-5-NO 2 -2-Py], [BA1962; 4-CN-5-NO 2 -2-Py], [BA1963; 6-CN-5-NO ₂ -2-Py !, [BA1964; 3-OMe-5-NO ₂ -2-Py], [BA 1 965; 4-OMe-5-NO ₂ -2-Py], [BA1966; 6-OMe-5- NO ₂ -2-Py !, [BA 1967; 6-NO ₂ -2-Py], [BA 1968; 3-Cl-6-NO ₂ -2-Py], [BA 1969; 4-Cl 6-NO ₂ − 2-Py], [BA1970; 5-Cl-6-NO 2 -2-Py], [BA1971; 3-Me-6-NO 2 -2-Py], [BA1972; 4-Me-6-NO 2 -2-Py], [BA1973; 5-Me-6-NO 2 -2-Py], [BA1974; 3-CF 3 -6-NO 2 -2-Py], [BA1975; 4-CF 3 -6 _{-NO 2 -2-Py], [} BA1976; 5-CF 3 -6-NO 2 -2-Py], [BA1977; 3-CN-6-NO 2 -2-Py], [BA1978; 4-CN _{-6-NO 2 -2-Py]} , [BA1979; 5-CN-6-NO 2 -2-Py], [BA1980; 3-OMe-6-NO 2 -2-Py], [BA1981; 4- _{OMe-6-NO 2 -2-} Py], [BA1982; 5-OMe-6-NO 2 -2-Py], [BA1983; 4-Cl-3-NH 2 -2-Py], [BA1984; 5 -Cl-3-NH ₂ -2-Py],

[BA1985; 6-Cl-3 -NH 2 -2-Py], [BA1986; 4-Me-3-NH 2 -2-Py], [BA1987; 5-Me-3-NH 2 -2-Py] , [BA1988; 6-Me- 3-NH 2 -2-Py], [BA1989; 4-CF 3 -3-NH 2 -2-Py], [BA1990; 5-CF 3 -3-NH 2 -2 -Py], [BA1991; 6- CF 3 -3-NH 2 -2-Py], [BA1992; 4-CN-3-NH 2 -2-Py], [BA1993; 5-CN-3-NH 2 -2-Py], [BA1994; 6-CN-3-NH 2 -2-Py], [BA1995; 4-OMe-3-NH 2 -2-Py], [BA1996; 5-OMe-3-NH _{2 -2-Py], [BA1997} ; 6-OMe-3-NH 2 -2-Py], [BA1998; 4-NH 2 -2-Py], [BA1999; 3-Cl-4-NH 2 -2 -Py], [BA2000; 5- Cl-4-NH 2 -2-Py], [BA2001; 6-Cl-4-NH 2 -2-Py], [BA2002; 3-Me-4-NH 2 - 2-Py], [BA2003; 5-Me-4-NH 2 -2-Py], [BA2004; 6-Me-4-NH 2 -2-Py], [BA2005; 3-CF 3 -4-NH _{2 -2-Py], [BA2006} ; 5-CF 3 -4-NH 2 -2-Py], [BA2007; 6-CF 3 -4-NH 2 -2-Py], [BA2008; 3-CN- _{4-NH 2 -2-Py]} , [BA2009; 5-CN-4-NH 2 -2-Py], [BA2010; 6-CN-4-NH 2 -2-Py], [BA2011; 3-OMe _{-4-NH 2 -2-Py]} , [BA2012; 5-OMe-4-NH 2 -2-Py], [BA2013; 6-OMe-4-NH 2 -2-Py], [BA2014; 5- _{NH 2 -2-Py], [} BA2015; 3-Cl-5-NH 2 -2-Py], [BA2016; 4-Cl-5-NH 2 -2-Py], [BA2017; 6-Cl-5 _{-NH 2 -2-Py], [} BA2018; 3-Me-5-NH 2 -2-Py], [BA2019; 4-Me-5-NH 2 -2-Py], [BA2020; 6-Me- 5-NH ₂ -2-Py, [BA 2021; 3-CF _{3 -5-NH 2 -2-Py]} , [BA2022; 4-CF 3 -5-NH 2 -2-Py], [BA2023; 6-CF 3 -5-NH 2 -2-Py], [BA2024; _{3-CN-5-NH 2} -2-Py], [BA2025; 4-CN-5-NH 2 -2-Py], [BA2026; 6-CN-5-NH 2 -2-Py], [BA2027 3-OMe-5-NH ₂ 2-Py !, [BA2028; 4-OMe-5-NH ₂ 2-Py], [BA 2029; 6-OMe-5-NH ₂ 2-Py], _{BA2030; 6-NH 2 -2-} Py], [BA2031; 3-Cl-6-NH 2 -2-Py], [BA2032; 4-Cl-6-NH 2 -2-Py], [BA2033; 5 _{-Cl-6-NH 2 -2-} Py], [BA2034; 3-Me-6-NH 2 -2-Py], [BA2035; 4-Me-6-NH 2 -2-Py], [BA2036; _{5-Me-6-NH 2} -2-Py], [BA2037; 3-CF 3 -6-NH 2 -2-Py], [BA2038; 4-CF 3 -6-NH 2 -2-Py], _{[BA2039; 5-CF 3 -6} -NH 2 -2-Py], [BA2040; 3-CN-6-NH 2 -2-Py], [BA2041; 4-CN-6-NH 2 -2-Py ], [BA2042; 5-CN -6-NH 2 -2-Py], [BA2043; 3-OMe-6-NH 2 -2-Py], [BA2044; 4-OMe-6-NH 2 -2- Py], [BA 2045; 5-OMe-6-NH ₂ 2-Py], [BA 2046; 3-NHMe-2-Py], [BA 2047; 4-Cl-3-NHMe-2-Py], [BA 2048 5-Cl-3-NHMe-2-Py !, [BA2049; 6-Cl-3-NHMe-2-Py], [BA2050; 4-Me-3-NHMe-2-Py], [BA2051; -Me-3-NHMe-2- Py], [BA2052; 6-Me-3-NHMe-2-Py], [BA2053; 4-CF 3 -3-NHMe-2-Py], [BA2054; 5- _{CF 3 -3-NHMe-2-} Py], [BA2055; 6-CF 3 -3-NHMe-2-Py], [BA2056; 4-CN-3-NHMe-2-Py], [BA2057; 5- CN-3-NHMe-2-Py], [BA2 058; 6-CN-3-NHMe-2-Py, [BA 2059; 4-OMe-3-NHMe-2-Py], [BA 2060; 5-OMe-3-NHMe-2-Py], [BA 2061; 6-OMe-3-NHMe-2-Py, [BA2062; 4-NHMe-2-Py], [BA2063; 3-Cl-4-NHMe-2-Py], [BA 2064; 5-Cl-4- NHMe-2-Py, [BA 2065; 6-Cl-4-NHMe-2-Py], [BA 2066; 3-Me-4-NHMe-2-Py], [BA 2067; 5-Me-4-NHMe- 2-Py], [BA2068; 6-Me-4-NHMe-2-Py], [BA2069; 3-CF 3 -4-NHMe-2-Py], [BA2070; 5-CF 3 -4-NHMe- 2-Py], [BA2071; 6-CF 3 -4-NHMe-2-Py], [BA2072; 3-CN-4-NHMe-2-Py], [BA2073; 5-CN-4-NHMe-2 -Py], [BA 2074; 6-CN-4-NHMe-2-Py], [BA 2075; 3-OMe-4-NHMe-2-Py], [BA 2076; 5-OMe-4-NHMe-2-Py ], [BA 2077; 6-OMe-4-NHMe-2-Py], [BA 2078; 5-NHMe-2-Py], [BA 2079; 3-Cl-5-NHMe-2-Py], [BA 2080; 4] -Cl-5-NHMe-2-Py, [BA2081; 6-Cl-5-NHMe-2-Py], [BA2082; 3-Me-5-NHMe-2-Py], [BA2083; 4-Me -5-NHMe-2-Py], [BA2084; 6-Me-5-NHMe-2-Py],

_{[BA2085; 3-CF 3 -5} -NHMe-2-Py], [BA2086; 4-CF 3 -5-NHMe-2-Py], [BA2087; 6-CF 3 -5-NHMe-2-Py] [BA 2088; 3-CN-5-NHMe-2-Py], [BA 2089; 4-CN-5-NHMe-2-Py], [BA 2090; 6-CN-5-NHMe-2-Py], [BA 20 88; BA2091; 3-OMe-5-NHMe-2-Py], [BA2092; 4-OMe-5-NHMe-2-Py], [BA2093; 6-OMe-5-NHMe-2-Py], [BA 2094; 6-NHMe-2-Py, [BA 2095; 3-Cl-6-NHMe-2-Py], [BA 2096; 4-Cl-6-NHMe-2-Py], [BA 2097; 5-Cl-6- NHMe-2-Py, [BA 2098; 3-Me-6-NHMe-2-Py], [BA 2099; 4-Me-6-NHMe-2-Py], [BA 2 100; 5-Me-6-NHMe- 2-Py], [BA2101; 3-CF 3 -6-NHMe-2-Py], [BA2102; 4-CF 3 -6-NHMe-2-Py], [BA2103; 5-CF 3 -6-NHMe -2-Py !, [BA2104; 3-CN-6-NHMe-2-Py], [BA2105; 4-CN-6-NHMe-2-Py], [BA2106; 5-CN-6-NHMe-2 -Py], [BA2107; 3-OMe-6-NHMe-2-Py], [BA2108; 4-OMe-6-NHMe-2-Py], [BA2109; 5-OMe-6-NHMe-2-Py ], [BA2110; 3-NMe 2 -2-Py], [BA2111; 4-Cl-3-NMe 2 -2-Py], [BA2112; 5-Cl-3-NMe 2 -2-Py], [ BA2113; 6-Cl-3- NMe 2 -2-Py], [BA2114; 4-Me-3-NMe 2 -2-Py], [BA2115; 5-Me-3-NMe 2 -2-Py], [BA2116; 6-Me-3 -NMe 2 -2-Py], [BA2117; 4-CF 3 -3-NMe 2 -2-Py], [BA2118; 5-CF 3 -3-NMe 2 -2- Py], [BA2119; 6- CF 3 -3-NMe 2 -2-Py], [BA2120; 4-CN-3-NMe 2 -2-Py], [BA2121; 5-CN-3-NMe _{2 -2-Py], [BA2122} ; 6-CN-3-NMe 2 -2-Py], [BA2123; 4-OMe-3-NMe 2 -2-Py], [BA2124; 5-OMe-3- _{NMe 2 -2-Py], [} BA2125; 6-OMe-3-NMe 2 -2-Py], [BA2126; 4-NMe 2 -2-Py], [BA2127; 3-Cl-4-NMe 2 - 2-Py], [BA2128; 5-Cl-4-NMe 2 -2-Py], [BA2129; 6-Cl-4-NMe 2 -2-Py], [BA2130; 3-Me-4-NMe 2 -2-Py], [BA2131; 5-Me-4-NMe 2 -2-Py], [BA2132; 6-Me-4-NMe 2 -2-Py], [BA2133; 3-CF 3 -4- _{NMe 2 -2-Py], [} BA2134; 5-CF 3 -4-NMe 2 -2-Py], [BA2135; 6-CF 3 -4-NMe 2 -2-Py], [BA2136; 3-CN _{-4-NMe 2 -2-Py]} , [BA2137; 5-CN-4-NMe 2 -2-Py], [BA2138; 6-CN-4-NMe 2 -2-Py], [BA2139; 3- _{OMe-4-NMe 2 -2-} Py], [BA2140; 5-OMe-4-NMe 2 -2-Py], [BA2141; 6-OMe-4-NMe 2 -2-Py], [BA2142; 5 _{-NMe 2 -2-Py], [} BA2143; 3-Cl-5-NMe 2 -2-Py], [BA2144; 4-Cl-5-NMe 2 -2-Py], [BA2145; 6-Cl- _{5-NMe 2 -2-Py]} , [BA2146; 3-Me-5-NMe 2 -2-Py], [BA2147; 4-Me-5-NMe 2 -2-Py], [BA2148; 6-Me -5-NMe ₂ -2-Py !, [BA 2149; 3-CF ₃ -5-NMe ₂ -2-Py], [BA 2 150; 4-CF ₃ -5-NMe ₂ -2-Py], [BA 2 51; _{6-CF 3 -5-NMe 2} -2-Py], [BA2152; 3-CN-5-NMe 2 -2-Py], [BA2153; 4-CN-5-NMe 2 -2-Py], [ BA2154; 6-CN-5- NMe 2 -2-Py], [BA2155; 3-OMe-5-NMe 2 -2-Py], [BA2156; 4-OMe-5-NMe 2 -2 -Py], [BA2157; 6- OMe-5-NMe 2 -2-Py], [BA2158; 6-NMe 2 -2-Py], [BA2159; 3-Cl-6-NMe 2 -2-Py] , [BA2160; 4-Cl- 6-NMe 2 -2-Py], [BA2161; 5-Cl-6-NMe 2 -2-Py], [BA2162; 3-Me-6-NMe 2 -2-Py ], [BA2163; 4-Me -6-NMe 2 -2-Py], [BA2164; 5-Me-6-NMe 2 -2-Py], [BA2165; 3-CF 3 -6-NMe 2 -2 -Py], [BA2166; 4- CF 3 -6-NMe 2 -2-Py], [BA2167; 5-CF 3 -6-NMe 2 -2-Py], [BA2168; 3-CN-6-NMe ₂ -2-Py !, [BA2169; 4-CN-6-NMe ₂ -2-Py], [BA 2170; 5-CN-6-NMe ₂ -2-Py], [BA 2171; 3-OMe -6- _{NMe 2 -2-Py], [} BA2172; 4-OMe-6-NMe 2 -2-Py], [BA2173; 5-OMe-6-NMe 2 -2-Py], [BA2174; 3-ACNH-2 -Py], [BA2175; 4-Cl-3-ACNH-2-Py], [BA2176; 5-Cl-3-ACNH-2-Py], [BA2177; 6-Cl-3-ACNH-2-Py ], [BA2178; 4-Me-3-ACNH-2-Py], [BA2179; 5-Me-3-ACNH-2-Py], [BA2180; 6-Me-3-ACNH-2-Py], _{[BA2181; 4-CF 3 -3} -ACNH-2-Py], [BA2182; 5-CF 3 -3-ACNH-2-Py], [BA2183; 6-CF 3 -3-ACNH-2-Py] , [BA 2184; 4-CN-3-ACNH-2-Py],

[BA2185; 5-CN-3-ACNH-2-Py], [BA2186; 6-CN-3-ACNH-2-Py], [BA2187; 4-OMe-3-ACNH-2-Py], [BA2188 5-OMe-3-ACNH-2-Py !, [BA2189; 6-OMe-3-ACNH-2-Py], [BA2190; 4-ACNH-2-Py], [BA2191; 3-Cl-4; -ACNH-2-Py], [BA2192; 5-Cl-4-ACNH-2-Py], [BA2193; 6-Cl-4-ACNH-2-Py], [BA2194; 3-Me-4-ACNH -2-Py], [BA2195; 5-Me-4-ACNH-2-Py], [BA2196; 6-Me-4-ACNH-2-Py], [BA2197; 3-CF 3 -4-ACNH- 2-Py], [BA2198; 5-CF 3 -4-ACNH-2-Py], [BA2199; 6-CF 3 -4-ACNH-2-Py], [BA2200; 3-CN-4-ACNH- 2-Py], [BA2201; 5-CN-4-ACNH-2-Py], [BA2202; 6-CN-4-ACNH-2-Py], [BA2203; 3-OMe-4-ACNH-2- Py], [BA2204; 5-OMe-4-ACNH-2-Py], [BA2205; 6-OMe-4-ACNH-2-Py], [BA2206; 5-ACNH-2-Py], [BA2207; 3-Cl-5-ACNH-2-Py, [BA2208; 4-Cl-5-ACNH-2-Py], [BA2209; 6-Cl-5-ACNH-2-Py], [BA2210; Me-5-ACNH-2- Py], [BA2211; 4-Me-5-ACNH-2-Py], [BA2212; 6-Me-5-ACNH-2-Py], [BA2213; 3-CF 3 -5-ACNH-2-Py] , [BA2214; 4-CF 3 -5-ACNH-2-Py], [BA2215; 6-CF 3 -5-ACNH-2-Py], [BA2216; 3-CN -5-ACNH-2-Py, [BA2217; 4-CN-5-ACNH-2-Py], [BA2218; 6-CN-5-ACNH-2-Py], [BA2219; 3-OMe-5 -ACNH-2-Py], [BA2220; 4-OMe-5-ACNH-2-Py], [BA2221; 6-OMe-5-ACNH-2-Py], [BA2222; 6-ACNH-2-Py ], [BA2223; 3-Cl-6-ACNH-2-Py], [BA2224; 4-Cl-6-ACNH-2-Py], [BA2225; 5-Cl-6-ACNH-2-Py], [BA2226] 3-Me-6-ACNH-2-Py !, [BA2227; 4-Me-6-ACNH-2-Py], [BA2228; 5-Me-6-ACNH-2-Py], [BA2229; _{-CF 3 -6-ACNH-2-} Py], [BA2230; 4-CF 3 -6-ACNH-2-Py], [BA2231; 5-CF 3 -6-ACNH-2-Py], [BA2232; 3-CN-6-ACNH-2-Py, [BA2233; 4-CN-6-ACNH-2-Py], [BA2234; 5-CN-6-ACNH-2-Py], [BA2235; OMe-6-ACNH-2-Py], [BA2236; 4-OMe-6-ACNH-2-Py], [BA2237; 5-OMe-6-ACNH-2-Py], [BA2238; (Ac) (Me))-2-Py] [BA2239; 4-Cl-3- (N (Ac) (Me))-2-Py], [BA2240; 5-Cl-3- (N (Ac)) (Me))-2-Py], [BA2241; 6-Cl-3- (N (Ac) (Me))-2-Py], [BA2242; 4-Me-3- (N (Ac) (Me) )) [2-Py], [BA 2243; 5-Me-3- (N (Ac) (Me))-2-Py], [BA 2244; 6-Me-3- (N (Ac) (Me)) -2-Py], [BA2245; 4-CF 3 -3- (N (Ac) (Me)) - 2-Py], [BA2246; 5-CF 3 -3- (N (Ac) (Me)) -2-Py], [BA2247; 6-CF 3 -3- (N (Ac) (Me)) - 2-Py], [BA2248; 4-CN-3- (N (Ac) (Me)) - 2-Py], [BA2249; 5-CN-3- (N (Ac) (Me))-2-Py], [BA2250; 6-CN-3- (N (Ac) (Me))-2-] Py], [BA2251; 4-OMe-3- (N (Ac) (Me))-2-Py], [BA2252; 5-OMe-3- (N (Ac) (Me))-2-Py] , [BA2253; 6-OMe-3- (N (Ac) (Me))-2-Py], [BA2254; 4- (N (Ac) (Me))-2-Py], [BA2255; Cl-4- (N (Ac) (Me))-2-Py], [BA 2256; 5-Cl-4- (N (Ac) (Me))-2-Py], [BA2257; 6-Cl-4- (N (Ac) (Me))-2-Py], [BA2258; 3-Me-4- (N (Ac) (Me))-2-Py], [BA2259; 5-Me-4- (N (Ac) (Me))-2-Py], [BA2260; 6- Me-4- (N (Ac) (Me)) - 2-Py], [BA2261; 3-CF 3 -4- (N (Ac) (Me)) - 2-Py], [BA2262; 5-CF _{3 -4- (N (Ac) (} Me)) - 2-Py], [BA2263; 6-CF 3 -4- (N (Ac) (Me)) - 2-Py], [BA2264; 3-CN -4- (N (Ac) (Me))-2-Py], [BA2265; 5-CN-4- (N (Ac) (Me))-2-Py], [BA2266; 6-CN-4 -(N (Ac) (Me))-2-Py], [BA2267; 3-OMe-4- (N (Ac) (Me))-2-Py], [BA2268; 5-OMe-4- (4) N (Ac) (Me))-2-Py], [BA2269; 6-OMe-4- (N (Ac) (Me))-2-Py], [BA2270; 5- (N (Ac) (Me) )) [2-Py], [BA2271; 3-Cl-5- (N (Ac) (Me))-2-Py], [BA2272; 4-Cl-5- (N (Ac) (Me)) -2-Py], [BA 2273; 6-Cl-5- (N (Ac) (Me))-2-Py], [BA 2274; 3-Me-5- (N (Ac) (Me))-2 -Py], [BA2275; 4-Me-5- (N (Ac) (Me))-2-Py], [BA2276; 6-Me-5- (N (Ac) (Me))-2-Py ], [BA2277; 3-CF 3 -5- (N (Ac) (Me)) - 2-Py], [BA2278; 4-CF 3 -5- (N (Ac) (Me)) - 2-Py ], [BA 2279; 6-CF ₃ -5- (N (Ac) (Me))-2-Py], [BA 2280; 3-CN-5- (N (Ac) (Me))-2-Py] , [BA2281; 4-CN-5- (N (Ac) (Me))-2-Py], [BA2282; 6-CN-5- (N (Ac) (Me))-2-Py], [BA2282; BA 2283; 3-OMe-5- (N (Ac) (Me))-2-Py], [BA2284; 4-OMe-5- (N (Ac) (Me))-2-Py],

[BA2285; 6-OMe-5- (N (Ac) (Me))-2-Py], [BA2286; 6- (N (Ac) (Me))-2-Py], [BA2287; 3-Cl -6- (N (Ac) (Me))-2-Py], [BA2288; 4-Cl-6- (N (Ac) (Me))-2-Py], [BA2289; 5-Cl-6 -(N (Ac) (Me))-2-Py], [BA 2290; 3-Me-6- (N (Ac) (Me))-2-Py], [BA 2291; 4-Me-6- ( N (Ac) (Me))-2-Py], [BA 2 229; 5-Me-6- (N (Ac) (Me))-2-Py], [BA 2293; 3-CF ₃ -6- (N (Ac) (Me)) - 2-Py], [BA2294; 4-CF 3 -6- (N (Ac) (Me)) - 2-Py], [BA2295; 5-CF 3 -6- (N (Ac) (Me))-2-Py], [BA2296; 3-CN-6- (N (Ac) (Me))-2-Py], [BA2297; 4-CN-6- (N (Ac) ) (Me))-2-Py], [BA2298; 5-CN-6- (N (Ac) (Me))-2-Py], [BA2299; 3-OMe-6- (N (Ac) ( Me))-2-Py], [BA2300; 4-OMe-6- (N (Ac) (Me))-2-Py], [BA2301; 5-OMe-6- (N (Ac) (Me)) )-[2-Py], [BA 2302; 3-AC-2-Py], [BA 2303; 4-Cl-3-AC-2-Py], [BA 2304; 5-Cl-3-AC-2-Py] , [BA2305; 6-Cl-3-AC-2-Py], [BA2306; 4-Me-3-AC-2-Py], [BA2307; 5-Me-3-AC-2-Py], [BA2305; BA 2308; 6-Me-3-AC-2-Py], [BA 2309; 4-CF ₃ -3-AC-2-Py], [BA 2310; 5-CF ₃ -3-AC-2-Py], [BA 23 10; _{BA2311; 6-CF 3 -3-} AC-2-Py], [BA2312; 4-CN-3-AC-2-Py], [BA2313; 5-CN-3-AC-2-Py], [BA2314 6-CN-3-AC-2-Py !, [BA2315; 4-OMe-3-AC-2-Py], [BA2316; 5-OMe-3-AC-2-Py], [BA2317; -OMe-3-AC-2-Py], [BA2318; 4-AC-2-Py], [BA2319; 3-Cl-4-AC-2-P y], [BA2320; 5-Cl-4-AC-2-Py], [BA2321; 6-Cl-4-AC-2-Py], [BA2322; 3-Me-4-AC-2-Py] , [BA2323; 5-Me- 4-AC-2-Py], [BA2324; 6-Me-4-AC-2-Py], [BA2325; 3-CF 3 -4-AC-2-Py], _{[BA2326; 5-CF 3 -4} -AC-2-Py], [BA2327; 6-CF 3 -4-AC-2-Py], [BA2328; 3-CN-4-AC-2-Py], [BA2329; 5-CN-4-AC-2-Py], [BA2330; 6-CN-4-AC-2-Py], [BA2331; 3-OMe-4-AC-2-Py], [BA2332 5-OMe-4-AC-2-Py !, [BA2333; 6-OMe-4-AC-2-Py], [BA2334; 5-AC-2-Py], [BA2335; 3-Cl-5; -AC-2-Py], [BA2336; 4-Cl-5-AC-2-Py], [BA2337; 6-Cl-5-AC-2-Py], [BA2338; 3-Me-5-AC -2-Py], [BA2339; 4-Me-5-AC-2-Py], [BA2340; 6-Me-5-AC-2-Py], [BA2341; 3-CF 3 -5-AC- 2-Py], [BA2342; 4-CF 3 -5-AC-2-Py], [BA2343; 6-CF 3 -5-AC-2-Py], [BA2344; 3-CN-5-AC- 2-Py], [BA2345; 4-CN-5-AC-2-Py], [BA2346; 6-CN-5-AC-2-Py], [BA2347; 3-OMe-5-AC-2-] Py], [BA2348; 4-OMe-5-AC-2-Py], [BA2349; 6-OMe-5-AC-2-Py], [BA2350; 6-AC-2-Py], [BA2351; 3-Cl-6-AC-2-Py], [BA2352; 4-Cl-6-AC-2-Py], [BA2353; 5-Cl-6-AC-2-Py], [BA2354; Me-6-AC-2- Py], [BA2355; 4-Me-6-AC-2-Py], [BA2356; 5-Me-6-AC-2-Py], [BA2357; 3-CF 3 -6-AC-2-Py] , [BA2358; 4-CF 3 -6-AC-2-Py], [BA2359; 5-CF 3 -6-AC-2-Py], [BA2360; 3-CN -6 -AC-2-Py], [BA2361; 4-CN-6-AC-2-Py], [BA2362; 5-CN-6-AC-2-Py], [BA2363; 3-OMe-6-AC -2-Py], [BA2364; 4-OMe-6-AC-2-Py], [BA2365; 5-OMe-6-AC-2-Py], [BA2366; 2-F-3-Py], [BA2367; 4-Cl-2-F-3-Py], [BA 2368; 5-Cl-2-F-3-Py], [BA 2369; 6-Cl-2-F-3-Py], [BA 2370] 4-Me-2-F-3-Py !, [BA 2371; 5-Me-2-F-3-Py], [BA 2372; 6-Me-2-F-3-Py], [BA 2373; _{-CF 3 -2-F-3-} Py], [BA2374; 5-CF 3 -2-F-3-Py], [BA2375; 6-CF 3 -2-F-3-Py], [BA2376; 4-CN-2-F-3-Py, [BA2377; 5-CN-2-F-3-Py], [BA2378; 6-CN-2-F-3-Py], [BA2379; OMe-2-F-3-Py, [BA2380; 5-OMe-2-F-3-Py], [BA2381; 6-OMe-2-F-3-Py], [BA2382; 4-F- 3-Py], [BA2383; 2-Cl-4-F-3-Py], [BA2384; 5-Cl-4-F-3-Py],

[BA2385; 6-Cl-4-F-3-Py], [BA2386; 2-Me-4-F-3-Py], [BA2387; 5-Me-4-F-3-Py], [BA2388] ; 6-Me-4-F -3-Py], [BA2389; 2-CF 3 -4-F-3-Py], [BA2390; 5-CF 3 -4-F-3-Py], [BA2391 _{; 6-CF 3 -4-F} -3-Py], [BA2392; 2-CN-4-F-3-Py], [BA2393; 5-CN-4-F-3-Py], [BA2394; 6-CN-4-F-3-Py !, [BA2395; 2-OMe-4-F-3-Py], [BA2396; 5-OMe-4-F-3-Py], [BA2397; OMe-4-F-3-Py], [BA2398; 5-F-3-Py], [BA2399; 2-Cl-5-F-3-Py], [BA2400; 4-Cl-5-F- 3-Py], [BA 2401; 6-Cl-5-F-3-Py], [BA 2402; 2-Me-5-F-3-Py], [BA 2403; 4-Me-5-F-3- Py], [BA2404; 6- Me-5-F-3-Py], [BA2405; 2-CF 3 -5-F-3-Py], [BA2406; 4-CF 3 -5-F-3- Py], [BA2407; 6- CF 3 -5-F-3-Py], [BA2408; 2-CN-5-F-3-Py], [BA2409; 4-CN-5-F-3-Py ], [BA 2410; 6-CN-5-F-3-Py], [BA 2411; 2-OMe-5-F-3-Py], [BA 2412; 4-OMe-5-F-3-Py], [BA2413; 6-OMe-5-F-3-Py], [BA2414; 6-F-3-Py], [BA2415; 2-Cl-6-F-3-Py], [BA2416; 4-Cl -6-F-3-Py], [BA2417; 5-Cl-6-F-3-Py], [BA2418; 2-Me-6-F-3-Py], [BA2419; 4-Me-6 -F-3-Py], [ BA2420; 5-Me-6-F-3-Py], [BA2421; 2-CF 3 -6-F-3-Py], [BA2422; 4-CF 3 -6 -F-3-Py], [ BA2423; 5-CF 3 -6-F-3-Py], [BA2424; 2-CN-6-F-3-Py], [BA2425; 4-CN-6- F-3-Py], [BA2426; 5-CN-6-F-3-Py], [BA2427; 2-O Me-6-F-3-Py], [BA2428; 4-OMe-6-F-3-Py], [BA2429; 5-OMe-6-F-3-Py], [BA2430; 2-Cl- 3-Py], [BA2431; 4-Cl-2-Cl-3-Py], [BA2432; 5-Cl-2-Cl-3-Py], [BA2433; 6-Cl-2-Cl-3- Py], [BA2434; 4-Me-2-Cl-3-Py], [BA2435; 5-Me-2-Cl-3-Py], [BA2436; 6-Me-2-Cl-3-Py] _{, [BA2437; 4-CF 3} -2-Cl-3-Py], [BA2438; 5-CF 3 -2-Cl-3-Py], [BA2439; 6-CF 3 -2-Cl-3-Py ], [BA2440; 4-CN-2-Cl-3-Py], [BA2441; 5-CN-2-Cl-3-Py], [BA2442; 6-CN-2-Cl-3-Py], [BA2443; 4-OMe-2-Cl-3-Py], [BA2444; 5-OMe-2-Cl-3-Py], [BA2445; 6-OMe-2-Cl-3-Py], [BA2446] 4-Cl-3-Py !, [BA2447; 2-Cl-4-Cl-3-Py], [BA2448; 5-Cl-4-Cl-3-Py], [BA2449; 6-Cl-4 -Cl-3-Py, [BA2450; 2-Me-4-Cl-3-Py], [BA2451; 5-Me-4-Cl-3-Py], [BA2452; 6-Me-4-Cl -3-Py], [BA2453; 2-CF 3 -4-Cl-3-Py], [BA2454; 5-CF 3 -4-Cl-3-Py], [BA2455; 6-CF 3 -4- Cl-3-Py, [BA2456; 2-CN-4-Cl-3-Py], [BA2457; 5-CN-4-Cl-3-Py], [BA2458; 6-CN-4-Cl- 3-Py], [BA2459; 2-OMe-4-Cl-3-Py], [BA2460; 5-OMe-4-Cl-3-Py], [BA2461; 6-OMe-4-Cl-3- Py], [BA2462; 5-Cl-3-Py], [BA2463; 4-Cl-5-Cl-3-Py], [BA2464; 5-Cl-5-Cl-3-Py], [BA2465; 6-Cl-5-Cl-3-Py, [BA2466; 4-Me-5-Cl-3-Py], [BA2467; 5-Me-5-Cl-3-Py], [BA2468; 6- Me-5-Cl- 3-Py], [BA2469; 4-CF 3 -5-Cl-3-Py], [BA2470; 5-CF 3 -5-Cl-3-Py], [BA2471; 6-CF 3 -5-Cl -3-Py !, [BA2472; 4-CN-5-Cl-3-Py], [BA2473; 3-CN-5-Cl-3-Py], [BA2474; 6-CN-5-Cl-3 -Py], [BA2475; 4-OMe-5-Cl-3-Py], [BA2476; 5-OMe-5-Cl-3-Py], [BA2477; 6-OMe-5-Cl-3-Py ], [BA2478; 6-Cl-3-Py], [BA2479; 2-Cl-6-Cl-3-Py], [BA2480; 4-Cl-6-Cl-3-Py], [BA2481; -Cl-6-Cl-3-Py], [BA2482; 2-Me-6-Cl-3-Py], [BA2483; 4-Me-6-Cl-3-Py], [BA2484; 5-Me -6-Cl-3-Py],

_{[BA2485; 2-CF 3 -6} -Cl-3-Py], [BA2486; 4-CF 3 -6-Cl-3-Py], [BA2487; 5-CF 3 -6-Cl-3-Py] , [BA2488; 2-CN-6-Cl-3-Py], [BA2489; 4-CN-6-Cl-3-Py], [BA2490; 5-CN-6-Cl-3-Py], [BA2488; BA2491; 2-OMe-6-Cl-3-Py], [BA2492; 4-OMe-6-Cl-3-Py], [BA2493; 5-OMe-6-Cl-3-Py], [BA2494; 2-Br-3-Py !, [BA2495; 4-Cl-2-Br-3-Py], [BA2496; 5-Cl-2-Br-3-Py], [BA 2497; 6-Cl-2- Br-3-Py, [BA2498; 4-Me-2-Br-3-Py], [BA2499; 5-Me-2-Br-3-Py], [BA2500; 6-Me-2-Br- 3-Py], [BA2501; 4-CF 3 -2-Br-3-Py], [BA2502; 5-CF 3 -2-Br-3-Py], [BA2503; 6-CF 3 -2-Br -3-Py !, [BA2504; 4-CN-2-Br-3-Py], [BA2505; 5-CN-2-Br-3-Py], [BA2506; 6-CN-2-Br-3 -Py], [BA2507; 4-OMe-2-Br-3-Py], [BA2508; 5-OMe-2-Br-3-Py], [BA2509; 6-OMe-2-Br-3-Py ], [BA 2510; 4-Br-3-Py], [BA 2511; 2-Cl-4-Br-3-Py], [BA 2512; 5-Cl-4-Br-3-Py], [BA 2513; 6] -Cl-4-Br-3-Py], [BA 2514; 2-Me-4-Br-3-Py], [BA 2515; 5-Me-4-Br-3-Py], [BA 2516; 6-Me -4-Br-3-Py] , [BA2517; 2-CF 3 -4-Br-3-Py], [BA2518; 5-CF 3 -4-Br-3-Py], [BA2519; 6-CF _{3 -4-Br-3-Py} ], [BA2520; 2-CN-4-Br-3-Py], [BA2521; 5-CN-4-Br-3-Py], [BA2522; 6-CN- 4-Br-3-Py, [BA2523; 2-OMe-4-Br-3-Py], [BA2524; 5-OMe-4-Br-3-Py], [BA2525; 6-OMe-4 -Br-3-Py], [BA2526; 5-Br-3-Py], [BA2527; 2-Cl-5-Br-3-Py], [BA2528; 4-Cl-5-Br-3-Py ], [BA 2529; 6-Cl-5-Br-3-Py], [BA 2530; 2-Me-5-Br-3-Py], [BA 2531; 4-Me-5-Br-3-Py], [BA2532; 6-Me-5 -Br-3-Py], [BA2533; 2-CF 3 -5-Br-3-Py], [BA2534; 4-CF 3 -5-Br-3-Py], _{[BA2535; 6-CF 3 -5} -Br-3-Py], [BA2536; 2-CN-5-Br-3-Py], [BA2537; 4-CN-5-Br-3-Py], [ 6-CN-5-Br-3-Py], [BA2539; 2-OMe-5-Br-3-Py], [BA2540; 4-OMe-5-Br-3-Py], [BA2541; 6-OMe-5-Br-3-Py, [BA 2542; 6-Br-3-Py], [BA 2543; 2-Cl-6-Br-3-Py], [BA 2544; 4-Cl-6- Br-3-Py, [BA2545; 5-Cl-6-Br-3-Py], [BA2546; 2-Me-6-Br-3-Py], [BA2547; 4-Me-6-Br- 3-Py], [BA2548; 5-Me-6-Br-3-Py], [BA2549; 2-CF 3 -6-Br-3-Py], [BA2550; 4-CF 3 -6-Br- 3-Py], [BA2551; 5-CF 3 -6-Br-3-Py], [BA2552; 2-CN-6-Br-3-Py], [BA2553; 4-CN-6-Br-3 -Py], [BA2554; 5-CN-6-Br-3-Py], [BA2555; 2-OMe-6-Br-3-Py], [BA2556; 4-OMe-6-Br-3-Py ], [BA2557; 5-OMe-6-Br-3-Py], [BA2558; 2-I-3-Py], [BA2559; 4-Cl-2-I-3-Py], [BA2560; -Cl-2-I-3-Py, [BA2561; 6-Cl-2-I-3-Py], [BA2562; 4-Me-2-I-3-Py], [BA2563; 5-Me -2-I-3-Py] , [BA2564; 6-Me-2-I-3-Py], [BA2565; 4-CF 3 -2-I-3-Py], [BA2566; 5-CF 3 -2-I-3-Py], _{[BA2567; 6-CF 3 -2} -I-3-Py], [BA2568; 4-CN-2-I-3-Py], [BA2569; 5-CN-2-I-3-Py], [ BA2570; 6-CN-2-I-3-Py], [BA2571; 4-OMe-2-I-3-Py], [BA2572; 5-OMe-2-I-3-Py], [BA2573; 6-OMe-2-I-3-Py, [BA2574; 4-I-3-Py], [BA2575; 2-Cl-4-I-3-Py], [BA2576; 5-Cl-4- I-3-Py, [BA2577; 6-Cl-4-I-3-Py], [BA2578; 2-Me-4-I-3-Py], [BA2579; 5-Me-4-I- 3-Py], [BA2580; 6-Me-4-I-3-Py], [BA2581; 2-CF 3 -4-I-3-Py], [BA2582; 5-CF 3 -4-I- 3-Py], [BA2583; 6-CF 3 -4-I-3-Py], [BA2584; 2-CN-4-I-3-Py],

[BA2585; 5-CN-4-I-3-Py], [BA2586; 6-CN-4-I-3-Py], [BA2587; 2-OMe-4-I-3-Py], [BA2588] 5-OMe-4-I-3-Py !, [BA2589; 6-OMe-4-I-3-Py], [BA2590; 5-I-3-Py], [BA2591; 2-Cl-5; -I-3-Py, [BA2592; 4-Cl-5-I-3-Py], [BA2593; 6-Cl-5-I-3-Py], [BA2594; 2-Me-5-I -3-Py], [BA2595; 4-Me-5-I-3-Py], [BA2596; 6-Me-5-I-3-Py], [BA2597; 2-CF 3 -5-I- 3-Py], [BA2598; 4-CF 3 -5-I-3-Py], [BA2599; 6-CF 3 -5-I-3-Py], [BA2600; 2-CN-5-I- 3-Py], [BA2601; 4-CN-5-I-3-Py], [BA2602; 6-CN-5-I-3-Py], [BA2603; 2-OMe-5-I-3-3 Py], [BA2604; 4-OMe-5-I-3-Py], [BA2605; 6-OMe-5-I-3-Py], [BA2606; 6-I-3-Py], [BA2607; 2-Cl-6-I-3-Py, [BA2608; 4-Cl-6-I-3-Py], [BA2609; 5-Cl-6-I-3-Py], [BA 2610; Me-6-I-3- Py], [BA2611; 4-Me-6-I-3-Py], [BA2612; 5-Me-6-I-3-Py], [BA2613; 2-CF 3 -6-I-3-Py] , [BA2614; 4-CF 3 -6-I-3-Py], [BA2615; 5-CF 3 -6-I-3-Py], [BA2616; 2-CN -6-I-3-Py !, [BA2617; 4-CN-6-I-3-Py], [BA2618; 5-CN-6-I-3-Py], [BA2619; 2-OMe-6 -I-3-Py], [BA2620; 4-OMe-6-I-3-Py], [BA2621; 5-OMe-6-I-3-Py], [BA2622; 2-Me-3-Py ], [BA2623; 4-Cl-2-Me-3-Py], [BA2624; 5-Cl-2-Me-3-Py], [BA2625; 6-Cl-2-Me-3-Py], [BA2626; 4-Me-2-Me-3-Py], [BA2627; 5-Me-2-Me -3-Py], [BA2628; 6-Me-2-Me-3-Py], [BA2629; 4-CF 3 -2-Me-3-Py], [BA2630; 5-CF 3 -2-Me -3-Py], [BA2631; 6-CF 3 -2-Me-3-Py], [BA2632; 4-CN-2-Me-3-Py], [BA2633; 5-CN-2-Me- 3-Py], [BA2634; 6-CN-2-Me-3-Py], [BA2635; 4-OMe-2-Me-3-Py], [BA2636; 5-OMe-2-Me-3- Py], [BA2637; 6-OMe-2-Me-3-Py], [BA2638; 4-Me-3-Py], [BA2639; 2-Cl-4-Me-3-Py], [BA2640; 5-Cl-4-Me-3-Py !, [BA2641; 6-Cl-4-Me-3-Py], [BA2642; 2-Me-4-Me-3-Py], [BA2643; 5- Me-4-Me-3- Py], [BA2644; 6-Me-4-Me-3-Py], [BA2645; 2-CF 3 -4-Me-3-Py], [BA2646; 5-CF ₃ -4-Me-3-Py !, [BA2647; 6-CF ₃ -4-Me-3-Py], [BA 2648; 2-CN-4-Me-3-Py], [BA 2649; 5-CN -4-Me-3-Py !, [BA2650; 6-CN-4-Me-3-Py], [BA2651; 2-OMe-4-Me-3-Py], [BA2652; 5-OMe-4 -Me-3-Py], [BA2653; 6-OMe-4-Me-3-Py], [BA2654; 5-Me-3-Py], [BA2655; 2-Cl-5-Me-3-Py ], [BA2656; 4-Cl-5-Me-3-Py], [BA2657; 6-Cl-5-Me-3-Py], [BA2658; 2-Me-5-Me-3-Py], [BA2659; 4-Me-5 -Me-3-Py], [BA2660; 6-Me-5-Me-3-Py], [BA2661; 2-CF 3 -5-Me-3-Py], [ _{BA2662; 4-CF 3 -5-} Me-3-Py], [BA2663; 6-CF 3 -5-Me-3-Py], [BA2664; 2-CN-5-Me-3-Py], [ BA2665; 4-CN-5-Me-3-Py], [BA2666; 6-CN-5-Me-3-Py], [BA2667; 2-OMe-5-Me-3-Py], [BA2668; Four -OMe-5-Me-3-Py], [BA2669; 6-OMe-5-Me-3-Py], [BA2670; 6-Me-3-Py], [BA 2671; 2-Cl-6-Me -3-Py], [BA 2672; 4-Cl-6-Me-3-Py], [BA 2673; 5-Cl-6-Me-3-Py], [BA 2674; 2-Me-6-Me-3 -Py], [BA2675; 4- Me-6-Me-3-Py], [BA2676; 5-Me-6-Me-3-Py], [BA2677; 2-CF 3 -6-Me-3- Py], [BA2678; 4- CF 3 -6-Me-3-Py], [BA2679; 5-CF 3 -6-Me-3-Py], [BA2680; 2-CN-6-Me-3- Py], [BA2681; 4-CN-6-Me-3-Py], [BA2682; 5-CN-6-Me-3-Py], [BA2683; 2-OMe-6-Me-3-Py] , [BA2684; 4-OMe-6-Me-3-Py],

[BA2685; 5-OMe-6-Me-3-Py], [BA2686; 2-OMe-3-Py], [BA2687; 4-Cl-2-OMe-3-Py], [BA2688; 5-Cl -2-OMe-3-Py !, [BA2689; 6-Cl-2-OMe-3-Py], [BA2690; 4-Me-2-OMe-3-Py], [BA2691; 5-Me-2 -OMe-3-Py], [ BA2692; 6-Me-2-OMe-3-Py], [BA2693; 4-CF 3 -2-OMe-3-Py], [BA2694; 5-CF 3 -2 -OMe-3-Py], [ BA2695; 6-CF 3 -2-OMe-3-Py], [BA2696; 4-CN-2-OMe-3-Py], [BA2697; 5-CN-2- OMe-3-Py, [BA2698; 6-CN-2-OMe-3-Py], [BA2699; 4-OMe-2-OMe-3-Py], [BA2700; 5-OMe-2-OMe- 3-Py], [BA2701; 6-OMe-2-OMe-3-Py], [BA2702; 4-OMe-3-Py], [BA2703; 2-Cl-4-OMe-3-Py], [BA2702; BA2704; 5-Cl-4-OMe-3-Py], [BA2705; 6-Cl-4-OMe-3-Py], [BA2706; 2-Me-4-OMe-3-Py], [BA2707; 5-Me-4-OMe- 3-Py], [BA2708; 6-Me-4-OMe-3-Py], [BA2709; 2-CF 3 -4-OMe-3-Py], [BA2710; 5 _{-CF 3 -4-OMe-3-} Py], [BA2711; 6-CF 3 -4-OMe-3-Py], [BA2712; 2-CN-4-OMe-3-Py], [BA2713; 5 -CN-4-OMe-3-Py], [BA2714; 6-CN-4-OMe-3-Py], [BA2715; 2-OMe-4-OMe-3-Py], [BA2716; 5-OMe -4-OMe-3-Py !, [BA2717; 6-OMe-4-OMe-3-Py], [BA2718; 5-OMe-3-Py], [BA2719; 2-Cl-5-OMe-3 -Py], [BA2720; 4-Cl-5-OMe-3-Py], [BA2721; 6-Cl-5-OMe-3-Py], [BA2722; 2-Me-5-OMe-3-Py ], [BA 2723; 4-Me-5-OMe-3-Py], [BA 2724; 6-Me-5-O Me-3-Py], [ BA2725; 2-CF 3 -5-OMe-3-Py], [BA2726; 4-CF 3 -5-OMe-3-Py], [BA2727; 6-CF 3 -5 -OMe-3-Py], [BA2728; 2-CN-5-OMe-3-Py], [BA2729; 4-CN-5-OMe-3-Py], [BA2730; 6-CN-5-OMe -3-Py, [BA 2731; 2-OMe-5-OMe-3-Py], [BA 2732; 4-OMe-5-OMe-3-Py], [BA 2733; 6-OMe-5-OMe-3 -Py], [BA2734; 6-OMe-3-Py], [BA2735; 2-Cl-6-OMe-3-Py], [BA2736; 4-Cl-6-OMe-3-Py], [BA2737] 5-Cl-6-OMe-3-Py !, [BA2738; 2-Me-6-OMe-3-Py], [BA2739; 4-Me-6-OMe-3-Py], [BA2740; -Me-6-OMe-3- Py], [BA2741; 2-CF 3 -6-OMe-3-Py], [BA2742; 4-CF 3 -6-OMe-3-Py], [BA2743; 5 _{-CF 3 -6-OMe-3-} Py], [BA2744; 2-CN-6-OMe-3-Py], [BA2745; 4-CN-6-OMe-3-Py], [BA2746; 5- CN-6-OMe-3-Py !, [BA2747; 2-OMe-6-OMe-3-Py], [BA2748; 4-OMe-6-OMe-3-Py], [BA2749; 5-OMe- 6-OMe-3-Py] , [BA2750; 2-CF 3 -3-Py], [BA2751; 4-Cl-2-CF 3 -3-Py], [BA2752; 5-Cl-2-CF 3 -3-Py], [BA2753; 6-Cl-2-CF 3 -3-Py], [BA2754; 4-Me-2-CF 3 -3-Py], [BA2755; 5-Me-2-CF _{3 -3-Py], [BA2756} ; 6-Me-2-CF 3 -3-Py], [BA2757; 4-CF 3 -2-CF 3 -3-Py], [BA2758; 5-CF 3 - _{2-CF 3 -3-Py]} , [BA2759; 6-CF 3 -2-CF 3 -3-Py], [BA2760; 4-CN-2-CF 3 -3-Py], [BA2761; 5- _{CN-2-CF 3 -3-} Py], [BA2762; 6-CN-2-CF 3 -3-Py], [BA2763; 4-OMe-2-CF 3 -3-Py], [BA2764; 5-OMe-2-CF 3 -3-Py], [BA2765; 6-OMe-2-CF _{3 -3-Py], [BA2766} ; 4-CF 3 -3-Py], [BA2767; 2-Cl-4-CF 3 -3-Py], [BA2768; 5-Cl-4-CF 3 -3 -Py], [BA2769; 6- Cl-4-CF 3 -3-Py], [BA2770; 2-Me-4-CF 3 -3-Py], [BA2771; 5-Me-4-CF 3 - 3-Py], [BA2772; 6-Me-4-CF 3 -3-Py], [BA2773; 2-CF 3 -4-CF 3 -3-Py], [BA2774; 5-CF 3 -4- _{CF 3 -3-Py], [} BA2775; 6-CF 3 -4-CF 3 -3-Py], [BA2776; 2-CN-4-CF 3 -3-Py], [BA2777; 5-CN- _{4-CF 3 -3-Py]} , [BA2778; 6-CN-4-CF 3 -3-Py], [BA2779; 2-OMe-4-CF 3 -3-Py], [BA2780; 5-OMe _{-4-CF 3 -3-Py]} , [BA2781; 6-OMe-4-CF 3 -3-Py], [BA2782; 5-CF 3 -3-Py], [BA2783; 2-Cl-5- CF ₃ -3-Py], [BA 2784; 4-Cl-5-CF ₃ -3-Py],

[BA2785; 6-Cl-5 -CF 3 -3-Py], [BA2786; 2-Me-5-CF 3 -3-Py], [BA2787; 4-Me-5-CF 3 -3-Py] , [BA2788; 6-Me- 5-CF 3 -3-Py], [BA2789; 2-CF 3 -5-CF 3 -3-Py], [BA2790; 4-CF 3 -5-CF 3 -3 -Py], [BA2791; 6- CF 3 -5-CF 3 -3-Py], [BA2792; 2-CN-5-CF 3 -3-Py], [BA2793; 4-CN-5-CF 3 -3-Py], [BA2794; 6-CN-5-CF 3 -3-Py], [BA2795; 2-OMe-5-CF 3 -3-Py], [BA2796; 4-OMe-5-CF _{3 -3-Py], [BA2797} ; 6-OMe-5-CF 3 -3-Py], [BA2798; 6-CF 3 -3-Py], [BA2799; 2-Cl-6-CF 3 -3 -Py], [BA2800; 4- Cl-6-CF 3 -3-Py], [BA2801; 5-Cl-6-CF 3 -3-Py], [BA2802; 2-Me-6-CF 3 - 3-Py], [BA2803; 4-Me-6-CF 3 -3-Py], [BA2804; 5-Me-6-CF 3 -3-Py], [BA2805; 2-CF 3 -6-CF _{3 -3-Py], [BA2806} ; 4-CF 3 -6-CF 3 -3-Py], [BA2807; 5-CF 3 -6-CF 3 -3-Py], [BA2808; 2-CN- _{6-CF 3 -3-Py]} , [BA2809; 4-CN-6-CF 3 -3-Py], [BA2810; 5-CN-6-CF 3 -3-Py], [BA2811; 2-OMe _{-6-CF 3 -3-Py]} , [BA2812; 4-OMe-6-CF 3 -3-Py], [BA2813; 5-OMe-6-CF 3 -3-Py], [BA2814; 2- _{OCF 3 -3-Py], [} BA2815; 4-Cl-2-OCF 3 -3-Py], [BA2816; 5-Cl-2-OCF 3 -3-Py], [BA2817; 6-Cl-2 _{-OCF 3 -3-Py], [} BA2818; 4-Me-2-OCF 3 -3-Py], [BA2819; 5-Me-2-OCF 3 -3-Py], [BA2820; 6-Me- 2-OCF ₃ -3-Py], [BA2821 _{; 4-CF 3 -2-OCF} 3 -3-Py], [BA2822; 5-CF 3 -2-OCF 3 -3-Py], [BA2823; 6-CF 3 -2-OCF 3 -3-Py ], [BA2824; 4-CN -2-OCF 3 -3-Py], [BA2825; 5-CN-2-OCF 3 -3-Py], [BA2826; 6-CN-2-OCF 3 -3- Py], [BA2827; 4- OMe-2-OCF 3 -3-Py], [BA2828; 5-OMe-2-OCF 3 -3-Py], [BA2829; 6-OMe-2-OCF 3 -3 -Py], [BA2830; 4- OCF 3 -3-Py], [BA2831; 2-Cl-4-OCF 3 -3-Py], [BA2832; 5-Cl-4-OCF 3 -3-Py] , [BA2833; 6-Cl- 4-OCF 3 -3-Py], [BA2834; 2-Me-4-OCF 3 -3-Py], [BA2835; 5-Me-4-OCF 3 -3-Py ], [BA2836; 6-Me -4-OCF 3 -3-Py], [BA2837; 2-CF 3 -4-OCF 3 -3-Py], [BA2838; 5-CF 3 -4-OCF 3 - 3-Py], [BA2839; 6-CF 3 -4-OCF 3 -3-Py], [BA2840; 2-CN-4-OCF 3 -3-Py], [BA2841; 5-CN-4-OCF _{3 -3-Py], [BA2842} ; 6-CN-4-OCF 3 -3-Py], [BA2843; 2-OMe-4-OCF 3 -3-Py], [BA2844; 5-OMe-4- _{OCF 3 -3-Py], [} BA2845; 6-OMe-4-OCF 3 -3-Py], [BA2846; 5-OCF 3 -3-Py], [BA2847; 2-Cl-5-OCF 3 - 3-Py], [BA2848; 4-Cl-5-OCF 3 -3-Py], [BA2849; 6-Cl-5-OCF 3 -3-Py], [BA2850; 2-Me-5-OCF 3 -3-Py], [BA2851; 4-Me-5-OCF 3 -3-Py], [BA2852; 6-Me-5-OCF 3 -3-Py], [BA2853; 2-CF 3 -5- OCF ₃ -3-Py], [BA 2 854; 4-CF ₃ -5-OCF ₃ -3-Py], [BA 2 855; 6-CF ₃ -5-OCF ₃ -3-Py], [BA 2 856; 2-CN-5- OCF 3 -3-Py], [BA2857; 4-CN-5-OCF 3 -3-Py], [BA2858; 6-CN-5-OCF 3 -3-Py], [BA 2859; 2-OMe-5-OCF ₃ -3-Py], [BA 2860; 4-OMe -5-OCF ₃ -3-Py], [BA 2 861; 6-OMe -5-OCF ₃ -3-Py] _{, [BA2862; 6-OCF 3} -3-Py], [BA2863; 2-Cl-6-OCF 3 -3-Py], [BA2864; 4-Cl-6-OCF 3 -3-Py], [BA2865 ; 5-Cl-6-OCF 3 -3-Py], [BA2866; 2-Me-6-OCF 3 -3-Py], [BA2867; 4-Me-6-OCF 3 -3-Py], [ BA2868; 5-Me-6- OCF 3 -3-Py], [BA2869; 2-CF 3 -6-OCF 3 -3-Py], [BA2870; 4-CF 3 -6-OCF 3 -3-Py ], [BA2871; 5-CF 3 -6-OCF 3 -3-Py], [BA2872; 2-CN-6-OCF 3 -3-Py], [BA2873; 4-CN-6-OCF 3 -3 -Py], [BA2874; 5- CN-6-OCF 3 -3-Py], [BA2875; 2-OMe-6-OCF 3 -3-Py], [BA2876; 4-OMe-6-OCF 3 - 3-Py], [BA2877; 5-OMe-6-OCF 3 -3-Py], [BA2878; 2-CHF 2 -3-Py], [BA2879; 4-Cl-2-CHF 2 -3-Py ], [BA2880; 5-Cl -2-CHF 2 -3-Py], [BA2881; 6-Cl-2-CHF 2 -3-Py], [BA2882; 4-Me-2-CHF 2 -3- Py], [BA2883; 5- Me-2-CHF 2 -3-Py], [BA2884; 6-Me-2-CHF 2 -3-Py],

_{[BA2885; 4-CF 3 -2} -CHF 2 -3-Py], [BA2886; 5-CF 3 -2-CHF 2 -3-Py], [BA2887; 6-CF 3 -2-CHF 2 -3 -Py], [BA2888; 4- CN-2-CHF 2 -3-Py], [BA2889; 5-CN-2-CHF 2 -3-Py], [BA2890; 6-CN-2-CHF 2 - 3-Py], [BA2891; 4-OMe-2-CHF 2 -3-Py], [BA2892; 5-OMe-2-CHF 2 -3-Py], [BA2893; 6-OMe-2-CHF 2 -3-Py], [BA2894; 4-CHF 2 -3-Py], [BA2895; 2-Cl-4-CHF 2 -3-Py], [BA2896; 5-Cl-4-CHF 2 -3- Py], [BA2897; 6- Cl-4-CHF 2 -3-Py], [BA2898; 2-Me-4-CHF 2 -3-Py], [BA2899; 5-Me-4-CHF 2 -3 -Py], [BA2900; 6- Me-4-CHF 2 -3-Py], [BA2901; 2-CF 3 -4-CHF 2 -3-Py], [BA2902; 5-CF 3 -4-CHF _{2 -3-Py], [BA2903} ; 6-CF 3 -4-CHF 2 -3-Py], [BA2904; 2-CN-4-CHF 2 -3-Py], [BA2905; 5-CN-4 _{-CHF 2 -3-Py], [} BA2906; 6-CN-4-CHF 2 -3-Py], [BA2907; 2-OMe-4-CHF 2 -3-Py], [BA2908; 5-OMe- _{4-CHF 2 -3-Py]} , [BA2909; 6-OMe-4-CHF 2 -3-Py], [BA2910; 5-CHF 2 -3-Py], [BA2911; 2-Cl-5-CHF _{2 -3-Py], [BA2912} ; 4-Cl-5-CHF 2 -3-Py], [BA2913; 6-Cl-5-CHF 2 -3-Py], [BA2914; 2-Me-5- _{CHF 2 -3-Py], [} BA2915; 4-Me-5-CHF 2 -3-Py], [BA2916; 6-Me-5-CHF 2 -3-Py], [BA2917; 2-CF 3 - _{5-CHF 2 -3-Py]} , [BA2918; 4-CF 3 -5-CHF 2 -3-Py], [BA2919; 6-CF 3 -5-CHF 2 -3-P y], [BA2920; 2- CN-5-CHF 2 -3-Py], [BA2921; 4-CN-5-CHF 2 -3-Py], [BA2922; 6-CN-5-CHF 2 -3 -Py], [BA2923; 2- OMe-5-CHF 2 -3-Py], [BA2924; 4-OMe-5-CHF 2 -3-Py], [BA2925; 6-OMe-5-CHF 2 - 3-Py], [BA2926; 6-CHF 2 -3-Py], [BA2927; 2-Cl-6-CHF 2 -3-Py], [BA2928; 4-Cl-6-CHF 2 -3-Py ], [BA2929; 5-Cl -6-CHF 2 -3-Py], [BA2930; 2-Me-6-CHF 2 -3-Py], [BA2931; 4-Me-6-CHF 2 -3- Py], [BA2932; 5- Me-6-CHF 2 -3-Py], [BA2933; 2-CF 3 -6-CHF 2 -3-Py], [BA2934; 4-CF 3 -6-CHF 2 -3-Py, [BA 2935; 5-CF ₃ -6-CHF ₂ -3-Py], [BA 2 936; 2-CN-6-CHF ₂ -3-Py], [BA ₂ 937; _{CHF 2 -3-Py], [} BA2938; 5-CN-6-CHF 2 -3-Py], [BA2939; 2-OMe-6-CHF 2 -3-Py], [BA2940; 4-OMe-6 _{-CHF 2 -3-Py], [} BA2941; 5-OMe-6-CHF 2 -3-Py], [BA2942; 2-OCHF 2 -3-Py], [BA2943; 4-Cl-2-OCHF 2 -3-Py !, [BA2944; 5-Cl-2-OCHF ₂ -3-Py], [BA 2945; 6-Cl-2-OCHF ₂ -3-Py], [BA 2946; 4-Me-2-OCHF _{2 -3-Py], [BA2947} ; 5-Me-2-OCHF 2 -3-Py], [BA2948; 6-Me-2-OCHF 2 -3-Py], [BA2949; 4-CF 3 -2 _{-OCHF 2 -3-Py], [} BA2950; 5-CF 3 -2-OCHF 2 -3-Py], [BA2951; 6-CF 3 -2-OCHF 2 -3-Py], [BA2952; 4- CN-2-OCHF ₂ -3-Py !, [BA 2953; 5-CN -2-OCHF ₂ -3-Py], [BA 2954; 6-CN -2-OCHF ₂ -3-Py, [BA 2 955; 4-OMe-2-OCHF ₂ -3-Py], [BA 2956; 5-OMe -2-OCHF ₂ -3-Py], [BA 2 957; 6-OMe -2- OFHF ₂ -3-Py, [BA 2958; 4-OCHF ₂ -3-Py], [BA 2959; 2-Cl 4-OCHF ₂ -3-Py], [BA ₂ 960; 5-Cl 4-OCHF _2- 3-Py], [BA2961; 6-Cl-4-OCHF 2 -3-Py], [BA2962; 2-Me-4-OCHF 2 -3-Py], [BA2963; 5-Me-4-OCHF 2 -3-Py], [BA2964; 6-Me-4-OCHF 2 -3-Py], [BA2965; 2-CF 3 -4-OCHF 2 -3-Py], [BA2966; 5-CF 3 -4 _{-OCHF 2 -3-Py], [} BA2967; 6-CF 3 -4-OCHF 2 -3-Py], [BA2968; 2-CN-4-OCHF 2 -3-Py], [BA2969; 5-CN _{-4-OCHF 2 -3-Py]} , [BA2970; 6-CN-4-OCHF 2 -3-Py], [BA2971; 2-OMe-4-OCHF 2 -3-Py], [BA2972; 5- _{OMe-4-OCHF 2 -3-} Py], [BA2973; 6-OMe-4-OCHF 2 -3-Py], [BA2974; 5-OCHF 2 -3-Py], [BA2975; 2-Cl-5 _{-OCHF 2 -3-Py], [} BA2976; 4-Cl-5-OCHF 2 -3-Py], [BA2977; 6-Cl-5-OCHF 2 -3-Py], [BA2978; 2-Me- _{5-OCHF 2 -3-Py]} , [BA2979; 4-Me-5-OCHF 2 -3-Py], [BA2980; 6-Me-5-OCHF 2 -3-Py], [BA2981; 2-CF _{3 -5-OCHF 2 -3-Py} ], [BA2982; 4-CF 3 -5-OCHF 2 -3-Py], [BA2983; 6-CF 3 -5-OCHF 2 -3-Py], [BA2984 2-CN-5-OCHF ₂ -3-Py],

[BA 2985; 4-CN-5-OCHF ₂ -3-Py], [BA 2986; 6-CN -5-OCHF ₂ -3-Py], [BA 2 987; 2-OMe -5-OCHF ₂ -3-Py] , [BA2988; 4-OMe- 5-OCHF 2 -3-Py], [BA2989; 6-OMe-5-OCHF 2 -3-Py], [BA2990; 6-OCHF 2 -3-Py], [BA2991 ; 2-Cl-6-OCHF 2 -3-Py], [BA2992; 4-Cl-6-OCHF 2 -3-Py], [BA2993; 5-Cl-6-OCHF 2 -3-Py], [ BA2994; 2-Me-6- OCHF 2 -3-Py], [BA2995; 4-Me-6-OCHF 2 -3-Py], [BA2996; 5-Me-6-OCHF 2 -3-Py], _{[BA2997; 2-CF 3 -6} -OCHF 2 -3-Py], [BA2998; 4-CF 3 -6-OCHF 2 -3-Py], [BA2999; 5-CF 3 -6-OCHF 2 -3 -Py], [BA3000; 2- CN-6-OCHF 2 -3-Py], [BA3001; 4-CN-6-OCHF 2 -3-Py], [BA3002; 5-CN-6-OCHF 2 - 3-Py], [BA3003; 2-OMe-6-OCHF 2 -3-Py], [BA3004; 4-OMe-6-OCHF 2 -3-Py], [BA3005; 5-OMe-6-OCHF 2 -3-Py], [BA 3006; 2-Et-3-Py], [BA 3007; 4-Cl-2-Et-3-Py], [BA 3008; 5-Cl-2-Et-3-Py], [BA3009; 6-Cl-2-Et-3-Py], [BA3010; 4-Me-2-Et-3-Py], [BA3011; 5-Me-2-Et-3-Py], [BA3012 ; 6-Me-2-Et -3-Py], [BA3013; 4-CF 3 -2-Et-3-Py], [BA3014; 5-CF 3 -2-Et-3-Py], [BA3015 _{; 6-CF 3 -2-Et} -3-Py], [BA3016; 4-CN-2-Et-3-Py], [BA3017; 5-CN-2-Et-3-Py], [BA3018; 6-CN-2-Et-3-Py], [BA3019; 4-OMe-2-Et-3-Py], [BA3020; 5-OMe-2-Et-3-Py], [BA3021; 6- OMe-2 -Et-3-Py], [BA3022; 4-Et-3-Py], [BA3023; 2-Cl-4-Et-3-Py], [BA3024; 5-Cl-4-Et-3-Py ], [BA3025; 6-Cl-4-Et-3-Py], [BA3026; 2-Me-4-Et-3-Py], [BA3027; 5-Me-4-Et-3-Py], [BA3028; 6-Me-4 -Et-3-Py], [BA3029; 2-CF 3 -4-Et-3-Py], [BA3030; 5-CF 3 -4-Et-3-Py], _{[BA3031; 6-CF 3 -4} -Et-3-Py], [BA3032; 2-CN-4-Et-3-Py], [BA3033; 5-CN-4-Et-3-Py], [ BA3034; 6-CN-4-Et-3-Py], [BA3035; 2-OMe-4-Et-3-Py], [BA3036; 5-OMe-4-Et-3-Py], [BA3037; 6-OMe-4-Et-3-Py], [BA3038; 5-Et-3-Py], [BA3039; 2-Cl-5-Et-3-Py], [BA3040; 4-Cl-5-4 Et-3-Py, [BA3041; 6-Cl-5-Et-3-Py], [BA3042; 2-Me-5-Et-3-Py], [BA3043; 4-Me-5-Et- 3-Py], [BA3044; 6-Me-5-Et-3-Py], [BA3045; 2-CF 3 -5-Et-3-Py], [BA3046; 4-CF 3 -5-Et- 3-Py], [BA3047; 6-CF 3 -5-Et-3-Py], [BA3048; 2-CN-5-Et-3-Py], [BA3049; 4-CN-5-Et-3 -Py], [BA3050; 6-CN-5-Et-3-Py], [BA3051; 2-OMe-5-Et-3-Py], [BA3052; 4-OMe-5-Et-3-Py ], [BA3053; 6-OMe-5-Et-3-Py], [BA3054; 6-Et-3-Py], [BA3055; 2-Cl-6-Et-3-Py], [BA3056; 4] -Cl-6-Et-3-Py], [BA3057; 5-Cl-6-Et-3-Py], [BA3058; 2-Me-6-Et-3-Py], [BA3059; 4-Me -6-Et-3-Py] , [BA3060; 5-Me-6-Et-3-Py], [BA3061; 2-CF 3 -6-Et-3-Py], [BA3062; 4-CF 3 -6- Et-3-Py], [ BA3063; 5-CF 3 -6-Et-3-Py], [BA3064; 2-CN-6-Et-3-Py], [BA3065; 4-CN-6-Et -3-Py, [BA 3066; 5-CN-6-Et-3-Py], [BA 3067; 2-OMe-6-Et-3-Py], [BA 3068; 4-OMe-6-Et-3 -Py], [BA3069; 5- OMe-6-Et-3-Py] 2691, [BA3070; 4-Cl-2-CH 2 CF 3 -3-Py], [BA3071; 5-Cl-2-CH _{2 CF 3 -3-Py],} [BA3072; 6-Cl-2-CH 2 CF 3 -3-Py], [BA3073; 4-Me-2-CH 2 CF 3 -3-Py], [BA3074; _{5-Me-2-CH 2} CF 3 -3-Py], [BA3075; 6-Me-2-CH 2 CF 3 -3-Py], [BA3076; 4-CF 3 -2-CH 2 CF 3 - 3-Py], [BA3077; 5-CF 3 -2-CH 2 CF 3 -3-Py], [BA3078; 6-CF 3 -2-CH 2 CF 3 -3-Py], [BA3079; 4- _{CN-2-CH 2 CF 3} -3-Py], [BA3080; 5-CN-2-CH 2 CF 3 -3-Py], [BA3081; 6-CN-2-CH 2 CF 3 -3-Py ], [BA3082; 4-OMe -2-CH 2 CF 3 -3-Py], [BA3083; 5-OMe-2-CH 2 CF 3 -3-Py], [BA3084; 6-OMe-2-CH ₂ CF ₃ -3-Py],

_{[BA3085; 4-CH 2 CF} 3 -3-Py], [BA3086; 2-Cl-4-CH 2 CF 3 -3-Py], [BA3087; 5-Cl-4-CH 2 CF 3 -3- Py], [BA3088; 6- Cl-4-CH 2 CF 3 -3-Py], [BA3089; 2-Me-4-CH 2 CF 3 -3-Py], [BA3090; 5-Me-4- _{CH 2 CF 3 -3-Py]} , [BA3091; 6-Me-4-CH 2 CF 3 -3-Py], [BA3092; 2-CF 3 -4-CH 2 CF 3 -3-Py], [ BA 3093; 5-CF ₃ -4-CH ₂ CF ₃ -3-Py], [BA 3094; 6-CF ₃ -4-CH ₂ CF ₃ -3-Py], [BA 3095; 2-CN -4-CH _{2 CF 3 -3-Py], [} BA3096; 5-CN-4-CH 2 CF 3 -3-Py], [BA3097; 6-CN-4-CH 2 CF 3 -3-Py], [BA3098; 2 _{-OMe-4-CH 2 CF 3} -3-Py], [BA3099; 5-OMe-4-CH 2 CF 3 -3-Py], [BA3100; 6-OMe-4-CH 2 CF 3 -3- Py], [BA3101; 5- CH 2 CF 3 -3-Py], [BA3102; 2-Cl-5-CH 2 CF 3 -3-Py], [BA3103; 4-Cl-5-CH 2 CF 3 -3-Py], [BA3104; 6-Cl-5-CH 2 CF 3 -3-Py], [BA3105; 2-Me-5-CH 2 CF 3 -3-Py], [BA3106; 4-Me _{-5-CH 2 CF 3 -3-} Py], [BA3107; 6-Me-5-CH 2 CF 3 -3-Py], [BA3108; 2-CF 3 -5-CH 2 CF 3 -3-Py ], [BA 3109; 4-CF ₃ -5-CH ₂ CF ₃ -3-Py], [BA 3110; 6-CF ₃ -5-CH ₂ CF ₃ -3-Py], [BA 3111; 2-CN-5] _{-CH 2 CF 3 -3-Py]} , [BA3112; 4-CN-5-CH 2 CF 3 -3-Py], [BA3113; 6-CN-5-CH 2 CF 3 -3-Py], [ BA3114; 2-OMe-5- CH 2 CF 3 -3-Py], [BA3115; 4-OMe-5-CH 2 CF 3 -3 -Py], [BA3116; 6- OMe-5-CH 2 CF 3 -3-Py], [BA3117; 6-CH 2 CF 3 -3-Py], [BA3118; 2-Cl-6-CH 2 CF _{3 -3-Py], [BA3119} ; 4-Cl-6-CH 2 CF 3 -3-Py], [BA3120; 5-Cl-6-CH 2 CF 3 -3-Py], [BA3121; 2- _{Me-6-CH 2 CF 3} -3-Py], [BA3122; 4-Me-6-CH 2 CF 3 -3-Py], [BA3123; 5-Me-6-CH 2 CF 3 -3-Py ], [BA3124; 2-CF 3 -6-CH 2 CF 3 -3-Py], [BA3125; 4-CF 3 -6-CH 2 CF 3 -3-Py], [BA3126; 5-CF 3 - _{6-CH 2 CF 3 -3-} Py], [BA3127; 2-CN-6-CH 2 CF 3 -3-Py], [BA3128; 4-CN-6-CH 2 CF 3 -3-Py], [BA3129; 5-CN-6 -CH 2 CF 3 -3-Py], [BA3130; 2-OMe-6-CH 2 CF 3 -3-Py], [BA3131; 4-OMe-6-CH 2 CF _{3 -3-Py], [BA3132} ; 5-OMe-6-CH 2 CF 3 -3-Py], [BA3133; 4-Cl-2-OEt-3-Py], [BA3134; 5-Cl-2 -OEt-3-Py], [BA3135; 6-Cl-2-OEt-3-Py], [BA3136; 4-Me-2-OEt-3-Py], [BA3137; 5-Me-2-OEt -3-Py], [BA3138; 6-Me-2-OEt-3-Py], [BA3139; 4-CF 3 -2-OEt-3-Py], [BA3140; 5-CF 3 -2-OEt -3-Py], [BA3141; 6-CF 3 -2-OEt-3-Py], [BA3142; 4-CN-2-OEt-3-Py], [BA3143; 5-CN-2-OEt- 3-Py], [BA3144; 6-CN-2-OEt-3-Py], [BA3145; 4-OMe-2-OEt-3-Py], [BA3146; 5-OMe-2-OEt-3- 3 Py], [BA3147; 6-OMe-2-OEt-3-Py], [BA3148; 4-OEt-3-Py], [BA3149; 2-Cl-4-OEt-3-Py], [BA3150; 5-C l-4-OEt-3-Py !, [BA3151; 6-Cl-4-OEt-3-Py], [BA3152; 2-Me-4-OEt-3-Py], [BA3153; 5-Me- 4-OEt-3-Py] , [BA3154; 6-Me-4-OEt-3-Py], [BA3155; 2-CF 3 -4-OEt-3-Py], [BA3156; 5-CF 3 - 4-OEt-3-Py] , [BA3157; 6-CF 3 -4-OEt-3-Py], [BA3158; 2-CN-4-OEt-3-Py], [BA3159; 5-CN-4 -OEt-3-Py], [BA3160; 6-CN-4-OEt-3-Py], [BA3161; 2-OMe-4-OEt-3-Py], [BA3162; 5-OMe-4-OEt -3-Py !, [BA3163; 6-OMe-4-OEt-3-Py], [BA3164; 5-OEt-3-Py], [BA3165; 2-Cl-5-OEt-3-Py], [BA3166; 4-Cl-5-OEt-3-Py], [BA3167; 6-Cl-5-OEt-3-Py], [BA3168; 2-Me-5-OEt-3-Py], [BA3169 ; 4-Me-5-OEt -3-Py], [BA3170; 6-Me-5-OEt-3-Py], [BA3171; 2-CF 3 -5-OEt-3-Py], [BA3172; _{4-CF 3 -5-OEt-} 3-Py], [BA3173; 6-CF 3 -5-OEt-3-Py], [BA3174; 2-CN-5-OEt-3-Py], [BA3175; 4-CN-5-OEt-3-Py], [BA3176; 6-CN-5-OEt-3-Py], [BA3177; 2-OMe-5-OEt-3-Py], [BA3178; OMe-5-OEt-3-Py !, [BA3179; 6-OMe-5-OEt-3-Py], [BA3180; 6-OEt-3-Py], [BA3181; 2-Cl-6-OEt- 3-Py], [BA3182; 4-Cl-6-OEt-3-Py], [BA3183; 5-Cl-6-OEt-3-Py], [BA3184; 2-Me-6-OEt-3- Py],

[BA3185; 4-Me-6 -OEt-3-Py], [BA3186; 5-Me-6-OEt-3-Py], [BA3187; 2-CF 3 -6-OEt-3-Py], [ _{BA3188; 4-CF 3 -6-} OEt-3-Py], [BA3189; 5-CF 3 -6-OEt-3-Py], [BA3190; 2-CN-6-OEt-3-Py], [ BA 3191; 4-CN-6-OEt-3-Py], [BA3192; 5-CN-6-OEt-3-Py], [BA3193; 2-OMe-6-OEt-3-Py], [BA3194; 4-OMe-6-OEt- 3-Py], [BA3195; 5-OMe-6-OEt-3-Py], [BA3196; 4-Cl-2-OCH 2 CF 3 -3-Py], [BA3197 ; 5-Cl-2-OCH 2 CF 3 -3-Py], [BA3198; 6-Cl-2-OCH 2 CF 3 -3-Py], [BA3199; 4-Me-2-OCH 2 CF 3 - 3-Py], [BA3200; 5-Me-2-OCH 2 CF 3 -3-Py], [BA3201; 6-Me-2-OCH 2 CF 3 -3-Py], [BA3202; 4-CF 3 -2-OCH ₂ CF ₃ -3-Py, [BA 3203; 5-CF ₃ -2-OCH ₂ CF ₃ -3-Py], [BA 3204; 6-CF ₃ -2-OCH ₂ CF ₃ -3- Py], [BA3205; 4- CN-2-OCH 2 CF 3 -3-Py], [BA3206; 5-CN-2-OCH 2 CF 3 -3-Py], [BA3207; 6-CN-2- _{OCH 2 CF 3 -3-Py]} , [BA3208; 4-OMe-2-OCH 2 CF 3 -3-Py], [BA3209; 5-OMe-2-OCH 2 CF 3 -3-Py], [BA3210 6-OMe-2-OCH ₂ CF ₃ -3-Py !, [BA 3211; 4-OCH ₂ CF ₃ -3-Py], [BA 3212; 2-Cl 4 -OCH ₂ CF ₃ -3-Py] , [BA3213; 5-Cl- 4-OCH 2 CF 3 -3-Py], [BA3214; 6-Cl-4-OCH 2 CF 3 -3-Py], [BA3215; 2-Me-4-OCH 2 CF ₃ -3-Py !, [BA 3216; 5-Me-4-OCH ₂ CF ₃ -3-Py], [BA 3217; 6-Me- _{4-OCH 2 CF 3 -3-} Py], [BA3218; 2-CF 3 -4-OCH 2 CF 3 -3-Py], [BA3219; 5-CF 3 -4-OCH 2 CF 3 -3-Py ], [BA3220; 6-CF 3 -4-OCH 2 CF 3 -3-Py], [BA3221; 2-CN-4-OCH 2 CF 3 -3-Py], [BA3222; 5-CN-4- _{OCH 2 CF 3 -3-Py]} , [BA3223; 6-CN-4-OCH 2 CF 3 -3-Py], [BA3224; 2-OMe-4-OCH 2 CF 3 -3-Py], [BA3225 ; 5-OMe-4-OCH 2 CF 3 -3-Py], [BA3226; 6-OMe-4-OCH 2 CF 3 -3-Py], [BA3227; 5-OCH 2 CF 3 -3-Py] , [BA3228; 2-Cl- 5-OCH 2 CF 3 -3-Py], [BA3229; 4-Cl-5-OCH 2 CF 3 -3-Py], [BA3230; 6-Cl-5-OCH 2 _{CF 3 -3-Py], [} BA3231; 2-Me-5-OCH 2 CF 3 -3-Py], [BA3232; 4-Me-5-OCH 2 CF 3 -3-Py], [BA3233; 6 _{-Me-5-OCH 2 CF 3} -3-Py], [BA3234; 2-CF 3 -5-OCH 2 CF 3 -3-Py], [BA3235; 4-CF 3 -5-OCH 2 CF 3 - 3-Py], [BA3236; 6-CF 3 -5-OCH 2 CF 3 -3-Py], [BA3237; 2-CN-5-OCH 2 CF 3 -3-Py], [BA3238; 4-CN _{-5-OCH 2 CF 3 -3-} Py], [BA3239; 6-CN-5-OCH 2 CF 3 -3-Py], [BA3240; 2-OMe-5-OCH 2 CF 3 -3-Py] , [BA3241; 4-OMe- 5-OCH 2 CF 3 -3-Py], [BA3242; 6-OMe-5-OCH 2 CF 3 -3-Py], [BA3243; 6-OCH 2 CF 3 -3 -Py], [BA3244; 2- Cl-6-OCH 2 CF 3 -3-Py], [BA3245; 4-Cl-6-OCH 2 CF 3 -3-Py], [BA3246; 5-Cl-6 -OCH ₂ CF ₃ -3-Py], [BA 3247; 2 _{-Me-6-OCH 2 CF 3} -3-Py], [BA3248; 4-Me-6-OCH 2 CF 3 -3-Py], [BA3249; 5-Me-6-OCH 2 CF 3 -3- Py], [BA3250; 2- CF 3 -6-OCH 2 CF 3 -3-Py], [BA3251; 4-CF 3 -6-OCH 2 CF 3 -3-Py], [BA3252; 5-CF 3 _{-6-OCH 2 CF 3 -3-} Py], [BA3253; 2-CN-6-OCH 2 CF 3 -3-Py], [BA3254; 4-CN-6-OCH 2 CF 3 -3-Py] , [BA3255; 5-CN- 6-OCH 2 CF 3 -3-Py], [BA3256; 2-OMe-6-OCH 2 CF 3 -3-Py], [BA3257; 4-OMe-6-OCH 2 _{CF 3 -3-Py], [} BA3258; 5-OMe-6-OCH 2 CF 3 -3-Py], [BA3259; 2-Pr-3-Py], [BA3260; 4-Cl-2-Pr- 3-Py], [BA3261; 5-Cl-2-Pr-3-Py], [BA3262; 6-Cl-2-Pr-3-Py], [BA 3263; 4-Me-2-Pr-3- Py], [BA3264; 5- Me-2-Pr-3-Py], [BA3265; 6-Me-2-Pr-3-Py], [BA3266; 4-CF 3 -2-Pr-3-Py ], [BA3267; 5-CF 3 -2-Pr-3-Py], [BA3268; 6-CF 3 -2-Pr-3-Py], [BA3269; 4-CN-2-Pr-3-Py ], [BA3270; 5-CN-2-Pr-3-Py], [BA3271; 6-CN-2-Pr-3-Py], [BA3272; 4-OMe-2-Pr-3-Py], [BA3273; 5-OMe-2-Pr-3-Py], [BA3274; 6-OMe-2-Pr-3-Py], [BA3275; 4-Pr-3-Py], [BA3276; -4-Pr-3-Py], [BA3277; 5-Cl-4-Pr-3-Py], [BA3278; 6-Cl-4-Pr-3-Py], [BA3279; 2-Me-4 -Pr-3-Py], [ BA3280; 5-Me-4-Pr-3-Py], [BA3281; 6-Me-4-Pr-3-Py], [BA3282; 2-CF 3 -4- Pr-3-Py, [BA3283; 5-CF ₃ -4-Pr -3-Py], [BA3284; 6-CF 3 -4-Pr-3-Py],

[BA3285; 2-CN-4-Pr-3-Py], [BA3286; 5-CN-4-Pr-3-Py], [BA3287; 6-CN-4-Pr-3-Py], [BA3288] 2-OMe-4-Pr-3-Py !, [BA3289; 5-OMe-4-Pr-3-Py], [BA3290; 6-OMe-4-Pr-3-Py], [BA3291; -Pr-3-Py], [BA3292; 2-Cl-5-Pr-3-Py], [BA3293; 4-Cl-5-Pr-3-Py], [BA3294; 6-Cl-5-Pr -3-Py, [BA3295; 2-Me-5-Pr-3-Py], [BA3296; 4-Me-5-Pr-3-Py], [BA3297; 6-Me-5-Pr-3 -Py], [BA3298; 2- CF 3 -5-Pr-3-Py], [BA3299; 4-CF 3 -5-Pr-3-Py], [BA3300; 6-CF 3 -5-Pr- 3-Py], [BA3301; 2-CN-5-Pr-3-Py], [BA3302; 4-CN-5-Pr-3-Py], [BA3303; 6-CN-5-Pr-3- 3 Py], [BA3304; 2-OMe-5-Pr-3-Py], [BA3305; 4-OMe-5-Pr-3-Py], [BA3306; 6-OMe-5-Pr-3-Py] , [BA3307; 6-Pr-3-Py], [BA3308; 2-Cl-6-Pr-3-Py], [BA3309; 4-Cl-6-Pr-3-Py], [BA 3310; Cl-6-Pr-3-Py], [BA3311; 2-Me-6-Pr-3-Py], [BA3312; 4-Me-6-Pr-3-Py], [BA3313; 5-Me- 6-Pr-3-Py] , [BA3314; 2-CF 3 -6-Pr-3-Py], [BA3315; 4-CF 3 -6-Pr-3-Py], [BA3316; 5-CF 3 -6-Pr-3-Py], [BA3317; 2-CN-6-Pr-3-Py], [BA3318; 4-CN-6-Pr-3-Py], [BA3319; 5-CN-6 -Pr-3-Py], [BA3320; 2-OMe-6-Pr-3-Py], [BA3321; 4-OMe-6-Pr-3-Py], [BA3322; 5-OMe-6-Pr -3-Py !, [BA3323; 2-OPr-3-Py], [BA3324; 4-Cl-2-OPr-3-Py], [BA3325; 5-Cl-2-OPr-3-Py], [ BA3326; 6-Cl-2-OPr-3-Py], [BA3327; 4-Me-2-OPr-3-Py], [BA3328; 5-Me-2-OPr-3-Py], [BA3329; 6-Me-2-OPr- 3-Py], [BA3330; 4-CF 3 -2-OPr-3-Py], [BA3331; 5-CF 3 -2-OPr-3-Py], [BA3332; _{6-CF 3 -2-OPr-} 3-Py], [BA3333; 4-CN-2-OPr-3-Py], [BA3334; 5-CN-2-OPr-3-Py], [BA3335; 6 -CN-2-OPr-3-Py, [BA3336; 4-OMe-2-OPr-3-Py], [BA3337; 5-OMe-2-OPr-3-Py], [BA3338; 6-OMe -2-OPr-3-Py, [BA3339; 4-OPr-3-Py], [BA3340; 2-Cl-4-OPr-3-Py], [BA3341; 5-Cl-4-OPr-3 -Py], [BA3342; 6-Cl-4-OPr-3-Py], [BA3343; 2-Me-4-OPr-3-Py], [BA3344; 5-Me-4-OPr-3-Py ], [BA3345; 6-Me -4-OPr-3-Py], [BA3346; 2-CF 3 -4-OPr-3-Py], [BA3347; 5-CF 3 -4-OPr-3-Py ], [BA3348; 6-CF 3 -4-OPr-3-Py], [BA3349; 2-CN-4-OPr-3-Py], [BA3350; 5-CN-4-OPr-3-Py] , [BA3351; 6-CN-4-OPr-3-Py], [BA3352; 2-OMe-4-OPr-3-Py], [BA3353; 5-OMe-4-OPr-3-Py], [BA 3352; 6-OMe-4-OPr-3-Py !, [BA3355; 5-OPr-3-Py], [BA3356; 2-Cl-5-OPr-3-Py], [BA3357; 4-Cl- 5-OPr-3-Py, [BA3358; 6-Cl-5-OPr-3-Py], [BA3359; 2-Me-5-OPr-3-Py], [BA3360; 4-Me-5- OPr-3-Py], [ BA3361; 6-Me-5-OPr-3-Py], [BA3362; 2-CF 3 -5-OPr-3-Py], [BA3363; 4-CF 3 -5- OPr-3-Py], [ BA3364; 6-CF 3 -5-OPr-3-Py], [BA 3365; 2-CN-5-OPr-3-Py], [BA3366; 4-CN-5-OPr-3-Py], [BA3367; 6-CN-5-OPr-3-Py], [BA3368; 2-OMe-5-OPr-3-Py], [BA3369; 4-OMe-5-OPr-3-Py], [BA3370; 6-OMe-5-OPr-3-Py], [BA3371; 6- OPr-3-Py, [BA3372; 2-Cl-6-OPr-3-Py], [BA3373; 4-Cl-6-OPr-3-Py], [BA3374; 5-Cl-6-OPr- 3-Py], [BA3375; 2-Me-6-OPr-3-Py], [BA3376; 4-Me-6-OPr-3-Py], [BA3377; 5-Me-6-OPr-3- Py], [BA 3378; 2-CF ₃ -6-OPr-3-Py], [BA 3379; 4-CF ₃ -6-OPr-3-Py], [BA 3380; 5-CF ₃ -6-OPr-3 -Py], [BA3381; 2-CN-6-OPr-3-Py], [BA3382; 4-CN-6-OPr-3-Py], [BA3383; 5-CN-6-OPr-3-Py ], [BA3384; 2-OMe-6-OPr-3-Py],

[BA3385; 4-OMe-6-OPr-3-Py], [BA3386; 5-OMe-6-OPr-3-Py], [BA3387; 2-SMe-3-Py], [BA3388; -2-SMe-3-Py !, [BA3389; 5-Cl-2-SMe-3-Py], [BA3390; 6-Cl-2-SMe-3-Py], [BA3391; 4-Me-2 5-SMe-3-Py !, [BA3392; 5-Me-2-SMe-3-Py], [BA3393; 6-Me-2-SMe-3-Py], [BA3394; 4-CF ₃ -2] SMe-3-Py], [ BA3395; 5-CF 3 -2-SMe-3-Py], [BA3396; 6-CF 3 -2-SMe-3-Py], [BA3397; 4-CN-2- SMe-3-Py !, [BA3398; 5-CN-2-SMe-3-Py], [BA3399; 6-CN-2-SMe-3-Py], [BA3400; 4-OMe-2-SMe- 3-Py], [BA3401; 5-OMe-2-SMe-3-Py], [BA3402; 6-OMe-2-SMe-3-Py], [BA3403; 4-SMe-3-Py], [BA3403; BA3404; 2-Cl-4-SMe-3-Py], [BA3405; 5-Cl-4-SMe-3-Py], [BA3406; 6-Cl-4-SMe-3-Py], [BA3407; 2-Me-4-SMe-3-Py !, [BA3408; 5-Me-4-SMe-3-Py], [BA3409; 6-Me-4-SMe-3-Py], [BA3410; _{CF 3 -4-SMe-3-} Py], [BA3411; 5-CF 3 -4-SMe-3-Py], [BA3412; 6-CF 3 -4-SMe-3-Py], [BA3413; 2 -CN-4-SMe-3-Py], [BA3414; 5-CN-4-SMe-3-Py], [BA3415; 6-CN-4-SMe-3-Py], [BA3416; 2-OMe -4-SMe-3-Py !, [BA3417; 5-OMe-4-SMe-3-Py], [BA3418; 6-OMe-4-SMe-3-Py], [BA3419; 5-SMe-3 -Py], [BA3420; 2-Cl-5-SMe-3-Py], [BA3421; 4-Cl-5-SMe-3-Py], [BA3422; 6-Cl-5-SMe-3-Py ], [BA 3423; 2-Me-5-SMe-3-Py], [BA 3424; 4-Me-5 -SMe-3-Py], [ BA3425; 6-Me-5-SMe-3-Py], [BA3426; 2-CF 3 -5-SMe-3-Py], [BA3427; 4-CF 3 -5 -SMe-3-Py], [ BA3428; 6-CF 3 -5-SMe-3-Py], [BA3429; 2-CN-5-SMe-3-Py], [BA3430; 4-CN-5- SMe-3-Py !, [BA3431; 6-CN-5-SMe-3-Py], [BA3432; 2-OMe-5-SMe-3-Py], [BA3433; 4-OMe-5-SMe- 3-Py], [BA3434; 6-OMe-5-SMe-3-Py], [BA3435; 6-SMe-3-Py], [BA3436; 2-Cl-6-SMe-3-Py], [BA3434; 4-Cl-6-SMe-3-Py !, [BA3438; 5-Cl-6-SMe-3-Py], [BA3439; 2-Me-6-SMe-3-Py], [BA3440; 4-Me-6-SMe- 3-Py], [BA3441; 5-Me-6-SMe-3-Py], [BA3442; 2-CF 3 -6-SMe-3-Py], [BA3443; 4 _{-CF 3 -6-SMe-3-} Py], [BA3444; 5-CF 3 -6-SMe-3-Py], [BA3445; 2-CN-6-SMe-3-Py], [BA3446; 4 -CN-6-SMe-3-Py], [BA3447; 5-CN-6-SMe-3-Py], [BA3448; 2-OMe-6-SMe-3-Py], [BA3449; 4-OMe -6-SMe-3-Py !, [BA3450; 5-OMe-6-SMe-3-Py], [BA3451; 2-SCF ₃ -3-Py], [BA3452; 4-Cl-2-SCF ₃ -3-Py !, [BA 3453; 5-Cl-2-SCF ₃ -3-Py], [BA 3454; 6-Cl-2-SCF ₃ -3-Py], [BA 3455; 4-Me-2-SCF _{3 -3-Py], [BA3456} ; 5-Me-2-SCF 3 -3-Py], [BA3457; 6-Me-2-SCF 3 -3-Py], [BA3458; 4-CF 3 -2 _{-SCF 3 -3-Py], [} BA3459; 5-CF 3 -2-SCF 3 -3-Py], [BA3460; 6-CF 3 -2-SCF 3 -3-Py], [BA3461; 4- CN-2-SCF ₃ -3-Py], [BA3462; _{5-CN-2-SCF 3} -3-Py], [BA3463; 6-CN-2-SCF 3 -3-Py], [BA3464; 4-OMe-2-SCF 3 -3-Py], [BA3465 ; 5-OMe-2-SCF 3 -3-Py], [BA3466; 6-OMe-2-SCF 3 -3-Py], [BA3467; 4-SCF 3 -3-Py], [BA3468; 2- _{Cl-4-SCF 3 -3-} Py], [BA3469; 5-Cl-4-SCF 3 -3-Py], [BA3470; 6-Cl-4-SCF 3 -3-Py], [BA3471; 2 _{-Me-4-SCF 3 -3-} Py], [BA3472; 5-Me-4-SCF 3 -3-Py], [BA3473; 6-Me-4-SCF 3 -3-Py], [BA3474; 2-CF ₃ -4-SCF ₃ -3-Py], [BA 3475; 5-CF ₃ -4-SCF ₃ -3-Py], [BA 3476; 6-CF ₃ -4-SCF ₃ -3-Py] , [BA3477; 2-CN- 4-SCF 3 -3-Py], [BA3478; 5-CN-4-SCF 3 -3-Py], [BA3479; 6-CN-4-SCF 3 -3-Py ], [BA3480; 2-OMe -4-SCF 3 -3-Py], [BA3481; 5-OMe-4-SCF 3 -3-Py], [BA3482; 6-OMe-4-SCF 3 -3- Py], [BA3483; 5- SCF 3 -3-Py], [BA3484; 2-Cl-5-SCF 3 -3-Py],

[BA3485; 4-Cl-5 -SCF 3 -3-Py], [BA3486; 6-Cl-5-SCF 3 -3-Py], [BA3487; 2-Me-5-SCF 3 -3-Py] , [BA3488; 4-Me-5-SCF ₃ -3-Py], [BA 3489; 6-Me-5-SCF ₃ -3-Py], [BA 3490; 2-CF ₃ -5-SCF ₃ -3- Py], [BA3491; 4- CF 3 -5-SCF 3 -3-Py], [BA3492; 6-CF 3 -5-SCF 3 -3-Py], [BA3493; 2-CN-5-SCF 3 -3-Py], [BA3494; 4-CN-5-SCF 3 -3-Py], [BA3495; 6-CN-5-SCF 3 -3-Py], [BA3496; 2-OMe-5-SCF _{3 -3-Py], [BA3497} ; 4-OMe-5-SCF 3 -3-Py], [BA3498; 6-OMe-5-SCF 3 -3-Py], [BA3499; 6-SCF 3 -3 -Py], [BA3500; 2- Cl-6-SCF 3 -3-Py], [BA3501; 4-Cl-6-SCF 3 -3-Py], [BA3502; 6-Cl-6-SCF 3 - 3-Py], [BA3503; 2-Me-6-SCF 3 -3-Py], [BA3504; 4-Me-6-SCF 3 -3-Py], [BA3505; 6-Me-6-SCF 3 -3-Py], [BA3506; 2-CF 3 -6-SCF 3 -3-Py], [BA3507; 4-CF 3 -6-SCF 3 -3-Py], [BA3508; 6-CF 3 - _{6-SCF 3 -3-Py]} , [BA3509; 2-CN-6-SCF 3 -3-Py], [BA3510; 4-CN-6-SCF 3 -3-Py], [BA3511; 6-CN _{-6-SCF 3 -3-Py]} , [BA3512; 2-OMe-6-SCF 3 -3-Py], [BA3513; 4-OMe-6-SCF 3 -3-Py], [BA3514; 6- OMe-6-SCF ₃ -3-Py !, [BA 3515; 2-S (O) Me-3-Py], [BA 3516; 4-Cl-2-S (O) Me-3-Py], [BA 3517 5-Cl-2-S (O) Me-3-Py], [BA3518; 6-Cl-2-S (O) Me-3-Py], [BA3519; 4-Me-2-S (O ) Me-3-Py], [BA 352] 0: 5-Me-2-S (O) Me-3-Py], [BA3521; 6-Me-2-S (O) Me-3-Py], [BA3522; 4-CF ₃ -2-S (O) Me-3-Py ], [BA3523; 5-CF 3 -2-S (O) Me-3-Py], [BA3524; 6-CF 3 -2-S (O) Me-3-Py ], [BA3525; 4-CN-2-S (O) Me-3-Py], [BA3526; 5-CN-2-S (O) Me-3-Py], [BA3527; 6-CN-2 -S (O) Me-3-Py], [BA3528; 4-OMe-2-S (O) Me-3-Py], [BA3529; 5-OMe-2-S (O) Me-3-Py ], [BA3530; 6-OMe-2-S (O) Me-3-Py], [BA3531; 4-S (O) Me-3-Py], [BA3532; 2-Cl-4-S (O) ) Me-3-Py], [BA3533; 5-Cl-4-S (O) Me-3-Py], [BA3534; 6-Cl-4-S (O) Me-3-Py], [BA3535] 2-Me-4-S (O) Me-3-Py], [BA3536; 5-Me-4-S (O) Me-3-Py], [BA3537; 6-Me-4-S (O ) Me-3-Py], [BA3538; 2-CF 3 -4-S (O) Me-3-Py], [BA3539; 5-CF 3 -4-S (O) Me-3-Py], _{[BA3540; 6-CF 3 -4} -S (O) Me-3-Py], [BA3541; 2-CN-4-S (O) Me-3-Py], [BA3542; 5-CN-4- S (O) Me-3-Py], [BA3543; 6-CN-4-S (O) Me-3-Py], [BA3544; 2-OMe-4-S (O) Me-3-Py] , [BA3545; 5-OMe-4-S (O) Me-3-Py], [BA3546; 6-OMe-4-S (O) Me-3-Py], [BA3547; 5-S (O) Me-3-Py !, [BA3548; 2-Cl-5-S (O) Me-3-Py], [BA3549; 4-Cl-5-S (O) Me-3-Py], [BA3550; 6-Cl-5-S (O) Me-3-Py], [BA3551; 2-Me-5-S (O) Me-3-Py], [BA3552; 4-Me-5-S (O) Me-3-Py], [ BA3553; 6-Me-5-S (O) Me-3-Py], [BA3554; 2-CF 3 -5-S (O) Me-3-Py], [BA3555 ;Four _{-CF 3 -5-S (O)} Me-3-Py], [BA3556; 6-CF 3 -5-S (O) Me-3-Py], [BA3557; 2-CN-5-S (O ) Me-3-Py], [BA3558; 4-CN-5-S (O) Me-3-Py], [BA3559; 6-CN-5-S (O) Me-3-Py], [BA3560] 2-OMe-5-S (O) Me-3-Py], [BA3561; 4-OMe-5-S (O) Me-3-Py], [BA3562; 6-OMe-5-S (O ) Me-3-Py], [BA 3563; 6-S (O) Me-3-Py], [BA 3564; 2-Cl-6-S (O) Me-3-Py], [BA 3 565; -6-S (O) Me-3-Py], [BA3566; 5-Cl-6-S (O) Me-3-Py], [BA3567; 2-Me-6-S (O) Me-3 -Py], [BA3568; 4-Me-6-S (O) Me-3-Py], [BA3569; 5-Me-6-S (O) Me-3-Py], [BA3570; 2-CF _{3 -6-S (O) Me} -3-Py], [BA3571; 4-CF 3 -6-S (O) Me-3-Py], [BA3572; 5-CF 3 -6-S (O) Me-3-Py !, [BA3573; 2-CN-6-S (O) Me-3-Py], [BA3574; 4-CN-6-S (O) Me-3-Py], [BA3575; 5-CN-6-S (O) Me-3-Py], [BA3576; 2-OMe-6-S (O) Me-3-Py], [BA3577; 4-OMe-6-S (O) Me-3-Py], [ BA3578; 5-OMe-6-S (O) Me-3-Py], [BA3579; 2-S (O) CF 3 -3-Py], [BA3580; 4-Cl _{-2-S (O) CF 3} -3-Py], [BA3581; 5-Cl-2-S (O) CF 3 -3-Py], [BA3582; 6-Cl-2-S (O) CF _{3 -3-Py], [BA3583} ; 4-Me-2-S (O) CF 3 -3-Py], [BA3584; 5-Me-2-S (O) CF 3 -3-Py],

[BA 3585; 6-Me-2-S (O) CF ₃ -3-Py], [BA 3586; 4-CF ₃ -2-S (O) CF ₃ -3-Py], [BA 3587; 5-CF _{3 -2-S (O) CF 3} -3-Py], [BA3588; 6-CF 3 -2-S (O) CF 3 -3-Py], [BA3589; 4-CN-2-S (O) _{CF 3 -3-Py], [} BA3590; 5-CN-2-S (O) CF 3 -3-Py], [BA3591; 6-CN-2-S (O) CF 3 -3-Py], [BA3592; 4-OMe-2 -S (O) CF 3 -3-Py], [BA3593; 5-OMe-2-S (O) CF 3 -3-Py], [BA3594; 6-OMe-2 _{-S (O) CF 3 -3-} Py], [BA3595; 4-S (O) CF 3 -3-Py], [BA3596; 2-Cl-4-S (O) CF 3 -3-Py] , [BA3597; 5-Cl- 4-S (O) CF 3 -3-Py], [BA3598; 6-Cl-4-S (O) CF 3 -3-Py], [BA3599; 2-Me- _{4-S (O) CF 3} -3-Py], [BA3600; 5-Me-4-S (O) CF 3 -3-Py], [BA3601; 6-Me-4-S (O) CF 3 -3-Py], [BA3602; 2-CF 3 -4-S (O) CF 3 -3-Py], [BA3603; 5-CF 3 -4-S (O) CF 3 -3-Py], _{[BA3604; 6-CF 3 -4} -S (O) CF 3 -3-Py], [BA3605; 2-CN-4-S (O) CF 3 -3-Py], [BA3606; 5-CN- _{4-S (O) CF 3} -3-Py], [BA3607; 6-CN-4-S (O) CF 3 -3-Py], [BA3608; 2-OMe-4-S (O) CF 3 -3-Py], [BA3609; 5-OMe-4-S (O) CF 3 -3-Py], [BA3610; 6-OMe-4-S (O) CF 3 -3-Py], [BA3611 ; 5-S (O) CF 3 -3-Py], [BA3612; 2-Cl-5-S (O) CF 3 -3-Py], [BA3613; 4-Cl-5-S (O) CF _{3 -3-Py], [BA3614} ; 6-Cl-5-S (O) CF 3 -3-Py], [BA3615; 2-Me-5-S (O) CF 3 -3-Py], [ BA 3616; 4-Me-5-S (O) CF _3- 3-Py], [BA3617; 6-Me-5-S (O) CF 3 -3-Py], [BA3618; 2-CF 3 -5-S (O) CF 3 -3-Py], [BA3619 _{; 4-CF 3 -5-S} (O) CF 3 -3-Py], [BA3620; 6-CF 3 -5-S (O) CF 3 -3-Py], [BA3621; 2-CN-5 _{-S (O) CF 3 -3-} Py], [BA3622; 4-CN-5-S (O) CF 3 -3-Py], [BA3623; 6-CN-5-S (O) CF 3 - 3-Py], [BA3624; 2-OMe-5-S (O) CF 3 -3-Py], [BA3625; 4-OMe-5-S (O) CF 3 -3-Py], [BA3626; 6-OMe-5-S ( O) CF 3 -3-Py], [BA3627; 6-S (O) CF 3 -3-Py], [BA3628; 2-Cl-6-S (O) CF 3 -3-Py], [BA3629; 4-Cl-6-S (O) CF 3 -3-Py], [BA3630; 5-Cl-6-S (O) CF 3 -3-Py], [BA3631 ; 2-Me-6-S (O) CF 3 -3-Py], [BA3632; 4-Me-6-S (O) CF 3 -3-Py], [BA3633; 5-Me-6-S _{(O) CF 3 -3-Py} ], [BA3634; 2-CF 3 -6-S (O) CF 3 -3-Py], [BA3635; 4-CF 3 -6-S (O) CF 3 - 3-Py], [BA3636; 5-CF 3 -6-S (O) CF 3 -3-Py], [BA3637; 2-CN-6-S (O) CF 3 -3-Py], [BA3638 ; 4-CN-6-S (O) CF 3 -3-Py], [BA3639; 5-CN-6-S (O) CF 3 -3-Py], [BA3640; 2-OMe-6-S _{(O) CF 3 -3-Py} ], [BA3641; 4-OMe-6-S (O) CF 3 -3-Py], [BA3642; 5-OMe-6-S (O) CF 3 -3- Py], [BA3643; 4- Cl-2-S (O) 2 Me-3-Py], [BA3644; 5-Cl-2-S (O) 2 Me-3-Py], [BA3645; 6- Cl-2-S (O) 2 Me-3-Py], [BA3646; 4-Me-2-S (O) 2 Me-3-Py], [BA3647; 5-Me-2-S (O) ₂ Me-3-Py], [BA 3648; 6-Me-2 _{-S (O) 2 Me-3} -Py], [BA3649; 4-CF 3 -2-S (O) 2 Me-3-Py], [BA3650; 5-CF 3 -2-S (O) 2 Me-3-Py], [ BA3651; 6-CF 3 -2-S (O) 2 Me-3-Py], [BA3652; 4-CN-2-S (O) 2 Me-3-Py], [BA3653; 5-CN-2 -S (O) 2 Me-3-Py], [BA3654; 6-CN-2-S (O) 2 Me-3-Py], [BA3655; 4-OMe-2 _{-S (O) 2 Me-3} -Py], [BA3656; 5-OMe-2-S (O) 2 Me-3-Py], [BA3657; 6-OMe-2-S (O) 2 Me- 3-Py], [BA3658; 4-S (O) 2 Me-3-Py], [BA3659; 2-Cl-4-S (O) 2 Me-3-Py], [BA3660; 5-Cl- _{4-S (O) 2 Me} -3-Py], [BA3661; 6-Cl-4-S (O) 2 Me-3-Py], [BA3662; 2-Me-4-S (O) 2 Me -3-Py !, [BA3663; 5-Me-4-S (O) ₂ Me-3-Py], [BA3664; 6-Me-4-S (O) ₂ Me-3-Py], [BA3665] _{; 2-CF 3 -4-S} (O) 2 Me-3-Py], [BA3666; 5-CF 3 -4-S (O) 2 Me-3-Py], [BA3667; 6-CF 3 - _{4-S (O) 2 Me} -3-Py], [BA3668; 2-CN-4-S (O) 2 Me-3-Py], [BA3669; 5-CN-4-S (O) 2 Me -3-Py !, [BA3670; 6-CN-4-S (O) ₂ Me-3-Py], [BA3671; 2-OMe-4-S (O) ₂ Me-3-Py], [BA3672] ; 5-OMe-4-S (O) 2 Me-3-Py], [BA3673; 6-OMe-4-S (O) 2 Me-3-Py], [BA3674; 5-S (O) 2 Me-3-Py !, [BA3675; 2-Cl-5-S (O) ₂ Me-3-Py], [BA3676; 4-Cl-5-S (O) ₂ Me-3-Py], BA3677; 6-Cl-5- S (O) 2 Me-3-Py], [BA3678; 2-Me-5-S (O) 2 Me-3-Py], [BA3679; 4-Me-5- _{S (O) 2 Me-3} -Py], [BA3680; 6-Me-5-S ( O) 2 Me-3-Py], [BA3681; 2-CF 3 -5-S (O) 2 Me-3-Py], [BA3682; 4-CF 3 -5- _{S (O) 2 Me-3} -Py], [BA3683; 6-CF 3 -5-S (O) 2 Me-3-Py], [BA3684; 2-CN-5-S (O) 2 Me- 3-Py],

[BA 3685; 4-CN-5-S (O) ₂ Me-3-Py], [BA 3686; 6-CN-5-S (O) ₂ Me-3-Py], [BA 3687; 2-OMe-5 _{-S (O) 2 Me-3} -Py], [BA3688; 4-OMe-5-S (O) 2 Me-3-Py], [BA3689; 6-OMe-5-S (O) 2 Me- 3-Py], [BA3690; 6-S (O) 2 Me-3-Py], [BA3691; 2-Cl-6-S (O) 2 Me-3-Py], [BA3692; 4-Cl- _{6-S (O) 2 Me} -3-Py], [BA3693; 5-Cl-6-S (O) 2 Me-3-Py], [BA3694; 2-Me-6-S (O) 2 Me -3-Py !, [BA3695; 4-Me-6-S (O) ₂ Me-3-Py], [BA3696; 5-Me-6-S (O) ₂ Me-3-Py], [BA3697] _{; 2-CF 3 -6-S} (O) 2 Me-3-Py], [BA3698; 4-CF 3 -6-S (O) 2 Me-3-Py], [BA3699; 5-CF 3 - _{6-S (O) 2 Me} -3-Py], [BA3700; 2-CN-6-S (O) 2 Me-3-Py], [BA3701; 4-CN-6-S (O) 2 Me -3-Py !, [BA3702; 5-CN-6-S (O) ₂ Me-3-Py], [BA3703; 2-OMe-6-S (O) ₂ Me-3-Py], [BA3704] ; 4-OMe-6-S (O) 2 Me-3-Py], [BA3705; 5-OMe-6-S (O) 2 Me-3-Py], [BA3706; 2-S (O) 2 _{CF 3 -3-Py], [} BA3707; 4-Cl-2-S (O) 2 CF 3 -3-Py], [BA3708; 5-Cl-2-S (O) 2 CF 3 -3-Py ], [BA3709; 6-Cl -2-S (O) 2 CF 3 -3-Py], [BA3710; 4-Me-2-S (O) 2 CF 3 -3-Py], [BA3711; 5 -Me-2-S (O) 2 CF 3 -3-Py], [BA3712; 6-Me-2-S (O) 2 CF 3 -3-Py], [BA3713; 4-CF 3 -2- _{S (O) 2 CF 3 -3} -Py], [BA3714; 5-CF 3 -2-S (O) 2 CF 3 -3-Py], [BA3715; 6-CF 3 -2-S (O) ₂ CF ₃ -3 -Py], [BA3716; 4- CN-2-S (O) 2 CF 3 -3-Py], [BA3717; 5-CN-2-S (O) 2 CF 3 -3-Py], [BA3718 ; 6-CN-2-S (O) 2 CF 3 -3-Py], [BA3719; 4-OMe-2-S (O) 2 CF 3 -3-Py], [BA3720; 5-OMe-2 _{-S (O) 2 CF 3 -3} -Py], [BA3721; 6-OMe-2-S (O) 2 CF 3 -3-Py], [BA3722; 4-S (O) 2 CF 3 -3 -Py], [BA3723; 2- Cl-4-S (O) 2 CF 3 -3-Py], [BA3724; 5-Cl-4-S (O) 2 CF 3 -3-Py], [BA3725 ; 6-Cl-4-S (O) 2 CF 3 -3-Py], [BA3726; 2-Me-4-S (O) 2 CF 3 -3-Py], [BA3727; 5-Me-4 _{-S (O) 2 CF 3 -3} -Py], [BA3728; 6-Me-4-S (O) 2 CF 3 -3-Py], [BA3729; 2-CF 3 -4-S (O) _{2 CF 3 -3-Py],} [BA3730; 5-CF 3 -4-S (O) 2 CF 3 -3-Py], [BA3731; 6-CF 3 -4-S (O) 2 CF 3 - 3-Py], [BA3732; 2-CN-4-S (O) 2 CF 3 -3-Py], [BA3733; 5-CN-4-S (O) 2 CF 3 -3-Py], [ BA3734; 6-CN-4- S (O) 2 CF 3 -3-Py], [BA3735; 2-OMe-4-S (O) 2 CF 3 -3-Py], [BA3736; 5-OMe- _{4-S (O) 2 CF} 3 -3-Py], [BA3737; 6-OMe-4-S (O) 2 CF 3 -3-Py], [BA3738; 5-S (O) 2 CF 3 - 3-Py], [BA3739; 2-Cl-5-S (O) 2 CF 3 -3-Py], [BA3740; 4-Cl-5-S (O) 2 CF 3 -3-Py], [ BA3741; 6-Cl-5- S (O) 2 CF 3 -3-Py], [BA3742; 2-Me-5-S (O) 2 CF 3 -3-Py], [BA3743; 4-Me- _{5-S (O) 2 CF} 3 -3-Py], [BA3744; 6-Me-5-S (O) 2 CF 3 -3-Py], [BA3 _{745; 2-CF 3 -5-} S (O) 2 CF 3 -3-Py], [BA3746; 4-CF 3 -5-S (O) 2 CF 3 -3-Py], [BA3747; 6- _{CF 3 -5-S (O)} 2 CF 3 -3-Py], [BA3748; 2-CN-5-S (O) 2 CF 3 -3-Py], [BA3749; 4-CN-5-S _{(O) 2 CF 3 -3-} Py], [BA3750; 6-CN-5-S (O) 2 CF 3 -3-Py], [BA3751; 2-OMe-5-S (O) 2 CF 3 -3-Py], [BA3752; 4-OMe-5-S (O) 2 CF 3 -3-Py], [BA3753; 6-OMe-5-S (O) 2 CF 3 -3-Py], [BA3754; 6-S (O ) 2 CF 3 -3-Py], [BA3755; 2-Cl-6-S (O) 2 CF 3 -3-Py], [BA3756; 4-Cl-6-S _{(O) 2 CF 3 -3-} Py], [BA3757; 5-Cl-6-S (O) 2 CF 3 -3-Py], [BA3758; 2-Me-6-S (O) 2 CF 3 -3-Py, [BA 3759; 4-Me-6-S (O) ₂ CF ₃ -3-Py], [BA 3760; 5-Me-6-S (O) ₂ CF ₃ -3-Py], _{[BA3761; 2-CF 3 -6} -S (O) 2 CF 3 -3-Py], [BA3762; 4-CF 3 -6-S (O) 2 CF 3 -3-Py], [BA3763; 5 _{-CF 3 -6-S (O)} 2 CF 3 -3-Py], [BA3764; 2-CN-6-S (O) 2 CF 3 -3-Py], [BA3765; 4-CN-6- _{S (O) 2 CF 3 -3} -Py], [BA3766; 5-CN-6-S (O) 2 CF 3 -3-Py], [BA3767; 2-OMe-6-S (O) 2 CF _{3 -3-Py], [BA3768} ; 4-OMe-6-S (O) 2 CF 3 -3-Py], [BA3769; 5-OMe-6-S (O) 2 CF 3 -3-Py] , [BA3770; 2-CN-3-Py], [BA3771; 4-Cl-2-CN-3-Py], [BA3772; 5-Cl-2-CN-3-Py], [BA3773; Cl-2-CN-3-Py, [BA3774; 4-Me-2-CN-3-Py], [BA3775; 5-Me-2-CN-3- Py], [BA3776; 6- Me-2-CN-3-Py], [BA3777; 4-CF 3 -2-CN-3-Py], [BA3778; 5-CF 3 -2-CN-3- Py], [BA3779; 6- CF 3 -2-CN-3-Py], [BA3780; 4-CN-2-CN-3-Py], [BA3781; 5-CN-2-CN-3-Py ], [BA3782; 6-CN-2-CN-3-Py], [BA3783; 4-OMe-2-CN-3-Py], [BA3784; 5-OMe-2-CN-3-Py],

[BA3785; 6-OMe-2-CN-3-Py], [BA3786; 4-CN-3-Py], [BA3787; 2-Cl-4-CN-3-Py], [BA3788; 5-Cl -4-CN-3-Py !, [BA3789; 6-Cl-4-CN-3-Py], [BA3790; 2-Me-4-CN-3-Py], [BA 3791; 5-Me-4 -CN-3-Py], [ BA3792; 6-Me-4-CN-3-Py], [BA3793; 2-CF 3 -4-CN-3-Py], [BA3794; 5-CF 3 -4 -CN-3-Py], [ BA3795; 6-CF 3 -4-CN-3-Py], [BA3796; 2-CN-4-CN-3-Py], [BA3797; 5-CN-4- CN-3-Py !, [BA 3798; 6-CN-4-CN-3-Py], [BA 3799; 2-OMe-4-CN-3-Py], [BA 3800; 5-OMe-4-CN- 3-Py], [BA3801; 6-OMe-4-CN-3-Py], [BA3802; 5-CN-3-Py], [BA3803; 2-Cl-5-CN-3-Py], [BA-380] 4-Cl-5-CN-3-Py !, [BA3805; 6-Cl-5-CN-3-Py], [BA3806; 2-Me-5-CN-3-Py], [BA3807; 4-Me-5-CN- 3-Py], [BA3808; 6-Me-5-CN-3-Py], [BA3809; 2-CF 3 -5-CN-3-Py], [BA3810; 4 _{-CF 3 -5-CN-3-} Py], [BA3811; 6-CF 3 -5-CN-3-Py], [BA3812; 2-CN-5-CN-3-Py], [BA3813; 4 -CN-5-CN-3-Py], [BA3814; 6-CN-5-CN-3-Py], [BA3815; 2-OMe-5-CN-3-Py], [BA3816; 4-OMe -5-CN-3-Py], [BA3817; 6-OMe-5-CN-3-Py], [BA3818; 6-CN-3-Py], [BA3819; 2-Cl-6-CN-3 -Py], [BA3820; 4-Cl-6-CN-3-Py], [BA3821; 5-Cl-6-CN-3-Py], [BA3822; 2-Me-6-CN-3-Py ], [BA3823; 4-Me -6-CN-3-Py], [BA3824; 5-Me-6-CN-3-Py], [BA3825; 2-CF 3 -6-CN-3-Py] , [BA _{3826; 4-CF 3 -6-} CN-3-Py], [BA3827; 5-CF 3 -6-CN-3-Py], [BA3828; 2-CN-6-CN-3-Py], [ BA3829; 4-CN-6-CN-3-Py], [BA3830; 5-CN-6-CN-3-Py], [BA3831; 2-OMe-6-CN-3-Py], [BA3832; 4-OMe-6-CN-3-Py], [BA3833; 5-OMe-6-CN-3-Py], [BA3834; 2-COOMe-3-Py], [BA3835; 4-Cl-2- COOMe-3-Py !, [BA3836; 5-Cl-2-COOMe-3-Py], [BA3837; 6-Cl-2-COOMe-3-Py], [BA3838; 4-Me-2-COOMe- 3-Py], [BA3839; 5-Me-2-COOMe-3-Py], [BA3840; 6-Me-2-COOMe-3-Py], [BA3841; 4-CF 3 -2-COOMe-3 -Py], [BA3842; 5- CF 3 -2-COOMe-3-Py], [BA3843; 6-CF 3 -2-COOMe-3-Py], [BA3844; 4-CN-2-COOMe-3 -Py], [BA3845; 5-CN-2-COOMe-3-Py], [BA3846; 6-CN-2-COOMe-3-Py], [BA3847; 4-OMe-2-COOMe-3-Py ], [BA3848; 5-OMe-2-COOMe-3-Py], [BA3849; 6-OMe-2-COOMe-3-Py], [BA3850; 4-COOMe-3-Py], [BA3851; 2] -Cl-4-COOMe-3-Py], [BA3852; 5-Cl-4-COOMe-3-Py], [BA3853; 6-Cl-4-COOMe-3-Py], [BA3854; 2-Me -4-COOMe-3-Py !, [BA3855; 5-Me-4-COOMe-3-Py], [BA3856; 6-Me-4-COOMe-3-Py], [BA3857; 2-CF _3- 4-COOMe-3-Py] , [BA3858; 5-CF 3 -4-COOMe-3-Py], [BA3859; 6-CF 3 -4-COOMe-3-Py], [BA3860; 2-CN- 4-COOMe-3-Py], [BA3861; 5-CN-4-COOMe-3-Py], [BA3862; 6-CN-4-COOMe-3-Py], [BA3863; 2-OMe-4-COOMe-3-Py], [BA3864; 5-OMe-4-COOMe-3-Py], [BA3865; 6-OMe-4-COOMe-3-Py], [BA3866; 5- COOMe-3-Py !, [BA 3867; 2-Cl-5-COOMe-3-Py], [BA 3868; 4-Cl-5-COOMe-3-Py], [BA 3869; 6-Cl-5-COOMe- 3-Py], [BA3870; 2-Me-5-COOMe-3-Py], [BA3871; 4-Me-5-COOMe-3-Py], [BA3872; 6-Me-5-COOMe-3- Py], [BA 3873; 2-CF ₃ -5-COOMe-3-Py], [BA 3874; 4-CF ₃ -5-COOMe-3-Py], [BA 3875; 6-CF ₃ -5-COOMe-3 -Py], [BA3876; 2-CN-5-COOMe-3-Py], [BA3877; 4-CN-5-COOMe-3-Py], [BA3878; 6-CN-5-COOMe-3-Py ], [BA3879; 2-OMe-5-COOMe-3-Py], [BA3880; 4-OMe-5-COOMe-3-Py], [BA3881; 6-OMe-5-COOMe-3-Py], [BA3882; 6-COOMe-3-Py], [BA3883; 2-Cl-6-COOMe-3-Py], [BA3884; 4-Cl-6-COOMe-3-Py],

[BA3885; 5-Cl-6-COOMe-3-Py], [BA3886; 2-Me-6-COOMe-3-Py], [BA3887; 4-Me-6-COOMe-3-Py], [BA3888] ; 5-Me-6-COOMe -3-Py], [BA3889; 2-CF 3 -6-COOMe-3-Py], [BA3890; 4-CF 3 -6-COOMe-3-Py], [BA3891 _{; 5-CF 3 -6-COOMe} -3-Py], [BA3892; 2-CN-6-COOMe-3-Py], [BA3893; 4-CN-6-COOMe-3-Py], [BA3894; 5-CN-6-COOMe-3-Py], [BA3895; 2-OMe-6-COOMe-3-Py], [BA3896; 4-OMe-6-COOMe-3-Py], [BA3897; 5- OMe-6-COOMe-3- Py], [BA3898; 2-NO 2 -3-Py], [BA3899; 4-Cl-2-NO 2 -3-Py], [BA3900; 5-Cl-2- _{NO 2 -3-Py], [} BA3901; 6-Cl-2-NO 2 -3-Py], [BA3902; 4-Me-2-NO 2 -3-Py], [BA3903; 5-Me-2 _{-NO 2 -3-Py], [} BA3904; 6-Me-2-NO 2 -3-Py], [BA3905; 4-CF 3 -2-NO 2 -3-Py], [BA3906; 5-CF _{3 -2-NO 2 -3-Py} ], [BA3907; 6-CF 3 -2-NO 2 -3-Py], [BA3908; 4-CN-2-NO 2 -3-Py], [BA3909; _{5-CN-2-NO 2} -3-Py], [BA3910; 6-CN-2-NO 2 -3-Py], [BA3911; 4-OMe-2-NO 2 -3-Py], [BA3912 ; 5-OMe-2-NO 2 -3-Py], [BA3913; 6-OMe-2-NO 2 -3-Py], [BA3914; 4-NO 2 -3-Py], [BA3915; 2- _{Cl-4-NO 2 -3-} Py], [BA3916; 5-Cl-4-NO 2 -3-Py], [BA3917; 6-Cl-4-NO 2 -3-Py], [BA3918; 2 _{-Me-4-NO 2 -3-} Py], [BA3919; 5-Me-4-NO 2 -3-Py], [BA3920; 6-Me-4-NO 2 -3-Py], [BA3921; 2-CF _{3 -4-NO 2 -3-Py]} , [BA3922; 5-CF 3 -4-NO 2 -3-Py], [BA3923; 6-CF 3 -4-NO 2 -3-Py], [BA3924; _{2-CN-4-NO 2} -3-Py], [BA3925; 5-CN-4-NO 2 -3-Py], [BA3926; 6-CN-4-NO 2 -3-Py], [BA3927 ; 2-OMe-4-NO 2 -3-Py], [BA3928; 5-OMe-4-NO 2 -3-Py], [BA3929; 6-OMe-4-NO 2 -3-Py], [ _{BA3930; 5-NO 2 -3-} Py], [BA3931; 2-Cl-5-NO 2 -3-Py], [BA3932; 4-Cl-5-NO 2 -3-Py], [BA3933; 6 _{-Cl-5-NO 2 -3-} Py], [BA3934; 2-Me-5-NO 2 -3-Py], [BA3935; 4-Me-5-NO 2 -3-Py], [BA3936; _{6-Me-5-NO 2} -3-Py], [BA3937; 2-CF 3 -5-NO 2 -3-Py], [BA3938; 4-CF 3 -5-NO 2 -3-Py], _{[BA3939; 6-CF 3 -5} -NO 2 -3-Py], [BA3940; 2-CN-5-NO 2 -3-Py], [BA3941; 4-CN-5-NO 2 -3-Py ], [BA3942; 6-CN -5-NO 2 -3-Py], [BA3943; 2-OMe-5-NO 2 -3-Py], [BA3944; 4-OMe-5-NO 2 -3- Py], [BA3945; 6- OMe-5-NO 2 -3-Py], [BA3946; 6-NO 2 -3-Py], [BA3947; 2-Cl-6-NO 2 -3-Py], [BA3948; 4-Cl-6 -NO 2 -3-Py], [BA3949; 5-Cl-6-NO 2 -3-Py], [BA3950; 2-Me-6-NO 2 -3-Py] , [BA3951; 4-Me- 6-NO 2 -3-Py], [BA3952; 5-Me-6-NO 2 -3-Py], [BA3953; 2-CF 3 -6-NO 2 -3- Py], [BA 3954; 4-CF ₃ -6-NO ₂ -3-Py], [BA ₃ 955; 5-CF ₃ -6-NO ₂ -3-Py], [BA 3956; 2-CN -6- NO ₂ -3-Py], [BA 3957; 4-CN-6-NO ₂ -3-Py], [BA3958; 5-CN-6-NO 2 -3-Py], [BA3959; 2-OMe-6-NO 2 -3-Py], [BA3960; 4-OMe-6-NO _{2 -3-Py], [BA3961} ; 5-OMe-6-NO 2 -3-Py], [BA3962; 4-Cl-2-NH 2 -3-Py], [BA3963; 5-Cl-2- NH ₂ -3-Py !, [BA 3964; 6-Cl-2-NH ₂ -3-Py], [BA 3 965; 4-Me-2-NH ₂ -3-Py], [BA 3966; 5-Me-2 _{-NH 2 -3-Py], [} BA3967; 6-Me-2-NH 2 -3-Py], [BA3968; 4-CF 3 -2-NH 2 -3-Py], [BA3969; 5-CF _{3 -2-NH 2 -3-Py} ], [BA3970; 6-CF 3 -2-NH 2 -3-Py], [BA3971; 4-CN-2-NH 2 -3-Py], [BA3972; _{5-CN-2-NH 2} -3-Py], [BA3973; 6-CN-2-NH 2 -3-Py], [BA3974; 4-OMe-2-NH 2 -3-Py], [BA3975 ; 5-OMe-2-NH 2 -3-Py], [BA3976; 6-OMe-2-NH 2 -3-Py], [BA3977; 4-NH 2 -3-Py], [BA3978; 2- _{Cl-4-NH 2 -3-} Py], [BA3979; 5-Cl-4-NH 2 -3-Py], [BA3980; 6-Cl-4-NH 2 -3-Py], [BA3981; 2 _{-Me-4-NH 2 -3-} Py], [BA3982; 5-Me-4-NH 2 -3-Py], [BA3983; 6-Me-4-NH 2 -3-Py], [BA3984; _{2-CF 3 -4-NH 2} -3-Py],

_{[BA3985; 5-CF 3 -4} -NH 2 -3-Py], [BA3986; 6-CF 3 -4-NH 2 -3-Py], [BA3987; 2-CN-4-NH 2 -3- Py], [BA3988; 5- CN-4-NH 2 -3-Py], [BA3989; 6-CN-4-NH 2 -3-Py], [BA3990; 2-OMe-4-NH 2 -3 -Py], [BA3991; 5- OMe-4-NH 2 -3-Py], [BA3992; 6-OMe-4-NH 2 -3-Py], [BA3993; 5-NH 2 -3-Py] , [BA3994; 2-Cl- 5-NH 2 -3-Py], [BA3995; 4-Cl-5-NH 2 -3-Py], [BA3996; 6-Cl-5-NH 2 -3-Py ], [BA3997; 2-Me -5-NH 2 -3-Py], [BA3998; 4-Me-5-NH 2 -3-Py], [BA3999; 6-Me-5-NH 2 -3- Py], [BA4000; 2- CF 3 -5-NH 2 -3-Py], [BA4001; 4-CF 3 -5-NH 2 -3-Py], [BA4002; 6-CF 3 -5-NH ₂ -3-Py !, [BA 4003; 2-CN-5-NH ₂ -3-Py], [BA 4004; 4-CN-5-NH ₂ -3-Py], [BA 4005; 6-CN -5- _{NH 2 -3-Py], [} BA4006; 2-OMe-5-NH 2 -3-Py], [BA4007; 4-OMe-5-NH 2 -3-Py], [BA4008; 6-OMe-5 _{-NH 2 -3-Py], [} BA4009; 6-NH 2 -3-Py], [BA4010; 2-Cl-6-NH 2 -3-Py], [BA4011; 4-Cl-6-NH 2 -3-Py], [BA4012; 5-Cl-6-NH 2 -3-Py], [BA4013; 2-Me-6-NH 2 -3-Py], [BA4014; 4-Me-6-NH _{2 -3-Py], [BA4015} ; 5-Me-6-NH 2 -3-Py], [BA4016; 2-CF 3 -6-NH 2 -3-Py], [BA4017; 4-CF 3 - _{6-NH 2 -3-Py]} , [BA4018; 5-CF 3 -6-NH 2 -3-Py], [BA4019; 2-CN-6-NH 2 -3-Py], [BA4020; 4- _{CN-6-NH 2 -3-} Py], [BA4021; _{5-CN-6-NH 2} -3-Py], [BA4022; 2-OMe-6-NH 2 -3-Py], [BA4023; 4-OMe-6-NH 2 -3-Py], [BA4024 ; 5-OMe-6-NH 2 -3-Py], [BA4025; 2-NHMe-3-Py], [BA4026; 4-Cl-2-NHMe-3-Py], [BA4027; 5-Cl- 2-NHMe-3-Py, [BA4028; 6-Cl-2-NHMe-3-Py], [BA4029; 4-Me-2-NHMe-3-Py], [BA4030; 5-Me-2- NHMe-3-Py], [ BA4031; 6-Me-2-NHMe-3-Py], [BA4032; 4-CF 3 -2-NHMe-3-Py], [BA4033; 5-CF 3 -2- NHMe-3-Py], [ BA4034; 6-CF 3 -2-NHMe-3-Py], [BA4035; 4-CN-2-NHMe-3-Py], [BA4036; 5-CN-2-NHMe -3-Py !, [BA4037; 6-CN-2-NHMe-3-Py], [BA4038; 4-OMe-2-NHMe-3-Py], [BA4039; 5-OMe-2-NHMe-3 -Py], [BA4040; 6-OMe-2-NHMe-3-Py], [BA4041; 4-NHMe-3-Py], [BA4042; 2-Cl-4-NHMe-3-Py], [BA4043] 5-Cl-4-NHMe-3-Py, [BA4044; 6-Cl-4-NHMe-3-Py], [BA4045; 2-Me-4-NHMe-3-Py], [BA4046; -Me-4-NHMe-3- Py], [BA4047; 6-Me-4-NHMe-3-Py], [BA4048; 2-CF 3 -4-NHMe-3-Py], [BA4049; 5- _{CF 3 -4-NHMe-3-} Py], [BA4050; 6-CF 3 -4-NHMe-3-Py], [BA4051; 2-CN-4-NHMe-3-Py], [BA4052; 5- CN-4-NHMe-3-Py, [BA4053; 6-CN-4-NHMe-3-Py], [BA4054; 2-OMe-4-NHMe-3-Py], [BA4055; 5-OMe- 4-NHMe-3-Py, [BA 4056; 6-OMe-4-NHMe-3-Py], [BA 4057; 5-NHMe-3-Py], [BA 4058; 2-Cl-5-NHMe-3- Py], [BA4 059; 4-Cl-5-NHMe-3-Py], [BA 4060; 6-Cl-5-NHMe-3-Py], [BA4061; 2-Me-5-NHMe-3-Py], [BA4062; 4-Me-5-NHMe- 3-Py], [BA4063; 6-Me-5-NHMe-3-Py], [BA4064; 2-CF 3 -5-NHMe-3-Py], [BA4065; 4 _{-CF 3 -5-NHMe-3-} Py], [BA4066; 6-CF 3 -5-NHMe-3-Py], [BA4067; 2-CN-5-NHMe-3-Py], [BA4068; 4 -CN-5-NHMe-3-Py, [BA4069; 6-CN-5-NHMe-3-Py], [BA4070; 2-OMe-5-NHMe-3-Py], [BA4071; 4-OMe -5-NHMe-3-Py, [BA4072; 6-OMe-5-NHMe-3-Py], [BA4073; 6-NHMe-3-Py], [BA4074; 2-Cl-6-NHMe-3 -Py], [BA4075; 4-Cl-6-NHMe-3-Py], [BA4076; 5-Cl-6-NHMe-3-Py], [BA4077; 2-Me-6-NHMe-3-Py ], [BA4078; 4-Me -6-NHMe-3-Py], [BA4079; 5-Me-6-NHMe-3-Py], [BA4080; 2-CF 3 -6-NHMe-3-Py] _{, [BA4081; 4-CF 3} -6-NHMe-3-Py], [BA4082; 5-CF 3 -6-NHMe-3-Py], [BA4083; 2-CN-6-NHMe-3-Py] , [BA4084; 4-CN-6-NHMe-3-Py],

[BA 4085; 5-CN-6-NHMe-3-Py], [BA 4086; 2-OMe-6-NHMe-3-Py], [BA 4087; 4-OMe-6-NHMe-3-Py], [BA 4088] ; 5-OMe-6-NHMe -3-Py], [BA4089; 2-NMe 2 -3-Py], [BA4090; 4-Cl-2-NMe 2 -3-Py], [BA4091; 5-Cl _{-2-NMe 2 -3-Py]} , [BA4092; 6-Cl-2-NMe 2 -3-Py], [BA4093; 4-Me-2-NMe 2 -3-Py], [BA4094; 5- _{Me-2-NMe 2 -3-} Py], [BA4095; 6-Me-2-NMe 2 -3-Py], [BA4096; 4-CF 3 -2-NMe 2 -3-Py], [BA4097; _{5-CF 3 -2-NMe 2} -3-Py], [BA4098; 6-CF 3 -2-NMe 2 -3-Py], [BA4099; 4-CN-2-NMe 2 -3-Py], [BA4100; 5-CN-2 -NMe 2 -3-Py], [BA4101; 6-CN-2-NMe 2 -3-Py], [BA4102; 4-OMe-2-NMe 2 -3-Py] , [BA4103; 5-OMe- 2-NMe 2 -3-Py], [BA4104; 6-OMe-2-NMe 2 -3-Py], [BA4105; 4-NMe 2 -3-Py], [BA4106 ; 2-Cl-4-NMe 2 -3-Py], [BA4107; 5-Cl-4-NMe 2 -3-Py], [BA4108; 6-Cl-4-NMe 2 -3-Py], [ BA4109; 2-Me-4- NMe 2 -3-Py], [BA4110; 5-Me-4-NMe 2 -3-Py], [BA4111; 6-Me-4-NMe 2 -3-Py], _{[BA4112; 2-CF 3 -4} -NMe 2 -3-Py], [BA4113; 5-CF 3 -4-NMe 2 -3-Py], [BA4114; 6-CF 3 -4-NMe 2 -3 -Py], [BA4115; 2- CN-4-NMe 2 -3-Py], [BA4116; 5-CN-4-NMe 2 -3-Py], [BA4117; 6-CN-4-NMe 2 - 3-Py], [BA4118; 2-OMe-4-NMe 2 -3-Py], [BA4119; 5-OMe-4-NMe 2 -3-Py], [BA4120; 6-OM _{e-4-NMe 2 -3-} Py], [BA4121; 5-NMe 2 -3-Py], [BA4122; 2-Cl-5-NMe 2 -3-Py], [BA4123; 4-Cl-5 _{-NMe 2 -3-Py], [} BA4124; 6-Cl-5-NMe 2 -3-Py], [BA4125; 2-Me-5-NMe 2 -3-Py], [BA4126; 4-Me- _{5-NMe 2 -3-Py]} , [BA4127; 6-Me-5-NMe 2 -3-Py], [BA4128; 2-CF 3 -5-NMe 2 -3-Py], [BA4129; 4- _{CF 3 -5-NMe 2 -3-} Py], [BA4130; 6-CF 3 -5-NMe 2 -3-Py], [BA4131; 2-CN-5-NMe 2 -3-Py], [BA4132 ; 4-CN-5-NMe 2 -3-Py], [BA4133; 6-CN-5-NMe 2 -3-Py], [BA4134; 2-OMe-5-NMe 2 -3-Py], [ BA4135; 4-OMe-5- NMe 2 -3-Py], [BA4136; 6-OMe-5-NMe 2 -3-Py], [BA4137; 6-NMe 2 -3-Py], [BA4138; 2 _{-Cl-6-NMe 2 -3-} Py], [BA4139; 4-Cl-6-NMe 2 -3-Py], [BA4140; 5-Cl-6-NMe 2 -3-Py], [BA4141; _{2-Me-6-NMe 2} -3-Py], [BA4142; 4-Me-6-NMe 2 -3-Py], [BA4143; 5-Me-6-NMe 2 -3-Py], [BA4144 _{; 2-CF 3 -6-NMe} 2 -3-Py], [BA4145; 4-CF 3 -6-NMe 2 -3-Py], [BA4146; 5-CF 3 -6-NMe 2 -3-Py ], [BA4147; 2-CN -6-NMe 2 -3-Py], [BA4148; 4-CN-6-NMe 2 -3-Py], [BA4149; 5-CN-6-NMe 2 -3- Py], [BA4150; 2- OMe-6-NMe 2 -3-Py], [BA4151; 4-OMe-6-NMe 2 -3-Py], [BA4152; 5-OMe-6-NMe 2 -3 -Py], [BA4153; 2-ACNH-3-Py], [BA4154; 4-Cl-2-ACNH-3-Py], [BA4155; 5-Cl-2-ACNH-3-Py], [BA4156; 6-Cl-2-ACNH-3-Py], [BA4157; 4-Me-2-ACNH-3-Py], [BA4158; 5-Me-2-ACNH-3-Py], [BA4159 ; 6-Me-2-ACNH -3-Py], [BA4160; 4-CF 3 -2-ACNH-3-Py], [BA4161; 5-CF 3 -2-ACNH-3-Py], [BA4162 _{; 6-CF 3 -2-ACNH} -3-Py], [BA4163; 4-CN-2-ACNH-3-Py], [BA4164; 5-CN-2-ACNH-3-Py], [BA4165; 6-CN-2-ACNH-3-Py, [BA4166; 4-OMe-2-ACNH-3-Py], [BA4167; 5-OMe-2-ACNH-3-Py], [BA4168; 6- OMe-2-ACNH-3-Py, [BA4169; 4-ACNH-3-Py], [BA4170; 2-Cl-4-ACNH-3-Py], [BA4171; 5-Cl-4-ACNH- 3-Py], [BA4172; 6-Cl-4-ACNH-3-Py], [BA4173; 2-Me-4-ACNH-3-Py], [BA4174; 5-Me-4-ACNH-3- Py], [BA4175; 6- Me-4-ACNH-3-Py], [BA4176; 2-CF 3 -4-ACNH-3-Py], [BA4177; 5-CF 3 -4-ACNH-3- Py], [BA4178; 6- CF 3 -4-ACNH-3-Py], [BA4179; 2-CN-4-ACNH-3-Py], [BA4180; 5-CN-4-ACNH-3-Py ], [BA4181; 6-CN-4-ACNH-3-Py], [BA4182; 2-OMe-4-ACNH-3-Py], [BA4183; 5-OMe-4-ACNH-3-Py], [BA 4184; 6-OMe-4-ACNH-3-Py],

[BA4185; 5-ACNH-3-Py], [BA4186; 2-Cl-5-ACNH-3-Py], [BA4187; 4-Cl-5-ACNH-3-Py], [BA4188; 6-Cl -5-ACNH-3-Py, [BA 4189; 2-Me-5-ACNH-3-Py], [BA 4190; 4-Me-5-ACNH-3-Py], [BA 4191; 6-Me-5 -ACNH-3-Py], [ BA4192; 2-CF 3 -5-ACNH-3-Py], [BA4193; 4-CF 3 -5-ACNH-3-Py], [BA4194; 6-CF 3 - 5-ACNH-3-Py, [BA4195; 2-CN-5-ACNH-3-Py], [BA4196; 4-CN-5-ACNH-3-Py], [BA4197; 6-CN-5- ACNH-3-Py], [BA 4198; 2-OMe-5-ACNH-3-Py], [BA 4199; 4-OMe-5-ACNH-3-Py], [BA 4200; 6-OMe-5-ACNH- 3-Py], [BA4201; 6-ACNH-3-Py], [BA4202; 2-Cl-6-ACNH-3-Py], [BA 4203; 4-Cl-6-ACNH-3-Py], [BA-420] BA4204; 5-Cl-6-ACNH-3-Py], [BA4205; 2-Me-6-ACNH-3-Py], [BA4206; 4-Me-6-ACNH-3-Py], [BA4207; 5-Me-6-ACNH- 3-Py], [BA4208; 2-CF 3 -6-ACNH-3-Py], [BA4209; 4-CF 3 -6-ACNH-3-Py], [BA4210; _{5-CF 3 -6-ACNH-} 3-Py], [BA4211; 2-CN-6-ACNH-3-Py], [BA4212; 4-CN-6-ACNH-3-Py], [BA4213; 5 -CN-6-ACNH-3-Py], [BA4214; 2-OMe-6-ACNH-3-Py], [BA4215; 4-OMe-6-ACNH-3-Py], [BA4216; 5-OMe -6-ACNH-3-Py], [BA4217; 2- (N-AC-N-Me-N) -3-Py], [BA4218; 4-Cl-2- (N (Ac) (Me)) -3-Py !, [BA 4219; 5-Cl-2- (N (Ac) (Me))-3-Py], [BA4220; 6-Cl-2- (N (Ac) (Me))-3] -Py], [BA 4221; 4-Me-2- (N (Ac)) (Me))-3-Py], [BA4222; 5-Me-2- (N (Ac) (Me))-3-Py], [BA4223; 6-Me-2- (N (Ac) (Me) )) 3-Py], [BA 4224; 4-CF ₃ -2- (N (Ac) (Me))-3-Py], [BA 4225; 5-CF ₃ -2- (N (Ac) (Me) )) 3-Py], [BA 4226; 6-CF ₃ -2- (N (Ac) (Me))-3-Py], [BA 4227; 4-CN-2- (N (Ac) (Me)) )-[3-Py], [BA4228; 5-CN-2- (N (Ac) (Me))-3-Py], [BA4229; 6-CN-2- (N (Ac) (Me))- 3-Py], [BA 4230; 4-OMe-2- (N (Ac) (Me))-3-Py], [BA4231; 5-OMe-2- (N (Ac) (Me))-3- Py], [BA4232; 6-OMe-2- (N (Ac) (Me))-3-Py], [BA4233; 4- (N-AC-N-Me-N) -3-Py], BA 4234; 2-Cl-4- (N (Ac) (Me))-3-Py], [BA4235; 5-Cl-4- (N (Ac) (Me))-3-Py], [BA4236; 6-Cl-4- (N (Ac) (Me))-3-Py], [BA4237; 2-Me-4- (N (Ac) (Me))-3-Py], [BA4238; 5- Me-4- (N (Ac) (Me)) - 3-Py], [BA4239; 6-Me-4- (N (Ac) (Me)) - 3-Py], [BA4240; 2-CF 3 -4- (N (Ac) (Me )) - 3-Py], [BA4241; 5-CF 3 -4- (N (Ac) (Me)) - 3-Py], [BA4242; 6-CF 3 -4- (N (Ac) (Me))-3-Py], [BA4243; 2-CN-4- (N (Ac) (Me))-3-Py], [BA4244; 5-CN-4 -(N (Ac) (Me))-3-Py], [BA4245; 6-CN-4- (N (Ac) (Me))-3-Py], [BA4246; 2-OMe-4- ( N (Ac) (Me))-3-Py], [BA4247; 5-OMe-4- (N (Ac) (Me))-3-Py], [BA4248; 6-OMe-4- (N ( Ac) (Me))-3-Py], [BA4249; 5- (N-AC-N-Me-N) -3-Py], [BA4250; 2-Cl-5- (N (Ac) (Me) ))-3-Py], [BA42] 51; 4-Cl-5- (N (Ac) (Me))-3-Py], [BA4252; 6-Cl-5- (N (Ac) (Me))-3-Py], [BA4253; 2-Me-5- (N (Ac) (Me))-3-Py], [BA 4254; 4-Me-5- (N (Ac) (Me))-3-Py], [BA 4255; 6- Me-5- (N (Ac) (Me)) - 3-Py], [BA4256; 2-CF 3 -5- (N (Ac) (Me)) - 3-Py], [BA4257; 4-CF _{3 -5- (N (Ac) (} Me)) - 3-Py], [BA4258; 6-CF 3 -5- (N (Ac) (Me)) - 3-Py], [BA4259; 2-CN -5- (N (Ac) (Me))-3-Py], [BA 4260; 4-CN-5- (N (Ac) (Me))-3-Py], [BA4261; 6-CN-5 -(N (Ac) (Me))-3-Py], [BA4262; 2-OMe-5- (N (Ac) (Me))-3-Py], [BA4263; 4-OMe-5- ( N (Ac) (Me))-3-Py], [BA4264; 6-OMe-5- (N (Ac) (Me))-3-Py], [BA4265; 6- (N-AC-N-) Me-N) -3-Py], [BA4266; 2-Cl-6- (N (Ac) (Me))-3-Py], [BA4267; 4-Cl-6- (N (Ac) (Me) )) 3-Py], [BA4268; 5-Cl-6- (N (Ac) (Me))-3-Py], [BA4269; 2-Me-6- (N (Ac) (Me)) -3-Py !, [BA4270; 4-Me-6- (N (Ac) (Me))-3-Py], [BA4271; 5-Me-6- (N (Ac) (Me))-3] -Py], [BA4272; 2- CF 3 -6- (N (Ac) (Me)) - 3-Py], [BA4273; 4-CF 3 -6- (N (Ac) (Me)) - 3 -Py], [BA4274; 5- CF 3 -6- (N (Ac) (Me)) - 3-Py], [BA4275; 2-CN-6- (N (Ac) (Me)) - 3- Py], [BA4276; 4-CN-6- (N (Ac) (Me))-3-Py], [BA4277; 5-CN-6- (N (Ac) (Me))-3-Py] , [BA4278; 2-OMe-6- (N (Ac) (Me))-3-Py], [BA4279; 4-OMe-6- (N (Ac) (Me))-3-Py], [BA4 2 BA 4280; 5-OMe-6- (N (Ac) (M) e))-3-Py], [BA4281; 2-AC-3-Py], [BA4282; 4-Cl-2-AC-3-Py], [BA4283; 5-Cl-2-AC-3- Py], [BA 4284; 6-Cl-2-AC-3-Py],

[BA4285; 4-Me-2-AC-3-Py], [BA4286; 5-Me-2-AC-3-Py], [BA4287; 6-Me-2-AC-3-Py], [BA4288] _{; 4-CF 3 -2-AC} -3-Py], [BA4289; 5-CF 3 -2-AC-3-Py], [BA4290; 6-CF 3 -2-AC-3-Py], [ BA4291; 4-CN-2-AC-3-Py !, [BA4292; 5-CN-2-AC-3-Py], [BA4293; 6-CN-2-AC-3-Py], [BA4294; 4-OMe-2-AC-3-Py], [BA4295; 5-OMe-2-AC-3-Py], [BA4296; 6-OMe-2-AC-3-Py], [BA4297; AC-3-Py !, [BA4298; 2-Cl-4-AC-3-Py], [BA4299; 5-Cl-4-AC-3-Py], [BA4300; 6-Cl-4-AC- 3-Py], [BA4301; 2-Me-4-AC-3-Py], [BA4302; 5-Me-4-AC-3-Py], [BA4303; 6-Me-4-AC-3- Py], [BA4304; 2- CF 3 -4-AC-3-Py], [BA4305; 5-CF 3 -4-AC-3-Py], [BA4306; 6-CF 3 -4-AC-3 -Py], [BA4307; 2-CN-4-AC-3-Py], [BA4308; 5-CN-4-AC-3-Py], [BA4309; 6-CN-4-AC-3-Py ], [BA 4310; 2-OMe-4-AC-3-Py], [BA4311; 5-OMe-4-AC-3-Py], [BA4312; 6-OMe-4-AC-3-Py], [BA4313; 5-AC-3-Py], [BA4314; 2-Cl-5-AC-3-Py], [BA4315; 4-Cl-5-AC-3-Py], [BA4316; 6-Cl -5-AC-3-Py, [BA 4317; 2-Me-5-AC-3-Py], [BA 4318; 4-Me-5-AC-3-Py], [BA 4319; 6-Me-5 -AC-3-Py], [ BA4320; 2-CF 3 -5-AC-3-Py], [BA4321; 4-CF 3 -5-AC-3-Py], [BA4322; 6-CF 3 - 5-AC-3-Py, [BA 4323; 2-CN-5-AC-3-Py], [BA 4324; 4-CN-5-AC-3-Py], [BA 4325; 6-CN-5- AC -3-Py, [BA4326; 2-OMe-5-AC-3-Py], [BA4327; 4-OMe-5-AC-3-Py], [BA4328; 6-OMe-5-AC-3 -Py], [BA4329; 6-AC-3-Py], [BA4330; 2-Cl-6-AC-3-Py], [BA4331; 4-Cl-6-AC-3-Py], [BA4332 5-Cl-6-AC-3-Py !, [BA4333; 2-Me-6-AC-3-Py], [BA4334; 4-Me-6-AC-3-Py], [BA4335; -Me-6-AC-3- Py], [BA4336; 2-CF 3 -6-AC-3-Py], [BA4337; 4-CF 3 -6-AC-3-Py], [BA4338; 5 _{-CF 3 -6-AC-3-} Py], [BA4339; 2-CN-6-AC-3-Py], [BA4340; 4-CN-6-AC-3-Py], [BA4341; 5- CN-6-AC-3-Py, [BA4342; 2-OMe-6-AC-3-Py], [BA4343; 4-OMe-6-AC-3-Py], [BA4344; 5-OMe- 6-AC-3-Py, [BA 4345; 4-Py], 0 [BA 4346; 3-F-4-Py], [BA 4347; 2-Cl-3-F-4-Py], [BA 4 348; 5 -Cl-3-F-4-Py, [BA4349; 6-Cl-3-F-4-Py], [BA4350; 2-Me-3-F-4-Py], [BA4351; 5-Me -3-F-4-Py] , [BA4352; 6-Me-3-F-4-Py], [BA4353; 2-CF 3 -3-F-4-Py], [BA4354; 5-CF 3 -3-F-4-Py] , [BA4355; 6-CF 3 -3-F-4-Py], [BA4356; 2-CN-3-F-4-Py], [BA4357; 5-CN- 3-F-4-Py], [BA4358; 6-CN-3-F-4-Py], [BA4359; 2-OMe-3-F-4-Py], [BA4360; 5-OMe-3- F-4-Py !, [BA4361; 6-OMe-3-F-4-Py], [BA4362; 2-F-4-Py], [BA4363; 3-Cl-2-F-4-Py] [BA 4364; 5-Cl-2-F-4-Py], [BA 4365; 6-Cl-2-F-4-Py], [BA 4366; 3-Me-2-F-4-Py], [BA 4 36 4 BA 4367; 5-Me-2-F-4-Py], [B A4368; 6-Me-2- F-4-Py], [BA4369; 3-CF 3 -2-F-4-Py], [BA4370; 5-CF 3 -2-F-4-Py], [ BA 4371; 6-CF ₃ -2-F-4-Py !, [BA 4372; 3-CN-2-F-4-Py], [BA 4373; 5-CN-2-F-4-Py], [BA 4374] 6-CN-2-F-4-Py !, [BA4375; 3-OMe-2-F-4-Py], [BA4376; 5-OMe-2-F-4-Py], [BA4377; -OMe-2-F-4-Py], [BA 4378; 5-F-4-Py], [BA 4379; 3-Cl-5-F-4-Py], [BA 4380; 2-Cl-5-F -4-Py], [BA4381; 6-Cl-5-F-4-Py], [BA4382; 3-Me-5-F-4-Py], [BA4383; 2-Me-5-F-4 -Py], [BA4384; 6-Me-5-F-4-Py],

_{[BA4385; 3-CF 3 -5} -F-4-Py], [BA4386; 2-CF 3 -5-F-4-Py], [BA4387; 6-CF 3 -5-F-4-Py] , [BA4388; 3-CN-5-F-4-Py], [BA4389; 2-CN-5-F-4-Py], [BA4390; 6-CN-5-F-4-Py], [BA4390; BA 4391; 3-OMe-5-F-4-Py], [BA4392; 2-OMe-5-F-4-Py], [BA4393; 6-OMe-5-F-4-Py], [BA4394; 6-F-4-Py], [BA4395; 3-Cl-6-F-4-Py], [BA4396; 2-Cl-6-F-4-Py], [BA 4397; 5-Cl-6- 6 F-4-Py !, [BA4398; 3-Me-6-F-4-Py], [BA4399; 2-Me-6-F-4-Py], [BA4400; 5-Me-6-F- 4-Py], [BA4401; 3-CF 3 -6-F-4-Py], [BA4402; 2-CF 3 -6-F-4-Py], [BA4403; 5-CF 3 -6-F -4-Py], [BA4404; 3-CN-6-F-4-Py], [BA4405; 2-CN-6-F-4-Py], [BA4406; 5-CN-6-F-4 -Py], [BA4407; 3-OMe-6-F-4-Py], [BA4408; 2-OMe-6-F-4-Py], [BA4409; 5-OMe-6-F-4-Py ], [BA4410; 3-Cl-4-Py], [BA4411; 2-Cl-3-Cl-4-Py], [BA4412; 5-Cl-3-Cl-4-Py], [BA4413; 6] -Cl-3-Cl-4-Py], [BA4414; 2-Me-3-Cl-4-Py], [BA4415; 5-Me-3-Cl-4-Py], [BA4416; 6-Me -3-Cl-4-Py] , [BA4417; 2-CF 3 -3-Cl-4-Py], [BA4418; 5-CF 3 -3-Cl-4-Py], [BA4419; 6-CF _{3 -3-Cl-4-Py} ], [BA4420; 2-CN-3-Cl-4-Py], [BA4421; 5-CN-3-Cl-4-Py], [BA4422; 6-CN- 3-Cl-4-Py], [BA4423; 2-OMe-3-Cl-4-Py], [BA4424; 5-OMe-3-Cl-4-Py], [BA4425; 6-OMe-3- Cl-4-Py], [BA 4426; 2-Cl-4- Py], [BA4427; 3-Cl-2-Cl-4-Py], [BA4428; 5-Cl-2-Cl-4-Py], [BA4429; 6-Cl-2-Cl-4-Py] , [BA4430; 3-Me-2-Cl-4-Py], [BA4431; 5-Me-2-Cl-4-Py], [BA4432; 6-Me-2-Cl-4-Py], [BA4432; _{BA4433; 3-CF 3 -2-} Cl-4-Py], [BA4434; 5-CF 3 -2-Cl-4-Py], [BA4435; 6-CF 3 -2-Cl-4-Py], [BA4436; 3-CN-2-Cl-4-Py], [BA4437; 5-CN-2-Cl-4-Py], [BA4438; 6-CN-2-Cl-4-Py], [BA4439] 3-OMe-2-Cl-4-Py !, [BA4440; 5-OMe-2-Cl-4-Py], [BA4441; 6-OMe-2-Cl-4-Py], [BA4442; -Cl-4-Py], [BA4443; 2-Cl-5-Cl-4-Py], [BA4444; 5-Cl-5-Cl-4-Py], [BA4445; 6-Cl-5-Cl] -4-Py], [BA4446; 2-Me-5-Cl-4-Py], [BA4447; 5-Me-5-Cl-4-Py], [BA 4448; 6-Me-5-Cl-4 -Py], [BA4449; 2- CF 3 -5-Cl-4-Py], [BA4450; 5-CF 3 -5-Cl-4-Py], [BA4451; 6-CF 3 -5-Cl- 4-Py], [BA4452; 2-CN-5-Cl-4-Py], [BA4453; 3-CN-5-Cl-4-Py], [BA4454; 6-CN-5-Cl-4- Py], [BA4455; 2-OMe-5-Cl-4-Py], [BA4456; 5-OMe-5-Cl-4-Py], [BA4457; 6-OMe-5-Cl-4-Py] , [BA4458; 6-Cl-4-Py], [BA4459; 3-Cl-6-Cl-4-Py], [BA4460; 2-Cl-6-Cl-4-Py], [BA4461; Cl-6-Cl-4-Py], [BA4462; 3-Me-6-Cl-4-Py], [BA4463; 2-Me-6-Cl-4-Py], [BA 4464; 5-Me- 6-Cl-4-Py] , [BA4465; 3-CF 3 -6-Cl-4-Py], [BA4466; 2-CF 3 -6-Cl-4-Py], [BA4467; 5-CF 3 - 6-Cl-4-Py, [BA4468; 3-CN-6-Cl-4-Py], [BA4469; 2-CN-6-Cl-4-Py], [BA4470; 5-CN-6- Cl-4-Py], [BA4471; 3-OMe-6-Cl-4-Py], [BA4472; 2-OMe-6-Cl-4-Py], [BA4473; 5-OMe-6-Cl- 4-Py], [BA4474; 3-Br-4-Py], [BA4475; 2-Cl-3-Br-4-Py], [BA4476; 5-Cl-3-Br-4-Py], [BA4 4 BA4477; 6-Cl-3-Br-4-Py], [BA4478; 2-Me-3-Br-4-Py], [BA4479; 5-Me-3-Br-4-Py], [BA4480; 6-Me-3-Br- 4-Py], [BA4481; 2-CF 3 -3-Br-4-Py], [BA4482; 5-CF 3 -3-Br-4-Py], [BA4483; _{6-CF 3 -3-Br-} 4-Py], [BA4484; 2-CN-3-Br-4-Py],

[BA4485; 5-CN-3-Br-4-Py], [BA4486; 6-CN-3-Br-4-Py], [BA4487; 2-OMe-3-Br-4-Py], [BA4488] 5-OMe-3-Br-4-Py !, [BA4489; 6-OMe-3-Br-4-Py], [BA4490; 2-Br-4-Py], [BA4491; 3-Cl-2 -Br-4-Py], [BA4492; 5-Cl-2-Br-4-Py], [BA4493; 6-Cl-2-Br-4-Py], [BA4494; 3-Me-2-Br -4-Py], [BA4495; 5-Me-2-Br-4-Py], [BA4496; 6-Me-2-Br-4-Py], [BA4497; 3-CF 3 -2-Br- 4-Py], [BA4498; 5-CF 3 -2-Br-4-Py], [BA4499; 6-CF 3 -2-Br-4-Py], [BA4500; 3-CN-2-Br- 4-Py], [BA4501; 5-CN-2-Br-4-Py], [BA4502; 6-CN-2-Br-4-Py], [BA4503; 3-OMe-2-Br-4- Py], [BA4504; 5-OMe-2-Br-4-Py], [BA4505; 6-OMe-2-Br-4-Py], [BA4506; 5-Br-4-Py], [BA4507; 3-Cl-5-Br-4-Py], [BA4508; 2-Cl-5-Br-4-Py], [BA4509; 6-Cl-5-Br-4-Py], [BA 4510; Me-5-Br-4- Py], [BA4511; 2-Me-5-Br-4-Py], [BA4512; 6-Me-5-Br-4-Py], [BA4513; 3-CF 3 -5-Br-4-Py] , [BA4514; 2-CF 3 -5-Br-4-Py], [BA4515; 6-CF 3 -5-Br-4-Py], [BA4516; 3-CN -5-Br-4-Py !, [BA4517; 2-CN-5-Br-4-Py], [BA4518; 6-CN-5-Br-4-Py], [BA4519; 3-OMe-5 -Br-4-Py], [BA4520; 2-OMe-5-Br-4-Py], [BA4521; 6-OMe-5-Br-4-Py], [BA4522; 6-Br-4-Py ], [BA4523; 3-Cl-6-Br-4-Py], [BA4524; 2-Cl-6-Br-4-Py], [BA4525; 5-Cl-6-Br-4-Py], [BA4 526; 3-Me-6-Br-4-Py], [BA4527; 2-Me-6-Br-4-Py], [BA4528; 5-Me-6-Br-4-Py], [BA4529; _{3-CF 3 -6-Br-} 4-Py], [BA4530; 2-CF 3 -6-Br-4-Py], [BA4531; 5-CF 3 -6-Br-4-Py], [BA4532 3-CN-6-Br-4-Py !, [BA4533; 2-CN-6-Br-4-Py], [BA4534; 5-CN-6-Br-4-Py], [BA4535; -OMe-6-Br-4-Py], [BA4536; 2-OMe-6-Br-4-Py], [BA4537; 5-OMe-6-Br-4-Py], [BA4538; 3-I -4-Py !, [BA4539; 2-Cl-3-I-4-Py], [BA4540; 5-Cl-3-I-4-Py], [BA4541; 6-Cl-3-I-4 -Py], [BA4542; 2-Me-3-I-4-Py], [BA4543; 5-Me-3-I-4-Py], [BA4544; 6-Me-3-I-4-Py ], [BA4545; 2-CF 3 -3-I-4-Py], [BA4546; 5-CF 3 -3-I-4-Py], [BA4547; 6-CF 3 -3-I-4- Py], [BA4548; 2-CN-3-I-4-Py], [BA4549; 5-CN-3-I-4-Py], [BA4550; 6-CN-3-I-4-Py] , [BA4551; 2-OMe-3-I-4-Py], [BA4552; 5-OMe-3-I-4-Py], [BA4553; 6-OMe-3-I-4-Py], [BA4552; BA 4554; 2-I-4-Py], [BA4555; 3-Cl-2-I-4-Py], [BA4556; 5-Cl-2-I-4-Py], [BA4557; 6-Cl- 2-I-4-Py, [BA4558; 3-Me-2-I-4-Py], [BA4559; 5-Me-2-I-4-Py], [BA4560; 6-Me-2- I-4-Py], [ BA4561; 3-CF 3 -2-I-4-Py], [BA4562; 5-CF 3 -2-I-4-Py], [BA4563; 6-CF 3 -2 -I-4-Py], [BA4564; 3-CN-2-I-4-Py], [BA4565; 5-CN-2-I-4-Py], [BA4566; 6-CN-2-I -4-Py], [BA4567; 3-OMe-2-I-4-Py], [B A4568; 5-OMe-2-I-4-Py, [BA4569; 6-OMe-2-I-4-Py], [BA4570; 5-I-4-Py], [BA4571; 3-Cl- 5-I-4-Py, [BA4572; 2-Cl-5-I-4-Py], [BA4573; 6-Cl-5-I-4-Py], [BA4574; 3-Me-5-5 I-4-Py], [ BA4575; 2-Me-5-I-4-Py], [BA4576; 6-Me-5-I-4-Py], [BA4577; 3-CF 3 -5-I -4-Py], [BA4578; 2-CF 3 -5-I-4-Py], [BA4579; 6-CF 3 -5-I-4-Py], [BA4580; 3-CN-5-I -4-Py !, [BA4581; 2-CN-5-I-4-Py], [BA4582; 6-CN-5-I-4-Py], [BA4583; 3-OMe-5-I-4 -Py], [BA4584; 2-OMe-5-I-4-Py],

[BA 4585; 6-OMe-5-I-4-Py], [BA 4586; 6-I-4-Py], [BA 4587; 3-Cl-6-I-4-Py], [BA 4588; 2-Cl -6-I-4-Py], [BA 4589; 5-Cl-6-I-4-Py], [BA 4590; 3-Me-6-I-4-Py], [BA 4591; 2-Me-6 -I-4-Py], [ BA4592; 5-Me-6-I-4-Py], [BA4593; 3-CF 3 -6-I-4-Py], [BA4594; 2-CF 3 -6 -I-4-Py], [ BA4595; 5-CF 3 -6-I-4-Py], [BA4596; 3-CN-6-I-4-Py], [BA4597; 2-CN-6- I-4-Py], [BA 4598; 5-CN-6-I-4-Py], [BA 4599; 3-OMe-6-I-4-Py], [BA4600; 2-OMe-6-I- 4-Py], [BA4601; 5-OMe-6-I-4-Py], [BA4602; 3-Me-4-Py], [BA4603; 2-Cl-3-Me-4-Py], [BA-460]; BA4604; 5-Cl-3-Me-4-Py], [BA4605; 6-Cl-3-Me-4-Py], [BA4606; 2-Me-3-Me-4-Py], [BA4607; 5-Me-3-Me- 4-Py], [BA4608; 6-Me-3-Me-4-Py], [BA4609; 2-CF 3 -3-Me-4-Py], [BA4610; 5 _{-CF 3 -3-Me-4-} Py], [BA4611; 6-CF 3 -3-Me-4-Py], [BA4612; 2-CN-3-Me-4-Py], [BA4613; 5 -CN-3-Me-4-Py], [BA4614; 6-CN-3-Me-4-Py], [BA4615; 2-OMe-3-Me-4-Py], [BA4616; 5-OMe -3-Me-4-Py !, [BA4617; 6-OMe-3-Me-4-Py], [BA4618; 2-Me-4-Py], [BA4619; 3-Cl-2-Me-4 -Py], [BA4620; 5-Cl-2-Me-4-Py], [BA4621; 6-Cl-2-Me-4-Py], [BA4622; 3-Me-2-Me-4-Py ], [BA4623; 5-Me -2-Me-4-Py], [BA4624; 6-Me-2-Me-4-Py], [BA4625; 3-CF 3 -2-Me-4-Py] , [BA4626; 5-CF ₃ -2-Me -4-Py], [BA4627; 6-CF 3 -2-Me-4-Py], [BA4628; 3-CN-2-Me-4-Py], [BA4629; 5-CN-2-Me- 4-Py], [BA4630; 6-CN-2-Me-4-Py], [BA4631; 3-OMe-2-Me-4-Py], [BA4632; 5-OMe-2-Me-4- 4 Py], [BA4633; 6-OMe-2-Me-4-Py], [BA4634; 5-Me-4-Py], [BA4635; 3-Cl-5-Me-4-Py], [BA4636; 2-Cl-5-Me-4-Py], [BA4637; 6-Cl-5-Me-4-Py], [BA4638; 3-Me-5-Me-4-Py], [BA4639; 2- Me-5-Me-4- Py], [BA4640; 6-Me-5-Me-4-Py], [BA4641; 3-CF 3 -5-Me-4-Py], [BA4642; 2-CF _{3 -5-Me-4-Py} ], [BA4643; 6-CF 3 -5-Me-4-Py], [BA4644; 3-CN-5-Me-4-Py], [BA4645; 2-CN -5-Me-4-Py], [BA4646; 6-CN-5-Me-4-Py], [BA4647; 3-OMe-5-Me-4-Py], [BA4648; 2-OMe-5 -Me-4-Py], [BA4649; 6-OMe-5-Me-4-Py], [BA4650; 6-Me-4-Py], [BA4651; 3-Cl-6-Me-4-Py ], [BA4652; 2-Cl-6-Me-4-Py], [BA4653; 5-Cl-6-Me-4-Py], [BA4654; 3-Me-6-Me-4-Py], [BA4655; 2-Me-6 -Me-4-Py], [BA4656; 5-Me-6-Me-4-Py], [BA4657; 3-CF 3 -6-Me-4-Py], [ _{BA4658; 2-CF 3 -6-} Me-4-Py], [BA4659; 5-CF 3 -6-Me-4-Py], [BA4660; 3-CN-6-Me-4-Py], [ BA4661; 2-CN-6-Me-4-Py], [BA4662; 5-CN-6-Me-4-Py], [BA4663; 3-OMe-6-Me-4-Py], [BA4664; 2-OMe-6-Me-4-Py], [BA4665; 5-OMe-6-Me-4-Py], [BA4666; 3-OMe-4-Py], [BA4667; 2-Cl-3- OM e-4-Py], [BA4668; 5-Cl-3-OMe-4-Py], [BA4669; 6-Cl-3-OMe-4-Py], [BA4670; 2-Me-3-OMe- 4-Py], [BA4671; 5-Me-3-OMe-4-Py], [BA4672; 6-Me-3-OMe-4-Py], [BA4673; 2-CF 3 -3-OMe-4 -Py], [BA4674; 5- CF 3 -3-OMe-4-Py], [BA4675; 6-CF 3 -3-OMe-4-Py], [BA4676; 2-CN-3-OMe-4 -Py], [BA4677; 5-CN-3-OMe-4-Py], [BA4678; 6-CN-3-OMe-4-Py], [BA4679; 2-OMe-3-OMe-4-Py ], [BA4680; 5-OMe-3-OMe-4-Py], [BA4681; 6-OMe-3-OMe-4-Py], [BA4682; 2-OMe-4-Py], [BA4683; 3] -Cl-2-OMe-4-Py], [BA4684; 5-Cl-2-OMe-4-Py],

[BA 4685; 6-Cl-2-OMe-4-Py], [BA 4686; 3-Me-2-OMe-4-Py], [BA4687; 5-Me-2-OMe-4-Py], [BA 4688] ; 6-Me-2-OMe -4-Py], [BA4689; 3-CF 3 -2-OMe-4-Py], [BA4690; 5-CF 3 -2-OMe-4-Py], [BA4691 _{; 6-CF 3 -2-OMe} -4-Py], [BA4692; 3-CN-2-OMe-4-Py], [BA4693; 5-CN-2-OMe-4-Py], [BA4694; 6-CN-2-OMe-4-Py], [BA4695; 3-OMe-2-OMe-4-Py], [BA4696; 5-OMe-2-OMe-4-Py], [BA4697; OMe-2-OMe-4-Py], [BA4698; 5-OMe-4-Py], [BA4699; 3-Cl-5-OMe-4-Py], [BA4700; 2-Cl-5-OMe- 4-Py], [BA4701; 6-Cl-5-OMe-4-Py], [BA4702; 3-Me-5-OMe-4-Py], [BA4703; 2-Me-5-OMe-4- Py], [BA4704; 6- Me-5-OMe-4-Py], [BA4705; 3-CF 3 -5-OMe-4-Py], [BA4706; 2-CF 3 -5-OMe-4- Py], [BA4707; 6- CF 3 -5-OMe-4-Py], [BA4708; 3-CN-5-OMe-4-Py], [BA4709; 2-CN-5-OMe-4-Py ], [BA 4710; 6-CN-5-OMe-4-Py], [BA4711; 3-OMe-5-OMe-4-Py], [BA4712; 2-OMe-5-OMe-4-Py], [BA4713; 6-OMe-5-OMe-4-Py], [BA4714; 6-OMe-4-Py], [BA4715; 3-Cl-6-OMe-4-Py], [BA4716; 2-Cl -6-OMe-4-Py !, [BA 4717; 5-Cl-6-OMe-4-Py], [BA 4718; 3-Me-6-OMe-4-Py], [BA 4719; 2-Me-6 -OMe-4-Py], [ BA4720; 5-Me-6-OMe-4-Py], [BA4721; 3-CF 3 -6-OMe-4-Py], [BA4722; 2-CF 3 -6 -OMe-4-Py], [ BA4723; 5-CF 3 -6-OMe-4-Py], [B A4724; 3-CN-6-OMe-4-Py], [BA4725; 2-CN-6-OMe-4-Py], [BA4726; 5-CN-6-OMe-4-Py], [BA4727; 3-OMe-6-OMe-4-Py], [BA4728; 2-OMe-6-OMe-4-Py], [BA4729; 5-OMe-6-OMe-4-Py], [BA4730; 3- _{CF 3 -4-Py], [} BA4731; 2-Cl-3-CF 3 -4-Py], [BA4732; 5-Cl-3-CF 3 -4-Py], [BA4733; 6-Cl-3 _{-CF 3 -4-Py], [} BA4734; 2-Me-3-CF 3 -4-Py], [BA4735; 5-Me-3-CF 3 -4-Py], [BA4736; 6-Me- _{3-CF 3 -4-Py]} , [BA4737; 2-CF 3 -3-CF 3 -4-Py], [BA4738; 5-CF 3 -3-CF 3 -4-Py], [BA4739; 6 _{-CF 3 -3-CF 3 -4-} Py], [BA4740; 2-CN-3-CF 3 -4-Py], [BA4741; 5-CN-3-CF 3 -4-Py], [BA4742 ; 6-CN-3-CF 3 -4-Py], [BA4743; 2-OMe-3-CF 3 -4-Py], [BA4744; 5-OMe-3-CF 3 -4-Py], [ BA4745; 6-OMe-3- CF 3 -4-Py], [BA4746; 2-CF 3 -4-Py], [BA4747; 3-Cl-2-CF 3 -4-Py], [BA4748; 5 _{-Cl-2-CF 3 -4-} Py], [BA4749; 6-Cl-2-CF 3 -4-Py], [BA4750; 3-Me-2-CF 3 -4-Py], [BA4751; _{5-Me-2-CF 3} -4-Py], [BA4752; 6-Me-2-CF 3 -4-Py], [BA4753; 3-CF 3 -2-CF 3 -4-Py], [ BA 4754; 5-CF ₃ -2-CF ₃ -4-Py], [BA 4 755; 6-CF ₃ -2-CF ₃ -4-Py], [BA 4 756; 3-CN-2-CF ₃ -4-Py ], [BA4757; 5-CN -2-CF 3 -4-Py], [BA4758; 6-CN-2-CF 3 -4-Py], [BA4759; 3-OMe-2-CF 3 -4- Py], [BA 4760; 5-OMe-2-CF ₃ -4-Py] , [BA4761; 6-OMe- 2-CF 3 -4-Py], [BA4762; 5-CF 3 -4-Py], [BA4763; 3-Cl-5-CF 3 -4-Py], [BA4764 ; 2-Cl-5-CF 3 -4-Py], [BA4765; 6-Cl-5-CF 3 -4-Py], [BA4766; 3-Me-5-CF 3 -4-Py], [ BA 4767; 2-Me-5-CF ₃ -4-Py], [BA 4768; 6-Me-5-CF ₃ -4-Py], [BA 4769; 3-CF ₃ -5-CF ₃ -4-Py] _{, [BA4770; 2-CF 3} -5-CF 3 -4-Py], [BA4771; 6-CF 3 -5-CF 3 -4-Py], [BA4772; 3-CN-5-CF 3 -4 -Py], [BA 4773; 2-CN-5-CF ₃ -4-Py], [BA 4774; 6-CN-5-CF ₃ -4-Py], [BA 4775; 3-OMe-5-CF _3- 4-Py], [BA4776; 2-OMe-5-CF 3 -4-Py], [BA4777; 6-OMe-5-CF 3 -4-Py], [BA4778; 6-CF 3 -4-Py ], [BA4779; 3-Cl -6-CF 3 -4-Py], [BA4780; 2-Cl-6-CF 3 -4-Py], [BA4781; 5-Cl-6-CF 3 -4- Py], [BA4782; 3- Me-6-CF 3 -4-Py], [BA4783; 2-Me-6-CF 3 -4-Py], [BA4784; 5-Me-6-CF 3 -4 -Py],

_{[BA4785; 3-CF 3 -6} -CF 3 -4-Py], [BA4786; 2-CF 3 -6-CF 3 -4-Py], [BA4787; 5-CF 3 -6-CF 3 -4 -Py], [BA4788; 3- CN-6-CF 3 -4-Py], [BA4789; 2-CN-6-CF 3 -4-Py], [BA4790; 5-CN-6-CF 3 - 4-Py], [BA4791; 3-OMe-6-CF 3 -4-Py], [BA4792; 2-OMe-6-CF 3 -4-Py], [BA4793; 5-OMe-6-CF 3 -4-Py], [BA4794; 3-OCF 3 -4-Py], [BA4795; 2-Cl-3-OCF 3 -4-Py], [BA4796; 5-Cl-3-OCF 3 -4- Py], [BA4797; 6- Cl-3-OCF 3 -4-Py], [BA4798; 2-Me-3-OCF 3 -4-Py], [BA4799; 5-Me-3-OCF 3 -4 -Py], [BA4800; 6- Me-3-OCF 3 -4-Py], [BA4801; 2-CF 3 -3-OCF 3 -4-Py], [BA4802; 5-CF 3 -3-OCF _{3 -4-Py], [BA4803} ; 6-CF 3 -3-OCF 3 -4-Py], [BA4804; 2-CN-3-OCF 3 -4-Py], [BA4805; 5-CN-3 _{-OCF 3 -4-Py], [} BA4806; 6-CN-3-OCF 3 -4-Py], [BA4807; 2-OMe-3-OCF 3 -4-Py], [BA4808; 5-OMe- _{3-OCF 3 -4-Py]} , [BA4809; 6-OMe-3-OCF 3 -4-Py], [BA4810; 2-OCF 3 -4-Py], [BA4811; 3-Cl-2-OCF ₃ -4-Py !, [BA 4812; 5-Cl-2-OCF ₃ -4-Py], [BA 4813; 6-Cl 2-OCF ₃ -4-Py], [BA 4814; _{OCF 3 -4-Py], [} BA4815; 5-Me-2-OCF 3 -4-Py], [BA4816; 6-Me-2-OCF 3 -4-Py], [BA4817; 3-CF 3 - _{2-OCF 3 -4-Py]} , [BA4818; 5-CF 3 -2-OCF 3 -4-Py], [BA4819; 6-CF 3 -2-OCF 3 -4-Py], [BA482 0; 3-CN-2- OCF 3 -4-Py], [BA4821; 5-CN-2-OCF 3 -4-Py], [BA4822; 6-CN-2-OCF 3 -4-Py], [BA4823; 3-OMe-2 -OCF 3 -4-Py], [BA4824; 5-OMe-2-OCF 3 -4-Py], [BA4825; 6-OMe-2-OCF 3 -4-Py] _{, [BA4826; 5-OCF 3} -4-Py], [BA4827; 3-Cl-5-OCF 3 -4-Py], [BA4828; 2-Cl-5-OCF 3 -4-Py], [BA4829 ; 6-Cl-5-OCF 3 -4-Py], [BA4830; 3-Me-5-OCF 3 -4-Py], [BA4831; 2-Me-5-OCF 3 -4-Py], [ BA 4832; 6-Me-5-OCF ₃ -4-Py !, [BA 4833; 3-CF ₃ -5-OCF ₃ -4-Py], [BA 4834; 2-CF ₃ -5-OCF ₃ -4-Py ], [BA4835; 6-CF 3 -5-OCF 3 -4-Py], [BA4836; 3-CN-5-OCF 3 -4-Py], [BA4837; 2-CN-5-OCF 3 -4 -Py], [BA4838; 6- CN-5-OCF 3 -4-Py], [BA4839; 3-OMe-5-OCF 3 -4-Py], [BA4840; 2-OMe-5-OCF 3 - 4-Py], [BA4841; 6-OMe-5-OCF 3 -4-Py], [BA4842; 6-OCF 3 -4-Py], [BA4843; 3-Cl-6-OCF 3 -4-Py ], [BA4844; 2-Cl -6-OCF 3 -4-Py], [BA4845; 5-Cl-6-OCF 3 -4-Py], [BA4846; 3-Me-6-OCF 3 -4- Py], [BA4847; 2- Me-6-OCF 3 -4-Py], [BA4848; 5-Me-6-OCF 3 -4-Py], [BA4849; 3-CF 3 -6-OCF 3 - 4-Py], [BA4850; 2-CF 3 -6-OCF 3 -4-Py], [BA4851; 5-CF 3 -6-OCF 3 -4-Py], [BA4852; 3-CN-6- _{OCF 3 -4-Py], [} BA4853; 2-CN-6-OCF 3 -4-Py], [BA4854; 5-CN-6-OCF 3 -4-Py], [BA4855; 3-OM _{e-6-OCF 3 -4-} Py], [BA4856; 2-OMe-6-OCF 3 -4-Py], [BA4857; 5-OMe-6-OCF 3 -4-Py], [BA4858; 3 _{-CHF 2 -4-Py], [} BA4859; 2-Cl-3-CHF 2 -4-Py], [BA4860; 5-Cl-3-CHF 2 -4-Py], [BA4861; 6-Cl- _{3-CHF 2 -4-Py]} , [BA4862; 2-Me-3-CHF 2 -4-Py], [BA4863; 5-Me-3-CHF 2 -4-Py], [BA4864; 6-Me -3-CHF ₂ -4-Py !, [BA 4865; 2-CF ₃ -3-CHF ₂ -4-Py], [BA 4866; 5-CF ₃ -3-CHF ₂ -4-Py], [BA 4867; _{6-CF 3 -3-CHF 2} -4-Py], [BA4868; 2-CN-3-CHF 2 -4-Py], [BA4869; 5-CN-3-CHF 2 -4-Py], [ BA4870; 6-CN-3- CHF 2 -4-Py], [BA4871; 2-OMe-3-CHF 2 -4-Py], [BA4872; 5-OMe-3-CHF 2 -4-Py], [BA4873; 6-OMe-3 -CHF 2 -4-Py], [BA4874; 4-CHF 2 -4-Py], [BA4875; 3-Cl-4-CHF 2 -4-Py], [BA4876; _{5-Cl-4-CHF 2} -4-Py], [BA4877; 6-Cl-4-CHF 2 -4-Py], [BA4878; 3-Me-4-CHF 2 -4-Py], [BA4879 ; 5-Me-4-CHF 2 -4-Py], [BA4880; 6-Me-4-CHF 2 -4-Py], [BA4881; 3-CF 3 -4-CHF 2 -4-Py], _{[BA4882; 5-CF 3 -4} -CHF 2 -4-Py], [BA4883; 6-CF 3 -4-CHF 2 -4-Py], [BA4884; 3-CN-4-CHF 2 -4- Py],

[BA4885; 5-CN-4 -CHF 2 -4-Py], [BA4886; 6-CN-4-CHF 2 -4-Py], [BA4887; 3-OMe-4-CHF 2 -4-Py] , [BA4888; 5-OMe- 4-CHF 2 -4-Py], [BA4889; 6-OMe-4-CHF 2 -4-Py], [BA4890; 5-CHF 2 -4-Py], [BA4891 ; 3-Cl-5-CHF 2 -4-Py], [BA4892; 2-Cl-5-CHF 2 -4-Py], [BA4893; 6-Cl-5-CHF 2 -4-Py], [ BA 4894; 3-Me-5-CHF ₂ -4-Py], [BA 4895; 2-Me-5-CHF ₂ -4-Py], [BA 4896; 6-Me-5-CHF ₂ -4-Py], [BA 4897; 3-CF ₃ -5-CHF ₂ -4-Py], [BA 4898; 2-CF ₃ -5-CHF ₂ -4-Py], [BA 4899; 6-CF ₃ -5-CHF _2-4 -Py], [BA4900; 3- CN-5-CHF 2 -4-Py], [BA4901; 2-CN-5-CHF 2 -4-Py], [BA4902; 6-CN-5-CHF 2 - 4-Py], [BA4903; 3-OMe-5-CHF ₂ -4-Py], [BA 4904; 2-OMe-5-CHF ₂ -4-Py], [BA 4905; 6-OMe-5-CHF ₂ -4-Py], [BA4906; 6-CHF 2 -4-Py], [BA4907; 3-Cl-6-CHF 2 -4-Py], [BA4908; 2-Cl-6-CHF 2 -4- Py], [BA4909; 5- Cl-6-CHF 2 -4-Py], [BA4910; 3-Me-6-CHF 2 -4-Py], [BA4911; 2-Me-6-CHF 2 -4 -Py], [BA4912; 5- Me-6-CHF 2 -4-Py], [BA4913; 3-CF 3 -6-CHF 2 -4-Py], [BA4914; 2-CF 3 -6-CHF ₂ -4-Py !, [BA 4915; 5-CF ₃ -6-CHF ₂ -4-Py], [BA 4916; 3-CN-6-CHF ₂ -4-Py], [BA 4917; 2-CN-6 _{-CHF 2 -4-Py], [} BA4918; 5-CN-6-CHF 2 -4-Py], [BA4919; 3-OMe-6-CHF 2 -4-Py], [BA49 20; 2-OMe-6- CHF 2 -4-Py], [BA4921; 5-OMe-6-CHF 2 -4-Py], [BA4922; 3-OCHF 2 -4-Py], [BA4923; 2 _{-Cl-3-OCHF 2 -4-} Py], [BA4924; 5-Cl-3-OCHF 2 -4-Py], [BA4925; 6-Cl-3-OCHF 2 -4-Py], [BA4926; 2-Me-3-OCHF ₂ -4-Py !, [BA 4927; 5-Me-3-OCHF ₂ -4-Py], [BA 4928; 6-Me-3-OCHF ₂ -4-Py], [BA 4929] _{; 2-CF 3 -3-OCHF} 2 -4-Py], [BA4930; 5-CF 3 -3-OCHF 2 -4-Py], [BA4931; 6-CF 3 -3-OCHF 2 -4-Py ], [BA4932; 2-CN -3-OCHF 2 -4-Py], [BA4933; 5-CN-3-OCHF 2 -4-Py], [BA4934; 6-CN-3-OCHF 2 -4- Py], [BA4935; 2- OMe-3-OCHF 2 -4-Py], [BA4936; 5-OMe-3-OCHF 2 -4-Py], [BA4937; 6-OMe-3-OCHF 2 -4 -Py], [BA4938; 4- OCHF 2 -4-Py], [BA4939; 3-Cl-4-OCHF 2 -4-Py], [BA4940; 5-Cl-4-OCHF 2 -4-Py] , [BA4941; 6-Cl- 4-OCHF 2 -4-Py], [BA4942; 3-Me-4-OCHF 2 -4-Py], [BA4943; 5-Me-4-OCHF 2 -4-Py ], [BA 4944; 6-Me-4-OCHF ₂ -4-Py], [BA 4945; 3-CF ₃ -4-OCHF ₂ -4-Py], [BA 4946; 5-CF ₃ -4-OCHF _2- 4-Py], [BA4947; 6-CF 3 -4-OCHF 2 -4-Py], [BA4948; 3-CN-4-OCHF 2 -4-Py], [BA4949; 5-CN-4-OCHF _{2 -4-Py], [BA4950} ; 6-CN-4-OCHF 2 -4-Py], [BA4951; 3-OMe-4-OCHF 2 -4-Py], [BA4952; 5-OMe-4- OHF ₂ -4-Py], [BA 4953; 6-OMe -4-OCHF ₂ -4-Py], [BA 49 _{54; 5-OCHF 2 -4-} Py], [BA4955; 3-Cl-5-OCHF 2 -4-Py], [BA4956; 2-Cl-5-OCHF 2 -4-Py], [BA4957; 6 -Cl-5-OCHF ₂ -4-Py], [BA 4958; 3-Me-5-OCHF ₂ -4-Py], [BA 4959; 2-Me-5-OCHF ₂ -4-Py], [BA 4960; _{6-Me-5-OCHF 2} -4-Py], [BA4961; 3-CF 3 -5-OCHF 2 -4-Py], [BA4962; 2-CF 3 -5-OCHF 2 -4-Py], _{[BA4963; 6-CF 3 -5} -OCHF 2 -4-Py], [BA4964; 3-CN-5-OCHF 2 -4-Py], [BA4965; 2-CN-5-OCHF 2 -4-Py ], [BA 4966; 6-CN-5-OCHF ₂ -4-Py], [BA 4967; 3-OMe-5-OCHF ₂ -4-Py], [BA 4968; 2-OMe -5-OCHF ₂ -4-] Py], [BA4969; 6- OMe-5-OCHF 2 -4-Py], [BA4970; 6-OCHF 2 -4-Py], [BA4971; 3-Cl-6-OCHF 2 -4-Py], [BA4972; 2-Cl-6 -OCHF 2 -4-Py], [BA4973; 5-Cl-6-OCHF 2 -4-Py], [BA4974; 3-Me-6-OCHF 2 -4-Py] , [BA4975; 2-Me- 6-OCHF 2 -4-Py], [BA4976; 5-Me-6-OCHF 2 -4-Py], [BA4977; 3-CF 3 -6-OCHF 2 -4- Py], [BA4978; 2- CF 3 -6-OCHF 2 -4-Py], [BA4979; 5-CF 3 -6-OCHF 2 -4-Py], [BA4980; 3-CN-6-OCHF 2 -4-Py], [BA4981; 2-CN-6-OCHF 2 -4-Py], [BA4982; 5-CN-6-OCHF 2 -4-Py], [BA4983; 3-OMe-6-OCHF ₂ -4-Py], [BA4984; 2-OMe-6-OCHF ₂ -4-Py],

[BA4985; 5-OMe-6 -OCHF 2 -4-Py], [BA4986; 3-Et-4-Py], [BA4987; 2-Cl-3-Et-4-Py], [BA4988; 5- Cl-3-Et-4-Py], [BA 4989; 6-Cl-3-Et-4-Py], [BA4990; 2-Me-3-Et-4-Py], [BA4991; 5-Me- 3-Et-4-Py] , [BA4992; 6-Me-3-Et-4-Py], [BA4993; 2-CF 3 -3-Et-4-Py], [BA4994; 5-CF 3 - 3-Et-4-Py] , [BA4995; 6-CF 3 -3-Et-4-Py], [BA4996; 2-CN-3-Et-4-Py], [BA4997; 5-CN-3 -Et-4-Py], [BA4998; 6-CN-3-Et-4-Py], [BA4999; 2-OMe-3-Et-4-Py], [BA5000; 5-OMe-3-Et -4-Py], [BA 5001; 6-OMe-3-Et-4-Py], [BA 5002; 2-Et-4-Py], [BA 5003; 3-Cl-2-Et-4-Py], [BA 5004; 5-Cl-2-Et-4-Py], [BA 5005; 6-Cl-2-Et-4-Py], [BA 5006; 3-Me-2-Et-4-Py], [BA 5007] ; 5-Me-2-Et -4-Py], [BA5008; 6-Me-2-Et-4-Py], [BA5009; 3-CF 3 -2-Et-4-Py], [BA5010; _{5-CF 3 -2-Et-} 4-Py], [BA5011; 6-CF 3 -2-Et-4-Py], [BA5012; 3-CN-2-Et-4-Py], [BA5013; 5-CN-2-Et-4-Py !, [BA5014; 6-CN-2-Et-4-Py], [BA5015; 3-OMe-2-Et-4-Py], [BA5016; 5- OMe-2-Et-4-Py], [BA5017; 6-OMe-2-Et-4-Py], [BA5018; 5-Et-4-Py], [BA5019; 3-Cl-5-Et- 4-Py], [BA 5020; 2-Cl-5-Et-4-Py], [BA 5021; 6-Cl-5-Et-4-Py], [BA 5022; 3-Me-5-Et-4- Py], [BA5023; 2- Me-5-Et-4-Py], [BA5024; 6-Me-5-Et-4-Py], [BA5025; 3-CF 3 -5-Et-4-Py ], [BA5026; 2-CF 3 -5-Et-4-Py], [BA5027; 6-CF 3 -5-Et-4-Py], [BA5028; 3-CN-5-Et-4-Py ], [BA5029; 2-CN-5-Et-4-Py], [BA5030; 6-CN-5-Et-4-Py], [BA5031; 3-OMe-5-Et-4-Py], [BA 5032; 2-OMe-5-Et-4-Py], [BA 5033; 6-OMe-5-Et-4-Py], [BA 5034; 6-Et-4-Py], [BA 50 35; 3-Cl -6-Et-4-Py], [BA 5036; 2-Cl-6-Et-4-Py], [BA 5037; 5-Cl-6-Et-4-Py], [BA 5038; 3-Me-6 -Et-4-Py], [BA5039; 2-Me-6-Et-4-Py], [BA5040; 5-Me-6-Et-4-Py], [BA5041; 3-CF ₃ -6- Et-4-Py], [ BA5042; 2-CF 3 -6-Et-4-Py], [BA5043; 5-CF 3 -6-Et-4-Py], [BA5044; 3-CN-6- Et-4-Py !, [BA5045; 2-CN-6-Et-4-Py], [BA5046; 5-CN-6-Et-4-Py], [BA5047; 3-OMe-6-Et- 4-Py], [BA5048; 2-OMe-6-Et-4-Py], [BA5049; 5-OMe-6-Et-4-Py], [BA5050; 3-CH ₂ CF ₃ -4-Py ], [BA5051; 2-Cl -3-CH 2 CF 3 -4-Py], [BA5052; 5-Cl-3-CH 2 CF 3 -4-Py], [BA5053; 6-Cl-3-CH _{2 CF 3 -4-Py],} [BA5054; 2-Me-3-CH 2 CF 3 -4-Py], [BA5055; 5-Me-3-CH 2 CF 3 -4-Py], [BA5056; _{6-Me-3-CH 2} CF 3 -4-Py], [BA5057; 2-CF 3 -3-CH 2 CF 3 -4-Py], [BA5058; 5-CF 3 -3-CH 2 CF 3 -4-Py], [BA5059; 6-CF 3 -3-CH 2 CF 3 -4-Py], [BA5060; 2-CN-3-CH 2 CF 3 -4-Py], [BA5061; 5- _{CN-3-CH 2 CF 3} -4-Py], [BA5062; 6-CN-3-CH _{2 CF 3 -4-Py],} [BA5063; 2-OMe-3-CH 2 CF 3 -4-Py], [BA5064; 5-OMe-3-CH 2 CF 3 -4-Py], [BA5065; _{6-OMe-3-CH 2} CF 3 -4-Py], [BA5066; 2-CH 2 CF 3 -4-Py], [BA5067; 3-Cl-2-CH 2 CF 3 -4-Py], [BA5068; 5-Cl-2 -CH 2 CF 3 -4-Py], [BA5069; 6-Cl-2-CH 2 CF 3 -4-Py], [BA5070; 3-Me-2-CH 2 CF _{3 -4-Py], [BA5071} ; 5-Me-2-CH 2 CF 3 -4-Py], [BA5072; 6-Me-2-CH 2 CF 3 -4-Py], [BA5073; 3- CF ₃ -2-CH ₂ CF ₃ -4-Py, [BA 5074; 5-CF ₃ -2-CH ₂ CF ₃ -4-Py], [BA 5075; 6-CF ₃ -2-CH ₂ CF _3- 4-Py], [BA5076; 3-CN-2-CH 2 CF 3 -4-Py], [BA5077; 5-CN-2-CH 2 CF 3 -4-Py], [BA5078; 6-CN- _{2-CH 2 CF 3 -4-} Py], [BA5079; 3-OMe-2-CH 2 CF 3 -4-Py], [BA5080; 5-OMe-2-CH 2 CF 3 -4-Py], [BA 5081; 6-OMe-2-CH ₂ CF ₃ -4-Py], [BA 5082; 5-CH ₂ CF ₃ -4-Py], [BA 5083; 3-Cl-5-CH ₂ CF ₃ -4- Py], [BA 5084; 2-Cl-5-CH ₂ CF ₃ -4-Py],

[BA5085; 6-Cl-5 -CH 2 CF 3 -4-Py], [BA5086; 3-Me-5-CH 2 CF 3 -4-Py], [BA5087; 2-Me-5-CH 2 CF _{3 -4-Py], [BA5088} ; 6-Me-5-CH 2 CF 3 -4-Py], [BA5089; 3-CF 3 -5-CH 2 CF 3 -4-Py], [BA5090; 2 _{-CF 3 -5-CH 2 CF 3} -4-Py], [BA5091; 6-CF 3 -5-CH 2 CF 3 -4-Py], [BA5092; 3-CN-5-CH 2 CF 3 - 4-Py], [BA5093; 2-CN-5-CH 2 CF 3 -4-Py], [BA5094; 6-CN-5-CH 2 CF 3 -4-Py], [BA5095; 3-OMe- _{5-CH 2 CF 3 -4-} Py], [BA5096; 2-OMe-5-CH 2 CF 3 -4-Py], [BA5097; 6-OMe-5-CH 2 CF 3 -4-Py], _{[BA5098; 6-CH 2 CF} 3 -4-Py], [BA5099; 3-Cl-6-CH 2 CF 3 -4-Py], [BA5100; 2-Cl-6-CH 2 CF 3 -4- Py], [BA5101; 5- Cl-6-CH 2 CF 3 -4-Py], [BA5102; 3-Me-6-CH 2 CF 3 -4-Py], [BA5103; 2-Me-6- _{CH 2 CF 3 -4-Py]} , [BA5104; 5-Me-6-CH 2 CF 3 -4-Py], [BA5105; 3-CF 3 -6-CH 2 CF 3 -4-Py], [ _{BA5106; 2-CF 3 -6-} CH 2 CF 3 -4-Py], [BA5107; 5-CF 3 -6-CH 2 CF 3 -4-Py], [BA5108; 3-CN-6-CH 2 _{CF 3 -4-Py], [} BA5109; 2-CN-6-CH 2 CF 3 -4-Py], [BA5110; 5-CN-6-CH 2 CF 3 -4-Py], [BA5111; 3 _{-OMe-6-CH 2 CF 3} -4-Py], [BA5112; 2-OMe-6-CH 2 CF 3 -4-Py], [BA5113; 5-OMe-6-CH 2 CF 3 -4- Py], [BA5114; 3-OEt-4-Py], [BA5115; 2-Cl-3-OEt-4-Py], [BA5116; 5-Cl-3-OEt-4-Py !, [BA5117; 6-Cl-3-OEt-4-Py], [BA5118; 2-Me-3-OEt-4-Py], [BA5119; 5- Me-3-OEt-4- Py], [BA5120; 6-Me-3-OEt-4-Py], [BA5121; 2-CF 3 -3-OEt-4-Py], [BA5122; 5-CF _{3 -3-OEt-4-Py} ], [BA5123; 6-CF 3 -3-OEt-4-Py], [BA5124; 2-CN-3-OEt-4-Py], [BA5125; 5-CN -3-OEt-4-Py !, [BA5126; 6-CN-3-OEt-4-Py], [BA5127; 2-OMe-3-OEt-4-Py], [BA5128; 5-OMe-3 -OEt-4-Py], [BA5129; 6-OMe-3-OEt-4-Py], [BA5130; 2-OEt-4-Py], [BA5131; 3-Cl-2-OEt-4-Py ], [BA5132; 5-Cl-2-OEt-4-Py], [BA5133; 6-Cl-2-OEt-4-Py], [BA5134; 3-Me-2-OEt-4-Py], [BA5135; 5-Me-2 -OEt-4-Py], [BA5136; 6-Me-2-OEt-4-Py], [BA5137; 3-CF 3 -2-OEt-4-Py], [ _{BA5138; 5-CF 3 -2-} OEt-4-Py], [BA5139; 6-CF 3 -2-OEt-4-Py], [BA5140; 3-CN-2-OEt-4-Py], [ BA5141; 5-CN-2-OEt-4-Py], [BA5142; 6-CN-2-OEt-4-Py], [BA5143; 3-OMe-2-OEt-4-Py], [BA5144; 5-OMe-2-OEt-4-Py !, [BA5145; 6-OMe-2-OEt-4-Py], [BA5146; 5-OEt-4-Py], [BA5147; 3-Cl-5- OEt-4-Py], [BA5148; 2-Cl-5-OEt-4-Py], [BA5149; 6-Cl-5-OEt-4-Py], [BA5150; 3-Me-5-OEt- 4-Py], [BA5151; 2-Me-5-OEt-4-Py], [BA5152; 6-Me-5-OEt-4-Py], [BA5153; 3-CF 3 -5-OEt-4 -Py], [BA5154; 2- CF 3 -5-OEt-4-Py], [BA5155; 6-CF _{3 -5-OEt-4-Py} ], [BA5156; 3-CN-5-OEt-4-Py], [BA5157; 2-CN-5-OEt-4-Py], [BA5158; 6-CN- 5-OEt-4-Py], [BA5159; 3-OMe-5-OEt-4-Py], [BA5160; 2-OMe-5-OEt-4-Py], [BA5161; 6-OMe-5- OEt-4-Py], [BA5162; 6-OEt-4-Py], [BA5163; 3-Cl-6-OEt-4-Py], [BA5164; 2-Cl-6-OEt-4-Py] , [BA5165; 5-Cl-6-OEt-4-Py], [BA5166; 3-Me-6-OEt-4-Py], [BA5167; 2-Me-6-OEt-4-Py], [BA5 165; BA5168; 5-Me-6- OEt-4-Py], [BA5169; 3-CF 3 -6-OEt-4-Py], [BA5170; 2-CF 3 -6-OEt-4-Py], [ BA 5171; 5-CF ₃ -6-OEt-4-Py], [BA5172; 3-CN-6-OEt-4-Py], [BA5173; 2-CN-6-OEt-4-Py], [BA5174] 5-CN-6-OEt-4-Py !, [BA5175; 3-OMe-6-OEt-4-Py], [BA5176; 2-OMe-6-OEt-4-Py], [BA5177; -OMe-6-OEt-4- Py], [BA5178; 3-OCH 2 CF 3 -4-Py], [BA5179; 2-Cl-3-OCH 2 CF 3 -4-Py], [BA5180; 5 _{-Cl-3-OCH 2 CF 3} -4-Py], [BA5181; 6-Cl-3-OCH 2 CF 3 -4-Py], [BA5182; 2-Me-3-OCH 2 CF 3 -4- Py], [BA5183; 5- Me-3-OCH 2 CF 3 -4-Py], [BA5184; 6-Me-3-OCH 2 CF 3 -4-Py],

[BA 5185; 2-CF ₃ -3-OCH ₂ CF ₃ -4-Py], [BA 5186; 5-CF ₃ -3-OCH ₂ CF ₃ -4-Py], [BA 5187; 6-CF ₃ -3- _{OCH 2 CF 3 -4-Py]} , [BA5188; 2-CN-3-OCH 2 CF 3 -4-Py], [BA5189; 5-CN-3-OCH 2 CF 3 -4-Py], [BA5190 ; 6-CN-3-OCH 2 CF 3 -4-Py], [BA5191; 2-OMe-3-OCH 2 CF 3 -4-Py], [BA5192; 5-OMe-3-OCH 2 CF 3 - 4-Py], [BA5193; 6-OMe-3-OCH 2 CF 3 -4-Py], [BA5194; 2-OCH 2 CF 3 -4-Py], [BA5195; 3-Cl-2-OCH 2 CF ₃ -4-Py !, [BA 5196; 5-Cl-2-OCH ₂ CF ₃ -4-Py], [BA 5197; 6-Cl-2-OCH ₂ CF ₃ -4-Py], [BA 5198; 3] _{-Me-2-OCH 2 CF 3} -4-Py], [BA5199; 5-Me-2-OCH 2 CF 3 -4-Py], [BA5200; 6-Me-2-OCH 2 CF 3 -4- Py], [BA5201; 3- CF 3 -2-OCH 2 CF 3 -4-Py], [BA5202; 5-CF 3 -2-OCH 2 CF 3 -4-Py], [BA5203; 6-CF 3 _{-2-OCH 2 CF 3 -4-} Py], [BA5204; 3-CN-2-OCH 2 CF 3 -4-Py], [BA5205; 5-CN-2-OCH 2 CF 3 -4-Py] , [BA5206; 6-CN- 2-OCH 2 CF 3 -4-Py], [BA5207; 3-OMe-2-OCH 2 CF 3 -4-Py], [BA5208; 5-OMe-2-OCH 2 _{CF 3 -4-Py], [} BA5209; 6-OMe-2-OCH 2 CF 3 -4-Py], [BA5210; 5-OCH 2 CF 3 -4-Py], [BA5211; 3-Cl-5 _{-OCH 2 CF 3 -4-Py]} , [BA5212; 2-Cl-5-OCH 2 CF 3 -4-Py], [BA5213; 6-Cl-5-OCH 2 CF 3 -4-Py], [ BA 5214; 3-Me-5-OCH ₂ CF ₃ -4- Py], [BA5215; 2- Me-5-OCH 2 CF 3 -4-Py], [BA5216; 6-Me-5-OCH 2 CF 3 -4-Py], [BA5217; 3-CF 3 -5 _{-OCH 2 CF 3 -4-Py]} , [BA5218; 2-CF 3 -5-OCH 2 CF 3 -4-Py], [BA5219; 6-CF 3 -5-OCH 2 CF 3 -4-Py] , [BA5220; 3-CN- 5-OCH 2 CF 3 -4-Py], [BA5221; 2-CN-5-OCH 2 CF 3 -4-Py], [BA5222; 6-CN-5-OCH 2 CF ₃ -4-Py], [BA 5223; 3-OMe-5-OCH ₂ CF ₃ -4-Py], [BA 5224; 2-OMe-5-OCH ₂ CF ₃ -4-Py], [BA 5225; 6 _{-OMe-5-OCH 2 CF 3} -4-Py], [BA5226; 6-OCH 2 CF 3 -4-Py], [BA5227; 3-Cl-6-OCH 2 CF 3 -4-Py], [ BA5228; 2-Cl-6- OCH 2 CF 3 -4-Py], [BA5229; 5-Cl-6-OCH 2 CF 3 -4-Py], [BA5230; 3-Me-6-OCH 2 CF 3 -4-Py], [BA5231; 2-Me-6-OCH 2 CF 3 -4-Py], [BA5232; 5-Me-6-OCH 2 CF 3 -4-Py], [BA5233; 3-CF _{3 -6-OCH 2 CF 3 -4} -Py], [BA5234; 2-CF 3 -6-OCH 2 CF 3 -4-Py], [BA5235; 5-CF 3 -6-OCH 2 CF 3 -4 -Py], [BA5236; 3- CN-6-OCH 2 CF 3 -4-Py], [BA5237; 2-CN-6-OCH 2 CF 3 -4-Py], [BA5238; 5-CN-6 _{-OCH 2 CF 3 -4-Py]} , [BA5239; 3-OMe-6-OCH 2 CF 3 -4-Py], [BA5240; 2-OMe-6-OCH 2 CF 3 -4-Py], [ BA5241; 5-OMe-6- OCH 2 CF 3 -4-Py], [BA5242; 3-Pr-4-Py], [BA5243; 2-Cl-3-Pr-4-Py], [BA5244; 5 -Cl-3-Pr-4-Py], [BA5245; 6-Cl-3-Pr-4 -Py], [BA5246; 2-Me-3-Pr-4-Py], [BA5247; 5-Me-3-Pr-4-Py], [BA5248; 6-Me-3-Pr-4-Py ], [BA5249; 2-CF 3 -3-Pr-4-Py], [BA5250; 5-CF 3 -3-Pr-4-Py], [BA5251; 6-CF 3 -3-Pr-4- Py], [BA5252; 2-CN-3-Pr-4-Py], [BA5253; 5-CN-3-Pr-4-Py], [BA5254; 6-CN-3-Pr-4-Py] , [BA5255; 2-OMe-3-Pr-4-Py], [BA5256; 5-OMe-3-Pr-4-Py], [BA5257; 6-OMe-3-Pr-4-Py], [BA5255; BA5258; 2-Pr-4-Py], [BA5259; 3-Cl-2-Pr-4-Py], [BA5260; 5-Cl-2-Pr-4-Py], [BA5261; 6-Cl- 2-Pr-4-Py], [BA5262; 3-Me-2-Pr-4-Py], [BA5263; 5-Me-2-Pr-4-Py], [BA5264; 6-Me-2- Pr-4-Py], [ BA5265; 3-CF 3 -2-Pr-4-Py], [BA5266; 5-CF 3 -2-Pr-4-Py], [BA5267; 6-CF 3 -2 -Pr-4-Py], [BA5268; 3-CN-2-Pr-4-Py], [BA5269; 5-CN-2-Pr-4-Py], [BA5270; 6-CN-2-Pr -4-Py !, [BA5271; 3-OMe-2-Pr-4-Py], [BA5272; 5-OMe-2-Pr-4-Py], [BA5273; 6-OMe-2-Pr-4 -Py], [BA5274; 5-Pr-4-Py], [BA5275; 3-Cl-5-Pr-4-Py], [BA5276; 2-Cl-5-Pr-4-Py], [BA5277 6-Cl-5-Pr-4-Py !, [BA5278; 3-Me-5-Pr-4-Py], [BA5279; 2-Me-5-Pr-4-Py], [BA5280; -Me-5-Pr-4- Py], [BA5281; 3-CF 3 -5-Pr-4-Py], [BA5282; 2-CF 3 -5-Pr-4-Py], [BA5283; 6 _{-CF 3 -5-Pr-4-} Py], [BA5284; 3-CN-5-Pr-4-Py],

[BA5285; 2-CN-5-Pr-4-Py], [BA5286; 6-CN-5-Pr-4-Py], [BA5287; 3-OMe-5-Pr-4-Py], [BA5288 2-OMe-5-Pr-4-Py !, [BA5289; 6-OMe-5-Pr-4-Py], [BA5290; 6-Pr-4-Py], [BA5291; 3-Cl-6 -Pr-4-Py], [BA5292; 2-Cl-6-Pr-4-Py], [BA5293; 5-Cl-6-Pr-4-Py], [BA5294; 3-Me-6-Pr -4-Py], [BA5295; 2-Me-6-Pr-4-Py], [BA5296; 5-Me-6-Pr-4-Py], [BA5297; 3-CF 3 -6-Pr- 4-Py], [BA5298; 2-CF 3 -6-Pr-4-Py], [BA5299; 5-CF 3 -6-Pr-4-Py], [BA5300; 3-CN-6-Pr- 4-Py], [BA5301; 2-CN-6-Pr-4-Py], [BA5302; 5-CN-6-Pr-4-Py], [BA5303; 3-OMe-6-Pr-4- Py], [BA5304; 2-OMe-6-Pr-4-Py], [BA5305; 5-OMe-6-Pr-4-Py], [BA5306; 3-OPr-4-Py], [BA5307; 2-Cl-3-OPr-4-Py !, [BA5308; 5-Cl-3-OPr-4-Py], [BA5309; 6-Cl-3-OPr-4-Py], [BA5310; Me-3-OPr-4- Py], [BA5311; 5-Me-3-OPr-4-Py], [BA5312; 6-Me-3-OPr-4-Py], [BA5313; 2-CF 3 -3-OPr-4-Py] , [BA5314; 5-CF 3 -3-OPr-4-Py], [BA5315; 6-CF 3 -3-OPr-4-Py], [BA5316; 2-CN -3-OPr-4-Py !, [BA5317; 5-CN-3-OPr-4-Py], [BA5318; 6-CN-3-OPr-4-Py], [BA5319; 2-OMe-3 -OPr-4-Py], [BA5320; 5-OMe-3-OPr-4-Py], [BA5321; 6-OMe-3-OPr-4-Py], [BA5322; 2-OPr-4-Py ], [BA5323; 3-Cl-2-OPr-4-Py], [BA5324; 5-Cl-2-OPr-4-Py], [BA5325; 6] -Cl-2-OPr-4-Py], [BA5326; 3-Me-2-OPr-4-Py], [BA5327; 5-Me-2-OPr-4-Py], [BA5328; 6-Me -2-OPr-4-Py] , [BA5329; 3-CF 3 -2-OPr-4-Py], [BA5330; 5-CF 3 -2-OPr-4-Py], [BA5331; 6-CF _3- 2-OPr-4-Py, [BA5332; 3-CN-2-OPr-4-Py], [BA5333; 5-CN-2-OPr-4-Py], [BA5334; 6-CN- 2-OPr-4-Py], [BA5335; 3-OMe-2-OPr-4-Py], [BA5336; 5-OMe-2-OPr-4-Py], [BA5337; 6-OMe-2- OPr-4-Py], [BA5338; 5-OPr-4-Py], [BA5339; 3-Cl-5-OPr-4-Py], [BA5340; 2-Cl-5-OPr-4-Py] , [BA5341; 6-Cl-5-OPr-4-Py], [BA5342; 3-Me-5-OPr-4-Py], [BA5343; 2-Me-5-OPr-4-Py], [BA5342; BA5344; 6-Me-5- OPr-4-Py], [BA5345; 3-CF 3 -5-OPr-4-Py], [BA5346; 2-CF 3 -5-OPr-4-Py], [ _{BA5347; 6-CF 3 -5-} OPr-4-Py], [BA5348; 3-CN-5-OPr-4-Py], [BA5349; 2-CN-5-OPr-4-Py], [BA5350 6-CN-5-OPr-4-Py !, [BA5351; 3-OMe-5-OPr-4-Py], [BA5352; 2-OMe-5-OPr-4-Py], [BA5353; -OMe-5-OPr-4-Py], [BA 5354; 6-OPr-4-Py], [BA 5355; 3-Cl-6-OPr-4-Py], [BA 5356; 2-Cl-6-OPr -4-Py !, [BA5357; 5-Cl-6-OPr-4-Py], [BA5358; 3-Me-6-OPr-4-Py], [BA5359; 2-Me-6-OPr-4 -Py], [BA5360; 5- Me-6-OPr-4-Py], [BA5361; 3-CF 3 -6-OPr-4-Py], [BA5362; 2-CF 3 -6-OPr-4 -Py], [BA5363; 5- CF 3 -6-OPr-4-Py], [BA5364; 3-C N-6-OPr-4-Py], [BA5365; 2-CN-6-OPr-4-Py], [BA5366; 5-CN-6-OPr-4-Py], [BA5367; 3-OMe- 6-OPr-4-Py], [BA5368; 2-OMe-6-OPr-4-Py], [BA5369; 5-OMe-6-OPr-4-Py], [BA5370; 3-SMe-4- Py], [BA5371; 2-Cl-3-SMe-4-Py], [BA5372; 5-Cl-3-SMe-4-Py], [BA5373; 6-Cl-3-SMe-4-Py] , [BA5374; 2-Me-3-SMe-4-Py], [BA5375; 5-Me-3-SMe-4-Py], [BA5376; 6-Me-3-SMe-4-Py], [BA-5376; _{BA5377; 2-CF 3 -3-} SMe-4-Py], [BA5378; 5-CF 3 -3-SMe-4-Py], [BA5379; 6-CF 3 -3-SMe-4-Py], [BA5380; 2-CN-3-SMe-4-Py], [BA5381; 5-CN-3-SMe-4-Py], [BA5382; 6-CN-3-SMe-4-Py], [BA5383 2-OMe-3-SMe-4-Py !, [BA5384; 5-OMe-3-SMe-4-Py],

[BA5385; 6-OMe-3-SMe-4-Py], [BA5386; 2-SMe-4-Py], [BA5387; 3-Cl-2-SMe-4-Py], [BA5388; -2-SMe-4-Py !, [BA5389; 6-Cl-2-SMe-4-Py], [BA5390; 3-Me-2-SMe-4-Py], [BA5391; 5-Me-2 -SMe-4-Py], [ BA5392; 6-Me-2-SMe-4-Py], [BA5393; 3-CF 3 -2-SMe-4-Py], [BA5394; 5-CF 3 -2 -SMe-4-Py], [ BA5395; 6-CF 3 -2-SMe-4-Py], [BA5396; 3-CN-2-SMe-4-Py], [BA5397; 5-CN-2- SMe-4-Py !, [BA5398; 6-CN-2-SMe-4-Py], [BA5399; 3-OMe-2-SMe-4-Py], [BA5400; 5-OMe-2-SMe- 4-Py], [BA5401; 6-OMe-2-SMe-4-Py], [BA5402; 5-SMe-4-Py], [BA5403; 3-Cl-5-SMe-4-Py], [BA5403; BA5404; 2-Cl-5-SMe-4-Py], [BA5405; 6-Cl-5-SMe-4-Py], [BA5406; 3-Me-5-SMe-4-Py], [BA5407; 2-Me-5-SMe- 4-Py], [BA5408; 6-Me-5-SMe-4-Py], [BA5409; 3-CF 3 -5-SMe-4-Py], [BA5410; 2 _{-CF 3 -5-SMe-4-} Py], [BA5411; 6-CF 3 -5-SMe-4-Py], [BA5412; 3-CN-5-SMe-4-Py], [BA5413; 2 -CN-5-SMe-4-Py], [BA5414; 6-CN-5-SMe-4-Py], [BA5415; 3-OMe-5-SMe-4-Py], [BA5416; 2-OMe -5-SMe-4-Py !, [BA5417; 6-OMe-5-SMe-4-Py], [BA5418; 6-SMe-4-Py], [BA5419; 3-Cl-6-SMe-4 -Py], [BA5420; 2-Cl-6-SMe-4-Py], [BA5421; 5-Cl-6-SMe-4-Py], [BA5422; 3-Me-6-SMe-4-Py ], [BA 5423; 2-Me-6-SMe-4-Py], [BA 5424; 5-Me-6- SMe-4-Py], [ BA5425; 3-CF 3 -6-SMe-4-Py], [BA5426; 2-CF 3 -6-SMe-4-Py], [BA5427; 5-CF 3 -6 -SMe-4-Py], [BA5428; 3-CN-6-SMe-4-Py], [BA5429; 2-CN-6-SMe-4-Py], [BA5430; 5-CN-6-SMe -4-Py], [BA5431; 3-OMe-6-SMe-4-Py], [BA5432; 2-OMe-6-SMe-4-Py], [BA5433; 5-OMe-6-SMe-4 -Py], [BA 5434; 3-SCF ₃ -4-Py], [BA 5435; 2-Cl-3-SCF ₃ -4-Py], [BA 5436; 5-Cl-3-SCF ₃ -4-Py] , [BA5437; 6-Cl- 3-SCF 3 -4-Py], [BA5438; 2-Me-3-SCF 3 -4-Py], [BA5439; 5-Me-3-SCF 3 -4-Py ], [BA5440; 6-Me -3-SCF 3 -4-Py], [BA5441; 2-CF 3 -3-SCF 3 -4-Py], [BA5442; 5-CF 3 -3-SCF 3 - 4-Py], [BA5443; 6-CF 3 -3-SCF 3 -4-Py], [BA5444; 2-CN-3-SCF 3 -4-Py], [BA5445; 5-CN-3-SCF ₆ -4-Py !, [BA5446; 6-CN-3-SCF ₃ -4-Py], [BA 5447; 2-OMe-3-SCF ₃ -4-Py], [BA 5448; 5-OMe -3- SCF ₃ -4-Py !, [BA 5449; 6-OMe -3-SCF ₃ -4-Py], [BA 5450; 2-SCF ₃ -4-Py], [BA 5451; 3-Cl-2-SCF _3- 4-Py], [BA5452; 5-Cl-2-SCF 3 -4-Py], [BA5453; 6-Cl-2-SCF 3 -4-Py], [BA5454; 3-Me-2-SCF 3 -4-Py], [BA5455; 5-Me-2-SCF 3 -4-Py], [BA5456; 6-Me-2-SCF 3 -4-Py], [BA5457; 3-CF 3 -2- SCF ₃ -4-Py !, [BA5458; 5-CF ₃ -2-SCF ₃ -4-Py], [BA 5459; 6-CF ₃ -2-SCF ₃ -4-Py], [BA 5460; 3-CN] -2 -SCF ₃ -4-Py !, [BA5461; 5-CN-2-SCF ₃ -4-Py], [BA5462; 6-CN-2-SCF ₃ -4-Py], [BA5463; 3-OMe- _{2-SCF 3 -4-Py]} , [BA5464; 5-OMe-2-SCF 3 -4-Py], [BA5465; 6-OMe-2-SCF 3 -4-Py], [BA5466; 5-SCF ₃ -4-Py !, [BA 5467; 3-Cl-5-SCF ₃ -4-Py], [BA 5468; 2-Cl-5-SCF ₃ -4-Py], [BA 5469; 6-Cl-5- SCF ₃ -4-Py !, [BA 5470; 3-Me-5-SCF ₃ -4-Py], [BA 5471; 2-Me-5-SCF ₃ -4-Py], [BA 5472; 6-Me-5 -SCF ₃ -4-Py], [BA 5473; 3-CF ₃ -5-SCF ₃ -4-Py], [BA 5474; 2-CF ₃ -5-SCF ₃ -4-Py], [BA 5475; 6- _{CF 3 -5-SCF 3 -4-} Py], [BA5476; 3-CN-5-SCF 3 -4-Py], [BA5477; 2-CN-5-SCF 3 -4-Py], [BA5478; 6-CN-5-SCF ₃ -4-Py !, [BA5479; 3-OMe-5-SCF ₃ -4-Py], [BA 5480; 2-OMe-5-SCF ₃ -4-Py], [BA5481] ; 6-OMe-5-SCF 3 -4-Py], [BA5482; 6-SCF 3 -4-Py], [BA5483; 3-Cl-6-SCF 3 -4-Py], [BA5484; 2- Cl-6-SCF ₃ -4-Py],

[BA5485; 6-Cl-6-SCF ₃ -4-Py], [BA 5486; 3-Me-6-SCF ₃ -4-Py], [BA 5487; 2-Me-6-SCF ₃ -4-Py] , [BA5488; 6-Me- 6-SCF 3 -4-Py], [BA5489; 3-CF 3 -6-SCF 3 -4-Py], [BA5490; 2-CF 3 -6-SCF 3 -4 -Py], [BA5491; 6- CF 3 -6-SCF 3 -4-Py], [BA5492; 3-CN-6-SCF 3 -4-Py], [BA5493; 2-CN-6-SCF 3 -4-Py], [BA5494; 6-CN-6-SCF 3 -4-Py], [BA5495; 3-OMe-6-SCF 3 -4-Py], [BA5496; 2-OMe-6-SCF ₃ -4-Py !, [BA5497; 6-OMe-6-SCF ₃ -4-Py], [BA 5498; 3-S (O) Me-4-Py], [BA5499; 2-Cl-3-S (O) Me-4-Py], [BA5500; 5-Cl-3-S (O) Me-4-Py], [BA5501; 6-Cl-3-S (O) Me-4-Py], [BA5502; 2-Me-3-S (O) Me-4-Py], [BA5503; 5-Me-3-S (O) Me-4-Py], [BA5504; 6-Me-3-S (O) Me-4-Py ], [BA5505; 2-CF 3 -3-S (O) Me-4-Py], [BA5506; 5-CF 3 -3-S (O) Me-4-Py ], [BA5507; 6-CF 3 -3-S (O) Me-4-Py], [BA5508; 2-CN-3-S (O) Me-4-Py], [BA5509; 5-CN- 3-S (O) Me-4-Py], [BA5510; 6-CN-3-S (O) Me-4-Py], [BA5511; 2-OMe-3-S (O) Me-4- 4 Py], [BA5512; 5-OMe-3-S (O) Me-4-Py], [BA5513; 6-OMe-3-S (O) Me-4-Py], [BA5514; O) Me-4-Py], [BA5515; 3-Cl-2-S (O) Me-4-Py], [BA5516; 5-Cl-2-S (O) Me-4-Py], [BA5516; BA 5517; 6-Cl-2-S (O) Me-4-Py], [BA5518; 3-Me-2-S (O) Me-4-Py], [BA5519; 5-Me-2-S ( O) Me-4-Py], [BA 552 0; 6-Me-2- S (O) Me-4-Py], [BA5521; 3-CF 3 -2-S (O) Me-4-Py], [BA5522; 5-CF 3 -2- S (O) Me-4- Py], [BA5523; 6-CF 3 -2-S (O) Me-4-Py], [BA5524; 3-CN-2-S (O) Me-4-Py ], [BA5525; 5-CN-2-S (O) Me-4-Py], [BA5526; 6-CN-2-S (O) Me-4-Py], [BA5527; 3-OMe-2 -S (O) Me-4-Py], [BA5528; 5-OMe-2-S (O) Me-4-Py], [BA5529; 6-OMe-2-S (O) Me-4-Py ], [BA5530; 5-S (O) Me-4-Py], [BA5531; 3-Cl-5-S (O) Me-4-Py], [BA5532; 2-Cl-5-S (O) ) Me-4-Py], [BA5533; 6-Cl-5-S (O) Me-4-Py], [BA5534; 3-Me-5-S (O) Me-4-Py], [BA5535] ; 2-Me-5-S (O) Me-4-Py], [BA5536; 6-Me-5-S (O) Me-4-Py], [BA5537; 3-CF 3 -5-S ( O) Me-4-Py] , [BA5538; 2-CF 3 -5-S (O) Me-4-Py], [BA5539; 6-CF 3 -5-S (O) Me-4-Py] , [BA5540; 3-CN-5-S (O) Me-4-Py], [BA5541; 2-CN-5-S (O) Me-4-Py], [BA5542; 6-CN-5- S (O) Me-4-Py], [BA5543; 3-OMe-5-S (O) Me-4-Py], [BA5544; 2-OMe-5-S (O) Me-4-Py] , [BA5545; 6-OMe-5-S (O) Me-4-Py], [BA5546; 6-S (O) Me-4-Py], [BA5547; 3-Cl-6-S (O) Me-4-Py !, [BA5548; 2-Cl-6-S (O) Me-4-Py], [BA5549; 5-Cl-6-S (O) Me-4-Py], [BA5550; 3-Me-6-S (O) Me-4-Py], [BA5551; 2-Me-6-S (O) Me-4-Py], [BA5552; 5-Me-6-S (O) Me-4-Py], [ BA5553; 3-CF 3 -6-S (O) Me-4-Py], [BA5554; 2-CF 3 -6-S (O) Me-4-Py], [ BA 555 _{5; 5-CF 3 -6-} S (O) Me-4-Py], [BA5556; 3-CN-6-S (O) Me-4-Py], [BA5557; 2-CN-6-S (O) Me-4-Py], [BA5558; 5-CN-6-S (O) Me-4-Py], [BA5559; 3-OMe-6-S (O) Me-4-Py], [BA5560; 2-OMe-6-S (O) Me-4-Py], [BA5561; 5-OMe-6-S (O) Me-4-Py], [BA5562; 3-S (O) CF ₃ -4-Py !, [BA5563; 2-Cl-3-S (O) CF ₃ -4-Py], [BA5564; 5-Cl-3-S (O) CF ₃ -4-Py], BA5565; 6-Cl-3- S (O) CF 3 -4-Py], [BA5566; 2-Me-3-S (O) CF 3 -4-Py], [BA5567; 5-Me-3- _{S (O) CF 3 -4-} Py], [BA5568; 6-Me-3-S (O) CF 3 -4-Py], [BA5569; 2-CF 3 -3-S (O) CF 3 - 4-Py], [BA5570; 5-CF 3 -3-S (O) CF 3 -4-Py], [BA5571; 6-CF 3 -3-S (O) CF 3 -4-Py], [ BA5572; 2-CN-3- S (O) CF 3 -4-Py], [BA5573; 5-CN-3-S (O) CF 3 -4-Py], [BA5574; 6-CN-3- _{S (O) CF 3 -4-} Py], [BA5575; 2-OMe-3-S (O) CF 3 -4-Py], [BA5576; 5-OMe-3-S (O) CF 3 -4 -Py], [BA5577; 6- OMe-3-S (O) CF 3 -4-Py], [BA5578; 2-S (O) CF 3 -4-Py], [BA5579; 3-Cl-2 _{-S (O) CF 3 -4-} Py], [BA5580; 5-Cl-2-S (O) CF 3 -4-Py], [BA5581; 6-Cl-2-S (O) CF 3 - 4-Py], [BA5582; 3-Me-2-S (O) CF 3 -4-Py], [BA5583; 5-Me-2-S (O) CF 3 -4-Py], [BA5584; 6-Me-2-S ( O) CF 3 -4-Py],

[BA 5585; 3-CF ₃ -2-S (O) CF ₃ -4-Py], [BA 5586; 5-CF ₃ -2-S (O) CF ₃ -4-Py], [BA 5587; 6-CF _{3 -2-S (O) CF} 3 -4-Py], [BA5588; 3-CN-2-S (O) CF 3 -4-Py], [BA5589; 5-CN-2-S (O) _{CF 3 -4-Py], [} BA5590; 6-CN-2-S (O) CF 3 -4-Py], [BA5591; 3-OMe-2-S (O) CF 3 -4-Py], [BA5592; 5-OMe-2 -S (O) CF 3 -4-Py], [BA5593; 6-OMe-2-S (O) CF 3 -4-Py], [BA5594; 5-S (O ) CF ₃ -4-Py !, [BA 5595; 3-Cl-5-S (O) CF ₃ -4-Py], [BA5596; 2-Cl-5-S (O) CF ₃ -4-Py] , [BA5597; 6-Cl- 5-S (O) CF 3 -4-Py], [BA5598; 3-Me-5-S (O) CF 3 -4-Py], [BA5599; 2-Me- _{5-S (O) CF 3} -4-Py], [BA5600; 6-Me-5-S (O) CF 3 -4-Py], [BA5601; 3-CF 3 -5-S (O) CF ₃ -4-Py !, [BA5602; 2-CF ₃ -5-S (O) CF ₃ -4-Py], [BA 5603; 6-CF ₃ -5-S (O) CF ₃ -4-Py] , [BA5604; 3-CN- 5-S (O) CF 3 -4-Py], [BA5605; 2-CN-5-S (O) CF 3 -4-Py], [BA5606; 6-CN- _{5-S (O) CF 3} -4-Py], [BA5607; 3-OMe-5-S (O) CF 3 -4-Py], [BA5608; 2-OMe-5-S (O) CF 3 -4-Py], [BA5609; 6-OMe-5-S (O) CF 3 -4-Py], [BA5610; 6-S (O) CF 3 -4-Py], [BA5611; 3-Cl _{-6-S (O) CF 3} -4-Py], [BA5612; 2-Cl-6-S (O) CF 3 -4-Py], [BA5613; 5-Cl-6-S (O) CF _{3 -4-Py], [BA5614} ; 3-Me-6-S (O) CF 3 -4-Py], [BA5615; 2-Me-6-S (O) CF 3 -4-Py], [ BA 5616; 5-Me-6-S (O) CF _3- 4-Py], [BA 5617; 3-CF ₃ -6-S (O) CF ₃ -4-Py], [BA 5618; 2-CF ₃ -6-S (O) CF ₃ -4-Py], [4 _{BA5619; 5-CF 3 -6-} S (O) CF 3 -4-Py], [BA5620; 3-CN-6-S (O) CF 3 -4-Py], [BA5621; 2-CN-6 _{-S (O) CF 3 -4-} Py], [BA5622; 5-CN-6-S (O) CF 3 -4-Py], [BA5623; 3-OMe-6-S (O) CF 3 - 4-Py], [BA5624; 2-OMe-6-S (O) CF 3 -4-Py], [BA5625; 5-OMe-6-S (O) CF 3 -4-Py], [BA5626; _{3-S (O) 2 Me} -4-Py], [BA5627; 2-Cl-3-S (O) 2 Me-4-Py], [BA5628; 5-Cl-3-S (O) 2 Me -4-Py], [BA5629; 6-Cl-3-S (O) 2 Me-4-Py], [BA5630; 2-Me-3-S (O) 2 Me-4-Py], [BA5631 ; 5-Me-3-S (O) 2 Me-4-Py], [BA5632; 6-Me-3-S (O) 2 Me-4-Py], [BA5633; 2-CF 3 -3- _{S (O) 2 Me-4} -Py], [BA5634; 5-CF 3 -3-S (O) 2 Me-4-Py], [BA5635; 6-CF 3 -3-S (O) 2 Me -4-Py !, [BA5636; 2-CN-3-S (O) ₂ Me-4-Py], [BA5637; 5-CN-3-S (O) ₂ Me-4-Py], [BA5638] ; 6-CN-3-S (O) 2 Me-4-Py], [BA5639; 2-OMe-3-S (O) 2 Me-4-Py], [BA5640; 5-OMe-3-S (O) ₂ Me-4-Py], [BA5641; 6-OMe-3-S (O) ₂ Me-4-Py], [BA5642; 2-S (O) ₂ Me-4-Py], BA5643; 3-Cl-2- S (O) 2 Me-4-Py], [BA5644; 5-Cl-2-S (O) 2 Me-4-Py], [BA5645; 6-Cl-2- _{S (O) 2 Me-4} -Py], [BA5646; 3-Me-2-S (O) 2 Me-4-Py], [BA5647; 5-Me-2-S (O) 2 Me-4 -Py], [BA 5648; 6-Me-2-S (O) _{2 Me-4-Py],} [BA5649; 3-CF 3 -2-S (O) 2 Me-4-Py], [BA5650; 5-CF 3 -2-S (O) 2 Me-4-Py ], [BA5651; 6-CF 3 -2-S (O) 2 Me-4-Py], [BA5652; 3-CN-2-S (O) 2 Me-4-Py], [BA5653; 5- CN-2-S (O) 2 Me-4-Py], [BA5654; 6-CN-2-S (O) 2 Me-4-Py], [BA5655; 3-OMe-2-S (O) ₂ Me-4-Py !, [BA5656; 5-OMe-2-S (O) ₂ Me-4-Py], [BA5657; 6-OMe-2-S (O) ₂ Me-4-Py], [BA5658; 5-S (O) ₂ Me-4-Py], [BA5659; 3-Cl-5-S (O) ₂ Me-4-Py], [BA 5660; 2-Cl-5-S (O ) ₂ Me-4-Py], [BA5661; 6-Cl-5-S (O) ₂ Me-4-Py], [BA5662; 3-Me-5-S (O) ₂ Me-4-Py] , [BA5663; 2-Me- 5-S (O) 2 Me-4-Py], [BA5664; 6-Me-5-S (O) 2 Me-4-Py], [BA5665; 3-CF 3 _{-5-S (O) 2 Me} -4-Py], [BA5666; 2-CF 3 -5-S (O) 2 Me-4-Py], [BA5667; 6-CF 3 -5-S (O ) ₂ Me-4-Py], [BA5668; 3-CN-5-S (O) ₂ Me-4-Py], [BA5669; 2-CN-5-S (O) ₂ Me-4-Py] , [BA 5670; 6-CN-5-S (O) ₂ Me-4-Py], [BA 5671; 3-OMe-5-S (O) ₂ Me-4-Py], [BA 5672; 2-OMe- _{5-S (O) 2 Me} -4-Py], [BA5673; 6-OMe-5-S (O) 2 Me-4-Py], [BA5674; 6-S (O) 2 Me-4-Py ], [BA 5675; 3-Cl-6-S (O) ₂ Me-4-Py], [BA 5676; 2-Cl-6-S (O) ₂ Me-4-Py], [BA 5677; 5-Cl] _{-6-S (O) 2 Me} -4-Py], [BA5678; 3-Me-6-S (O) 2 Me-4-Py], [BA5679; 2-Me-6-S (O) 2 Me-4-Py], [BA5680; 5-Me- _{6-S (O) 2 Me} -4-Py], [BA5681; 3-CF 3 -6-S (O) 2 Me-4-Py], [BA5682; 2-CF 3 -6-S (O) _{2 Me-4-Py],} [BA5683; 5-CF 3 -6-S (O) 2 Me-4-Py], [BA5684; 3-CN-6-S (O) 2 Me-4-Py] ,

[BA5685; 2-CN-6 -S (O) 2 Me-4-Py], [BA5686; 5-CN-6-S (O) 2 Me-4-Py], [BA5687; 3-OMe-6 _{-S (O) 2 Me-4} -Py], [BA5688; 2-OMe-6-S (O) 2 Me-4-Py], [BA5689; 5-OMe-6-S (O) 2 Me- 4-Py], [BA5690; 3-S (O) 2 CF 3 -4-Py], [BA5691; 2-Cl-3-S (O) 2 CF 3 -4-Py], [BA5692; 5- Cl-3-S (O) 2 CF 3 -4-Py], [BA5693; 6-Cl-3-S (O) 2 CF 3 -4-Py], [BA5694; 2-Me-3-S ( O) ₂ CF ₃ -4-Py], [BA 5 695; 5-Me-3-S (O) ₂ CF ₃ -4-Py], [BA 5 696; 6-Me-3-S (O) ₂ CF _3- 4-Py], [BA5697; 2-CF 3 -3-S (O) 2 CF 3 -4-Py], [BA5698; 5-CF 3 -3-S (O) 2 CF 3 -4-Py] _{, [BA5699; 6-CF 3} -3-S (O) 2 CF 3 -4-Py], [BA5700; 2-CN-3-S (O) 2 CF 3 -4-Py], [BA5701; 5 -CN-3-S (O) 2 CF 3 -4-Py], [BA5702; 6-CN-3-S (O) 2 CF 3 -4-Py], [BA5703; 2-OMe-3-S _{(O) 2 CF 3 -4-} Py], [BA5704; 5-OMe-3-S (O) 2 CF 3 -4-Py], [BA5705; 6-OMe-3-S (O) 2 CF 3 -4-Py], [BA5706; 2-S (O) 2 CF 3 -4-Py], [BA5707; 3-Cl-2-S (O) 2 CF 3 -4-Py], [BA5708; 5 -Cl-2-S (O) 2 CF 3 -4-Py], [BA5709; 6-Cl-2-S (O) 2 CF 3 -4-Py], [BA5710; 3-Me-2-S _{(O) 2 CF 3 -4-} Py], [BA5711; 5-Me-2-S (O) 2 CF 3 -4-Py], [BA5712; 6-Me-2-S (O) 2 CF 3 -4-Py], [BA 5713; 3-CF ₃ -2-S (O) ₂ CF ₃ -4-Py], [BA 5714; 5-CF ₃ -2-S (O _{) 2 CF 3 -4-Py]} , [BA5715; 6-CF 3 -2-S (O) 2 CF 3 -4-Py], [BA5716; 3-CN-2-S (O) 2 CF 3 - 4-Py], [BA5717; 5-CN-2-S (O) 2 CF 3 -4-Py], [BA5718; 6-CN-2-S (O) 2 CF 3 -4-Py], [ BA5719; 3-OMe-2- S (O) 2 CF 3 -4-Py], [BA5720; 5-OMe-2-S (O) 2 CF 3 -4-Py], [BA5721; 6-OMe- _{2-S (O) 2 CF} 3 -4-Py], [BA5722; 5-S (O) 2 CF 3 -4-Py], [BA5723; 3-Cl-5-S (O) 2 CF 3 - 4-Py], [BA5724; 2-Cl-5-S (O) 2 CF 3 -4-Py], [BA5725; 6-Cl-5-S (O) 2 CF 3 -4-Py], [ BA5726; 3-Me-5- S (O) 2 CF 3 -4-Py], [BA5727; 2-Me-5-S (O) 2 CF 3 -4-Py], [BA5728; 6-Me- _{5-S (O) 2 CF} 3 -4-Py], [BA5729; 3-CF 3 -5-S (O) 2 CF 3 -4-Py], [BA5730; 2-CF 3 -5-S ( O) ₂ CF ₃ -4-Py], [BA 5731; 6-CF ₃ -5-S (O) ₂ CF ₃ -4-Py], [BA 573 2; 3-CN-5-S (O) ₂ CF ₃ -4-Py], [BA5733; 2-CN-5-S (O) 2 CF 3 -4-Py], [BA5734; 6-CN-5-S (O) 2 CF 3 -4-Py], [BA5735; 3-OMe-5 -S (O) 2 CF 3 -4-Py], [BA5736; 2-OMe-5-S (O) 2 CF 3 -4-Py], [BA5737; 6-OMe _{-5-S (O) 2 CF} 3 -4-Py], [BA5738; 6-S (O) 2 CF 3 -4-Py], [BA5739; 3-Cl-6-S (O) 2 CF 3 -4-Py], [BA5740; 2-Cl-6-S (O) 2 CF 3 -4-Py], [BA5741; 5-Cl-6-S (O) 2 CF 3 -4-Py], [BA5742; 3-Me-6 -S (O) 2 CF 3 -4-Py], [BA5743; 2-Me-6-S (O) 2 CF ₃ -4-Py !, [BA 5744; 5-Me-6-S (O) ₂ CF ₃ -4-Py], [BA 5745; 3-CF ₃ -6-S (O) ₂ CF ₃ -4-Py ], [BA5746; 2-CF 3 -6-S (O) 2 CF 3 -4-Py], [BA5747; 5-CF 3 -6-S (O) 2 CF 3 -4-Py], [BA5748 ; 3-CN-6-S (O) 2 CF 3 -4-Py], [BA5749; 2-CN-6-S (O) 2 CF 3 -4-Py], [BA5750; 5-CN-6 _{-S (O) 2 CF 3 -4} -Py], [BA5751; 3-OMe-6-S (O) 2 CF 3 -4-Py], [BA5752; 2-OMe-6-S (O) 2 _{CF 3 -4-Py], [} BA5753; 5-OMe-6-S (O) 2 CF 3 -4-Py], [BA5754; 3-CN-4-Py], [BA5755; 2-Cl-3 -CN-4-Py], [BA5756; 5-Cl-3-CN-4-Py], [BA5757; 6-Cl-3-CN-4-Py], [BA5758; 2-Me-3-CN -4-Py], [BA5759; 5-Me-3-CN-4-Py], [BA5760; 6-Me-3-CN-4-Py], [BA5761; 2-CF 3 -3-CN- 4-Py], [BA5762; 5-CF 3 -3-CN-4-Py], [BA5763; 6-CF 3 -3-CN-4-Py], [BA5764; 2-CN-3-CN- 4-Py], [BA5765; 5-CN-3-CN-4-Py], [BA5766; 6-CN-3-CN-4-Py], [BA5767; 2-OMe-3-CN-4-] Py], [BA5768; 5-OMe-3-CN-4-Py], [BA5769; 6-OMe-3-CN-4-Py], [BA5770; 2-CN-4-Py], [BA5771; 3-Cl-2-CN-4-Py !, [BA 5772; 5-Cl-2-CN-4-Py], [BA 5773; 6-Cl-2-CN-4-Py], [BA 5774; Me-2-CN-4- Py], [BA5775; 5-Me-2-CN-4-Py], [BA5776; 6-Me-2-CN-4-Py], [BA5777; 3-CF 3 -2-CN-4-Py !, [BA 5778; 5-CF ₃ -2-CN-4-Py], [BA 5779; 6-CF ₃ 2-CN-4-Py], [BA 5780; 3-CN-2-CN-4-Py !, [BA5781; 5-CN-2-CN-4-Py], [BA5782; 6-CN-2-CN-4-Py], [BA5783; 3-OMe-2-CN-4-Py], [BA5784; 5-OMe-2-CN-4-Py],

[BA 5785; 6-OMe-2-CN-4-Py], [BA 5786; 5-CN-4-Py], [BA 5787; 3-Cl-5-CN-4-Py], [BA 5788; 2-Cl -5-CN-4-Py !, [BA5789; 6-Cl-5-CN-4-Py], [BA5790; 3-Me-5-CN-4-Py], [BA5791; 2-Me-5 -CN-4-Py], [ BA5792; 6-Me-5-CN-4-Py], [BA5793; 3-CF 3 -5-CN-4-Py], [BA5794; 2-CF 3 -5 -CN-4-Py], [ BA5795; 6-CF 3 -5-CN-4-Py], [BA5796; 3-CN-5-CN-4-Py], [BA5797; 2-CN-5- CN-4-Py], [BA5798; 6-CN-5-CN-4-Py], [BA5799; 3-OMe-5-CN-4-Py], [BA5800; 2-OMe-5-CN- 4-Py], [BA5801; 6-OMe-5-CN-4-Py], [BA5802; 6-CN-4-Py], [BA5803; 3-Cl-6-CN-4-Py], [BA-580] BA5804; 2-Cl-6-CN-4-Py], [BA5805; 5-Cl-6-CN-4-Py], [BA5806; 3-Me-6-CN-4-Py], [BA5807; 2-Me-6-CN- 4-Py], [BA5808; 5-Me-6-CN-4-Py], [BA5809; 3-CF 3 -6-CN-4-Py], [BA5810; 2 _{-CF 3 -6-CN-4-} Py], [BA5811; 5-CF 3 -6-CN-4-Py], [BA5812; 3-CN-6-CN-4-Py], [BA5813; 2 -CN-6-CN-4-Py], [BA5814; 5-CN-6-CN-4-Py], [BA5815; 3-OMe-6-CN-4-Py], [BA5816; 2-OMe -6-CN-4-Py !, [BA5817; 5-OMe-6-CN-4-Py], [BA5818; 3-COOMe-4-Py], [BA5819; 2-Cl-3-COOMe-4 -Py], [BA5820; 5-Cl-3-COOMe-4-Py], [BA5821; 6-Cl-3-COOMe-4-Py], [BA5822; 2-Me-3-COOMe-4-Py ], [BA 5823; 5-Me-3-COOMe-4-Py], [BA 5824; 6-Me-3-COOMe-4-Py], [BA 5825; 2] _{-CF 3 -3-COOMe-4-} Py], [BA5826; 5-CF 3 -3-COOMe-4-Py], [BA5827; 6-CF 3 -3-COOMe-4-Py], [BA5828; 2-CN-3-COOMe-4-Py !, [BA5829; 5-CN-3-COOMe-4-Py], [BA5830; 6-CN-3-COOMe-4-Py], [BA5831; OMe-3-COOMe-4-Py], [BA5832; 5-OMe-3-COOMe-4-Py], [BA5833; 6-OMe-3-COOMe-4-Py], [BA5834; 2-COOMe- 4-Py], [BA5835; 3-Cl-2-COOMe-4-Py], [BA5836; 5-Cl-2-COOMe-4-Py], [BA5837; 6-Cl-2-COOMe-4-] Py], [BA5838; 3-Me-2-COOMe-4-Py], [BA5839; 5-Me-2-COOMe-4-Py], [BA5840; 6-Me-2-COOMe-4-Py] _{, [BA5841; 3-CF 3} -2-COOMe-4-Py], [BA5842; 5-CF 3 -2-COOMe-4-Py], [BA5843; 6-CF 3 -2-COOMe-4-Py ], [BA5844; 3-CN-2-COOMe-4-Py], [BA5845; 5-CN-2-COOMe-4-Py], [BA5846; 6-CN-2-COOMe-4-Py], [BA 5847; 3-OMe-2-COOMe-4-Py], [BA 5848; 5-OMe-2-COOMe-4-Py], [BA 5849; 6-OMe-2-COOMe-4-Py], [BA 5850] 5-COOMe-4-Py !, [BA5851; 3-Cl-5-COOMe-4-Py], [BA5852; 2-Cl-5-COOMe-4-Py], [BA5853; 6-Cl-5; -COOMe-4-Py], [BA5854; 3-Me-5-COOMe-4-Py], [BA5855; 2-Me-5-COOMe-4-Py], [BA5856; 6-Me-5-COOMe -4-Py], [BA5857; 3-CF 3 -5-COOMe-4-Py], [BA5858; 2-CF 3 -5-COOMe-4-Py], [BA5859; 6-CF 3 -5- COOMe-4-Py], [BA 5860; 3-CN-5-COOMe-4-Py], [BA 586 1; 2-CN-5 -COOMe-4-Py], [BA5862; 6-CN-5-COOMe-4-Py], [BA5863; 3-OMe-5-COOMe-4-Py], [BA5864; 2-OMe-5-COOMe -4-Py], [BA5865; 6-OMe-5-COOMe-4-Py], [BA5866; 6-COOMe-4-Py], [BA5867; 3-Cl-6-COOMe-4-Py], [BA5868; 2-Cl-6-COOMe-4-Py], [BA5869; 5-Cl-6-COOMe-4-Py], [BA5870; 3-Me-6-COOMe-4-Py], [BA5871] ; 2-Me-6-COOMe -4-Py], [BA5872; 5-Me-6-COOMe-4-Py], [BA5873; 3-CF 3 -6-COOMe-4-Py], [BA5874; _{2-CF 3 -6-COOMe-} 4-Py], [BA5875; 5-CF 3 -6-COOMe-4-Py], [BA5876; 3-CN-6-COOMe-4-Py], [BA5877; 2-CN-6-COOMe-4-Py], [BA5878; 5-CN-6-COOMe-4-Py], [BA5879; 3-OMe-6-COOMe-4-Py], [BA5880; OMe-6-COOMe-4- Py], [BA5881; 5-OMe-6-COOMe-4-Py], [BA5882; 3-NO 2 -4-Py], [BA5883; 2-Cl-3-NO ₂ -4-Py], [BA 5884; 5-Cl-3-NO ₂ -4-Py],

[BA5885; 6-Cl-3 -NO 2 -4-Py], [BA5886; 2-Me-3-NO 2 -4-Py], [BA5887; 5-Me-3-NO 2 -4-Py] , [BA5888; 6-Me-3-NO ₂ -4-Py], [BA 5889; 2-CF ₃ -3-NO ₂ -4-Py], [BA 5890; 5-CF ₃ -3-NO _2-4 -Py], [BA5891; 6- CF 3 -3-NO 2 -4-Py], [BA5892; 2-CN-3-NO 2 -4-Py], [BA5893; 5-CN-3-NO 2 -4-Py], [BA5894; 6-CN-3-NO 2 -4-Py], [BA5895; 2-OMe-3-NO 2 -4-Py], [BA5896; 5-OMe-3-NO ₂ -4-Py], [BA 5897; 6-OMe-3-NO ₂ -4-Py], [BA 5898; 2-NO ₂ -4-Py], [BA 5899; 3-Cl-2-NO _2-4 -Py], [BA5900; 5- Cl-2-NO 2 -4-Py], [BA5901; 6-Cl-2-NO 2 -4-Py], [BA5902; 3-Me-2-NO 2 - 4-Py], [BA5903; 5-Me-2-NO 2 -4-Py], [BA5904; 6-Me-2-NO 2 -4-Py], [BA5905; 3-CF 3 -2-NO _{2 -4-Py], [BA5906} ; 5-CF 3 -2-NO 2 -4-Py], [BA5907; 6-CF 3 -2-NO 2 -4-Py], [BA5908; 3-CN- _{2-NO 2 -4-Py]} , [BA5909; 5-CN-2-NO 2 -4-Py], [BA5910; 6-CN-2-NO 2 -4-Py], [BA5911; 3-OMe -2-NO ₂ -4-Py !, [BA5912; 5-OMe-2-NO ₂ -4-Py], [BA5913; 6-OMe-2-NO ₂ -4-Py], [BA5914; _{NO 2 -4-Py], [} BA5915; 3-Cl-5-NO 2 -4-Py], [BA5916; 2-Cl-5-NO 2 -4-Py], [BA5917; 6-Cl-5 _{-NO 2 -4-Py], [} BA5918; 3-Me-5-NO 2 -4-Py], [BA5919; 2-Me-5-NO 2 -4-Py], [BA5920; 6-Me- 5-NO ₂ -4-Py], [BA 5921; 3-CF _{3 -5-NO 2 -4-Py]} , [BA5922; 2-CF 3 -5-NO 2 -4-Py], [BA5923; 6-CF 3 -5-NO 2 -4-Py], [BA5924; _{3-CN-5-NO 2} -4-Py], [BA5925; 2-CN-5-NO 2 -4-Py], [BA5926; 6-CN-5-NO 2 -4-Py], [BA5927 ; 3-OMe-5-NO 2 -4-Py], [BA5928; 2-OMe-5-NO 2 -4-Py], [BA5929; 6-OMe-5-NO 2 -4-Py], [ _{BA5930; 6-NO 2 -4-} Py], [BA5931; 3-Cl-6-NO 2 -4-Py], [BA5932; 2-Cl-6-NO 2 -4-Py], [BA5933; 5 _{-Cl-6-NO 2 -4-} Py], [BA5934; 3-Me-6-NO 2 -4-Py], [BA5935; 2-Me-6-NO 2 -4-Py], [BA5936; _{5-Me-6-NO 2} -4-Py], [BA5937; 3-CF 3 -6-NO 2 -4-Py], [BA5938; 2-CF 3 -6-NO 2 -4-Py], _{[BA5939; 5-CF 3 -6} -NO 2 -4-Py], [BA5940; 3-CN-6-NO 2 -4-Py], [BA5941; 2-CN-6-NO 2 -4-Py ], [BA5942; 5-CN -6-NO 2 -4-Py], [BA5943; 3-OMe-6-NO 2 -4-Py], [BA5944; 2-OMe-6-NO 2 -4- Py], [BA5945; 5- OMe-6-NO 2 -4-Py], [BA5946; 3-NH 2 -4-Py], [BA5947; 2-Cl-3-NH 2 -4-Py], [BA5948; 5-Cl-3 -NH 2 -4-Py], [BA5949; 6-Cl-3-NH 2 -4-Py], [BA5950; 2-Me-3-NH 2 -4-Py] , [BA5951; 5-Me- 3-NH 2 -4-Py], [BA5952; 6-Me-3-NH 2 -4-Py], [BA5953; 2-CF 3 -3-NH 2 -4- Py], [BA5954; 5- CF 3 -3-NH 2 -4-Py], [BA5955; 6-CF 3 -3-NH 2 -4-Py], [BA5956; 2-CN-3-NH 2 -4-Py], [BA 5957; 5-CN-3-NH ₂ -4-Py], [BA5958; 6-CN-3-NH 2 -4-Py], [BA5959; 2-OMe-3-NH 2 -4-Py], [BA5960; 5-OMe-3-NH _{2 -4-Py], [BA5961} ; 6-OMe-3-NH 2 -4-Py], [BA5962; 2-NH 2 -4-Py], [BA5963; 3-Cl-2-NH 2 -4 -Py], [BA5964; 5- Cl-2-NH 2 -4-Py], [BA5965; 6-Cl-2-NH 2 -4-Py], [BA5966; 3-Me-2-NH 2 - 4-Py], [BA5967; 5-Me-2-NH 2 -4-Py], [BA5968; 6-Me-2-NH 2 -4-Py], [BA5969; 3-CF 3 -2-NH ₂ -4-Py], [BA 5970; 5-CF ₃ -2-NH ₂ -4-Py], [BA 597 1; 6-CF ₃ -2-NH ₂ -4-Py], [BA 5 972; _{2-NH 2 -4-Py]} , [BA5973; 5-CN-2-NH 2 -4-Py], [BA5974; 6-CN-2-NH 2 -4-Py], [BA5975; 3-OMe _{-2-NH 2 -4-Py]} , [BA5976; 5-OMe-2-NH 2 -4-Py], [BA5977; 6-OMe-2-NH 2 -4-Py], [BA5978; 5- _{NH 2 -4-Py], [} BA5979; 3-Cl-5-NH 2 -4-Py], [BA5980; 2-Cl-5-NH 2 -4-Py], [BA5981; 6-Cl-5 _{-NH 2 -4-Py], [} BA5982; 3-Me-5-NH 2 -4-Py], [BA5983; 2-Me-5-NH 2 -4-Py], [BA5984; 6-Me- 5-NH ₂ -4-Py],

_{[BA5985; 3-CF 3 -5} -NH 2 -4-Py], [BA5986; 2-CF 3 -5-NH 2 -4-Py], [BA5987; 6-CF 3 -5-NH 2 -4 -Py], [BA5988; 3- CN-5-NH 2 -4-Py], [BA5989; 2-CN-5-NH 2 -4-Py], [BA5990; 6-CN-5-NH 2 - 4-Py], [BA5991; 3-OMe-5-NH 2 -4-Py], [BA5992; 2-OMe-5-NH 2 -4-Py], [BA5993; 6-OMe-5-NH 2 -4-Py], [BA5994; 6-NH 2 -4-Py], [BA5995; 3-Cl-6-NH 2 -4-Py], [BA5996; 2-Cl-6-NH 2 -4- Py], [BA5997; 5- Cl-6-NH 2 -4-Py], [BA5998; 3-Me-6-NH 2 -4-Py], [BA5999; 2-Me-6-NH 2 -4 -Py], [BA6000; 5- Me-6-NH 2 -4-Py], [BA6001; 3-CF 3 -6-NH 2 -4-Py], [BA6002; 2-CF 3 -6-NH ₂ -4-Py !, [BA 6003; 5-CF ₃ -6-NH ₂ -4-Py], [BA 6004; 3-CN-6-NH ₂ -4-Py], [BA 6005; 2-CN-6 _{-NH 2 -4-Py], [} BA6006; 5-CN-6-NH 2 -4-Py], [BA6007; 3-OMe-6-NH 2 -4-Py], [BA6008; 2-OMe- _{6-NH 2 -4-Py]} , [BA6009; 5-OMe-6-NH 2 -4-Py], [BA6010; 3-NHMe-4-Py], [BA6011; 2-Cl-3-NHMe- 4-Py], [BA6012; 5-Cl-3-NHMe-4-Py], [BA6013; 6-Cl-3-NHMe-4-Py], [BA6014; 2-Me-3-NHMe-4- Py], [BA6015; 5- Me-3-NHMe-4-Py], [BA6016; 6-Me-3-NHMe-4-Py], [BA6017; 2-CF 3 -3-NHMe-4-Py ], [BA6018; 5-CF 3 -3-NHMe-4-Py], [BA6019; 6-CF 3 -3-NHMe-4-Py], [BA6020; 2-CN-3-NHMe-4-Py ], [BA 6021; 5-CN-3-N HMe-4-Py], [BA6022; 6-CN-3-NHMe-4-Py], [BA6023; 2-OMe-3-NHMe-4-Py], [BA6024; 5-OMe-3-NHMe- 4-Py], [BA6025; 6-OMe-3-NHMe-4-Py], [BA6026; 2-NHMe-4-Py], [BA6027; 3-Cl-2-NHMe-4-Py], [BA6027] BA6028; 5-Cl-2-NHMe-4-Py], [BA6029; 6-Cl-2-NHMe-4-Py], [BA6030; 3-Me-2-NHMe-4-Py], [BA6031; 5-Me-2-NHMe- 4-Py], [BA6032; 6-Me-2-NHMe-4-Py], [BA6033; 3-CF 3 -2-NHMe-4-Py], [BA6034; 5 _{-CF 3 -2-NHMe-4-} Py], [BA6035; 6-CF 3 -2-NHMe-4-Py], [BA6036; 3-CN-2-NHMe-4-Py], [BA6037; 5 -CN-2-NHMe-4-Py], [BA6038; 6-CN-2-NHMe-4-Py], [BA6039; 3-OMe-2-NHMe-4-Py], [BA6040; 5-OMe -2-NHMe-4-Py !, [BA6041; 6-OMe-2-NHMe-4-Py], [BA6042; 5-NHMe-4-Py], [BA6043; 3-Cl-5-NHMe-4 -Py], [BA6044; 2-Cl-5-NHMe-4-Py], [BA6045; 6-Cl-5-NHMe-4-Py], [BA6046; 3-Me-5-NHMe-4-Py ], [BA6047; 2-Me -5-NHMe-4-Py], [BA6048; 6-Me-5-NHMe-4-Py], [BA6049; 3-CF 3 -5-NHMe-4-Py] _{, [BA6050; 2-CF 3} -5-NHMe-4-Py], [BA6051; 6-CF 3 -5-NHMe-4-Py], [BA6052; 3-CN-5-NHMe-4-Py] , [BA6053; 2-CN-5-NHMe-4-Py], [BA6054; 6-CN-5-NHMe-4-Py], [BA6055; 3-OMe-5-NHMe-4-Py], [BA6053; BA6056; 2-OMe-5-NHMe-4-Py], [BA6057; 6-OMe-5-NHMe-4-Py], [BA6058; 6-NHMe-4-Py], [BA6059; 3-Cl- 6-N HMe-4-Py !, [BA6060; 2-Cl-6-NHMe-4-Py], [BA6061; 5-Cl-6-NHMe-4-Py], [BA6062; 3-Me-6-NHMe- 4-Py], [BA6063; 2-Me-6-NHMe-4-Py], [BA6064; 5-Me-6-NHMe-4-Py], [BA6065; 3-CF 3 -6-NHMe-4 -Py], [BA6066; 2- CF 3 -6-NHMe-4-Py], [BA6067; 5-CF 3 -6-NHMe-4-Py], [BA6068; 3-CN-6-NHMe-4 -Py], [BA6069; 2-CN-6-NHMe-4-Py], [BA 6070; 5-CN-6-NHMe-4-Py], [BA6071; 3-OMe-6-NHMe-4-Py ], [BA6072; 2-OMe -6-NHMe-4-Py], [BA6073; 5-OMe-6-NHMe-4-Py], [BA6074; 3-NMe 2 -4-Py], [BA6075; _{2-Cl-3-NMe 2} -4-Py], [BA6076; 5-Cl-3-NMe 2 -4-Py], [BA6077; 6-Cl-3-NMe 2 -4-Py], [BA6078 ; 2-Me-3-NMe 2 -4-Py], [BA6079; 5-Me-3-NMe 2 -4-Py], [BA6080; 6-Me-3-NMe 2 -4-Py], [ _{BA6081; 2-CF 3 -3-} NMe 2 -4-Py], [BA6082; 5-CF 3 -3-NMe 2 -4-Py], [BA6083; 6-CF 3 -3-NMe 2 -4- Py], [BA6084; 2- CN-3-NMe 2 -4-Py],

[BA 6085; 5-CN-3-NMe ₂ -4-Py], [BA 6086; 6-CN -3-NMe ₂ -4-Py], [BA 6087; 2-OMe -3-NMe ₂ -4-Py] , [BA 6088; 5-OMe-3-NMe _2-4 -Py], [BA 6089; 6-OMe-3-NMe _2-4 -Py], [BA 6090; 4-NMe _2-4 -Py], [BA 60 01 ; 3-Cl-4-NMe 2 -4-Py], [BA6092; 5-Cl-4-NMe 2 -4-Py], [BA6093; 6-Cl-4-NMe 2 -4-Py], [ BA6094; 3-Me-4- NMe 2 -4-Py], [BA6095; 5-Me-4-NMe 2 -4-Py], [BA6096; 6-Me-4-NMe 2 -4-Py], [BA 6097; 3-CF ₃ -4-NMe ₂ -4-Py], [BA 6098; 5-CF ₃ -4-NMe ₂ -4-Py], [BA 6099; 6-CF ₃ -4-NMe _2-4 -Py], [BA6100; 3- CN-4-NMe 2 -4-Py], [BA6101; 5-CN-4-NMe 2 -4-Py], [BA6102; 6-CN-4-NMe 2 - 4-Py], [BA6103; 3-OMe-4-NMe 2 -4-Py], [BA6104; 5-OMe-4-NMe 2 -4-Py], [BA6105; 6-OMe-4-NMe 2 -4-Py], [BA6106; 5-NMe 2 -4-Py], [BA6107; 3-Cl-5-NMe 2 -4-Py], [BA6108; 2-Cl-5-NMe 2 -4- Py], [BA6109; 6- Cl-5-NMe 2 -4-Py], [BA6110; 3-Me-5-NMe 2 -4-Py], [BA6111; 2-Me-5-NMe 2 -4 -Py], [BA6112; 6- Me-5-NMe 2 -4-Py], [BA6113; 3-CF 3 -5-NMe 2 -4-Py], [BA6114; 2-CF 3 -5-NMe ₂ -4-Py], [BA 6115; 6-CF ₃ -5-NMe ₂ -4-Py], [BA 6116; 3-CN-5-NMe ₂ -4-Py], [BA 6117; 2-CN-5 _{-NMe 2 -4-Py], [} BA6118; 6-CN-5-NMe 2 -4-Py], [BA6119; 3-OMe-5-NMe 2 -4-Py], [BA61 20; 2-OMe-5- NMe 2 -4-Py], [BA6121; 6-OMe-5-NMe 2 -4-Py], [BA6122; 6-NMe 2 -4-Py], [BA6123; 3 _{-Cl-6-NMe 2 -4-} Py], [BA6124; 2-Cl-6-NMe 2 -4-Py], [BA6125; 5-Cl-6-NMe 2 -4-Py], [BA6126; _{3-Me-6-NMe 2} -4-Py], [BA6127; 2-Me-6-NMe 2 -4-Py], [BA6128; 5-Me-6-NMe 2 -4-Py], [BA6129 _{; 3-CF 3 -6-NMe} 2 -4-Py], [BA6130; 2-CF 3 -6-NMe 2 -4-Py], [BA6131; 5-CF 3 -6-NMe 2 -4-Py ], [BA6132; 3-CN -6-NMe 2 -4-Py], [BA6133; 2-CN-6-NMe 2 -4-Py], [BA6134; 5-CN-6-NMe 2 -4- Py], [BA6135; 3- OMe-6-NMe 2 -4-Py], [BA6136; 2-OMe-6-NMe 2 -4-Py], [BA6137; 5-OMe-6-NMe 2 -4 -Py], [BA6138; 3-ACNH-4-Py], [BA6139; 2-Cl-3-ACNH-4-Py], [BA6140; 5-Cl-3-ACNH-4-Py], [BA6141 6-Cl-3-ACNH-4-Py !, [BA6142; 2-Me-3-ACNH-4-Py], [BA6143; 5-Me-3-ACNH-4-Py], [BA6144; -Me-3-ACNH-4- Py], [BA6145; 2-CF 3 -3-ACNH-4-Py], [BA6146; 5-CF 3 -3-ACNH-4-Py], [BA6147; 6 _{-CF 3 -3-ACNH-4-} Py], [BA6148; 2-CN-3-ACNH-4-Py], [BA6149; 5-CN-3-ACNH-4-Py], [BA6150; 6- CN-3-ACNH-4-Py, [BA6151; 2-OMe-3-ACNH-4-Py], [BA6152; 5-OMe-3-ACNH-4-Py], [BA6153; 6-OMe- 3-ACNH-4-Py], [BA6154; 2-ACNH-4-Py], [BA6155; 3-Cl-2-ACNH-4-Py], [BA6156; 5-Cl-2-ACNH-4- Py], [BA6157; 6-Cl-2-ACNH-4-Py], [BA6158; 3-Me-2-ACNH-4-Py], [BA6159; 5-Me-2-ACNH-4-Py] , [BA6160; 6-Me- 2-ACNH-4-Py], [BA6161; 3-CF 3 -2-ACNH-4-Py], [BA6162; 5-CF 3 -2-ACNH-4-Py] _{, [BA6163; 6-CF 3} -2-ACNH-4-Py], [BA6164; 3-CN-2-ACNH-4-Py], [BA6165; 5-CN-2-ACNH-4-Py], [BA 6166; 6-CN-2-ACNH-4-Py], [BA 6167; 3-OMe-2-ACNH-4-Py], [BA 6168; 5-OMe-2-ACNH-4-Py], [BA 6169] 6-OMe-2-ACNH-4-Py !, [BA6170; 5-ACNH-4-Py], [BA6171; 3-Cl-5-ACNH-4-Py], [BA6172; 2-Cl-5; -ACNH-4-Py], [BA6173; 6-Cl-5-ACNH-4-Py], [BA6174; 3-Me-5-ACNH-4-Py], [BA6175; 2-Me-5-ACNH -4-Py], [BA6176; 6-Me-5-ACNH-4-Py], [BA6177; 3-CF 3 -5-ACNH-4-Py], [BA6178; 2-CF 3 -5-ACNH -4-Py], [BA6179; 6-CF 3 -5-ACNH-4-Py], [BA6180; 3-CN-5-ACNH-4-Py], [BA6181; 2-CN-5-ACNH- 4-Py], [BA6182; 6-CN-5-ACNH-4-Py], [BA6183; 3-OMe-5-ACNH-4-Py], [BA6184; 2-OMe-5-ACNH-4- Py],

[BA 6185; 6-OMe-5-ACNH-4-Py], [BA 6186; 6-ACNH-4-Py], [BA 6187; 3-Cl-6-ACNH-4-Py], [BA 6188; 2-Cl -6-ACNH-4-Py !, [BA6189; 5-Cl-6-ACNH-4-Py], [BA6190; 3-Me-6-ACNH-4-Py], [BA6191; 2-Me-6 -ACNH-4-Py], [ BA6192; 5-Me-6-ACNH-4-Py], [BA6193; 3-CF 3 -6-ACNH-4-Py], [BA6194; 2-CF 3 -6 -ACNH-4-Py], [ BA6195; 5-CF 3 -6-ACNH-4-Py], [BA6196; 3-CN-6-ACNH-4-Py], [BA6197; 2-CN-6- ACNH-4-Py !, [BA6198; 5-CN-6-ACNH-4-Py], [BA6199; 3-OMe-6-ACNH-4-Py], [BA6200; 2-OMe-6-ACNH- 4-Py], [BA6201; 5-OMe-6-ACNH-4-Py], [BA6202; 3- (N (Ac) (Me))-4-Py], [BA6203; 2-Cl-3- (N (Ac) (Me))-4-Py], [BA6204; 5-Cl-3- (N (Ac) (Me))-4-Py], [BA6205; 6-Cl-3- (N) (Ac) (Me))-4-Py], [BA6206; 2-Me-3- (N (Ac) (Me))-4-Py], [BA6207; 5-Me-3- (N (Ac) ) (Me))-4-Py], [BA6208; 6-Me-3- (N (Ac) (Me))-4-Py], [BA6209; 2-CF ₃ -3- (N (Ac)) (Me)) - 4-Py ], [BA6210; 5-CF 3 -3- (N (Ac) (Me)) - 4-Py], [BA6211; 6-CF 3 -3- (N (Ac) (Me))-4-Py], [BA6212; 2-CN-3- (N (Ac) (Me))-4-Py], [BA6213; 5-CN-3- (N (Ac) (Me) )) 4-Py], [BA 6214; 6-CN-3- (N (Ac) (Me))-4-Py], [BA 6215; 2-OMe-3- (N (Ac) (Me)) -4-Py], [BA6216; 5-OMe-3- (N (Ac) (Me))-4-Py], [BA6217; 6-OMe-3- (N (Ac) (Me))-4 -Py], [BA 6218; 2- (N (Ac ) (Me))-4-Py], [BA6219; 3-Cl-2- (N (Ac) (Me))-4-Py], [BA6220; 5-Cl-2- (N (Ac) ( Me))-4-Py], [BA 6221; 6-Cl-2- (N (Ac) (Me))-4-Py], [BA6222; 3-Me-2- (N (Ac) (Me)) )-[4-Py], [BA6223; 5-Me-2- (N (Ac) (Me))-4-Py], [BA6224; 6-Me-2- (N (Ac) (Me))- 4-Py], [BA6225; 3-CF 3 -2- (N (Ac) (Me)) - 4-Py], [BA6226; 5-CF 3 -2- (N (Ac) (Me)) - 4-Py], [BA6227; 6-CF 3 -2- (N (Ac) (Me)) - 4-Py], [BA6228; 3-CN-2- (N (Ac) (Me)) - 4 -Py], [BA6229; 5-CN-2- (N (Ac) (Me))-4-Py], [BA6230; 6-CN-2- (N (Ac) (Me))-4-Py ], [BA6231; 3-OMe-2- (N (Ac) (Me))-4-Py], [BA6232; 5-OMe-2- (N (Ac) (Me))-4-Py], [BA 6233; 6-OMe-2- (N (Ac) (Me))-4-Py], [BA6234; 5- (N (Ac) (Me))-4-Py], [BA6235; 3-Cl -5- (N (Ac) (Me))-4-Py], [BA6236; 2-Cl-5- (N (Ac) (Me))-4-Py], [BA 6237; 6-Cl-5 -(N (Ac) (Me))-4-Py], [BA6238; 3-Me-5- (N (Ac) (Me))-4-Py], [BA6239; 2-Me-5- ( N (Ac) (Me)) - 4-Py], [BA6240; 6-Me-5- (N (Ac) (Me)) - 4-Py], [BA6241; 3-CF 3 -5- (N (Ac) (Me)) - 4-Py], [BA6242; 2-CF 3 -5- (N (Ac) (Me)) - 4-Py], [BA6243; 6-CF 3 -5- (N (Ac) (Me))-4-Py], [BA6244; 3-CN-5- (N (Ac) (Me))-4-Py], [BA6245; 2-CN-5- (N (Ac) ) (Me))-4-Py], [BA6246; 6-CN-5- (N (Ac) (Me))-4-Py], [BA6247; 3-OMe-5- (N (Ac) ( Me))-4-Py], [BA 6248; 2-OMe -5- (N (Ac) (Me))-4-Py], [BA6249; 6-OMe-5- (N (Ac) (Me))-4-Py], [BA6250; 6- (N ( Ac) (Me))-4-Py], [BA6251; 3-Cl-6- (N (Ac) (Me))-4-Py], [BA6252; 2-Cl-6- (N (Ac)) (Me))-4-Py], [BA6253; 5-Cl-6- (N (Ac) (Me))-4-Py], [BA6254; 3-Me-6- (N (Ac) (Me) )) 4-Py], [BA 6255; 2-Me-6- (N (Ac) (Me))-4-Py], [BA 6 256; 5-Me-6- (N (Ac) (Me)) -4-Py], [BA6257; 3-CF 3 -6- (N (Ac) (Me)) - 4-Py], [BA6258; 2-CF 3 -6- (N (Ac) (Me)) -4-Py], [BA6259; 5-CF 3 -6- (N (Ac) (Me)) - 4-Py], [BA6260; 3-CN-6- (N (Ac) (Me)) - 4-Py], [BA6261; 2-CN-6- (N (Ac) (Me))-4-Py], [BA6262; 5-CN-6- (N (Ac) (Me))-4-] Py], [BA6263; 3-OMe-6- (N (Ac) (Me))-4-Py], [BA6264; 2-OMe-6- (N (Ac) (Me))-4-Py] , [BA6265; 5-OMe-6- (N (Ac) (Me))-4-Py], [BA6266; 3-AC-4-Py], [BA6267; 2-Cl-3-AC-4- Py], [BA6268; 5-Cl-3-AC-4-Py], [BA6269; 6-Cl-3-AC-4-Py], [BA6270; 2-Me-3-AC-4-Py] , [BA6271; 5-Me- 3-AC-4-Py], [BA6272; 6-Me-3-AC-4-Py], [BA6273; 2-CF 3 -3-AC-4-Py], _{[BA6274; 5-CF 3 -3} -AC-4-Py], [BA6275; 6-CF 3 -3-AC-4-Py], [BA6276; 2-CN-3-AC-4-Py], [BA 6277; 5-CN-3-AC-4-Py], [BA 6278; 6-CN-3-AC-4-Py], [BA 6279; 2-OMe-3-AC-4-Py], [BA 6280] 5-OMe-3-AC-4-Py !, [BA6281; 6-OMe-3-AC-4-Py], [BA6282; 2-AC-4-Py], [BA6283; 3-Cl-2-AC-4-Py], [BA6284; 5-Cl-2-AC-4-Py],

[BA6285; 6-Cl-2-AC-4-Py], [BA6286; 3-Me-2-AC-4-Py], [BA6287; 5-Me-2-AC-4-Py], [BA6288] ; 6-Me-2-AC -4-Py], [BA6289; 3-CF 3 -2-AC-4-Py], [BA6290; 5-CF 3 -2-AC-4-Py], [BA6291 _{; 6-CF 3 -2-AC} -4-Py], [BA6292; 3-CN-2-AC-4-Py], [BA6293; 5-CN-2-AC-4-Py], [BA6294; 6-CN-2-AC-4-Py !, [BA6295; 3-OMe-2-AC-4-Py], [BA6296; 5-OMe-2-AC-4-Py], [BA6297; OMe-2-AC-4-Py], [BA6298; 5-AC-4-Py], [BA6299; 3-Cl-5-AC-4-Py], [BA6300; 2-Cl-5-AC- 4-Py], [BA6301; 6-Cl-5-AC-4-Py], [BA6302; 3-Me-5-AC-4-Py], [BA6303; 2-Me-5-AC-4- 4 Py], [BA6304; 6- Me-5-AC-4-Py], [BA6305; 3-CF 3 -5-AC-4-Py], [BA6306; 2-CF 3 -5-AC-4- Py], [BA6307; 6- CF 3 -5-AC-4-Py], [BA6308; 3-CN-5-AC-4-Py], [BA6309; 2-CN-5-AC-4-Py ], [BA6310; 6-CN-5-AC-4-Py], [BA6311; 3-OMe-5-AC-4-Py], [BA6312; 2-OMe-5-AC-4-Py], [BA6313; 6-OMe-5-AC-4-Py], [BA6314; 6-AC-4-Py], [BA6315; 3-Cl-6-AC-4-Py], [BA6316; 2-Cl -6-AC-4-Py], [BA 6317; 5-Cl-6-AC-4-Py], [BA 6318; 3-Me-6-AC-4-Py], [BA 6319; 2-Me-6 -AC-4-Py], [ BA6320; 5-Me-6-AC-4-Py], [BA6321; 3-CF 3 -6-AC-4-Py], [BA6322; 2-CF 3 -6 -AC-4-Py], [ BA6323; 5-CF 3 -6-AC-4-Py], [BA6324; 3-CN-6-AC-4-Py], [BA6325; 2-CN-6- AC -4-Py], [BA6326; 5-CN-6-AC-4-Py], [BA6327; 3-OMe-6-AC-4-Py], [BA6328; 2-OMe-6-AC-4 -Py], [BA6329; 5-OMe-6-AC-4-Py], [BA6330; 3,4- (methylenedioxy) phenyl], [BA6331; 2,3-dihydrobenzofuran-5-yl], [BA6332; 2,3-dihydrobenzofuran-6-yl], [BA6333; 1,3-dihydroisobenzofuran-5-yl], [BA6334; benzofuran-5-yl], [BA6335; benzofuran-6-yl] [BA 6336; 2,3-dihydrobenzothiophen-5-yl], [BA 6337; 2,3-dihydrobenzothiophen-6-yl], [BA 6338; 1,3-dihydroisobenzothiophen-5-yl], [BA6339; benzothiophen-5-yl], [BA6340; benzothiophen-6-yl], [BA6341; 1,4-benzodioxane-6-yl], [BA6342; chroman-6-yl], [BA6343; Chroman-7-yl], [BA 6344; isochroman-6-yl], [BA 6345; isochroman-7-yl], [BA 6346; 2-quinolyl], [BA 6347; (Methylenedioxy) phenyl], [BA 6349; 2-indolyl ], [BA 6350; 3-indolyl], [BA 6351; 2-benzoimidazolyl], [BA 6352; 2-thienyl], [BA 6353; 3-thienyl], [BA 6354; 2,3-dihydrobenzofuran-7-yl], [BA 6352; 2-pyrimidinyl], [BA 6356; 5-pyrimidinyl], [BA 6357; 2-thiazolyl], [BA 6358; 4-thiazolyl], [BA 6359; 5-thiazolyl], [BA 6 360; 2-pyrazinyl], [BA 6361; 3-Pyridazinyl], [BA6362; 2-benzoxazolyl], [BA6363; 2-benzothiazolyl], [BA6364; 2-quinazolinyl], [BA6365; 2-quinoxalinyl].

  Further, the present compounds AB1-BB1 to AB119-BB511 and the present compounds AB1-BB1001 to AB119-BB3016 can also be obtained according to the method described above.

The present compounds AB1-BB1 to AB119-BB511 and the present compounds AB1-BB1001 to AB119-BB3016 are compounds represented by the following formula (ABBB).

[Wherein, X ^{121 to} X ¹²⁷ each represent a substituent corresponding to each of substituent numbers (MB1) AB 1 to AB 319 shown below, and in the formula, E ¹⁰² represents a substituent number (MB 2) BB 1 shown below ~ BB 511 is represented. ]
For example, the present compound AB2-BB1, in the compounds of formula (ABBB), X ¹²¹ ~X ¹²⁷ substituents ID AB2 (X ¹²¹ and X ¹²⁴ to X ¹²⁶ is a hydrogen atom, X ¹²² and X ¹²⁷ is an oxygen atom And ^X123 represents a fluorine atom, and E ¹⁰² represents a compound in which the substituent number (MB2) is BB1 (phenyl group), and is represented by the following formula.
Further, the AB2-BB1001, the compounds of formula (AB2), X ¹²¹ ~X ¹²⁷ substituents ID AB2 (X ¹²¹ and X ¹²⁴ to X ¹²⁶ is a hydrogen atom, X ¹²² and X ¹²⁷ is an oxygen atom, The compound represented by the following formula is a compound wherein X ¹²³ is a fluorine atom) and the moiety of E ¹⁰² is a substituent number (MB2) of BB1001 (R201 to R206 and R250 to R252 are hydrogen atoms E201).
[Substituent group number ^{(MB1); X 121, X} 122, X 123, X 124, X 125, X 126, X 127], [AB1; H, O, H, H, H, H, O], [AB2 H, O, F, H, H, H, O, [AB 3; H, O, Cl, H, H, H, O], [AB 4; H, O, Br, H, H, H, O] ], [AB5; H, O, I, H, H, H, O], [AB 6; H, O, Me, H, H, H, O], [AB 7; H, O, Et, H, H] , H, O], [AB 8; H, O, Pr, H, H, H, O], [AB 9; H, O, i-Pr, H, H, H, O], [AB 10; H, O _{, CH = CH 2, H,} H, H, O], [AB11; H, O, C (CH 3) = CH 2, H, H, H, O], [AB12; H, O, C≡CH , H, H, H, O], [AB 13; H, O, C≡CCH ₃ , H, H, H, O], [AB 14; H, O, c-Pr, H, H, H, O] , [AB15; H, O, OMe, H, H, H, O], [AB16; H, O, OEt, H, H, H, O], [AB17; H, O, Oi-Pr, H, H, H, O], [AB 18; H, O, S Me, H, H, H, O], [AB 19; H, O, SE t, H, H, H, O], [AB 20; H, O, _{CH 2 F, H, H,} H, O], [AB21; H, O, CHF 2, H, H, H, O], [AB22; H, O, CF 3, H, H, H, O] , [AB23; H, O, OCH 2 F, H, H, H, O], [AB24; H, O, OCHF 2, H, H, H, O], [AB25; H, O, OCF 3, H, H, H, O], [AB 26; H, O, SCH ₂ F, H, H, H, O], [AB 27; H, O, SCHF ₂ , H, H, H, O], [AB 28 _{; H, O, SCF 3,} H, H, H, O], [AB29; H, O, CN, H, H, H, O], [AB30; H, O, NO 2, H, H, H , O], [AB31; Me, O, H, H, H, H, O], [AB 32; Me, O, F, H, H, H, O], [AB 33; Me, O, Cl, H , H, H, O], [AB34; Me, O, Br, H, H, H, O], [AB 35; Me, O, I, H, H, H, O], [AB 36; Me, O , Me, H, H, H, O], [AB 37; Me, O, Et, H, H, H, O], [AB 38; Me, O, Pr, H, H, H, O], [AB 39 ; Me, O, i-Pr, H, H, H, O] , [AB40; Me, O, CH = CH 2, H, H, H, O], [AB41; Me, O, C (CH 3) = CH 2, H, H, H, O], [AB 42; Me, O, C≡CH, H, H, H, O], [AB 43; Me, O, C≡ CCH ₃ , H, H, H, O], [AB 44; Me , O, c-Pr, H, H, H, O], [AB 45; Me, O, OMe, H, H, H, O], [AB 46; Me, O, OEt, H, H, H, O ], [AB 47; Me, O, Oi-Pr, H, H, H, O], [AB 48; Me, O, SMe, H, H, H, O], [AB 49; Me, O, SEt, H , H, H, O], [AB50; Me, O, CH 2 F, H, H, H, O], [AB51; Me, O, CHF 2, H, H, H, O], [AB52; _{Me, O, CF 3, H} , H, H, O], [AB53; Me, O, OCH 2 F, H, H, H, O], [AB54; Me, O, OCHF 2, H, H, H, O], [AB55; Me, O, OCF 3, H, H, H, O], [AB56; Me, O, SCH 2 F, H, H, H, O], [AB57; Me, O , SCHF ₂ , H, H, H, O], [AB 58; Me, O, SCF ₃ , H, H, H, O], [AB 59; Me, O, CN, H, H, H, O], [AB60; Me, O, NO 2, H, H, H, O], [AB61; Et, O, H, H, H, H, O], [AB62; Et, O, F, H, H, H, O], [AB 63; Et, O, Cl, H, H, H, O], [AB 64; Et, O, Br, H, H, H, O], [AB 65; Et, O, I, H, H, H, O], [AB 66; Et, O, Me, H, H, H, O], [AB 67; Et, O, Et, H, H, H, O], [AB 68; Et, Et, O, Pr, H, H, H, O], [AB69; Et, O, i-Pr, H, H, H, O], [AB70; Et, O, CH = CH 2, H, H, H , O], [AB71; Et , O, C (CH 3) = CH 2, H, H, H, O], [AB72; Et, O, C≡CH, H, H, H, O], [ AB 73; Et, O, C≡CCH ₃ , H, H, H, O], [AB 74; Et, O, c-Pr, H, H, H, O], [AB 75; Et, O, OMe, H , H, H, O], [AB 76; Et, O, OEt, H, H, H, O], [AB 77; Et, O, Oi-Pr, H, H, H, O], [AB 78; Et, O, SMe, H, H, H, O], [AB 79; Et, O, SEt, H, H, H, O], [AB 80; Et, O, CH ₂ F, H, H , H, O], [AB81 ; Et, O, CHF 2, H, H, H, O], [AB82; Et, O, CF 3, H, H, H, O], [AB83; Et, O OCH ₂ F, H, H, H, O], [AB 84; Et, O, OCHF ₂ , H, H, H, O], [AB 85; Et, O, OCF ₃ , H, H, H, O ], [AB 86; Et, O, SCH ₂ F, H, H, H, O], [AB 87; Et, O, SCHF ₂ , H, H, H, O], [AB 88; Et, O, SCF ₃ , H, H, H, O], [AB 89; Et, O, CN, H, H, H, O], [AB 90; Et, O, NO ₂ , H, H, H, O], [AB 91; Pr, O, H, H, H, H, H, O], [AB 92; Pr, O, F, H, H, H, O], [AB 93; Pr, O, Cl, H, H, H, O] , [AB 94; Pr, O, Br, H, H, H, O], [AB 95; Pr, O, I, H, H, H, O], [AB 96; Pr, O, Me, H, H, H, H, O], [AB 97; Pr, O, Et, H, H, H, O], [AB 98; Pr, O, Pr, H, H, H, O], [AB 99; Pr, O, i- Pr, H, H, H, O],

[AB100; Pr, O, CH = CH 2, H, H, H, O], [AB101; Pr, O, C (CH 3) = CH 2, H, H, H, O], [AB102; Pr , O, C≡CH, H, H, H, H, O], [AB 103; Pr, O, C≡ CCH ₃ , H, H, H, O], [AB 104; Pr, O, c-Pr, H, H, H, O], [AB 105; Pr, O, OMe, H, H, H, O], [AB 106; Pr, O, OEt, H, H, H, O], [AB 107; Pr, O, Oi-Pr, H, H, H, O], [AB 108; Pr, O, SMe, H, H, H, O], [AB 109; Pr, O, SEt, H, H, H, O], [[ _{AB110; Pr, O, CH 2} F, H, H, H, O], [AB111; Pr, O, CHF 2, H, H, H, O], [AB112; Pr, O, CF 3, H, H, H, O], [ AB113; Pr, O, OCH 2 F, H, H, H, O], [AB114; Pr, O, OCHF 2, H, H, H, O], [AB115; Pr _{, O, OCF 3, H,} H, H, O], [AB116; Pr, O, SCH 2 F, H, H, H, O], [AB117; Pr, O, SCHF 2, H, H, H , O], [AB 118; Pr, O, SCF ₃ , H, H, H, O], [AB 119; Pr, O, CN, H, H, H, O], [AB 120; Pr, O, NO ₂ , H, H, H, O], [AB 121; i-Pr, O, H, H, H, H, O], [AB 122; i-Pr, O, F, H, H, H, O], [AB 123; i-Pr, O, Cl, H, H, H, O], [AB 124; i-Pr, O, Br, H, H, H, O], [AB 125; i-Pr, O, I , H, H, H, O], [AB 126; i-Pr, O, Me, H, H, H, O], [AB 127; i-Pr, O, Et, H, H, H, O], [AB 128; i-Pr, O, Pr, H, H, H, O], [AB 129; i-Pr, O, i-Pr, H, H, H, O], [AB 130; i-Pr, O , CH = CH ₂ , H, H, H, O, [AB 131; i-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AB 132; i-Pr, O , C≡CH, H, H, H, O, [AB133; i-Pr, O, C≡CCH ₃ , H, H, H, O], [AB 134; i-Pr, O, c-Pr, H, H, H, O], [AB 135; i-Pr, O, OMe, H, H, H, O], [AB136; i-Pr, O, OEt, H, H, H, O], [AB 137; i-Pr, O, Oi-Pr, H, H, H, O], [A AB138; i-Pr, O, SMe, H, H, H, O], [AB139; i-Pr, O, SEt, H, H, H, O], [AB 140; i-Pr, O, CH ₂ F, H, H, H, O], [AB141; i-Pr, O, CHF 2, H, H, H, O], [AB142; i-Pr, O, CF 3, H, H, H, O], [AB143; i- Pr, O, OCH 2 F, H, H, H, O], [AB144; i-Pr, O, OCHF 2, H, H, H, O], [AB145; i _{-Pr, O, OCF 3, H} , H, H, O], [AB146; i-Pr, O, SCH 2 F, H, H, H, O], [AB147; i-Pr, O, SCHF 2 , H, H, H, O], [AB 148; i-Pr, O, SCF ₃ , H, H, H, O], [AB 149; i-Pr, O, CN, H, H, H, O] , [AB150; i-Pr, O, NO 2, H, H, H, O], [AB151; c-Pr, O, H, H, H, H, O], [AB152; c-Pr, O , F, H, H, H, O], [AB153; c-Pr, O, Cl, H, H, H, O], [AB 154; c-Pr, O, Br, H, H, H, O ], [AB 155; c-Pr, O, I, H, H, H, O], [AB 156; c-Pr, O, Me, H, H, H, O], [AB 157; c-Pr, O , Et, H, H, H, O], [AB158; c-Pr, O, Pr, H, H, H, O], [AB 159; c-Pr, O, i-Pr, H, H, H , O], [AB 160; c-Pr, O, CH = CH ₂ , H, H, H, O], [AB 161; c-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H , O], [AB 162; c-Pr, O, C≡CH, H, H, H, O], [AB 163; c-Pr, O, C≡ CCH ₃ , H, H, H, O], [[ AB 164; c-Pr, O, c-Pr, H, H, H, O], [AB 165; c-Pr, O, OMe, H, H, H, O], [AB 166; c-Pr, O, OEt, H, H, H, O], [AB 167; c-Pr, O, Oi-Pr, H, H, H, O], [AB 168; c-Pr, O, SMe, H, H, H, O], [AB 169; c-Pr, O, SEt, H, H, H, O], [AB 170; c-Pr, O, CH ₂ F, H, H, H, O], [ AB171; c-Pr, O, CHF 2, H, H, H, O], [AB172; c-Pr, O, CF 3, H, H, H, O], [ AB173; c-Pr, O, OCH 2 F, H, H, H, O], [AB174; c-Pr, O, OCHF 2, H, H, H, O], [AB175; c-Pr, O , OCF ₃ , H, H, H, O], [AB176; c-Pr, O, SCH ₂ F, H, H, H, O], [AB 177; c-Pr, O, SCHF ₂ , H, H , H, O], [AB 178; c-Pr, O, SCF ₃ , H, H, H, O], [AB 179; c-Pr, O, CN, H, H, H, O], [AB 180; _{c-Pr, O, NO 2} , H, H, H, O], [AB181; SMe, O, H, H, H, H, O], [AB182; SMe, O, F, H, H, H , O], [AB183; SMe, O, Cl, H, H, H, O], [AB 184; SMe, O, Br, H, H, H, O], [AB 185; SMe, O, I, H , H, H, O], [AB 186; SMe, O, Me, H, H, H, O], [AB 187; SMe, O, Et, H, H, H, O], [AB 188; SMe, O , Pr, H, H, H , O], [AB189; SMe, O, i-Pr, H, H, H, O], [AB190; SMe, O, CH = CH 2, H, H, H, O], [AB191; SMe, O, C (CH 3) = CH 2, H, H, H, O], [AB192; SMe, O, C≡CH, H, H, H, O], [AB193 SMe, O, C≡CCH ₃ , H, H, H, O], [AB194; SMe, O, c-Pr, H, H, H, O], [AB 195; SMe, O, OMe, H, H, H, O], [AB 196; SMe, O, OEt, H, H, H, O], [AB 197; SMe, O, Oi-Pr, H, H, H, O], [AB 198; SMe, O, SMe, H, H, H, O], [AB 199; SMe, O, SEt, H, H, H, O],

[AB200; SMe, O, CH 2 F, H, H, H, O], [AB201; SMe, O, CHF 2, H, H, H, O], [AB202; SMe, O, CF 3, H , H, H, O], [AB203; SMe, O, OCH 2 F, H, H, H, O], [AB204; SMe, O, OCHF 2, H, H, H, O], [AB205; _{SMe, O, OCF 3, H} , H, H, O], [AB206; SMe, O, SCH 2 F, H, H, H, O], [AB207; SMe, O, SCHF 2, H, H, H, O], [AB208; SMe, O, SCF 3, H, H, H, O], [AB209; SMe, O, CN, H, H, H, O], [AB210; SMe, O, NO ₂ , H, H, H, O], [AB 211; OMe, O, H, H, H, H, O], [AB 212; OMe, O, F, H, H, H, O], [AB 213; OMe, O, Cl, H, H, H, O], [AB 214; OMe, O, Br, H, H, H, O], [AB 215; OMe, O, I, H, H, H, O] , [AB 216; OMe, O, Me, H, H, H, O], [AB 217; OMe, O, Et, H, H, H, O], [AB 218; OMe, O, Pr, H, H, H, O], [AB219; OMe, O, i-Pr, H, H, H, O], [AB220; OMe, O, CH = CH 2, H, H, H, O], [AB221; OMe , O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AB 222; OMe, O, C≡CH, H, H, H, O], [AB 223; OMe, O, C≡ _{CCH 3, H, H, H} , O], [AB224; OMe, O, c-Pr, H, H, H, O], [AB225; OMe, O, OMe, H, H, H, O], [AB226; OMe, O, OEt, H, H, H, O], [AB 227; OMe, O, Oi-Pr, H, H, H, O], [AB 228; OMe, O, SMe, H, H , H, O], [AB 229; OMe, O, SEt, H, H, H, O], [AB 230; OMe, O, CH ₂ F, H, H, H, O], [AB 231; OMe, O _{, CHF 2, H, H,} H, O], [AB232; OMe, O, CF 3, H, H, H, O], [AB233; OMe, O, OCH 2 F, H, H, H, O ], [AB 234; OMe, O, OCHF ₂ , H, H, H, O], [AB 235; OMe, O, OCF ₃ , H, H, H, O], [AB 236; OMe, O, SCH ₂ F, H, H, H, O], [AB 237; OMe, O, SCHF ₂ , H, H, H, O], [AB 238; OMe, O , SCF ₃ , H, H, H, O], [AB 239; OMe, O, CN, H, H, H, O], [AB 240; OMe, O, NO ₂ , H, H, H, O], [AB241; H, S, H, H, H, H, H, O], [AB 242; H, S, F, H, H, H, O], [AB 243; H, S, Cl, H, H, H , O], [AB244; H, S, Br, H, H, O], [AB245; H, S, I, H, H, H, O], [AB 246; H, S, Me, H , H, H, O], [AB 247; H, S, Et, H, H, H, O], [AB 248; H, S, Pr, H, H, H, O], [AB 249; H, S , i-Pr, H, H , H, O], [AB250; H, S, CH = CH 2, H, H, H, O], [AB251; H, S, C (CH 3) = CH 2 , H, H, H, O], [AB 252; H, S, C≡CH, H, H, H, O], [AB 253; H, S, C≡ CCH ₃ , H, H, H, O] , [AB254; H, S, c-Pr, H, H, H, O], [AB 255; H, S, OMe, H, H, H, O], [AB 256; H, S, OEt, H, H, H, O], [AB 257; H, S, Oi-Pr, H, H, H, O], [AB 258; H, S, S Me, H, H, H, O], [AB 259; H, S, SEt, H, H, H, O], [AB 260; H, S, CH ₂ F, H, H, H, O], [AB 261; H, S, CHF ₂ , H, H, H, O ], [AB262; H, S , CF 3, H, H, H, O], [AB263; H, S, OCH 2 F, H, H, H, O], [AB264; H, S, OCHF 2 , H, H, H, O ], [AB265; H, S, OCF 3, H, H, H, O], [AB266; H, S, SCH 2 F, H, H, H, O], [ _{AB267; H, S, SCHF 2} , H, H, H, O], [AB268; H, S, SCF 3, H, H, H, O], [AB269; H, S, CN, H, H, H, O], [AB 270; H, S, NO ₂ , H, H, H, O], [AB 271; Me, S, H, H, H, H, O], [AB 272; Me, S, F , H, H, H, O], [AB 273; Me, S, Cl, H, H, H, O], [AB 274; Me, S, B r, H, H, H, O], [AB 275; Me, S, I, H, H, H, O], [AB 276; Me, S, Me, H, H, H, O], [AB 277; Me, S, Et, H, H, H, O], [AB 278; Me, S, Pr, H, H, H, O], [AB 279; Me, S, i-Pr, H, H, H, H, O], [AB280; Me, S, CH = CH 2, H, H, H, O], [AB281; Me, S, C (CH 3) = CH 2, H, H, H, O], [ AB282; Me, S, C≡CH, H, H, H, O], [AB 283; Me, S, C≡CCH ₃ , H, H, H, O], [AB 284: Me, S, c-Pr , H, H, H, O], [AB 285; Me, S, OMe, H, H, H, O], [AB 286; Me, S, OEt, H, H, H, O], [AB 287; Me , S, Oi-Pr, H, H, H, O], [AB 288; Me, S, SMe, H, H, H, O], [AB 289; Me, S, SE t, H, H, H, O ], [AB290; Me, S , CH 2 F, H, H, H, O], [AB291; Me, S, CHF 2, H, H, H, O], [AB292; Me, S, CF 3 , H, H, H, O ], [AB293; Me, S, OCH 2 F, H, H, H, O], [AB294; Me, S, OCHF 2, H, H, H, O], [ _{AB295; Me, S, OCF 3} , H, H, H, O], [AB296; Me, S, SCH 2 F, H, H, H, O], [AB297; Me, S, SCHF 2, H, H, H, O], [AB 298; Me, S, SCF ₃ , H, H, H, O], [AB 299; Me, S, CN, H, H, H, O],

[AB300; Me, S, NO 2, H, H, H, O], [AB301; Et, S, H, H, H, H, O], [AB302; Et, S, F, H, H, H, O], [AB 303; Et, S, Cl, H, H, H, O], [AB 304; Et, S, Br, H, H, H, O], [AB 305; Et, S, I, H, H, H, O], [AB 306; Et, S, Me, H, H, H, O], [AB 307; Et, S, Et, H, H, H, O], [AB 308; S, Pr, H, H, H, O], [AB309; Et, S, i-Pr, H, H, H, O], [AB310; Et, S, CH = CH 2, H, H, H , O], [AB311; Et , S, C (CH 3) = CH 2, H, H, H, O], [AB312; Et, S, C≡CH, H, H, H, O], [ _{AB313; Et, S, C≡CCH 3} , H, H, H, O], [AB314; Et, S, c-Pr, H, H, H, O], [AB315; Et, S, OMe, H , H, H, O], [AB 316; Et, S, OEt, H, H, H, O], [AB 317; Et, S, Oi-Pr, H, H, H, O], [AB 318; Et , S, SMe, H, H, H, O], [AB 319; Et, S, SEt, H, H, H, O], [AB 320; Et, S, CH ₂ F, H, H, H, O ], [AB321; Et, S , CHF 2, H, H, H, O], [AB322; Et, S, CF 3, H, H, H, O], [AB323; Et, S, OCH 2 F , H, H, H, O ], [AB324; Et, S, OCHF 2, H, H, H, O], [AB325; Et, S, OCF 3, H, H, H, O], [AB326 Et, S, SCH ₂ F, H, H, H, H, O], [AB 327; Et, S, SCHF ₂ , H, H, H, O], [AB 328; Et, S, SCF ₃ , H, H , H, O], [AB329 ; Et, S, CN, H, H, H, O], [AB330; Et, S, NO 2, H, H, H, O], [AB331; H, O, H, H, H, H, S], [AB332; H, O, F, H, H, H, S], [AB 333; H, O, Cl, H, H, H, S], [AB334; H, O, Br, H, H, H, S], [AB 335; H, O, I, H, H, H, S], [AB 336; H, O, Me, H, H, H, S] , [AB 337; H, O, Et, H, H, H, S], [AB 338; H, O, Pr, H , H, H, S], [AB339; H, O, i-Pr, H, H, H, S], [AB340; H, O, CH = CH 2, H, H, H, S], [ AB 341; H, O, C (CH ₃ ) = CH ₂ , H, H, H, S], [AB 342; H, O, C≡CH, H, H, H, S], [AB 343; H, O , C≡CCH ₃ , H, H, H, S], [AB 344; H, O, c-Pr, H, H, H, S], [AB 345; H, O, OMe, H, H, H, S, [AB346; H, O, OEt, H, H, H, S], [AB 347; H, O, Oi-Pr, H, H, H, S], [AB 348; H, O, SMe, H, H, H, S] , [AB349; H, O, SEt, H, H, H, S], [AB350; H, O, CH 2 F, H, H, H, S], [AB351; _{H, O, CHF 2, H} , H, H, S], [AB352; H, O, CF 3, H, H, H, S], [AB353; H, O, OCH 2 F, H, H, H, S], [AB354; H, O, OCHF 2, H, H, H, S], [AB355; H, O, OCF 3, H, H, H, S], [AB356; H, O, SCH ₂ F, H, H, H, S], [AB 357; H, O, SCHF ₂ , H, H, H, S], [AB 358; H, O, SCF ₃ , H, H, H, S] , [AB 359; H, O, CN, H, H, H, S], [AB 360; H, O, NO ₂ , H, H, H, S], [AB 361; Me, O, H, H, H , H, S], [AB 362; Me, O, F, H, H, H, S], [AB 363; Me, O, Cl, H, H, H, S], [AB 364; Me, O, Br] , H, H, H, S], [AB365; Me, O, I, H, H, H, S], [AB 366; Me, O, Me, H, H, H, S], [AB 367; Me , O, Et, H, H, H, S], [AB 368; Me, O, Pr, H, H, H, S], [AB 369; Me, O, i-Pr, H, H, H, S Me, O, CH = CH ₂ , H, H, H, S], [AB 371; Me, O, C (CH ₃ ) = CH ₂ , H, H, H, S], [AB 372] Me, O, C≡CH, H, H, H, S, [AB 373; Me, O, C≡CCH ₃ , H, H, H, S], [AB 374; Me, O, c-Pr, H, H, H, S], [AB 375; Me, O, OMe, H, H, H, S], [AB 376; Me, O , OEt, H, H, H, S], [AB 377; Me, O, Oi-Pr, H, H, H, S], [AB 378; Me, O, SMe, H, H, H, S], [AB379; Me, O, SEt , H, H, H, S], [AB380; Me, O, CH 2 F, H, H, H, S], [AB381; Me, O, CHF 2, H, H, H, S], [ AB382; Me, O, CF 3, H, H, H, S], [AB383; Me, O, OCH 2 F, H, H, H, S], [AB384; Me , O, OCHF ₂ , H, H, H, S], [AB 385; Me, O, OCF ₃ , H, H, H, S], [AB 386; Me, O, SCH ₂ F, H, H, H , S], [AB 387; Me, O, SCHF ₂ , H, H, H, S], [AB 388; Me, O, SCF ₃ , H, H, H, S], [AB 389; Me, O, CN , H, H, H, S ], [AB390; Me, O, NO 2, H, H, H, S], [AB391; Et, O, H, H, H, H, S], [AB392; Et, O, F, H, H, H, S], [AB 393; Et, O, Cl, H, H, H, S], [AB 394; Et, O, Br, H, H, H, S] , [AB 395; Et, O, I, H, H, H, S], [AB 396; Et, O, Me, H, H, H, S], [AB 397; Et, O, Et, H, H, H, S], [AB 398; Et, O, Pr, H, H, H, S], [AB 399; Et, O, i-Pr, H, H, H, S],

[AB400; Et, O, CH = CH 2, H, H, H, S], [AB401; Et, O, C (CH 3) = CH 2, H, H, H, S], [AB402; Et , O, C≡CH, H, H, H, S, [AB 403; Et, O, C≡ CCH ₃ , H, H, H, S], [AB 404; Et, O, c-Pr, H, H, H, S], [AB 405; Et, O, OMe, H, H, H, S], [AB 406; Et, O, OEt, H, H, H, S], [AB 407; Et, O, Oi-Pr, H, H, H, S], [AB 408; Et, O, SMe, H, H, H, S], [AB 409; Et, O, SEt, H, H, H, S], [ _{AB410; Et, O, CH 2} F, H, H, H, S], [AB411; Et, O, CHF 2, H, H, H, S], [AB412; Et, O, CF 3, H, H, H, S], [ AB413; Et, O, OCH 2 F, H, H, H, S], [AB414; Et, O, OCHF 2, H, H, H, S], [AB415; Et _{, O, OCF 3, H,} H, H, S], [AB416; Et, O, SCH 2 F, H, H, H, S], [AB417; Et, O, SCHF 2, H, H, H , S], [AB418; Et , O, SCF 3, H, H, H, S], [AB419; Et, O, CN, H, H, H, S], [AB420; H, O, H, F, H, H, O], [AB 421; H, O, F, F, H, H, O], [AB 422; H, O, Cl, F, H, H, O], [AB 423; H, O, Br, F, H, H, O], [AB 424; H, O, I, F, H, H, O], [AB 425; H, O, Me, F, H, H, O], [AB AB 426; H, O, Et, F, H, H, O], [AB 427; H, O, Pr, F, H, H, O], [AB 428; H, O, i-Pr, F, H, H, O], [AB429; H, O, CH = CH 2, F, H, H, O], [AB430; H, O, C (CH 3) = CH 2, F, H, H, O] , [AB 431; H, O, C≡CH, F, H, H, O], [AB 432; H, O, C≡ CCH ₃ , F, H, H, O], [AB 433; H, O, c -Pr, F, H, H, O], [AB 434; H, O, OMe, F, H, H, O], [AB 435; H, O, OEt, F, H, H, O], [AB 436 H, O, Oi-Pr, F, H, H, O], [AB 437; H, O, SMe, F, H, H, O], [AB 438; H, O, SE t, F, H, H, O], [AB 439; H, O, CH ₂ F, F, H, H, O], [AB 440; _{H, O, CHF 2, F} , H, H, O], [AB441; H, O, CF 3, F, H, H, O], [AB442; H, O, OCH 2 F, F, H, H, O], [AB443; H, O, OCHF 2, F, H, H, O], [AB444; H, O, OCF 3, F, H, H, O], [AB445; H, O, SCH ₂ F, F, H, H, O], [AB 446; H, O, SCHF ₂ , F, H, H, O], [AB 447; H, O, SCF ₃ , F, H, H, O] , [AB 448; H, O, CN, F, H, H, O], [AB 449; H, O, NO ₂ , F, H, H, O], [AB 450; Me, O, H, F, H , H, O], [AB 451; Me, O, F, F, H, H, O], [AB 452; Me, O, Cl, F, H, H, O], [AB 453; Me, O, Br] , F, H, H, O], [AB 454; Me, O, I, F, H, H, O], [AB 455; Me, O, Me, F, H, H, O], [AB 456; , O, Et, F, H, H, O], [AB 457; Me, O, Pr, F, H, H, O], [AB 458; Me, O, i-Pr, F, H, H, O ], [AB459; Me, O , CH = CH 2, F, H, H, O], [AB460; Me, O, C (CH 3) = CH 2, F, H, H, O], [AB461 Me, O, C≡CH, F, H, H, O], [AB 462; Me, O, C≡CCH ₃ , F, H, H, O], [AB 463; Me, O, c-Pr, F, H, H, O], [AB464; Me, O, OMe, F, H, H, O], [AB 465; Me, O, OEt, F, H, H, O], [AB466; O, Oi-Pr, F, H, H, O], [AB 467; Me, O, SMe, F, H, H, O], [AB 468; Me, O, SEt, F, H, H, O] , [AB 469; Me, O, CH ₂ F, F, H, H, O], [AB 470; Me, O, CHF ₂ , F, H, H, O], [AB 471; Me, O, CF ₃ , F, H, H, O] , [AB472; Me, O, OCH 2 F, F, H, H, O], [AB473; Me, O, OCHF 2, F, H, H, O], [AB474 _{; Me, O, OCF 3,} F, H, H, O], [AB475; Me , O, SCH ₂ F, F, H, H, O], [AB 476; Me, O, SCHF ₂ , F, H, H, O], [AB 477; Me, O, SCF ₃ , F, H, H , O], [AB 478; Me, O, CN, F, H, H, O], [AB 479; Me, O, NO ₂ , F, H, H, O], [AB 480; Et, O, H, F, H, H, O], [AB 481; Et, O, F, F, H, H, O], [AB 482; Et, O, Cl, F, H, H, O], [AB 483; Et, O, Br, F, H, H, O], [AB 484; Et, O, I, F, H, H, O], [AB 485; Et, O, Me, F, H, H, O], [A AB 486; Et, O, Et, F, H, H, O], [AB 487; Et, O, Pr, F, H, H, O], [AB 488; Et, O, i-Pr, F, H, H, O], [AB489; Et, O, CH = CH 2, F, H, H, O], [AB490; Et, O, C (CH 3) = CH 2, F, H, H, O] , [AB 491; Et, O, C≡CH, F, H, H, O], [AB 492; Et, O, C≡ CCH ₃ , F, H, H, O], [AB 493; Et, O, c -Pr, F, H, H, O], [AB 494; Et, O, OMe, F, H, H, O], [AB 495; Et, O, OEt, F, H, H, O], [AB 496 Et, O, Oi-Pr, F, H, H, O], [AB 497; Et, O, SMe, F, H, H, O], [AB 498; Et, O, SEt, F, H, H , O], [AB 499; Et, O, CH ₂ F, F, H, H, O],

[AB500; Et, O, CHF 2, F, H, H, O], [AB501; Et, O, CF 3, F, H, H, O], [AB502; Et, O, OCH 2 F, F , H, H, O], [AB503; Et, O, OCHF 2, F, H, H, O], [AB504; Et, O, OCF 3, F, H, H, O], [AB505; Et , O, SCH ₂ F, F, H, H, O], [AB 506; Et, O, SCHF ₂ , F, H, H, O], [AB 507; Et, O, SCF ₃ , F, H, H , O], [AB 508; Et, O, CN, F, H, H, O], [AB 509; Et, O, NO ₂ , F, H, H, O], [AB 510; H, O, Pr, H, F, H, O] , [AB511; H, O, i-Pr, H, F, H, O], [AB512; H, O, CH = CH 2, H, F, H, O], [AB513; H, O, C (CH 3) = CH 2, H, F, H, O], [AB514; H, O, C≡CH, H, F, H, O], [AB515; H, O, C≡CCH ₃ , H, F, H, O], [AB 516; H, O, c-Pr, H, F, H, O], [AB 517; H, O, OMe, H, F, H , O], [AB518; H, O, OEt, H, F, H, O], [AB519; H, O, Oi-Pr, H, F, H, O], [AB520; H, O, SMe , H, F, H, O], [AB 521; H, O, SE t, H, F, H, O], [AB 522; H, O, CH ₂ F, H, F, H, O], [AB 523] _{; H, O, CHF 2,} H, F, H, O], [AB524; H, O, CF 3, H, F, H, O], [AB525; H, O, OCH 2 F, H, F , H, O], [AB526 ; H, O, OCHF 2, H, F, H, O], [AB527; H, O, OCF 3, H, F, H, O], [AB528; H, O , SCH ₂ F, H, F, H, O], [AB 529; H, O, SCHF ₂ , H, F, H, O], [AB 530; H, O, SCF ₃ , H, F, H, O H, O, CN, H, F, H, O], [AB 532; H, O, NO ₂ , H, F, H, O], [AB 533: Me, O, H, H, F, H, O], [AB 534; Me, O, F, H, F, H, O], [AB 535: Me, O, Cl, H, F, H, O], [AB 536: Me, O, Br, H, F, H, O], [AB 537; Me, O, I, H, F, H, O], [AB 538; Me, O, Me, H, F, H, O], [AB 539; Me, O, Et, H, F, H, O], [AB 540; Me, O, Pr, H, F, H, O], [AB541; Me, O, i-Pr, H, F, H, O], [AB542; Me, O, CH = CH 2, H, F, H, O ], [AB543; Me, O , C (CH 3) = CH 2, H, F, H, O], [AB544; Me, O, C≡CH, H, F, H, O], [AB545; Me, O, C≡CCH ₃ , H, F, H, O], [AB 546; Me, O, c-Pr, H, F, H, O], [AB 547; Me, O, OMe, H, F , H, O], [AB 548; Me, O, OEt, H, F, H, O], [AB 549; Me, O, Oi-Pr, H, F, H, O], [AB 550; Me, O , SMe, H, F, H, O], [AB 551; Me, O, SEt, H, F, H, O], [AB 552; Me, O, CH ₂ F, H, F, H, O], [AB553; Me, O, CHF 2, H, F, H, O], [AB554; Me, O, CF 3, H, F, H, O], [AB555; Me, O, OCH 2 F, H , F, H, O], [AB 556; Me, O, OCHF ₂ , H, F, H, O], [AB 557; Me, O, OCF ₃ , H, F, H, O], [AB 558; Me , O, SCH ₂ F, H, F, H, O], [AB 559; Me, O, SCHF ₂ , H, F, H, O], [AB 560; Me, O, SCF ₃ , H, F, H , O], [AB 561; Me, O, CN, H, F, H, O], [AB 562; Me, O, NO ₂ , H, F, H, O], [AB 563; Et, O, H, H, F, H, O], [AB 564; Et, O, F, H, F, H, O], [AB 565; Et, O, Cl, H, F, H, O], [AB 566; Et, Et, O, Br, H, F, H, O], [AB 567; Et, O, I, H, F, H, O], [AB 568; Et, O, Me, H, F, H, O], [A AB569; Et, O, Et, H, F, H, O], [AB 570; Et, O, Pr, H, F, H, O], [AB 571; Et, O, i-Pr, H, F, H, O], [AB572; Et, O, CH = CH 2, H, F, H, O], [AB573; Et, O, C (CH 3) = CH 2, H, F, H, O] , [AB 574; Et, O, C≡CH, H, F, H, O], [A AB575; Et, O, C≡CCH ₃ , H, F, H, O], [AB 576; Et, O, c-Pr, H, F, H, O], [AB 577; Et, O, OMe, H , F, H, O], [AB 578; Et, O, OEt, H, F, H, O], [AB 579; Et, O, Oi-Pr, H, F, H, O], [AB 580; , O, SMe, H, F, H, O], [AB 581; Et, O, SE t, H, F, H, O], [AB 582; Et, O, CH ₂ F, H, F, H, O ], [AB583; Et, O , CHF 2, H, F, H, O], [AB584; Et, O, CF 3, H, F, H, O], [AB585; Et, O, OCH 2 F , H, F, H, O ], [AB586; Et, O, OCHF 2, H, F, H, O], [AB587; Et, O, OCF 3, H, F, H, O], [AB588 Et, O, SCH ₂ F, H, F, H, O], [AB 589; Et, O, SCHF ₂ , H, F, H, O], [AB 590; Et, O, SCF ₃ , H, F , H, O], [AB 591; Et, O, CN, H, F, H, O], [AB 592; Et, O, NO ₂ , H, F, H, O], [AB 593; H, O, Pr, H, H, F, O], [AB594; H, O, i-Pr, H, H, F, O], [AB595; H, O, CH = CH 2, H, H, F, O ], [AB596; H, O , C (CH 3) = CH 2, H, H, F, O], [AB597; H, O, C≡CH, H, H, F, O], [AB598; H, O, C≡CCH ₃ , H, H, F, O], [AB 599; H, O, c-Pr, H, H, F, O],

[AB600; H, O, OMe, H, H, F, O], [AB601; H, O, OEt, H, H, F, O], [AB 602; H, O, Oi-Pr, H, H , F, O], [AB603; H, O, SMe, H, H, F, O], [AB 604; H, O, SEt, H, H, F, O], [AB 605; H, O, CH ₂ F, H, H, F, O], [AB 606; H, O, CHF ₂ , H, H, F, O], [AB 607; H, O, CF ₃ , H, H, F, O], [AB608; H, O, OCH 2 F, H, H, F, O], [AB609; H, O, OCHF 2, H, H, F, O], [AB610; H, O, OCF 3, H , H, F, O], [AB 611; H, O, SCH ₂ F, H, H, F, O], [AB 612; H, O, SCHF ₂ , H, H, F, O], [AB 613; _{H, O, SCF 3, H} , H, F, O], [AB614; H, O, CN, H, H, F, O], [AB615; H, O, NO 2, H, H, F, O], [AB 616; Me, O, H, H, H, F, O], [AB 617; Me, O, F, H, H, F, O], [AB 618; Me, O, Cl, H, H, F, O], [AB 619; Me, O, Br, H, F, O], [AB 620; Me, O, I, H, H, F, O], [AB 621; Me, O, Me, H, H, F, O], [AB 622; Me, O, Et, H, H, F, O], [AB 623; Me, O, Pr, H, H, F, O], [AB 624; Me, O, i-Pr, H, H, F, O], [AB625; Me, O, CH = CH 2, H, H, F, O], [AB626; Me, O, C (CH 3) = CH ₂ , H, H, F, O], [AB 627; Me, O, C≡CH, H, H, F, O], [AB 628; Me, O, C≡CCH ₃ , H, H, F , O], [AB629; Me, O, c-Pr, H, H, F, O], [AB 630; Me, O, OMe, H, F, O], [AB 631; Me, O, OEt , H, H, F, O], [AB 632; Me, O, Oi-Pr, H, H, F, O], [AB 633; Me, O, SMe, H, H, F, O], [AB 634 Me, O, SEt, H, H, F, O], [AB 635; Me, O, CH ₂ F, H, H, F, O], [AB 636; Me, O, CHF ₂ , H, H, H F, O], [AB637; Me, O, CF 3, H, H, F, O], [AB638 _{; Me, O, OCH 2 F} , H, H, F, O], [AB639; Me, O, OCHF 2, H, H, F, O], [AB640; Me, O, OCF 3, H, H , F, O], [AB 641; Me, O, SCH ₂ F, H, H, F, O], [AB 642; Me, O, SCHF ₂ , H, H, F, O], [AB 643: Me, O, SCF ₃ , H, H, F, O], [AB 644; Me, O, CN, H, H, F, O], [AB 645; Me, O, NO ₂ , H, H, F, O] , [AB 646; Et, O, H, H, H, H, F, O], [AB 647; Et, O, F, H, H, F, O], [AB 648; Et, O, Cl, H, H, F, O], [AB 649; Et, O, Br, H, H, F, O], [AB 650; Et, O, I, H, H, F, O], [AB 651; Et, O, Me, H, H, F, O], [AB 652; Et, O, Et, H, H, F, O], [AB 653; Et, O, Pr, H, H, F, O], [AB 654; Et, O, i-Pr, H, H, F, O], [AB655; Et, O, CH = CH 2, H, H, F, O], [AB656; Et, O, C (CH 3) = CH ₂ , H, H, F, O], [AB657; Et, O, C≡CH, H, H, F, O], [AB658; Et, O, C≡ CCH ₃ , H, H, F, O ], [AB 659; Et, O, c-Pr, H, H, F, O], [AB 660; Et, O, OMe, H, F, O], [AB 661; Et, O, OEt, H , H, F, O], [AB 662; Et, O, Oi-Pr, H, H, F, O], [AB 663; Et, O, SMe, H, H, F, O], [AB 664; , O, SEt, H, H , F, O], [AB665; Et, O, CH 2 F, H, H, F, O], [AB666; Et, O, CHF 2, H, H, F, O], [AB667; Et, O, CF 3, H, H, F, O], [AB668; Et, O, OCH 2 F, H, H, F, O], [AB669; Et, O, OCHF _{2, H, H, F,} O], [AB670; Et, O, OCF 3, H, H, F, O], [AB671; Et, O, SCH 2 F, H, H, F, O], [AB672; Et, O, SCHF 2, H, H, F, O], [AB673; Et, O, SCF 3, H, H, F, O], [AB674; Et, O, CN, H, H , F, O], [AB 675; Et, _{O, NO 2, H, H} , F, O].

[Substituent group number ^{(MB2); E 102],} [BB1; phenyl], [BB2; 2-fluorophenyl], [BB3; 3- fluorophenyl], [BB4; 4-fluorophenyl], [BB5; 2, 3-difluorophenyl], [BB6; 2,4-difluorophenyl], [BB7; 2, 5-difluorophenyl], [BB 8; 2, 6-difluorophenyl], [BB 9; 3,4-difluorophenyl], [BB10; 3,5-Difluorophenyl], [BB11; 2,3,4-Trifluorophenyl], [BB12; 2,3,5-Trifluorophenyl], [BB 13; 2,4,5-Trifluoro Phenyl], [BB14; 2,3,6-trifluorophenyl], [BB15; 2,4,6-trifluorophenyl], [BB16; 3,4,5-trifluorophenyl], [BB17; Chlorophenyl], [BB 18; 4-chlorophenyl], [BB 19; 3,4-dichlorophenyl], [BB 20; 3,5-dichlorophenyl], [BB 21; 3, 4, 5-trichlorophenyl], [BB 22; 3-bromo Phenyl], [BB23; 4-bromophenyl], [BB24; 3,4-dibromophenyl], [BB25; 3,5-dibromofe] [BB26; 3,4,5-tribromophenyl], [BB27; 3-iodophenyl], [BB28; 4-iodophenyl], [BB29; 3,4-diiodophenyl], [BB30; 3,5-diiodophenyl], [BB31; 3,4,5-triiodophenyl], [BB32; 2-fluoro-3-chlorophenyl], [BB33; 2-fluoro-3-bromophenyl], [BB34 2-fluoro-3-iodophenyl], [BB35; 2-fluoro-4-chlorophenyl], [BB36; 2-fluoro-4-bromophenyl], [BB37; 2-fluoro-4-iodophenyl], BB38; 2-fluoro-5-chlorophenyl], [BB 39; 2-fluoro-5-bromophenyl], [BB 40; 2-fluoro-5-iodophenyl], [BB 41; 2-fluoro-6-chlorophenyl], [BB 2-fluoro-6-bromophenyl], [BB 43; 2-fluoro-6-iodophenyl], [BB 44; 3-fluoro-4-chlorophenyl], [BB 45; 3-fluoro-4-bromophenyl], [BB46; 3-fluoro-4-iodophenyl], [BB47; 3-fluoro-5-chloropheny ], [BB 48; 3-fluoro-5-bromophenyl], [BB 49; 3-fluoro-5-iodophenyl], [BB 50; 3-chloro-4-fluorophenyl], [BB 51; 3-chloro-4- Bromophenyl], [BB 52; 3-chloro-4-iodophenyl], [BB 53; 3-chloro-5-bromophenyl], [BB 54; 3-chloro-5-iodophenyl], [BB 55; 3-iodo- 4-fluorophenyl], [BB56; 3-iodo-4-chlorophenyl], [BB57; 3-iodo-4-bromophenyl], [BB58; 3-chloro-4, 5-difluorophenyl], [BB59; 3 -Bromo-4,5-difluorophenyl], [BB60; 3-iodo-4,5-difluorophenyl], [BB61; 3-fluoro-4,5-dichlorophenyl], [BB62; 3-bromo-4,5 -Dichlorophenyl], [BB63; 3-iodo-4,5-dichlorophenyl], [BB64; 3-fluoro-4,5-dibromophenyl], [BB65; 3-chloro-4,5-dibromophenyl], [BB66 3-iodo-4,5-dibromophenyl], [BB 67; 3-fluoro-4, 5-diiodophenyl], [BB 68; 3-chloro; Ro-4,5-diiodophenyl], [BB69; 3-bromo-4,5-diiodophenyl], [BB70; 4-chloro-3,5-difluorophenyl], [BB71; 4-bromo-3 4, 5-Difluorophenyl], [BB 72; 4-iodo-3,5-difluorophenyl], [BB 73; 4-fluoro-3,5-dichlorophenyl], [BB 74; 4-bromo-3,5-dichlorophenyl], [BB 75; 4-iodo-3,5-dichlorophenyl], [BB 76; 4-fluoro-3,5-dibromophenyl], [BB 77; 4-chloro-3,5-dibromophenyl], [BB 78; 4-iodo -3,5-dibromophenyl], [BB 79; 4-fluoro-3,5-diiodophenyl], [BB 80; 4-chloro-3,5-diiodophenyl], [BB 81; 4-bromo-3, 5-diiodophenyl], [BB 82; 2-methylphenyl], [BB 83; 3-methylphenyl], [BB 84; 4-methylphenyl], [BB 85; 2,3-dimethylphenyl], [BB 86; 4-dimethylphenyl], [BB 87; 2, 5-dimethylphenyl], [BB 88; 2, 6-dimethylphenyl], [BB 89; 3,4-dimethylphenyl], [BB 90; 3 , 5-Dimethylphenyl], [BB91; 2,3,4-trimethylphenyl], [BB 92; 2,3,5-trimethylphenyl], [BB 93; 4- (2,2,3,3,3-penta] Fluoropropyl) phenyl], [BB94; 2,3,6-trimethylphenyl], [BB95; 2,4,5-trimethylphenyl], [BB96; 2,4,6-trimethylphenyl], [BB97; 4,5-trimethylphenyl], [BB 98; 2-ethylphenyl], [BB 99; 3-ethylphenyl], [BB 100; 4-ethylphenyl],

[BB101; 2,3-diethylphenyl], [BB102; 2,4-diethylphenyl], [BB103; 2,5-diethylphenyl], [BB104; 2,6-diethylphenyl], [BB105; 3,4 -Diethylphenyl], [BB 106; 3,5-diethylphenyl], [BB 107; 2, 3,4-triethylphenyl], [BB 108; 2, 3, 5-triethylphenyl], [BB 109; -Triethylphenyl], [BB110; 2,4,5-triethylphenyl], [BB111; 2,4,6-triethylphenyl], [BB112; 3,4,5-triethylphenyl], [BB113; 3-propyl] Phenyl], [BB114; 4-propylphenyl], [BB115; 3,4-di-propylphenyl], [BB116; 3,5-di-propylphenyl], [BB117; 3,4,5-tri-propyl] Phenyl], [BB118; 3-isopropylphenyl], [BB119; 4-isopropylphenyl], [BB120; 3,4-diisopropylphenyl], [BB121; 3,5-diisopropylphenyl], [BB122; 5-triisopropylphenyl], [BB 123; 3-butylphenyl], [BB 124; Nyl], [BB 125; 3,4-di-butylphenyl], [BB 126; 3,5-di-butylphenyl], [BB 127; 3-s-butylphenyl], [BB 128; 4-s-butylphenyl] [BB129; 3,4-di-s-butylphenyl], [BB130; 3,5-di-s-butylphenyl], [BB131; 3-isobutylphenyl], [BB132; 4-isobutylphenyl], [BB BB133; 3,4-diisobutylphenyl], [BB134; 3,5-diisobutylphenyl], [BB135; 3-t-butylphenyl], [BB136; 4-t-butylphenyl], [BB 137; 3,4-] Di-t-butylphenyl], [BB 138; 3,5-di-t-butylphenyl], [BB 139; 3-cyclopropylphenyl], [BB 140; 4-cyclopropylphenyl], [BB 141; 3,4- Dicyclopropylphenyl], [BB142; 3,5-dicyclopropylphenyl], [BB143; 3-cyclobutylphenyl], [BB144; 4-cyclobutylphenyl], [BB145; 3,4-dicyclobutylphenyl] ], [BB 146; 3,5-dicyclobutylphenyl], [BB 147; 3-vinylphenyl], [BB 148; Phenyl], [BB149; 3- (1-propenyl) phenyl], [BB150; 4- (1-propenyl) phenyl], [BB151; 3- (2-propenyl) phenyl], [BB152; Propenyl) phenyl], [BB153; 3- (1-butenyl) phenyl], [BB154; 4- (1-butenyl) phenyl], [BB155; 3- (2-butenyl) phenyl], [BB156; 2-butenyl) phenyl], [BB157; 3- (3-butenyl) phenyl], [BB158; 4- (3-butenyl) phenyl], [BB159; 3- (1-methyl-2-propynyl) phenyl], [BB160; 4- (1-methyl-2-propynyl) phenyl], [BB161; 3- (1-ethyl-2-propynyl) phenyl], [BB162; 4- (1-ethyl-2-propynyl) phenyl] , [BB163; 3- (1,1-dimethyl-2-propynyl) phenyl], [BB164; 4- (1,1-dimethyl-2-propynyl) phenyl], [BB165; 3- (1,1-diethyl] -2-propynyl) phenyl], [BB166; 4- (1,1-diethyl-2-propynyl) phenyl], [BB167; 3-ethynylphenyl], [BB168; 4-ethynylphenyl], [BB169; 3- (1-Pro 4- (1-propynyl) phenyl], [BB 171; 3- (2-propynyl) phenyl], [BB 172; 4- (2-propynyl) phenyl], [BB 173; 1-butynyl) phenyl], [BB174; 4- (1-butynyl) phenyl], [BB175; 3- (2-butynyl) phenyl], [BB176; 4- (2-butynyl) phenyl], [BB177; 3 -(3-butynyl) phenyl], [BB 178; 4- (3-butynyl) phenyl], [BB 179; 3- (1-methyl-2-propynyl) phenyl], [BB 180; 4- (1-methyl-2) -Propynyl) phenyl], [BB181; 3-methoxyphenyl], [BB182; 4-methoxyphenyl], [BB183; 3-ethoxyphenyl], [BB184; 4-ethoxyphenyl], [BB185; 3-propyloxyphenyl] ], [BB 186; 4-propyloxyphenyl], [BB 187; 3-isopropyloxyphenyl], [BB 188; 4-isopropyloxyphenyl], [BB 189; 3-cyclopropyloxyphenyl], [BB 190; 4-cyclopropyl] Oxyphenyl], [BB191; 3-butoxypheny ], [BB192; 4-butoxyphenyl], [BB193; 3-s-butoxyphenyl], [BB194; 4-s-butoxyphenyl], [BB195; 3-isobutoxyphenyl], [BB196; 4-isobutoxy Phenyl], [BB 197; 3-t-butoxyphenyl], [BB 198; 4-t-butoxyphenyl], [BB 199; 3,4-dimethoxyphenyl], [BB 200; 3,5-dimethoxyphenyl],

[BB201; 3,4,5-trimethoxyphenyl], [BB202; 3-vinyloxyphenyl], [BB203; 4-vinyloxyphenyl], [BB204; 3- (1-propenyloxy) phenyl], [BB205 4- (1-propenyloxy) phenyl], [BB206; 3- (2-propenyloxy) phenyl], [BB207; 4- (2-propenyloxy) phenyl], [BB208; 3- (1-butenyloxy) Phenyl], [BB209; 4- (1-butenyloxy) phenyl], [BB210; 3- (2-butenyloxy) phenyl], [BB211; 4- (2-butenyloxy) phenyl], [BB212; Butenyloxy) phenyl], [BB213; 4- (3-butenyloxy) phenyl], [BB214; 3- (1-methyl-2-propynyloxy) phenyl], [BB215; 4- (1-methyl-2-propynyloxy] ) Phenyl], [BB216; 3- (1,1-dimethyl-2-propynyloxy) phenyl], [BB217; 4- (1,1-dimethyl-2-propynyloxy) phenyl], [BB218; 1-Methyl-2-butenyloxy) phenyl], [BB 219; 4- (1-methyl) -2-butenyloxy) phenyl], [BB220; 3- (1,1-dimethyl-2-butenyloxy) phenyl], [BB221; 4- (1,1-dimethyl-2-butenyloxy) phenyl], [BB222; 3 -Methoxymethylphenyl], [BB223; 4-methoxymethylphenyl], [BB224; 3-fluoromethylphenyl], [BB225; 4-fluoromethylphenyl], [BB226; 3-difluoromethylphenyl], [BB227; 4 -Difluoromethylphenyl], [BB 228; 3-trifluoromethylphenyl], [BB 229; 4-trifluoromethylphenyl], [BB 230; 3- (1-fluoroethyl) phenyl], [BB 231; 4- (1-) Fluoroethyl) phenyl], [BB232; 3- (2-fluoroethyl) phenyl], [BB233; 4- (2-fluoroethyl) phenyl], [BB234; 3- (1,1-difluoroethyl) phenyl], [BB235; 4- (1,1-difluoroethyl) phenyl], [BB236; 3- (1,2-difluoroethyl) phenyl], [BB237; 4- (1,2-difluoroethyl) phenyl], [BB238 3- (2, 2-di) Fluoroethyl) phenyl], [BB 239; 4- (2, 2-difluoroethyl) phenyl], [BB 240; 3- (1, 1, 2-trifluoroethyl) phenyl], [BB 241; 2-trifluoroethyl) phenyl], [BB 242; 3- (1,2,2-trifluoroethyl) phenyl], [BB 243; 4- (1,2,2-trifluoroethyl) phenyl], [BB 244; 3- (2,2,2-trifluoroethyl) phenyl], [BB245; 4- (2,2,2-trifluoroethyl) phenyl], [BB246; 3- (1,1,2,2-tetra] Fluoroethyl) phenyl], [BB 247; 4- (1,1,2,2-tetrafluoroethyl) phenyl], [BB248; 3-perfluoroethylphenyl], [BB249; 4-perfluoroethylphenyl], [BB BB 250; 3- (1-fluoropropyl) phenyl], [BB 251; 4- (1-fluoropropyl) phenyl], [BB 252; 3- (2-fluoropropyl) phenyl], [BB 253; 4- (2-fluoro) Propyl) phenyl], [BB254; 3- (3-fluoropropyl) phenyl], [BB255; 4- (3-fluoropropyl) phenyl] , [BB256; 3- (1,1-difluoropropyl) phenyl], [BB 257; 4- (1,1-difluoropropyl) phenyl], [BB258; 3- (1,2-difluoropropyl) phenyl], [BB BB 259; 4- (1,2-difluoropropyl) phenyl], [BB 260; 3- (1,3-difluoropropyl) phenyl], [BB 261; 4- (1,3-difluoropropyl) phenyl], [BB 262; 3- (2,2-difluoropropyl) phenyl], [BB 263; 4- (2, 2-difluoropropyl) phenyl], [BB 264; 3- (2,3-difluoropropyl) phenyl], [BB 265; (2,3-difluoropropyl) phenyl], [BB 266; 3- (3, 3-difluoropropyl) phenyl], [BB 267; 4- (3, 3- difluoropropyl) phenyl], [BB 268; 1,2-trifluoropropyl) phenyl], [BB 269; 4- (1,1,2-trifluoropropyl) phenyl], [BB 270; 3- (1,1,3-trifluoropropyl) phenyl], [BB 271; 4- (1,1,3-trifluoropropyl) phenyl], [BB 272; 3- (1,2,2-trifluoropropyl) Phenyl], [BB 273; 4- (1, 2, 2- trifluoropropyl) phenyl], [BB 274; 3- (1, 2, 3- trifluoropropyl) phenyl], [BB 275; , 3-trifluoropropyl) phenyl], [BB 276; 3- (1,3,3-trifluoropropyl) phenyl], [BB 277; 4- (1,3,3-trifluoropropyl) phenyl], [BB 278 3- (2,2,3-trifluoropropyl) phenyl], [BB279; 4- (2,2,3-trifluoropropyl) phenyl], [BB280; 3- (2,3,3-trifluoro] Propyl) phenyl], [BB 281; 4- (2, 3, 3- trifluoropropyl) phenyl], [BB 282; 3- (3, 3, 3- trifluoropropyl) phenyl], [BB 283; 3,3,3-Trifluoropropyl) phenyl], [BB 284; 3- (1,1,2,2-tetrafluoropropyl) phenyl], [BB 285; 4- (1,1,2,2-tetrafluoropropyl] ) Phenyl], [BB 286; 3- (1, 1, 3, 3- tetrafluoropropyl) phenyl], [BB 287; 4- (1, 1, 3, 3- tetrafluoropropyl) phenyl], [BB 288; -(2, 2, 3, 3-te Trafluoropropyl) phenyl], [BB 289; 4- (2,2,3,3-tetrafluoropropyl) phenyl], [BB290; 3- (1,1,3,3,3-pentafluoropropyl) phenyl] , [BB 291; 4- (1,1,3,3,3-pentafluoropropyl) phenyl], [BB292; 3- (2,2,3,3,3-pentafluoropropyl) phenyl], [BB293; 3- (1,1,2,2,3,3-hexafluoropropyl) phenyl], [BB 294; 4- (1,1,2,2,3,3-hexafluoropropyl) phenyl], [BB 295; 3-perfluoropropylphenyl], [BB 296; 4-perfluoropropylphenyl], [BB 297; 3-perfluoropropylphenyl], [BB 298; 4-perfluoropropylphenyl], [BB 299; 3- [2, 2 , 2-trifluoro-1- (trifluoromethyl) ethylphenyl], [BB 300; 4- [2,2,2-trifluoro-1- (trifluoromethyl) ethylphenyl],

[BB301; 3- [1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylphenyl], [BB302; 4- [1,2,2,2-tetrafluoro-1- (trifluoro) Methyl) ethylphenyl], [BB 303; 3-perfluorobutylphenyl], [BB 304; 4-perfluorobutylphenyl], [BB 305; 3- [1, 2, 2, 3, 3, 3-hexafluoro-1] -(Trifluoromethyl) propylphenyl], [BB306; [1,2,2,3,3,3-hexafluoro-1- (trifluoromethyl) propylphenyl], [BB307; 3- [1,1,6 2,3,3,3-hexafluoro-2- (trifluoromethyl) propylphenyl], [BB 308; 4- [1,1,2,3,3,3-hexafluoro-2- (trifluoromethyl) Propylphenyl], [BB309; 5-fluoro-3-trifluoromethylphenyl], [BB310; 6-fluoro-3-trifluoromethylphenyl], [BB311; 2,4-difluoro-3-trifluoromethylphenyl] , [BB 312; 2, 5-difluoro-3-trifluoromethylphenyl], [BB 313; 2, 6-di Fluoro-3-trifluoromethylphenyl], [BB 314; 4, 5-difluoro-3- trifluoromethylphenyl], [BB 315; 4, 6-difluoro-3- trifluoromethylphenyl], [BB 316; -Difluoro-3-trifluoromethylphenyl], [BB 317; 2,4,5-trifluoro-3-trifluoromethylphenyl], [BB 318; 2,4,6-trifluoro-3-trifluoromethylphenyl] , [BB319; 4,5,6-trifluoro-3-trifluoromethylphenyl], [BB320; 2,4,5,6-tetrafluoro-3-trifluoromethylphenyl], [BB321; 4-chloro- 3-trifluoromethylphenyl], [BB 322; 5-chloro-3-trifluoromethylphenyl], [BB 323; 4-methyl-3-trifluoromethylphenyl], [BB 324; 5-methyl-3-trifluoromethyl Phenyl], [BB 325; 4-ethyl-3-trifluoromethylphenyl], [BB 326; 5-ethyl-3-trifluoromethylphenyl], [BB 327; -3-trifluoromethylphenyl], [BB 328; 5-cyclopropyl-3-trifluoromethylphenyl], [BB 329; 4-methoxy-3-trifluoromethylphenyl], [BB 330; Fluoromethylphenyl], [BB331; 3-fluoromethoxyphenyl], [BB332; 4-fluoromethoxyphenyl], [BB333; 3-difluoromethoxyphenyl], [BB334; 4-difluoromethoxyphenyl], [BB335; Trifluoromethoxyphenyl], [BB 336; 4-trifluoromethoxyphenyl], [BB 337; 3- (1-fluoroethoxy) phenyl], [BB 338; 4- (1-fluoroethoxy) phenyl], [BB 339; 3- (2-fluoroethoxy) phenyl], [BB340; 4- (2-fluoroethoxy) phenyl], [BB341; 3- (1,1-difluoroethoxy) phenyl], [BB342; 4- (1,1-difluoro) Ethoxy) phenyl], [BB 343; 3- (1,2-difluoroethoxy) phenyl], [BB 344; 4- (1,2-difluoroethoxy) phenyl] Phenyl], [BB 345; 3- (2, 2-difluoroethoxy) phenyl], [BB 346; 4- (2, 2- difluoroethoxy) phenyl], [BB 347; 3- (1, 1, 2- trifluoroethoxy) ) Phenyl], [BB 348; 4- (1,1,2-trifluoroethoxy) phenyl], [BB 349; 3- (1,2,2-trifluoroethoxy) phenyl], [BB 350; 2,2-trifluoroethoxy) phenyl], [BB 351; 3- (2,2,2-trifluoroethoxy) phenyl], [BB 352; 4- (2,2,2-trifluoroethoxy) phenyl], [ BB 353; 3- (1,1,2,2-tetrafluoroethoxy) phenyl], [BB 354; 4- (1,1,2,2-tetrafluoroethoxy) phenyl], [BB 355; 3- (perfluoroethoxy) ) Phenyl], [BB 356; 4- (perfluoroethoxy) phenyl], [BB 357; 3- (1- fluoropropyloxy) phenyl], [BB 358; 4- (1- fluoropropyloxy) phenyl], [BB 359; 3- (2-fluoropropyloxy) phenyl], [BB 360; 4- (2-fluoropropyloxy) pheny ], [BB 361; 3- (3-fluoropropyloxy) phenyl], [BB 362; 4- (3-fluoropropyloxy) phenyl], [BB 363; 3- (1,1-difluoropropyloxy) phenyl], [BB 361; BB 364; 4- (1,1-difluoropropyloxy) phenyl], [BB365; 3- (1,2-difluoropropyloxy) phenyl], [BB 366; 4- (1,2-difluoropropyloxy) phenyl], [BB 367; 3- (1,3-difluoropropyloxy) phenyl], [BB 368; 4- (1,3-difluoropropyloxy) phenyl], [BB 369; 3- (2,2-difluoropropyloxy) phenyl] [BB 370; 4- (2, 2-difluoropropyloxy) phenyl], [BB 371; 3- (2,3-difluoropropyloxy) phenyl], [BB 372; 4- (2,3-difluoropropyloxy) phenyl ], [BB 373; 3- (3, 3-difluoropropyloxy) phenyl], [BB 374; 4- (3, 3- difluoropropyloxy) phenyl], [BB 375; 3- (1, 1, 2-trifluoro) Propyloxy) pheny ], [BB 376; 4- (1,1,2-trifluoropropyloxy) phenyl], [BB 377; 3- (1,1,3-trifluoropropyloxy) phenyl], [BB 378; 1,3-trifluoropropyloxy) phenyl], [BB379; 3- (1,2,2-trifluoropropyloxy) phenyl], [BB380; 4- (1,2,2-trifluoropropyloxy) phenyl ], [BB 381; 3- (1,2,3-trifluoropropyloxy) phenyl], [BB 382; 4- (1,2,3-trifluoropropyloxy) phenyl], [BB 383; 3- (1, 1 3,3-trifluoropropyloxy) phenyl], [BB 384; 4- (1,3,3-trifluoropropyloxy) phenyl], [BB 385; 3- (2,2,3-trifluoropropyloxy) phenyl ], [BB 386; 4- (2,2,3-trifluoropropyloxy) phenyl], [BB 387; 3- (2,3,3-trifluoropropyloxy) phenyl], [BB 388; 4- (2, 3,3-Trifluoropropyloxy) phenyl], [BB 389; 3- (3,3,3-trifluoropropyloxy) ester Phenyl], [BB390; 4- (3,3,3-trifluoropropyloxy) phenyl], [BB391; 3- (1,1,2,2-tetrafluoropropyloxy) phenyl], [BB392; 4- (1,1,2,2-tetrafluoropropyloxy) phenyl], [BB 393; 3- (1,1,3,3-tetrafluoropropyloxy) phenyl], [BB 394; 4- (1,1,3) , 3-Tetrafluoropropyloxy) phenyl], [BB 395; 3- (2,2,3,3-tetrafluoropropyloxy) phenyl], [BB 396; 4- (2,2,3,3-tetrafluoropropyl] Oxy) phenyl], [BB 397; 3- (1,1,3,3,3-pentafluoropropyloxy) phenyl], [BB 398; 4- (1,1,3,3,3-pentafluoropropyloxy) Phenyl], [BB 399; 3- (2,2,3,3,3-pentafluoropropyloxy) phenyl], [BB400; 4- (2,2,3,3,3-pentafluoropropyloxy) phenyl] ,

[BB 401; 3- (1,1,2,2,3,3-hexafluoropropyloxy) phenyl], [BB402; 4- (1,1,2,2,3,3-hexafluoropropyloxy) phenyl ], [BB 403; 3-perfluoropropyloxyphenyl], [BB 404; 4-perfluoropropyloxyphenyl], [BB 405; 3- (2,2,2,2,2,2-hexafluoroisopropyloxy) phenyl ], [BB406; 4- (2,2,2,2,2,2-hexafluoroisopropyloxy) phenyl], [BB407; 3-perfluoroisopropyloxyphenyl], [BB408; 4-perfluoroisopropyloxyphenyl] ], [BB 409; 3-perfluoro-butyloxyphenyl], [BB 410; 4-perfluoro-butyloxyphenyl], [BB 411; 3-perfluoro-s-butyloxyphenyl], [BB 412; 4-perfluoro] -s-butyloxyphenyl], [BB 413; 3-perfluoro-isobutyloxyphenyl], [BB 414; 4-perfluoro-isobutyloxyphenyl], [BB 415 4-chloro-3-trifluoromethoxyphenyl], [BB 416; 5-chloro-3-trifluoromethoxyphenyl], [BB 417; 4-methyl-3-trifluoromethoxyphenyl], [BB 418; 5-methyl-3 -Trifluoromethoxyphenyl], [BB 419; 4-ethyl-3-trifluoromethoxyphenyl], [BB 420; 5-ethyl-3-trifluoromethoxyphenyl], [BB 421; 4-cyclopropyl-3-trifluoromethoxy Phenyl], [BB 422; 5-cyclopropyl-3-trifluoromethoxyphenyl], [BB 423; 4-methoxy-3-trifluoromethoxyphenyl], [BB 424; 5-methoxy-3-trifluoromethoxyphenyl], [BB BB 425; 3-nitrophenyl], [BB 426; 4-nitrophenyl], [BB 427; 3-cyanophenyl], [BB 428; 4-cyanophenyl], [BB 429; 3-methylthiophenyl], [BB 430; 4-methylthio Phenyl], [BB 431; 3-trifluoromethylthiophenyl], [BB 432; 4-thiophenyl], [BB 433; 3- (methylamino) phenyl], [BB 436; 4- (methylamino) phenyl], [BB 437; -(Dimethylamino) phenyl], [BB 438; 4- (dimethylamino) phenyl], [BB 439; 3- (ethylamino) phenyl], [BB 440; 4- (ethylamino) phenyl], [BB 441; Diethylamino) phenyl], [BB 442; 4- (diethylamino) phenyl], [BB 443; 3- (ethylmethylamino) phenyl], [BB 444; 4- (ethylmethylamino) phenyl], [BB 445; 3- (propylamino) ) Phenyl], [BB 446; 4- (propylamino) phenyl], [BB 447; 3- (propylamino) phenyl], [BB 448; 4- (propylamino) phenyl], [BB 449; 3- (isopropylamino) phenyl ], [BB 450; 4- (isopropylamino) phenyl], [BB 451; 3- (diisopropylamino) phenyl], [BB 452; 4- (diisopropylamino) phenyl], [BB 453; 4-hydroxyphenyl], [BB 455; 3-methylthiophenyl], [BB 456; 4-methylthiophenyl], [BB 457; 3- (fluoromethylamino) phenyl], [BB 458; (Fluoromethylamino) phenyl], [BB 459; 3- (difluoromethylamino) phenyl], [BB 460; 4- (difluoromethylamino) phenyl], [BB 461; 3- (trifluoromethylamino) phenyl], [BB 462 4- (trifluoromethylamino) phenyl], [BB463; 3-methylcarbonylphenyl], [BB464; 4-methylcarbonylphenyl], [BB465; 3-ethylcarbonylphenyl], [BB466; 4-ethylcarbonylphenyl ], [BB 467; 3-methoxycarbonylphenyl], [BB 468; 4-methoxycarbonylphenyl], [BB 469; 3-ethoxycarbonylphenyl], [BB 470; 4-ethoxycarbonylphenyl], [BB 471; 3-aminocarbonylphenyl] ], [BB 472; 4-amino carbonyl fe N, N, N, B: BB473; 3-methylaminocarbonylphenyl, BB474; 4-methylaminocarbonylphenyl, BB 475; 3- (formylamino) phenyl !, BB 476; 4- (N-formylamino) phenyl] [BB 477; 3- (N-formyl-N-methylamino) phenyl], [BB 478; 4- (N-formyl-N-methylamino) phenyl], [BB 479; 3-trimethylsilylphenyl], [BB 480; -Trimethylsilylphenyl], [BB 481; 1-naphthyl], [BB 482; 2-naphthyl], [BB 483; indan-1-yl], [BB 484; indan-2-yl], [BB 485; 5, 6, 7, 7, 8-tetrahydronaphthalen-1-yl], [BB 486; 5, 6, 7, 8, 8-tetrahydronaphthalen-2-yl], [BB 487; 1-cyclohexenyl], [BB 488; cyclohexyl], [BB 489; -1-cyclohexenyl], [BB 490; 2-methyl-1-cyclohexenyl], [BB 491; 4-chloro-1-cyclohexenyl], [BB 492; 4-methyl-1-cyclohexenyl], [BB 493; -Chloro-1-cyclohexenyl ], [BB 494; 6-methyl-1-cyclohexenyl], [BB 495; 3-chloro-1-cyclohexenyl], [BB 496; 3-methyl-1-cyclohexenyl], [BB 497; 3-methoxy-1-cyclohexenyl] Cyclohexenyl], [BB 498; 3- (trifluoromethyl) -1-cyclohexenyl], [BB 499; 3- (difluoromethyl) -1-cyclohexenyl], [BB 500; 3- (trifluoromethoxy) -1-] Cyclohexenyl],

[BB501; 5-chloro-1-cyclohexenyl], [BB 502; 5-methyl-1-cyclohexenyl], [BB 503; 5-methoxy-1-cyclohexenyl], [BB 504; 5- (trifluoromethyl)- 1-cyclohexenyl], [BB 505; 5- (difluoromethyl) -1-cyclohexenyl], [BB 506; 5- (trifluoromethoxy) -1-cyclohexenyl], [BB 507; 1-butenyl], [BB 508; 3-Methyl-1-butenyl], [BB509; 4-chloro-3-chloromethyl-1-butenyl], [BB510; 3-chlorocyclohexyl], [BB511; 3-trifluoromethylcyclohexyl].

  The substituent numbers (MB2) BB1001 to BB3016 are described below.

The substituent number (MB2) BB1001 to BB3016 represents one of the following E201 to E262. Represents a binding site. ). For example, in the following E201, R ⁴⁰¹ is a fluorine atom, and R ⁴⁰² , R ⁴⁰³ , R ⁴⁰⁴ , R ⁴⁰⁵ , R ⁴⁰⁶ , R ⁴⁵⁰ , R ⁴⁵¹ , and R ⁴⁵² are hydrogen in the following E201: Represents a group that is an atom.

[Substituent No. (MB2); E ¹⁰² ], [BB 1001; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1002; E 201, E ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1003; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1004; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1005; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1006; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1007; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1008; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1009; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1010; E 201, E ^401, H ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H , R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1011; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1012 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB1013; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1014; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H] [BB 1015; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1016; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1017; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1018; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1019; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1020; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H , R ⁴⁵² : H], [BB 1021; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1022; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1023; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H , R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1024; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1025; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1026; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1027; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1028; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1029; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1030; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1031; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1032; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1033; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H , R ⁴⁵² : H], [BB 1034; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1035; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1036; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1037; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1038; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1039; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1040; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1041; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1042; E 201, R ⁴⁰¹ : H, R ^{4 02} : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1043; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1044; E201, R ⁴⁰¹ : F , R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1045; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1046; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1047; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1048; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1049; E 201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1050; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1051 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB1052; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1053; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, ^{R 406: Cl, R 450:} Cl, R 451: H, R 452: H], [BB1054; E201, R 401: H, R 402: H, R 403: Br, R 404: H, R 405: H , R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1055; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1056; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1057; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1058; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵
: H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1059; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1060; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1061; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1062; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1063; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1064; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1065; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1066; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F , R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1067; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1068; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1069; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H , R ⁴⁵² : H], [BB 1070; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1071; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1072; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1073; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1074; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : Br , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1075; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1076; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1077; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1078; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1079; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1080; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1081; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1082; E201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1083; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1084 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1085; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1086; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H] [BB 1087; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1088; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1089; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1090; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1091; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1092; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1093; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1094; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl , R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1095; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1096; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1097; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1098; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1099; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : Me , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1100; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H],

[BB1101; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H] [BB 1102; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB1103; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1104; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1105; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1106; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H , R ⁴⁵² : H], [BB 1107; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1108; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1109; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1110; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ^{450 _{: CF 3, R 451: H}} , R 452: H], [BB1111; E201, R 4 ⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1112; E 201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1113 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1114; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1115; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1116; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1117; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1118; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1119; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1120; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1121; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1122; E 201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1123 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1124; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1125; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1126; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1127; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H , R ⁴⁵² : H], [BB 1 128; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1129; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1130; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1131; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1132; E 201, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1133; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1134; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1135; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1136; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1137; E 201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1138; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1139 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1140; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1141; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1142; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1143; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H , R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1144; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1145; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1146; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1147; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1148; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1149; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1150; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1151; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1152; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1153; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1154; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1155; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1156; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ^40
4 : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1157; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl , R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1158; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1159; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1160; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1161; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1162; E201, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1163; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1164; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1165; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1166; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1167; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1168; E 201, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1169; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1170; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1171; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1172; E201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1173; E201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1174 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB1 175; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1176; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ^{4 04} : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1177; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1178; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl , R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1179; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1180; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1181; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1182; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1183; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1184; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1185; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1186; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1187; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me , R ⁴⁰⁶ : Me, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1188; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1189; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1190; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB1191; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB1192; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H , R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1193; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1194; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1195; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1196; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H] [BB 1197; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H ], [BB 1198; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1 199; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1200; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H],

[BB 1201; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H] [BB1202; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H ], [BB1203; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1204; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1205; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1206; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1207; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F , R ⁴⁵² : H], [BB 1208; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1209; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1210; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1211; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ^{4 03} : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1212; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1213; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1214; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1215; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1216; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1217; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1218; E 201, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1219; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1220; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1221; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1222; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1223; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1224; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1225; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1226; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1227; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1228; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H , R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1229; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1230; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1231; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1232; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1233; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1234; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br , R ⁴⁵² : H], [BB 1235; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1236; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1237; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1238; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1239; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H , R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1240; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1241; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1242; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1243; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1244; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1245; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1246; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1247; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1248; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1249; E 201, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1250; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1251; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1252; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1253; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1254; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1 255; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1256; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1257; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1258; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H
, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1259; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1260; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1261; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1262; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1263; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1264; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1265; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1266; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1267; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1268; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me , R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : M e, R ⁴⁵² : H], [BB 1269; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1270; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1271; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1272; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H , R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1273; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1274; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1275; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1276; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1277; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1278; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H , R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1 279; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H] [BB 1280; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1281; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB1282; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1283; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1284; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R _{^{451: CF 3, R 452:}} H], [BB1285; E201, R 401: H, R 402: H, R 403: Br, R 404: H, R 405: H, R 406: H, R 450: H , R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1286; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1287; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1288; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [B B1289; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H] [BB1290; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1291; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ^{452: H], [BB1292;} E201, R 401: H, R 402: H, R 403: H, R 404: H, R 405: Me, R 406: Me, R 450: H, R 451: CF 3 , R ⁴⁵² : H], [BB 1293; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1294; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R _{^{451: CF 3, R 452:}} H], [BB1295; E201, R 401: H, R 402: H, R 403: H, R 404: H, R 405: H, R 406: H, R 450: H , R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1296; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1297; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1298; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1299; E 2 01, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1300 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H],

[BB1301; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H] [BB1302; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H ], [BB1303; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB1304; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1305; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1306; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1307; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe , R ⁴⁵² : H], [BB 1308; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1309; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1310; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1311; E 201, R ^{40 1} : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1312; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1313; E 201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1314; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1315 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [ BB 1316; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H] ^{, [BB1317; E201, R 401} : F, R 402: H, R 403: H, R 404: H, R 405: H, R 406: H, R 450: H, R 451: OCF 3, R 452: H], [BB1318; E201, R 401: H, R 402: H, R 403: F, R 404: H, R 405: H, R 406: H, R 450: H, R 451: OCF 3, R ⁴⁵² : H], [BB 1319; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1320; E 201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1321; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1322; E 201, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1323; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1324; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1325; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [ BB 1326; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H] [BB1327; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1328; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1329; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1330; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1331; E 20 1, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [ BB1332; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H] ^{, [BB1333; E201, R 401} : H, R 402: H, R 403: Me, R 404: Me, R 405: H, R 406: H, R 450: H, R 451: OCF 3, R 452: H], [BB 1334; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1335; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1336; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1337; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1338; E 201, R ⁴⁰¹ : F, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1339; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H , R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1340; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB1341; E201, R ⁴⁰¹ : F, R ⁴⁰² : F, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB1342; E201 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB1343; E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1344 E201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [ BB 1345; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1346; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H] [BB 1347; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H ], [BB 1348; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1349; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1350; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Br, R ⁴⁰⁴ : Br, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1351; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Br, R ⁴⁰⁶ : Br, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1352; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1353; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1354; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1355; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1356; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : OMe, R ⁴⁰⁴ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰
: H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1357; E 201, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁵ : OMe, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1358; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1359; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1 360; E202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1361; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1362; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1363; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1364; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1365; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1366; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1367; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1368; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1369; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1370; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1371; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : F , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1372; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1373; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1374; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1375; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1376; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl , R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1377; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : ^{H, R 452: H],} [BB1378; E202, R 401: H, R 402: H, R 403: Me, R 404: Me, R 450: Cl, R 451: H, R 452: H], [ BB 1379; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1380; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1381; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F , R ⁴⁰⁴ : F, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB1382; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1383; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1384; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me , R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1385; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1386; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1387; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1388; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1389; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1390; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1391; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ^{451 : H, R 452: H]} , [BB1392; E202, R 401: H, R 402: H, R 403: Me, R 404: Me, R 450: Me, R 451: H, R 452: H], [BB 1393; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1394; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1395; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1396; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1397; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1398: E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1399; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1400; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H],

[BB 1401; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1402; E 202, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1403; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1404; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1405; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1406; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1407; E 202 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1408; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1409; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1410; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1411; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1412; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1413 E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1414; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H , R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1415; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1416; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1417; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1418; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1419; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1420; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1421; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1422; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1423; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1424; E 202, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1425; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ^{4 52} : H], [BB 1426; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1427; E 202 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1428; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1429; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1430; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1431; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H] [BB 1432; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1433; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1434; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1435; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1436; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1437; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1438; E202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1439; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br , R ⁴⁵² : H], [BB 1440; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1441 E202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1442; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1443; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1444; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H , R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1445; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1446; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1447; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1448; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1449; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1450; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1451; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB1452; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1453; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1454; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R _{^{451: CF 3, R 452:}} H], [BB1455; E202, R 401: H, R 402: H, R 403: Me, R 404: Me, R 450: H, R 451: CF 3, R 452: H], [BB 1456; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1457; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1458; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1459; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1460; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : ^{OMe, R 452: H],} [BB1461; E202, R 401: H, R 402: H, R 403: Me, R 404: H, R 450: H, R 451: OMe, R 452: H], [ BB 1462; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1463; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1464; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1465; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H ], [BB 1466; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1467; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1468; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1469; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1470; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1471; E 202, R ⁴⁰¹ : H,
R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : S Me, R ⁴⁵² : H], [BB 1472; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F , R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1473; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1474; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1475; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1476; E 202, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1477; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1478; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1479; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1480; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1481; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1482; E 203, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1483; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1484; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1485; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1486; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1487; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H , R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1488; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1489; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1490; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1491; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1492; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F , R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1493; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1494; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1495; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1496; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1497; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1498; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1499; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1500; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H],

[BB 1501; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1502; E 203, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1503; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1504; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : Br, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1505; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1506; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1507; E203 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1508; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1509; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1510; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1511; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H] [BB 1512; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1513; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1514; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1515; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H] [BB 1516; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1517; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1518; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1519; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1520; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1521; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1522; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1523; E 203, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1524; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1525; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1526; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1527; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1528; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1529; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1530; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1531; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1532; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1533; E 203 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1534; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1535; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1536; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1537; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H] , [BB1538; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1539; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1540; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1541; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1542; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1543; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1544; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB1545; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ^{404: H, R 450: H} , R 451: F, R 452: H], [BB1546; E203, R 401: H, R 402: H, R 403: Me, R 404: Me, R 450: H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1547; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H ], [BB 1548; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1 549; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB1550; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [ BB 1551; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1552; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1553; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me , R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1554; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1555; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1556; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1557; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1558; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1559; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1560; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Br, R ⁴⁵² : H], [BB 1561; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB1562; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1563; E 203, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1564; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB1 565; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1 566; E 203 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB1567; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1568; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1569; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1570; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1571; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ^4
50 : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1572; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1573; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1574; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1575: E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1576; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1577; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1578; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1579; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1580; E203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1581; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1582; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1583; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H , R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1584; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1585; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1586; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1587; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1588; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1589; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H] [BB 1590; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1591; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB1592; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1593; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1594; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1595; E 203, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1596; E 204, R ⁴⁰¹ : H, R ^{4 02} : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1597; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1598; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F , R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1599; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1600; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H],

[BB 1601; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1602; E 204 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1603; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1604, E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1605; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1606; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1607; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl , R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1608; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1609; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1610; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1611; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1612; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1613; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1614; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1615; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1616; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : c-Pr, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1617; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1618; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1619; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1620; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1621; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1622; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB1623; E204, R 401: H, R 402: H, R 403: Me, R 404: Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1624; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1625; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1626; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1627; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1628; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1629; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1630; E 204 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : F, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1631; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1632; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1633; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1634; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1635; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1636; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1637; E 204 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1638; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1639; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1640; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1641; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1642; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl , R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1643; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1644; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1645; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1646; E 204, R ^{40 1} : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1647; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1648; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1649; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1650; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1651; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1652; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1653; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1654; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1655; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1656; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1657; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me , R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1658; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1659; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1660; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1661; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1662; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1663; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1664; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³
: Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1665; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1666; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1667; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1668; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et , R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1669; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ^{450 _{: CF 3, R 451: H}} , R 452: H], [BB1670; E204, R 401: H, R 402: H, R 403: Cl, R 404: Cl, R 407: Et, R 450: CF 3 , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1671; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1672; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1673; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H ], [BB 1674; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1675 E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1676; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl , R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1677; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1678; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1679; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1680; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1681; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H , R ⁴⁵² : H], [BB1682; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1683; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1684; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1685; E 204, E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1686; E 204, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1687; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1688; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me , R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1689; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1690; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1691; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB1692; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H] [BB 1693; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1694; E204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1695; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB1696; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1697; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1698; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H], [BB 1699; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H] [BB1700; E204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : F, R ⁴⁵² : H],

[BB 1701; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1702; E 204 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1703; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1704; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1705; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1706; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1707; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me , R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1708; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1709; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1710; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1711; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1712; E 204, R ⁴⁰¹ : H, R ^{4 02} : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1713; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1714; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me , R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1715; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1716; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1717; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1718; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1719; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me , R ⁴⁵² : H], [BB 1720; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB1721; E204, R 401: H, R 402: H, R 403: Me, R 404: Me, R 407: Me, R 450: H, R 451: Me, R 452: H], [ BB 1722; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1723; E 204, E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1724; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1725; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1726; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H , R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1727; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1728; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : Me, R ⁴⁵² : H], [BB 1729; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H] [BB 1730; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1731 E204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1732; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1733; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1734; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ^{40 7} : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1735; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Me , R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1736; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1737; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1738; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1739; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1740; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1741; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1742; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1743; E204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1744; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1745; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F , R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1746; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1747; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1 748; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ^{451: OMe, R 452: H} ], [BB1749; E204, R 401: H, R 402: H, R 403: Me, R 404: Me, R 407: Me, R 450: H, R 451: OMe, R ⁴⁵² : H], [BB 1750; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H ], [BB 1751; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1752 E204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1753; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1754; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1755; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰³ : Me, R ⁴⁰⁴ : H, R ⁴⁰⁷ : Et, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1756; E 204, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁰⁷ : E t, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1757; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1758; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1759; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1760; E 205, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1761; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1762; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1763; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1764; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ :
F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1765; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1766; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1 767; E205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1 768; , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1769; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1770; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1771; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1772; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H] [BB1773; E205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1774; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1775; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1776; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [B B1777; E205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1778; E 205, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1779; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1780; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1781; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1782; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [ BB 1783; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1784; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1785; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me , R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1786; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1787; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1 788; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1 789; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1790; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1791; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H ], [BB 1792; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1793; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1794; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1795; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1796; E 205, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R _{^{451: CF 3, R 452:}} H], [BB1797; E205, R 401: H, R 402: H, R 405: Me, R 406: H, R 450: H, R 451: CF 3, R 452: H], [BB 1798; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1799; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1800; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H],

[BB 1801; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1802; E 206, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1803; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1804; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1805; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1806; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1807; E 206 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1808; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1809; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1810; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1811; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H] [BB 1812; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1813; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1814; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1815; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1816; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1817; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H , R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1818; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1819; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1820; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1821; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1822; E 206 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1823; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1824; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1825; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1826; E 2 06, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1827; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1828; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1829; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1830; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H ], [BB 1831; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1832; E 206, R ^401] : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1833; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1834; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1835; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1836; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1837; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1838; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Cl, R ⁴⁰⁶ : C l, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1839; E 206, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R _{^{451: CF 3, R 452:}} H], [BB1840; E206, R 401: H, R 402: H, R 405: Me, R 406: Me, R 450: H, R 451: CF 3, R 452: H], [BB 1841; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1842; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1843; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1844; E 207, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1845; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1846; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1847; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1848; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1849; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁰⁸ : Me , R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1850; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1851; E207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1852; E 207, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : Me, R ⁴⁰⁶ : Me, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1853; E 208, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1854; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1855; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1856; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1 857; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1858 E208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1859; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1860; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1861; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1862; E 2 08, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1863; E 208, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1864; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1865; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1866; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1867; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1868; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1869; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ^{4
51: H, R 452: H} ], [BB1870; E209, R 401: H, R 402: H, R 403: H, R 404: H, R 450: H, R 451: Cl, R 452: H] , [BB 187 1; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 187 2; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1873; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1874; E 209, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1875; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1876; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1877; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1878; E 210, R ⁴⁰¹ : H , R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1879; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1880; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1881; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1 882; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1883; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1884; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1885; E 210, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H] [BB 1886; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1887; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1888; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1889; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1890; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OCF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1891; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB1892; E211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1893; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1894; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1895; E 211, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OCF ₃ , R ⁴⁵² : H], [BB 1896; E 211 , R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1897; E 212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1898; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [ BB 1899; E 212, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1900; E 212, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H],

[BB1901; E212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1902; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : Cl , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1903; E 212, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1904; E 212, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1905; E 212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1906; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1907; E 212, R ⁴⁰³ : Cl, R ^{404 _{: Cl, R 450: CF 3}} , R 451: H, R 452: H], [BB1908; E212, R 403: Me, R 404: Me, R 450: CF 3, R 451: H, R 452: H ], [BB 1909; E 212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1910; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ^450] : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1911; E 212, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1912; E 212, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1913; E 212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl , R ⁴⁵² : H], [BB 1914; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1915; E 212, R ⁴⁰³ : Cl, R ^{404 : Cl, R 450: H,} R 451: Cl, R 452: H], [BB1916; E212, R 403: Me, R 404: Me, R 450: H, R 451: Cl, R 452: H], [BB 1917; E212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1918; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1919; E 212, R ⁴⁰³ : Cl, R ⁴⁰⁴ : Cl, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1920; E 212, R ⁴⁰³ : Me, R ⁴⁰⁴ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB1921; E 212, R ⁴⁰³ : H, R ⁴⁰⁴ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1 922; E 212, R ⁴⁰³ : F, R ⁴⁰⁴ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1923; E 212, R ⁴⁰³ : Cl, R ⁴⁰⁴ : ^{Cl, R 450: H, R} 451: OMe, R 452: H], [BB1924; E212, R 403: Me, R 404: Me, R 450: H, R 451: OMe, R 452: H], [ BB 1925; E 213, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1926; E 214, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1927; E 215, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁷ : Me , R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1928; E 216, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1929; E 217, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1930; E 218, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1931; E219, R ⁴⁰¹ : H, R ⁴⁰² : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H] , [BB1932; E220, R ⁴⁰¹ : H, R ^{4 02} : H, R ⁴⁰⁸ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1933; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1934; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H , R ⁴⁵² : H], [BB 1935; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1936 E221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1937; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1938; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : H, ^{R 406: H, R 450:} Cl, R 451: H, R 452: H], [BB1939; E221, R 401: H, R 403: H, R 405: F, R 406: F, R 450: Cl , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1940; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1941; E221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1942; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1943; E221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1944; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F , R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1945; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1946; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me , R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1947; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1948; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1949; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1950; E221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : H, R ⁴⁰⁶ : H, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1951; E 221, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1952; E221, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁵ : F, R ⁴⁰⁶ : F, R ⁴⁵⁰ : S Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1953; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1954; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1 955 E222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1956; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1957; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1958; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1959; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1960; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1961; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : S Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1962; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1963; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB1964; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1965; E222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB1966; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1967; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1968; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1969; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB1970; E 222, R ⁴⁰¹ : H, R ⁴⁰³ : Me, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1971; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1972; E 223, R ⁴⁰¹ : H , R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1973; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1974; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1975; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : S Me, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1976; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : Cl, R ⁴⁵² : H], [BB 1977; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1978; E 223, R ⁴⁰¹ : H , R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1979; E 223, R ⁴⁰¹ : H, R ⁴⁵⁰ : H, R ⁴⁵¹ : S Me, R ⁴⁵² : H], [BB1980; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1981; E224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : Cl, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1982; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : OMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1983; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : CF ₃ , R ⁴⁵¹ : H, R ⁴⁵² : H], [BB 1984; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : SMe, R ⁴⁵¹ : H, R ⁴⁵² : H], [BB1985; E224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹
: Cl, R ⁴⁵² : H], [BB 1986; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : OMe, R ⁴⁵² : H], [BB 1987; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : CF ₃ , R ⁴⁵² : H], [BB 1988; E 224, R ⁴⁰¹ : H, R ⁴⁰⁷ : Me, R ⁴⁵⁰ : H, R ⁴⁵¹ : SMe, R ⁴⁵² : H], [BB 1989; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 1990; E 225, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 1991; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 1992; E 225 , R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 1993; E 225, R ⁴⁰⁹ : F, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 1994; E 225, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 1995; E 225, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : F], [BB 1996; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H] [BB 1997; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : F, R ⁴¹³ : H], [BB 1998; E 225, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 1999; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2000; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H],

[BB 2001; E 225, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2002; E 225, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : Cl , R ⁴¹² : H, R ⁴¹³ : H], [BB 2003; E 225, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Cl], [BB 2004; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2005; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : Cl, R ⁴¹³ : H], [BB 2006; E 225, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2007; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2008; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H] ^{, [BB2009; E225, R 409} : CF 3, R 410: CF 3, R 411: H, R 412: H, R 413: H], [BB2010; E225, R 409: CF 3, R 410: H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2011; E 225, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : CF ₃ ], ^{[BB2012; E225, R 409:} H, R 410: CF 3, R 411: CF 3, R 412: H, R 413: H], [BB2013; E225, R 409: H, R 410: CF 3, R ⁴¹¹ : H, R ⁴¹² : CF ₃ , R ⁴¹³ : H], [BB 2014; E 225, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2015; E225, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB2016; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2017; E 225, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2018; E 225, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2019; E 225, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : OMe] [BB 2020; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2021; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : OMe, R ⁴¹³ : H], [BB 2022; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : Br, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2023; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Br, R ⁴¹² : H, R ⁴¹³ : H], [BB 2024; E 225, R ⁴⁰⁹ : Br, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Br], [BB 2025; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : Me, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2026; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Me, R ⁴¹² : H, R ⁴¹³ : H], [BB 2027; E 225, R ⁴⁰⁹ : Me, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Me], [[ ^{BB2028; E225, R 409: H} , R 410: c-Pr, R 411: H, R 412: H, R 413: H], [BB2029; E225, R 409: H, R 410: H, R 411: c-Pr, R ⁴¹² : H, R ⁴¹³ : H], [BB 2030; E 225, R ⁴⁰⁹ : c-Pr, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : c-Pr], ^{[BB2031; E225, R 409:} H, R 410: OCHF 2, R 411: H, R 412: H, R 413: H], [BB2032; E225, R 409: H, R 410: H, R 411: OCHF ₂ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2033; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2034; E 225, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2035; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2036; E 226, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2037; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H , R ⁴¹² : H, R ⁴¹³ : H], [BB 2038; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2039; E 226, R ⁴⁰⁹ : F, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2040; E 226, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2041; E 226, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : F], [BB 2042; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : F , R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2043; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : F, R ⁴¹³ : H], [BB 2044 E226, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2045; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2046; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2047; E 226, R ⁴⁰⁹ : Cl , R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2048; E 226, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2049; E 226, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Cl], [BB 2050; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2051 E226, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : Cl, R ⁴¹³ : H], [BB 2052; E 226, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2053; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2054; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2055; E 226, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2056; E 226, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2057; E 226, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : CF ₃ ], [BB 2058; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : CF ₃ , R ⁴¹² : H , R ⁴¹³ : H], [BB 2059; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : CF ₃ , R ⁴¹³ : H], [BB 2060; E 226, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2061; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H ], [BB2062; E226, R 409: H, R 410: H, R 411: OMe, R 412: H, R 413: H], [BB2063; E226, R 409: OMe, R 410: OMe, R 411 : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2064; E 226, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2065; E 226, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : OMe], [BB 2066; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2067; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : OMe, R ⁴¹³ : H], [BB 2068; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : Br, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2069; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Br, R ⁴¹² : H, R ⁴¹³ : H], [ ^{BB2070; E226, R 409: Br} , R 410: H, R 411: H, R 412: H, R 413: Br], [BB2071; E226, R 409: H, R 410: Me, R 411: H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2072; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Me, R ⁴¹² : H, R ⁴¹³ : H], [BB 2073; E 226, R ⁴⁰⁹ : Me, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Me], [BB 2074; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : c-Pr, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2075; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : c-Pr, R ⁴¹² : H, R ⁴¹³ : H], [BB 2076; E 226, R ⁴⁰⁹ : c-Pr , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : c-Pr], [BB 2077; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCHF ₂ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2078; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCHF ₂ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2079; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2080; E 226, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCF ₃ , R ⁴¹² : H, R ⁴¹³ : H ], [BB2081; E227, R ^{40 9} : H, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2082; E 227, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2083; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2084; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2085; E 227, R ⁴⁰⁹ : F, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [ BB 2086; E 227, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2087; E 227, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : F], [BB 2088; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2089; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : F, R ⁴¹³ : H], [BB 2090; E 227, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2091; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2092; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2093; E 227, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³
: H], [BB 2094; E 227, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2095; E 227, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Cl], [BB 2096; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2097; E227, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : Cl, R ⁴¹³ : H], [BB 2098; E 227, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2099; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2100; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H],

[BB2101; E227, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2102; E 227, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2103; E 227, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : CF ₃ ], [ BB 2104; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2105; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : CF ₃ , R ⁴¹³ : H], [BB 2106; E 227, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2107; E 227 , R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2108; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2109; E 227, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2110; E 227, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2111; E 227, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : OMe] [BB 2112; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 113; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : OMe, R ⁴¹³ : H], [BB 2114; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : Br, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 115; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Br, R ⁴¹² : H, R ⁴¹³ : H], [BB 2116; E 227, R ⁴⁰⁹ : Br, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Br], [BB 2117; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : Me, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2118; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Me, R ⁴¹² : H, R ⁴¹³ : H], [BB 2119; E 227, R ⁴⁰⁹ : Me, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Me ], [BB 2120; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : c-Pr, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2121, E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : c-Pr, R ⁴¹² : H, R ⁴¹³ : H], [BB 2122; E 227, R ⁴⁰⁹ : c-Pr, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : c- Pr], [BB 2123; E227, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCHF ₂ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2124; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCHF ₂ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2 125; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [ BB 2 126; E 227, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2127; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : H , R ⁴¹² : H, R ⁴¹³ : H], [BB 2128; E 228, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2129; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2130; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2131; E 228, R ⁴⁰⁹ : F, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2132; E 228, R ⁴⁰⁹ : F, R ⁴¹⁰ : H , R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 133; E 228, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : F], [BB 2 134; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2135; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : F, R ⁴¹³ : H], [BB 2136; E 228, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2137; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2138; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2139; E 228, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2140; E 228, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2141; ^{E228, R 409: Cl, R} 410: H, R 411: H, R 412: H, R 413: Cl], [BB2142; E228, R 409: H, R 410: Cl, R 411: Cl, R 412 : H, R ⁴¹³ : H], [BB 2143; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : Cl, R ⁴¹³ : H], [BB 2144; E 228, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2145; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2146; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2147; E 228, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2148; E 228, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H ], [BB 2149; E 228, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : CF ₃ ], [BB 2150; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2151; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : CF ₃ , R ⁴¹³ : H], [BB 2152; E 228, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2153; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2154; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 155; E 228, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2156; E 228, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 157; E228, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : OMe], [BB 2158; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2159; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : OMe, R ⁴¹³ : H], [BB 2 160; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : Br, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2161; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Br, R ⁴¹² : H, R ⁴¹³ : H ], [BB2162; E228, R 409: Br, R 410: H, R 411: H, R 412: H, R 413: Br], [BB2163; E228, R 409: H, R 410: Me, R 411 : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 164; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Me, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 165; E 228, R ⁴⁰⁹ : Me, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Me], [BB 2166; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : c-Pr, R ⁴¹¹ : H, R ⁴¹² : H , R ⁴¹³ : H], [BB 2 167; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : c-Pr, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 168; E 228, R ⁴⁰⁹ : c- Pr, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : c-Pr], [BB 2169; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCHF ₂ , R ⁴¹¹ : H, R ⁴¹² : H , R ⁴¹³ : H], [BB 2170; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCHF ₂ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2171; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2172; E 228, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2173; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2174; E 229, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2175; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2176; E 229 , R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2177; E 229, R ⁴⁰⁹ : F, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2178; E 229, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2179; E 229, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : F], [BB 2180; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H] [BB2181; E229, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H , R ⁴¹² : F, R ⁴¹³ : H], [BB 2182; E 229, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2183; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2184; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2185; E 229, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2186; E 229, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H , R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2187; E 229, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Cl], [BB 2188 E229, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2189; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : Cl, R ⁴¹³ : H], [BB 2190; E 229, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2191; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 192; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2193; E 229, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ^41
2 : H, R ⁴¹³ : H], [BB 2194; E 229, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2 195; E 229, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : CF ₃ ], [BB 2196; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2197; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : CF ₃ , R ⁴¹³ : H], [BB 2198; E 229, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2199; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2200; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H],

^{[BB2201; E229, R 409:} OMe, R 410: OMe, R 411: H, R 412: H, R 413: H], [BB2202; E229, R 409: OMe, R 410: H, R 411: OMe , R ⁴¹² : H, R ⁴¹³ : H], [BB 2203; E 229, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : OMe], [BB 2 204; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2205; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : OMe, R ⁴¹³ : H], [BB 2206; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : Br, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2207; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H , R ⁴¹¹ : Br, R ⁴¹² : H, R ⁴¹³ : H], [BB 2208; E 229, R ⁴⁰⁹ : Br, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Br], [BB 2209 E229, R ⁴⁰⁹ : H, R ⁴¹⁰ : Me, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2210; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Me, R ⁴¹² : H, R ⁴¹³ : H], [BB 2211; E 229, R ⁴⁰⁹ : Me, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Me], [BB 22 12; E 229, R ⁴⁰⁹ : H , R ⁴¹⁰ : c-Pr, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2213; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : c-Pr, R ⁴¹² : H , R ⁴¹³ : H], [BB 2214; E 229, R ⁴⁰⁹ : c-Pr, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : c-Pr], [BB 2215; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCHF ₂ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2216; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCHF ₂ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2 217; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2218; E 229, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2219; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2220; E 230, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2221; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2222; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2223; E 230, R ⁴⁰⁹ : F, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2224; E 230, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [ BB 2225; E 230, R ⁴⁰⁹ : F, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : F], [BB 2226; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : F, R ⁴¹² : H, R ⁴¹³ : H], [BB 2227; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : F, R ⁴¹¹ : H, R ⁴¹² : F, R ⁴¹³ : H], [BB 2 228; E 230, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2229; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2230; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2231; E 230, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2232; E 230, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2233; E230, R ⁴⁰⁹ : Cl, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Cl], [BB 2234; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : Cl, R ⁴¹¹ : Cl, R ⁴¹² : H, R ⁴¹³ : H], [BB 2235; E 230, R ⁴⁰⁹ : H , R ⁴¹⁰ : Cl, R ⁴¹¹ : H, R ⁴¹² : Cl, R ⁴¹³ : H], [BB 2236; E 230, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2237; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2238; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H , R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2239; E 230, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H] , [BB 2240; E 230, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2241; E 230, R ⁴⁰⁹ : CF ₃ , R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : CF ₃ ], [BB 2242; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : CF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2243; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : CF ₃ , R ⁴¹¹ : H, R ⁴¹² : CF ₃ , R ⁴¹³ : H], [BB 2244; E 230, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2245; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2246; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2247; E 230, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : OMe, R ⁴¹¹ : H, R ⁴¹² : H , R ⁴¹³ : H], [BB 2248; E 230, R ⁴⁰⁹ : OMe, R ⁴¹⁰ : H, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H], [BB 2249; E 230, R ⁴⁰⁹ : OMe, R ^{4 10} : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : OMe], [BB 2250; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : OMe, R ⁴¹¹ : OMe, R ⁴¹² : H, R ⁴¹³ : H] ^{, [BB2251; E230, R 409} : H, R 410: OMe, R 411: H, R 412: OMe, R 413: H], [BB2252; E230, R 409: H, R 410: Br, R 411: H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2253; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Br, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 254; E 230, R ⁴⁰⁹ : Br, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Br], [BB 2 255; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : Me, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2256; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : Me, R ⁴¹² : H, R ⁴¹³ : H], [BB 2257; E 230, R ⁴⁰⁹ : Me, R ⁴¹⁰ : H, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : Me], [BB 2258; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : c-Pr, R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H] , [BB 2259; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : c-Pr, R ⁴¹² : H, R ⁴¹³ : H], [BB 2 260; E 230, R ⁴⁰⁹ : c-Pr, R ⁴¹⁰ : H , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : c-Pr], [BB 2261; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCHF ₂ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H] , [BB 2262; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCHF ₂ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2263; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : OCF ₃ , R ⁴¹¹ : H, R ⁴¹² : H, R ⁴¹³ : H], [BB 2264; E 230, R ⁴⁰⁹ : H, R ⁴¹⁰ : H, R ⁴¹¹ : OCF ₃ , R ⁴¹² : H, R ⁴¹³ : H], [BB 2265; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2266; E 231, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [[ ^{BB2267; E231, R 414: H} , R 415: F, R 416: H, R 417: H, R 418: H], [BB2268; E231, R 414: H, R 415: H, R 416: F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2269; E 231, R ⁴¹⁴ : F, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 270; E 231, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2271; E 231, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : F], [BB 2272; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2273; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : F, R ⁴¹⁸ : H], [BB 2274; E 231, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2275; E231, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2276; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2277; E 231, R ⁴¹⁴ : Cl, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2278; E 231, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2279; E 231, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Cl ], [BB 2280; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2281; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : Cl, R ⁴¹⁸ : H], [BB2282; E231, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2283; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2284; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2285; E 231, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2286; E 231, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H , R ⁴¹⁸ : H], [BB 2287; E 231, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : CF ₃ ], [BB 2 288; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2289; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : CF ₃ , R ⁴¹⁸ : H], [BB 2290; E 231, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2291; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 229; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ BB 2293; E 231, R ⁴¹⁴ : OMe, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸
: H], [BB 2294; E 231, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2295; E 231, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : OMe], [BB 2296; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2297; E231, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : OMe, R ⁴¹⁸ : H], [BB 2298; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : Br, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2299; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Br, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2300; E 231, R ⁴¹⁴ : Br, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Br],

[BB 2301; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : Me, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2302: E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Me , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2303; E 231, R ⁴¹⁴ : Me, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Me], [BB 2304; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : c-Pr, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2305; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : c-Pr, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2306; E 231, R ⁴¹⁴ : c-Pr, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : c-Pr], [BB 2307; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : OCHF ₂ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2308; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCHF ₂ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2309; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : OCF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2310; E 231, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2311; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2312; E 232, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2313; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2314; E232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2315; E 232 , R ⁴¹⁴ : F, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2316; E 232, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2317; E 232, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : F], [BB 2318; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2319; E232, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : F, R ⁴¹⁸ : H], [BB 2320; E 232, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2321; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2322 E232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2323; E 232, R ⁴¹⁴ : Cl, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2324; E 232, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2325; E 232, R ⁴¹⁴ : Cl , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Cl], [BB 2326; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2327; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : Cl, R ⁴¹⁸ : H], [BB 2328; E 232, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2329; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 330 E232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2331; E 232, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2332; E 232, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2333; E 232 , R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : CF ₃ ], [BB 2334; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H ], [BB 2335; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : CF ₃ , R ⁴¹⁸ : H], [BB 2336; E 232, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2337; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 338; E232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2339; E 232, R ⁴¹⁴ : OMe, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2340; E 232, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2341; E 232, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : OMe], [BB 2342; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H ], [BB 2343; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : OMe, R ⁴¹⁸ : H], [BB 2344; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : Br, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2345; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Br, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2346; E 232, R ⁴¹⁴ : Br, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Br], [BB 2347; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : Me, R ⁴¹⁶ : H, R ⁴¹⁷ : H , R ⁴¹⁸ : H], [BB 2348; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Me, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2349; E 232, R ⁴¹⁴ : Me, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Me], [BB 2 350; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : c-Pr, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 351 E232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : c-Pr, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2352; E 232, R ⁴¹⁴ : c-Pr, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : c-Pr], [BB 2353; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : OCHF ₂ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2354 E232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCHF ₂ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 355; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : OCF ₃ , R ⁴¹⁶ : H , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2356; E 232, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 357: E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2358; E233, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2359; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 360; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2361; E 233, R ⁴¹⁴ : F, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ BB2362; E233, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2363; E 233, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : F], [BB 2364; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2365; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : F, R ^{41 8} : H], [BB 2366; E233, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2367; E233, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2368; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2369 E233, R ⁴¹⁴ : Cl, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2370; E 233, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2371; E233, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Cl], [BB 2372; E 233, R ⁴¹⁴ : H , R ⁴¹⁵ : Cl, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2373; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : Cl, R ⁴¹⁸ : H], [BB2374; E233, R 414: CF 3, R 415: H, R 416: H, R 417: H, R 418: H], [BB2375; E233, R 414: H, R 415: CF 3 , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2376; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ ^{BB2377; E233, R 414: CF} 3, R 415: CF 3, R 416: H, R 417: H, R 418: H], [BB2378; E233, R 414: CF 3, R 415: H, R 416 : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2379; E 233, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : CF ₃ ], [BB 2 380 E233, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2381; E233, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : C F ₃ , R ⁴¹⁸ : H], [BB 2382; E 233, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2383; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2384; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H ], [BB2385; E233, R 414: OMe, R 415: OMe, R 416: H, R 417: H, R 418: H], [BB2386; E233, R 414: OMe, R 415: H, R 416 : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2387; E 233, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : OMe], [BB 2388; E 233, E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2389; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : OMe ^{, R 418: H], [} BB2390; E233, R 414: H, R 415: Br, R 416: H, R 417: H, R 418: H], [BB2391; E233, R 414: H, R 415 : H, R ⁴¹⁶ : Br, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2392; E233, R ⁴¹⁴ : Br, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Br], [BB 2393; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : Me, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸
: H], [BB 2394; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Me, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2395; E 233, R ⁴¹⁴ : Me, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Me], [BB 2396; E 233, R ⁴¹⁴ : H, R ⁴¹⁵ : c-Pr, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ BB2397; E233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : c-Pr, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2398; E233, R ⁴¹⁴ : c-Pr, R ⁴¹⁵ : H, R ^{416: H, R 417: H} , R 418: c-Pr], [BB2399; E233, R 414: H, R 415: OCHF 2, R 416: H, R 417: H, R 418: H], [ BB2400; E233, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCHF ₂ , R ⁴¹⁷ : H, R ⁴¹⁸ : H],

^{[BB2401; E233, R 414:} H, R 415: OCF 3, R 416: H, R 417: H, R 418: H], [BB2402; E233, R 414: H, R 415: H, R 416: OCF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2403; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2404; E 234, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2405; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H , R ⁴¹⁸ : H], [BB 2406; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2407; E 234, R ⁴¹⁴ : F, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2408; E 234, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2409; E234, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : F], [BB 2410; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : F , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2411; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : F, R ⁴¹⁸ : H], [BB 2412; E 234, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2413; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2414; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2415; E 234, R ⁴¹⁴ : Cl, R ⁴¹⁵ : Cl , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2416; E 234, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2417 E234, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Cl], [BB 2418; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2419; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : Cl, R ⁴¹⁸ : H], [BB 2420; E234, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H , R ⁴¹⁸ : H], [BB 2421; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2422; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2423; E 234, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2424; E234, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2425; E 234, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : CF ₃ ], [BB 2426; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2427; E234, R 414: H, R 415: CF 3, R 416: H, R 417: CF 3, R 418: H], [BB2428; E234, R 414: OMe, R 415: H , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2429; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2430 E234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2431; E 234, R ⁴¹⁴ : OMe, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2432; E 234, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2433; E 234, R ⁴¹⁴ : OMe , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : OMe], [BB 2434; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2435; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : OMe, R ⁴¹⁸ : H], [BB 2436; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : Br, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2437; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Br, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2438; , R ⁴¹⁴ : Br, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Br], [BB 2439; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : Me, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2440; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Me, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2441; E 234, R ⁴¹⁴ : Me, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Me], [BB 2442; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : c-Pr, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2443; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : c-Pr, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2444; E234, R ⁴¹⁴ : c-Pr, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : c-Pr], [BB 2445; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : OCHF ₂ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2446; E234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCHF ₂ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2 447: E234, R ⁴¹⁴ : H, R ⁴¹⁵ : OCF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2448; E 234, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ BB 2449; E 235, R ⁴¹⁴ : H, R ^{4 15} : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2450; E 235, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H] [BB2451; E235, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2452; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2453; E 235, R ⁴¹⁴ : F, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2454; E 235, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2455; E 235, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : F], [BB 2456; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2457; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : F, R ⁴¹⁸ : H], [BB 2458; E 235, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ BB 2459; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2460; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, ^{R 417: H, R 418:} H], [BB2461; E235, R 414: Cl, R 415: Cl, R 416: H, R 417: H, R 418: H], [BB2462; E235, R 414: Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2463; E 235, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Cl], [BB 2464; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2465; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : Cl, R ⁴¹⁸ : H], [BB 2466; E 235, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2467; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2468; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2469; E 235, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2470; E 235, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2471; E 235, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : CF ₃ ], [BB 2472; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2473; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : CF ₃ , R ⁴¹⁸ : H], [BB 2474; E 235, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2475; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2476; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H] ^{, [BB2477; E235, R 414} : OMe, R 415: OMe, R 416: H, R 417: H, R 418: H], [BB2478; E235, R 414: OMe, R 415: H, R 416: OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2479; E 235, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : OMe], [BB 2480; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2481; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : O ^{Me, R 418: H],} [BB2482; E235, R 414: H, R 415: Br, R 416: H, R 417: H, R 418: H], [BB2483; E235, R 414: H, R ⁴¹⁵ : H, R ⁴¹⁶ : Br, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2484; E 235, R ⁴¹⁴ : Br, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Br] [BB2485; E235, R ⁴¹⁴ : H, R ⁴¹⁵ : Me, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2486; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Me, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2487; E 235, R ⁴¹⁴ : Me, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Me], [BB 2488; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : c-Pr, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2489; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : c-Pr, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2490; E 235, R ⁴¹⁴ : c-Pr, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : c-Pr], [BB 2491; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : OCHF ₂ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2492; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCHF ₂ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2493; E 235, R ⁴¹⁴ : H, R ⁴¹⁵ : OCF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R
^{418: H], [BB2494;} E235, R 414: H, R 415: H, R 416: OCF 3, R 417: H, R 418: H], [BB2495; E236, R 414: H, R 415: H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2496; E 236, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [ BB2497; E236, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2498; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2499; E 236, R ⁴¹⁴ : F, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2500; E 236, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : F, R ⁴¹⁷ : H, R ⁴¹⁸ : H],

[BB 2501; E 236, R ⁴¹⁴ : F, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : F], [BB 2502: E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : F , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2503; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : F, R ⁴¹⁶ : H, R ⁴¹⁷ : F, R ⁴¹⁸ : H], [BB 2504; E 236, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2505; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2506; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2507; E 236, R ⁴¹⁴ : Cl, R ⁴¹⁵ : Cl , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2508; E 236, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2509 E236, R ⁴¹⁴ : Cl, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Cl], [BB 2510; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : Cl, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2511; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : Cl, R ⁴¹⁶ : H, R ⁴¹⁷ : Cl, R ⁴¹⁸ : H], [BB 2512; E 236, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2513; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ^{418: H], [BB2514;} E236, R 414: H, R 415: H, R 416: CF 3, R 417: H, R 418: H], [BB2515; E236, R 414: CF 3, R 415 : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2516; E 236, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB2517; E236, R ⁴¹⁴ : CF ₃ , R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : CF ₃ ], [BB 2518; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : CF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2519; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : CF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : CF ₃ , R ⁴¹⁸ : H], [BB 25 20; E 236, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2521; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2522; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2523; E 236, R ⁴¹⁴ : OMe, R ⁴¹⁵ : OMe , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2524; E 236, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 25 25 E236, R ⁴¹⁴ : OMe, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : OMe], [BB 2526; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : OMe, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2527; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : OMe, R ⁴¹⁶ : H, R ⁴¹⁷ : OMe, R ⁴¹⁸ : H], [BB 2528; E 236, R ⁴¹⁴ : H , R ⁴¹⁵ : Br, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2529; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Br, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2530; E 236, R ⁴¹⁴ : Br, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Br], [BB 2531; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : Me, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2532; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : Me, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2533; E 236 , R ⁴¹⁴ : Me, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : Me], [BB 2534; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : c-Pr, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2535; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : c-Pr, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2536; E 236, R ⁴¹⁴ : c -Pr, R ⁴¹⁵ : H, R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : c-Pr], [BB 2537; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : OCHF ₂ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2538; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCHF ₂ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2539; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : OCF ₃ , R ⁴¹⁶ : H, R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2540; E 236, R ⁴¹⁴ : H, R ⁴¹⁵ : H, R ⁴¹⁶ : OCF ₃ , R ⁴¹⁷ : H, R ⁴¹⁸ : H], [BB 2541; E 237, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²² : H], [BB 2542; E 237, R ⁴²⁰ : Me, R ⁴²¹ : H, R ⁴²² : H], [BB 2543; , R ⁴²⁰ : H, R ⁴²¹ : Me, R ⁴²² : H], [BB 2544; E 237, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²² : Me], [BB 2545; E 237, R ⁴²⁰ : Me, R ⁴²¹ : Me, R ⁴²² : H], [BB 2546; E 237, R ⁴²⁰ : Me, R ⁴²¹ : H, R ⁴²² : Me], [BB 2547; E 237, R ⁴²⁰ : H, R ⁴²¹ : Me, R ⁴²² : Me] , [BB 2548; E 237, R ⁴²⁰ : Me, R ⁴²¹ : Me, R ⁴²² : Me], [BB 2 549; E 237, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²² : Cl], [BB 2550; E 237, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²² : CF ₃ ], [BB 2551; E 237, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²² : OMe], [BB 2552; E 238, R ⁴²⁰ : H, R ⁴²¹ : H , R ⁴²³ : H], [BB 2553; E 238, R ⁴²⁰ : Me, R ⁴²¹ : H, R ⁴²³ : H], [BB 2554; E 238, R ⁴²⁰ : H, R ⁴²¹ : Me, R ⁴²³ : H], [BB 2555; E 238 , R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²³ : Me], [BB 2556; E 238, R ⁴²⁰ : Me, R ⁴²¹ : Me, R ⁴²³ : H], [BB 2557; E 238, R ⁴²⁰ : Me, R ⁴²¹ : H, R ⁴²³ : Me], [BB 2558; E 238, R ⁴²⁰ : H, R ⁴²¹ : Me, R ⁴²³ : Me], [BB 2559; E 238, R ⁴²⁰ : Me, R ⁴²¹ : Me, R ⁴²³ : Me] , [BB 2560; E 238, R ⁴²⁰ : H, R ⁴²¹ : Cl, R ⁴²³ : H], [BB 2561; E 238, R ⁴²⁰ : H, R ⁴²¹ : CF ₃ , R ⁴²³ : H], [BB 2562; E 238, R ⁴²⁰ : H, R ⁴²¹ : OMe, R ⁴²³ : H], [BB 2563; E 238, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²³ : Cl], [BB 2564; E 238, R ⁴²⁰ : H, R ⁴²¹ : H , R ⁴²³ : CF ₃ ], [BB 2565; E 238, R ⁴²⁰ : H, R ⁴²¹ : H, R ⁴²³ : OMe], [BB 2566; E 239, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁶ : H], [BB2567; E239, R ⁴²⁴ : Me, R ⁴²⁵ : H, R ⁴²⁶ : H], [BB 2568; E 239, R ⁴²⁴ : H, R ⁴²⁵ : Me, R ⁴²⁶ : H], [BB 2569; E 239, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁶ : Me], [BB 2570; E 239, R ⁴²⁴ : Me, R ⁴²⁵ : Me, R ⁴²⁶ : H], [BB 2571; E 239, R ⁴²⁴ : Me, R ⁴²⁵ : H, R ⁴²⁶ : Me], [BB2572; E239, R ⁴²⁴ : H, R ⁴²⁵ : Me, R ⁴²⁶ : Me], [BB 2573; E239, R ⁴²⁴ : Me, R ⁴²⁵ : Me, R ⁴²⁶ : Me], [BB 2574; E239, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁶ : Cl], [BB 2575; E 239, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁶ : CF ₃ ], [BB 2 576; E 2 39, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁶ : OMe], [BB 2577; E 240, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁷ : H], [BB 2578; E 240, R ⁴²⁴ : Me, R ⁴²⁵ : H, R ⁴²⁷ : H], [BB 2579; E 240, R ⁴²⁴ : H, R ⁴²⁵ : Me, R ⁴²⁷ : H], [BB 2580; E 240, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁷ : Me ], [BB 2581; E 240, R ⁴²⁴ : Me, R ⁴²⁵ : Me, R ⁴²⁷ : H], [BB 2582; E 240, R ⁴²⁴ : Me, R ⁴²⁵ : H, R ⁴²⁷ : Me], [BB 2583; E 240, R ⁴²⁴ : H, R ⁴²⁵ : Me, R ⁴²⁷ : Me], [BB 2584; E 240, R ⁴²⁴ : Me, R ⁴²⁵ : Me, R ⁴²⁷ : Me], [BB 2585; E 240, R ⁴²⁴ : H, R ⁴²⁵ : Cl , R ⁴²⁷ : H], [BB 2586; E 240, R ⁴²⁴ : H, R ⁴²⁵ : CF ₃ , R ⁴²⁷ : H], [BB 2587; E 240, R ⁴²⁴ : H, R ⁴²⁵ : OMe, R ⁴²⁷ : H], [BB2588; E240, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁷ : Cl], [BB 2589; E 240, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁷ : CF ₃ ], [BB 2590; E 240, R ⁴²⁴ : H, R ⁴²⁵ : H, R ⁴²⁷ : OMe], [BB 2591; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2 592; E 241, R ⁴²⁸ : H, R ⁴²⁹ : F, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2593; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : F, R ⁴³¹ : H , R ⁴³² : H], [BB 2594; E 241, R ⁴²⁸ : F, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : F], [BB 2595; E 241, R ⁴²⁸ : H, R ⁴²⁹ : F, R ⁴³⁰ : H, R ⁴³¹ : F, R ⁴³² : H], [BB 2596; E 241, R ⁴²⁸ : H, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB2597; E241 , R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Cl, R ⁴³¹ : H, R ⁴³² : H], [BB 2598; E 241, R ⁴²⁸ : Cl, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2599; E 241, R ⁴²⁸ : Cl, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Cl], [BB 2600; E 241, R ⁴²⁸ : H, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : Cl, R ⁴³² : H],

^{[BB2601; E241, R 428:} H, R 429: CF 3, R 430: H, R 431: H, R 432: H], [BB2602; E241, R 428: H, R 429: H, R 430: CF ₃ , R ⁴³¹ : H, R ⁴³² : H], [BB 2603; E 241, R ⁴²⁸ : H, R ⁴²⁹ : OMe, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2604; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OMe, R ⁴³¹ : H, R ⁴³² : H], [BB 2605; E 241, R ⁴²⁸ : OMe, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H , R ⁴³² : OMe], [BB 2606; E 241, R ⁴²⁸ : H, R ⁴²⁹ : OMe, R ⁴³⁰ : H, R ⁴³¹ : OMe, R ⁴³² : H], [BB 2607; E 241, R ⁴²⁸ : H, R ⁴²⁹ : Br, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2608; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Br, R ⁴³¹ : H, R ⁴³² : H], [BB2609; E241, R ⁴²⁸ : Br, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Br], [BB 2610; E 241, R ⁴²⁸ : H, R ⁴²⁹ : Me, R ⁴³⁰ : H , R ⁴³¹ : H, R ⁴³² : H], [BB 2611; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Me, R ⁴³¹ : H, R ⁴³² : H], [BB 2612; E 241, R ⁴²⁸ : Me, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Me], [BB 2613; E 241, R ⁴²⁸ : H, R ⁴²⁹ : c-Pr, R ⁴³⁰ : H, R ⁴³¹ : H , R ⁴³² : H], [BB 2614; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : c-Pr, R ⁴³¹ : H, R ⁴³² : H], [BB 2615; E 241, R ⁴²⁸ : c- Pr, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : c-Pr], [BB 2616; E 241, R ⁴²⁸ : H, R ⁴²⁹ : OCHF ₂ , R ⁴³⁰ : H, R ⁴³¹ : H , R ⁴³² : H], [BB 2617; E 2 41, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OCHF ₂ , R ⁴³¹ : H, R ⁴³² : H], [BB 2618; E 241, R ⁴²⁸ : H, R ⁴²⁹ : OCF ₃ , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2619; E 241, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OCF ₃ , R ⁴³¹ : H, R ⁴³² : H], [BB 2620; E 242, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2621; E 242, R ⁴²⁸ : H, R ⁴²⁹ : F, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2622; E 242, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : F, R ⁴³¹ : H, R ⁴³² : H], [BB 2623; E 242, R ⁴²⁸ : F, R ⁴²⁹ : H , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : F], [BB 2624; E 242, R ⁴²⁸ : H, R ⁴²⁹ : F, R ⁴³⁰ : H, R ⁴³¹ : F, R ⁴³² : H], [BB 2625 E242, R ⁴²⁸ : H, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2626; E 242, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Cl, R ⁴³¹ : H, R ⁴³² : H], [BB 2627; E 242, R ⁴²⁸ : Cl, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2628; E 242, R ⁴²⁸ : Cl , R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Cl], [BB 2629; E 242, R ⁴²⁸ : H, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : Cl, R ⁴³² : H], [BB2630; E242, R 428: H, R 429: CF 3, R 430: H, R 431: H, R 432: H], [BB2631; E242, R 428: H, R 429: H, R ⁴³⁰ : CF ₃ , R ⁴³¹ : H, R ⁴³² : H], [BB 2632; E 242, R ⁴²⁸ : H, R ⁴²⁹ : OMe, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2633 E 242, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OMe, R ⁴³¹ : H, R ⁴³² : H], [BB 2634; E 242, R ⁴²⁸ : OMe, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : OMe], [BB 26 35; E 242 , R ⁴²⁸ : H, R ⁴²⁹ : OMe, R ⁴³⁰ : H, R ⁴³¹ : OMe, R ⁴³² : H], [BB 2636; E 242, R ⁴²⁸ : H, R ⁴²⁹ : Br, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2637; E 242, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Br, R ⁴³¹ : H, R ⁴³² : H], [BB 2638; E 242, R ⁴²⁸ : Br, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Br], [BB 2639; E 242, R ⁴²⁸ : H, R ⁴²⁹ : Me, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H] ^{, [BB2640; E242, R 428} : H, R 429: H, R 430: Me, R 431: H, R 432: H], [BB2641; E242, R 428: Me, R 429: H, R 430: H, R ⁴³¹ : H, R ⁴³² : Me], [BB 2642; E 242, R ⁴²⁸ : H, R ⁴²⁹ : c-Pr, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2643; E 242 , R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : c-Pr, R ⁴³¹ : H, R ⁴³² : H], [BB 2644; E 242, R ⁴²⁸ : c-Pr, R ⁴²⁹ : H, R ⁴³⁰ : H , R ⁴³¹ : H, R ⁴³² : c-Pr], [BB 2645; E 242, R ⁴²⁸ : H, R ⁴²⁹ : OCHF ₂ , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2 646: E 242 , R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OCHF ₂ , R ⁴³¹ : H, R ⁴³² : H], [BB 2647; E 242, R ⁴²⁸ : H, R ⁴²⁹ : OCF ₃ , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2648; E 242, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OCF ₃ , R ⁴³¹ : H, R ⁴³² : H], [BB 2649; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2650; E 243, R ⁴²⁸ : H, R ⁴²⁹ : F, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2651; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : F, R ⁴³¹ : H, R ⁴³² : H], [BB 2652; E 243, R ⁴²⁸ : F, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H , R ⁴³² : F], [BB 2653; E 243, R ⁴²⁸ : H, R ⁴²⁹ : F, R ⁴³⁰ : H, R ⁴³¹ : F, R ⁴³² : H], [BB 2654; E 243, R ⁴²⁸ : H, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2655; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Cl, R ⁴³¹ : H, R ⁴³² : H], ^{[BB2656; E243, R 428:} Cl, R 429: Cl, R 430: H, R 431: H, R 432: H], [BB2657; E243, R 428: Cl, R 429: H, R 430: H , R ⁴³¹ : H, R ⁴³² : Cl], [BB 2658; E 243, R ⁴²⁸ : H, R ⁴²⁹ : Cl, R ⁴³⁰ : H, R ⁴³¹ : Cl, R ⁴³² : H], [BB 2659; E 243, R ⁴²⁸ : H, R ⁴²⁹ : CF ₃ , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2660; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : CF ₃ , R ⁴³¹ : H , R ⁴³² : H], [BB 2661; E 243, R ⁴²⁸ : H, R ⁴²⁹ : OMe, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2662; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OMe, R ⁴³¹ : H, R ⁴³² : H], [BB 2663; E 243, R ⁴²⁸ : OMe, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : OMe], ^{[BB2664; E243, R 428:} H, R 429: OMe, R 430: H, R 431: OMe, R 432: H], [BB2665; E243, R 428: H, R 429: Br, R 430: H , R ⁴³¹ : H, R ⁴³² : H], [BB 2 666; E243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Br, R ⁴³¹ : H, R ⁴³² : H], [BB 2667; E 243, R ⁴²⁸ : Br, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Br], [BB 2668; E 243, R ⁴²⁸ : H, R ⁴²⁹ : Me, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2669; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : Me, R ⁴³¹ : H, R ⁴³² : H], [BB 2670; E 243, R ⁴²⁸ : Me, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : Me], [BB 2671; E 243, R ⁴²⁸ : H, R ⁴²⁹ : c-Pr, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2672; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : c-Pr, R ⁴³¹ : H, R ⁴³² : H], [BB 2673; E 243, R ⁴²⁸ : c-Pr, R ⁴²⁹ : H, R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : c-Pr], [BB 2674; E 243, R ⁴²⁸ : H, R ⁴²⁹ : OCHF ₂ , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H], [BB 2 675: E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OCHF ₂ , R ⁴³¹ : H, R ⁴³² : H], [BB 2676; E 243, R ⁴²⁸ : H, R ⁴²⁹ : OCF ₃ , R ⁴³⁰ : H, R ⁴³¹ : H, R ⁴³² : H] [BB 2677; E 243, R ⁴²⁸ : H, R ⁴²⁹ : H, R ⁴³⁰ : OCF ₃ , R ⁴³¹ : H, R ⁴³² : H], [BB 2 678: E 244, R ⁴³³ : H, R ⁴³⁴ : H, R ⁴³⁵ : H], [BB 2679; E244, R ⁴³³ : Me, R ⁴³⁴ : H, R ⁴³⁵ : H], [BB 2 680: E 244, R ⁴³³ : H, R ⁴³⁴ : Me, R ⁴³⁵ : H], [BB 2 6 8 , R ⁴³³ : H, R ⁴³⁴ : H, R ⁴³⁵ : Me], [BB 2682; E 244, R ⁴³³ : Me, R ⁴³⁴ : Me, R ⁴³⁵ : H], [BB 2683; E 244, R ⁴³³ : Me, R ⁴³⁴ : H, R ⁴³⁵ : Me], [B ^{B2684; E244, R 433: H} , R 434: Me, R 435: Me], [BB2685; E244, R 433: Me, R 434: Me, R 435: Me], [BB2686; E244, R 433: H , R ⁴³⁴ : H, R ⁴³⁵ : Cl], [BB 2687; E 244, R ⁴³³ : H, R ⁴³⁴ : H, R ⁴³⁵ : CF ₃ ], [BB 2688; E 244, R ⁴³³ : H, R ⁴³⁴ : H, R ⁴³⁵ : OMe], [BB 2689; E245, R ⁴³³ : H, R ⁴³⁴ : H, R ⁴³⁶ : H], [BB 2690; E 245, R ⁴³³ : Me, R ⁴³⁴ : H, R ⁴³⁶ : H], [BB 2691; ^{E245, R 433: H, R} 434: Me, R 436: H], [BB2692; E245, R 433: H, R 434: H, R 436: Me], [BB2693; E245, R 433: Me, R ^{434: Me, R 436: H} ], [BB2694; E245, R 433: Me, R 434: H, R 436: Me], [BB2695; E245, R 433: H, R 434: Me, R 436: Me ], [BB2696; E245, R 433: Me, R 434: Me, R 436: Me], [BB2697; E245, R 433: H, R 434: Cl, R 436: H], [BB2698; E245, R ^{433: H, R 434: CF} 3, R 436: H], [BB2699; E245, R 433: H, R 434: OMe, R 436: H], [BB2700; E245, R 433: H, R 434: H, R ⁴³⁶ : Cl],

^{[BB2701; E245, R 433:} H, R 434: H, R 436: CF 3], [BB2702; E245, R 433: H, R 434: H, R 436: OMe], [BB2703; E246, R 437 : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2704; E 246, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2705; E 246, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2706; E 246, R ⁴³⁷ : H, R ⁴³⁸ : H , R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2707; E 246, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl], [BB 2708 E246, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H], [BB 2709; E 246, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2710; E 246, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2711; E 246, R ⁴³⁷ : H , R ⁴³⁸ : H, R ⁴³⁹ : Me, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2712; E 246, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me], [BB2713; E246, R 437: H, R 438: Me, R 439: H, R 440: Me, R 441: H], [BB2714; E246, R 437: H, R 438: H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2715; E 247, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2716; , R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2717; E 247, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2718; E 24 7, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2719; E 247, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl], [BB 2720; E 247, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H], [BB 2721; E 247, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2722; E 247, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H ], [BB2723; E247, R 437: H, R 438: H, R 439: Me, R 440: H, R 441: H], [BB2724; E247, R 437: Me, R 438: H, R 439 : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me], [BB 2725; E 247, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H], [BB 2726; E 247, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2727; E 248, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H , R ⁴⁴¹ : H], [BB 2728; E 248, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2 729; E 248, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2730; E 248, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2731; E248, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl], [BB 2732; E 248, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H , R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H], [BB 2733; E 248, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2734; E 248, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2735; E 248, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Me, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2 736: E 248, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me], [BB 2 737: E 248, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H ], [BB 2738; E 248, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2739; E 249, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2740; E 249, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2741; E 249, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB2742; E249, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H , R ⁴⁴¹ : H], [BB 2743; E 249, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl], [BB 2 744; E 249, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H], [BB 2745; E249, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB2746; E249, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2 747: E249, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Me , R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2 748; E 249, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me], [BB 2749; E 249, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H], [BB 2750; E249, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2751; E 250, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2752; E 250, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H] [BB 2753; E 250, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2754; E 250, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2755; E 250, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl], [BB 2756; E 250, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H], [BB 2757; E 250, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2758; E 250, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2759; E 250, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Me, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2760; E 250, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me], [, BB2761; E250, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H], [BB 2762; E 250, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2763; E 251, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2764; E 251, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2765; E 251, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2766; E 251, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2 767: E 251, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl], [B B2768; E251, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H], [BB 2769; E 251, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2770; E 251, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 277 1; E 251, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Me, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2772; E 251, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me], [BB 2773; E 251, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H], [BB 2 774; E 251, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H], [BB 2775; E 252, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H ], [BB2776; E252, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2777; E 252, R ⁴³⁷ : H, R ^438] : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2778; E 252, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2779; E 252, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Cl, R ⁴⁴² : H], [BB 2 780; E 252 , R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB2781; E252, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2782; E 252, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2783; E 252, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Me, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2784; E 252, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me, R ⁴⁴² : H], [BB 2 785; E 252, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H, R ⁴⁴² : H], [BB 2786; E 252 , R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2787; E 252, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2 788; E 252, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2789; E 252, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2 790: E 252, R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : Cl, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2791; E 252, R ⁴³⁷ : Cl, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H , R ⁴⁴¹ : Cl, R ⁴⁴² : Me], [BB 2792; E 252, R ⁴³⁷ : H, R ⁴³⁸ : Cl, R ⁴³⁹ : H, R ⁴⁴⁰ : Cl, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2793 E252, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2794; E 252, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2795; E 252, R ⁴³⁷ : H, R ⁴³⁸
: H, R ⁴³⁹ : Me, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2796; E 252, R ⁴³⁷ : Me, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : Me, R ⁴⁴² : Me], [BB 2797; E 252, R ⁴³⁷ : H, R ⁴³⁸ : Me, R ⁴³⁹ : H, R ⁴⁴⁰ : Me, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2798; E 252 , R ⁴³⁷ : H, R ⁴³⁸ : H, R ⁴³⁹ : H, R ⁴⁴⁰ : H, R ⁴⁴¹ : H, R ⁴⁴² : Me], [BB 2799; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2800; E 253, R ⁴⁵³ : F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H],

^{[BB2801; E253, R 453:} H, R 454: F, R 455: H, R 456: H], [BB2802; E253, R 453: H, R 454: H, R 455: F, R 456: H ], [BB2803; E253, R 453: H, R 454: H, R 455: H, R 456: F], [BB2804; E253, R 453: Cl, R 454: H, R 455: H, R 456 : H], [BB 2805; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2806; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, ^{R 456: H], [BB2807} ; E253, R 453: H, R 454: H, R 455: H, R 456: Cl], [BB2808; E253, R 453: Me, R 454: H, R 455: H, R ⁴⁵⁶ : H], [BB 2809; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : Me, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2810: E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Me, R ⁴⁵⁶ : H], [BB 2811; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2812; E 253, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H ^{, R 455: H, R 456} : H], [BB2813; E253, R 453: H, R 454: OMe, R 455: H, R 456: H], [BB2814; E253, R 453: H, R 454 : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [BB 2815; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : OMe], [BB 2816; E 253, R ⁴⁵³ : CF ₃ , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2817; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : CF ₃ , R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2818; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : CF ₃ , R ⁴⁵⁶ : H], [BB 2819; E 253, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : CF ₃ ], [BB 2820 E254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2821; E 254, R ⁴⁵³ : F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2822; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2823; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2824; E254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : F], [BB 2825; E 254, R ⁴⁵³ : Cl, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [ BB2826; E254, R ⁴⁵³ : H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2827; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H] ^{, [BB2828; E254, R 453} : H, R 454: H, R 455: H, R 456: Cl], [BB2829; E254, R 453: Me, R 454: H, R 455: H, R 456: H], [BB2830; E254, R 453: H, R 454: Me, R 455: H, R 456: H], [BB2831; E254, R 453: H, R 454: H, R 455: Me, R ⁴⁵⁶ : H], [BB 2832; E254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2833; E 254, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H , R ⁴⁵⁶ : H], [BB 2834; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : OMe, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2 835; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [BB 2836; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : OMe], [BB 2837; E 254, R ⁴⁵³ : CF ₃ , R ⁴⁵⁴ : H , R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2838; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : CF ₃ , R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2839; E 254, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : CF ₃ , ^{R 456: H], [BB2840} ; E254, R 453: H, R 454: H, R 455: H, R 456: CF 3], [BB2841; E255, R 453: H, R 454: H, R 455 : H, R ⁴⁵⁶ : H], [BB 2842; E 255, R ⁴⁵³ : F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2843; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2844; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2845; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : ^{H, R 455: H, R} 456: F], [BB2846; E255, R 453: Cl, R 454: H, R 455: H, R 456: H], [BB2847; E255, R 453: H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2848; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H], [BB 2849; E 255, R ⁴⁵³ : H , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Cl], [BB 2850; E 255, R ⁴⁵³ : Me, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2 851; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : Me, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2852; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Me, R ⁴⁵⁶ : H], [BB 2853; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2854; E 255, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2855; E255, R ⁴⁵³ : H, R ⁴⁵⁴ : OMe, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2856; E 255, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [ ^{BB2857; E255, R 453: H} , R 454: H, R 455: H, R 456: OMe], [BB2858; E255, R 453: CF 3, R 454: H, R 455: H, R 456: H ], [BB 2859; E 255, R ^{4 53: H, R 454: CF} 3, R 455: H, R 456: H], [BB2860; E255, R 453: H, R 454: H, R 455: CF 3, R 456: H], [BB2861 E255, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : CF ₃ ], [BB2862; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H] [BB 2863; E 256, R ⁴⁵³ : F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2864; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2865; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2866; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : F], [BB 2867; E 256, R ⁴⁵³ : Cl, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2 868: E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H , R ⁴⁵⁶ : H], [BB 2869; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H], [BB 2870; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Cl], [BB2871; E 256, R ⁴⁵³ : Me, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2 872; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : Me, ^{R 455: H, R 456:} H], [BB2873; E256, R 453: H, R 454: H, R 455: Me, R 456: H], [BB2874; E256, R 453: H, R 454: H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2875; E 256, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2876; E 256, R ⁴⁵³ : H, R ^{454: OMe, R 455: H} , R 456: H], [BB2877; E256, R 453: H, R 454: H, R 455: OMe, R 456: H], [BB2878; E256, R 453: H , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : OMe], [BB 2879; E 256, R ⁴⁵³ : CF ₃ , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2 880; E 256, R ⁴⁵³ : H, R ⁴⁵⁴ : CF ₃ , R ^{455: H, R 456: H} ], [BB2881; E256, R 453: H, R 454: H, R 455: CF 3, R 456: H], [BB2882; E256, R 453: H, R 454: ^{H, R 455: H, R} 456: CF 3], [BB2883; E257, R 453: H, R 454: H, R 455: H, R 456: H], [BB2884; E257, R 453: F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2885; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2886; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2887; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : F], [BB 2 888; E 257, R ⁴⁵³ : Cl, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2889; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2890; E 257 , R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H], [BB 2891; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Cl], [BB 2 89 2 E257, R ⁴⁵³ : Me, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2893; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : Me, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2894; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Me, R ⁴⁵⁶ : H], [BB 2895; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me ], [BB 2896; E 257, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2897; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : OMe, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2898; E 2 57, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [BB 2899; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : OMe], [ BB 2900; E 257, R ⁴⁵³ : CF ₃ , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H],

[BB 2901; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : CF ₃ , R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2902; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : CF ₃ , R ⁴⁵⁶ : H], [BB 2903; E 257, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : CF ₃ ], [BB 2904; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H , R ⁴⁵⁶ : H], [BB 2 905; E 258, R ⁴⁵³ : F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2906; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2907; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2 908; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, ^{R 455: H, R 456:} F], [BB2909; E258, R 453: Cl, R 454: H, R 455: H, R 456: H], [BB2910; E258, R 453: H, R 454: Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2911; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H], [BB 2912; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Cl], [BB 2913; E258, R ⁴⁵³ : Me, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2914; E 258, R ⁴⁵³ : H , R ⁴⁵⁴ : Me, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2915; E258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Me, R ⁴⁵⁶ : H], [BB 2916; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2917; E258, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2918; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : OMe, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2919; E 258, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [BB 2920; E258, R ⁴⁵³ : H, R ^{454: H, R 455: H} , R 456: OMe], [BB2921; E258, R 453: CF 3, R 454: H, R 455: H, R 456: H], [BB2922; E258, R 453: _{^{H, R 454: CF 3,}} R 455: H, R 456: H], [BB2923; E258, R 453: H, R 454: H, R 455: CF 3, R 456: H], [BB2924; E258 , R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : CF ₃ ], [BB 2925; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [ BB 2926; E 259, R ⁴⁵³ : F, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2 927; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H] [BB 2 928; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2 929: E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : F], [BB 2930; E 259, R ⁴⁵³ : Cl, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2931; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB2932; E259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H], [BB 2933; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H , R ⁴⁵⁶ : Cl], [BB 2934; E 259, R ⁴⁵³ : Me, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2935; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : Me, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2936; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Me, R ⁴⁵⁶ : H], [BB 2 937; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2938; E 259, R ⁴⁵³ : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2939; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : OMe, R ⁴⁵⁵ : H, R ^{45 6} : H], [BB 2940; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [BB 2941; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H , R ⁴⁵⁶ : OMe], [BB2942; E259, R ⁴⁵³ : CF ₃ , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2943; E 259, R ⁴⁵³ : H, R ⁴⁵⁴ : CF ₃ , ^{R 455: H, R 456:} H], [BB2944; E259, R 453: H, R 454: H, R 455: CF 3, R 456: H], [BB2945; E259, R 453: H, R 454 : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : CF ₃ ], [BB 2946; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2947; E 260, R ⁴⁵³ : F , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2948; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : F, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2949; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : F, R ⁴⁵⁶ : H], [BB 2950; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : F], [BB 2951; E 260, R ⁴⁵³ : Cl, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2952; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : Cl, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2953; E260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Cl, R ⁴⁵⁶ : H], [BB 2954; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Cl], [ BB 2 955; E 260, R ⁴⁵³ : Me, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2956; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : Me, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H] [BB 2957; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : Me, R ⁴⁵⁶ : H], [BB 2958; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : Me], [BB 2959; E 260, R ^{4 53} : OMe, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2960; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : OMe, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 296 1; E 260 , R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : OMe, R ⁴⁵⁶ : H], [BB 2962; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : OMe], [BB 2 63 3 E260, R ⁴⁵³ : CF ₃ , R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : H], [BB 2964; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : CF ₃ , R ⁴⁵⁵ : H, R ⁴⁵⁶ : H ], [BB 2 965; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : CF ₃ , R ⁴⁵⁶ : H], [BB 2966; E 260, R ⁴⁵³ : H, R ⁴⁵⁴ : H, R ⁴⁵⁵ : H, R ⁴⁵⁶ : CF ₃ ], [BB2967; E261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H ], [BB2968; E261, R ⁴⁴² : F, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2969] E261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : F, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2 970; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : F, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2971; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : F, R ⁴⁴⁹ : H], [BB 2972; E 261, R ⁴⁴² : Cl, R ⁴⁴³ : H , R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2973; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : Cl, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : ^{H, R 449: H],} [BB2974; E261, R 442: H, R 443: H, R 444: H, R 445: H, R 446: Cl, R 447: H, R 448: H, R 449 : H], [BB 2 975; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : Cl, R ⁴⁴⁹ : H], [BB2976; E261, R ⁴⁴² : Me, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2977; E 261 , R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : Me, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2978; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : Me, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2979; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : Me, R ⁴⁴⁹ : H], [BB 2980; E 261, R ⁴⁴² : OMe, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2981; E261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : OMe, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2982; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H , R ⁴⁴⁶ : OMe, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2983; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : OMe, R ⁴⁴⁹ : H], [BB 2984; E 261, R ⁴⁴² : CF ₃ , R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2985; E 261, R ⁴⁴² : H, R ^{443: H, R 444: CF} 3, R 445: H, R 446: H, R 447: H, R 448: H, R 449: H], [BB2986; E261, R 442: H, R 443: H , R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : CF ₃ , R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2987; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : CF ₃ , R ⁴⁴⁹ : H], [BB 2988; E 261, R ⁴⁴² : F, R ⁴⁴³ : F, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2989; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : F, R ⁴⁴⁵ : F , R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2990; E 261, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : ^{F, R 447: F, R} 448: H, R 449: H], [BB2991; E261, R 442: H, R 443: H, R 444: H, R 445: H, R 446: H, R 447 ^{: H, R 448: F,} R 449: F], [BB2992; E262, R 442: H, R 443: H, R 444: H, R 445: H, R 446: H, R 447: H, R ^{448: H, R 449: H} ], [BB2993; E262, R 442: F, R 443: H, R 444: H, R 445: H, R 446: H, R 447: H, R 448: H, R ^4
49 : H], [BB 2994; E262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : F, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H] [BB2995; E262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : F, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2996; E262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : F, R ⁴⁴⁹ : H], [BB 2 997; E 262, R ⁴⁴² : Cl, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2998; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : Cl, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 2 999; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : Cl, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3000; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H , R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : Cl, R ⁴⁴⁹ : H],

[BB3001; E262, R ⁴⁴² : Me, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3002; E 262 , R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : Me, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3003; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : Me, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3004; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : Me, R ⁴⁴⁹ : H], [BB 3005; E 262, R ⁴⁴² : OMe, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3006; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : OMe, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3007; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H , R ⁴⁴⁶ : OMe, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3008; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : OMe, R ⁴⁴⁹ : H], [BB 3009; E 262, R ⁴⁴² : CF ₃ , R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ^{447: H, R 448: H} , R 449: H], [BB3010; E262, R 442: H, R 443: H, R 444: CF 3, R 445: H, R 446: H, R 447: H , R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3011; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : CF ₃ , R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3012; E 262, R ⁴⁴² : H, R ⁴⁴³ : H , R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : CF ₃ , R ⁴⁴⁹ : H], [BB 3013; E 262, R ⁴⁴² : F, R ⁴⁴³ : F, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3014; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : F, R ⁴⁴⁵ : F, R ⁴⁴⁶ : H, R ⁴⁴⁷ : H, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3015; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : F, R ⁴⁴⁷ : F, R ⁴⁴⁸ : H, R ⁴⁴⁹ : H], [BB 3016; E 262, R ⁴⁴² : H, R ⁴⁴³ : H, R ⁴⁴⁴ : H, R ⁴⁴⁵ : H, R ⁴⁴⁶ : H , R ⁴⁴⁷ : H, R ⁴⁴⁸ : F, R ⁴⁴⁹ : F].

Further, the present compounds AC1-BC1 to AC10200-BC5278 can be obtained according to the above-mentioned method. The present compounds AC1-BC1 to AC10200-BC5278 are compounds represented by the following formula (ACBC).
[Wherein, X ^{30 to} X ³⁹ each represent a substituent corresponding to each of the substituent numbers (MC1) AC 1 to AC 10 200 shown below, and E ¹⁰³ represents a substituent number (MC 2) BC 1 to BC 5278 shown below Each represents a corresponding substituent. ]
For example, AC 1 -BC 1 is a compound represented by the formula (ACBC), wherein X ^{30 to} X ³⁹ are substituent numbers AC 1 (X ³⁴ and X ³⁹ are oxygen atoms, X ^{30 to} X ³³ and X ^{35 to} X ³⁸ are hydrogen Represents an atom), and E ¹⁰³ represents a compound in which the substituent number (MC 2) is BC 1 (pyrazol-1-yl group), and is represented by the following formula.

[Substituent group number ^{(MC1); X 30, X} 31, X 32, X 33, X 34, X 35, X 36, X 37, X 38, X 39], [AC1; H, H, H, H, O, H, H, H, H, O], [AC 2; H, H, H, H, H, O, F, H, H, O], [AC 3; H, H, H, H, O, Cl, H, H, H, O], [AC 4; H, H, H, H, O, Br, H, H, H, O], [AC 5; H, H, H, H, O, I, I, H, H, H, O], [AC 6; H, H, H, H, O, Me, H, H, H, O], [AC 7; H, H, H, H, O, Et, H, O, H, H, O], [AC 8; H, H, H, H, O, Pr, H, H, H, O], [AC 9; H, H, H, H, O, i-Pr, H, H, H, O], [ AC10; H, H, H, H, O, CH = CH 2, H, H, H, O], [AC11; H, H, H, H, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 12; H, H, H, H, O, C≡CH, H, H, H, O], [AC 13; H, H, H, H H, O, C≡CCH ₃ , H, H, H, O], [AC 14; H, H, H, H, O, c-Pr, H, H, O], [AC 15; H, H , H, H, O, OMe, H, H, H, O], [AC 16; H, H, H, H, O, OEt, H, H, H, O], [AC 17; H, H, H , H, O, Oi-Pr, H, H, H, O, [AC 18; H, H, H, H, O, SMe, H, H, O], [AC 19; H, H, H , H, O, SEt, H , H, H, O], [AC20; H, H, H, H, O, CH 2 F, H, H, H, O], [AC21; H, H, H _{, H, O, CHF 2,} H, H, H, O], [AC22; H, H, H, H, O, CF 3, H, H, H, O], [AC23; H, H, H _{, H, O, OCH 2 F} , H, H, H, O], [AC24; H, H, H, H, O, OCHF 2, H, H, H, O], [AC25; H, H, _{H, H, O, OCF 3} , H, H, H, O], [AC26; H, H, H, H, O, SCH 2 F, H, H, H, O], [AC27; H, H , H, H, O, SCHF 2, H, H, H, O], [AC28; H, H, H, H, O, SCF 3, H, H, H, O], [AC29; H, H , H, H, O, CN , H, H, H, O], [AC30; H, H, H, H, O, NO 2, H, H, H, O], [AC31; H, H, H, Me, O, H, H, H, O], [AC 32; H, H, H, Me, O, F, H, H, O], [AC 33 H, H, H, H, Me, O, Cl, H, H, H, O], [AC 34; H, H, H, Me, O, Br, H, H, O], [AC 35; H , H, H, Me, O, I, H, H, H, O], [AC 36; H, H, H, Me, O, Me, H, H, H, O], [AC 37; H, H , H, Me, O, Et, H, H, H, O], [AC 38; H, H, H, Me, O, Pr, H, H, H, O], [AC 39; H, H, H] , Me, O, i-Pr , H, H, H, O], [AC40; H, H, H, Me, O, CH = CH 2, H, H, H, O], [AC41; H, H, H, Me, O, C (CH 3) = CH 2, H, H, H, O], [AC42; H, H, H, Me, O, C≡CH, H, H, H, O ], [AC 43; H, H, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 44; H, H, H, Me, O, c-Pr, H, H, H, O], [AC 45; H, H, H, Me, O, OMe, H, H, H, O], [AC 46; H, H, H, Me, O, OE t, H, H, H, H O], [AC 47; H, H, H, Me, O, Oi-Pr, H, H, H, O], [AC 48; H, H, H, Me, O, SMe, H, H, H, H, O], [AC 49; H, H, H, Me, O, SE t, H, H, H, O], [AC 50; H, H, H, Me, O, CH ₂ F, H, H, H, H, O], [AC51; H, H, H, Me, O, CHF 2, H, H, H, O], [AC52; H, H, H, Me, O, CF 3, H, H, H, O], [AC 53; H, H, H, Me, O, OCH ₂ F, H, H, H, O], [AC 54; H, H, H, Me, O, OCHF ₂ , H, H, H , O], [AC 55; H, H, H, Me, O, OCF ₃ , H, H, O], [AC 56; H, H, H, Me, O, SCH ₂ F, H, H, H H, O], [AC 57; H, H, H, Me, O, SCHF ₂ , H, H, H, O], [AC 58; H, H, H, Me, O, SCF ₃ , H, H, H, H, O], [AC 59; H, H, H, Me, O, CN, H, H, H, O], [AC 60; H, H, H, Me, O, NO ₂ , H, H, H , O], [AC 61; H, H, H, Et, O, H, H, H, O], [AC 62; H, H, H, Et, O, F, H, H , H, O], [AC 63; H, H, H, Et, O, Cl, H, H, O], [AC 64; H, H, H, Et, O, Br, H, H, H , O], [AC 65; H, H, H, Et, O, I, H, H, H, O], [AC 66; H, H, H, Et, O, Me, H, H, H, O ], [AC 67; H, H, H, H, Et, O, Et, H, H, H, O], [AC 68; H, H, H, Et, O, Pr, H, H, H, O], [AC69; H, H, H , Et, O, i-Pr, H, H, H, O], [AC70; H, H, H, Et, O, CH = CH 2, H, H, H, O], [AC 71; H, H, H, Et, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 72; H, H, H, Et, O, C≡CH H, H, H, O], [AC 73; H, H, H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 74; H, H, H, Et, O, c-Pr, H, H, H, O], [AC 75; H, H, H, Et, O, OMe, H, H, H, O], [AC 76; H, H, H, Et, O, O Et, H, H, H, O], [AC 77; H, H, H, Et, O, Oi-Pr, H, H, H, O], [AC 78; H, H, H, Et, O, SMe, H, H, H, O], [AC 79; H, H, H, Et, O, SE, H, H, H, O], [AC 80; H, H, H, Et, O, CH ₂ F, H, H, H, O], [AC81; H, H, H, Et, O, CHF 2, H, H, H, O], [AC82; H, H, H, Et, O, CF ₃ , H, H, H, O], [AC 83; H, H, H, Et, O, OCH ₂ F, H, H, H, O], [AC 84; H, H, H, Et, O, _{OCHF 2, H, H, H} , O], [AC85; H, H, H, Et, O, OCF 3, H, H, H, O], [AC86; H, H, H, Et, O, SCH ₂ F, H, H, H, O], [AC 87; H, H, H, Et, O, SCHF ₂ , H, H, H, O], [AC 88; H, H, H, Et, O , SCF ₃ , H, H, H, O], [AC 89; H, H, H, Et, O, CN, H, H, H, O], [AC 90; H, H, H, Et, O, _{NO 2, H, H, H} , O], [AC91; H, H, H, Pr, O, H, H, H, H, O], [AC92; H, H, H, Pr, O, F H, H, H, O], [AC 93; H, H, H, Pr, O, Cl, H, H, H, O], [AC 94; H, H, H, Pr, O, Br, H, H, H, O], [AC95; H, H, H, Pr, O, I, H, H, H, O], [AC 96; H, H, H, Pr, O, Me, H, H, H, O], [AC 97; H, H, H, Pr, O, Et, H, H, H, O], [AC 98; H, H, H, Pr, O, Pr, H, H, H, O], [AC 99; H, H, H, Pr, O, i-Pr, H, H, H, O],

[AC100; H, H, H , Pr, O, CH = CH 2, H, H, H, O], [AC101; H, H, H, Pr, O, C (CH 3) = CH 2, H , H, H, O], [AC 102; H, H, H, Pr, O, C≡CH, H, H, H, O], [AC 103; H, H, H, Pr, O, C≡ CCH ₃ , H, H, H, O], [AC 104; H, H, H, Pr, O, c-Pr, H, H, H, O], [AC 105; H, H, H, Pr, O, OMe, H, H, H, O], [AC 106; H, H, H, Pr, O, OEt, H, H, H, O], [AC 107; H, H, H, Pr, O, Oi- Pr, H, H, H, O], [AC 108; H, H, H, Pr, O, SMe, H, H, H, O], [AC 109; H, H, H, Pr, O, SEt, H, H, H, O], [AC 110; H, H, H, Pr, O, CH ₂ F, H, H, H, O], [AC 111; H, H, H, Pr, O, CHF ₂ , H, H, H, O ], [AC112; H, H, H, Pr, O, CF 3, H, H, H, O], [AC113; H, H, H, Pr, O, OCH 2 F, H, H, H, O], [AC114; H, H, H, Pr, O, OCHF 2, H, H, H, O], [AC115; H, H, H, Pr, O, OCF _{3, H, H, H,} O], [AC116; H, H, H, Pr, O, SCH 2 F, H, H, H, O], [AC117; H, H, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 118; H, H, H, H, Pr, O, SCF ₃ , H, H, H, O], [AC 119; H, H, H, Pr, O, CN, H, H, H, O], [AC 120; H, H, H, Pr, O, NO ₂ , H, H, H, O], [AC 121; H, H, H, i-Pr, O , H, H, H, H, O], [AC 122; H, H, H, i-Pr, O, F, H, H, H, O], [AC 123; H, H, H, i-Pr , O, Cl, H, H, H, O, [AC 124; H, H, H, i-Pr, O, Br, H, H, H, O], [AC 125; H, H, H, i -Pr, O, I, H, H, H, O], [AC 126; H, H, H, i-Pr, O, Me, H, H, H, O], [AC 127; H, H, H , i-Pr, O, Et, H, H, H, O], [AC 128; H, H, H, i-Pr, O, Pr, H, H, H, O], [AC 129; H, H , H, i-Pr, O, i-Pr, H, H, H, O], [A C130; H, H, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC131; H, H, H, i-Pr, O, C (CH 3) = CH ₂ , H, H, H, O], [AC 132; H, H, H, i-Pr, O, C≡CH, H, H, H, O], [AC 133; H, H, H, i- Pr, O, C≡CCH ₃ , H, H, H, O], [AC 134; H, H, H, i-Pr, O, c-Pr, H, H, H, O], [AC 135; H , H, H, i-Pr, O, OMe, H, H, H, O], [AC 136; H, H, H, i-Pr, O, OEt, H, H, H, O], [AC 137 H, H, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 138; H, H, H, i-Pr, O, SMe, H, H, H, O ], [AC 139; H, H, H, i, Pr, O, SEt, H, H, H, O], [AC 140; H, H, H, i, Pr, O, CH ₂ F, H, H , H, O], [AC 141; H, H, H, i-Pr, O, CHF ₂ , H, H, H, O], [AC 142; H, H, H, i-Pr, O, CF ₃ , H, H, H, O], [AC 143; H, H, H, i-Pr, O, OCH ₂ F, H, H, H, O], [AC 144; H, H, H, i-Pr , O, OCHF ₂ , H, H, H, O], [AC145; H, H, H, i-Pr, O, OCF ₃ , H, H, H, O], [AC 146; H, H, H , i-Pr, O, SCH ₂ F, H, H, H, O], [AC 147; H, H, H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 148; H, H, H, i- Pr, O, SCF 3, H, H, H, O], [AC149; H, H, H, i-Pr, O, CN, H, H, H, O], [AC 150; H, H, H, i-Pr, O, NO ₂ , H, H, O], [AC 151; H, H, H, c, Pr, O, H, H, H, H, H, O], [AC 152; H, H, H, c, Pr, O, F, H, H, O], [AC 153; H, H, H, c, Pr, O, Cl, H, H, H, H, O], [AC 154; H, H, H, c-Pr, O, Br, H, H, H, O], [AC 155; H, H, H, c-Pr, O, I, H, H, H, O], [AC 156; H, H, H, c-Pr, O, Me, H, H, H, O], [AC 157; H, H, H, c-Pr, O, Et, Et, H, H, H, O], [AC158; H, H, H, c-Pr, O, Pr, H, H, H , O], [AC 159; H, H, H, c-Pr, O, i-Pr, H, H, H, O], [AC 160; H, H, H, c-Pr, O, CH = CH _{2, H, H, H,} O], [AC161; H, H, H, c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC162; H, H , H, c-Pr, O, C≡CH, H, H, H, O], [AC 163; H, H, H, c, Pr, O, C≡ CCH ₃ , H, H, H, O] , [AC 164; H, H, H, c-Pr, O, c-Pr, H, H, H, O], [AC 165; H, H, H, c-Pr, O, OMe, H, H, H, H, O], [AC 166; H, H, H, c-Pr, O, OEt, H, H, H, O], [AC 167; H, H, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 168; H, H, H, c-Pr, O, SMe, H, H, H, O], [AC 169; H, H, H, c-Pr, O, SEt, H, H, H, O], [AC 170; H, H, H, c-Pr, O, CH ₂ F, H, H, H, O], [AC 171; H, H, H, c- _{Pr, O, CHF 2, H} , H, H, O], [AC172; H, H, H, c-Pr, O, CF 3, H, H, H, O], [AC173; H, H, H, c-Pr, O, OCH 2 F, H, H, H, O], [AC174; H, H, H, c-Pr, O, OCHF 2, H, H, H, O], [AC175 ; H, H, H, c -Pr, O, OCF 3, H, H, H, O], [AC176; H, H, H, c-Pr, O, SCH 2 F, H, H, H, O], [AC 177; H, H, H, c, Pr, O, SCHF ₂ , H, H, H, O], [AC 178; H, H, H, c, Pr, O, SCF ₃ , H, H, H, H, O], [AC 179; H, H, H, c-Pr, O, CN, H, H, H, O], [AC 180; H, H, H, c-Pr, O, NO ₂ , H, H, H, O], [AC181; H, H, H, SMe, O, H, H, H, H, O], [AC 182; H, H, H, SMe, O, F, H , H, H, O], [AC183; H, H, H, SMe, O, Cl, H, H, H, O], [AC 184; H, H, H, SMe, O, Br, H, H , H, O], [AC 185; H, H, H, SMe, O, I, H, H, H, O], [AC 186; H, H, H, SMe, O, Me, H, H, H, H , O], [AC 187; H, H, H, SMe, O, Et, H, H, H, O], [AC 188; H, H, H, SMe, O, Pr, H, H, H, O], [AC 189; H, H, H, SMe, O, i-Pr, H, H, H, O], [AC190; H, H, H, SMe, O, CH = CH 2, H, H, H, O], [AC191; H, H, H, SMe, O, C (CH 3) = CH ₂ , H, H, H, O], [AC 192; H, H, H, SMe, O, C≡CH, H, H, H, O], [AC 193; H, H, H, SMe, O, C≡CCH ₃ , H, H, H, O], [AC 194; H, H, H, SMe, O, c-Pr, H, H, H, O], [AC 195; H, H, H , SMe, O, OMe, H, H, H, O], [AC 196; H, H, H, SMe, O, OEt, H, H, H, O], [AC 197; H, H, H, SMe , O, Oi-Pr, H, H, H, O, [AC 198; H, H, H, SMe, O, SMe, H, H, H, O], [AC 199; H, H, H, SMe , O, SEt, H, H, H, O],

[AC200; H, H, H , SMe, O, CH 2 F, H, H, H, O], [AC201; H, H, H, SMe, O, CHF 2, H, H, H, O] , [AC202; H, H, H, SMe, O, CF 3, H, H, H, O], [AC203; H, H, H, SMe, O, OCH 2 F, H, H, H, O ], [AC204; H, H , H, SMe, O, OCHF 2, H, H, H, O], [AC205; H, H, H, SMe, O, OCF 3, H, H, H, O ], [AC206; H, H , H, SMe, O, SCH 2 F, H, H, H, O], [AC207; H, H, H, SMe, O, SCHF 2, H, H, H, O], [AC208; H, H, H, SMe, O, SCF 3, H, H, H, O], [AC209; H, H, H, SMe, O, CN, H, H, H, O ], [AC 210; H, H, H, SMe, O, NO ₂ , H, H, O], [AC 211; H, H, H, OMe, O, H, H, H, H, O] , [AC212; H, H, H, OMe, O, F, H, H, O], [AC 213; H, H, H, OMe, O, Cl, H, H, H, O], [AC 212; AC 214; H, H, H, OMe, O, Br, H, H, O], [AC 215; H, H, H, OMe, O, I, H, H, H, O], [AC 216; H, H, H, OMe, O, Me, H, H, H, O], [AC 217; H, H, H, OMe, O, Et, H, H, H, O], [AC 218; H, H, H, OMe, O, Pr, H, H, H, O], [AC 219; H, H, H, OMe, O, i-Pr, H, H, H, O], [AC 220; H, H, H, OMe, O, CH = CH 2, H, H, H, O], [AC221; H, H, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC 222; H, H, H, H, OMe, O, C≡CH, H, H, H, O], [AC 223; H, H, H, OMe, O, C≡ CCH ₃ , H, H , H, O], [AC224; H, H, H, OMe, O, c-Pr, H, H, H, O], [AC 225; H, H, H, OMe, O, OMe, H, H , H, O], [AC226; H, H, H, OMe, O, OEt, H, H, H, O], [AC 227; H, H, H, OMe, O, Oi-Pr, H, H , H, O], [AC 228; H, H, H, OMe, O, SMe, H, H, H, O], [AC 229; H, H, H, OMe, O, SE t , H, H, H, O ], [AC230; H, H, H, OMe, O, CH 2 F, H, H, H, O], [AC231; H, H, H, OMe, O, CHF _{2, H, H, H,} O], [AC232; H, H, H, OMe, O, CF 3, H, H, H, O], [AC233; H, H, H, OMe, O, OCH ₂ F, H, H, H, O], [AC 234; H, H, H, OMe, O, OCHF ₂ , H, H, H, O], [AC 235; H, H, H, OMe, O, OCF ₃ , H, H, H, O], [AC 236; H, H, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 237; H, H, H, OMe, O , SCHF ₂ , H, H, H, O], [AC 238; H, H, H, OMe, O, SCF ₃ , H, H, H, O], [AC 239: H, H, H, OMe, O , CN, H, H, H, O], [AC 240; H, H, H, OMe, O, NO ₂ , H, H, H, O], [AC 241; H, H, H, F, O, H, H, H, H, O], [AC 242; H, H, H, F, O, F, H, H, H, O], [AC 243; H, H, H, F, O, Cl, H, H, H, O], [AC244; H, H, H, F, O, Br, H, H, H, O], [AC 245; H, H, H, F, O, I, H, H, H, O], [AC 246; H, H, H, F, O, Me, H, H, H, O], [AC 247; H, H, H, F, O, Et, H, H, H, H, O], [AC 248; H, H, H, F, O, Pr, H, H, H, O], [AC 249; H, H, H, F, O, i-Pr, H, H, H, H, O], [AC250; H, H, H, F, O, CH = CH 2, H, H, H, O], [AC251; H, H, H, F, O, C (CH 3) = CH ₂ , H, H, H, O], [AC 252; H, H, H, F, O, C≡CH, H, H, H, O], [AC 253; H, H, H, F, O, C≡CCH ₃ , H, H, H, O], [AC254; H, H, H, F, O, c-Pr, H, H, H, O], [AC 255; H, H, H , F, O, OMe, H, H, H, O], [AC 256; H, H, H, F, O, OEt, H, H, H, O], [AC 257; H, H, H, F , O, Oi-Pr, H, H, H, O, [AC258; H, H, H, F, O, SMe, H, H, H, O], [AC 259: H, H, H, F , O, SEt, H, H, H, O], [AC 260; H, H, H, F, O, C H ₂ F, H, H, H, O], [AC 261; H, H, H, F, O, CHF ₂ , H, H, H, O], [AC 262; H, H, H, F, O _{, CF 3, H, H,} H, O], [AC263; H, H, H, F, O, OCH 2 F, H, H, H, O], [AC264; H, H, H, F, _{O, OCHF 2, H, H} , H, O], [AC265; H, H, H, F, O, OCF 3, H, H, H, O], [AC266; H, H, H, F, O, SCH ₂ F, H, H, H, O], [AC 267; H, H, H, F, O, SCHF ₂ , H, H, H, O], [AC 268; H, H, H, F , O, SCF ₃ , H, H, H, O], [AC 269; H, H, H, F, O, CN, H, H, H, O], [AC 270; H, H, H, F, _{O, NO 2, H, H} , H, O], [AC271; H, H, H, Cl, O, H, H, H, H, O], [AC272; H, H, H, Cl, O , F, H, H, H, O], [AC 273; H, H, H, H, Cl, O, Cl, H, H, H, O], [AC 274; H, H, H, Cl, O, Br , H, H, H, O], [AC 275; H, H, H, Cl, O, I, H, H, H, O], [AC 276; H, H, H, Cl, O, Me, H , H, H, O], [AC 277; H, H, H, Cl, O, Et, H, H, H, O], [AC 278; H, H, H, Cl, O, Pr, H, H , H, O], [AC 279; H, H, H, Cl, O, i-Pr, H, H, H, O], [AC 280; H, H, H, Cl, O, CH = CH ₂ , H, H, H, O] , [AC281; H, H, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC282; H, H, H, Cl , O, C≡CH, H, H, H, O, [AC 283; H, H, H, Cl, O, C≡ CCH ₃ , H, H, H, O], [AC 284; H, H, H, H, Cl, O, c-Pr, H, H, H, O], [AC 285; H, H, H, H, Cl, O, OMe, H, H, H, O], [AC 286; H, H, H, H H, Cl, O, OEt, H, H, H, O], [AC 287; H, H, H, H, Cl, O, Oi-Pr, H, H, H, O], [AC 288; H, H, H H, Cl, O, SMe, H, H, H, O], [AC 289; H, H, H, Cl, O, SE t, H, H, H, O], [AC 290; H, H, H, _{Cl, O, CH 2 F,} H, H, H, O], [AC291; H, H, H, Cl _{, O, CHF 2, H,} H, H, O], [AC292; H, H, H, Cl, O, CF 3, H, H, H, O], [AC293; H, H, H, Cl _{, O, OCH 2 F, H} , H, H, O], [AC294; H, H, H, Cl, O, OCHF 2, H, H, H, O], [AC295; H, H, H, _{Cl, O, OCF 3, H} , H, H, O], [AC296; H, H, H, Cl, O, SCH 2 F, H, H, H, O], [AC297; H, H, H _{, Cl, O, SCHF 2,} H, H, H, O], [AC298; H, H, H, Cl, O, SCF 3, H, H, H, O], [AC299; H, H, H , Cl, O, CN, H, H, H, O],

[AC 300; H, H, H, H, Cl, O, NO ₂ , H, H, H, O], [AC 301; H, H, H, Br, O, H, H, H, H, O], [AC 300 AC 302; H, H, H, H, Br, O, F, H, H, O], [AC 303; H, H, H, Br, O, Cl, H, H, H, O], [AC 304; H, H, H, H, Br, O, Br, H, H, H, O], [AC 305; H, H, H, Br, O, I, H, H, O], [AC 306; H, H, H, H, Br, O, Me, H, H, H, O], [AC 307; H, H, H, Br, O, Et, H, H, H, O], [AC 308; H, H, H, H H, Br, O, Pr, H, H, H, O], [AC 309; H, H, H, Br, O, i-Pr, H, H, H, O], [AC 310; H, H, H, H H, Br, O, CH = CH 2, H, H, H, O], [AC311; H, H, H, Br, O, C (CH 3) = CH 2, H, H, H, O] , [AC 312; H, H, H, H, Br, O, C≡CH, H, H, H, O], [AC 313; H, H, H, H, Br, O, C≡ CCH ₃ , H, H, H H, H, H, Br, O, c-Pr, H, H, H, O], [AC 315; H, H, H, Br, O, OMe, H, H, H] H, H, H, Br, O, OEt, H, H, H, O], [AC 317; H, H, H, H, Br, O, Oi-Pr, H, H, H H, H, H, Br, O, SMe, H, H, H, O], [AC 319: H, H, H, Br, O, SE t, H, H, H, O ], [AC320; H, H , H, Br, O, CH 2 F, H, H, H, O], [AC321; H, H, H, Br, O, CHF 2, H, H, H, O], [AC322; H, H, H, Br, O, CF 3, H, H, H, O], [AC323; H, H, H, Br, O, OCH 2 F, H, H, H , O], [AC 324; H, H, H, Br, O, OCHF ₂ , H, H, H, O], [AC 325; H, H, H, H, Br, O, OCF ₃ , H, H, H H, H, H, Br, O, SCH ₂ F, H, H, H, O], [AC 327; H, H, H, H, Br, O, SCHF ₂ , H, H, H H, O], [AC 328; H, H, H, Br, O, SCF ₃ , H, H, H, O], [AC 329: H, H, H, Br, O, CN, H, H, H , O], [AC 330; H, H, H, Br, O, NO ₂ , H, H, H, O], [AC 331; H, Me, H, H, O, H, H, H, H, O], [AC 332; H, Me, H, H, O, F, F, H, H, H, O], [AC333; H, Me, H, H, O, Cl, H, H, H, O], [AC 334; H, Me, H, H, O, Br, H, H H, H, O], [AC 335; H, Me, H, H, O, I, H, H, H, O], [AC 336: H, Me, H, H, O, Me, H, H, H, H, O], [AC 337; H, Me, H, H, O, Et, H, H, H, O], [AC 338; H, Me, H, H, O, Pr, H, H, H, H, H, Me, H, H, O, i-Pr, H, H, H, O], [AC 340; H, Me, H, H, O, CHHCH ₂ , H, H] , H, O], [AC341 ; H, Me, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC342; H, Me, H, H, O, C≡CH, H, H, H, O], [AC 343; H, Me, H, H, O, C≡CCH ₃ , H, H, H, O], [AC 344; H, Me, H, H , O, c-Pr, H, H, H, O], [AC 345; H, Me, H, H, O, OMe, H, H, H, O], [AC346; H, Me, H, H] , O, OEt, H, H, H, O, [AC 347; H, Me, H, H, O, Oi-Pr, H, H, H, O], [AC 348: H, Me, H, H , O, SMe, H, H, H, O], [AC 349; H, Me, H, H, O, SE, H, H, H, O], [AC 350; H, Me, H, H, O _{, CH 2 F, H, H} , H, O], [AC351; H, Me, H, H, O, CHF 2, H, H, H, O], [AC352; H, Me, H, H, _{O, CF 3, H, H} , H, O], [AC353; H, Me, H, H, O, OCH 2 F, H, H, H, O], [AC354; H, Me, H, H , O, OCHF ₂ , H, H, H, O], [AC 355; H, Me, H, H, O, OCF ₃ , H, H, H, O], [AC 356; H, Me, H, H , O, SCH ₂ F, H, H, H, O, [AC 357; H, Me, H, H, O, SCHF ₂ , H, H, H, O], [AC 358; H, Me, H, O _{H, O, SCF 3, H} , H, H, O], [AC359; H, Me, H, H, O, CN, H, H, H, O], [AC360; H, Me, H, H , O, NO ₂ , H, H, H, O], [AC 361; H, Me, H, Me, O, H, H, H, H, O], [AC 362; H, Me, H, Me, O, F, H, H, O], [AC 363; H, Me, H, Me, O, Cl, H, H, H, O], [AC 364; H, Me, H, Me, O, Br, H, H, H, O], [AC 365; H, Me, H, Me, O, I, H, H, H, O], [AC 366; H, Me, H, Me, O, Me, H, H, H, O], [AC 367; H, Me, H, O Me, O, Et, H, H, H, O, [AC 368; H, Me, H, Me, O, Pr, H, H, H, O], [AC 369; H, Me, H, Me, O, i-Pr, H, H, H, O], [AC370; H, Me, H, Me, O, CH = CH 2, H, H, H, O], [AC371; H, Me, H , Me, O, C (CH 3) = CH 2, H, H, H, O], [AC372; H, Me, H, Me, O, C≡CH, H, H, H, O], [ AC 373; H, Me, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 374; H, Me, H, Me, O, c-Pr, H, H, H, O H, Me, H, Me, O, OMe, H, H, H, O], [AC 376; H, Me, H, Me, O, OEt, H, H, H, O], [AC 377; H, Me, H, Me, O, Oi-Pr, H, H, H, O], [AC 378; H, Me, H, Me, O, SMe, H, H, H, O], [AC 379; H, Me, H, Me, O, SEt, H, H, H, O], [AC 380; H, Me, H, Me, O, CH ₂ F, H, H, H, O], [AC381; H, Me, H , Me, O, CHF 2, H, H, H, O], [AC382; H, Me, H, Me, O, CF 3, H, H, H, O], [AC 383; H, Me, H, Me, O, OCH ₂ F, H, H, H, O], [AC 384; H, Me, H, Me, O, OCHF ₂ , H, H, H, O] , [AC385; H, Me, H, Me, O, OCF 3, H, H, H, O], [AC386; H, Me, H, Me, O, SCH 2 F, H, H, H, O H, Me, H, Me, O, SCHF ₂ , H, H, H, O], [AC 388; H, Me, H, Me, O, SCF ₃ , H, H, H, O] H, Me, H, Me, O, CN, H, H, H, O], [AC 390; H, Me, H, Me, O, NO ₂ , H, H, H, H] O], [AC 391; H, Me, H, Et, O, H, H, H, O], [AC 392; H, Me, H, Et, O, F, H, H, H, O] , [AC 393; H, Me, H, Et, O, Cl, H, H, O], [AC 394; H, Me, H, Et, O, Br, H, H, H, O], [AC 394; AC 395; H, Me, H, Et, O, I, H, H, O], [AC 396; H, Me, H, Et, O, Me, H, H, H, O], [AC 397; H, Me, H, Et, O, Et, H, H, H, O], [AC 398; H, Me, H, Et, O, Pr, H, H, H, O],

[AC399; H, Me, H , Et, O, i-Pr, H, H, H, O], [AC400; H, Me, H, Et, O, CH = CH 2, H, H, H, O], [AC 401; H, Me, H, Et, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 402; H, Me, H, Et, O, C≡CH H, H, H, O], [AC 403; H, Me, H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 404; H, Me, H, Et, O, c-Pr, H, H, H, O], [AC 405; H, Me, H, Et, O, OMe, H, H, H, O], [AC 406; H, Me, H, Et, O, OEt, H, H, H, O], [AC 407; H, Me, H, Et, O, Oi-Pr, H, H, H, O], [AC 408; H, Me, H, Et, O, SMe, H, H, H, O], [AC 409; H, Me, H, Et, O, SE t, H, H, H, O], [AC 410; H, Me, H, Et, O, CH ₂ F, H, H, H, O], [AC411; H, Me, H, Et, O, CHF 2, H, H, H, O], [AC412; H, Me, H, Et, O, CF _{3, H, H, H,} O], [AC413; H, Me, H, Et, O, OCH 2 F, H, H, H, O], [AC414; H, Me, H, Et, O, _{OCHF 2, H, H, H} , O], [AC415; H, Me, H, Et, O, OCF 3, H, H, H, O], [AC416; H, Me, H, Et, O, SCH ₂ F, H, H, H, O], [AC 417; H, Me, H, Et, O, SCHF ₂ , H, H, H, O], [AC 418; H, Me, H, Et, O , SCF ₃ , H, H, H, O], [AC 419; H, Me, H, Et, O, CN, H, H, H, O], [AC 420; H, Me, H, Et, O, _{NO 2, H, H, H} , O], [AC421; H, Me, H, Pr, O, H, H, H, H, O], [AC422; H, Me, H, Pr, O, F H, H, H, O], [AC 423; H, Me, H, Pr, O, Cl, H, H, H, O], [AC 424; H, Me, H, Pr, O, Br, H , H, H, O], [AC 425; H, Me, H, Pr, O, I, H, H, H, O], [AC 426; H, Me, H, Pr, O, Me, H, H , H, O], [AC 427; H, Me, H, Pr, O, Et, H, H, H, O], [AC 428; H, Me, H, Pr, O, Pr , H, H, H, O], [AC 429; H, Me, H, Pr, O, i-Pr, H, H, H, O], [AC 430; H, Me, H, Pr, O, CH _{= CH 2, H, H,} H, O], [AC431; H, Me, H, Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC432; H, Me , H, Pr, O, C≡CH, H, H, H, O], [AC 433; H, Me, H, Pr, O, C≡ CCH ₃ , H, H, H, O], [AC 434; H, Me, H, Pr, O, c-Pr, H, H, H, O], [AC 435; H, Me, H, Pr, O, OMe, H, H, H, O], [AC 436; H, Me, H, Pr, O, OEt, H, H, H, O], [AC 437; H, Me, H, Pr, O, Oi-Pr, H, H, H, O], [AC 438; H, Me, H, Pr, O, SMe, H, H, H, O], [AC 439: H, Me, H, Pr, O, SE t, H, H, H, O], [AC 440; H, Me, H, Pr, O, CH 2 F, H, H, H, O], [AC441; H, Me, H, Pr, O, CHF 2, H, H, H, O], [AC442; H , Me, H, Pr, O , CF 3, H, H, H, O], [AC443; H, Me, H, Pr, O, OCH 2 F, H, H, H, O], [AC444; H, Me, H, Pr, O, OCHF 2, H, H, H, O], [AC445; H, Me, H, Pr, O, OCF 3, H, H, H, O], [AC446; H, Me, H, Pr, O, SCH ₂ F, H, H, H, O], [AC 447; H, Me, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 448 H, Me, H, Pr, O, SCF ₃ , H, H, H, O], [AC 449; H, Me, H, Pr, O, CN, H, H, H, O], [AC 450; H, Me, H, Pr, O, NO 2, H, H, H, O], [AC451; H, Me, H, i-Pr, O, H, H, H, H, O], [AC452 H, Me, H, i-Pr, O, F, H, H, H, O], [AC 453; H, Me, H, i-Pr, O, Cl, H, H, H, O], [AC454; H, Me, H, i-Pr, O, Br, H, H, O], [AC 455; H, Me, H, i-Pr, O, I, H, H, H, O H, Me, H, i-Pr, O, Me, H, H, H, O], [AC 457; H, Me, H, i-Pr, O, Et, H, H, H] , O], [AC 458; H, Me, H, i-Pr, O, Pr, H, H, H, O], [AC 459; H, Me, H, i-Pr, O, i-Pr, H, H, H, O], [ AC460; H, Me, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC461; H, Me, H, i-Pr, O , C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 462; H, Me, H, i-Pr, O, C≡CH, H, H, H, O], [AC 463; H, Me, H, i-Pr, O, C≡CCH ₃ , H, H, H, O], [AC464; H, Me, H, i-Pr, O, c-Pr, H, H, H , O], [AC 465; H, Me, H, i-Pr, O, OMe, H, H, H, O], [AC 466: H, Me, H, i-Pr, O, OEt, H, H , H, O], [AC 467; H, Me, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 468; H, Me, H, i-Pr, O, SMe H, H, H, O], [AC 469; H, Me, H, i-Pr, O, SEt, H, H, H, O], [AC 470; H, Me, H, i-Pr, O _{, CH 2 F, H, H} , H, O], [AC471; H, Me, H, i-Pr, O, CHF 2, H, H, H, O], [AC472; H, Me, H, _{i-Pr, O, CF 3} , H, H, H, O], [AC473; H, Me, H, i-Pr, O, OCH 2 F, H, H, H, O], [AC474; H , Me, H, i-Pr , O, OCHF 2, H, H, H, O], [AC475; H, Me, H, i-Pr, O, OCF 3, H, H, H, O], [AC 476; H, Me, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 477; H, Me, H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC478; H, Me, H, i-Pr, O, SCF 3, H, H, H, O], [AC479; H, Me, H, i-Pr, O, CN, H H, H, O], [AC 480; H, Me, H, i-Pr, O, NO ₂ , H, H, H, O], [AC 481; H, Me, H, c-Pr, O, H, H, H, H, O], [AC 482; H, Me, H, c-Pr, O, F, H, H, H, O], [AC 483; H, Me, H, c-Pr, O, Cl, H, H, H, O], [AC 484; H, Me, H, c-Pr, O, Br, H, H, H, O], [AC 485; H, Me, H, c- Pr, O, I, H, H, H, O], [AC 486; H, Me, H, c-Pr, O, Me, H, H, H, O], [AC 487; H, Me, H, c-Pr, O, Et, Et, H, H, H, O], [AC 488; H, Me, H, c-Pr, O, Pr, H, H, H, O], [AC 489; H, Me, H, c-Pr, O, i-Pr, H, H, H, O], [AC490; H, Me, H, c-Pr, O, CH = CH 2, H, H, H, O], [AC491; H, Me, H , c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC492; H, Me, H, c-Pr, O, C≡CH, H, H, H, O], [AC 493; H, Me, H, c-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 494; H, Me, H, c-Pr, O, c-Pr H, H, H, O], [AC 495; H, Me, H, c-Pr, O, OMe, H, H, H, O], [AC 496; H, Me, H, c-Pr, O , OEt, H, H, H, O], [AC 497; H, Me, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 498; H, Me, H, c -Pr, O, SMe, H, H, H, O],

[AC499; H, Me, H , c-Pr, O, SEt, H, H, H, O], [AC500; H, Me, H, c-Pr, O, CH 2 F, H, H, H , O], [AC 501; H, Me, H, c-Pr, O, CHF ₂ , H, H, H, O], [AC 502; H, Me, H, c-Pr, O, CF ₃ , H ₃ , H, H, O], [AC 503; H, Me, H, c-Pr, O, OCH ₂ F, H, H, H, O], [AC 504; H, Me, H, c-Pr, O _{, OCHF 2, H, H,} H, O], [AC505; H, Me, H, c-Pr, O, OCF 3, H, H, H, O], [AC506; H, Me, H, c -Pr, O, SCH ₂ F, H, H, H, O, [AC 507; H, Me, H, c-Pr, O, SCHF ₂ , H, H, H, O], [AC 508; H, Me, H, c-Pr, O, SCF 3, H, H, H, O], [AC509; H, Me, H, c-Pr, O, CN, H, H, H, O], [AC510 H, Me, H, c-Pr, O, NO ₂ , H, H, H, O], [AC 511; H, Me, H, SMe, O, H, H, H, H, O], [AC 511; AC 512; H, Me, H, SMe, O, F, H, H, H, O], [AC 513: H, Me, H, SMe, O, Cl, H, H, H, O], [AC 514; H, Me, H, SMe, O, Br, H, H, H, O], [AC 515; H, Me, H, SMe, O, I, H, H, O, [AC 516: H, Me, H, SMe, O, Me, H, H, H, O], [AC 517; H, Me, H, SMe, O, Et, H, H, H, O], [AC 518: H, Me, H, SMe, O, Pr, H, H, H, O], [AC519; H, Me, H, SMe, O, i-Pr, H, H, H, O], [AC 520; H, Me, H, SMe, O, CH = CH 2, H, H, H, O], [AC521; H, Me, H, SMe, O, C (CH 3) = CH 2, H, H, H, O] [AC522; H, Me, H, SMe, O, C≡CH, H, H, H, O], [AC523; H, Me, H, SMe, O, C≡CCH ₃ , H, H, H H, Me, H, SMe, O, c-Pr, H, H, H, O], [AC 525; H, Me, H, SMe, O, OMe, H, H, H , O], [AC 526; H, Me, H, SMe, O, OEt, H, H, H, O], [AC 527; H, Me, H, SM e, O, Oi-Pr, H, H, H, O, [AC 528; H, Me, H, SMe, O, SMe, H, H, O, [AC 529; H, Me, H, SMe, O, SEt, H, H, H, O], [AC 530; H, Me, H, SMe, O, CH ₂ F, H, H, H, O], [AC 531; H, Me, H, _{SMe, O, CHF 2, H} , H, H, O], [AC532; H, Me, H, SMe, O, CF 3, H, H, H, O], [AC533; H, Me, H, _{SMe, O, OCH 2 F,} H, H, H, O], [AC534; H, Me, H, SMe, O, OCHF 2, H, H, H, O], [AC535; H, Me, H _{, SMe, O, OCF 3,} H, H, H, O], [AC536; H, Me, H, SMe, O, SCH 2 F, H, H, H, O], [AC537; H, Me, _{H, SMe, O, SCHF 2} , H, H, H, O], [AC538; H, Me, H, SMe, O, SCF 3, H, H, H, O], [AC539; H, Me, H, SMe, O, CN, H, H, H, H, O], [AC 540; H, Me, H, SMe, O, NO ₂ , H, H, H, O], [AC 541; H, Me, H , OMe, O, H, H, H, H, O], [AC 542; H, Me, H, OMe, O, F, H, H, H, O], [AC 543; H, Me, H, OMe , O, Cl, H, H, H, O], [AC 544; H, Me, H, OMe, O, Br, H, H, H, O], [AC 545; H, Me, H, OMe, O , I, H, H, H, O], [AC 546; H, Me, H, OMe, O, Me, H, H, H, O], [AC 547; H, Me, H, OMe, O, Et H, H, H, O], [AC 548; H, Me, H, OMe, O, Pr, H, H, H, O], [AC 549; H, Me, H, OMe, O, i-Pr , H, H, H, O ], [AC550; H, Me, H, OMe, O, CH = CH 2, H, H, H, O], [AC551; H, Me, H, OMe, O, _{C (CH 3) = CH 2} , H, H, H, O], [AC552; H, Me, H, OMe, O, C≡CH, H, H, H, O], [AC553; H, Me , H, OMe, O, C≡CCH ₃ , H, H, H, O], [AC 554; H, Me, H, OMe, O, c-Pr, H, H, H, O], [AC 555; H, Me, H, OMe, O, OMe, H, H, H, O], [AC 556; H, Me, H, OMe, O, OEt, H, H, H, O], [AC 557; H, Me, H, OMe, O, Oi-Pr, H, H, H, O], [AC 558; H, Me, H, OMe, O, SMe, H, H, H, O], [AC559; H, Me, H, OMe, O, SE t, H, H, H, O], [AC 560; H, Me, _{H, OMe, O, CH 2} F, H, H, H, O], [AC561; H, Me, H, OMe, O, CHF 2, H, H, H, O], [AC562; H, Me , H, OMe, O, CF 3, H, H, H, O], [AC563; H, Me, H, OMe, O, OCH 2 F, H, H, H, O], [AC564; H, Me, H, OMe, O, OCHF 2, H, H, H, O], [AC565; H, Me, H, OMe, O, OCF 3, H, H, H, O], [AC566; H, Me, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 567; H, Me, H, OMe, O, SCHF ₂ , H, H, H, O], [AC 568; H , Me, H, OMe, O, SCF ₃ , H, H, H, O], [AC 569; H, Me, H, OMe, O, CN, H, H, H, O], [AC 570; H, Me, H, OMe, O, NO 2, H, H, H, O], [AC571; H, Me, H, F, O, H, H, H, H, O], [AC572; H, Me , H, F, O, F, H, H, H, O], [AC 573; H, Me, H, F, O, Cl, H, H, H, O], [AC 574; H, Me, H , F, O, Br, H, H, H, O], [AC575; H, Me, H, F, O, I, H, H, O], [AC 576; H, Me, H, F] H, Me, H, H, H, O], [AC 577; H, Me, H, F, O, Et, H, H, H, O], [AC 578; H, Me, H, F, O , Pr, H, H, H, O], [AC579; H, Me, H, F, O, i-Pr, H, H, H, O], [AC 580; H, Me, H, F, O _{, CH = CH 2, H,} H, H, O], [AC581; H, Me, H, F, O, C (CH 3) = CH 2, H, H, H, O], [AC582; H , Me, H, F, O, C≡CH, H, H, H, O], [AC 583; H, Me, H, F, O, C≡ CCH ₃ , H, H, H, O], [C AC 584; H, Me, H, F, O, c-Pr, H, H, H, O], [AC 585; H, Me, H, F, O, OMe, H, H, H, O] [AC586; H, Me, H, F, O, OEt, H, H, H, O], [AC587; H, Me, H, F, O, Oi-Pr, H, H, H, O] , [AC 588; H, Me, H, F, O, S Me, H, H, H, O], [AC 589; H, Me, H, F, O, SE t, H, H, H, O], [AC 588; AC590; H, Me, H, F, O, CH 2 F, H, H, H, O], [AC591; H, Me, H, F, O, CHF 2, H, H, H, O], [AC 592; H, Me, H, F, O, CF ₃ , H, H, H, O], [AC 593; H, Me, H, F, O, OCH ₂ F, H, H, H, O] [AC 594; H, Me, H, F, O, OCHF ₂ , H, H, H, O], [AC 595; H, Me, H, F, O, OCF ₃ , H, H, H, O] , [AC 596; H, Me, H, F, O, SCH ₂ F, H, H, H, O], [AC 597; H, Me, H, F, O, SCHF ₂ , H, H, H, O ], [AC598; H, Me, H, F, O, SCF ₃ , H, H, H, O],

[AC599; H, Me, H , F, O, CN, H, H, H, O], [AC600; H, Me, H, F, O, NO 2, H, H, H, O], [ AC601; H, Me, H, Cl, O, H, H, H, O], [AC 602; H, Me, H, Cl, O, F, H, H, H, O], [AC 603; H, Me, H, Cl, O, Cl, H, H, H, O], [AC 604; H, Me, H, Cl, O, Br, H, H, O], [AC 605; H, Me, H, Cl, O, I, H, H, H, O], [AC 606; H, Me, H, Cl, O, Me, H, H, H, O], [AC 607; H, Me, H, Cl, O, Et, H, H, H, O], [AC 608; H, Me, H, Cl, O, Pr, H, H, H, O], [AC 609; H, Me, H, O Cl, O, i-Pr, H, H, H, O], [AC610; H, Me, H, Cl, O, CH = CH 2, H, H, H, O], [AC611; H, Me , H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC612; H, Me, H, Cl, O, C≡CH, H, H, H, O] [AC 613; H, Me, H, Cl, O, C≡CCH ₃ , H, H, H, O], [AC 614; H, Me, H, Cl, O, c-Pr, H, H, H , O], [AC 615; H, Me, H, Cl, O, OMe, H, H, H, O], [AC 616; H, Me, H, Cl, O, OEt, H, H, H, O H, Me, H, Cl, O, Oi-Pr, H, H, H, O], [AC 618; H, Me, H, Cl, O, SMe, H, H, H, O] H, Me, H, Cl, O, SEt, H, H, H, O], [AC 620; H, Me, H, Cl, O, CH ₂ F, H, H, H, O] ], [AC621; H, Me , H, Cl, O, CHF 2, H, H, H, O], [AC622; H, Me, H, Cl, O, CF 3, H, H, H, O H, Me, H, Cl, O, OCH ₂ F, H, H, H, O], [AC 624; H, Me, H, Cl, O, OCHF ₂ , H, H, H, O], [AC625; H, Me, H, Cl, O, OCF 3, H, H, H, O], [AC626; H, Me, H, Cl, O, SCH 2 F, H, H, H , O], [AC627; H , Me, H, Cl, O, SCHF 2, H, H, H, O], [AC628; H, Me, H, Cl, O, SCF 3, H , H, H, O], [AC 629; H, Me, H, Cl, O, CN, H, H, H, O], [AC 630; H, Me, H, Cl, O, NO ₂ , H, H, H, H, O], [AC 631; H, Me, H, Br, O, H, H, H, O], [AC 632; H, Me, H, Br, O, F, H, H, H, H, O], [AC 633; H, Me, H, Br, O, Cl, H, H, H, O], [AC 634; H, Me, H, Br, O, Br, H, H, H, H, O], [AC 635; H, Me, H, Br, O, I, H, H, O], [AC 636; H, Me, H, Br, O, Me, H, H, H, O] , [AC 637; H, Me, H, Br, O, Et, H, H, H, O], [AC 638; H, Me, H, Br, O, Pr, H, H, H, O], [AC 637; AC639; H, Me, H, Br, O, i-Pr, H, H, H, O], [AC640; H, Me, H, Br, O, CH = CH 2, H, H, H, O ], [AC641; H, Me , H, Br, O, C (CH 3) = CH 2, H, H, H, O], [AC642; H, Me, H, Br, O, C≡CH, H, H, H, O], [AC643; H, Me, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 644; H, Me, H, Br, O, c -Pr, H, H, H, O], [AC 645; H, Me, H, Br, O, OMe, H, H, H, O], [AC 646; H, Me, H, Br, O, OEt , H, H, H, O], [AC 647; H, Me, H, Br, O, Oi-Pr, H, H, H, O], [AC 648; H, Me, H, Br, O, SMe H, H, H, O], [AC 649; H, Me, H, Br, O, SE t, H, H, H, O], [AC 650; H, Me, H, Br, O, CH ₂ F , H, H, H, O ], [AC651; H, Me, H, Br, O, CHF 2, H, H, H, O], [AC652; H, Me, H, Br, O, CF 3 , H, H, H, O], [AC 653; H, Me, H, Br, O, OCH ₂ F, H, H, H, O], [AC 654; H, Me, H, Br, O, OCHF _{2, H, H, H,} O], [AC655; H, Me, H, Br, O, OCF 3, H, H, H, O], [AC656; H, Me, H, Br, O, SCH ₂ F, H, H, H, O], [AC 657; H, Me, H, Br, O, SCHF ₂ , H, H, H, O], [AC 658; H, Me, H, Br, O, SCF ₃ , H, H, H, O], [AC 659; H, Me, H, Br, O, CN, H, H, H, O], [AC 660; H, Me, H, Br, O , NO ₂ , H, H, H, O], [AC 661; H, Et, H, H, O, H, H, H, H, O], [AC 662; H, Et, H, H, O, F, H, H, H, O], [AC 663; H, Et, H, H, O, Cl, H, H, H, O], [AC 664; H, Et, H, H, O, Br, H, H, H, O], [AC 665; H, Et, H, H, O, I, H, H, H, O], [AC 666; H, Et, H, H, O, Me, H, H, H, O], [AC 667; H, Et, H, H, O, Et, H, H, H, O], [AC 668; H, Et, H, H, O, Pr, H, H, H, H, O], [AC669; H, Et, H, H, O, i-Pr, H, H, H, O], [AC670; H, Et, H, H, O, CH = CH 2, H , H, H, O], [AC671; H, Et, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC672; H, Et, H, H, O, C≡CH, H, H, H, O, [AC 673; H, Et, H, H, O, C≡ CCH ₃ , H, H, H, O], [AC 674; H, Et, H , H, O, c-Pr, H, H, H, O, [AC 675; H, Et, H, H, O, OMe, H, H, H, O], [AC 676; H, Et, H , H, O, OEt, H, H, H, O], [AC 677; H, Et, H, H, O, Oi-Pr, H, H, H, O], [AC 678; H, Et, H , H, O, SMe, H, H, H, O, [AC 679; H, Et, H, H, O, SE, H, H, H, O], [AC 680; H, Et, H, H] _{, O, CH 2 F, H} , H, H, O], [AC681; H, Et, H, H, O, CHF 2, H, H, H, O], [AC682; H, Et, H, _{H, O, CF 3, H} , H, H, O], [AC683; H, Et, H, H, O, OCH 2 F, H, H, H, O], [AC684; H, Et, H _{, H, O, OCHF 2,} H, H, H, O], [AC685; H, Et, H, H, O, OCF 3, H, H, H, O], [AC686; H, Et, H , H, O, SCH ₂ F, H, H, H, O], [AC 687; H, Et, H, H, O, SCHF ₂ , H, H, H, O], [AC 688; H, Et, H, H, O, SCF ₃ , H, H, H, O], [AC 689; H, Et, H, H, O, CN, H, H, H, O], [AC 690; H, Et, H, H, O, NO ₂ , H, H, H, O], [AC AC 691; H, Et, H, Me, O, H, H, H, O], [AC 692; H, Et, H, Me, O, F, H, H, H, O], [AC 693; H, Et, H, Me, O, Cl, H, H, H, O], [AC 694; H, Et, H, Me, O, Br, H, H, O], [AC 695; H, Et, H, Me, O, I, H, H, H, O], [AC 696; H, Et, H, Me, O, Me, H, H, H, O], [AC 697; H, Et, H, Me, O, Et, H, H, H, O],

[AC 698; H, Et, H, Me, O, Pr, H, H, H, O], [AC 699; H, Et, H, Me, O, i-Pr, H, H, H, O], [AC700; H, Et, H , Me, O, CH = CH 2, H, H, H, O], [AC701; H, Et, H, Me, O, C (CH 3) = CH 2, H , H, H, O], [AC 702; H, Et, H, Me, O, C≡CH, H, H, H, O], [AC 703; H, Et, H, Me, O, C≡ CCH ₃ , H, H, H, O], [AC 704; H, Et, H, Me, O, c-Pr, H, H, H, O], [AC 705; H, Et, H, Me, O, OMe, H, H, H, O], [AC 706; H, Et, H, Me, O, OEt, H, H, H, O], [AC 707; H, Et, H, Me, O, Oi- Pr, H, H, H, O], [AC 708; H, Et, H, Me, O, SMe, H, H, H, O], [AC 709; H, Et, H, Me, O, SE t, H, H, H, O] , [AC710; H, Et, H, Me, O, CH 2 F, H, H, H, O], [AC711; H, Et, H, Me, O, CHF 2 , H, H, H, O ], [AC712; H, Et, H, Me, O, CF 3, H, H, H, O], [AC713; H, Et, H, Me, O, OCH 2 F, H, H, H, O], [AC714; H, Et, H, Me, O, OCHF 2, H, H, H, O], [AC715; H, Et, H, Me, O, OCF ₃ , H, H, H, O], [AC 716; H, Et, H, Me, O, SCH ₂ F, H, H, H, O], [AC 717; H, Et, H, Me, O, _{SCHF 2, H, H, H} , O], [AC718; H, Et, H, Me, O, SCF 3, H, H, H, O], [AC719; H, Et, H, Me, O, CN, H, H, H, O], [AC 720; H, Et, H, Me, O, NO ₂ , H, H, H, O], [AC 721; H, Et, H, Et, O, H , H, H, H, O], [AC722; H, Et, H, Et, O, F, H, H, H, O], [AC 723; H, Et, H, Et, O, Cl, H H, H, O], [AC 724; H, Et, H, Et, O, Br, H, H, H, O], [AC 725; H, Et, H, Et, O, I, H, H H, O], [AC 726; H, Et, H, Et, O, Me, H, H, H, O], [AC 727; H, Et, H, Et, O, Et, , H, H, H, O], [AC 728; H, Et, H, Et, O, Pr, H, H, H, O], [AC 729; H, Et, H, Et, O, i-Pr , H, H, H, O ], [AC730; H, Et, H, Et, O, CH = CH 2, H, H, H, O], [AC731; H, Et, H, Et, O, _{C (CH 3) = CH 2} , H, H, H, O], [AC732; H, Et, H, Et, O, C≡CH, H, H, H, O], [AC733; H, Et , H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 734; H, Et, H, Et, O, c-Pr, H, H, H, O], [AC 735; H, Et, H, Et, O, OMe, H, H, H, O], [AC 736; H, Et, H, Et, O, OEt, H, H, H, O], [AC 737; H, Et, H, Et, O, Oi-Pr, H, H, H, O], [AC 738; H, Et, H, Et, O, SMe, H, H, H, O], [AC 739; H, Et, H, Et, O, SEt, H, H, H, O], [AC740; H, Et, H, Et, O, CH 2 F, H, H, H, O], [AC741; H, Et, H, Et, O, CHF 2, H, H, H, O], [AC742; H, Et, H, Et, O, CF 3, H, H, H, O], [AC743; H, Et, H, Et, O, OCH 2 F, H, H, H, O], [AC744; H, Et, H, Et, O, OCHF 2, H, H, H, O], [AC745; H , Et, H, Et, O , OCF 3, H, H, H, O], [AC746; H, Et, H, Et, O, SCH 2 F, H, H, H, O], [AC747; H, Et, H, Et, O, SCHF 2, H, H, H, O], [AC748; H, Et, H, Et, O, SCF 3, H, H, H, O], [AC749; H, Et, H, Et, O, CN, H, H, H, O], [AC 750; H, Et, H, Et, O, NO ₂ , H, H, H, O], [AC 751; H , Et, H, Pr, O, H, H, H, H, O], [AC 752; H, Et, H, Pr, O, F, H, H, H, O], [AC 753; H, Et , H, Pr, O, Cl, H, H, H, O], [AC 754; H, Et, H, Pr, O, Br, H, H, H, O], [AC 755; H, Et, H , Pr, O, I, H, H, H, O], [AC 756; H, Et, H, Pr, O, Me, H, H, H, O], [AC 757; H, Et , H, Pr, O, Et, H, H, H, O], [AC 758; H, Et, H, Pr, O, Pr, H, H, H, O], [AC 759; H, Et, H , Pr, O, i-Pr , H, H, H, O], [AC760; H, Et, H, Pr, O, CH = CH 2, H, H, H, O], [AC761; H, Et, H, Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC762; H, Et, H, Pr, O, C≡CH, H, H, H, O ], [AC 763; H, Et, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 764; H, Et, H, Pr, O, c-Pr, H, H, H, O], [AC 765; H, Et, H, Pr, O, OMe, H, H, H, O], [AC 766; H, Et, H, Pr, O, OEt, H, H, H, O, [AC 767; H, Et, H, Pr, O, Oi-Pr, H, H, H, O], [AC 768; H, Et, H, Pr, O, SMe, H, H, H, H, H, Et, H, Pr, O, SEt, H, H, H, O], [AC 770; H, Et, H, Pr, O, CH ₂ F, H, H, H, O], [AC 769; O], [AC 771; H, Et, H, Pr, O, CHF ₂ , H, H, H, O], [AC 772; H, Et, H, Pr, O, CF ₃ , H, H, H, H, O], [AC 773; H, Et, H, Pr, O, OCH ₂ F, H, H, H, O], [AC 774; H, Et, H, Pr, O, OCHF ₂ , H, H, H , O], [AC775; H , Et, H, Pr, O, OCF 3, H, H, H, O], [AC776; H, Et, H, Pr, O, SCH 2 F, H, H, H, O], [AC 777; H, Et, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 778; H, Et, H, Pr, O, SCF ₃ , H, H, H, H, O], [AC779; H, Et, H, Pr, O, CN, H, H, H, O], [AC780; H, Et, H, Pr, O, NO 2, H, H, H , O], [AC 781; H, Et, H, i-Pr, O, H, H, H, H, O], [AC 782; H, Et, H, i-Pr, O, F, H, H , H, O], [AC 783; H, Et, H, i-Pr, O, Cl, H, H, H, O], [AC 784; H, Et, H, i-Pr, O, Br, H , H, H, O], [AC 785; H, Et, H, i-Pr, O, I, H, H, H, O], [AC 786; H, Et, H, i-Pr, O, M e, H, H, H, O], [AC 787; H, Et, H, i-Pr, O, Et, H, H, H, O], [AC 788; H, Et, H, i-Pr, O, Pr, H, H, H, O], [AC 789; H, Et, H, i-Pr, O, i-Pr, H, H, H, O], [AC 790; H, Et, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC791; H, Et, H, i-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC 792; H, Et, H, i-Pr, O, C≡CH, H, H, H, O], [AC 793; H, Et, H, i-Pr, O, C≡ CCH ₃ , H, H, H, O], [AC 794; H, Et, H, i-Pr, O, c-Pr, H, H, H, O], [AC795; H, Et, H, i-Pr , O, OMe, H, H, H, O], [AC796; H, Et, H, i-Pr, O, OEt, H, H, H, O], [AC 797; H, Et, H, i -Pr, O, Oi-Pr, H, H, H, O],

[AC 798; H, Et, H, i-Pr, O, SMe, H, H, H, O], [AC 799; H, Et, H, i-Pr, O, SEt, H, H, H, O ], [AC800; H, Et , H, i-Pr, O, CH 2 F, H, H, H, O], [AC801; H, Et, H, i-Pr, O, CHF 2, H, H, H, O], [ AC802; H, Et, H, i-Pr, O, CF 3, H, H, H, O], [AC803; H, Et, H, i-Pr, O, OCH ₂ F, H, H, H, O], [AC 804; H, Et, H, i-Pr, O, OCHF ₂ , H, H, H, O], [AC 805; H, Et, H, i- _{Pr, O, OCF 3, H} , H, H, O], [AC806; H, Et, H, i-Pr, O, SCH 2 F, H, H, H, O], [AC807; H, Et , H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 808; H, Et, H, i-Pr, O, SCF ₃ , H, H, H, O], [AC 809 H, Et, H, i-Pr, O, CN, H, H, H, O], [AC 810; H, Et, H, i-Pr, O, NO ₂ , H, H, H, O] , [AC 811; H, Et, H, c-Pr, O, H, H, H, H, O], [AC 812; H, Et, H, c-Pr, O, F, H, H, H, H, O], [AC 813; H, Et, H, c-Pr, O, Cl, H, H, H, O], [AC 814; H, Et, H, c-Pr, O, Br, H, H, H, H, O], [AC 815; H, Et, H, c-Pr, O, I, H, H, H, O], [AC 816; H, Et, H, c-Pr, O, Me, H, H, H, O], [AC 817; H, Et, H, c-Pr, O, Et, H, H, H, O], [AC 818; H, Et, H, c-Pr, O, Pr, H, H, H, O], [AC 819; H, Et, H, c-Pr, O, i-Pr, H, H, H, O], [AC 820; H, Et, H, c-Pr, _{O, CH = CH 2, H} , H, H, O], [AC821; H, Et, H, c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [ AC 822; H, Et, H, c-Pr, O, C≡CH, H, H, H, O], [AC 823; H, Et, H, c-Pr, O, C≡ CCH ₃ , H, H , H, O], [AC 824; H, Et, H, c-Pr, O, c-Pr, H, H, H, O], [AC 825; H, Et, H, c-Pr, O, OMe , H, H, H, O], [AC 826; H, Et, H, c-Pr, O, OEt, H, H, H, O], [AC 827; H, Et, H, c-Pr, O, Oi-Pr, H, H, H H, Et, H, c-Pr, O, SMe, H, H, H, O], [AC 829; H, Et, H, c-Pr, O, SEt, H, H , H, O], [AC830 ; H, Et, H, c-Pr, O, CH 2 F, H, H, H, O], [AC831; H, Et, H, c-Pr, O, CHF _{2, H, H, H,} O], [AC832; H, Et, H, c-Pr, O, CF 3, H, H, H, O], [AC833; H, Et, H, c-Pr _{, O, OCH 2 F, H} , H, H, O], [AC834; H, Et, H, c-Pr, O, OCHF 2, H, H, H, O], [AC835; H, Et, H, c-Pr, O, OCF 3, H, H, H, O], [AC836; H, Et, H, c-Pr, O, SCH 2 F, H, H, H, O], [AC837 H, Et, H, c-Pr, O, SCHF ₂ , H, H, H, O], [AC 838; H, Et, H, c-Pr, O, SCF ₃ , H, H, H, O ], [AC 839; H, Et, H, c-Pr, O, CN, H, H, H, O], [AC 840; H, Et, H, c-Pr, O, NO ₂ , H, H, H, O], [AC 841; H, Et, H, SMe, O, H, H, H, H, O], [AC 842; H, Et, H, SMe, O, F, H, H, H, H, O], [AC 843; H, Et, H, SMe, O, Cl, H, H, H, O], [AC 844; H, Et, H, SMe, O, Br, H, H, H, O] , [AC845; H, Et, H, SMe, O, I, H, H, H, O], [AC 846; H, Et, H, SMe, O, Me, H, H, H, O], [AC 845; AC 847; H, Et, H, SMe, O, Et, H, H, H, O], [AC 848; H, Et, H, SMe, O, Pr, H, H, H, O], [AC 849; H, Et, H, SMe, O, i-Pr, H, H, H, O], [AC850; H, Et, H, SMe, O, CH = CH 2, H, H, H, O], [AC851; H, Et, H , SMe, O, C (CH 3) = CH 2, H, H, H, O], [AC852; H, Et, H, SMe, O, C≡CH, H, H, H, O], [AC 853; H, Et, H, SMe, O, C≡CCH ₃ , H, H, H, O], [AC 854; H, Et, H, SMe, O, c-Pr, H, H, H, O], [AC 855; H, Et, H, SMe, O, OMe, H, H, H, O], [AC 856; H, Et, H, SMe, O, OEt, H, H, H, O], [AC 857; H, Et, H, SMe, O, Oi-Pr, H, H, H, O], [AC 858; H, Et, H, SMe, O, SMe, H, H, H, O, [AC 859; H, Et, H, SMe, O, SE t, H, H, H, O], [AC 860; H, Et, H, _{SMe, O, CH 2 F,} H, H, H, O], [AC861; H, Et, H, SMe, O, CHF 2, H, H, H, O], [AC862; H, Et, H _{, SMe, O, CF 3,} H, H, H, O], [AC863; H, Et, H, SMe, O, OCH 2 F, H, H, H, O], [AC864; H, Et, _{H, SMe, O, OCHF 2} , H, H, H, O], [AC865; H, Et, H, SMe, O, OCF 3, H, H, H, O], [AC866; H, Et, H, SMe, O, SCH ₂ F, H, H, H, O], [AC 867; H, Et, H, SMe, O, SCHF ₂ , H, H, H, O], [AC 868; H, Et , H, SMe, O, SCF ₃ , H, H, H, O], [AC 869; H, Et, H, SMe, O, CN, H, H, H, O], [AC 870; H, Et, _{H, SMe, O, NO 2} , H, H, H, O], [AC871; H, Et, H, OMe, O, H, H, H, H, O], [AC872; H, Et, H , OMe, O, F, H, H, H, O], [AC 873; H, Et, H, OMe, O, Cl, H, H, H, O], [AC 874; H, Et, H, OMe , O, Br, H, H, H, O], [AC 875; H, Et, H, OMe, O, I, H, H, H, O], [AC 876; H, Et, H, OMe, O , Me, H, H, H, O], [AC 877; H, Et, H, OMe, O, Et, H, H, H, O], [AC 878; H, Et, H, OMe, O, Pr , H, H, H, O], [AC 879; H, Et, H, OMe, O, i-Pr, H, H, H, O], [AC 880; H, Et, H, OMe, O, CH _{= CH 2, H, H,} H, O], [AC881; H, Et, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC882; H, Et , H, OMe, O, C≡CH, H, H, H, O], [AC 883; H, Et, _{H, OMe, O, C≡CCH 3} , H, H, H, O], [AC884; H, Et, H, OMe, O, c-Pr, H, H, H, O], [AC885; H Et, H, OMe, O, OMe, H, H, H, O], [AC 886; H, Et, H, OMe, O, OEt, H, H, H, O], [AC 887; H, Et , H, OMe, O, Oi-Pr, H, H, H, O], [AC 888; H, Et, H, OMe, O, SMe, H, H, H, O], [AC 889; H, Et , H, OMe, O, SEt , H, H, H, O], [AC890; H, Et, H, OMe, O, CH 2 F, H, H, H, O], [AC891; H, Et , H, OMe, O, CHF 2, H, H, H, O], [AC892; H, Et, H, OMe, O, CF 3, H, H, H, O], [AC893; H, Et , H, OMe, O, OCH 2 F, H, H, H, O], [AC894; H, Et, H, OMe, O, OCHF 2, H, H, H, O], [AC895; H, Et, H, OMe, O, OCF 3, H, H, H, O], [AC896; H, Et, H, OMe, O, SCH 2 F, H, H, H, O], [AC897; H , Et, H, OMe, O, SCHF ₂ , H, H, H, O],

[AC 898; H, Et, H, OMe, O, SCF ₃ , H, H, H, O], [AC 899; H, Et, H, OMe, O, CN, H, H, H, O], [AC AC 900; H, Et, H, OMe, O, NO ₂ , H, H, H, O], [AC 901; H, Et, H, F, O, H, H, H, H, O], [AC 902 H, Et, H, F, O, F, H, H, H, O], [AC 903; H, Et, H, F, O, Cl, H, H, H, O], [AC 904; H , Et, H, F, O, Br, H, H, H, O], [AC 905; H, Et, H, F, O, I, H, H, H, O], [AC 906; H, Et , H, F, O, Me, H, H, H, O], [AC 907; H, Et, H, F, O, Et, H, H, H, O], [AC 908; H, Et, H , F, O, Pr, H, H, H, O, [AC 909; H, Et, H, F, O, i-Pr, H, H, H, O], [AC 910; H, Et, H , F, O, CH = CH 2, H, H, H, O], [AC911; H, Et, H, F, O, C (CH 3) = CH 2, H, H, H, O], [AC 912; H, Et, H, F, O, C≡CH, H, H, H, O], [AC 913; H, Et, H, F, O, C≡ CCH ₃ , H, H, H, H O], [AC 914; H, Et, H, F, O, c-Pr, H, H, H, O], [AC 915; H, Et, H, F, O, OMe, H, H, H, H, O], [AC 916; H, Et, H, F, O, OEt, H, H, H, O], [AC 917; H, Et, H, F, O, Oi-Pr, H, H, H, O], [AC 918; H, Et, H, F, O, SMe, H, H, H, O], [AC 919; H, Et, H, F, O, SE t, H, H, H, O] , [AC920; H, Et, H, F, O, CH 2 F, H, H, H, O], [AC921; H, Et, H, F, O, CHF 2, H, H, H, O ], [AC922; H, Et , H, F, O, CF 3, H, H, H, O], [AC923; H, Et, H, F, O, OCH 2 F, H, H, H, O], [AC924; H, Et, H, F, O, OCHF 2, H, H, H, O], [AC925; H, Et, H, F, O, OCF 3, H, H, H, O], [AC 926; H, Et, H, F, O, SCH ₂ F, H, H, H, O], [AC 927; H, Et, H, F, O, SCHF ₂ , H, H, H , O], [AC 928; H, Et, H, F, O, SCF ₃ , H, H, H, O], [AC 929; H, Et, H, F, O, CN, H, H, H, O], [AC 930; H, Et, H, F _{, O, NO 2, H,} H, H, O], [AC931; H, Et, H, Cl, O, H, H, H, H, O], [AC932; H, Et, H, Cl, O, F, H, H, H, O, [AC 933; H, Et, H, Cl, O, Cl, H, H, H, O], [AC 934; H, Et, H, Cl, O, Br, H, H, H, O], [AC 935; H, Et, H, Cl, O, I, H, H, H, O], [AC 936; H, Et, H, Cl, O, Me, H, H, H, O], [AC 937; H, Et, H, Cl, O, Et, H, H, H, O], [AC 938; H, Et, H, Cl, O, Pr, H, H, H, O], [ AC939; H, Et, H, Cl, O, i-Pr, H, H, H, O], [AC940; H, Et, H, Cl, O, CH = CH 2 , H, H, H, O ], [AC941; H, Et, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC942; H, Et, H, Cl, O, C≡CH, H, H, H, H, O], [AC 943; H, Et, H, Cl, O, C≡ CCH ₃ , H, H, H, O], [AC 944; H, Et , H, Cl, O, c-Pr, H, H, H, O], [AC 945; H, Et, H, Cl, O, OMe, H, H, H, O], [AC 946; H, Et , H, Cl, O, OEt, H, H, H, O], [AC 947; H, Et, H, Cl, O, Oi-Pr, H, H, H, O], [AC 948; H, Et , H, Cl, O, SMe, H, H, H, O], [AC 949; H, Et, H, Cl, O, SE t, H, H, H, O], [AC 950; H, Et, H _{, Cl, O, CH 2 F} , H, H, H, O], [AC951; H, Et, H, Cl, O, CHF 2, H, H, H, O], [AC952; H, Et, _{H, Cl, O, CF 3} , H, H, H, O], [AC953; H, Et, H, Cl, O, OCH 2 F, H, H, H, O], [AC954; H, Et , H, Cl, O, OCHF 2, H, H, H, O], [AC955; H, Et, H, Cl, O, OCF 3, H, H, H, O], [AC956; H, Et , H, Cl, O, SCH ₂ F, H, H, H, O], [AC 957; H, Et, H, Cl, O, SCHF ₂ , H, H, H, O], [AC 958; H, Et, H, Cl, O, SCF 3, H, H, H, O], [AC959; H, Et, H, Cl, O, CN, H, H, H, O], [AC960; H , Et, H, Cl, O , NO 2, H, H, H, O], [AC961; H, Et, H, Br, O, H, H, H, H, O], [AC962; H, Et, H, Br, O, F, H, H, H, O], [AC 963; H, Et, H, Br, O, Cl, H, H, H, O], [AC 964; H, Et, H, Br, O, Br, H, H, H, O], [AC 965; H, Et, H, Br, O, I, H, H, H, O], [AC 966; H, Et, H, Br, O, Me, H, H, H, O, [AC 967; H, Et, H, Br, O, Et, H, H, H, O], [AC 968; H, Et, H, Br, O, Pr, H, H, H, O], [AC 969; H, Et, H, Br, O, i-Pr, H, H, H, O], [AC 970; H, Et, H, Br, _{O, CH = CH 2, H} , H, H, O], [AC971; H, Et, H, Br, O, C (CH 3) = CH 2, H, H, H, O], [AC972; H, Et, H, Br, O, C≡CH, H, H, H, O], [AC 973; H, Et, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 974; H, Et, H, Br, O, c-Pr, H, H, H, O], [AC 975; H, Et, H, Br, O, OMe, H, H, H, O], [AC 976; H, Et, H, Br, O, OEt, H, H, H, O], [AC 977; H, Et, H, Br, O, Oi-Pr, H, H, H, O], [AC978; H, Et, H, Br, O, SMe, H, H, H, O], [AC 979; H, Et, H, Br, O, SEt, H, H, H, O], [AC 980 ; H, Et, H, Br , O, CH 2 F, H, H, H, O], [AC981; H, Et, H, Br, O, CHF 2, H, H, H, O], [ AC982; H, Et, H, Br, O, CF 3, H, H, H, O], [AC983; H, Et, H, Br, O, OCH 2 F, H, H, H, O], [AC984; H, Et, H , Br, O, OCHF 2, H, H, H, O], [AC985; H, Et, H, Br, O, OCF 3, H, H, H, O], [AC986; H, Et, H, Br, O, SCH ₂ F, H, H, H, O], [AC 987; H, Et, H, Br, O, SCHF ₂ , H, H, H, H O], [AC 988; H, Et, H, Br, O, SCF ₃ , H, H, H, O], [AC 989; H, Et, H, Br, O, CN, H, H, H, O H, Et, H, Br, O, NO ₂ , H ₂ , H, O], [AC 991; H, Pr, H, H, O, H, H, H, H, O] , [AC 992; H, Pr, H, H, O, F, H, H, O], [AC 993; H, Pr, H, H, O, Cl, H, H, H, O], [AC 993; AC 994; H, Pr, H, H, O, Br, H, H, O], [AC 995; H, Pr, H, H, O, I, H, H, H, O], [AC 996; H, Pr, H, H, O, Me, H, H, H, O],

[AC 997; H, Pr, H, H, O, Et, H, H, H, O], [AC 998; H, Pr, H, H, O, Pr, H, H, H, O], [AC 999 H, Pr, H, H, O, i-Pr, H, H, H, O], [AC 1000; H, Pr, H, H, O, CH, CH ₂ , H, H, H, O] , [AC1001; H, Pr, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC1002; H, Pr, H, H, O, C≡CH, H , H, H, O], [AC 1003; H, Pr, H, H, O, C≡CCH ₃ , H, H, H, O], [AC 1004; H, Pr, H, H, O, c- Pr, H, H, H, O], [AC 1005; H, Pr, H, H, O, OMe, H, H, H, O], [AC 1006; H, Pr, H, H, O, OE t, H, H, H, O], [AC 1007; H, Pr, H, H, O, Oi-Pr, H, H, H, O], [AC 1008; H, Pr, H, H, O, SMe, H, H, H, O], [AC 1009; H, Pr, H, H, O, SE t, H, H, H, O], [AC 1010; H, Pr, H, H, O, CH ₂ F, H, H, H, O], [AC 1011; H, Pr, H, H, O, CHF ₂ , H, H, H, O], [AC 1012; H, Pr, H, H, O, CF ₃ , H, H, H, O] , [AC1013; H, Pr, H, H, O, OCH 2 F, H, H, H, O], [AC1014; H, Pr, H, H, O, OCHF 2 , H, H, H, O ], [AC1015; H, Pr, H, H, O, OCF 3, H, H, H, O], [AC1016; H, Pr, H, H, O, SCH 2 F, H, H, H, O], [AC 1017; H, Pr, H, H, O, SCHF ₂ , H, H, H, O], [AC 1018; H, Pr, H, H, O, SCF ₃ , H, H, H, O], [AC 1019; H, Pr, H, H, O, CN, H, H, H, O], [AC 1020; H, Pr, H, H, O, NO ₂ H, H, H, O], [AC 1021; H, Pr, H, Me, O, H, H, H, H, O], [AC 1022; H, Pr, H, Me, O, F, H H, H, O], [AC1023; H, Pr, H, Me, O, Cl, H, H, H, O], [AC 1024; H, Pr, H, Me, O, Br, H, H , H, O], [AC 1025; H, Pr, H, Me, O, I, H, H, H, O], [AC 1026; H, Pr, H, Me, O , Me, H, H, H, O], [AC 1027; H, Pr, H, Me, O, Et, H, H, H, O], [AC 1028; H, Pr, H, Me, O, Pr , H, H, H, O], [AC 1029; H, Pr, H, Me, O, i-Pr, H, H, H, O], [AC 1030; H, Pr, H, Me, O, CH _{= CH 2, H, H,} H, O], [AC1031; H, Pr, H, Me, O, C (CH 3) = CH 2, H, H, H, O], [AC1032; H, Pr , H, Me, O, C≡CH, H, H, H, O], [AC 1033; H, Pr, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 1034; H, Pr, H, Me, O, c-Pr, H, H, H, O], [AC 1035; H, Pr, H, Me, O, OMe, H, H, H, O], [AC 1036; H, Pr, H, Me, O, OEt, H, H, H, O], [AC 1037; H, Pr, H, Me, O, Oi-Pr, H, H, H, O], [AC 1038; H, Pr, H, Me, O, SMe, H, H, H, O], [AC 1039; H, Pr, H, Me, O, SE, H, H, H, O], [AC 1040; H, Pr, H, Me, O, CH 2 F, H, H, H, O], [AC1041; H, Pr, H, Me, O, CHF 2, H, H, H, O], [AC1042; H , Pr, H, Me, O , CF 3, H, H, H, O], [AC1043; H, Pr, H, Me, O, OCH 2 F, H, H, H, O], [AC1044; H, Pr, H, Me, O, OCHF 2, H, H, H, O], [AC1045; H, Pr, H, Me, O, OCF 3, H, H, H, O], [AC1046; H, Pr, H, Me, O, SCH ₂ F, H, H, H, O], [AC 1047; H, Pr, H, Me, O, SCHF ₂ , H, H, H, O], [AC 1048 ; H, Pr, H, Me , O, SCF 3, H, H, H, O], [AC1049; H, Pr, H, Me, O, CN, H, H, H, O], [AC1050; H, Pr, H, Me, O, NO 2, H, H, H, O], [AC1051; H, Pr, H, Et, O, H, H, H, H, O], [AC1052; H , Pr, H, Et, O, F, H, H, H, O], [AC1053; H, Pr, H, Et, O, Cl, H, H, H, O], [AC 1054; H, Pr , H, Et, O, Br, H, H, H, O], [AC1055; H, Pr, H, Et, O, I, H, H, H, O], [AC 1056; H, Pr, H, Et, O, Me, H, H, O, [AC 1057; H, Pr, H, Et, O, Et, H, H, H, O], [AC 1058; H, Pr, H, Et, O, Pr, H, H, H, O], [AC 1059; H, Pr, H, Et, O, i-Pr, H, H, H, H, O], [AC 1060; H, Pr, H, Et, O, CH = CH ₂ , H, H, H, O], [AC 1061; H, Pr , H, Et, O, C (CH 3) = CH 2, H, H, H, O], [AC1062; H, Pr, H, Et, O, C≡CH, H, H, H, O] , [AC 1063; H, Pr, H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 1064; H, Pr, H, Et, O, c-Pr, H, H, H H, Pr, H, Et, O, OMe, H, H, H, O], [AC 1066; H, Pr, H, Et, O, OEt, H, H, H, O H, Pr, H, Et, O, Oi-Pr, H, H, H, O], [AC 1068; H, Pr, H, Et, O, SMe, H, H, H, O] H, Pr, H, Et, O, SEt, H, H, H, O], [AC 1070; H, Pr, H, Et, O, CH ₂ F, H, H, H, O] ], [AC1071; H, Pr , H, Et, O, CHF 2, H, H, H, O], [AC1072; H, Pr, H, Et, O, CF 3, H, H, H, O ], [AC1073; H, Pr , H, Et, O, OCH 2 F, H, H, H, O], [AC1074; H, Pr, H, Et, O, OCHF 2, H, H, H, O], [AC1075; H, Pr, H, Et, O, OCF 3, H, H, H, O], [AC1076; H, Pr, H, Et, O, SCH 2 F, H, H, H H, Pr, H, Et, O, SCHF ₂ , H, H, H, O], [AC 1078; H, Pr, H, Et, O, SCF ₃ , H, H, H H, Pr, H, Et, O, CN, H, H, H, O], [AC 1080; H, Pr, H, Et, O, NO ₂ , H, H, H, H, H] O], [AC1081; H, Pr, H, Pr, O, H, H, H, O], [AC1082; H, Pr, H, Pr, O, F, H, H, H, O] , [AC1083; H, Pr, H, Pr, O, Cl, H, H, H, O], [A H, Pr, H, Pr, O, Br, H, H, O], [AC 1085; H, Pr, H, Pr, O, I, H, H, H, O], [AC 1086; H, Pr, H, Pr, O, Me, H, H, H, O], [AC 1087; H, Pr, H, Pr, O, Et, H, H, H, O], [AC 1088; H, Pr, H, Pr, O, Pr, H, H, H, O], [AC 1089; H, Pr, H, Pr, O, i-Pr, H, H, H, O], [AC 1090; H, Pr, H, Pr, O, CH = CH 2, H, H, H, O], [AC1091; H, Pr, H, Pr, O, C (CH 3) = CH 2, H, H, H, O, [AC1092; H, Pr, H, Pr, O, C≡CH, H, H, H, O], [AC1093; H, Pr, H, Pr, O, C≡ CCH ₃ , H, H , H, O], [AC1094; H, Pr, H, Pr, O, c-Pr, H, H, H, O], [AC 1095; H, Pr, H, Pr, O, OMe, H, H , H, O], [AC 1096; H, Pr, H, Pr, O, OEt, H, H, H, O],

[AC 1097; H, Pr, H, Pr, O, Oi-Pr, H, H, H, O], [AC 1098; H, Pr, H, Pr, O, SMe, H, H, H, O], [AC 1099; H, Pr, H, Pr, O, SEt, H, H, H, O], [AC 1100; H, Pr, H, Pr, O, CH ₂ F, H, H, H, O], [AC1101; H, Pr, H , Pr, O, CHF 2, H, H, H, O], [AC1102; H, Pr, H, Pr, O, CF 3, H, H, H, O], [AC1103; H, Pr, H , Pr, O, OCH 2 F, H, H, H, O], [AC1104; H, Pr, H, Pr, O, OCHF 2, H, H, H, O] , [AC1105; H, Pr, H, Pr, O, OCF 3, H, H, H, O], [AC1106; H, Pr, H, Pr, O, SCH 2 F, H, H, H, O H, Pr, H, Pr, O, SCHF ₂ , H, H, O], [AC 1108; H, Pr, H, Pr, O, SCF ₃ , H, H, H, O] ], [AC 1109; H, Pr, H, Pr, O, CN, H, H, H, O], [AC 1110; H, Pr, H, Pr, O, NO ₂ , H, H, H, O] , [AC1 111; H, Pr, H, i-Pr, O, H, H, H, H, O], [AC 1112; H, Pr, H, i-Pr, O, F, H, H, H, O], [AC1113; H, Pr, H, i-Pr, O, Cl, H, H, O], [AC 1114; H, Pr, H, i-Pr, O, Br, H, H, H, O], [AC 1115; H, Pr, H, i-Pr, O, I, H, H, H, O], [AC 1116; H, Pr, H, i-Pr, O, Me, H, H, H, O], [AC 1 117; H, Pr, H, i-Pr, O, Et, H, H, H, O], [AC 1118; H, Pr, H, i-Pr, O, Pr, H, H, H, O], [AC 1119; H, Pr, H, i-Pr, O, i-Pr, H, H, H, O], [AC 1 120; H, Pr, H, i-Pr, O, CH = CH ₂ , H, H, H, O, [AC 1121; H, Pr, H, i-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [[ AC1122; H, Pr, H, i-Pr, O, C≡CH, H, H, H, O], [AC 1123; H, Pr, H, i-Pr, O, C≡ CCH ₃ , H, H , H, O], [AC 1 124; H, Pr, H, i-Pr, O, c-Pr, H, H, H, O H, Pr, H, i-Pr, O, OMe, H, H, H, O], [AC 1126; H, Pr, H, i-Pr, O, OEt, H, H, H] , O], [AC 1127; H, Pr, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 1 128; H, Pr, H, i-Pr, O, SMe, H , H, H, O], [AC 1129; H, Pr, H, i-Pr, O, SE t, H, H, H, O], [AC 1130; H, Pr, H, i-Pr, O, CH ₂ F, H, H, H, O], [AC 1131; H, Pr, H, i-Pr, O, CHF ₂ , H, H, H, O], [AC 1132; H, Pr, H, i- _{Pr, O, CF 3, H} , H, H, O], [AC1133; H, Pr, H, i-Pr, O, OCH 2 F, H, H, H, O], [AC1134; H, Pr , H, i-Pr, O , OCHF 2, H, H, H, O], [AC1135; H, Pr, H, i-Pr, O, OCF 3, H, H, H, O], [AC1136 H, Pr, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 1137; H, Pr, H, i-Pr, O, SCHF ₂ , H, H, H, H O], [AC 1138; H, Pr, H, i-Pr, O, SCF ₃ , H, H, H, O], [AC 1139; H, Pr, H, i-Pr, O, CN, H, H , H, O], [AC 1 140; H, Pr, H, i-Pr, O, NO ₂ , H, H, H, O], [AC 1141; H, Pr, H, c-Pr, O, H, H, H, H, O], [AC1142; H, Pr, H, c-Pr, O, F, H, H, H, O], [AC 1143; H, Pr, H, c-Pr, O, Cl, H, H, H, O], [AC 1144; H, Pr, H, c-Pr, O, Br, H, H, H, O], [AC 1145; H, Pr, H, c-Pr, O, I, H, H, H, O], [AC 1146; H, Pr, H, c-Pr, O, Me, H, H, H, O], [AC 1147; H, Pr, H, c- Pr, O, Et, H, H, H, O, [AC1148; H, Pr, H, c-Pr, O, Pr, H, H, H, O], [AC 1149; H, Pr, H, c-Pr, O, i-Pr, H, H, H, O], [AC 1150; H, Pr, H, c-Pr, O, CH = CH ₂ , H, H, H, O], [AC 1151 ; H, Pr, H, c -Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC1152; H, Pr, H , c-Pr, O, C≡CH, H, H, H, O], [AC 1153; H, Pr, H, c-Pr, O, C≡ CCH ₃ , H, H, H, O], [[ AC1154; H, Pr, H, c-Pr, O, c-Pr, H, H, H, O], [AC 1155; H, Pr, H, c-Pr, O, OMe, H, H, H, O, [AC 1156; H, Pr, H, c-Pr, O, OEt, H, H, H, O], [AC 1 157; H, Pr, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 1158; H, Pr, H, c-Pr, O, SMe, H, H, H, O], [AC 1159; H, Pr, H, c-Pr, O, SEt, H, H, H, O] , [AC1160; H, Pr, H, c-Pr, O, CH 2 F, H, H, H, O], [AC1161; H, Pr, H, c-Pr, _{O, CHF 2, H, H} , H, O], [AC1162; H, Pr, H, c-Pr, O, CF 3, H, H, H, O], [AC1163; H, Pr, H, _{c-Pr, O, OCH 2} F, H, H, H, O], [AC1164; H, Pr, H, c-Pr, O, OCHF 2, H, H, H, O], [AC1165; H , Pr, H, c-Pr , O, OCF 3, H, H, H, O], [AC1166; H, Pr, H, c-Pr, O, SCH 2 F, H, H, H, O] H, Pr, H, c-Pr, O, SCHF ₂ , H, H, H, O], [AC 1168; H, Pr, H, c-Pr, O, SCF ₃ , H, H, H, O], [AC 1169; H, Pr, H, c-Pr, O, CN, H, H, H, O], [AC 1170; H, Pr, H, c-Pr, O, NO ₂ , H H, H, O], [AC1171; H, Pr, H, SMe, O, H, H, H, H, O], [AC1172; H, Pr, H, SMe, O, F, H, H , H, O], [AC1173; H, Pr, H, SMe, O, Cl, H, H, H, O], [AC 1174; H, Pr, H, SMe, O, Br, H, H, H H, Pr, H, SMe, O, I, H, H, H, O], [AC 1176; H, Pr, H, SMe, O, Me, H, H, H, O] H, Pr, H, SMe, O, Et, H, H, H, O], [AC 1178; H, Pr, H, SMe, O, Pr, H, H, H, O], [AC1179; H, Pr, H, SMe, O, i-Pr, H, H, H, O], [AC 1180; H , Pr, H, SMe, O , CH = CH 2, H, H, H, O], [AC1181; H, Pr, H, SMe, O, C (CH 3) = CH 2, H, H, H H, Pr, H, SMe, O, C≡CH, H, H, H, O], [AC1183; H, Pr, H, SMe, O, C≡CCH ₃ , H, H, H, O], [AC 1184; H, Pr, H, SMe, O, c-Pr, H, H, H, O], [AC 1185; H, Pr, H, SMe, O, OMe, H, H, H, O], [AC1186; H, Pr, H, SMe, O, OEt, H, H, H, O], [AC 1187; H, Pr, H, SMe, O, Oi-Pr, H, H, H, O], [AC1188; H, Pr, H, SMe, O, SMe, H, H, H, O], [AC 1189; H, Pr, H, SMe, O, SEt, H, H, H, H, O], [AC1190; H, Pr, H, SMe, O, CH 2 F, H, H, H, O], [AC1191; H, Pr, H, SMe, O, CHF 2, H, H , H, O], [AC1192 ; H, Pr, H, SMe, O, CF 3, H, H, H, O], [AC1193; H, Pr, H, SMe, O, OCH 2 F, H, H, H, O], [ AC1194; H, Pr, H, SMe, O, OCHF 2, H, H, H, O], [AC1195; H, Pr, H, SMe, O, OCF 3, H, H, H, O], [AC 1196; H, Pr, H, SMe, O, SCH ₂ F, H, H, H, O],

[AC 1197; H, Pr, H, SMe, O, SCHF ₂ , H, H, H, O], [AC 1198; H, Pr, H, SMe, O, SCF ₃ , H, H, H, O], [AC1199; H, Pr, H , SMe, O, CN, H, H, H, O], [AC1200; H, Pr, H, SMe, O, NO 2, H, H, H, O], [ AC1201; H, Pr, H, OMe, O, H, H, H, H, O], [AC1202; H, Pr, H, OMe, O, F, H, H, H, O], [AC 1203; H, Pr, H, OMe, O, Cl, H, H, H, O], [AC 1204; H, Pr, H, OMe, O, Br, H, H, H, O], [AC 1205; H, Pr, H, OMe, O, I, H, H, H, O], [AC 1206; H, Pr, H, OMe, O, Me, H, H, H, O], [AC 1207; H, Pr, H, OMe, O, Et, H, H, H, O], [AC 1208; H, Pr, H, OMe, O, Pr, H, H, H, O], [AC 1209; H, Pr, H, OMe, O, i-Pr, H, H, H, O], [AC1210; H, Pr, H, OMe, O, CH = CH 2, H, H, H, O], [AC1211; H, Pr , H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC1212; H, Pr, H, OMe, O, C≡CH, H, H, H, O] , [AC 1213; H, Pr, H, OMe, O, C≡CCH ₃ , H, H, H, O], [AC 1214; H, Pr, H, OMe, O, c-Pr, H, H, H H, Pr, H, OMe, O, OMe, H, H, H, O], [AC 1216; H, Pr, H, OMe, O, OEt, H, H, H, O H, Pr, H, OMe, O, Oi-Pr, H, H, H, O], [AC 1218; H, Pr, H, OMe, O, SMe, H, H, H, O] H, Pr, H, OMe, O, SEt, H, H, H, O], [AC 1220; H, Pr, H, OMe, O, CH ₂ F, H, H, H, O] ], [AC1221; H, Pr , H, OMe, O, CHF 2, H, H, H, O], [AC1222; H, Pr, H, OMe, O, CF 3, H, H, H, O ], [AC1223; H, Pr , H, OMe, O, OCH 2 F, H, H, H, O], [AC1224; H, Pr, H, OMe, O, OCHF 2, H, H, H, O], [AC12 25; H, Pr, H, OMe, O, OCF 3, H, H, H, O], [AC1226; H, Pr, H, OMe, O, SCH 2 F, H, H, H, O], [AC1227; H, Pr, H , OMe, O, SCHF 2, H, H, H, O], [AC1228; H, Pr, H, OMe, O, SCF 3, H, H, H, O], [AC 1229; H, Pr, H, OMe, O, CN, H, H, H, O], [AC 1230; H, Pr, H, OMe, O, NO ₂ , H, H, H, O], [AC 12 30 AC 1231; H, Pr, H, F, O, H, H, H, O], [AC 1232; H, Pr, H, F, O, F, H, H, H, O], [AC 1233; H, Pr, H, F, O, Cl, H, H, H, O], [AC 1234; H, Pr, H, F, O, Br, H, H, O], [AC 1235; H, Pr, H, F, O, I, H, H, H, O], [AC 1236; H, Pr, H, F, O, Me, H, H, O], [AC 1237; H, Pr, H, F, O, Et, H, H, H, O], [AC1238; H, Pr, H, F, O, Pr, H, H, H, O], [AC 1239; H, Pr, H, F, O, i-Pr, H, H, H, H, O], [AC 1240; H, Pr, H, F, O, CH = CH ₂ , H, H, H, O], [AC 1241; H, Pr , H, F, O, C (CH 3) = CH 2, H, H, H, O], [AC1242; H, Pr, H, F, O, C≡CH, H, H, H, O] , [AC 1243; H, Pr, H, F, O, C≡CCH ₃ , H, H, H, O], [AC 1244; H, Pr, H, F, O, c-Pr, H, H, H H, Pr, H, F, O, OMe, H, H, H, O], [AC 1246; H, Pr, H, F, O, OEt, H, H, H, O H, Pr, H, F, O, Oi-Pr, H, H, H, O], [AC 1248; H, Pr, H, F, O, SMe, H, H, H, O] H, Pr, H, F, O, SE t, H, H, H, O], [AC 1250; H, Pr, H, F, O, CH ₂ F, H, H, H, O] ], [AC1251; H, Pr , H, F, O, CHF 2, H, H, H, O], [AC1252; H, Pr, H, F, O, CF 3, H, H, H, O ], [AC1253; H, Pr , H, F, O, OCH 2 F, H, H, H, O], [AC1254; H, Pr, H, F, O, _{OCHF 2, H, H, H} , O], [AC1255; H, Pr, H, F, O, OCF 3, H, H, H, O], [AC1256; H, Pr, H, F, O, SCH ₂ F, H, H, H, O], [AC 1257; H, Pr, H, F, O, SCHF ₂ , H, H, H, O], [AC 1258; H, Pr, H, F, O , SCF ₃ , H, H, H, O], [AC 1259; H, Pr, H, F, O, CN, H, H, H, O], [AC 1260; H, Pr, H, F, O, _{NO 2, H, H, H} , O], [AC1261; H, Pr, H, Cl, O, H, H, H, H, O], [AC1262; H, Pr, H, Cl, O, F H, H, H, O], [AC 1263; H, Pr, H, Cl, O, Cl, H, H, H, O], [AC 1264; H, Pr, H, Cl, O, Br, H , H, H, O], [AC 1265; H, Pr, H, Cl, O, I, H, H, H, O], [AC 1266; H, Pr, H, Cl, O, Me, H, H , H, O], [AC 1267; H, Pr, H, Cl, O, Et, H, H, H, O], [AC 1268; H, Pr, H, Cl, O, Pr, H, H, H H, Pr, H, Cl, O, i-Pr, H, H, H, O], [AC 1270; H, Pr, H, Cl, O, CH = CH ₂ , H, H, H, O], [ AC1271; H, Pr, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC1272; H, Pr, H, Cl, O , C≡CH, H, H, H, O], [AC 1273; H, Pr, H, Cl, O, C≡CCH ₃ , H, H, H, O], [AC 1274; H, Pr, H, Cl, O, c-Pr, H, H, H, H, O], [AC 1275; H, Pr, H, Cl, O, OMe, H, H, H, O], [AC 1276; H, Pr, H, Cl, O, OEt, H, H, H, O], [AC 1277; H, Pr, H, Cl, O, Oi-Pr, H, H, H, O], [AC 1278; H, Pr, H, Cl, O, SMe, H, H, H, O, [AC 1279; H, Pr, H, Cl, O, SE t, H, H, H, O], [AC 1280; H, Pr, H, Cl, _{O, CH 2 F, H,} H, H, O], [AC1281; H, Pr, H, Cl, O, CHF 2, H, H, H, O], [AC1282; H, Pr, H, Cl , O, CF ₃ , H, H, H, O], [AC1283; H, Pr, H, Cl, O, OCH _{2 F, H, H, H} , O], [AC1284; H, Pr, H, Cl, O, OCHF 2, H, H, H, O], [AC1285; H, Pr, H, Cl, O, _{OCF 3, H, H, H} , O], [AC1286; H, Pr, H, Cl, O, SCH 2 F, H, H, H, O], [AC1287; H, Pr, H, Cl, O , SCHF ₂ , H, H, H, O], [AC 1 288; H, Pr, H, Cl, O, SCF ₃ , H, H, H, O], [AC 1 289; H, Pr, H, Cl, O , CN, H, H, H, O], [AC 1290; H, Pr, H, Cl, O, NO ₂ , H, H, H, O], [AC 1291; H, Pr, H, Br, O, H, H, H, H, O], [AC1292; H, Pr, H, Br, O, F, H, H, H, O], [AC1293; H, Pr, H, Br, O, Cl, H, H, H, O], [AC 1294; H, Pr, H, Br, O, Br, H, H, H, O], [AC 1295; H, Pr, H, Br, O, I, H, H, H, O],

[AC1296; H, Pr, H, Br, O, Me, H, H, H, O], [AC 1297; H, Pr, H, Br, O, Et, H, H, H, O], [AC 1298 H, Pr, H, Br, O, Pr, H, H, H, O], [AC 1299; H, Pr, H, Br, O, i-Pr, H, H, H, O], [AC 1300] ; H, Pr, H, Br , O, CH = CH 2, H, H, H, O], [AC1301; H, Pr, H, Br, O, C (CH 3) = CH 2, H, H H, O], [AC1302; H, Pr, H, Br, O, C≡CH, H, H, H, O], [AC1303; H, Pr, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC1304; H, Pr, H, Br, O, c-Pr, H, H, H, O], [AC 1305; H, Pr, H, Br, O, OMe, H, H, H, O], [AC 1306; H, Pr, H, Br, O, OEt, H, H, H, O], [AC 1307; H, Pr, H, Br, O, Oi-Pr, H, H, H, O], [AC 1308; H, Pr, H, Br, O, SMe, H, H, H, O], [AC 1309; H, Pr, H, Br, O, SEt, H, H, H, O], [AC 1310; H, Pr, H, Br, O, CH ₂ F, H, H, H, O], [AC 1311; H, Pr, H, Br, O, CHF ₂ , H , H, H, O], [AC1312; H, Pr, H, Br, O, CF 3, H, H, H, O], [AC1313; H, Pr, H, Br, O, OCH 2 F, H, H, H, O], [AC 1314; H, Pr, H, Br, O, OCHF ₂ , H, H, H, O], [AC 1315; H, Pr, H, Br, O, OCF ₃ , H, H, H, O], [AC 1316; H, Pr, H, Br, O, SCH ₂ F, H, H, H, O], [AC 1317; H, Pr, H, Br, O, SCHF ₂ , H, H, H, O ], [AC1318; H, Pr, H, Br, O, SCF 3, H, H, H, O], [AC1319; H, Pr, H, Br, O, CN, H, H, H, O], [AC 1320; H, Pr, H, Br, O, NO ₂ , H, H, H, O], [AC 1321; H, i-Pr, H, H, O, H , H, H, H, O], [AC1322; H, i-Pr, H, H, O, F, H, H, O], [AC 1323; H, i-Pr, H, H, O , Cl, H, H, H, O], [AC 1324; H, i-Pr, H, H, O , Br, H, H, H, O], [AC 1325; H, i-Pr, H, H, O, I, H, H, H, O], [AC 1326; H, i-Pr, H, H , O, Me, H, H, H, O, [AC 1327; H, i-Pr, H, H, O, Et, H, H, H, O], [AC 1328; H, i-Pr, H , H, O, Pr, H, H, H, O], [AC 1329; H, i-Pr, H, H, O, i-Pr, H, H, H, O], [AC 1330; H, i -Pr, H, H, O, CH = CH 2, H, H, H, O], [AC1331; H, i-Pr, H, H, O, C (CH 3) = CH 2, H, H , H, O], [AC1332; H, i-Pr, H, H, O, C≡CH, H, H, H, O], [AC 1333; H, i-Pr, H, H, O, C ≡ CCH ₃ , H, H, H, O], [AC 1334; H, i-Pr, H, H, O, c-Pr, H, H, H, O], [AC 1335; H, i-Pr, H, H, O, OMe, H, H, H, O], [AC 1336; H, i-Pr, H, H, O, OEt, H, H, H, O], [AC 1337; H, i- Pr, H, H, H, O, Oi-Pr, H, H, H, O], [AC 1338; H, i-Pr, H, H, O, SMe, H, H, H, O], [AC 1339; H, i-Pr, H, H, O, SEt, H, H, H, O], [AC1340; H, i-Pr, H, H, O, CH 2 F, H, H, H, O] , [AC1341; H, i- Pr, H, H, O, CHF 2, H, H, H, O], [AC1342; H, i-Pr, H, H, O, CF 3, H, H, H, O], [AC1343; H, i-Pr, H, H, O, OCH 2 F, H, H, H, O], [AC1344; H, i-Pr, H, H, O, OCHF 2 , H, H, H, O ], [AC1345; H, i-Pr, H, H, O, OCF 3, H, H, H, O], [AC1346; H, i-Pr, H, H, O, SCH ₂ F, H, H, H, O, [AC 1347; H, i-Pr, H, H, O, SCHF ₂ , H, H, H, O], [AC 1348; H, i-Pr , H, H, O, SCF 3, H, H, H, O], [AC1349; H, i-Pr, H, H, O, CN, H, H, H, O], [AC1350; H, i-Pr, H, H, O, NO 2, H, H, H, O], [AC1351; H, i-Pr, H, Me, O, H, H, H, H, O], [AC1352 H, i-Pr , H, Me, O, F, H, H, H, O], [AC1353; H, i-Pr, H, Me, O, Cl, H, H, O], [AC 1354; H, i -Pr, H, Me, O, Br, H, H, H, O], [AC1 355; H, i-Pr, H, Me, O, I, H, H, O, [AC 1356; H , i-Pr, H, Me, O, Me, H, H, H, O], [AC 1357; H, i-Pr, H, Me, O, Et, H, H, H, O], [AC 1358 H, i-Pr, H, Me, O, Pr, H, H, H, O], [AC 1359; H, i-Pr, H, Me, O, i-Pr, H, H, H, O; H, i-Pr, H, Me, O, CH = CH ₂ , H, H, H, O], [AC 1361; H, i-Pr, H, Me, O, C (CH ₃₎ ) = CH ₂ , H, H, H, O], [AC1362; H, i-Pr, H, Me, O, C≡CH, H, H, H, O], [AC1363; H, i-Pr , H, Me, O, C≡CCH ₃ , H, H, H, O], [AC1364; H, i-Pr, H, Me, O, c-Pr, H, H, H, O], [[ AC 1365; H, i-Pr, H, Me, O, OMe, H, H, H, O], [AC 1366; H, i-Pr, H, Me, O, OEt, H, H, H, O] , [AC 1367; H, i-Pr, H, Me, O, Oi-Pr, H, H, H, O], [AC 1368; H, i-Pr, H, Me, O, SMe, H, H, H, O], [AC1369; H, i-Pr, H, Me, O, SEt, H, H, H, O], [AC1370; H, i-Pr, H, Me, O, CH 2 F, H, H, H, O] , [AC1371; H, i-Pr, H, Me, O, CHF 2, H, H, H, O], [AC1372; H, i-Pr, H, Me, O _{, CF 3, H, H,} H, O], [AC1373; H, i-Pr, H, Me, O, OCH 2 F, H, H, H, O], [AC1374; H, i-Pr, _{H, Me, O, OCHF 2} , H, H, H, O], [AC1375; H, i-Pr, H, Me, O, OCF 3, H, H, H, O], [AC1376; H, i-Pr, H, Me, O, SCH ₂ F, H, H, H, O], [AC 1377; H, i-Pr, H, Me, O, SCHF ₂ , H, H, H, O], [AC 1378; H, i-Pr, H, Me, O, SCF ₃ , H, H, H, O], [AC 1379; H, i-Pr, H, M e, O, CN, H, H, H, O, [AC 1380; H, i-Pr, H, Me, O, NO ₂ , H, H, H, O], [AC 1381; H, i-Pr , H, Et, O, H, H, H, H, O], [AC1382; H, i-Pr, H, Et, O, F, H, H, O], [AC 1383; H, i -Pr, H, Et, O, Cl, H, H, H, O], [AC 1384; H, i-Pr, H, Et, O, Br, H, H, H, O], [AC 1385; H , i-Pr, H, Et, O, I, H, H, O], [AC 1386; H, i-Pr, H, Et, O, Me, H, H, H, O], [AC 1387 H, i-Pr, H, Et, O, Et, H, H, H, O], [AC 1388; H, i-Pr, H, Et, O, Pr, H, H, H, O], [AC 1 389; H, i-Pr, H, Et, O, i-Pr, H, H, H, O], [AC 1390; H, i-Pr, H, Et, O, CH = CH ₂ , H, H, H, O], [ AC1391; H, i-Pr, H, Et, O, C (CH 3) = CH 2, H, H, H, O], [AC1392; H, i-Pr, H , Et, O, C≡CH, H , H, H, O], [AC1393; H, i-Pr, H, Et, O, C≡CCH 3, H, H, H, O], [AC1394; H, i-Pr, H, Et, O, c-Pr, H, H, H, O], [AC 1395; H, i-Pr, H, Et, O, OMe, H, H, H, O] ,

[AC1396; H, i-Pr, H, Et, O, OEt, H, H, H, O], [AC 1397; H, i-Pr, H, Et, O, Oi-Pr, H, H, H H, i-Pr, H, Et, O, SMe, H, H, H, O], [AC 1399; H, i-Pr, H, Et, O, SEt, H, H , H, O], [AC1400 ; H, i-Pr, H, Et, O, CH 2 F, H, H, H, O], [AC1401; H, i-Pr, H, Et, O, CHF ₂ , H, H, H, O], [AC 1402; H, i-Pr, H, Et, O, CF ₃ , H, H, H, O], [AC 1403; H, i-Pr, H, Et _{, O, OCH 2 F, H} , H, H, O], [AC1404; H, i-Pr, H, Et, O, OCHF 2, H, H, H, O], [AC1405; H, i- Pr, H, Et, O, OCF 3, H, H, H, O], [AC1406; H, i-Pr, H, Et, O, SCH 2 F, H, H, H, O], [AC1407 H, i-Pr, H, Et, O, SCHF ₂ , H, H, H, O], [AC 1408; H, i-Pr, H, Et, O, SCF ₃ , H, H, H, O H, i-Pr, H, Et, O, CN, H, H, H, O], [AC 1410; H, i-Pr, H, Et, O, NO ₂ , H, H, H, O], [AC 1411; H, i-Pr, H, Pr, O, H, H, H, H, O], [AC 1412; H, i-Pr, H, Pr, O, F, H, H, H, O], [AC 1413; H, i-Pr, H, Pr, O, Cl, H, H, H, O], [AC 1414; H, i-Pr, H, Pr, O, Br, H, H, H, O], [AC 1415; H, i-Pr, H, Pr, O, I, H, H, H, O], [AC 1416; H, i-Pr, H, Pr, O, Me, H, H, H, O], [AC1417; H, i-Pr, H, Pr, O, Et, H, H, H, O], [AC 1418; H, i-Pr, H, Pr, O, Pr, H, H, H, O], [AC 1419; H, i-Pr, H, Pr, O, i-Pr, H, H, H, O], [AC 1420; H, i-Pr, H, Pr, O, CH = CH 2, H, H, H, O], [AC1421; H, i-Pr, H, Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC 1422; H, i-Pr, H, Pr, O, C≡CH, H, H, H, O], [AC 1423; H, iP r, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 1424; H, i-Pr, H, Pr, O, c-Pr, H, H, H, O], [AC 1425; H, i-Pr, H, Pr, O, OMe, H, H, H, O], [AC 1426; H, i-Pr, H, Pr, O, OEt, H, H, H, O H, i-Pr, H, Pr, O, Oi-Pr, H, H, H, O], [AC 1428; H, i-Pr, H, Pr, O, SMe, H, H] , H, O], [AC 1429; H, i-Pr, H, Pr, O, SE t, H, H, H, O], [AC 1430; H, i-Pr, H, Pr, O, CH ₂ F , H, H, H, O ], [AC1431; H, i-Pr, H, Pr, O, CHF 2, H, H, H, O], [AC1432; H, i-Pr, H, Pr, _{O, CF 3, H, H} , H, O], [AC1433; H, i-Pr, H, Pr, O, OCH 2 F, H, H, H, O], [AC1434; H, i-Pr , H, Pr, O, OCHF 2, H, H, H, O], [AC1435; H, i-Pr, H, Pr, O, OCF 3, H, H, H, O], [AC1436; H , i-Pr, H, Pr, O, SCH ₂ F, H, H, H, O], [AC 1437; H, i-Pr, H, Pr, O, SCHF ₂ , H, H, H, O] , [AC 1438; H, i-Pr, H, Pr, O, SCF ₃ , H, H, H, O], [AC 1439; H, i-Pr, H, Pr, O, CN, H, H, H , O], [AC 1440; H, i-Pr, H, Pr, O, NO ₂ , H, H, H, O], [AC 1441; H, i-Pr, H, i-Pr, O, H, H, H, H, O], [AC1442; H, i-Pr, H, i-Pr, O, F, H, H, H, O], [AC 1443; H, i-Pr, H, i- Pr, O, Cl, H, H, H, H, O], [AC 1444; H, i-Pr, H, i-Pr, O, Br, H, H, O], [AC 1445; H, i- Pr, H, i-Pr, O, I, H, H, H, O], [AC 1446; H, i-Pr, H, i-Pr, O, Me, H, H, H, O], [[ AC1447; H, i-Pr, H, i-Pr, O, Et, H, H, H, O], [AC 1448; H, i-Pr, H, i-Pr, O, Pr, H, H, H, O], [AC1449; H, i-Pr, H, i-Pr, O, i-Pr, H, H, H, O], [AC 1450; H, i-Pr, H, i- _{Pr, O, CH = CH 2} , H, H, H, O], [AC1451; H, i-Pr, H, i-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC1452; H, i-Pr, H, i-Pr, O, C≡CH, H, H, H, O], [AC1453; H, i-Pr, H, i-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 1454; H, i-Pr, H, i-Pr, O, c-Pr, H, H, H, O], [AC 1455; H, i -Pr, H, i-Pr, O, OMe, H, H, H, O], [AC 1456; H, i-Pr, H, i-Pr, O, OEt, H, H, H, O], [AC 1457; H, i-Pr, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 1458; H, i-Pr, H, i-Pr, O, SMe, H , H, H, O], [AC 1459; H, i-Pr, H, i-Pr, O, SE t, H, H, H, O], [AC 1460; H, i-Pr, H, i-Pr _{, O, CH 2 F, H} , H, H, O], [AC1461; H, i-Pr, H, i-Pr, O, CHF 2, H, H, H, O], [AC1462; H, i-Pr, H, i- Pr, O, CF 3, H, H, H, O], [AC1463; H, i-Pr, H, i-Pr, O, OCH 2 F, H, H, H , O], [AC1464; H , i-Pr, H, i-Pr, O, OCHF 2, H, H, H, O], [AC1465; H, i-Pr, H, i-Pr, O, OCF ₃ , H, H, H, O], [AC 1466; H, i-Pr, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 1467; H, i-Pr , H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 1468; H, i-Pr, H, i-Pr, O, SCF ₃ , H, H, H, O], [AC1469; H, i-Pr , H, i-Pr, O, CN, H, H, H, O], [AC1470; H, i-Pr, H, i-Pr, O, NO 2, H, H, H, O], [AC1471; H, i-Pr, H, c-Pr, O, H, H, H, H, O], [AC 1472; H, i-Pr, H, c-Pr, O, F, H, H, H, O], [AC 1473; H, i-Pr, H, c-Pr, O, Cl, H, H, H, O], [AC 1474; H, i-Pr, H, c-Pr, O, Br, H, H, H, O], [AC1475; H, i-Pr, H, c-Pr, O, I, H, H, H, O], [AC 14 76; H, i-Pr, H, c-Pr, O, Me, H, H, H, O], [AC 1477; H, i-Pr, H, c-Pr, O, Et, H, H, H, H, O], [AC1478; H, i-Pr, H, c-Pr, O, Pr, H, H, H, O], [AC1479; H, i-Pr, H, c-Pr, O, i-Pr, H, H, H, O], [AC1480; H, i-Pr, H, c-Pr, O, CH = CH 2, H, H, H, O], [AC1481; H, i -Pr, H, c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC1482; H, i-Pr, H, c-Pr, O, C≡CH, H, H, H, O], [AC 1483; H, i-Pr, H, c-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 1484; H, i-Pr, H , c-Pr, O, c-Pr, H, H, H, O], [AC 1485; H, i-Pr, H, c-Pr, O, OMe, H, H, H, O], [AC 1486 H, i-Pr, H, c-Pr, O, OEt, H, H, H, O], [AC 1487; H, i-Pr, H, c-Pr, O, Oi-Pr, H, H , H, O], [AC 1 488; H, i-Pr, H, c-Pr, O, SMe, H, H, H, O], [AC 1489; H, i-Pr, H, c-Pr, O , SEt, H, H, H, O], [AC 1490; H, i-Pr, H, c-Pr, O, CH ₂ F, H, H, H, O], [AC 1491; H, i-Pr , H, c-Pr, O , CHF 2, H, H, H, O], [AC1492; H, i-Pr, H, c-Pr, O, CF 3, H, H, H, O], [AC 1493; H, i-Pr, H, c-Pr, O, OCH ₂ F, H, H, H, O], [AC 1494; H, i-Pr, H, c-Pr, O, OCHF ₂ , H, H, H, O] , [AC1495; H, i-Pr, H, c-Pr, O, OCF 3, H, H, H, O],

[AC 1496; H, i-Pr, H, c-Pr, O, SCH ₂ F, H, H, H, O], [AC 1497; H, i-Pr, H, c-Pr, O, SCHF ₂ , H, H, H, O] , [AC1498; H, i-Pr, H, c-Pr, O, SCF 3, H, H, H, O], [AC1499; H, i-Pr, H, c -Pr, O, CN, H, H, H, H, O], [AC 1500; H, i-Pr, H, c-Pr, O, NO ₂ , H, H, H, O], [AC 1501; H, i-Pr, H, SMe, O, H, H, H, H, O], [AC1502; H, i-Pr, H, SMe, O, F, H, H, H, O], [AC 1503; H, i-Pr, H, SMe, O, Cl, H, H, H, O], [AC 1504; H, i-Pr, H, SMe, O, Br, H, H, H, O], [, AC1505; H, i-Pr, H, SMe, O, I, H, H, H, O], [AC 1506; H, i-Pr, H, SMe, O, Me, H, H, H, O] , [AC1507; H, i-Pr, H, SMe, O, Et, H, H, H, O], [AC 1508; H, i-Pr, H, SMe, O, Pr, H, H, H, O], [AC 1509; H, i-Pr, H, SMe, O, i-Pr, H, H, H, O], [AC 1510; H, i-Pr, H, SMe, O, CH = CH ₂ , H, H, H, O ], [AC1511; H, i-Pr, H, SMe, O, C (CH 3) = CH 2, H, H, H, O], [AC1512; H, i- Pr, H, SMe, O, C≡CH, H, H, H, O], [AC 1513; H, i-Pr, H, SMe, O, C≡ CCH ₃ , H, H, H, O], [AC 1514; H, i-Pr, H, SMe, O, c-Pr, H, H, H, O], [AC 1515; H, i-Pr, H, SMe, O, OMe, H, H, H H, i-Pr, H, SMe, O, OEt, H, H, H, O], [AC 1517; H, i-Pr, H, SMe, O, Oi-Pr, H , H, H, O], [AC1518; H, i-Pr, H, SMe, O, SMe, H, H, H, O], [AC 1519; H, i-Pr, H, SMe, O, SEt , H, H, H, O ], [AC1520; H, i-Pr, H, SMe, O, CH 2 F, H, H, H, O], [AC1521; H, i-Pr, H, SMe _{, O, CHF 2, H,} H, H, O], [AC1522; H, i-Pr, H, SMe, O _{, CF 3, H, H,} H, O], [AC1523; H, i-Pr, H, SMe, O, OCH 2 F, H, H, H, O], [AC1524; H, i-Pr, _{H, SMe, O, OCHF 2} , H, H, H, O], [AC1525; H, i-Pr, H, SMe, O, OCF 3, H, H, H, O], [AC1526; H, i-Pr, H, SMe, O, SCH 2 F, H, H, H, O], [AC1527; H, i-Pr, H, SMe, O, SCHF 2, H, H, H, O], [AC1528; H, i-Pr , H, SMe, O, SCF 3, H, H, H, O], [AC1529; H, i-Pr, H, SMe, O, CN, H, H, H, O], [AC 1530; H, i-Pr, H, SMe, O, NO ₂ , H, H, H, O], [AC 1531; H, i-Pr, H, OMe, O, H, H, H , H, O], [AC 1532; H, i-Pr, H, OMe, O, F, H, H, H, O], [AC 1533; H, i-Pr, H, OMe, O, Cl, H , H, H, O], [AC1534; H, i-Pr, H, OMe, O, Br, H, H, H, O], [AC1535; H, i-Pr, H, OMe, O, I , H, H, H, O], [AC 1536; H, i-Pr, H, OMe, O, Me, H, H, H, O], [AC 1537; H, i-Pr, H, OMe, O , Et, H, H, H, O], [AC1538; H, i-Pr, H, OMe, O, Pr, H, H, H, O], [AC1539; H, i-Pr, H, OMe , O, i-Pr, H , H, H, O], [AC1540; H, i-Pr, H, OMe, O, CH = CH 2, H, H, H, O], [AC1541; H, i-Pr, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC1542; H, i-Pr, H, OMe, O, C≡CH, H, H , H, O], [AC 1543; H, i-Pr, H, OMe, O, C≡CCH ₃ , H, H, H, O], [AC 1544; H, i-Pr, H, OMe, O, c-Pr, H, H, H, O], [AC1545; H, i-Pr, H, OMe, O, OMe, H, H, H, O], [AC 1546; H, i-Pr, H, OMe, O, OEt, H, H, H, O], [AC1547; H, i-Pr, H, OMe, O, Oi-Pr, H, H, H, O], [AC1548; H, i- Pr, H, OMe, O, SMe, H, H, H, O], [AC154 9; H, i-Pr, H, OMe, O, SEt, H, H, H, O], [AC1550; H, i-Pr, H, OMe, O, CH 2 F, H, H, H, O], [AC1551; H, i-Pr, H, OMe, O, CHF 2, H, H, H, O], [AC1552; H, i-Pr, H, OMe, O, CF 3, H, H, H, O], [ AC1553; H, i-Pr, H, OMe, O, OCH 2 F, H, H, H, O], [AC1554; H, i-Pr, H, OMe, O, _{OCHF 2, H, H, H} , O], [AC1555; H, i-Pr, H, OMe, O, OCF 3, H, H, H, O], [AC1556; H, i-Pr, H, _{OMe, O, SCH 2 F,} H, H, H, O], [AC1557; H, i-Pr, H, OMe, O, SCHF 2, H, H, H, O], [AC1558; H, i -Pr, H, OMe, O, SCF 3, H, H, H, O], [AC1559; H, i-Pr, H, OMe, O, CN, H, H, H, O], [AC1560; H, i-Pr, H, OMe, O, NO 2, H, H, H, O], [AC1561; H, i-Pr, H, F, O, H, H, H, H, O], [AC1562; H, i-Pr, H, F, O, F, H, H, O], [AC 1563; H, i-Pr, H, F, O, Cl, H, H, H, O H, i-Pr, H, F, O, Br, H, H, O], [AC 1565; H, i-Pr, H, F, O, I, H, H, H] H, i-Pr, H, F, O, Me, H, H, H, O], [AC 1567; H, i-Pr, H, F, O, Et, H, H , H, O], [AC1568; H, i-Pr, H, F, O, Pr, H, H, H, O], [AC 1569; H, i-Pr, H, F, O, i-Pr , H, H, H, O ], [AC1570; H, i-Pr, H, F, O, CH = CH 2, H, H, H, O], [AC1571; H, i-Pr, H, _{F, O, C (CH 3} ) = CH 2, H, H, H, O], [AC1572; H, i-Pr, H, F, O, C≡CH, H, H, H, O], [AC 1573; H, i-Pr, H, F, O, C≡CCH ₃ , H, H, H, O], [AC 1574; H, i-Pr, H, F, O, c-Pr, H, H, H, O], [AC1575; H, i-Pr, H, F, O, OMe, H, H, H, O], [AC 1576; H, i-Pr, H , F, O, OEt, H, H, H, O], [AC 1577; H, i-Pr, H, F, O, Oi-Pr, H, H, H, O], [AC 1578; H, i -Pr, H, F, O, SMe, H, H, H, O], [AC1579; H, i-Pr, H, F, O, SEt, H, H, H, O], [AC 1580; H , i-Pr, H, F , O, CH 2 F, H, H, H, O], [AC1581; H, i-Pr, H, F, O, CHF 2, H, H, H, O] , [AC1582; H, i- Pr, H, F, O, CF 3, H, H, H, O], [AC1583; H, i-Pr, H, F, O, OCH 2 F, H, H , H, O], [AC 1584; H, i-Pr, H, F, O, OCHF ₂ , H, H, H, O], [AC 1585; H, i-Pr, H, F, O, OCF ₃ , H, H, H, O], [AC 1586; H, i-Pr, H, F, O, SCH ₂ F, H, H, H, O], [AC 1587; H, i-Pr, H, F , O, SCHF ₂ , H, H, H, O], [AC1588; H, i-Pr, H, F, O, SCF ₃ , H, H, H, O], [AC1589; H, i-Pr , H, F, O, CN, H, H, H, O], [AC 1590; H, i-Pr, H, F, O, NO ₂ , H, H, H, O], [AC 1591; H, i-Pr, H, Cl, O, H, H, H, H, O], [AC1592; H, i-Pr, H, Cl, O, F, H, H, H, O], [AC1593; H, i-Pr, H, Cl, O, Cl, H, H, H, O], [AC1594; H, i-Pr, H, Cl, O, Br, H, H, H, O],

[AC 1595; H, i-Pr, H, Cl, O, I, H, H, H, O], [AC 1596; H, i-Pr, H, Cl, O, Me, H, H, H, O H, i-Pr, H, Cl, O, Et, H, H, H, O], [AC 1598; H, i-Pr, H, Cl, O, Pr, H, H, H] H, i-Pr, H, Cl, O, i-Pr, H, H, H, O], [AC1600; H, i-Pr, H, Cl, O, CH = CH _{2, H, H, H,} O], [AC1601; H, i-Pr, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC1602; H, i -Pr, H, Cl, O, C≡CH, H, H, H, O], [AC 1603; H, i-Pr, H, Cl, O, C≡ CCH ₃ , H, H, H, O] [AC1604; H, i-Pr, H, Cl, O, c-Pr, H, H, H, O], [AC 1605; H, i-Pr, H, Cl, O, OMe, H, H, H, O], [AC 1 606; H, i-Pr, H, Cl, O, OEt, H, H, H, O], [AC 1607; H, i-Pr, H, Cl, O, Oi-Pr, H, H, H, O], [AC 1608; H, i-Pr, H, Cl, O, SMe, H, H, H, O], [AC 1609; H, i-Pr, H, Cl, O, SEt, H, H, H, O], [AC 1610; H, i-Pr, H, Cl, O, CH ₂ F, H, H, H, O], [AC 1611; H, i-Pr, H, _{Cl, O, CHF 2, H} , H, H, O], [AC1612; H, i-Pr, H, Cl, O, CF 3, H, H, H, O], [AC1613; H, i- Pr, H, Cl, O, OCH 2 F, H, H, H, O], [AC1614; H, i-Pr, H, Cl, O, OCHF 2, H, H, H, O], [AC1615 ; H, i-Pr, H , Cl, O, OCF 3, H, H, H, O], [AC1616; H, i-Pr, H, Cl, O, SCH 2 F, H, H, H, O, [AC1617; H, i-Pr, H, Cl, O, SCHF ₂ , H, H, H, O], [AC 1618; H, i-Pr, H, Cl, O, SCF ₃ , H, H, H, O], [AC 1619; H, i-Pr, H, Cl, O, CN, H, H, H, O], [AC 1620; H, i-Pr, H, Cl, O, NO ₂ , H, H, H, O], [AC1621; H, i-Pr, H, Br, O, H, H, H, H, O], [[ AC1622; H, i-Pr, H, Br, O, F, H, H, O], [AC1623; H, i-Pr, H, Br, O, Cl, H, H, H, O] [AC1624; H, i-Pr, H, Br, O, Br, H, H, O], [AC1625; H, i-Pr, H, Br, O, I, H, H, H, H, O], [AC 1626; H, i-Pr, H, Br, O, Me, H, H, H, O], [AC 1627; H, i-Pr, H, Br, O, Et, H, H, H, H, O], [AC 1628; H, i-Pr, H, Br, O, Pr, H, H, H, O], [AC 1629; H, i-Pr, H, Br, O, i-Pr, H, H, H, O] , [AC1630; H, i-Pr, H, Br, O, CH = CH 2, H, H, H, O], [AC1631; H, i-Pr, H, Br _{, O, C (CH 3)} = CH 2, H, H, H, O], [AC1632; H, i-Pr, H, Br, O, C≡CH, H, H, H, O], [ AC1633; H, i-Pr, H, Br, O, C≡CCH 3, H, H, H, O], [AC1634; H, i-Pr, H, Br, O, c-Pr, H, H , H, O], [AC 1635; H, i-Pr, H, Br, O, H, H, H, O], [AC 1636; H, i-Pr, H, Br, O, OEt, H , H, H, O], [AC 1637; H, i-Pr, H, Br, O, Oi-Pr, H, H, H, O], [AC 1638; H, i-Pr, H, Br, O , SMe, H, H, H, O], [AC 1639; H, i-Pr, H, Br, O, SEt, H, H, H, O], [AC 1640; H, i-Pr, H, Br _{, O, CH 2 F, H} , H, H, O], [AC1641; H, i-Pr, H, Br, O, CHF 2, H, H, H, O], [AC1642; H, i- Pr, H, Br, O, CF 3, H, H, H, O], [AC1643; H, i-Pr, H, Br, O, OCH 2 F, H, H, H, O], [AC1644 ; H, i-Pr, H , Br, O, OCHF 2, H, H, H, O], [AC1645; H, i-Pr, H, Br, O, OCF 3, H, H, H, O H, i-Pr, H, Br, O, SCH ₂ F, H, H, H, O], [AC 1647; H, i-Pr, H, Br, O, SCHF ₂ , H, H, H, O], [AC 1648; H, i-Pr, H, Br, O, SCF ₃ , H, H, H, O], [AC 16 49; H, i-Pr, H, Br, O, CN, H, H, H, O], [AC1650; H, i-Pr, H, Br, O, NO 2, H, H, H, O H, c-Pr, H, H, O, H, H, H, H, O], [AC 1652; H, c-Pr, H, H, O, F, H, H, H] H, c-Pr, H, H, H, O, Cl, H, H, O], [AC1654; H, c-Pr, H, H, O, Br, H, H , H, O], [AC 1655; H, c-Pr, H, H, O, I, H, H, H, O], [AC 1656; H, c-Pr, H, H, O, Me, H , H, H, O], [AC 1657; H, c-Pr, H, H, O, Et, H, H, H, O], [AC 1658; H, c-Pr, H, H, O, Pr , H, H, H, O], [AC 1659; H, c-Pr, H, H, O, i-Pr, H, H, H, O], [AC 1660; H, c-Pr, H, H _{, O, CH = CH 2,} H, H, H, O], [AC1661; H, c-Pr, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC1662; H, c-Pr, H, H, O, C≡CH, H, H, H, O], [AC1663; H, c-Pr, H, H, O, C≡ CCH ₃ , H, H, H, O], [AC1664; H, c-Pr, H, H, O, c-Pr, H, H, H, O], [AC 1665; H, c-Pr, H, H, O, OMe, H, H, H, O], [AC 1 666; H, c-Pr, H, H, O, OEt, H, H, H, O], [AC 1 667; H, c-Pr, H, H, O, Oi-Pr, H, H, H, O, [AC 1668; H, c-Pr, H, H, O, SMe, H, H, O], [AC 1669; H, c-Pr, H, H, O, SEt, H, H, H, O], [AC1670; H, c-Pr, H, H, O, CH 2 F, H, H, H, O], [AC1671; H, c-Pr, H, H, O, CHF 2, H, H, H, O], [AC1672; H, c-Pr, H, H, O, CF 3, H, H, H, O], [ AC1673; H, c-Pr, H, H, O, OCH 2 F, H, H, H, O], [AC1674; H, c-Pr, H, H, O, OCHF 2, H, H, H , O], [AC1675; H , c-Pr, H, H, O, OCF 3, H, H, H, O], [AC1676; H, c-Pr, H, H, O, SCH 2 F, H, H, H, O], [AC 1677; H, c-Pr, H, H, O, SCHF 2, H, H, H, O], [AC1678; H, c-Pr, H, H, O, SCF 3, H, H, H, O] , [AC1679; H, c- Pr, H, H, O, CN, H, H, H, O], [AC1680; H, c-Pr, H, H, O, NO 2, H, H, H H, c-Pr, H, Me, O, H, H, H, H, O], [AC 1682; H, c-Pr, H, Me, O, F, H, H , H, O], [AC 1683; H, c-Pr, H, Me, O, Cl, H, H, H, O], [AC 1684; H, c-Pr, H, Me, O, Br, H , H, H, O], [AC 1 685; H, c-Pr, H, Me, O, I, H, H, H, O], [AC 1686; H, c-Pr, H, Me, O, Me , H, H, H, O], [AC 1687; H, c-Pr, H, Me, O, Et, H, H, H, O], [AC 1688; H, c-Pr, H, Me, O , Pr, H, H, H, O], [AC 1689; H, c-Pr, H, Me, O, i-Pr, H, H, H, O], [AC 1690; H, c-Pr, H , Me, O, CH = CH 2, H, H, H, O], [AC1691; H, c-Pr, H, Me, O, C (CH 3) = CH 2, H, H, H, O H, c-Pr, H, Me, O, C≡CH, H, H, H, O], [AC 1693; H, c-Pr, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 1694; H, c-Pr, H, Me, O, c-Pr, H, H, H, O],

[AC1695; H, c-Pr, H, Me, O, OMe, H, H, H, O], [AC 1 696; H, c-Pr, H, Me, O, OEt, H, H, H, O H, c-Pr, H, Me, O, Oi-Pr, H, H, H, O], [AC 1698; H, c-Pr, H, Me, O, SMe, H, H] , H, O], [AC1699 ; H, c-Pr, H, Me, O, SEt, H, H, H, O], [AC1700; H, c-Pr, H, Me, O, CH 2 F , H, H, H, O ], [AC1701; H, c-Pr, H, Me, O, CHF 2, H, H, H, O], [AC1702; H, c-Pr, H, Me, _{O, CF 3, H, H} , H, O], [AC1703; H, c-Pr, H, Me, O, OCH 2 F, H, H, H, O], [AC1704; H, c-Pr , H, Me, O, OCHF 2, H, H, H, O], [AC1705; H, c-Pr, H, Me, O, OCF 3, H, H, H, O], [AC1706; H , c-Pr, H, Me, O, SCH ₂ F, H, H, H, O], [AC 1707; H, c-Pr, H, Me, O, SCHF ₂ , H, H, H, O] , [AC1708; H, c- Pr, H, Me, O, SCF 3, H, H, H, O], [AC1709; H, c-Pr, H, Me, O, CN, H, H, H , O], [AC 1710; H, c-Pr, H, Me, O, NO ₂ , H, H, H, O], [AC 1711; H, c-Pr, H, Et, O, H, H, H, H, O], [AC 1712; H, c-Pr, H, Et, O, F, H, H, H, O], [AC 1713; H, c-Pr, H, Et, O, Cl, H, H, H, O], [AC1714; H, c-Pr, H, Et, O, Br, H, H, H, O], [AC 1715; H, c-Pr, H, Et, O, H, c-Pr, H, Et, O, Me, H, H, H, O], [AC 1717; H, c-Pr, H, Et, I, H, H, H, O], [AC1716; O, Et, H, H, H, O, [AC1718; H, c-Pr, H, Et, O, Pr, H, H, H, O], [AC1719; H, c-Pr, H, Et, O, i-Pr, H, H, H, O], [AC1720; H, c-Pr, H, Et, O, CH = CH 2, H, H, H, O], [AC1721; H , c-Pr, H, Et , O, C (CH 3) = CH 2, H, H, H, O], [AC1722; H, c-Pr, H , Et, O, C≡CH, H , H, H, O], [AC1723; H, c-Pr, H, Et, O, C≡CCH 3, H, H, H, O], [AC1724; H, c-Pr, H, Et, O, c-Pr, H, H, H, O], [AC 1725; H, c-Pr, H, Et, O, OMe, H, H, H, O] H, c-Pr, H, Et, O, OEt, H, H, H, O], [AC 1727; H, c-Pr, H, Et, O, Oi-Pr, H, H, H, O], [AC1728; H, c-Pr, H, Et, O, SMe, H, H, H, O], [AC 1729; H, c-Pr, H, Et, O, SEt, H, H, H, O], [ AC1730; H, c-Pr, H, Et, O, CH 2 F, H, H, H, O], [AC1731; H, c-Pr, H, Et, O, _{CHF 2, H, H, H} , O], [AC1732; H, c-Pr, H, Et, O, CF 3, H, H, H, O], [AC1733; H, c-Pr, H, _{Et, O, OCH 2 F,} H, H, H, O], [AC1734; H, c-Pr, H, Et, O, OCHF 2, H, H, H, O], [AC1735; H, c -Pr, H, Et, O, OCF 3, H, H, H, O], [AC1736; H, c-Pr, H, Et, O, SCH 2 F, H, H, H, O], [ AC1737; H, c-Pr, H, Et, O, SCHF 2, H, H, H, O], [AC1738; H, c-Pr, H, Et, O, SCF 3, H, H, H, H, c-Pr, H, Et, O, CN, H, H, H, O], [AC 1740; H, c-Pr, H, Et, O, NO ₂ , H, H] , H, O], [AC 1741; H, c-Pr, H, Pr, O, H, H, H, H, O], [AC 1742; H, c-Pr, H, Pr, O, F, H , H, H, O], [AC 1743; H, c-Pr, H, Pr, O, Cl, H, H, H, O], [AC 1744; H, c-Pr, H, Pr, O, Br , H, H, H, O], [AC 1745; H, c-Pr, H, Pr, O, I, H, H, H, O], [AC 1746; H, c-Pr, H, Pr, O , Me, H, H, H, O], [AC 1747; H, c-Pr, H, Pr, O, Et, H, H, H, O], [AC 1 748; H, c-Pr, H, Pr , O, Pr, H, H, H, O], [AC 1749; H, c-Pr, H, Pr, O, i-Pr, H, H, H, O], [A C1750; H, c-Pr, H, Pr, O, CH = CH 2, H, H, H, O], [AC1751; H, c-Pr, H, Pr, O, C (CH 3) = CH ₂ , H, H, H, O], [AC1752; H, c-Pr, H, Pr, O, C≡CH, H, H, H, O], [AC1753; H, c-Pr, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 1754; H, c-Pr, H, Pr, O, c-Pr, H, H, H, O], [AC 1755; H , c-Pr, H, Pr, O, OMe, H, H, H, O], [AC 1756; H, c-Pr, H, Pr, O, OEt, H, H, H, O], [AC 1757 H, c-Pr, H, Pr, O, Oi-Pr, H, H, H, O], [AC 1758; H, c-Pr, H, Pr, O, SMe, H, H, H, O H, c-Pr, H, Pr, O, SEt, H, H, H, O], [AC 1760; H, c-Pr, H, Pr, O, CH ₂ F, H, H] , H, O], [AC1761 ; H, c-Pr, H, Pr, O, CHF 2, H, H, H, O], [AC1762; H, c-Pr, H, Pr, O, CF 3 , H, H, H, O], [AC1763; H, c-Pr, H, Pr, O, OCH ₂ F, H, H, H, O], [AC 1764; H, c-Pr, H, Pr , O, OCHF ₂ , H, H, H, O], [AC 1765; H, c-Pr, H, Pr, O, OCF ₃ , H, H, H, O], [AC 1766; H, c-Pr , H, Pr, O, SCH ₂ F, H, H, H, O], [AC 1767; H, c-Pr, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 1768; H, c-Pr, H, Pr, O, SCF 3, H, H, H, O], [AC1769; H, c-Pr, H, Pr, O, CN, H, H, H, O], [AC 1 770; H, c-Pr, H, Pr, O, NO ₂ , H, H, O], [AC 1771; H, c-Pr, H, i-Pr, O, H, H, H, H, O], [AC1772; H, c-Pr, H, i-Pr, O, F, H, H, H, O], [AC1773; H, c-Pr, H, i-Pr, O, Cl, H, H, H, O], [AC 1774; H, c-Pr, H, i-Pr, O, Br, H, H, H, O], [AC 1 775; H, c-Pr, H, i-Pr, O, I, H, H, H, O], [AC 1776; H, c-Pr, H, i-Pr, O, Me, H, H , H, O], [AC1 777; H, c-Pr, H, i-Pr, O, Et, H, H, H, O], [AC 1778; H, c-Pr, H, i-Pr, O , Pr, H, H, H, O], [AC 1779; H, c-Pr, H, i-Pr, O, i-Pr, H, H, H, O], [AC 1 780; H, c-Pr , H, i-Pr, O , CH = CH 2, H, H, H, O], [AC1781; H, c-Pr, H, i-Pr, O, C (CH 3) = CH 2, H , H, H, O], [AC 1782; H, c-Pr, H, i-Pr, O, C≡CH, H, H, H, O], [AC 1783; H, c-Pr, H, i -Pr, O, C≡CCH ₃ , H, H, H, O], [AC 1784; H, c-Pr, H, i-Pr, O, c-Pr, H, H, H, O], [[ AC 1785; H, c-Pr, H, i-Pr, O, OMe, H, H, H, O], [AC 1786; H, c-Pr, H, i-Pr, O, OEt, H, H, H, O], [AC 1787; H, c-Pr, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 1788; H, c-Pr, H, i-Pr, O, SMe, H, H, H, O], [AC 1 789; H, c-Pr, H, i-Pr, O, SE t, H, H, H, O], [AC 1 790; H, c-Pr, H, i-Pr, O, CH 2 F, H, H, H, O], [AC1791; H, c-Pr, H, i-Pr, O, CHF 2, H, H, H, O], [AC1792; H, c-Pr , H, i-Pr, O, CF 3, H, H, H, O], [AC1793; H, c-Pr, H, i-Pr, O, OCH 2 F, H, H, H, O] , [AC1794; H, c-Pr, H, i-Pr, O, OCHF 2, H, H, H, O],

[AC1795; H, c-Pr , H, i-Pr, O, OCF 3, H, H, H, O], [AC1796; H, c-Pr, H, i-Pr, O, SCH 2 F, H, H, H, O], [AC 1 797; H, c-Pr, H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 1798; H, c-Pr, H, i _{-Pr, O, SCF 3, H} , H, H, O], [AC1799; H, c-Pr, H, i-Pr, O, CN, H, H, H, O], [AC1800; H, c-Pr, H, i-Pr, O, NO ₂ , H, H, H, O], [AC 1801; H, c-Pr, H, c-Pr, O, H, H, H, H, O H, c-Pr, H, c-Pr, O, F, H, H, H, O], [AC 1803; H, c-Pr, H, c-Pr, O, Cl, H] , H, H, O], [AC 1804, H, c-Pr, H, c-Pr, O, Br, H, H, H, O], [AC 1805; H, c-Pr, H, c-Pr , O, I, H, H, H, O, [AC 1 806; H, c-Pr, H, c-Pr, O, Me, H, H, H, O], [AC 1 807; H, c-Pr , H, c-Pr, O, Et, H, H, H, O], [AC 1808; H, c-Pr, H, c-Pr, O, Pr, H, H, H, O], [AC 1809 H, c-Pr, H, c-Pr, O, i-Pr, H, H, H, O], [AC 1810; H, c-Pr, H, c-Pr, O, CH = CH ₂ , H, H, H, O] , [AC1811; H, c-Pr, H, c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC1812; H, c -Pr, H, c-Pr, O, C≡CH, H, H, H, O], [AC 1813; H, c-Pr, H, c-Pr, O, C≡ CCH ₃ , H, H, H H, O], [AC 1814; H, c-Pr, H, c-Pr, O, c-Pr, H, H, H, O], [AC 1815; H, c-Pr, H, c-Pr, O, OMe, H, H, H, O], [AC1816; H, c-Pr, H, c-Pr, O, OEt, H, H, H, O], [AC 1817; H, c-Pr, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC1818; H, c-Pr, H, c-Pr, O, SMe, H, H, H, O], [[ AC 1819; H, c-Pr, H, c-Pr, O, SEt, H, H, H, O], [AC 1820; H, c-Pr, H, c-Pr, O, CH ₂ F, H, H, H, O], [ AC1821; H, c-Pr, H, c-Pr, O, CHF 2, H, H, H, O], [AC1822; H, c-Pr, H, c-Pr, O, CF 3, H, H, H, O], [ AC1823; H, c-Pr, H, c-Pr, O, OCH 2 F, H, H, H, O], [AC1824; H, c-Pr, H, c- _{Pr, O, OCHF 2, H} , H, H, O], [AC1825; H, c-Pr, H, c-Pr, O, OCF 3, H, H, H, O], [AC1826; H, c-Pr, H, c-Pr, O, SCH ₂ F, H, H, H, O], [AC 1827; H, c-Pr, H, c-Pr, O, SCHF ₂ , H, H, H , O], [AC1828; H , c-Pr, H, c-Pr, O, SCF 3, H, H, H, O], [AC1829; H, c-Pr, H, c-Pr, O, CN, H, H, H, O], [AC1830; H, c-Pr, H, c-Pr, O, NO 2, H, H, H, O], [AC1831; H, c-Pr, H , SMe, O, H, H, H, H, H, O], [AC 1832; H, c-Pr, H, SMe, O, F, H, H, O], [AC 1833; H, c-Pr , H, SMe, O, Cl, H, H, H, O], [AC 1834; H, c-Pr, H, SMe, O, Br, H, H, O], [AC 1835; H, c -Pr, H, SMe, O, I, H, H, H, O], [AC 1836; H, c-Pr, H, SMe, O, Me, H, H, H, O], [AC 1837; H , c-Pr, H, SMe, O, Et, H, H, O], [AC 1838; H, c-Pr, H, SMe, O, Pr, H, H, H, O], [AC 1839 ; H, c-Pr, H , SMe, O, i-Pr, H, H, H, O], [AC1840; H, c-Pr, H, SMe, O, CH = CH 2, H, H, H, O], [AC1841; H, c-Pr, H, SMe, O, C (CH 3) = CH 2, H, H, H, O], [AC1842; H, c-Pr, H, SMe , O, C≡CH, H, H, H, O], [AC 1843; H, c-Pr, H, SMe, O, C≡ CCH ₃ , H, H, H, O], [AC 1844; H, c-Pr, H, SMe, O, c-Pr, H, H, H, O], [AC 1845; H, c-Pr, H, SMe, O, OMe, H, H, H, O], [ AC 1846; H, c-Pr, H, SMe, O, OEt, H, H, H, O], [AC 1 847; H, c-Pr, H, SMe, O, Oi-Pr, H, H, H, O], [AC1848; H, c-Pr, H, SMe, O, SMe, H, H, H, O], [ AC1849; H, c-Pr, H, SMe, O, SEt, H, H, H, O], [AC1850; H, c-Pr, H, SMe, O, CH 2 F, H, H, H, O], [AC1851; H, c-Pr, H, SMe, O, CHF 2, H, H, H, O], [AC1852; H, c-Pr, H, SMe, O, CF 3, H, H, H, O], [ AC1853; H, c-Pr, H, SMe, O, OCH 2 F, H, H, H, O], [AC1854; H, c-Pr, H, SMe, O, _{OCHF 2, H, H, H} , O], [AC1855; H, c-Pr, H, SMe, O, OCF 3, H, H, H, O], [AC1856; H, c-Pr, H, SMe, O, SCH ₂ F, H, H, H, O, [AC 1857; H, c-Pr, H, SMe, O, SCHF ₂ , H, H, H, O], [AC 1858; H, c -Pr, H, SMe, O, SCF 3, H, H, H, O], [AC1859; H, c-Pr, H, SMe, O, CN, H, H, H, O], [AC1860; H, c-Pr, H, SMe, O, NO 2, H, H, H, O], [AC1861; H, c-Pr, H, OMe, O, H, H, H, H, O], [AC1862; H, c-Pr, H, OMe, O, F, H, H, H, O], [AC1863; H, c-Pr, H, OMe, O, Cl, H, H, H, O H, c-Pr, H, OMe, O, Br, H, H, O], [AC 1865; H, c-Pr, H, OMe, O, I, H, H, H] H, c-Pr, H, OMe, O, Me, H, H, H, O], [AC 1867; H, c-Pr, H, OMe, O, Et, H, H , H, O], [AC 1868; H, c-Pr, H, OMe, O, Pr, H, H, H, O], [AC 1869; H, c-Pr, H, OMe, O, i-Pr , H, H, H, O ], [AC1870; H, c-Pr, H, OMe, O, CH = CH 2, H, H, H, O], [AC1871; H, c-Pr, H, _{OMe, O, C (CH 3} ) = CH 2, H, H, H, O], [AC1872; H, c-Pr, H, OMe, O, C≡CH, H, H, H, O], [AC1873; H, c-Pr, H, OMe, O, C≡CCH ₃ , H, H, H, O], [AC 1874; H, c-Pr, H, OMe, O, c-Pr, H, H, H, O], [AC 1875; H, c-Pr, H, OMe , O, OMe, H, H, H, O], [AC1876; H, c-Pr, H, OMe, O, OEt, H, H, H, O], [AC 1877; H, c-Pr, H , OMe, O, Oi-Pr, H, H, H, O], [AC 1878; H, c-Pr, H, OMe, O, SMe, H, H, H, O], [AC 1879; H, c -Pr, H, OMe, O, SEt, H, H, H, O], [AC1880; H, c-Pr, H, OMe, O, CH 2 F, H, H, H, O], [AC1881 ; H, c-Pr, H , OMe, O, CHF 2, H, H, H, O], [AC1882; H, c-Pr, H, OMe, O, CF 3, H, H, H, O H, c-Pr, H, OMe, O, OCH ₂ F, H, H, H, O], [AC 1884; H, c-Pr, H, OMe, O, OCHF ₂ , H, H, H, O], [ AC1885; H, c-Pr, H, OMe, O, OCF 3, H, H, H, O], [AC1886; H, c-Pr, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 1887; H, c-Pr, H, OMe, O, SCHF ₂ , H, H, H, O], [AC 1888; H, c-Pr, H, _{OMe, O, SCF 3, H} , H, H, O], [AC1889; H, c-Pr, H, OMe, O, CN, H, H, H, O], [AC1890; H, c-Pr , H, OMe, O, NO 2, H, H, H, O], [AC1891; H, c-Pr, H, F, O, H, H, H, H, O], [AC1892; H, c-Pr, H, F, O, F, H, H, H, O], [AC 1893; H, c-Pr, H, F, O, Cl, H, H, H, O],

[AC1894; H, c-Pr, H, F, O, Br, H, H, O], [AC 1895; H, c-Pr, H, F, O, I, H, H, H, O H, c-Pr, H, F, O, Me, H, H, H, O], [AC 1897; H, c-Pr, H, F, O, Et, H, H, H] H, c-Pr, H, F, O, Pr, H, H, H, O], [AC 1899; H, c-Pr, H, F, O, i-Pr, H , H, H, O], [AC1900; H, c-Pr, H, F, O, CH = CH 2, H, H, H, O], [AC1901; H, c-Pr, H, F, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC1902; H, c-Pr, H, F, O, C≡CH, H, H, H, O], [AC 1903 H, c-Pr, H, F, O, C≡CCH ₃ , H, H, H, O], [AC 1904; H, c-Pr, H, F, O, c-Pr, H, H, H H, O], [AC 1905; H, c-Pr, H, F, O, OMe, H, H, H, O], [AC 1906; H, c-Pr, H, F, O, OEt, H, H, H, O], [AC 1907; H, c-Pr, H, F, O, Oi-Pr, H, H, H, O], [AC 1908; H, c-Pr, H, F, O, SMe, H, H, H, O], [AC 1 909; H, c-Pr, H, F, O, SE t, H, H, H, O], [AC 1910; H, c-Pr, H, F, _{O, CH 2 F, H,} H, H, O], [AC1911; H, c-Pr, H, F, O, CHF 2, H, H, H, O], [AC1912; H, c-Pr , H, F, O, CF 3, H, H, H, O], [AC1913; H, c-Pr, H, F, O, OCH 2 F, H, H, H, O], [AC1914; H, c-Pr, H, F, O, OCHF 2, H, H, H, O], [AC1915; H, c-Pr, H, F, O, OCF 3, H, H, H, O] H, c-Pr, H, F, O, SCH ₂ F, H, H, H, O], [AC 1917; H, c-Pr, H, F, O, SCHF ₂ , H, H , H, O], [AC 1918; H, c-Pr, H, F, O, SCF ₃ , H, H, H, O], [AC 1919; H, c-Pr, H, F, O, CN, H, H, H, O] , [AC1920; H, c-Pr, H, F, O, NO 2, H, H, H, O], [AC1921; H, c-Pr, H, Cl, O , H, H, H , H, O], [AC1922; H, c-Pr, H, Cl, O, F, H, H, H, O], [AC 1 923; H, c-Pr, H, Cl, O, Cl, H , H, H, O], [AC 1 924; H, c-Pr, H, Cl, O, Br, H, H, H, O], [AC 1 925; H, c-Pr, H, Cl, O, I , H, H, H, O], [AC 1926; H, c-Pr, H, Cl, O, Me, H, H, H, O], [AC 1 927; H, c-Pr, H, Cl, O , Et, H, H, H, O], [AC 1928; H, c-Pr, H, Cl, O, Pr, H, H, H, O], [AC 1 929; H, c-Pr, H, Cl , O, i-Pr, H , H, H, O], [AC1930; H, c-Pr, H, Cl, O, CH = CH 2, H, H, H, O], [AC1931; H, c-Pr, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC1932; H, c-Pr, H, Cl, O, C≡CH, H, H , H, O], [AC 1933; H, c-Pr, H, Cl, O, C≡CCH ₃ , H, H, H, O], [AC 1934; H, c-Pr, H, Cl, O, c-Pr, H, H, H, O], [AC 1935; H, c-Pr, H, Cl, O, OMe, H, H, H, O], [AC 1 936; H, c-Pr, H, Cl, O, OEt, H, H, H, O], [AC 1937; H, c-Pr, H, Cl, O, Oi-Pr, H, H, H, O], [AC 1938; H, c- Pr, H, Cl, O, SMe, H, H, H, O], [AC 1939; H, c-Pr, H, Cl, O, SE t, H, H, H, O], [AC 1940; H, c-Pr, H, Cl, O, CH 2 F, H, H, H, O], [AC1941; H, c-Pr, H, Cl, O, CHF 2, H, H, H, O], [AC1942; H, c-Pr , H, Cl, O, CF 3, H, H, H, O], [AC1943; H, c-Pr, H, Cl, O, OCH 2 F, H, H, H, O], [AC 1 944; H, c-Pr, H, Cl, O, OCHF ₂ , H, H, H, O], [AC 1945; H, c-Pr, H, Cl, O, OCF ₃ , H, H, H, O], [AC 1946; H, c-Pr, H, Cl, O, SCH ₂ F, H, H, H, O], [AC 1947; H, c-Pr, H, Cl, O, SCHF ₂ , H, H, H, O], [AC 1948; H, c-Pr, H, Cl, O, SCF ₃ , H, H, H, O ], [AC1949; H, c -Pr, H, Cl, O, CN, H, H, H, O], [AC1950; H, c-Pr, H, Cl, O, NO 2, H, H, H, O], [AC1951; H, c-Pr, H, Br, O, H, H, H, H, O], [AC 1952; H, c-Pr, H, Br, O, F, H, H, H, O], [AC1953; H, c-Pr, H, Br, O, Cl, H, H, H, O], [AC1954; H, c-Pr, H, Br, O, Br, H, H, H, O], [AC 1 955; H, c-Pr, H, Br, O, I, H, H, H, O], [AC 1956; H, c-Pr, H, Br, O, Me, H, H, H, O], [AC 1957; H, c-Pr, H, Br, O, Et, H, H, H, O], [AC 1958; H, c-Pr, H, Br, O, Pr, H, H, H, O], [AC 1959; H, c-Pr, H, Br, O, i-Pr, H, H, H, O], [AC1960; H, c-Pr, H, Br, O, CH = CH 2, H, H, H, O], [AC1961; H, c-Pr, H, Br, O, C (CH 3) = CH 2, H, H, H, H, c-Pr, H, Br, O, C≡CH, H, H, H, O], [AC1963; H, c-Pr, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 1964; H, c-Pr, H, Br, O, c-Pr, H, H, H, O], [AC 1965; H, c-Pr, H, Br , O, OMe, H, H, H, O], [AC 1966; H, c-Pr, H, Br, O, OEt, H, H, H, O], [AC 1967; H, c-Pr, H , Br, O, Oi-Pr, H, H, H, O], [AC1968; H, c-Pr, H, Br, O, SMe, H, H, O], [AC1969; H, c -Pr, H, Br, O, SEt, H, H, H, O], [AC1970; H, c-Pr, H, Br, O, CH 2 F, H, H, H, O], [AC1971 ; H, c-Pr, H , Br, O, CHF 2, H, H, H, O], [AC1972; H, c-Pr, H, Br, O, CF 3, H, H, H, O ], [AC1973; H, c -Pr, H, Br, O, OCH 2 F, H, H, H, O], [AC1974; H, c-Pr, H, Br, O, OCHF 2, H, H, H, O], [ AC1975; H, c-Pr, H, Br, O, OCF 3, H, H, H, O], [AC1976; H, c-Pr , H, Br, O, SCH ₂ F, H, H, H, O], [AC 1977; H, c-Pr, H, Br, O, SCHF ₂ , H, H, H, O], [AC 1978; H, c-Pr, H, Br, O, SCF 3, H, H, H, O], [AC1979; H, c-Pr, H, Br, O, CN, H, H, H, O], [AC1980; H, c-Pr , H, Br, O, NO 2, H, H, H, O], [AC1981; H, F, H, H, O, H, H, H, H, O] [AC 1982; H, F, H, H, O, F, H, H, O], [AC 1983; H, F, H, H, O, Cl, H, H, H, O], [AC 1982; AC 1984; H, F, H, H, H, O, Br, H, H, O], [AC 1985; H, F, H, H, O, I, H, H, O], [AC 1986; H, F, H, H, H, O, Me, H, H, H, O], [AC 1987; H, F, H, H, O, Et, H, H, H, O], [AC 1988; H, H, F, H, H, H, O, Pr, H, H, H, O], [AC 1989; H, F, H, H, O, i-Pr, H, H, H, O], [AC 1990; H, F, H, H, O, CH = CH 2, H, H, H, O], [AC1991; H, F, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC 1992; H, F, H, H, O, C≡CH, H, H, H, O], [AC1993; H, F, H, H, O, C≡ CCH ₃ , H, H , H, O],

[AC 1994; H, F, H, H, H, O, c-Pr, H, H, H, O], [AC 1995; H, F, H, H, O, OMe, H, H, H, O], [AC1996; H, F, H, H, H, O, OEt, H, H, H, O], [AC 1997; H, F, H, H, O, Oi-Pr, H, H, H, O], [AC1998; H, F, H, H, H, O, SMe, H, H, H, O], [AC1999; H, F, H, H, O, SE t, H, H, H, O], [AC 2000 ; H, F, H, H , O, CH 2 F, H, H, H, O], [AC2001; H, F, H, H, O, CHF 2, H, H, H, O], [ AC 2002; H, F, H, H, H, O, CF ₃ , H, H, H, O], [AC 2003; H, F, H, H, O, OCH ₂ F, H, H, H, O], [AC2004; H, F, H , H, O, OCHF 2, H, H, H, O], [AC2005; H, F, H, H, O, OCF 3, H, H, H, O], [AC2006; H, F, H, H, H, O, SCH ₂ F, H, H, H, O], [AC 2007; H, F, H, H, O, SCHF ₂ , H, H, H, O] , [AC2008; H, F, H, H, O, SCF 3, H, H, H, O], [AC2009; H, F, H, H, O, CN, H, H, H, O], [AC2010; H, F, H , H, O, NO 2, H, H, H, O], [AC2011; H, F, H, Me, O, H, H, H, H, O], [ AC 2012; H, F, H, Me, O, F, H, H, O], [AC 2013; H, F, H, Me, O, Cl, H, H, H, O], [AC 2014; H, F, H, Me, O, Br, H, H, H, O], [AC2015; H, F, H, Me, O, I, H, H, O], [AC 2016; H, H, F, H, Me, O, Me, H, H, H, O], [AC 2017; H, F, H, Me, O, Et, H, H, H, O], [AC 2018; H, F, H, Me, O, Pr, H, H, H, O], [AC 2019; H, F, H, Me, O, i-Pr, H, H, H, O], [AC 2020; H, F, H, Me, O, CH = CH 2, H, H, H, O], [AC2021; H, F, H, Me, O, C (CH 3) = CH 2, H, H, H, O] , [AC 2022; H, F, H, Me, O, C, CH, H, H, H, O], [AC 2023; H, F, H, Me, O, C≡ CCH ₃ , H, H, H , O], [AC2024 H, F, H, Me, O, c, Pr, H, H, H, O], [AC 2025; H, F, H, Me, O, OM, H, H, H, O], [AC 2026 H, F, H, Me, O, OEt, H, H, H, O], [AC2027; H, F, H, Me, O, Oi-Pr, H, H, H, O], [AC2028 H, F, H, Me, O, SMe, H, H, H, O], [AC 2029; H, F, H, Me, O, SE t, H, H, O], [AC 2030; H , F, H, Me, O , CH 2 F, H, H, H, O], [AC2031; H, F, H, Me, O, CHF 2, H, H, H, O], [AC2032; H, F, H, Me, O, CF 3, H, H, H, O], [AC2033; H, F, H, Me, O, OCH 2 F, H, H, H, O], [AC2034 H, F, H, Me, O, OCHF ₂ , H, H, H, O], [AC 2035; H, F, H, Me, O, OCF ₃ , H, H, H, O], [AC 2036 H, F, H, Me, O, SCH ₂ F, H, H, H, O], [AC 2037; H, F, H, Me, O, SCHF ₂ , H, H, H, O], [[ AC2038; H, F, H, Me, O, SCF 3, H, H, H, O], [AC2039; H, F, H, Me, O, CN, H, H, H, O], [AC2040 H, F, H, Me, O, NO, NO ₂ , H, H, H, O], [AC 2041; H, F, H, Et, O, H, H, H, H, O], [AC 2042; H, F, H, Et, O, F, H, H, H, O], [AC 2043; H, F, H, Et, O, Cl, H, H, O], [AC 2044; H, F, H, Et, O, Br, H, H, H, O], [AC 2045; H, F, H, Et, O, I, H, H, O], [AC 2046; H, F, H, Et, O, Me, H, H, H, O, [AC 2047; H, F, H, Et, O, Et, H, H, H, O], [AC 2048; H, F, H, Et, O, Pr, H, H, H, O, [AC 2049; H, F, H, Et, O, i-Pr, H, H, H, O], [AC 2050; H, F, H, _{Et, O, CH = CH 2} , H, H, H, O], [AC2051; H, F, H, Et, O, C (CH 3) = CH 2, H, H, H, O], [ AC 2052; H, F, H, Et, O, C≡CH, H, H, H, O], [AC 2053; H, F, H, Et, O, C≡CCH ₃ , H, H, H, O, [AC2054; H, F, H, Et, O, c-Pr, H, H, H, O], [AC 2055; H, F, H, Et, O, OMe, H, H, H, O, [AC2056; H, F, H, Et, O, OEt, H, H, H, O], [AC 2057; H, F, H, Et, O, Oi-Pr, H, H, H, O, [AC2058; H, F, H, Et, O, SMe, H, H, H, O], [AC 2059; H, F, H, Et, O, SEt, H, H, H, O] , [AC2060; H, F, H, Et, O, CH 2 F, H, H, H, O], [AC2061; H, F, H, Et, O, CHF 2, H, H, H, O ], [AC2062; H, F , H, Et, O, CF 3, H, H, H, O], [AC2063; H, F, H, Et, O, OCH 2 F, H, H, H, O, [AC 2064; H, F, H, Et, O, OCHF ₂ , H, H, H, O], [AC 2065; H, F, H, Et, O, OCF ₃ , H, H, H, O, [AC 2066; H, F, H, Et, O, SCH ₂ F, H, H, H, O], [AC 2067; H, F, H, Et, O, SCHF ₂ , H, H, H , O], [AC 2068; H, F, H, Et, O, SCF ₃ , H, H, H, O], [AC 2069; H, F, H, Et, O, CN, H, H, H, H, O, [AC2070; H, F, H, Et, O, NO ₂ , H, H, O], [AC 2071; H, F, H, Pr, O, H, H, H, H, O H, F, H, Pr, O, F, H, H, O], [AC 2073; H, F, H, Pr, O, Cl, H, H, H, O], [AC 2074; H, F, H, Pr, O, Br, H, H, O], [AC 2075; H, F, H, Pr, O, I, H, H, O], [AC 2076 H, F, H, Pr, O, Me, H, H, H, O], [AC 2077; H, F, H, Pr, O, Et, H, H, H, O], [AC 2078; H , F, H, Pr, O, Pr, H, H, H, O], [AC 2079; H, F, H, Pr, O, i-Pr, H, H, H, O], [AC 2080; H , F, H, Pr, O , CH = CH 2, H, H, H, O], [AC2081; H, F, H, Pr, O, C (CH 3) = CH 2, H, H, H H, F, H, Pr, O, C≡CH, H, H, H, O], [AC 2083; H, F, H, Pr, O, C≡ CCH ₃ H, H, H, O], [AC 2084; H, F, H, Pr, O, c-Pr, H, H, H, O], [AC 2085; H, F, H, Pr, O, OMe, H, H, H, O], [AC 2086; H, F, H, Pr, O, OEt, H, H, H, O], [AC 2087; H, F, H, Pr, O, Oi- Pr, H, H, H, O], [AC 2088; H, F, H, Pr, O, SMe, H, H, H, O], [AC 2089; H, F, H, Pr, O, SE t, H, H, H, O], [AC 2090; H, F, H, Pr, O, CH ₂ F, H, H, H, O], [AC 2091; H, F, H, Pr, O, CHF ₂ , H, H, H, O ], [AC2092; H, F, H, Pr, O, CF 3, H, H, H, O], [AC2093; H, F, H, Pr, O, OCH 2 F, H, H, H, O],

[AC 2094; H, F, H, Pr, O, OCHF ₂ , H, H, H, O], [AC 2095; H, F, H, Pr, O, OCF ₃ , H, H, H, O], [AC 2096; H, F, H, Pr, O, SCH ₂ F, H, H, H, O], [AC 2097; H, F, H, Pr, O, SCHF ₂ , H, H, H, O] [AC 2098; H, F, H, Pr, O, SCF ₃ , H, H, H, O], [AC 2099; H, F, H, Pr, O, CN, H, H, H, O], [AC 2 100; H, F, H, Pr, O, NO ₂ , H, H, O], [AC 2101; H, F, H, i-Pr, O, H, H, H, H, O] , [AC2102; H, F, H, i-Pr, O, F, H, H, H, O], [AC 2103; H, F, H, i-Pr, O, Cl, H, H, H, O], [AC 2104; H, F, H, i-Pr, O, Br, H, H, O], [AC 2 105; H, F, H, i-Pr, O, I, H, H, H, O], [AC 2106; H, F, H, i-Pr, O, Me, H, H, H, O], [AC 2107; H, F, H, i-Pr, O, Et, H, H, H, O], [AC 2108; H, F, H, i-Pr, O, Pr, H, H, H, O], [AC 2109; H, F, H, i-Pr, O, i- Pr, H, H, H, O], [AC2110; H, F, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC2111; H, F, H, i _{-Pr, O, C (CH 3} ) = CH 2, H, H, H, O], [AC2112; H, F, H, i-Pr, O, C≡CH, H, H, H, O] [AC 2 113; H, F, H, i-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 2114; H, F, H, i-Pr, O, c-Pr, H H, H, O], [AC 2115; H, F, H, i-Pr, O, OMe, H, H, H, O], [AC 2116; H, F, H, i-Pr, O, OEt H, H, H, O], [AC 2117; H, F, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 2118; H, F, H, i-Pr , O, SMe, H, H, H, O], [AC 2119; H, F, H, i-Pr, O, SE t, H, H, H, O], [AC 2 120; H, F, H, i _{-Pr, O, CH 2 F,} H, H, H, O], [AC2121; H, F, H, i-Pr, O, CHF 2, H, H, H, O], [AC2122; H, F, H, i-Pr , O, CF ₃ , H, H, H, O], [AC 2 123; H, F, H, i-Pr, O, OCH ₂ F, H, H, O], [AC 2 124; H, F, H, i-Pr, O, OCHF 2, H, H, H, O], [AC2125; H, F, H, i-Pr, O, OCF 3, H, H, H, O], [AC2126; H, F, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 2127; H, F, H, i-Pr, O, SCHF ₂ , H, H, H, O H, F, H, i-Pr, O, SCF ₃ , H, H, H, O], [AC 2129; H, F, H, i-Pr, O, CN, H, H, H, O], [AC 2130; H, F, H, i-Pr, O, NO ₂ , H, H, H, O], [AC 2131; H, F, H, c-Pr, O, H, H , H, H, O], [AC2132; H, F, H, c-Pr, O, F, H, H, H, O], [AC 2133; H, F, H, c-Pr, O, Cl H, H, H, O], [AC 2 134; H, F, H, c-Pr, O, Br, H, H, H, O], [AC 2 135; H, F, H, c-Pr, O , I, H, H, H, O], [AC 2136; H, F, H, c-Pr, O, Me, H, H, H, O], [AC 2 137; H, F, H, c-Pr , O, Et, H, H, H, O], [AC 2138; H, F, H, c-Pr, O, Pr, H, H, H, O], [AC 2 139; H, F, H, c -Pr, O, i-Pr, H, H, H, O, [AC 2 140; H, F, H, c-Pr, O, CH = CH ₂ , H, H, H, O], [AC 2141; H, F, H, c- Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC2142; H, F, H, c-Pr, O, C≡CH, H , H, H, O], [AC2143; H, F, H, c-Pr, O, C≡CCH 3, H, H, H, O], [AC2144; H, F, H, c-Pr, O, c-Pr, H, H, H, O], [AC 2145; H, F, H, c-Pr, O, OMe, H, H, H, O], [AC 2146; H, F, H, c-Pr, O, OEt, H, H, H, O], [AC 2147; H, F, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 2 148; H, F, H, c-Pr, O, SMe, H, H, H, O], [AC 2149; H, F, H, c-Pr, O, SE t, H, H, H, O], [AC 2 150; H, F, H, c-Pr, O, C _{H 2 F, H, H,} H, O], [AC2151; H, F, H, c-Pr, O, CHF 2, H, H, H, O], [AC2152; H, F, H, c _{-Pr, O, CF 3, H} , H, H, O], [AC2153; H, F, H, c-Pr, O, OCH 2 F, H, H, H, O], [AC2154; H, F, H, c-Pr, O, OCHF 2, H, H, H, O], [AC2155; H, F, H, c-Pr, O, OCF 3, H, H, H, O], [ AC 2156; H, F, H, c-Pr, O, SCH ₂ F, H, H, H, O], [AC 2 157; H, F, H, c-Pr, O, SCHF ₂ , H, H, H , O], [AC2158; H , F, H, c-Pr, O, SCF 3, H, H, H, O], [AC2159; H, F, H, c-Pr, O, CN, H, H, H, O], [AC 2 160; H, F, H, c-Pr, O, NO ₂ , H, H, H, O], [AC 2161; H, F, H, S Me, O, H, H , H, H, O], [AC2162; H, F, H, SMe, O, F, H, H, H, O], [AC 2163; H, F, H, SMe, O, Cl, H, H , H, O], [AC2164; H, F, H, SMe, O, Br, H, H, H, O], [AC 2165; H, F, H, SMe, O, I, H, H, H H, F, H, SMe, O, Me, H, H, H, O], [AC 2 167; H, F, H, SMe, O, Et, H, H, H, O H, F, H, SMe, O, Pr, H, H, H, O], [AC 2169; H, F, H, SMe, O, i-Pr, H, H, H, O] ], [AC2170; H, F , H, SMe, O, CH = CH 2, H, H, H, O], [AC2171; H, F, H, SMe, O, C (CH 3) = CH 2 H, H, H, O], [AC2172; H, F, H, SMe, O, C≡CH, H, H, H, O], [AC 2173; H, F, H, SMe, O, C ≡ CCH ₃ , H, H, H, O], [AC 2174; H, F, H, SMe, O, c-Pr, H, H, H, O], [AC 2 175; H, F, H, SMe, O, OMe, H, H, H, O], [AC 2176; H, F, H, SMe, O, OEt, H, H, H, O], [AC 2177; H, F, H, SMe, O, Oi-Pr, H, H, H, O], [AC 2178; H, F, H, SMe, O, SMe, H, H, H, O], [AC 2 179; H, F, H, SMe, O, SEt, H, H, H, O], [AC2180; H, F, H, SMe, O, CH 2 F, H, H, H, O], [ AC2181; H, F, H, SMe, O, CHF 2, H, H, H, O], [AC2182; H, F, H, SMe, O, CF 3, H, H, H, O], [ AC 2 183; H, F, H, SMe, O, OCH ₂ F, H, H, H, O], [AC 2 184; H, F, H, SMe, O, OCHF ₂ , H, H, H, O], [AC2185; H, F, H , SMe, O, OCF 3, H, H, H, O], [AC2186; H, F, H, SMe, O, SCH 2 F, H, H, H, O] , [AC2187; H, F, H, SMe, O, SCHF 2, H, H, H, O], [AC2188; H, F, H, SMe, O, SCF 3, H, H, H, O] H, F, H, SMe, O, CN, H, H, H, O], [AC 2190; H, F, H, SMe, O, NO ₂ , H, H, H, O], [AC2191; H, F, H, OMe, O, H, H, H, H, O], [AC 2 192; H, F, H, OMe, O, F, H, H, H, O],

[AC2193; H, F, H, OMe, O, Cl, H, H, H, O], [AC 2194; H, F, H, OMe, O, Br, H, H, H, O], [AC 2195 H, F, H, OMe, O, I, H, H, H, O], [AC 2196; H, F, H, OMe, O, Me, H, H, H, O], [AC 2 197; H , F, H, OMe, O, Et, H, H, H, O], [AC 2198; H, F, H, OMe, O, Pr, H, H, H, O], [AC 2199; H, F , H, OMe, O, i-Pr, H, H, H, O], [AC 2200; H, F, H, OMe, O, CH = CH ₂ , H, H, H, O], [AC 2201; H, F, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC2202; H, F, H, OMe, O, C≡CH, H, H, H H, F, H, OMe, O, C≡CCH ₃ , H, H, H, O], [AC 2204; H, F, H, OMe, O, c-Pr, H, H, H, O], [AC 2205; H, F, H, OMe, O, OMe, H, H, H, O], [AC 2206; H, F, H, OMe, O, OE t, H, H, H, H, O], [AC2207; H, F, H, OMe, O, Oi-Pr, H, H, H, O], [AC 2208; H, F, H, OMe, O, SMe, H, H, H, H, O], [AC 2 209; H, F, H, OMe, O, SE t, H, H, H, O], [AC 2210; H, F, H, OMe, O, CH ₂ F, H, H, H, O], [AC2211; H, F, H, OMe, O, CHF 2, H, H, H, O], [AC2212; H, F, H, OMe, O, CF 3, H, H, H, O], [AC2213; H, F, H, OMe, O, OCH 2 F, H, H, H, O], [AC2214; H, F, H, OMe, O, OCHF 2, H, H , H, O], [AC2215 ; H, F, H, OMe, O, OCF 3, H, H, H, O], [AC2216; H, F, H, OMe, O, SCH 2 F, H, H, H, O], [AC2217; H, F, H, OMe, O, SCHF ₂ , H, H, H, O], [AC 2218; H, F, H, OMe, O, SCF ₃ , H, H, H, O], [AC2219; H, F, H, OMe, O, CN, H, H, H, O], [AC 2220; H, F, H, OMe, O, NO ₂ , H, H , H, O], [AC 2221; H, F, H, F, O, H, H, H, H, O], [AC2222; H, F, H, F, O, F, H, H, H, O], [AC2223; H, F, H, F, O, Cl, H, H, H, O], [AC2224; H, F, H, F, O, Br, H, H, O], [AC2225; H, F, H, F, O, I, H, H, H, H O], [AC2226; H, F, H, F, O, Me, H, H, H, O], [AC 2 227; H, F, H, F, O, Et, H, H, H, O] , [AC 2 228; H, F, H, F, O, Pr, H, H, H, O], [AC 2 229; H, F, H, F, O, i-Pr, H, H, H, O] , [AC2230; H, F, H, F, O, CH = CH 2, H, H, H, O], [AC2231; H, F, H, F, O, C (CH 3) = CH 2, H, H, H, O], [AC 2232; H, F, H, F, O, C≡CH, H, H, H, O], [AC 2233; H, F, H, F, O, C ≡ _{CCH 3, H, H, H} , O], [AC2234; H, F, H, F, O, c-Pr, H, H, H, O], [AC2235; H, F, H, F, O , OMe, H, H, H, O], [AC 2236; H, F, H, F, O, OEt, H, H, H, O], [AC 2237; H, F, H, F, O, Oi -Pr, H, H, H, O], [AC2238; H, F, H, F, O, SMe, H, H, H, O], [AC 2239; H, F, H, F, O, SEt H, H, H, O], [AC 2 240; H, F, H, F, O, CH ₂ F, H, H, H, O], [AC 2241; H, F, H, F, O, CHF _{2, H, H, H,} O], [AC2242; H, F, H, F, O, CF 3, H, H, H, O], [AC2243; H, F, H, F, O, OCH ₂ F, H, H, H, O], [AC 2244; H, F, H, F, O, OCHF ₂ , H, H, H, O], [AC 2 245; H, F, H, F, O, OCF ₃ , H, H, H, O], [AC 2246; H, F, H, F, O, SCH ₂ F, H, H, H, O], [AC 2247; H, F, H, F, O , SCHF ₂ , H, H, H, O], [AC 2248; H, F, H, F, O, SCF ₃ , H, H, H, O], [AC 2249; H, F, H, F, O , CN, H, H, H, O], [AC 2250; H, F, H, F, O, NO ₂ , H, H, H, O], [AC 2251; H, F, H, Cl, O, H, H, H, H, O], [AC 2252; H, F, H, Cl, O, F, H, H, H, O], [AC 2253; H, F, H, Cl, O, Cl, H, H, H, O], [AC 2 254; H, F, H, Cl, O, Br, H, H, H, O], [AC 2 255; H, F, H, Cl, O, I, H, H, H, O], [AC 2 256; H, F, H, Cl, O, Me, H, H, H, O], [AC 2 257; H, F, H, Cl, O, Et, H, H, H, O], [AC 2 258; H, F, H, Cl, O, Pr, H, H, H, O], [AC 2259; H, F, H, Cl, O, i-Pr, H, H, H, O], [AC 2 260; H, F, H, Cl, O, _{CH = CH 2, H, H} , H, O], [AC2261; H, F, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC2262; H, F, H, Cl, O, C≡CH, H, H, H, O], [AC 2263; H, F, H, Cl, O, C≡ CCH ₃ , H, H, H, O], [AC 2 264 H, F, H, Cl, O, c-Pr, H, H, H, O], [AC2265; H, F, H, Cl, O, OMe, H, H, H, O], [AC 2266 H, F, H, Cl, O, OEt, H, H, H, O], [AC 2267; H, F, H, Cl, O, Oi-Pr, H, H, H, O], [AC 2268 H, F, H, Cl, O, SMe, H, H, H, O], [AC 2269; H, F, H, Cl, O, SE t, H, H, O], [AC 2270; H , F, H, Cl, O , CH 2 F, H, H, H, O], [AC2271; H, F, H, Cl, O, CHF 2, H, H, H, O], [AC2272; H, F, H, Cl, O, CF 3, H, H, H, O], [AC2273; H, F, H, Cl, O, OCH 2 F, H, H, H, O], [AC2274 ; H, F, H, Cl , O, OCHF 2, H, H, H, O], [AC2275; H, F, H, Cl, O, OCF 3, H, H, H, O], [AC2276 H, F, H, Cl, O, SCH ₂ F, H, H, H, O], [AC 2277; H, F, H, Cl, O, SCHF ₂ , H, H, H, O], [[ AC 2 278; H, F, H, Cl, O, SCF ₃ , H, H, H, O], [AC 2279; H, F, H, Cl, O, CN, H, H, H, O], [AC 2 280 H, F, H, Cl, O, NO ₂ , H, H, H, O], [AC2281; H, F, H, Br, O, H, H, H, H, O], [A H, F, H, Br, O, F, H, H, O], [AC 2283; H, F, H, Br, O, Cl, H, H, H, O], [AC 2284; H, F, H, Br, O, Br, H, H, H, O], [AC 2285; H, F, H, Br, O, I, H, H, O], [AC 2286; H, F, H, Br, O, Me, H, H, H, O], [AC 2 287; H, F, H, Br, O, Et, H, H, H, O], [AC 2 288; H, F, H, Br, O, Pr, H, H, H, O], [AC 2289; H, F, H, Br, O, i-Pr, H, H, H, O], [AC 2290; H, F, H, Br, O, CH = CH 2, H, H, H, O], [AC2291; H, F, H, Br, O, C (CH 3) = CH 2, H, H, H, O] [AC 2 229; H, F, H, Br, O, C≡CH, H, H, H, O],

[AC 2 293; H, F, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 2 294; H, F, H, Br, O, c-Pr, H, H, H, O], [AC2295; H, F, H, Br, O, OMe, H, H, H, O], [AC 2296; H, F, H, Br, O, OEt, H, H, H, O] , [AC2 297; H, F, H, Br, O, Oi-Pr, H, H, H, O], [AC 2298; H, F, H, Br, O, SMe, H, H, H, O] , [AC 2 299; H, F, H, Br, O, SE t, H, H, H, O], [AC 2300; H, F, H, Br, O, CH ₂ F, H, H, H, O] , [AC2301; H, F, H, Br, O, CHF 2, H, H, H, O], [AC2302; H, F, H, Br, O, CF 3, H, H, H, O] , [AC2303; H, F, H, Br, O, OCH 2 F, H, H, H, O], [AC2304; H, F, H, Br, O, OCHF 2, H, H, H, O ], [AC2305; H, F , H, Br, O, OCF 3, H, H, H, O], [AC2306; H, F, H, Br, O, SCH 2 F, H, H, H, O], [AC 2307; H, F, H, Br, O, SCHF ₂ , H, H, H, O], [AC 2308; H, F, H, Br, O, SCF ₃ , H, H, H, O], [AC 2309; H, F, H, Br, O, CN, H, H, H, O], [AC 2310; H, F, H, Br, O, NO ₂ , H, H, H, O H, Cl, H, H, O, H, H, H, H, O], [AC 2312; H, Cl, H, H, O, F, H, H, H, O], [AC2313; H, Cl, H, H, O, Cl, H, H, O], [AC 2314; H, Cl, H, H, O, Br, H, H, H, O], [AC 2315 H, Cl, H, H, H, O, I, H, H, O, [AC2316; H, Cl, H, H, O, Me, H, H, O], [AC 2317; H , Cl, H, H, O, Et, H, H, H, O], [AC 2318; H, Cl, H, H, O, Pr, H, H, H, O], [AC 2319; H, Cl , H, H, O, i -Pr, H, H, H, O], [AC2320; H, Cl, H, H, O, CH = CH 2, H, H, H, O], [AC2321; H, Cl, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC2322; H, Cl, H, H, O, C≡CH , H, H, H, O], [AC 2323; H, Cl, H, H, O, C≡CCH ₃ , H, H, H, O], [AC 2324; H, Cl, H, H, O, c-Pr, H, H, H, O], [AC2325; H, Cl, H, H, O, OMe, H, H, H, O], [AC 2326; H, Cl, H, H, O, H, Cl, H, H, H, O, Oi-Pr, H, H, H, O], [AC2328; H, Cl, H, H, O, OEt, H, H, H, O], [AC2327; SMe, H, H, H, O], [AC 2329; H, Cl, H, H, O, SE, H, H, H, O], [AC 2330; H, Cl, H, H, O, CH ₂ F, H, H, H, O], [AC2331; H, Cl, H, H, O, CHF 2, H, H, H, O], [AC2332; H, Cl, H, H, O, CF _{3, H, H, H,} O], [AC2333; H, Cl, H, H, O, OCH 2 F, H, H, H, O], [AC2334; H, Cl, H, H, O, _{OCHF 2, H, H, H} , O], [AC2335; H, Cl, H, H, O, OCF 3, H, H, H, O], [AC2336; H, Cl, H, H, O, SCH ₂ F, H, H, H, O], [AC 2 337; H, Cl, H, H, O, SCHF ₂ , H, H, H, O], [AC 2 338; H, Cl, H, H, O , SCF ₃ , H, H, H, O], [AC 2339; H, Cl, H, H, O, CN, H, H, H, O], [AC 2 340; H, Cl, H, H, O, _{NO 2, H, H, H} , O], [AC2341; H, Cl, H, Me, O, H, H, H, H, O], [AC2342; H, Cl, H, Me, O, F H, H, H, O], [AC 2343; H, Cl, H, Me, O, Cl, H, H, H, O], [AC 2344; H, Cl, H, Me, O, Br, H H, H, O], [AC2345; H, Cl, H, Me, O, I, H, H, H, O], [AC 2346; H, Cl, H, Me, O, Me, H, H , H, O], [AC 2347; H, Cl, H, Me, O, Et, H, H, H, O], [AC 2348; H, Cl, H, Me, O, Pr, H, H, H H, Cl, H, Me, O, i-Pr, H, H, H, O], [AC 2 350; H, Cl, H, Me, O, CH = CH ₂ , H, H, H, O], [ AC2351; H, Cl, H, Me, O, C (CH 3) = CH 2, H, H, H, O], [AC2 H, Cl, H, Me, O, C≡CH, H, H, H, O], [AC 2 353; H, Cl, H, Me, O, C≡CCH ₃ , H, H, H, O H, Cl, H, Me, O, c-Pr, H, H, H, O], [AC 2 355; H, Cl, H, Me, O, OMe, H, H, H, O] ], [AC 2356; H, Cl, H, Me, O, OEt, H, H, H, O], [AC 2 357; H, Cl, H, Me, O, Oi-Pr, H, H, H, O H, Cl, H, Me, O, SMe, H, H, H, O], [AC 2359; H, Cl, H, Me, O, SE t, H, H, H, O], [AC 2 360; H, Cl, H, Me, O, CH ₂ F, H, H, H, O], [AC 2361; H, Cl, H, Me, O, CHF ₂ , H, H, H, O] , [AC2362; H, Cl, H, Me, O, CF 3, H, H, H, O], [AC2363; H, Cl, H, Me, O, OCH 2 F, H, H, H, O H, Cl, H, Me, O, OCHF ₂ , H, H, H, O], [AC 2365; H, Cl, H, Me, O, OCF ₃ , H, H, H, O] H, Cl, H, Me, O, SCH ₂ F, H, H, H, O], [AC 2367; H, Cl, H, Me, O, SCHF ₂ , H, H, H, O], [AC 2368; H, Cl, H, Me, O, SCF ₃ , H, H, H, O], [AC 2369; H, Cl, H, Me, O, CN, H, H, H, O ], [AC 2370; H, Cl, H, Me, O, NO ₂ , H, H, O], [AC 2371; H, Cl, H, Et, O, H, H, H, H, O] [AC 2372; H, Cl, H, Et, O, F, H, H, O], [AC 2373; H, Cl, H, Et, O, Cl, H, H, H, O], [AC 2373; AC 2 374; H, Cl, H, Et, O, Br, H, H, O], [AC 2 375; H, Cl, H, Et, O, I, H, H, H, O], [AC 2 376; H, Cl, H, Et, O, Me, H, H, H, O], [AC2 377; H, Cl, H, Et, O, Et, H, H, H, O], [AC 2378; H, Cl, H, Et, O, Pr, H, H, H, O], [AC 2379; H, Cl, H, Et, O, i-Pr, H, H, H, O], [AC 2 380; H, Cl, H, Et, O, CH = CH 2, H, H, H, O], [AC2381; H, Cl, H, Et, O, C (CH 3) = CH 2, H, H, H, O], [AC2382; H, Cl, H, Et, O, C≡CH, H, H, H H, Cl, H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 2384; H, Cl, H, Et, O, c-Pr, H, H, H, O], [AC2385; H, Cl, H, Et, O, OMe, H, H, H, O], [AC 2386; H, Cl, H, Et, O, OEt, H, H, H, O], [AC 2387; H, Cl, H, Et, O, Oi-Pr, H, H, H, O], [AC 2388; H, Cl, H, Et, O, SMe, H, H, H, O], [AC 2 389; H, Cl, H, Et, O, SE t, H, H, H, O], [AC 2 390; H, Cl, H, Et, O, CH ₂ F, H, H, H, O], [AC2391; H, Cl, H, Et, O, CHF 2, H, H, H, O], [AC2392; H, Cl, H, Et, O, CF 3, H, H, H, O],

[AC2393; H, Cl, H , Et, O, OCH 2 F, H, H, H, O], [AC2394; H, Cl, H, Et, O, OCHF 2, H, H, H, O] , [AC2395; H, Cl, H, Et, O, OCF 3, H, H, H, O], [AC2396; H, Cl, H, Et, O, SCH 2 F, H, H, H, O H, Cl, H, Et, O, SCHF ₂ , H, H, H, O], [AC 2398; H, Cl, H, Et, O, SCF ₃ , H, H, H, O] ], [AC2399; H, Cl , H, Et, O, CN, H, H, H, O], [AC2400; H, Cl, H, Et, O, NO 2, H, H, H, O] , [AC 2401; H, Cl, H, Pr, O, H, H, H, O], [AC 2402; H, Cl, H, Pr, O, F, H, H, H, O], [AC 2402; AC2403; H, Cl, H, Pr, O, Cl, H, H, O], [AC 2404; H, Cl, H, Pr, O, Br, H, H, H, O], [AC 2405; H, Cl, H, Pr, O, I, H, H, H, O], [AC 2406; H, Cl, H, Pr, O, Me, H, H, O], [AC 2407; H, Cl, H, Pr, O, Et, H, H, H, O], [AC 2408; H, Cl, H, Pr, O, Pr, H, H, H, O], [AC 2 409; H, Cl, H, Pr, O, i- Pr, H, H, H, O], [AC2410; H, Cl, H, Pr, O, CH = CH 2, H, H, H, O], [AC2411; H , Cl, H, Pr, O , C (CH 3) = CH 2, H, H, H, O], [AC2412; H, Cl, H, Pr, O, C≡CH, H, H, H, H, Cl, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 2414; H, Cl, H, Pr, O, c-Pr, H, H , H, O], [AC 2415; H, Cl, H, Pr, O, OMe, H, H, H, O], [AC 2416; H, Cl, H, Pr, O, OEt, H, H, H H, Cl, H, Pr, O, Oi-Pr, H, H, H, O], [AC 2418; H, Cl, H, Pr, O, SMe, H, H, H] H, Cl, H, Pr, O, SEt, H, H, H, O], [AC 2420; H, Cl, H, Pr, O, CH ₂ F, H, H, H , O], [AC2421; H, Cl, H, Pr, O, CHF ₂ , H, H, H, O], [AC2422; H, Cl, H, Pr, O, CF 3, H, H, H, O], [AC2423; H, Cl, H, Pr, O, OCH 2 F, H, H , H, O], [AC2424 ; H, Cl, H, Pr, O, OCHF 2, H, H, H, O], [AC2425; H, Cl, H, Pr, O, OCF 3, H, H , H, O], [AC 2426; H, Cl, H, Pr, O, SCH ₂ F, H, H, H, O], [AC 2427; H, Cl, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 2428; H, Cl, H, Pr, O, SCF ₃ , H, H, H, O], [AC 2429; H, Cl, H, Pr, O, CN, H, H , H, O], [AC 2430; H, Cl, H, Pr, O, NO ₂ , H, H, H, O], [AC 2431; H, Cl, H, i-Pr, O, H, H, H, H, O], [AC 2432; H, Cl, H, i-Pr, O, F, H, H, H, O], [AC 2433; H, Cl, H, i-Pr, O, Cl, H, H, H, O], [AC2434; H, Cl, H, i-Pr, O, Br, H, H, H, O], [AC 2435; H, Cl, H, i-Pr, O, H, Cl, H, i-Pr, O, Me, H, H, H, O], [AC 2437; H, Cl, H, i-Pr, I, H, H, H, O], [AC2436; O, Et, H, H, H, O], [AC2438; H, Cl, H, i-Pr, O, Pr, H, H, H, O], [AC2439; H, Cl, H, i- Pr, O, i-Pr, H, H, H, O], [AC2440; H, Cl, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC2441; H , Cl, H, i-Pr , O, C (CH 3) = CH 2, H, H, H, O], [AC2442; H, Cl, H, i-Pr, O, C≡CH, H, H, H, O], [AC2443; H, Cl, H, i-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 2444; H, Cl, H, i-Pr, O , c-Pr, H, H, H, O], [AC 2445; H, Cl, H, i-Pr, O, OMe, H, H, H, O], [AC 2446; H, Cl, H, i -Pr, O, OEt, H, H, H, O], [AC2447; H, Cl, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 2448; H, Cl , H, i-Pr, O, SMe, H, H, H, O], [AC2449; H, Cl, H, i-Pr, O, SE t, H, H, H, O], [AC2450; H, Cl, H, i-Pr, O, CH 2 F, H, H, H, O], [AC2451; H, Cl, H, i- _{Pr, O, CHF 2, H} , H, H, O], [AC2452; H, Cl, H, i-Pr, O, CF 3, H, H, H, O], [AC2453; H, Cl, H, i-Pr, O, OCH 2 F, H, H, H, O], [AC2454; H, Cl, H, i-Pr, O, OCHF 2, H, H, H, O], [AC2455 ; H, Cl, H, i -Pr, O, OCF 3, H, H, H, O], [AC2456; H, Cl, H, i-Pr, O, SCH 2 F, H, H, H, H, Cl, H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 2458; H, Cl, H, i-Pr, O, SCF ₃ , H, O], [AC 2 457; H, H, O], [AC 2459; H, Cl, H, i-Pr, O, CN, H, H, H, O], [AC 2460; H, Cl, H, i-Pr, O, NO ₂ H, H, H, O], [AC2461; H, Cl, H, c-Pr, O, H, H, H, H, O], [AC 2462; H, Cl, H, c-Pr, O , F, H, H, H, O], [AC2463; H, Cl, H, c-Pr, O, Cl, H, H, H, O], [AC 2464; H, Cl, H, c-Pr , O, Br, H, H, H, O], [AC 2465; H, Cl, H, c-Pr, O, I, H, H, H, O], [AC 2466; H, Cl, H, c -Pr, O, Me, H, H, H, O, [AC2467; H, Cl, H, c-Pr, O, Et, H, H, H, O], [AC 2468; H, Cl, H , c-Pr, O, Pr, H, H, H, O, [AC 2469; H, Cl, H, c-Pr, O, i-Pr, H, H, H, O], [AC 2 470; H , Cl, H, c-Pr , O, CH = CH 2, H, H, H, O], [AC2471; H, Cl, H, c-Pr, O, C (CH 3) = CH 2, H , H, H, O], [AC2472; H, Cl, H, c-Pr, O, C≡CH, H, H, H, O], [AC 2473; H, Cl, H, c-Pr, O , C≡CCH ₃ , H, H, H, O], [AC 2474; H, Cl, H, c-Pr, O, c-Pr, H, H, H, O], [AC 2475; H, Cl, H, c-Pr, O, OMe, H, H, H, O], [AC 2476; H, Cl, H, c-Pr, O, OEt, H, H, H H, Cl, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 2478; H, Cl, H, c-Pr, O, SMe, H H, H, O], [AC2479; H, Cl, H, c-Pr, O, SEt, H, H, H, O], [AC 2480; H, Cl, H, c-Pr, O, CH _{2 F, H, H, H} , O], [AC2481; H, Cl, H, c-Pr, O, CHF 2, H, H, H, O], [AC2482; H, Cl, H, c- _{Pr, O, CF 3, H} , H, H, O], [AC2483; H, Cl, H, c-Pr, O, OCH 2 F, H, H, H, O], [AC2484; H, Cl , H, c-Pr, O , OCHF 2, H, H, H, O], [AC2485; H, Cl, H, c-Pr, O, OCF 3, H, H, H, O], [AC2486 H, Cl, H, c-Pr, O, SCH ₂ F, H, H, H, O], [AC 2487; H, Cl, H, c-Pr, O, SCHF ₂ , H, H, H, H O], [AC2488; H, Cl, H, c-Pr, O, SCF 3, H, H, H, O], [AC2489; H, Cl, H, c-Pr, O, CN, H, H , H, O], [AC2490 ; H, Cl, H, c-Pr, O, NO 2, H, H, H, O], [AC2491; H, Cl, H, SMe, O, H, H, H, H, O],

[AC2492; H, Cl, H, SMe, O, F, H, H, H, O], [AC2493; H, Cl, H, SMe, O, Cl, H, H, H, O], [AC 2494 H, Cl, H, SMe, O, Br, H, H, O], [AC2495; H, Cl, H, SMe, O, I, H, H, H, O], [AC 2496; H , Cl, H, SMe, O, Me, H, H, H, O], [AC2497; H, Cl, H, SMe, O, Et, H, H, H, O], [AC 2498; H, Cl , H, SMe, O, Pr, H, H, H, O], [AC 2499; H, Cl, H, SMe, O, i-Pr, H, H, H, O], [AC 2500; H, Cl , H, SMe, O, CH = CH 2, H, H, H, O], [AC2501; H, Cl, H, SMe, O, C (CH 3) = CH 2, H, H, H, O H, Cl, H, SMe, O, C≡CH, H, H, H, O], [AC 2503; H, Cl, H, SMe, O, C≡CCH ₃ , H, H, H] H, O], [AC 2504; H, Cl, H, SMe, O, c-Pr, H, H, H, O], [AC 2505; H, Cl, H, SMe, O, OMe, H, H, H H, O], [AC 2506; H, Cl, H, SMe, O, OEt, H, H, H, O], [AC 2507; H, Cl, H, SMe, O, Oi-Pr, H, H, H, H, O], [AC2508; H, Cl, H, SMe, O, SMe, H, H, H, O], [AC 2509; H, Cl, H, SMe, O, SEt, H, H, H, H, O], [AC2510; H, Cl, H, SMe, O, CH 2 F, H, H, H, O], [AC2511; H, Cl, H, SMe, O, CHF 2, H, H, H , O], [AC2512; H , Cl, H, SMe, O, CF 3, H, H, H, O], [AC2513; H, Cl, H, SMe, O, OCH 2 F, H, H, H, O], [AC 2514; H, Cl, H, SMe, O, OCHF ₂ , H, H, H, O], [AC 2515; H, Cl, H, SMe, O, OCF ₃ , H, H, H H, O], [AC 2516; H, Cl, H, SMe, O, SCH ₂ F, H, H, H, O], [AC 2517; H, Cl, H, SMe, O, SCHF ₂ , H, H , H, O], [AC2518 ; H, Cl, H, SMe, O, SCF 3, H, H, H, O], [AC2519; H, Cl, H, SMe, O, CN, H, H, H, O ], [AC 2520; H, Cl, H, SMe, O, NO ₂ , H, H, O], [AC 2521; H, Cl, H, OMe, O, H, H, H, H, O] , [AC2522; H, Cl, H, OMe, O, F, H, H, H, O], [AC 2523; H, Cl, H, OMe, O, Cl, H, H, H, O], [, AC2524; H, Cl, H, OMe, O, Br, H, H, O], [AC2525; H, Cl, H, OMe, O, I, H, H, H, O], [AC2526; H, Cl, H, OMe, O, Me, H, H, H, O], [AC 2527; H, Cl, H, OMe, O, Et, H, H, H, O], [AC 2528; H, Cl, H, OMe, O, Pr, H, H, H, O], [AC 2529; H, Cl, H, OMe, O, i-Pr, H, H, H, O], [AC 2530; H, Cl, H, OMe, O, CH = CH 2, H, H, H, O], [AC2531; H, Cl, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC 2532; H, Cl, H, OMe, O, C≡CH, H, H, H, O], [AC 2533; H, Cl, H, OMe, O, C≡ CCH ₃ , H, H , H, O], [AC 2534; H, Cl, H, OMe, O, c-Pr, H, H, H, O], [AC 2535; H, Cl, H, OMe, O, OMe, H, H , H, O], [AC 2536; H, Cl, H, OMe, O, OEt, H, H, H, O], [AC 2537; H, Cl, H, OMe, O, Oi-Pr, H, H , H, O], [AC2538; H, Cl, H, OMe, O, SMe, H, H, H, O], [AC 2539; H, Cl, H, OMe, O, SEt, H, H, H , O], [AC2540; H , Cl, H, OMe, O, CH 2 F, H, H, H, O], [AC2541; H, Cl, H, OMe, O, CHF 2, H, H, H, O], [AC2542; H, Cl, H, OMe, O, CF 3, H, H, H, O], [AC2543; H, Cl, H, OMe, O, OCH 2 F, H, H , H, O], [AC2544 ; H, Cl, H, OMe, O, OCHF 2, H, H, H, O], [AC2545; H, Cl, H, OMe, O, OCF 3, H, H , H, O], [AC 2546; H, Cl, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 2547; H, Cl, H, OMe, O, SCHF ₂ , H, H, H, O ], [AC2548; H, Cl , H, OMe, O, SCF 3, H, H, H, O], [AC2549; H, Cl, H, OMe, O, CN, H, H, H, O] [AC 2550; H, Cl, H, OMe, O, NO ₂ , H ₂ , H, O], [AC 2551; H, Cl, H, F, O, H, H, H, H, O], [AC2552; H, Cl, H, F, O, F, H, H, O], [AC 2553; H, Cl, H, F, O, Cl, H, H, H, O], [AC 2554 H, Cl, H, F, O, Br, H, H, O], [AC 2 555; H, Cl, H, F, O, I, H, H, H, O], [AC 2 556; H , Cl, H, F, O, Me, H, H, H, O], [AC 2557; H, Cl, H, F, O, Et, H, H, H, O], [AC 2 558; H, Cl , H, F, O, Pr, H, H, H, O], [AC 2559; H, Cl, H, F, O, i-Pr, H, H, H, O], [AC 2560; H, Cl , H, F, O, CH = CH 2, H, H, H, O], [AC2561; H, Cl, H, F, O, C (CH 3) = CH 2, H, H, H, O H, Cl, H, F, O, C≡CH, H, H, H, O], [AC 2563; H, Cl, H, F, O, C≡ CCH ₃ , H, H, H, O], [AC 2564; H, Cl, H, F, O, c-Pr, H, H, H, O], [AC 2565; H, Cl, H, F, O, OMe, H, H, H, O], [AC 2566; H, Cl, H, F, O, OEt, H, H, H, O], [AC 2 567; H, Cl, H, F, O, Oi-Pr, H, H, H, O], [AC2568; H, Cl, H, F, O, SMe, H, H, H, O], [AC 2569; H, Cl, H, F, O, SE t, H, H, H, O], [AC 2570; H, Cl, H, F, O, CH ₂ F, H, H, H, O], [AC 2571; H, Cl, H, F, O, CHF ₂ , H, H, H , O], [AC2572; H , Cl, H, F, O, CF 3, H, H, H, O], [AC2573; H, Cl, H, F, O, OCH 2 F, H, H, H, O], [AC 2574; H, Cl, H, F, O, OCHF ₂ , H, H, H, O], [AC 2575; H, Cl, H, F, O, OCF ₃ , H, H, H, O], [AC 2576; H, Cl, H, F, O, SCH ₂ F, H, H, H, O], [AC 2577; H, Cl, H, F, O _{, SCHF 2, H, H,} H, O], [AC2578; H, Cl, H, F, O, SCF 3, H, H, H, O], [AC2579; H, Cl, H, F, O , CN, H, H, H, O], [AC 2580; H, Cl, H, F, O, NO ₂ , H, H, H, O], [AC 2581; H, Cl, H, Cl, O, H, H, H, H, O], [AC 2582; H, Cl, H, Cl, O, F, H, H, H, O], [AC 2583; H, Cl, H, Cl, O, Cl, H, H, H, O], [AC 2584; H, Cl, H, Cl, O, Br, H, H, H, O], [AC 2585; H, Cl, H, Cl, O, I, H, H, H, O], [AC2586; H, Cl, H, Cl, O, Me, H, H, H, O], [AC2587; H, Cl, H, Cl, O, Et, H, H, H, H, O], [AC2588; H, Cl, H, Cl, O, Pr, H, H, H, O], [AC 2589; H, Cl, H, Cl, O, i-Pr, H, H, H, O], [AC2590; H, Cl, H, Cl, O, CH = CH 2, H, H, H, O], [AC2591; H, Cl, H, Cl, O, C (CH 3) = CH ₂ , H, H, H, O],

[AC 2592; H, Cl, H, Cl, O, C≡CH, H, H, H, O], [AC 2593; H, Cl, H, Cl, O, C≡ CCH ₃ , H, H, H, O], [AC2594; H, Cl, H, Cl, O, c-Pr, H, H, H, O], [AC 2595; H, Cl, H, Cl, O, OMe, H, H, H, O, [AC 2596; H, Cl, H, Cl, O, OEt, H, H, H, O], [AC 2597; H, Cl, H, Cl, O, Oi-Pr, H, H, H, O, [AC2598; H, Cl, H, Cl, O, SMe, H, H, H, O], [AC 2599; H, Cl, H, Cl, O, SEt, H, H, H, O] , [AC2600; H, Cl, H, Cl, O, CH 2 F, H, H, H, O], [AC2601; H, Cl, H, Cl, O, CHF 2, H, H, H, O ], [AC2602; H, Cl , H, Cl, O, CF 3, H, H, H, O], [AC2603; H, Cl, H, Cl, O, OCH 2 F, H, H, H, O], [AC2604; H, Cl, H, Cl, O, OCHF 2, H, H, H, O], [AC2605; H, Cl, H, Cl, O, OCF 3, H, H, H, O], [AC 2606; H, Cl, H, Cl, O, SCH ₂ F, H, H, H, O], [AC 2607; H, Cl, H, Cl, O, SCHF ₂ , H, H, H , O], [AC2608; H , Cl, H, Cl, O, SCF 3, H, H, H, O], [AC2609; H, Cl, H, Cl, O, CN, H, H, H, O], [AC 2610; H, Cl, H, Cl, O, NO ₂ , H ₂ , H, H, O], [AC 2611; H, Cl, H, Br, O, H, H, H, H, O H, Cl, H, Br, O, F, H, H, O], [AC 2613; H, Cl, H, Br, O, Cl, H, H, H, O], [AC2614; H, Cl, H, Br, O, Br, H, H, O], [AC 2615; H, Cl, H, Br, O, I, H, H, H, O], [AC 2616 H, Cl, H, Br, O, Me, H, H, H, O], [AC2617; H, Cl, H, Br, O, Et, H, H, H, O], [AC 2618; H , Cl, H, Br, O, Pr, H, H, H, O], [AC 2619; H, Cl, H, Br, O, i-Pr, H, H, H, O], [AC 2620; H , Cl, H, Br, O, CH = CH ₂ , H, H, H, O], [AC 2 621; H, Cl, H, Br, O, C (CH 3) = CH 2, H, H, H, O], [AC2622; H, Cl, H, Br, O, C≡CH, H, H , H, O], [AC 2623; H, Cl, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 2624; H, Cl, H, Br, O, c-Pr, H, H, H, O], [AC 2625; H, Cl, H, Br, O, OMe, H, H, H, O], [AC 2626; H, Cl, H, Br, O, OE t, H, H, H, O], [AC2627; H, Cl, H, Br, O, Oi-Pr, H, H, H, O], [AC2628; H, Cl, H, Br, O, SMe, H, H, H, O], [AC 2629; H, Cl, H, Br, O, SE t, H, H, H, O], [AC 2630; H, Cl, H, Br, O, CH ₂ F, H, H, H, O], [ AC2631; H, Cl, H, Br, O, CHF 2, H, H, H, O], [AC2632; H, Cl, H, Br, O, CF 3, H, H, H, O], [ AC2633; H, Cl, H, Br, O, OCH 2 F, H, H, H, O], [AC2634; H, Cl, H, Br, O, OCHF 2, H , H, H, O], [AC2635; H, Cl, H, Br, O, OCF 3, H, H, H, O], [AC2636; H, Cl, H, Br, O, SCH 2 F, H, H, H, O], [AC 2637; H, Cl, H, Br, O, SCHF ₂ , H, H, H, O], [AC 2638; H, Cl, H, Br, O, SCF ₃ , H, H, H, O], [AC 2639; H, Cl, H, Br, O, CN, H, H, H, O], [AC 2640; H, Cl, H, Br, O, NO ₂ , H H, H, O], [AC2641; H, Br, H, H, O, H, H, H, H, O], [AC2642; H, Br, H, H, O, F, H, H , H, O], [AC 2643; H, Br, H, H, O, Cl, H, H, O], [AC 2 644; H, Br, H, H, O, Br, H, H, H H, Br, H, H, O, I, H, H, H, O], [AC 2646; H, Br, H, H, O, Me, H, H, H, O H, Br, H, H, O, Et, H, H, H, O], [AC 2648; H, Br, H, H, O, Pr, H, H, H, O], [AC2649; H, Br, H, H, O, i-Pr, H, H, H, O], [AC 2650; H, B r, H, H, O, CH = CH 2, H, H, H, O], [AC2651; H, Br, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC2652; H, Br, H, H, O, C≡CH, H, H, H, O], [AC2653; H, Br, H, H, O, C≡ CCH ₃ , H, H , H, O], [AC2654; H, Br, H, H, O, c-Pr, H, H, H, O], [AC 2655; H, Br, H, H, O, OMe, H, H , H, O], [AC 2656; H, Br, H, H, O, OEt, H, H, H, O], [AC 2657; H, Br, H, H, O, Oi-Pr, H, H H, O], [AC 2658; H, Br, H, H, O, SMe, H, H, H, O], [AC 2659; H, Br, H, H, O, SEt, H, H, H , O], [AC2660; H , Br, H, H, O, CH 2 F, H, H, H, O], [AC2661; H, Br, H, H, O, CHF 2, H, H, H, O], [AC2662; H, Br, H, H, O, CF 3, H, H, H, O], [AC2663; H, Br, H, H, O, OCH 2 F, H, H , H, O], [AC 2664; H, Br, H, H, O, OCHF ₂ , H, H, H, O], [AC 2 665; H, Br, H, H, O, OCF ₃ , H, H H, O], [AC 2 666; H, Br, H, H, O, SCH ₂ F, H, H, H, O], [AC 2 667; H, Br, H, H, O, SCHF ₂ , H, H, H, O], [AC 2668; H, Br, H, H, O, SCF ₃ , H, H, H, O], [AC 2 669; H, Br, H, H, O, CN, H, H , H, O], [AC 2 670; H, Br, H, H, O, NO ₂ , H, H, H, O], [AC 2671; H, Br, H, Me, O, H, H, H, H, H, O], [AC 2672; H, Br, H, Me, O, F, H, H, O], [AC 2673; H, Br, H, Me, O, Cl, H, H, H, H, O], [AC 2674; H, Br, H, Me, O, Br, H, H, O], [AC 2 675; H, Br, H, Me, O, I, H, H, H, O] , [AC 2 676; H, Br, H, Me, O, Me, H, H, H, O], [AC 2677; H, Br, H, Me, O, Et, H, H, H, O], [ AC 2678; H, Br, H, Me, O, Pr, H, H, H, O], [AC 2679; H, Br, H, Me, O, i-Pr, H , H, H, O], [AC 2 680; H, Br, H, Me, O, CH = CH ₂ , H, H, H, O], [AC2681; H, Br, H, Me, O, C ( _{CH 3) = CH 2, H} , H, H, O], [AC2682; H, Br, H, Me, O, C≡CH, H, H, H, O], [AC2683; H, Br, H , Me, O, C≡CCH ₃ , H, H, H, O], [AC 2684; H, Br, H, Me, O, c-Pr, H, H, H, O], [AC 2685; H, Br, H, Me, O, OMe, H, H, H, O], [AC 2 686; H, Br, H, Me, O, OEt, H, H, H, O], [AC 2687; H, Br, H, Me, O, Oi-Pr, H, H, H, O], [AC 2688; H, Br, H, Me, O, SMe, H, H, H, O], [AC 2689; H, Br, H, Me, O, SEt, H, H, H, O], [AC2690; H, Br, H, Me, O, CH 2 F, H, H, H, O], [AC2691; H, Br, _{H, Me, O, CHF 2} , H, H, H, O],

[AC2692; H, Br, H , Me, O, CF 3, H, H, H, O], [AC2693; H, Br, H, Me, O, OCH 2 F, H, H, H, O] , [AC 2694; H, Br, H, Me, O, OCHF ₂ , H, H, H, O], [AC 2695; H, Br, H, Me, O, OCF ₃ , H, H, H, O] H, Br, H, Me, O, SCH ₂ F, H, H, H, O], [AC 2697; H, Br, H, Me, O, SCHF ₂ , H, H, H, O H, Br, H, Me, O, SCF ₃ , H, H, H, O], [AC 2699; H, Br, H, Me, O, CN, H, H, H, O] [AC 2700; H, Br, H, Me, O, NO ₂ , H, H, O], [AC 2701; H, Br, H, Et, O, H, H, H, H, O], [AC 2702; H, Br, H, Et, O, F, H, H, O], [AC 2703; H, Br, H, Et, O, Cl, H, H, H, O], [AC 2704 H, Br, H, Et, O, Br, H, H, H], [AC 2 705; H, Br, H, Et, O, I, H, H, H, O], [AC 2706; H , Br, H, Et, O, Me, H, H, H, O], [AC 2707; H, Br, H, Et, O, Et, H, H, H, O], [AC 2 708; H, Br , H, Et, O, Pr, H, H, H, O], [AC 2709; H, Br, H, Et, O, i-Pr, H, H, H, O], [AC 2710; H, Br , H, Et, O, CH = CH 2, H, H, H, O], [AC2711; H, Br, H, Et, O, C (CH 3) = CH 2, H, H, H, O H, Br, H, Et, O, C≡CH, H, H, H, O], [AC 2713; H, Br, H, Et, O, C≡CCH ₃ , H, H, H] H, O], [AC 2714; H, Br, H, Et, O, c-Pr, H, H, H, O], [AC 2715; H, Br, H, Et, O, OMe, H, H, H, O], [AC 2716; H, Br, H, Et, O, OEt, H, H, H, O], [AC 2717; H, Br, H, Et, O, Oi-Pr, H, H, H, O], [AC 2718; H, Br, H, Et, O, SMe, H, H, H, O], [AC 2719; H, Br, H, Et, O, SE t, H, H, H, O], [AC 2720; H, Br, H, Et, O, CH ₂ F, H, H, H , O], [AC2721; H , Br, H, Et, O, CHF 2, H, H, H, O], [AC2722; H, Br, H, Et, O, CF 3, H, H, H , O], [AC2723; H , Br, H, Et, O, OCH 2 F, H, H, H, O], [AC2724; H, Br, H, Et, O, OCHF 2, H, H, H, O], [AC2725; H, Br, H, Et, O, OCF 3, H, H, H, O], [AC2726; H, Br, H, Et, O, SCH 2 F, H, H H, O], [AC 2 727; H, Br, H, Et, O, SCHF ₂ , H, H, H, O], [AC 2 728; H, Br, H, Et, O, SCF ₃ , H, H H, O], [AC 2729; H, Br, H, Et, O, CN, H, H, H, O], [AC 2730; H, Br, H, Et, O, NO ₂ , H, H, H, O], [AC 2731; H, Br, H, Pr, O, H, H, H, O], [AC 2732; H, Br, H, Pr, O, F, H, H, H, H, O], [AC2733; H, Br, H, Pr, O, Cl, H, H, O], [AC 2734; H, Br, H, Pr, O, Br, H, H, H, O] , [AC 2 735; H, Br, H, Pr, O, I, H, H, O], [AC 2 736; H, Br, H, Pr, O, Me, H, H, H, O], [AC 2 736 AC 2 737; H, Br, H, Pr, O, Et, H, H, O], [AC 2738; H, Br, H, Pr, O, Pr, H, H, H, O], [AC 2739; H, Br, H, Pr, O, i-Pr, H, H, H, O], [AC2740; H, Br, H, Pr, O, CH = CH 2, H, H, H, O], [AC2741; H, Br, H , Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC2742; H, Br, H, Pr, O, C≡CH, H, H, H, O], [AC 2743; H, Br, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 2744; H, Br, H, Pr, O, c-Pr H, H, H, O], [AC 2745; H, Br, H, Pr, O, OMe, H, H, H, O], [AC 2746; H, Br, H, Pr, O, OEt, H H, H, O], [AC 2 747; H, Br, H, Pr, O, Oi-Pr, H, H, H, O], [AC 2 748; H, Br, H, Pr, O, SMe, H , H, H, O], [AC 2749; H, Br, H, Pr, O, SEt, H , H, H, O], [AC2750; H, Br, H, Pr, O, CH 2 F, H, H, H, O], [AC2751; H, Br, H, Pr, O, CHF 2, H, H, H, O] , [AC2752; H, Br, H, Pr, O, CF 3, H, H, H, O], [AC2753; H, Br, H, Pr, O, OCH 2 F H, H, H, O], [AC 2754; H, Br, H, Pr, O, OCHF ₂ , H, H, H, O], [AC 2755; H, Br, H, Pr, O, OCF ₃ H, H, H, O], [AC 2756; H, Br, H, Pr, O, SCH ₂ F, H, H, H, O], [AC 2757; H, Br, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 2758; H, Br, H, Pr, O, SCF ₃ , H, H, H, O], [AC 2759; H, Br, H, Pr, O, CN , H, H, H, O ], [AC2760; H, Br, H, Pr, O, NO 2, H, H, H, O], [AC2761; H, Br, H, i-Pr, O, H, H, H, H, O], [AC2762; H, Br, H, i-Pr, O, F, H, H, H] O, [AC2763; H, Br, H, i-Pr, O, Cl, H, H, H, O], [AC 2764; H, Br, H, i-Pr, O, Br, H, H, H, O], [AC 2 765; H, Br, H, i- Pr, O, I, H, H, H, O], [AC 2 766; H, Br, H, i-Pr, O, Me, H, H, H, O], [AC 2 767; H, Br, H, i-Pr, O, Et, H, H, H, O], [AC 2768; H, Br, H, i-Pr, O, Pr, H, H, H, O], [AC 2769; H, Br, H, i-Pr, O, i-Pr, H, H, H, O], [AC2770; H, Br, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC2771; H, Br, H , i-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC2772; H, Br, H, i-Pr, O, C≡ CH, H, H, H, O], [AC2773; H, Br, H, i-Pr, O, C≡CCH 3, H, H, H, O], [AC2774; H, Br, H, i -Pr, O, c-Pr, H, H, H, O], [AC 2775; H, Br, H, i-Pr, O, OMe, H, H, H, O], [AC 2776; H, Br , H, i-Pr, O, OEt, H, H, H, O], [AC 2777; H, Br, H, i-Pr, O , Oi-Pr, H, H, H, O], [AC 2778; H, Br, H, i-Pr, O, SMe, H, H, H, O], [AC 2779; H, Br, H, i -Pr, O, SEt, H, H, H, O], [AC 2 780; H, Br, H, i-Pr, O, CH ₂ F, H, H, O], [AC 2781; H, Br , H, i-Pr, O , CHF 2, H, H, H, O], [AC2782; H, Br, H, i-Pr, O, CF 3, H, H, H, O], [AC2783 ; H, Br, H, i -Pr, O, OCH 2 F, H, H, H, O], [AC2784; H, Br, H, i-Pr, O, OCHF 2, H, H, H, O], [AC2785; H, Br, H, i-Pr, O, OCF 3, H, H, H, O], [AC2786; H, Br, H, i-Pr, O, SCH 2 F, H H, H, O], [AC 2787; H, Br, H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 2788; H, Br, H, i-Pr, O, SCF ₃ , H, H, H, O], [AC 2 789; H, Br, H, i-Pr, O, CN, H, H, H, O], [AC 2 790; H, Br, H, i-Pr , O, NO ₂ , H, H, H, O],

[AC 2791; H, Br, H, c-Pr, O, H, H, H, H, O], [AC 2792; H, Br, H, c-Pr, O, F, H, H, H, O H, Br, H, c-Pr, O, Cl, H, H, H, O], [AC 2794; H, Br, H, c-Pr, O, Br, H, H, H] H, Br, H, c-Pr, O, I, H, H, H, O], [AC 2796; H, Br, H, c-Pr, O, Me, H, H H, O], [AC 2 797; H, Br, H, c-Pr, O, Et, H, H, H, O], [AC 2798; H, Br, H, c-Pr, O, Pr, H H, H, O], [AC2799; H, Br, H, c-Pr, O, i-Pr, H, H, H, O], [AC 2800; H, Br, H, c-Pr, O _{, CH = CH 2, H,} H, H, O], [AC2801; H, Br, H, c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC2802 H, Br, H, c-Pr, O, C≡CH, H, H, H, O], [AC 2803; H, Br, H, c-Pr, O, C≡CCH ₃ , H, H, H H, O], [AC2804; H, Br, H, c-Pr, O, c-Pr, H, H, H, O], [AC 2805; H, Br, H, c-Pr, O, OMe, H, H, H, O], [AC 2806; H, Br, H, c-Pr, O, OEt, H, H, H, O], [AC 2807; H, Br, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 2 808; H, Br, H, c-Pr, O, SMe, H, H, H, O], [AC 2809; H, Br, H, c- Pr, O, SEt, H, H, H, O], [AC 2810; H, Br, H, c-Pr, O, CH ₂ F, H, H, O], [AC 2811; H, Br, H, c-Pr, O, CHF 2, H, H, H, O], [AC2812; H, Br, H, c-Pr, O, CF 3, H, H, H, O], [AC2813; H, Br, H, c- Pr, O, OCH 2 F, H, H, H, O], [AC2814; H, Br, H, c-Pr, O, OCHF 2, H, H, H, O ], [AC2815; H, Br , H, c-Pr, O, OCF 3, H, H, H, O], [AC2816; H, Br, H, c-Pr, O, SCH 2 F, H, H, H, O], [AC 2817; H, Br, H, c-Pr, O, SCHF ₂ , H, H, H, O], [AC 2818; H , Br, H, c-Pr , O, SCF 3, H, H, H, O], [AC2819; H, Br, H, c-Pr, O, CN, H, H, H, O], [ AC 2820; H, Br, H, c-Pr, O, NO ₂ , H, H, O], [AC 2821; H, Br, H, SMe, O, H, H, H, H, O], [AC2822; H, Br, H, SMe, O, F, H, H, H, O], [AC2823; H, Br, H, SMe, O, Cl, H, H, H, O], [AC2824 H, Br, H, SMe, O, Br, H, H, H, O], [AC2825; H, Br, H, SMe, O, I, H, H, H, O], [AC2826; H , Br, H, SMe, O, Me, H, H, H, O], [AC2827; H, Br, H, SMe, O, Et, H, H, H, O], [AC2828; H, Br , H, SMe, O, Pr, H, H, H, O], [AC 2829; H, Br, H, SMe, O, i-Pr, H, H, H, O], [AC 2830; H, Br , H, SMe, O, CH = CH 2, H, H, H, O], [AC2831; H, Br, H, SMe, O, C (CH 3) = CH 2, H, H, H, O H, Br, H, SMe, O, C≡CH, H, H, H, O], [AC 2833; H, Br, H, SMe, O, C≡CCH ₃ , H, H, H] H, O], [AC2834; H, Br, H, SMe, O, c-Pr, H, H, H, O], [AC 2 835; H, Br, H, SMe, O, OMe, H, H, H H, O], [AC 2836; H, Br, H, SMe, O, OEt, H, H, H, O], [AC 2837; H, Br, H, SMe, O, Oi-Pr, H, H, H H, O], [AC 2838; H, Br, H, SMe, O, SMe, H, H, H, O], [AC 2839; H, Br, H, SMe, O, SE t, H, H, H, H O], [AC2840; H, Br, H, SMe, O, CH 2 F, H, H, H, O], [AC2841; H, Br, H, SMe, O, CHF 2, H, H, H , O], [AC2842; H , Br, H, SMe, O, CF 3, H, H, H, O], [AC2843; H, Br, H, SMe, O, OCH 2 F, H, H, H, O], [AC 2844; H, Br, H, SMe, O, OCHF ₂ , H, H, H, O], [AC 2845; H, Br, H, SMe, O, OCF ₃ , H, H, H H, O], [AC 2846; H, Br , H, SMe, O, SCH 2 F, H, H, H, O], [AC2847; H, Br, H, SMe, O, SCHF 2, H, H, H, O], [AC2848; H, Br, H, SMe, O, SCF 3, H, H, H, O], [AC2849; H, Br, H, SMe, O, CN, H, H, H, O], [AC2850; H, Br , H, SMe, O, NO 2, H, H, H, O], [AC2851; H, Br, H, OMe, O, H, H, H, H, O], [AC2852; H, Br, H, OMe, O, F, H, H, H, O], [AC2853; H, Br, H, OMe, O, Cl, H, H, O], [AC 2854; H, Br, H, OMe, O, Br, H, H, H, O], [AC 2 855; H, Br, H, OMe, O, I, H, H, H, O], [AC 2856; H, Br, H, OMe, O, Me, H, H, H, O], [AC 2857; H, Br, H, OMe, O, Et, H, H, H, O], [AC 2858; H, Br, H, OMe, O, Pr, H, H, H, O], [AC 2859; H, Br, H, OMe, O, i-Pr, H, H, H, O], [AC 2860; H, Br, H, OMe, O, _{CH = CH 2, H, H} , H, O], [AC2861; H, Br, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC2862; H, Br, H, OMe, O, C≡CH, H, H, H, O], [AC2863; H, Br, H, OMe, O, C≡CCH ₃ , H, H, H, O], [AC 2864 H, Br, H, OMe, O, c-Pr, H, H, H, O], [AC 2865; H, Br, H, OMe, O, OMe, H, H, H, O], [AC 2866 H, Br, H, OMe, O, OEt, H, H, H, O], [AC 2867; H, Br, H, OMe, O, Oi-Pr, H, H, H, O], [AC 2868 H, Br, H, OMe, O, SMe, H, H, H, O], [AC 2869; H, Br, H, OMe, O, SE t, H, H, H, O], [AC 2870; H , Br, H, OMe, O , CH 2 F, H, H, H, O], [AC2871; H, Br, H, OMe, O, CHF 2, H, H, H, O], [AC2872; H, Br, H, OMe, O, CF 3, H, H, H, O], [AC2873; H, Br, H, OMe, O, OCH 2 F, H, H, H, O], [AC2874 H, Br, H, OM _{e, O, OCHF 2, H} , H, H, O], [AC2875; H, Br, H, OMe, O, OCF 3, H, H, H, O], [AC2876; H, Br, H, OMe, O, SCH ₂ F, H, H, H, O, [AC 2877; H, Br, H, OMe, O, SCHF ₂ , H, H, H, O], [AC 2878; H, Br, H _{, OMe, O, SCF 3,} H, H, H, O], [AC2879; H, Br, H, OMe, O, CN, H, H, H, O], [AC2880; H, Br, H, _{OMe, O, NO 2, H} , H, H, O], [AC2881; H, Br, H, F, O, H, H, H, H, O], [AC2882; H, Br, H, F , O, F, H, H, H, O], [AC2883; H, Br, H, F, O, Cl, H, H, H, O], [AC 2884; H, Br, H, F, O , Br, H, H, H, O], [AC 2885; H, Br, H, F, O, I, H, H, H, O], [AC 2886; H, Br, H, F, O, Me H, H, H, O], [AC 2887; H, Br, H, F, O, Et, H, H, H, O], [AC 2 888; H, Br, H, F, O, Pr, H , H, H, O], [AC 2889; H, Br, H, F, O, i-Pr, H, H, H, O], [AC 2890; H, Br, H, F, O, CH = CH ₂ , H, H, H, O],

[AC2891; H, Br, H , F, O, C (CH 3) = CH 2, H, H, H, O], [AC2892; H, Br, H, F, O, C≡CH, H, H, H, O], [AC 2893; H, Br, H, F, O, C≡CCH ₃ , H, H, H, O], [AC 2894; H, Br, H, F, O, c-Pr , H, H, H, O], [AC2895; H, Br, H, F, O, OMe, H, H, H, O], [AC 2896; H, Br, H, F, O, OEt, H H, H, O], [AC 2897; H, Br, H, F, O, Oi-Pr, H, H, H, O], [AC 2898; H, Br, H, F, O, SMe, H H, H, O], [AC 2899; H, Br, H, F, O, SE t, H, H, H, O], [AC 2900; H, Br, H, F, O, CH ₂ F, H , H, H, O], [AC2901; H, Br, H, F, O, CHF ₂ , H, H, H, O], [AC 2902; H, Br, H, F, O, CF ₃ , H H, H, O], [AC 2903; H, Br, H, F, O, OCH ₂ F, H, H, H, O], [AC 2904; H, Br, H, F, O, OCHF ₂ , H, H, H, O] , [AC2905; H, Br, H, F, O, OCF 3, H, H, H, O], [AC2906; H, Br, H, F, O, SCH 2 F H, H, H, O], [AC 2 907; H, Br, H, F, O, SCHF ₂ , H, H, H, O], [AC 2 908; H, Br, H, F, O, SCF ₃ H, H, H, O], [AC 2 909; H, Br, H, F, O, CN, H, H, H, O], [AC 2910; H, Br, H, F, O, NO ₂ , H, H, H, O], [AC2911; H, Br, H, Cl, O, H, H, H, H, O], [AC 2912; H, Br, H, Cl, O, F, H, H, H, O], [AC 2913; H, Br, H, Cl, O, Cl, H, H, H, O], [AC 2914; H, Br, H, Cl, O, Br, H, H, H, H, O], [AC 2915; H, Br, H, Cl, O, I, H, H, H, O], [AC 2916; H, Br, H, Cl, O, Me, H, H, H, H, O], [AC2917; H, Br, H, Cl, O, Et, H, H, H, O], [AC 2918; H, Br, H, Cl, O, Pr, H, H, H, O] [AC 2919; H, Br, H, Cl, O, i-Pr, H, H, H, O], [AC 2920; H, Br, H, Cl, _{O, CH = CH 2, H} , H, H, O], [AC2921; H, Br, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC2922; H, Br, H, Cl, O, C≡CH, H, H, H, O], [AC 2923; H, Br, H, Cl, O, C≡CCH ₃ , H, H, H, O], [AC2924; H, Br, H, Cl, O, c-Pr, H, H, H, O], [AC 2925; H, Br, H, Cl, O, OMe, H, H, H, O], [AC 2 926; H, Br, H, Cl, O, OEt, H, H, H, O], [AC 2 927; H, Br, H, Cl, O, Oi-Pr, H, H, H, O], [AC 2 928; H, Br, H, Cl, O, SMe, H, H, H, O], [AC 2 929; H, Br, H, Cl, O, SE t, H, H, H, O], [AC 2930 ; H, Br, H, Cl , O, CH 2 F, H, H, H, O], [AC2931; H, Br, H, Cl, O, CHF 2, H, H, H, O], [ AC2932; H, Br, H, Cl, O, CF 3, H, H, H, O], [AC2933; H, Br, H, Cl, O, OCH 2 F, H, H, H, O], [AC 2 934; H, Br, H, Cl, O, OCHF ₂ , H, H, H, O], [AC 2935; H, Br, H, Cl, O, OCF ₃ , H, H, H, O], [AC 2 936; H, Br, H, Cl, O, SCH ₂ F, H, H, H, O], [AC 2 937; H, Br, H, Cl, O, SCHF ₂ , H, H, H, O] , [AC 2938; H, Br, H, Cl, O, SCF ₃ , H, H, H, O], [AC 2939; H, Br, H, Cl, O, CN, H, H, H, O], [AC 2 940; H, Br, H, Cl, O, NO ₂ , H, H, H, O], [AC 2941; H, Br, H, Br, O, H, H, H, H, O], AC2942; H, Br, H, Br, O, F, H, H, O], [AC2943; H, Br, H, Br, O, Cl, H, H, H, O], [AC 2944; H, Br, H, Br, O, Br, H, H, H, O], [AC2945; H, Br, H, Br, O, I, H, H, H, O], [AC 2946; H, Br, H, Br, O, Me, H, H, H, O], [AC 2947; H, Br, H, Br, O, Et, H, H, H, O], [AC 2948; H, Br, H, Br, O, Pr, H, H, H, O], [AC 2949; H, Br , H, Br, O, i -Pr, H, H, H, O], [AC2950; H, Br, H, Br, O, CH = CH 2, H, H, H, O], [AC2951; H, Br, H, Br, O, C (CH 3) = CH 2, H, H, H, O], [AC2952; H, Br, H, Br, O, C≡CH, H, H, H H, Br, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 2954; H, Br, H, Br, O, c-Pr, H, H, H, O], [AC 2 955; H, Br, H, Br, O, OMe, H, H, H, O], [AC 2956; H, Br, H, Br, O, OE t, H, H, H, O], [AC 2957; H, Br, H, Br, O, Oi-Pr, H, H, H, O], [AC 2958; H, Br, H, Br, O, SMe, H, H, H, O], [AC 2959; H, Br, H, Br, O, SE t, H, H, H, O], [AC 2 960; H, Br, H, Br, O, CH ₂ F, H, H, H, O], [AC2961; H, Br, H, Br, O, CHF 2, H, H, H, O], [AC2962; H, Br, H, Br, O, CF 3, H, H, H, O], [AC 2963; H, Br, H, Br, O, OCH ₂ F, H, H, H, O], [AC 2964; H, Br, H, Br, O, OCHF ₂ , H, H , H, O], [AC2965 ; H, Br, H, Br, O, OCF 3, H, H, H, O], [AC2966; H, Br, H, Br, O, SCH 2 F, H, H, H, O], [AC 2967; H, Br, H, Br, O, SCHF ₂ , H, H, H, O], [AC 2968; H, Br, H, Br, O, SCF ₃ , H, H, H, O], [AC 2969; H, Br, H, Br, O, CN, H, H, H, O], [AC 2970; H, Br, H, Br, O, NO ₂ , H, H , H, O], [AC2971; H, OMe, H, H, O, H, H, H, H, O], [AC 2972; H, OMe, H, H, O, F, H, H, H H, OMe, H, H, O, Cl, H, H, O], [AC 2974; H, OMe, H, H, O, Br, H, H, H, O H, OMe, H, H, O, I, H, H, H, O], [AC 2976; H, OMe, H, H, O, Me, H, H, H, O], [AC 2977; H, OMe, H, H, O, Et, H, H, H, O], [AC 2 978; H, OMe, H, H, O, Pr, H, H, H, O], [AC 2979; H, OMe, H, H, O, i-Pr, H, H, H, O], [, AC 2 980; H, OMe, H, H, O, CH = CH ₂ , H, H, H, O], [AC 2981; H, OMe, H, H, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC2982; H, OMe, H, H, O, C≡CH, H, H, H, O], [AC2983; H, OMe, H, H, O, C, CCH ₃ H, H, H, O], [AC 2984; H, OMe, H, H, O, c-Pr, H, H, H, O], [AC 2985; H, OMe, H, H, O, OMe H, H, H, O], [AC2986; H, OMe, H, H, O, OEt, H, H, H, O], [AC 2987; H, OMe, H, H, O, Oi-Pr H, H, H, O], [AC2988; H, OMe, H, H, O, SMe, H, H, H, O], [AC2989; H, OMe, H, H, O, SEt, H , H, H, O], [AC 2 990; H, OMe, H, H, O, CH ₂ F, H, H, H, O],

[AC2991; H, OMe, H , H, O, CHF 2, H, H, H, O], [AC2992; H, OMe, H, H, O, CF 3, H, H, H, O], [AC 299; H, OMe, H, H, O, OCH ₂ F, H, H, H, O], [AC 2994; H, OMe, H, H, O, OCHF ₂ , H, H, H, O] , [AC2995; H, OMe, H, H, O, OCF 3, H, H, H, O], [AC2996; H, OMe, H, H, O, SCH 2 F, H, H, H, O H, OMe, H, H, O, SCHF ₂ , H, H, H, O], [AC 2998; H, OMe, H, H, O, SCF ₃ , H, H, H, O] H, OMe, H, H, O, CN, H, H, H, O], [AC 3000; H, OMe, H, H, O, NO ₂ , H, H, H, O] [AC3001; H, OMe, H, Me, O, H, H, H, O], [AC3002; H, OMe, H, Me, O, F, H, H, H, O], [AC 3002; AC 3003; H, OMe, H, Me, O, Cl, H, H, O], [AC 3004; H, OMe, H, Me, O, Br, H, H, O], [AC 3005; H, OMe, H, Me, O, I, H, H, H, O], [AC 3006; H, OMe, H, Me, O, Me, H, H, H, O], [AC 3007; H, OMe, H, Me, O, Et, H, H, H, O], [AC 3008; H, OMe, H, Me, O, Pr, H, H, H, O], [AC 3009; H, OMe, H, Me, O, i-Pr, H, H, H, O, [AC 3010; H, OMe, H, Me, O, CH = CH ₂ , H, H, H, O], [AC 3011; H , OMe, H, Me, O , C (CH 3) = CH 2, H, H, H, O], [AC3012; H, OMe, H, Me, O, C≡CH, H, H, H, O, [AC 3013; H, OMe, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 3014; H, OMe, H, Me, O, c-Pr, H, H , H, O], [AC 3015; H, OMe, H, Me, O, OMe, H, H, H, O], [AC 3016; H, OMe, H, Me, O, OEt, H, H, H , O], [AC 3017; H, OMe, H, Me, O, Oi-Pr, H, H, H, O], [AC 3018; H, OMe, H, Me, O, SMe, H, H, H , O], [AC 3019; H, O Me, H, Me, O, SEt, H, H, H, O], [AC 3020; H, OMe, H, Me, O, CH ₂ F, H, H, H, O], [AC 3021; H, OMe, H, Me, O, CHF 2, H, H, H, O], [AC3022; H, OMe, H, Me, O, CF 3, H, H, H, O], [AC3023; H, OMe, H, Me, O, OCH 2 F, H, H, H, O], [AC3024; H, OMe, H, Me, O, OCHF 2, H, H, H, O], [AC3025; H , OMe, H, Me, O , OCF 3, H, H, H, O], [AC3026; H, OMe, H, Me, O, SCH 2 F, H, H, H, O], [AC3027; H, OMe, H, Me, O, SCHF 2, H, H, H, O], [AC3028; H, OMe, H, Me, O, SCF 3, H, H, H, O], [AC3029; H, OMe, H, Me, O, CN, H, H, H, O], [AC3030; H, OMe, H, Me, O, NO 2, H, H, H, O], [AC3031; H , OMe, H, Et, O, H, H, H, H, O], [AC 3032; H, OMe, H, Et, O, F, H, H, H, O], [AC 3033; H, OMe , H, Et, O, Cl, H, H, H, O], [AC 3034; H, OMe, H, Et, O, Br, H, H, H, O], [AC 3035; H, OMe, H , Et, O, I, H, H, H, O], [AC3036; H, OMe, H, Et, O, Me, H, H, H, O], [AC 3037; H, OMe, H, Et , O, Et, H, H, H, O], [AC3038; H, OMe, H, Et, O, Pr, H, H, H, O], [AC 3039; H, OMe, H, Et, O , i-Pr, H, H, H, O], [AC 3040; H, OMe, H, Et, O, CH = CH ₂ , H, H, H, O], [AC 3041; H, OMe, H, _{Et, O, C (CH 3} ) = CH 2, H, H, H, O], [AC3042; H, OMe, H, Et, O, C≡CH, H, H, H, O], [AC3043 H, OMe, H, Et, O, C≡CCH ₃ , H, H, H, O], [AC3044; H, OMe, H, Et, O, c-Pr, H, H, H, O] , [AC 3045; H, OMe, H, Et, O, OMe, H, H, H, O], [AC 3046; H, OMe, H, Et, O, OEt, H, H, H, O], [, AC 3047; H, O Me, H, Et, O, Oi-Pr, H, H, H, O], [AC 3048; H, OMe, H, Et, O, SMe, H, H, H, O], [AC 3049; H, OMe, H, Et, O, SEt, H, H, H, O], [AC3050; H, OMe, H, Et, O, CH 2 F, H, H, H, O], [AC3051; H, OMe, H, Et, O, CHF 2, H, H, H, O], [AC3052; H, OMe, H, Et, O, CF 3, H, H, H, O], [AC3053; H, OMe, H, Et, O, OCH 2 F, H, H, H, O], [AC3054; H, OMe, H, Et, O, OCHF 2, H, H, H, O], [AC3055; H , OMe, H, Et, O , OCF 3, H, H, H, O], [AC3056; H, OMe, H, Et, O, SCH 2 F, H, H, H, O], [AC3057; H, OMe, H, Et, O, SCHF 2, H, H, H, O], [AC3058; H, OMe, H, Et, O, SCF 3, H, H, H, O], [AC3059; H, OMe, H, Et, O, CN, H, H, H, O], [AC3060; H, OMe, H, Et, O, NO 2, H, H, H, O], [AC3061; H , OMe, H, Pr, O, H, H, H, H, O], [AC3062; H, OMe, H, Pr, O, F, H, H, H, O], [AC3063; H, OMe , H, Pr, O, Cl, H, H, H, O], [AC 3064; H, OMe, H, Pr, O, Br, H, H, H, O], [AC 3065; H, OMe, H , Pr, O, I, H, H, H, O], [AC 3066; H, OMe, H, Pr, O, Me, H, H, H, O], [AC 3067; H, OMe, H, Pr , O, Et, H, H, H, O], [AC 3068; H, OMe, H, Pr, O, Pr, H, H, H, O], [AC 3069; H, OMe, H, Pr, O , i-Pr, H, H , H, O], [AC3070; H, OMe, H, Pr, O, CH = CH 2, H, H, H, O], [AC3071; H, OMe, H, Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 3072; H, OMe, H, Pr, O, C≡CH, H, H, H, O], [AC 3073 H, OMe, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 3074; H, OMe, H, Pr, O, c-Pr, H, H, H, O] , [AC 3075; H , OMe, H, Pr, O, OMe, H, H, H, O], [AC3076; H, OMe, H, Pr, O, OEt, H, H, H, O], [AC3077; H, OMe , H, Pr, O, Oi-Pr, H, H, H, O], [AC 3078; H, OMe, H, Pr, O, SMe, H, H, H, O], [AC 3079; H, OMe , H, Pr, O, SEt , H, H, H, O], [AC3080; H, OMe, H, Pr, O, CH 2 F, H, H, H, O], [AC3081; H, OMe , H, Pr, O, CHF 2, H, H, H, O], [AC3082; H, OMe, H, Pr, O, CF 3, H, H, H, O], [AC3083; H, OMe , H, Pr, O, OCH 2 F, H, H, H, O], [AC3084; H, OMe, H, Pr, O, OCHF 2, H, H, H, O], [AC3085; H, OMe, H, Pr, O, OCF 3, H, H, H, O], [AC3086; H, OMe, H, Pr, O, SCH 2 F, H, H, H, O], [AC3087; H , OMe, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 3088; H, OMe, H, Pr, O, SCF ₃ , H, H, O], [AC 3089; H , OMe, H, Pr, O, CN, H, H, H, O],

[AC 3090; H, OMe, H, Pr, O, NO ₂ , H, H, O], [AC 3091; H, OMe, H, i-Pr, O, H, H, H, H, O] , [AC3092; H, OMe, H, i-Pr, O, F, H, H, H, O], [AC 3093; H, OMe, H, i-Pr, O, Cl, H, H, H, O, [AC 3094; H, OMe, H, i-Pr, O, Br, H, H, O], [AC 3095; H, OMe, H, i-Pr, O, I, H, H, H, O], [AC 3096; H, OMe, H, i-Pr, O, Me, H, H, H, O], [AC 3097; H, OMe, H, i-Pr, O, Et, H, H, H, O], [AC 3098; H, OMe, H, i-Pr, O, Pr, H, H, H, O], [AC 3099; H, OMe, H, i-Pr, O, i- Pr, H, H, H, O], [AC3100; H, OMe, H, i-Pr, O, CH = CH 2, H, H, H, O], [AC3101; H, OMe, H, i _{-Pr, O, C (CH 3} ) = CH 2, H, H, H, O], [AC3102; H, OMe, H, i-Pr, O, C≡CH, H, H, H, O] , [AC 3103; H, OMe, H, i-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 3104; H, OMe, H, i-Pr, O, c-Pr, H , H, H, O], [AC 3105; H, OMe, H, i-Pr, O, OMe, H, H, H, O], [AC 3106; H, OMe, H, i-Pr, O, OEt , H, H, H, O], [AC 3107; H, OMe, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC 3108; H, OMe, H, i-Pr , O, SMe, H, H, H, O], [AC 3109; H, OMe, H, i-Pr, O, SE t, H, H, H, O], [AC 3110; H, OMe, H, i _{-Pr, O, CH 2 F,} H, H, H, O], [AC3111; H, OMe, H, i-Pr, O, CHF 2, H, H, H, O], [AC3112; H, OMe, H, i-Pr, O, CF 3, H, H, H, O], [AC3113; H, OMe, H, i-Pr, O, OCH 2 F, H, H, H, O], [AC 3 114; H, OMe, H, i-Pr, O, OCHF ₂ , H, H, H, O], [AC 3 115; H, OMe, H, i-Pr, O, OCF ₃ , H, H, H , O], [AC 3116; H, OMe, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 3 117; H, OMe, H, i-Pr, O, SCHF ₂ , H, H, H, O], [AC 3118; H, OMe, H, i- _{Pr, O, SCF 3, H} , H, H, O], [AC3119; H, OMe, H, i-Pr, O, CN, H, H, H, O], [AC3120; H, OMe, H , i-Pr, O, NO ₂ , H, H, H, O], [AC 3121; H, OMe, H, c-Pr, O, H, H, H, H, O], [AC 3122; H, OMe, H, c-Pr, O, F, H, H, H, O], [AC 3123; H, OMe, H, c-Pr, O, Cl, H, H, H, O], [AC 3 124; H, OMe, H, c-Pr, O, Br, H, H, H, O], [AC 3 125; H, OMe, H, c-Pr, O, I, H, H, H, O], [[ AC 3126; H, OMe, H, c-Pr, O, Me, H, H, H, O], [AC 3127; H, OMe, H, c-Pr, O, Et, H, H, H, O] , [AC3128; H, OMe, H, c-Pr, O, Pr, H, H, H, O], [AC 3129; H, OMe, H, c-Pr, O, i-Pr, H, H, H, O], [AC 3130; H, OMe, H, c-Pr, O, CH = CH ₂ , H, H, H, O], [AC 3131; H, OMe, H, c-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 3132; H, OMe, H, c-Pr, O, C≡CH, H, H, H, O], [AC 3133; H, OMe, H, c-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 3134; H, OMe, H, c-Pr, O, c-Pr, H, H, H, O H, OMe, H, c-Pr, O, OMe, H, H, H, O], [AC 3136; H, OMe, H, c-Pr, O, OEt, H, H, H] , O], [AC 3137; H, OMe, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC 3138; H, OMe, H, c-Pr, O, SMe, H H, H, O], [AC 3139; H, OMe, H, c-Pr, O, SEt, H, H, H, O], [AC 3140; H, OMe, H, c-Pr, O, CH ₂ F, H, H, H, O], [AC 3141; H, OMe, H, c-Pr, O, CHF ₂ , H, H, H, O], [AC 3142; H, OMe, H, c- Pr, O, CF ₃ , H, H, H, O], [AC 3143; H, OMe, H , c-Pr, O, OCH 2 F, H, H, H, O], [AC3144; H, OMe, H, c-Pr, O, OCHF 2, H, H, H, O], [AC3145; H, OMe, H, c- Pr, O, OCF 3, H, H, H, O], [AC3146; H, OMe, H, c-Pr, O, SCH 2 F, H, H, H, O H, OMe, H, c-Pr, O, SCHF ₂ , H, H, H, O], [AC 3148; H, OMe, H, c-Pr, O, SCF ₃ , H, H] H, O], [AC 3149; H, OMe, H, c-Pr, O, CN, H, H, H, O], [AC 3150; H, OMe, H, c-Pr, O, NO ₂ , H, H, H, O], [AC3151; H, OMe, H, SMe, O, H, H, H, H, O], [AC3152; H, OMe, H, SMe, O, F, H, H, H, H, O], [AC3153; H, OMe, H, SMe, O, Cl, H, H, H, O], [AC 3154; H, OMe, H, SMe, O, Br, H, H, H, H, O], [AC 3 155; H, OMe, H, SMe, O, I, H, H, H, O], [AC 3156; H, OMe, H, SMe, O, Me, H, H, H, H, O], [AC 3 157; H, OMe, H, SMe, O, Et, H, H, H, O], [AC 3158; H, OMe, H, SMe, O, Pr, H, H, H, O] , [AC3159; H, OMe, H, SMe, O, i-Pr, H, H, H, O], [AC3160; H, OMe, H, SMe, O, CH = CH 2, H, H, H , O], [AC3161; H , OMe, H, SMe, O, C (CH 3) = CH 2, H, H, H, O], [AC3162; H, OMe, H, SMe, O, C≡ CH, H, H, H, O], [AC 3163; H, OMe, H, SMe, O, C≡CCH ₃ , H, H, H, O], [AC 3 164; H, OMe, H, SMe, O , c-Pr, H, H, H, O], [AC 3165; H, OMe, H, SMe, O, OMe, H, H, H, O], [AC 3166; H, OMe, H, SMe, O , OEt, H, H, H, O], [AC 3 167; H, OMe, H, SMe, O, Oi-Pr, H, H, H, O], [AC 3168; H, OMe, H, SMe, O , SMe, H, H, H, O], [AC 3169; H, OMe, H, SMe, O, SEt, H, H, H, O], [AC 3170; H, OMe, H, SMe, _{O, CH 2 F, H,} H, H, O], [AC3171; H, OMe, H, SMe, O, CHF 2, H, H, H, O], [AC3172; H, OMe, H, SMe , O, CF ₃ , H, H, H, O], [AC 3173; H, OMe, H, SMe, O, OCH ₂ F, H, H, H, O], [AC 3174; H, OMe, H, _{SMe, O, OCHF 2, H} , H, H, O], [AC3175; H, OMe, H, SMe, O, OCF 3, H, H, H, O], [AC3176; H, OMe, H, SMe, O, SCH ₂ F, H, H, H, O, [AC 3177; H, OMe, H, SMe, O, SCHF ₂ , H, H, H, O], [AC 3178; H, OMe, H _{, SMe, O, SCF 3,} H, H, H, O], [AC3179; H, OMe, H, SMe, O, CN, H, H, H, O], [AC3180; H, OMe, H, _{SMe, O, NO 2, H} , H, H, O], [AC3181; H, OMe, H, OMe, O, H, H, H, H, O], [AC3182; H, OMe, H, OMe , O, F, H, H, H, O], [AC 3183; H, OMe, H, OMe, O, Cl, H, H, H, O], [AC 3184; H, OMe, H, OMe, O , Br, H, H, H, O], [AC 3185; H, OMe, H, OMe, O, I, H, H, H, O], [AC 3186; H, OMe, H, OMe, O, Me H, H, H, O], [AC 3187; H, OMe, H, OMe, O, Et, H, H, H, O], [AC 3188; H, OMe, H, OMe, O, Pr, H , H, H, O], [AC 3189; H, OMe, H, OMe, O, i-Pr, H, H, H, O],

[AC 3190; H, OMe, H, OMe, O, CH = CH ₂ , H, H, H, O], [AC 3191; H, OMe, H, OMe, O, C (CH ₃ ) = CH ₂ , H , H, H, O], [AC 3192; H, OMe, H, OMe, O, C≡CH, H, H, H, O], [AC 3193; H, OMe, H, OMe, O, C≡ CCH ₃ , H, H, H, O], [AC 3194; H, OMe, H, OMe, O, c-Pr, H, H, H, O], [AC 3195; H, OMe, H, OMe, O, OMe, H, H, H, O], [AC 3196; H, OMe, H, OMe, O, OEt, H, H, H, O], [AC 3 197; H, OMe, H, OMe, O, Oi- Pr, H, H, H, O], [AC 3198; H, OMe, H, OMe, O, SMe, H, H, H, O], [AC 3199; H, OMe, H, OMe, O, SEt, H, H, H, O], [AC 3200; H, OMe, H, OMe, O, CH ₂ F, H, H, H, O], [AC 3201; H, OMe, H, OMe, O, CHF ₂ , H, H, H, O ], [AC3202; H, OMe, H, OMe, O, CF 3, H, H, H, O], [AC3203; H, OMe, H, OMe, O, OCH 2 F, H, H, H, O], [AC 3204; H, OMe, H, OMe, O, OCHF ₂ , H, H, H, O], [AC 3205; H, OMe, H, OMe, O, OCF ₃ , H, H, H, O], [AC 3206; H, OMe, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 3207; H, OMe, H, OMe, O, SCHF ₂ , H, H, H, O], [AC 3208; H, OMe, H, OMe, O, SCF ₃ , H, H, H, O], [AC 3209; H, OMe, H, OMe, O, CN, H, H, H, O], [AC 3210; H, OMe, H, OMe, O, NO ₂ , H, H, H, O], [AC 3211; H, OMe, H, F, O, H H, H, H, O], [AC 3212; H, OMe, H, F, O, F, H, H, H, O], [AC 3213; H, OMe, H, F, O, Cl, H , H, H, O], [AC 3214; H, OMe, H, F, O, Br, H, H, H, O], [AC 3215; H, OMe, H, F, O, I, H, H H, O], [AC 3216; H, OMe, H, F, O, Me, H, H, H, O], [AC 3217; H, OMe, H, O F, O, Et, H, H, H, O], [AC 3218; H, OMe, H, F, O, Pr, H, H, H, O], [AC 3219; H, OMe, H, F, O, i-Pr, H, H, H, O], [AC3220; H, OMe, H, F, O, CH = CH 2, H, H, H, O], [AC3221; H, OMe, H , F, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 3222; H, OMe, H, F, O, C≡CH, H, H, H, O], [[ AC 3223; H, OMe, H, F, O, C≡CCH ₃ , H, H, H, O], [AC 3224; H, OMe, H, F, O, c-Pr, H, H, H, O H, OMe, H, F, O, OMe, H, H, H, O], [AC 3226; H, OMe, H, F, O, OEt, H, H, H, O], [AC 3227; H, OMe, H, F, O, Oi-Pr, H, H, H, O], [AC 3228; H, OMe, H, F, O, SMe, H, H, H, O], [AC 3229; H, OMe, H, F, O, SEt, H, H, H, O], [AC 3230; H, OMe, H, F, O, CH ₂ F, H, H, H, O], [AC3231; H, OMe, H , F, O, CHF 2, H, H, H, O], [AC3232; H, OMe, H, F, O, CF 3, H, H, H, O], [AC3233; H, OMe, H , F, O, OCH 2 F, H, H, H, O], [AC3234; H, OMe, H, F, O, OCHF 2, H, H, H, O] , [AC3235; H, OMe, H, F, O, OCF 3, H, H, H, O], [AC3236; H, OMe, H, F, O, SCH 2 F, H, H, H, O H, OMe, H, F, O, SCHF ₂ , H, H, H, O], [AC 3238; H, OMe, H, F, O, SCF ₃ , H, H, H, O] H, OMe, H, F, O, CN, H, H, H, O], [AC 3240; H, OMe, H, F, O, NO ₂ , H, H, H, O] [AC3241; H, OMe, H, Cl, O, H, H, H, O], [AC3242; H, OMe, H, Cl, O, F, H, H, H, O], [AC3241; AC 3243; H, OMe, H, Cl, O, Cl, H, H, H, O], [AC 3244; H, OMe, H, Cl, O, Br, H, H, H, O], [AC 3245; H, OMe, H, Cl, O, I, H, H, H, O], [AC 3246; H, OMe, H, Cl, O, Me, H, H, H, O], [AC 3247; H, OMe, H, Cl, O, Et, H, H, H, O], [AC 3248; H, OMe, H, Cl, O, Pr, H, H, H, O], [AC 3249; H, OMe, H, Cl, O, i-Pr, H, H, H, O], [AC 3250; H, OMe, H, Cl, O, CH = CH 2, H, H, H, O], [AC3251; H, OMe, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC 3252; H, OMe, H, Cl, O, C≡CH, H, H, H, O], [AC 3253; H, OMe, H, Cl, O, C≡ CCH ₃ , H H, H, O], [AC 3254; H, OMe, H, Cl, O, c-Pr, H, H, H, O], [AC 3 255; H, OMe, H, Cl, O, OMe, H , H, H, O], [AC 3 256; H, OMe, H, Cl, O, OEt, H, H, H, O], [AC 3 257; H, OMe, H, Cl, O, Oi-Pr, H , H, H, O], [AC3258; H, OMe, H, Cl, O, SMe, H, H, H, O], [AC 3259; H, OMe, H, Cl, O, SEt, H, H , H, O], [AC 3 260; H, OMe, H, Cl, O, CH ₂ F, H, H, H, O], [AC 3261; H, OMe, H, Cl, O, CHF ₂ , H, H, H, O], [ AC3262; H, OMe, H, Cl, O, CF 3, H, H, H, O], [AC3263; H, OMe, H, Cl, O, OCH 2 F, H H, H, O], [AC 3264; H, OMe, H, Cl, O, OCHF ₂ , H, H, H, O], [AC 3265; H, OMe, H, Cl, O, OCF ₃ , H , H, H, O], [AC 3266; H, OMe, H, Cl, O, SCH ₂ F, H, H, H, O], [AC 3 267; H, OMe, H, Cl, O, SCHF ₂ , H, H, H, O], [AC 3268; H, OMe, H, Cl, O, SCF ₃ , H, H, H, O], [AC 3269; H, OMe, H, Cl, O, CN, H , H, H, O], [AC 3270; H, OMe, H, Cl, O, NO ₂ , H, H, H, O], [AC 3271; H, OMe, H, Br, O, H, H, H, H, O], [AC3272; H, OMe, H, Br, O, F, H, H, H, O], [AC 3273; H, OMe, H, Br, O, Cl, H, H, H, O H, OMe, H, Br, O, Br, H, H, H, O], [AC 3275; H, OMe, H, Br, O, I, H, H, H, O], [AC 3276; H, OMe, H, Br, O, Me, H, H, H, O], [AC 3277; H, OMe, H, Br, O, Et, H, H, H, O], [AC 3278 H, OMe, H, Br, O, Pr, H, H, H, O], [AC 3279; H, OMe, H, Br, O, i-Pr, H, H, H, O], [AC 3280 ; H, OMe, H, Br , O, CH = CH 2, H, H, H, O], [AC3281; H, OMe, H, Br, O, C (CH 3) = CH 2, H, H H, O], [AC3282; H, OMe, H, Br, O, C≡CH, H, H, H, O], [AC 3283; H, OMe, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 3284; H, OMe, H, Br, O, c-Pr, H, H, H, O], [AC 3285; H, OMe, H, Br, O, OMe, H, H, H, O], [AC 3286; H, OMe, H, Br, O, OEt, H, H, H, O], [AC 3287; H, OMe, H, Br, O, Oi-Pr, H, H, H, O], [AC3288; H, OMe, H, Br, O, SMe, H, H, H, O], [AC 3289; H, OMe, H, Br, O, SEt, H, H, H, O],

[AC3290; H, OMe, H , Br, O, CH 2 F, H, H, H, O], [AC3291; H, OMe, H, Br, O, CHF 2, H, H, H, O] , [AC3292; H, OMe, H, Br, O, CF 3, H, H, H, O], [AC3293; H, OMe, H, Br, O, OCH 2 F, H, H, H, O ], [AC3294; H, OMe , H, Br, O, OCHF 2, H, H, H, O], [AC3295; H, OMe, H, Br, O, OCF 3, H, H, H, O H, OMe, H, Br, O, SCH ₂ F, H, H, H, O], [AC 3 297; H, OMe, H, Br, O, SCHF ₂ , H, H, H, H] O], [AC 3298; H, OMe, H, Br, O, SCF ₃ , H, H, H, O], [AC 3 299; H, OMe, H, Br, O, CN, H, H, H, O ], [AC3300; H, OMe , H, Br, O, NO 2, H, H, H, O], [AC3301; H, OEt, H, H, O, H, H, H, H, O] [AC3302; H, OEt, H, H, O, F, H, H, O], [AC 3303; H, OEt, H, H, O, Cl, H, H, H, O], [AC 3302; AC 3304; H, OEt, H, H, H, O, Br, H, H, O], [AC 3 305; H, OEt, H, H, O, I, H, H, O, [AC 3306; H, OEt, H, H, O, Me, H, H, H, O], [AC 3307; H, OEt, H, H, O, Et, H, H, H, O], [AC 3308; H, OEt, H, H, H, O, Pr, H, H, H, O], [AC 3309; H, OEt, H, H, O, i-Pr, H, H, H, O], [AC 3310; H, OEt, H, H, O, CH = CH 2, H, H, H, O], [AC3311; H, OEt, H, H, O, C (CH 3) = CH 2, H, H, H, O, [AC3312; H, OEt, H, H, O, C≡CH, H, H, H, O], [AC3313; H, OEt, H, H, O, C≡ CCH ₃ , H, H H, O], [AC3314; H, OEt, H, H, O, c-Pr, H, H, H, O], [AC 3315; H, OEt, H, H, O, OMe, H, H , H, O], [AC3316; H, OEt, H, H, O, OEt, H, H, H, O], [AC 3317; H, OEt, H, H, O, Oi-Pr, H, H , H, O], [AC 3318; H, OE t, H , H, O, SMe, H, H, H, O], [AC3319; H, OEt, H, H, O, SEt, H, H, H, O], [AC3320; H, OEt, H, H] _{, O, CH 2 F, H} , H, H, O], [AC3321; H, OEt, H, H, O, CHF 2, H, H, H, O], [AC3322; H, OEt, H, _{H, O, CF 3, H} , H, H, O], [AC3323; H, OEt, H, H, O, OCH 2 F, H, H, H, O], [AC3324; H, OEt, H _{, H, O, OCHF 2,} H, H, H, O], [AC3325; H, OEt, H, H, O, OCF 3, H, H, H, O], [AC3326; H, OEt, H , H, O, SCH ₂ F, H, H, H, O], [AC 3327; H, OEt, H, H, O, SCHF ₂ , H, H, H, O], [AC 3328; H, OE t, _{H, H, O, SCF 3} , H, H, H, O], [AC3329; H, OEt, H, H, O, CN, H, H, H, O], [AC3330; H, OEt, H _{, H, O, NO 2,} H, H, H, O], [AC3331; H, OEt, H, Me, O, H, H, H, H, O], [AC3332; H, OEt, H, Me, O, F, H, H, H, O], [AC3333; H, OEt, H, Me, O, Cl, H, H, H, O], [AC3334; H, OEt, H, Me, O, Br, H, H, H, O], [AC3335; H, OEt, H, Me, O, I, H, H, H, O], [AC 3336; H, OEt, H, Me, O, Me, H, H, H, O], [AC 3337; H, OEt, H, Me, O, Et, H, H, H, O], [AC 3338; H, OEt, H, Me, O, Pr, H, H, H, O], [AC3339; H, OEt, H, Me, O, i-Pr, H, H, H, O], [AC 3340; H, OEt, H, Me, O, CH = _{CH 2, H, H, H} , O], [AC3341; H, OEt, H, Me, O, C (CH 3) = CH 2, H, H, H, O], [AC3342; H, OEt, H, Me, O, C≡CH, H, H, H, O], [AC 3343; H, OEt, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 3344; H , OEt, H, Me, O, c-Pr, H, H, H, O], [AC3345; H, OEt, H, Me, O, OMe, H, H, H, O], [AC 3346; H , OEt, H, Me, O, OEt, H, H H, O], [AC 3347; H, OEt, H, Me, O, Oi-Pr, H, H, H, O], [AC 3348; H, OEt, H, Me, O, SMe, H, H , H, O], [AC3349 ; H, OEt, H, Me, O, SEt, H, H, H, O], [AC3350; H, OEt, H, Me, O, CH 2 F, H, H , H, O], [AC3351 ; H, OEt, H, Me, O, CHF 2, H, H, H, O], [AC3352; H, OEt, H, Me, O, CF 3, H, H , H, O], [AC3353 ; H, OEt, H, Me, O, OCH 2 F, H, H, H, O], [AC3354; H, OEt, H, Me, O, OCHF 2, H, H, H, O], [ AC3355; H, OEt, H, Me, O, OCF 3, H, H, H, O], [AC3356; H, OEt, H, Me, O, SCH 2 F, H , H, H, O], [AC 3357; H, OEt, H, Me, O, SCHF ₂ , H, H, H, O], [AC 3358; H, OE t, H, Me, O, SCF ₃ , H , H, H, O], [AC 3359; H, OEt, H, Me, O, CN, H, H, H, O], [AC 3360; H, OE t, H, Me, O, NO ₂ , H, H, H, O], [AC3361; H, OEt, H, Et, O, H, H, H, H, O], [AC3362; H, OEt, H, Et, O, F, H, H, H, O], [AC3363; H, OEt, H, Et, O, Cl, H, H, H] O, [AC 3364; H, OEt, H, Et, O, Br, H, H, H, H, O], [AC3365; H, OEt, H, Et, O, I, H, H, H, O], [AC 3366; H, OEt, H, Et, O, Me, H, H, H, O] H, OEt, H, Et, O, Et, H, H, H, O], [AC 3368; H, OEt, H, Et, O, Pr, H, H, H, O], [AC 3367; AC 3369; H, OEt, H, Et, O, i-Pr, H, H, H, O], [AC 3370; H, OEt, H, Et, O, CH = CH ₂ , H, H, H, O ], [AC3371; H, OEt , H, Et, O, C (CH 3) = CH 2, H, H, H, O], [AC3372; H, OEt, H, Et, O, C≡CH, H, H, H, O], [AC 3373; H, OEt, H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 3374; H, OE t, H, Et, O, c -Pr, H , H, H, O], [AC 3375; H, OEt, H, Et, O, OMe, H, H, H, O], [AC 3376; H, OEt, H, Et, O, OE t, H, H H, O], [AC 3377; H, OEt, H, Et, O, Oi-Pr, H, H, H, O], [AC 3378; H, OEt, H, Et, O, SMe, H, H , H, O], [AC 3379; H, OEt, H, Et, O, SE, H, H, H, O], [AC 3380; H, OE t, H, Et, O, CH ₂ F, H, H , H, O], [AC3381 ; H, OEt, H, Et, O, CHF 2, H, H, H, O], [AC3382; H, OEt, H, Et, O, CF 3, H, H , H, O], [AC3383 ; H, OEt, H, Et, O, OCH 2 F, H, H, H, O], [AC3384; H, OEt, H, Et, O, OCHF 2, H, H, H, O], [ AC3385; H, OEt, H, Et, O, OCF 3, H, H, H, O], [AC3386; H, OEt, H, Et, O, SCH 2 F, H , H, H, O], [AC3387; H, OEt, H, Et, O, SCHF 2, H, H, H, O], [AC3388; H, OEt, H, Et, O, SCF 3, H , H, H, O],

[AC 3 389; H, OEt, H, Et, O, CN, H, H, H, O], [AC 3390; H, OEt, H, Et, O, NO ₂ , H, H, H, O], [AC 3390; AC3391; H, OEt, H, Pr, O, H, H, H, O], [AC3392; H, OEt, H, Pr, O, F, H, H, H, O], [AC3393; H, OEt, H, Pr, O, Cl, H, H, H, O], [AC 3394; H, OEt, H, Pr, O, Br, H, H, H, O], [AC 3395; H, OEt, H, Pr, O, I, H, H, H, O], [AC3396; H, OEt, H, Pr, O, Me, H, H, H, O], [AC3397; H, OEt, H, Pr, O, Et, H, H, H, O], [AC3398; H, OEt, H, Pr, O, Pr, H, H, H, O], [AC 3399; H, OEt, H, Pr, O, i-Pr, H, H, H, O, [AC 3400; H, OEt, H, Pr, O, CH = CH ₂ , H, H, H, O], [AC 3401; H, OEt , H, Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC3402; H, OEt, H, Pr, O, C≡CH, H, H, H, O] , [AC3403; H, OEt, H, Pr, O, C≡CCH 3, H, H, H, O], [AC3404; H, OEt, H, Pr, O, c-Pr, H, H, H , O], [AC 3405; H, OEt, H, Pr, O, OMe, H, H, H, O], [AC 3406; H, OEt, H, Pr, O, OEt, H, H, H, O H, OEt, H, Pr, O, Oi-Pr, H, H, H, O], [AC 3408; H, OEt, H, Pr, O, SMe, H, H, H, O] ], [AC3409; H, OEt , H, Pr, O, SEt, H, H, H, O], [AC3410; H, OEt, H, Pr, O, CH 2 F, H, H, H, O ], [AC3411; H, OEt , H, Pr, O, CHF 2, H, H, H, O], [AC3412; H, OEt, H, Pr, O, CF 3, H, H, H, O ], [AC3413; H, OEt , H, Pr, O, OCH 2 F, H, H, H, O], [AC3414; H, OEt, H, Pr, O, OCHF 2, H, H, H, O], [AC3415; H, OEt, H, Pr, O, OCF 3, H, H, H, O], [AC3416; H, OEt, H, Pr, O, SCH 2 F, H, H, H , O], [AC34 17; H, OEt, H, Pr, O, SCHF ₂ , H, H, H, O], [AC 3418; H, OEt, H, Pr, O, SCF ₃ , H, H, H, O], [[ AC 3419; H, OEt, H, Pr, O, CN, H, H, H, O], [AC 3420; H, OEt, H, Pr, O, NO ₂ , H, H, H, O], [AC 3421 H, OEt, H, i-Pr, O, H, H, H, H, O], [AC3422; H, OEt, H, i-Pr, O, F, H, H, H, O], [AC3423; H, OEt, H, i-Pr, O, Cl, H, H, H, O], [AC 3424; H, OEt, H, i-Pr, O, Br, H, H, H, O , [AC3425; H, OEt, H, i-Pr, O, I, H, H, H, O], [AC 3426; H, OEt, H, i-Pr, O, Me, H, H, H] , O], [AC3427; H, OEt, H, i-Pr, O, Et, H, H, H, O], [AC 3428; H, OEt, H, i-Pr, O, Pr, H, H H, O], [AC3429; H, OEt, H, i-Pr, O, i-Pr, H, H, H, O], [AC 3430; H, OEt, H, i-Pr, O, CH _{= CH 2, H, H,} H, O], [AC3431; H, OEt, H, i-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC3432; H , OEt, H, i-Pr, O, C≡CH, H, H, H, O], [AC3433; H, OEt, H, i-Pr, O, C≡CCH ₃ , H, H, H, O, [AC3434; H, OEt, H, i-Pr, O, c-Pr, H, H, H, O], [AC 3435; H, OEt, H, i-Pr, O, OMe, H, H, H, O], [AC3436; H, OEt, H, i-Pr, O, OEt, H, H, H, O], [AC 3437; H, OEt, H, i-Pr, O, Oi- Pr, H, H, H, O], [AC 3438; H, OEt, H, i-Pr, O, SMe, H, H, H, O], [AC 3439; H, OEt, H, i-Pr, O, SEt, H, H, H, O], [AC3440; H, OEt, H, i-Pr, O, CH 2 F, H, H, H, O], [AC3441; H, OEt, H, _{i-Pr, O, CHF 2} , H, H, H, O], [AC3442; H, OEt, H, i-Pr, O, CF 3, H, H, H, O], [AC3443; H, OEt, H, i-Pr, O, OCH ₂ F, H, H, H, O], [A C3444; H, OEt, H, i-Pr, O, OCHF 2, H, H, H, O], [AC3445; H, OEt, H, i-Pr, O, OCF 3, H, H, H, O], [AC 3446; H, OEt, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 3447; H, OEt, H, i-Pr, O, SCHF ₂ , H , H, H, O], [AC 3448; H, OEt, H, i-Pr, O, SCF ₃ , H, H, H, O], [AC 3449; H, OEt, H, i-Pr, O, CN, H, H, H, O], [AC3450; H, OEt, H, i-Pr, O, NO 2, H, H, H, O], [AC3451; H, OEt, H, c-Pr , O, H, H, H, H, O], [AC3452; H, OEt, H, c-Pr, O, F, H, H, H, O], [AC3453; H, OEt, H, c -Pr, O, Cl, H, H, H, O, [AC 3454; H, OEt, H, c-Pr, O, Br, H, H, O], [AC 3455; H, OE t, H , c-Pr, O, I, H, H, H, O], [AC 3456; H, OEt, H, c-Pr, O, Me, H, H, O], [AC 3457; H, OEt , H, c-Pr, O, Et, H, H, H, O], [AC 3458; H, OEt, H, c-Pr, O, Pr, H, H, H, O], [AC 3459; H , OEt, H, c-Pr , O, i-Pr, H, H, H, O], [AC3460; H, OEt, H, c-Pr, O, CH = CH 2, H, H, H, O], [AC3461; H, OEt, H, c-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC3462; H, OEt, H, c-Pr, O , C≡CH, H, H, H, O], [AC3463; H, OEt, H, c-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 3464; H, OEt, H, c-Pr, O, c-Pr, H, H, H, O], [AC3465; H, OEt, H, c-Pr, O, OMe, H, H, H, O], [AC 3466; H, OEt, H, c-Pr, O, OEt, H, H, H, O], [AC 3467; H, OEt, H, c-Pr, O, Oi-Pr, H, H, H, O] , [AC 3468; H, OEt, H, c-Pr, O, SMe, H, H, H, O], [AC 3469; H, OEt, H, c-Pr, O, SEt, H, H, H, H, O], [AC 3470; H, OEt, H, c-Pr, O, CH ₂ F, H, H, H, O], [AC 3471; H, OEt, H, c-Pr, O, CHF ₂ , H, H, H, O], [AC 3472; H, OE t, H, c-Pr , O, CF ₃ , H, H, H, O], [AC 3473; H, OEt, H, c-Pr, O, OCH ₂ F, H, H, H, O], [AC 3474; H, OE t, H, c-Pr, O, OCHF 2, H, H, H, O], [AC3475; H, OEt, H, c-Pr, O, OCF 3, H, H, H, O], [AC3476; H, OEt, H, c- Pr, O, SCH 2 F, H, H, H, O], [AC3477; H, OEt, H, c-Pr, O, SCHF 2, H, H, H, O ], [AC3478; H, OEt , H, c-Pr, O, SCF 3, H, H, H, O], [AC3479; H, OEt, H, c-Pr, O, CN, H, H, H, O], [AC3480; H, OEt, H, c-Pr, O, NO 2, H, H, H, O], [AC3481; H, OEt, H, SMe, O, H, H, H H, O], [AC3482; H, OEt, H, SMe, O, F, H, H, H, O], [AC3483; H, OEt, H, SMe, O, Cl, H, H, H , O], [AC3484; H, OEt, H, SMe, O, Br, H, H, O], [AC 3485; H, OEt, H, SMe, O, I, H, H, H, O H, OEt, H, SMe, O, Me, H, H, H, O], [AC 3487; H, OEt, H, SMe, O, Et, H, H, H, O], [AC3488; H, OEt, H, SMe, O, Pr, H, H, H, O],

[AC 3489; H, OEt, H, SMe, O, i-Pr, H, H, H, O], [AC 3490; H, OEt, H, SMe, O, CH = CH ₂ , H, H, H, H O], [AC3491; H, OEt, H, SMe, O, C (CH 3) = CH 2, H, H, H, O], [AC3492; H, OEt, H, SMe, O, C≡CH H, H, H, O], [AC3493; H, OEt, H, SMe, O, C≡CCH ₃ , H, H, H, O], [AC 3494; H, OEt, H, SMe, O, c-Pr, H, H, H, O], [AC 3495; H, OEt, H, SMe, O, OMe, H, H, H, O], [AC 3496; H, OEt, H, SMe, O, OEt, H, H, H, O], [AC 3497; H, OEt, H, SMe, O, Oi-Pr, H, H, H, O], [AC 3498; H, OEt, H, SMe, O, SMe, H, H, H, O], [AC 3499; H, OEt, H, SMe, O, SE, H, H, H, O], [AC 3500] H, OEt, H, SMe, O, CH ₂ F, H, H, H, O], [AC 3501; H, OEt, H, SMe, O, CHF ₂ , H, H, H, O], [AC 3502; H, OE t, H, SMe, O, CF ₃ , H, H, H, O], [AC 3503; H, OEt, H, SMe, O, OCH ₂ F, H, H, H, O], [AC 3504; H, OEt, H, SMe, O, _{OCHF 2, H, H, H} , O], [AC3505; H, OEt, H, SMe, O, OCF 3, H, H, H, O], [AC3506; H, OEt, H, SMe, O, SCH ₂ F, H, H, H, O], [AC 3507; H, OEt, H, SMe, O, SCHF ₂ , H, H, H, O], [AC 3508; H, OEt, H, SMe, O , SCF ₃ , H, H, H, O], [AC 3509; H, OEt, H, SMe, O, CN, H, H, H, O], [AC 3510; H, OEt, H, SMe, O, _{NO 2, H, H, H} , O], [AC3511; H, OEt, H, OMe, O, H, H, H, H, O], [AC3512; H, OEt, H, OMe, O, F H, H, H, O], [AC 3513; H, OEt, H, OMe, O, Cl, H, H, H, O], [AC 3514; H, OE t, H, OMe, O, Br, H , H, H, O], [AC 3515; H, OEt, H, OMe, O, I, H, H, H, O], [A H, OEt, H, OMe, O, Me, H, H, H, O], [AC 3517; H, OEt, H, OMe, O, Et, H, H, H, O], [AC 3518; H, OEt, H, OMe, O, Pr, H, H, H, O], [AC 3519; H, OEt, H, OMe, O, i-Pr, H, H, H, O], [AC 3520; H, OEt, H, OMe, O, CH = CH 2, H, H, H, O], [AC3521; H, OEt, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC3522; H, OEt, H, OMe, O, C≡CH, H, H, H, O], [AC3523; H, OEt, H, OMe, O, C≡CCH ₃ , H , H, H, O], [AC 3524; H, OEt, H, OMe, O, c-Pr, H, H, H, O], [AC 3525; H, OEt, H, OMe, O, OMe, H , H, H, O], [AC 3526; H, OEt, H, OMe, O, OEt, H, H, H, O], [AC 3527; H, OEt, H, OMe, O, Oi-Pr, H , H, H, O], [AC3528; H, OEt, H, OMe, O, SMe, H, H, H, O], [AC 3529; H, OEt, H, OMe, O, SEt, H, H , H, O], [AC3530 ; H, OEt, H, OMe, O, CH 2 F, H, H, H, O], [AC3531; H, OEt, H, OMe, O, CHF 2, H, H, H, O], [ AC3532; H, OEt, H, OMe, O, CF 3, H, H, H, O], [AC3533; H, OEt, H, OMe, O, OCH 2 F, H , H, H, O], [AC3534; H, OEt, H, OMe, O, OCHF 2, H, H, H, O], [AC3535; H, OEt, H, OMe, O, OCF 3, H H, H, O], [AC 3536; H, OEt, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 3537; H, OE t, H, OMe, O, SCHF ₂ , H, H, H, O] , [AC3538; H, OEt, H, OMe, O, SCF 3, H, H, H, O], [AC3539; H, OEt, H, OMe, O, CN, H , H, H, O], [AC 3540; H, OEt, H, OMe, O, NO ₂ , H, H, H, O], [AC 3541; H, OEt, H, F, O, H, H, H, H, H, O], [AC3542; H, OEt, H, F, O, F, H, H, H, O], [AC 3543 H, OEt, H, F, O, Cl, H, H, O], [AC 3544; H, OEt, H, F, O, Br, H, H, H, O], [AC 3545; H , OEt, H, F, O, I, H, H, H, O], [AC 3546; H, OEt, H, F, O, Me, H, H, O, [AC 3547; H, OEt , H, F, O, Et, H, H, H, O], [AC 3548; H, OEt, H, F, O, Pr, H, H, H, O], [AC 3549; H, OE t, H , F, O, i-Pr , H, H, H, O], [AC3550; H, OEt, H, F, O, CH = CH 2, H, H, H, O], [AC3551; H, OEt, H, F, O, C (CH 3) = CH 2, H, H, H, O], [AC3552; H, OEt, H, F, O, C≡CH, H, H, H, O H, OEt, H, F, O, C≡CCH ₃ , H, H, H, O], [AC 3554; H, OEt, H, F, O, c-Pr, H, H, H] H, O], [AC 3 555; H, OEt, H, F, O, OMe, H, H, H, O], [AC 3556; H, OE t, H, F, O, OE t, H, H, H, H, H, OEt, H, F, O, Oi-Pr, H, H, H, O], [AC 3 558; H, OEt, H, F, O, SMe, H, H, H, H] O], [AC3559; H, OEt, H, F, O, SEt, H, H, H, O], [AC3560; H, OEt, H, F, O, CH 2 F, H, H, H, O], [AC3561; H, OEt, H, F, O, CHF 2, H, H, H, O], [AC3562; H, OEt, H, F, O, CF 3, H, H, H, O], [AC3563; H, OEt, H, F, O, OCH 2 F, H, H, H, O], [AC3564; H, OEt, H, F, O, OCHF 2, H, H, H , O], [AC3565; H , OEt, H, F, O, OCF 3, H, H, H, O], [AC3566; H, OEt, H, F, O, SCH 2 F, H, H, H, O], [AC3567; H, OEt, H, F, O, SCHF 2, H, H, H, O], [AC3568; H, OEt, H, F, O, SCF 3, H, H, H, O], [AC 3569; H, OEt, H, F, O, CN, H, H, H, O], [AC 3570; H, OEt, H, F, O, NO ₂ , H, H, H H, OEt, H, Cl, O, H, H, H, H, O], [AC3572; H, OEt, H, Cl, O, F, H, H, O], [AC3573; H, OEt, H, Cl, O, Cl, H, H, H, O] H, OEt, H, Cl, O, Br, H, H, O], [AC 3575; H, OEt, H, Cl, O, I, H, H, H, O], [AC 3574; AC 3576; H, OEt, H, Cl, O, Me, H, H, H, O], [AC 3577; H, OEt, H, Cl, O, Et, H, H, H, O], [AC 3578; H, OEt, H, Cl, O, Pr, H, H, H, O], [AC 3579; H, OEt, H, Cl, O, i-Pr, H, H, H, O], [AC 3 580; H, OEt, H, Cl, O, CH = CH 2, H, H, H, O], [AC3581; H, OEt, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC3582; H, OEt, H, Cl, O, C≡CH, H, H, H, O], [AC3583; H, OEt, H, Cl, O, C≡CCH ₃ , H H, H, O], [AC3584; H, OEt, H, Cl, O, c-Pr, H, H, H, O], [AC 3585; H, OEt, H, Cl, O, OMe, H , H, H, O], [AC3586; H, OEt, H, Cl, O, OEt, H, H, H, O], [AC 3587; H, OEt, H, Cl, O, Oi-Pr, H , H, H, O], [AC 3588; H, OEt, H, Cl, O, SMe, H, H, H, O],

[AC3589; H, OEt, H , Cl, O, SEt, H, H, H, O], [AC3590; H, OEt, H, Cl, O, CH 2 F, H, H, H, O], [AC3591; H, OEt, H , Cl, O, CHF 2, H, H, H, O], [AC3592; H, OEt, H, Cl, O, CF 3, H, H, H, O], [AC3593; H, OEt, H , Cl, O, OCH 2 F, H, H, H, O], [AC3594; H, OEt, H, Cl, O, OCHF 2, H, H, H, O] , [AC3595; H, OEt, H, Cl, O, OCF 3, H, H, H, O], [AC3596; H, OEt, H, Cl, O, SCH 2 F, H, H, H, O H, OEt, H, Cl, O, SCHF ₂ , H, H, H, O], [AC 3598; H, OEt, H, Cl, O, SCF ₃ , H, H, H, O] H, OEt, H, Cl, O, CN, H, H, H, O], [AC 3600; H, OEt, H, Cl, O, NO ₂ , H, H, H, O] H, OEt, H, Br, O, H, H, H, O], [AC 3602; H, OEt, H, Br, O, F, H, H, H, O], [AC 3601; AC 3603; H, OEt, H, Br, O, Cl, H, H, O], [AC 3604; H, OEt, H, Br, O, Br, H, H, H, O], [AC 3605; H, OEt, H, Br, O, I, H, H, O, [AC3606; H, OEt, H, Br, O, Me, H, H, H, O], [AC 3607; H, OEt, H, Br, O, Et, H, H, H, O], [AC 3608; H, OEt, H, Br, O, Pr, H, H, H, O], [AC 3609; H, OEt, H, Br, O, i- Pr, H, H, H, O], [AC3610; H, OEt, H, Br, O, CH = CH 2, H, H, H, O], [AC3611; H , OEt, H, Br, O , C (CH 3) = CH 2, H, H, H, O], [AC3612; H, OEt, H, Br, O, C≡CH, H, H, H, O], [AC 3613; H, OEt, H, Br, O, C≡CCH ₃ , H, H, H, O], [AC 3614; H, OEt, H, Br, O, c-Pr, H, H , H, O], [AC3615; H, OEt, H, Br, O, H, H, H, O], [AC 3616; H, OEt, H, Br, O, OEt, H, H, H] , O], [AC 3617; H, OEt, H, Br, O, Oi-Pr, H, H, H, O], [AC 3618; H, OEt, H, Br, O, SMe, H, H, H, O], [AC 3619; H, OEt, H, Br, O, SEt, H, H, H, O], [AC 3620; H, OEt, H, Br, O, CH ₂ F, H, H, H, O], [AC3621; H, OEt, H , Br, O, CHF 2, H, H, H, O], [AC3622; H, OEt, H, Br, O, CF 3, H, H, H, O], [AC3623; H, OEt, H , Br, O, OCH 2 F, H, H, H, O], [AC3624; H, OEt, H, Br, O, OCHF 2, H, H, H, O] , [AC3625; H, OEt, H, Br, O, OCF 3, H, H, H, O], [AC3626; H, OEt, H, Br, O, SCH 2 F, H, H, H, O H, OEt, H, Br, O, SCHF ₂ , H, H, H, O], [AC 3628; H, OEt, H, Br, O, SCF ₃ , H, H, H, O] ], [AC3629; H, OEt , H, Br, O, CN, H, H, H, O], [AC3630; H, OEt, H, Br, O, NO 2, H, H, H, O] _{, [AC3631; H, CHF 2} , H, H, O, H, H, H, H, O], [AC3632; H, CHF 2, H, H, O, F, H, H, H, O] _{, [AC3633; H, CHF 2} , H, H, O, Cl, H, H, H, O], [AC3634; H, CHF 2, H, H, O, Br, H, H, H, O] _{, [AC3635; H, CHF 2} , H, H, O, I, H, H, H, O], [AC3636; H, CHF 2, H, H, O, Me, H, H, H, O] _{, [AC3637; H, CHF 2} , H, H, O, Et, H, H, H, O], [AC3638; H, CHF 2, H, H, O, Pr, H, H, H, O] _{, [AC3639; H, CHF 2} , H, H, O, i-Pr, H, H, H, O], [AC3640; H, CHF 2, H, H, O, CH = CH 2, H, H , H, O], [AC3641 ; H, CHF 2, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC3642; H, CHF 2, H, H, O, C≡CH, H, H, H, O, [AC3643; H, CHF ₂ , H, H, O, C≡CCH ₃ , H, H, H, O], [AC 3644 _{; H, CHF 2, H,} H, O, c-Pr, H, H, H, O], [AC3645; H, CHF 2, H, H, O, OMe, H, H, H, O], _{[AC3646; H, CHF 2,} H, H, O, OEt, H, H, H, O], [AC3647; H, CHF 2, H, H, O, Oi-Pr, H, H, H, O ], [AC3648; H, CHF 2, H, H, O, SMe, H, H, H, O], [AC3649; H, CHF 2, H, H, O, SEt, H, H, H, O ], [AC3650; H, CHF 2, H, H, O, CH 2 F, H, H, H, O], [AC3651; H, CHF 2, H, H, O, CHF 2, H, H, H, O], [AC3652; H, CHF 2, H, H, O, CF 3, H, H, H, O], [AC3653; H, CHF 2, H, H, O, OCH 2 F, H , H, H, O], [AC3654; H, CHF 2, H, H, O, OCHF 2, H, H, H, O], [AC3655; H, CHF 2, H, H, O, OCF 3 H, H, H, O], [AC 3656; H, CHF ₂ , H, H, O, SCH ₂ F, H, H, H, O], [AC 3657; H, CHF ₂ , H, H, O _{, SCHF 2, H, H,} H, O], [AC3658; H, CHF 2, H, H, O, SCF 3, H, H, H, O], [AC3659; H, CHF 2, H, H , O, CN, H, H , H, O], [AC3660; H, CHF 2, H, H, O, NO 2, H, H, H, O], [AC3661; H, CHF 2, H, Me, O, H, H, H, H, O], [AC3662; H, CHF 2, H, Me, O, F, H, H, H, O], [AC3663; H, CHF 2, H, Me, O, Cl, H, H, H, O], [AC3664; H, CHF 2, H, Me, O, Br, H, H, H, O], [AC3665; H, CHF 2, H, Me, O, I, H, H, H, O], [AC 3 666; H, CHF ₂ , H, Me, O, Me, H, H, H, O], [AC 3 667; H, CHF ₂ , H, Me, O, Et, H, H, H, O], [AC 3668; H, CHF ₂ , H, Me, O, Pr, H, H, H, O], [AC 3 669; H, CHF ₂ , H, Me, O, i-Pr, H, H, H, O], [AC 3 670; H, CHF ₂ , H, Me, O, CH = CH ₂ , H, H, H H, CHF ₂ , H, Me, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 3672; H, CHF ₂ , H, Me, O, C≡CH, H, H, H, O], [AC 3673; H, CHF ₂ , H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 3674; H, CHF ₂ , H , Me, O, c-Pr , H, H, H, O], [AC3675; H, CHF 2, H, Me, O, OMe, H, H, H, O], [AC3676; H, CHF 2 , H, Me, O, OEt, H, H, H, O], [AC 3677; H, CHF ₂ , H, Me, O, Oi-Pr, H, H, H, O], [AC 3678; H, CHF ₂ , H, Me, O, SMe, H, H, H, O], [AC 3679; H, CHF ₂ , H, Me, O, SE t, H, H, H, O], [AC 3680; H, _{CHF 2, H, Me, O} , CH 2 F, H, H, H, O], [AC3681; H, CHF 2, H, Me, O, CHF 2, H, H, H, O], [AC3682 _{; H, CHF 2, H,} Me, O, CF 3, H, H, H, O], [AC3683; H, CHF 2, H, Me, O, OCH 2 F, H, H, H, O] _{, [AC3684; H, CHF 2} , H, Me, O, OCHF 2, H, H, H, O], [AC3685; H, CHF 2, H, Me, O, OCF 3, H, H, H, O], [AC3686; H, CHF 2, H, Me, O, SCH 2 F, H, H, H, O], [AC3687; H, CHF 2, H, Me, O, SCHF 2, H, H , H, O],

_{[AC3688; H, CHF 2,} H, Me, O, SCF 3, H, H, H, O], [AC3689; H, CHF 2, H, Me, O, CN, H, H, H, O] , [AC 3690; H, CHF ₂ , H, Me, O, NO ₂ , H, H, O], [AC 369 1; H, CHF ₂ , H, Et, O, H, H, H, H, O ], [AC3692; H, CHF 2, H, Et, O, F, H, H, H, O], [AC3693; H, CHF 2, H, Et, O, Cl, H, H, H, O ], [AC3694; H, CHF 2, H, Et, O, Br, H, H, H, O], [AC3695; H, CHF 2, H, Et, O, I, H, H, H, O ], [AC3696; H, CHF 2, H, Et, O, Me, H, H, H, O], [AC3697; H, CHF 2, H, Et, O, Et, H, H, H, O ], [AC3698; H, CHF 2, H, Et, O, Pr, H, H, H, O], [AC3699; H, CHF 2, H, Et, O, i-Pr, H, H, H , O], [AC3700; H , CHF 2, H, Et, O, CH = CH 2, H, H, H, O], [AC3701; H, CHF 2, H, Et, O, C (CH 3 ) = CH ₂ , H, H, H, O], [AC 3702; H, CHF ₂ , H, Et, O, C≡CH, H, H, H, O], [AC 3703; H, CHF ₂ , H , Et, O, C≡CCH ₃ , H, H, H, O], [AC 3704; H, CHF ₂ , H, Et, O, c-Pr, H, H, H, O], [AC 3705; H _{, CHF 2, H, Et,} O, OMe, H, H, H, O], [AC3706; H, CHF 2, H, Et, O, OEt, H, H, H, O], [AC3707; H , CHF ₂ , H, Et, O, Oi-Pr, H, H, H, O], [AC 3708; H, CHF ₂ , H, Et, O, SMe, H, H, H, O], [AC 3709 _{; H, CHF 2, H,} Et, O, SEt, H, H, H, O], [AC3710; H, CHF 2, H, Et, O, CH 2 F, H, H, H, O], _{[AC3711; H, CHF 2,} H, Et, O, CHF 2, H, H, H, O], [AC3712; H, CHF 2, H, Et, O, CF 3, H, H, H, O ], [AC3713; H, CHF 2, H, Et, O, OCH 2 F, H, H, H, O], [AC _{3714; H, CHF 2, H} , Et, O, OCHF 2, H, H, H, O], [AC3715; H, CHF 2, H, Et, O, OCF 3, H, H, H, O] _{, [AC3716; H, CHF 2} , H, Et, O, SCH 2 F, H, H, H, O], [AC3717; H, CHF 2, H, Et, O, SCHF 2, H, H, H , O], [AC3718; H , CHF 2, H, Et, O, SCF 3, H, H, H, O], [AC3719; H, CHF 2, H, Et, O, CN, H, H, H, O], [AC3720; H, CHF 2, H, Et, O, NO 2, H, H, H, O], [AC3721; H, CHF 2, H, Pr, O, H, H, H , H, O], [AC3722 ; H, CHF 2, H, Pr, O, F, H, H, H, O], [AC3723; H, CHF 2, H, Pr, O, Cl, H, H , H, O], [AC3724 ; H, CHF 2, H, Pr, O, Br, H, H, H, O], [AC3725; H, CHF 2, H, Pr, O, I, H, H , H, O], [AC3726 ; H, CHF 2, H, Pr, O, Me, H, H, H, O], [AC3727; H, CHF 2, H, Pr, O, Et, H, H , H, O], [AC3728 ; H, CHF 2, H, Pr, O, Pr, H, H, H, O], [AC3729; H, CHF 2, H, Pr, O, i-Pr, H , H, H, O], [AC3730; H, CHF 2, H, Pr, O, CH = CH 2, H, H, H, O], [AC3731; H, CHF 2, H, Pr, O, _{C (CH 3) = CH 2} , H, H, H, O], [AC3732; H, CHF 2, H, Pr, O, C≡CH, H, H, H, O], [AC3733; H, CHF ₂ , H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 3734; H, CHF ₂ , H, Pr, O, c-Pr, H, H, H, O], _{[AC3735; H, CHF 2,} H, Pr, O, OMe, H, H, H, O], [AC3736; H, CHF 2, H, Pr, O, OEt, H, H, H, O], _{[AC3737; H, CHF 2,} H, Pr, O, Oi-Pr, H, H, H, O], [AC3738; H, CHF 2, H, Pr, O, SMe, H, H, H, O ], [AC 3739; H, CHF ₂ , H, Pr, O, SE t, H, H, H, O], [AC _{3740; H, CHF 2, H} , Pr, O, CH 2 F, H, H, H, O], [AC3741; H, CHF 2, H, Pr, O, CHF 2, H, H, H, O ], [AC3742; H, CHF 2, H, Pr, O, CF 3, H, H, H, O], [AC3743; H, CHF 2, H, Pr, O, OCH 2 F, H, H, H, O], [AC3744; H, CHF 2, H, Pr, O, OCHF 2, H, H, H, O], [AC3745; H, CHF 2, H, Pr, O, OCF 3, H, H, H, O], [ AC3746; H, CHF 2, H, Pr, O, SCH 2 F, H, H, H, O], [AC3747; H, CHF 2, H, Pr, O, SCHF 2 H, H, H, O], [AC 3748; H, CHF ₂ , H, Pr, O, SCF ₃ , H, H, H, O], [AC 3749; H, CHF ₂ , H, Pr, O, CN, H, H, H, O], [AC3750; H, CHF 2, H, Pr, O, NO 2, H, H, H, O], [AC3751; H, CHF 2, H, i-Pr , O, H, H, H , H, O], [AC3752; H, CHF 2, H, i-Pr, O, F, H, H, H, O], [AC3753; H, CHF 2, H , i-Pr, O, Cl, H, H, H, O], [AC 3754; H, CHF ₂ , H, i-Pr, O, Br, H, H, O], [AC 3755; H, CHF ₂ , H, i-Pr, O, I, H, H, H, O], [AC 3756; H, CHF ₂ , H, i-Pr, O, Me, H, H, H, O], [[ _{AC3757; H, CHF 2, H} , i-Pr, O, Et, H, H, H, O], [AC3758; H, CHF 2, H, i-Pr, O, Pr, H, H, H, O, [AC 3759; H, CHF ₂ , H, i-Pr, O, i-Pr, H, H, H, O], [AC 3760; H, CHF ₂ , H, i-Pr, O, CH = _{CH 2, H, H, H} , O], [AC3761; H, CHF 2, H, i-Pr, O, C (CH 3) = CH 2, H, H, H, O], [AC3762; H _{, CHF 2, H, i-} Pr, O, C≡CH, H, H, H, O], [AC3763; H, CHF 2, H, i-Pr, O, C≡CCH 3, H, H, H, O], [AC 3764; H, CHF ₂ , H, i-Pr, O, c-Pr, H, H, H, O], [A _{C3765; H, CHF 2, H} , i-Pr, O, OMe, H, H, H, O], [AC3766; H, CHF 2, H, i-Pr, O, OEt, H, H, H, O], [AC3767; H, CHF 2, H, i-Pr, O, Oi-Pr, H, H, H, O], [AC3768; H, CHF 2, H, i-Pr, O, SMe, H, H, H, O] , [AC3769; H, CHF 2, H, i-Pr, O, SEt, H, H, H, O], [AC3770; H, CHF 2, H, i-Pr, _{O, CH 2 F, H,} H, H, O], [AC3771; H, CHF 2, H, i-Pr, O, CHF 2, H, H, H, O], [AC3772; H, CHF 2 , H, i-Pr, O , CF 3, H, H, H, O], [AC3773; H, CHF 2, H, i-Pr, O, OCH 2 F, H, H, H, O], _{[AC3774; H, CHF 2,} H, i-Pr, O, OCHF 2, H, H, H, O], [AC3775; H, CHF 2, H, i-Pr, O, OCF 3, H, H , H, O], [AC 3776; H, CHF ₂ , H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 3777; H, CHF ₂ , H, i-Pr, O , SCHF ₂ , H, H, H, O], [AC 3778; H, CHF ₂ , H, i-Pr, O, SCF ₃ , H, H, H, O], [AC 3779; H, CHF ₂ , H , i-Pr, O, CN, H, H, H, H, O], [AC 3780; H, CHF ₂ , H, i-Pr, O, NO ₂ , H, H, H, O], [AC 3781; H _{, CHF 2, H, c-} Pr, O, H, H, H, H, O], [AC3782; H, CHF 2, H, c-Pr, O, F, H, H, H, O], _{[AC3783; H, CHF 2,} H, c-Pr, O, Cl, H, H, H, O], [AC3784; H, CHF 2, H, c-Pr, O, Br, H, H, H , O], [AC3785; H , CHF 2, H, c-Pr, O, I, H, H, H, O], [AC3786; H, CHF 2, H, c-Pr, O, Me, H , H, H, O], [AC 3787; H, CHF ₂ , H, c-Pr, O, Et, H, H, H, O],

_{[AC3788; H, CHF 2,} H, c-Pr, O, Pr, H, H, H, O], [AC3789; H, CHF 2, H, c-Pr, O, i-Pr, H, H , H, O], [AC3790 ; H, CHF 2, H, c-Pr, O, CH = CH 2, H, H, H, O], [AC3791; H, CHF 2, H, c-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 3792; H, CHF ₂ , H, c-Pr, O, C≡CH, H, H, H, O], [[ _{AC3793; H, CHF 2, H} , c-Pr, O, C≡CCH 3, H, H, H, O], [AC3794; H, CHF 2, H, c-Pr, O, c-Pr, H , H, H, O], [AC3795; H, CHF 2, H, c-Pr, O, OMe, H, H, H, O], [AC3796; H, CHF 2, H, c-Pr, O , OEt, H, H, H , O], [AC3797; H, CHF 2, H, c-Pr, O, Oi-Pr, H, H, H, O], [AC3798; H, CHF 2, H , c-Pr, O, SMe , H, H, H, O], [AC3799; H, CHF 2, H, c-Pr, O, SEt, H, H, H, O], [AC3800; H, _{CHF 2, H, c-Pr} , O, CH 2 F, H, H, H, O], [AC3801; H, CHF 2, H, c-Pr, O, CHF 2, H, H, H, O ], [AC3802; H, CHF 2, H, c-Pr, O, CF 3, H, H, H, O], [AC3803; H, CHF 2, H, c-Pr, O, OCH 2 F, H, H, H, O] , [AC3804; H, CHF 2, H, c-Pr, O, OCHF 2, H, H, H, O], [AC3805; H, CHF 2, H, c-Pr _{, O, OCF 3, H,} H, H, O], [AC3806; H, CHF 2, H, c-Pr, O, SCH 2 F, H, H, H, O], [AC3807; H, CHF _{2, H, c-Pr,} O, SCHF 2, H, H, H, O], [AC3808; H, CHF 2, H, c-Pr, O, SCF 3, H, H, H, O], _{[AC3809; H, CHF 2,} H, c-Pr, O, CN, H, H, H, O], [AC3810; H, CHF 2, H, c-Pr, O, NO 2, H, H, H, O], [AC3811; H, CHF 2, H, SMe, O, H, H, H, H, O], [AC3812 _{; H, CHF 2, H,} SMe, O, F, H, H, H, O], [AC3813; H, CHF 2, H, SMe, O, Cl, H, H, H, O], [AC3814 _{; H, CHF 2, H,} SMe, O, Br, H, H, H, O], [AC3815; H, CHF 2, H, SMe, O, I, H, H, H, O], [AC3816 _{; H, CHF 2, H,} SMe, O, Me, H, H, H, O], [AC3817; H, CHF 2, H, SMe, O, Et, H, H, H, O], [AC3818 _{; H, CHF 2, H,} SMe, O, Pr, H, H, H, O], [AC3819; H, CHF 2, H, SMe, O, i-Pr, H, H, H, O], _{[AC3820; H, CHF 2,} H, SMe, O, CH = CH 2, H, H, H, O], [AC3821; H, CHF 2, H, SMe, O, C (CH 3) = CH 2 , H, H, H, O ], [AC3822; H, CHF 2, H, SMe, O, C≡CH, H, H, H, O], [AC3823; H, CHF 2, H, SMe, O , C≡CCH ₃ , H, H, H, O], [AC 3824; H, CHF ₂ , H, SMe, O, c-Pr, H, H, H, O], [AC 3825; H, CHF ₂ , H, SMe, O, OMe, H, H, H, O], [AC3826; H, CHF 2, H, SMe, O, OEt, H, H, H, O], [AC3827; H, CHF 2, H, SMe, O, Oi- Pr, H, H, H, O], [AC3828; H, CHF 2, H, SMe, O, SMe, H, H, H, O], [AC3829; H, CHF _{2, H, SMe, O,} SEt, H, H, H, O], [AC3830; H, CHF 2, H, SMe, O, CH 2 F, H, H, H, O], [AC3831; H _{, CHF 2, H, SMe,} O, CHF 2, H, H, H, O], [AC3832; H, CHF 2, H, SMe, O, CF 3, H, H, H, O], [AC3833 _{; H, CHF 2, H,} SMe, O, OCH 2 F, H, H, H, O], [AC3834; H, CHF 2, H, SMe, O, OCHF 2, H, H, H, O] _{, [AC3835; H, CHF 2} , H, SMe, O, OCF 3, H, H, H, O], [AC3836; H, CHF 2, H, SMe, O, SCH 2 F, H, H, H , O], [AC 3837; H, CHF ₂ , H, SMe, O, SCHF ₂ , H, H, H, O], [AC 3838; H, CHF ₂ , H, SMe, O, SCF ₃ , H, H, H, O], [AC 3839; H _{, CHF 2, H, SMe,} O, CN, H, H, H, O], [AC3840; H, CHF 2, H, SMe, O, NO 2, H, H, H, O], [AC3841; _{H, CHF 2, H, OMe} , O, H, H, H, H, O], [AC3842; H, CHF 2, H, OMe, O, F, H, H, H, O], [AC3843; _{H, CHF 2, H, OMe} , O, Cl, H, H, H, O], [AC3844; H, CHF 2, H, OMe, O, Br, H, H, H, O], [AC3845; _{H, CHF 2, H, OMe} , O, I, H, H, H, O], [AC3846; H, CHF 2, H, OMe, O, Me, H, H, H, O], [AC3847; _{H, CHF 2, H, OMe} , O, Et, H, H, H, O], [AC3848; H, CHF 2, H, OMe, O, Pr, H, H, H, O], [AC3849; _{H, CHF 2, H, OMe} , O, i-Pr, H, H, H, O], [AC3850; H, CHF 2, H, OMe, O, CH = CH 2, H, H, H, O ], [AC3851; H, CHF 2, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC3852; H, CHF 2, H, OMe, O, C≡ CH, H, H, H, O], [AC3853; H, CHF 2, H, OMe, O, C≡CCH 3, H, H, H, O], [AC3854; H, CHF 2, H, OMe , O, c-Pr, H , H, H, O], [AC3855; H, CHF 2, H, OMe, O, OMe, H, H, H, O], [AC3856; H, CHF 2, H , OMe, O, OEt, H, H, H, O], [AC 3857; H, CHF ₂ , H, OMe, O, Oi-Pr, H, H, H, O], [AC 3858; H, CHF ₂ , H, OMe, O, SMe, H, H, H, O], [AC 3859; H, CHF ₂ , H, OMe, O, SE t, H, H, H, O], [AC 3860; H, CHF ₂ , H, OMe, O, CH 2 F, H, H, H, O], [AC3861; H, CHF 2, H, OMe, O, CHF 2, H, H, H, O], [AC3862; H , CHF ₂ , H, OMe, O, CF ₃ , H, H, H, O ], [AC3863; H, CHF 2, H, OMe, O, OCH 2 F, H, H, H, O], [AC3864; H, CHF 2, H, OMe, O _{, OCHF 2, H, H,} H, O], [AC3865; H, CHF 2, H, OMe, O, OCF 3, H, H, H, O], [AC3866; H, CHF 2, H, OMe , O, SCH ₂ F, H, H, H, O], [AC3867; H, CHF ₂ , H, OMe, O, SCHF ₂ , H, H, H, O], [AC 3868; H, CHF ₂ , _{H, OMe, O, SCF 3} , H, H, H, O], [AC3869; H, CHF 2, H, OMe, O, CN, H, H, H, O], [AC3870; H, CHF 2 , H, OMe, O, NO ₂ , H, H, H, O], [AC 3871; H, CHF ₂ , H, F, O, H, H, H, H, O], [AC 3872; H, CHF _{2, H, F, O,} F, H, H, H, O], [AC3873; H, CHF 2, H, F, O, Cl, H, H, H, O], [AC3874; H, CHF _{2, H, F, O,} Br, H, H, H, O], [AC3875; H, CHF 2, H, F, O, I, H, H, H, O], [AC3876; H, CHF ₂ , H, F, O, Me, H, H, H, O, [AC 3877; H, CHF ₂ , H, F, O, Et, H, H, O], [AC 3878; H, CHF ₂ , H, F, O, Pr, H, H, H, O], [AC 3879; H, CHF ₂ , H, F, O, i-Pr, H, H, H, O], [AC 3880; H _{, CHF 2, H, F,} O, CH = CH 2, H, H, H, O], [AC3881; H, CHF 2, H, F, O, C (CH 3) = CH 2, H, H , H, O], [AC3882 ; H, CHF 2, H, F, O, C≡CH, H, H, H, O], [AC3883; H, CHF 2, H, F, O, C≡CCH _{3, H, H, H,} O], [AC3884; H, CHF 2, H, F, O, c-Pr, H, H, H, O], [AC3885; H, CHF 2, H, F, O, OMe, H, H, H, O], [AC 3886; H, CHF ₂ , H, F, O, OE t, H, H, H, O], [AC 3887; H, CHF ₂ , H, F, O, Oi-Pr, H, H, H, O],

_{[AC3888; H, CHF 2,} H, F, O, SMe, H, H, H, O], [AC3889; H, CHF 2, H, F, O, SEt, H, H, H, O], _{[AC3890; H, CHF 2,} H, F, O, CH 2 F, H, H, H, O], [AC3891; H, CHF 2, H, F, O, CHF 2, H, H, H, O], [AC3892; H, CHF 2, H, F, O, CF 3, H, H, H, O], [AC3893; H, CHF 2, H, F, O, OCH 2 F, H, H , H, O], [AC3894 ; H, CHF 2, H, F, O, OCHF 2, H, H, H, O], [AC3895; H, CHF 2, H, F, O, OCF 3, H , H, H, O], [AC3896; H, CHF 2, H, F, O, SCH 2 F, H, H, H, O], [AC3897; H, CHF 2, H, F, O, SCHF ₂ , H, H, H, O], [AC 3898; H, CHF ₂ , H, F, O, SCF ₃ , H, H, H, O], [AC 3899; H, CHF ₂ , H, F, O , CN, H, H, H, O], [AC 3900; H, CHF ₂ , H, F, O, NO ₂ , H, H, H, O], [AC 3901; H, CHF ₂ , H, Cl, O, H, H, H, H, O], [AC3902; H, CHF 2, H, Cl, O, F, H, H, H, O], [AC3903; H, CHF 2, H, Cl, O, Cl, H, H, H, O], [AC3904; H, CHF 2, H, Cl, O, Br, H, H, H, O], [AC3905; H, CHF 2, H, Cl, O, I, H, H, H, O], [AC3906; H, CHF 2, H, Cl, O, Me, H, H, H, O], [AC3907; H, CHF 2, H, Cl, O, Et, H, H, H, O], [AC3908; H, CHF 2, H, Cl, O, Pr, H, H, H, O], [AC3909; H, CHF 2, H, Cl, O, i-Pr, H, H, H, O], [AC3910; H, CHF 2, H, Cl, O, CH = CH 2, H, H, H, O], [AC3911; H, CHF 2 , H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC3912; H, CHF 2, H, Cl, O, C≡CH, H, H, H, O ], [AC3913; H, CHF 2, H, Cl, O, C≡CCH 3, H, H, H, O], [AC3 _{914; H, CHF 2, H} , Cl, O, c-Pr, H, H, H, O], [AC3915; H, CHF 2, H, Cl, O, OMe, H, H, H, O] _{, [AC3916; H, CHF 2} , H, Cl, O, OEt, H, H, H, O], [AC3917; H, CHF 2, H, Cl, O, Oi-Pr, H, H, H, O], [AC3918; H, CHF 2, H, Cl, O, SMe, H, H, H, O], [AC3919; H, CHF 2, H, Cl, O, SEt, H, H, H, O], [AC3920; H, CHF 2, H, Cl, O, CH 2 F, H, H, H, O], [AC3921; H, CHF 2, H, Cl, O, CHF 2, H, H , H, O], [AC3922 ; H, CHF 2, H, Cl, O, CF 3, H, H, H, O], [AC3923; H, CHF 2, H, Cl, O, OCH 2 F, H, H, H, O] , [AC3924; H, CHF 2, H, Cl, O, OCHF 2, H, H, H, O], [AC3925; H, CHF 2, H, Cl, O, OCF ₃ , H, H, H, O], [AC 3926; H, CHF ₂ , H, Cl, O, SCH ₂ F, H, H, H, O], [AC 3 927; H, CHF ₂ , H, Cl, O, SCHF ₂ , H, H, H, O], [AC3928; H, CHF ₂ , H, Cl, O, SCF ₃ , H, H, H, O], [AC 3929; H, CHF ₂ , H, H, Cl, O, CN, H, H, H, O], [AC3930; H, CHF 2, H, Cl, O, NO 2, H, H, H, O], [AC3931; H, CHF 2, H , Br, O, H, H , H, H, O], [AC3932; H, CHF 2, H, Br, O, F, H, H, H, O], [AC3933; H, CHF 2, H , Br, O, Cl, H , H, H, O], [AC3934; H, CHF 2, H, Br, O, Br, H, H, H, O], [AC3935; H, CHF 2, H , Br, O, I, H, H, H, O], [AC 3936; H, CHF ₂ , H, Br, O, Me, H, H, H, O], [AC 3937; H, CHF ₂ , H , Br, O, Et, H , H, H, O], [AC3938; H, CHF 2, H, Br, O, Pr, H, H, H, O], [AC3939; H, CHF 2, H , Br, O, i-Pr, H, H, H, O], [AC 3940; H, CHF ₂ , H , Br, O, CH = CH 2, H, H, H, O], [AC3941; H, CHF 2, H, Br, O, C (CH 3) = CH 2, H, H, H, O] _{, [AC3942; H, CHF 2} , H, Br, O, C≡CH, H, H, H, O], [AC3943; H, CHF 2, H, Br, O, C≡CCH 3, H, H , H, O], [AC 3944; H, CHF ₂ , H, Br, O, c-Pr, H, H, H, O], [AC 3945; H, CHF ₂ , H, Br, O, OMe, H , H, H, O], [AC3946; H, CHF 2, H, Br, O, OEt, H, H, H, O], [AC3947; H, CHF 2, H, Br, O, Oi-Pr , H, H, H, O ], [AC3948; H, CHF 2, H, Br, O, SMe, H, H, H, O], [AC3949; H, CHF 2, H, Br, O, SEt , H, H, H, O ], [AC3950; H, CHF 2, H, Br, O, CH 2 F, H, H, H, O], [AC3951; H, CHF 2, H, Br, O _{, CHF 2, H, H,} H, O], [AC3952; H, CHF 2, H, Br, O, CF 3, H, H, H, O], [AC3953; H, CHF 2, H, Br , O, OCH ₂ F, H, H, H, O, [AC 3954; H, CHF ₂ , H, Br, O, OCHF ₂ , H, H, H, O], [AC 3 955; H, CHF ₂ , _{H, Br, O, OCF 3} , H, H, H, O], [AC3956; H, CHF 2, H, Br, O, SCH 2 F, H, H, H, O], [AC3957; H, _{CHF 2, H, Br, O} , SCHF 2, H, H, H, O], [AC3958; H, CHF 2, H, Br, O, SCF 3, H, H, H, O], [AC3959; _{H, CHF 2, H, Br} , O, CN, H, H, H, O], [AC3960; H, CHF 2, H, Br, O, NO 2, H, H, H, O], [AC3961 _{; H, CF 3, H,} H, O, H, H, H, H, O], [AC3962; H, CF 3, H, H, O, F, H, H, H, O], [AC3963 _{; H, CF 3, H,} H, O, Cl, H, H, H, O], [AC3964; H, CF 3, H, H, O, Br, H, H, H, O], [AC3965 _{; H, CF 3, H,} H, O, I, H, H, H, O], [AC3966; H, CF 3 , H, H, O, Me , H, H, H, O], [AC3967; H, CF 3, H, H, O, Et, H, H, H, O], [AC3968; H, CF 3 , H, H, O, Pr, H, H, H, O], [AC 3969; H, CF ₃ , H, H, O, i-Pr, H, H, H, O], [AC 3 970; H, _{CF 3, H, H, O} , CH = CH 2, H, H, H, O], [AC3971; H, CF 3, H, H, O, C (CH 3) = CH 2, H, H, H, O], [AC ₃ 972; H, CF ₃ , H, H, O, C≡CH, H, H, H, O], [AC ₃ 973; H, CF ₃ , H, H, O, C≡ CCH ₃ , H, H, H, O ], [AC3974; H, CF 3, H, H, O, c-Pr, H, H, H, O], [AC3975; H, CF 3, H, H, O , OMe, H, H, H , O], [AC3976; H, CF 3, H, H, O, OEt, H, H, H, O], [AC3977; H, CF 3, H, H, O , Oi-Pr, H, H, H, O], [AC 3978; H, CF ₃ , H, H, O, S Me, H, H, H, O], [AC 3979; H, CF ₃ , H, H , O, SEt, H, H, H, O], [AC ₃ 980; H, CF ₃ , H, H, O, CH ₂ F, H, H, H, O], [AC 3981; H, CF ₃ , H _{, H, O, CHF 2,} H, H, H, O], [AC3982; H, CF 3, H, H, O, CF 3, H, H, H, O], [AC3983; H, CF 3 , H, H, O, OCH 2 F, H, H, H, O], [AC3984; H, CF 3, H, H, O, OCHF 2, H, H, H, O], [AC3985; H , CF ₃ , H, H, O, OCF ₃ , H, H, H, O], [AC 3986; H, CF ₃ , H, H, O, SCH ₂ F, H, H, H, O],

_{[AC3987; H, CF 3,} H, H, O, SCHF 2, H, H, H, O], [AC3988; H, CF 3, H, H, O, SCF 3, H, H, H, O ], [AC3989; H, CF 3, H, H, O, CN, H, H, H, O], [AC3990; H, CF 3, H, H, O, NO 2, H, H, H, O], [AC3991; H, CF 3, H, Me, O, H, H, H, H, O], [AC3992; H, CF 3, H, Me, O, F, H, H, H, O], [AC3993; H, CF 3, H, Me, O, Cl, H, H, H, O], [AC3994; H, CF 3, H, Me, O, Br, H, H, H, O, [AC 3995; H, CF ₃ , H, Me, O, I, H, H, O], [AC 3996; H, CF ₃ , H, Me, O, Me, H, H, H, H, O], [AC3997; H, CF 3, H, Me, O, Et, H, H, H, O], [AC3998; H, CF 3, H, Me, O, Pr, H, H, H, O], [AC3999; H, CF 3, H, Me, O, i-Pr, H, H, H, O], [AC4000; H, CF 3, H, Me, O, CH = CH 2, H , H, H, O], [AC4001; H, CF 3, H, Me, O, C (CH 3) = CH 2, H, H, H, O], [AC4002; H, CF 3, H, Me, O, C≡CH, H, H, H, O, [AC 4003; H, CF ₃ , H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 4004; H, _{CF 3, H, Me, O} , c-Pr, H, H, H, O], [AC4005; H, CF 3, H, Me, O, OMe, H, H, H, O], [AC4006; _{H, CF 3, H, Me} , O, OEt, H, H, H, O], [AC4007; H, CF 3, H, Me, O, Oi-Pr, H, H, H, O], [ _{AC4008; H, CF 3, H} , Me, O, SMe, H, H, H, O], [AC4009; H, CF 3, H, Me, O, SEt, H, H, H, O], [ AC 4010; H, CF ₃ , H, Me, O, CH ₂ F, H, H, H, O], [AC 4011; H, CF ₃ , H, Me, O, CHF ₂ , H, H, H, O H, CF ₃ , H, Me, O, CF ₃ , H, H, H, O], [AC 4013; H, CF ₃ , H, Me, O, OCH ₂ F, H, H] H, H, O], [AC 4014; H, CF ₃ , H, Me, O, OCHF ₂ , H, H, H, O], [AC 4015; H, CF ₃ , H, Me, O, OCF ₃ , H, H, H, O] , [AC4016; H, CF 3, H, Me, O, SCH 2 F, H, H, H, O], [AC4017; H, CF 3, H, Me, O, SCHF ₂ , H, H, H, O], [AC 4018; H, CF ₃ , H, Me, O, SCF ₃ , H, H, H, O], [AC 4019; H, CF ₃ , H, Me, O, CN, H, H, H, O], [AC 4020; H, CF ₃ , H, Me, O, NO ₂ , H, H, H, O], [AC 4021; H, CF ₃ , H, Et , O, H, H, H, H, O, [AC 4022; H, CF ₃ , H, Et, O, F, H, H, H, O], [AC 4023; H, CF ₃ , H, Et , O, Cl, H, H, H, O, [AC 4024; H, CF ₃ , H, Et, O, Br, H, H, H, O], [AC 4025; H, CF ₃ , H, Et , O, I, H, H, H, O, [AC 4026; H, CF ₃ , H, Et, O, Me, H, H, H, O], [AC 4027; H, CF ₃ , H, Et , O, Et, H, H, H, O, [AC 4028; H, CF ₃ , H, Et, O, Pr, H, H, H, O], [AC 4029; H, CF ₃ , H, Et , O, i-Pr, H, H, H, O], [AC 4030; H, CF ₃ , H, Et, O, CHCHCH ₂ , H, H, H, O], [AC 4031; H, CF _{3, H, Et, O,} C (CH 3) = CH 2, H, H, H, O], [AC4032; H, CF 3, H, Et, O, C≡CH, H, H, H, H, CF ₃ , H, Et, O, C≡CCH ₃ , H, H, H, O], [AC 4034; H, CF ₃ , H, Et, O, c-Pr, H , H, H, O], [AC4035; H, CF 3, H, Et, O, OMe, H, H, H, O], [AC4036; H, CF 3, H, Et, O, OEt, H , H, H, O], [AC4037; H, CF 3, H, Et, O, Oi-Pr, H, H, H, O], [AC4038; H, CF 3, H, Et, O, SMe , H, H, H, O], [AC 4039; H, CF ₃ , H, Et, O, SE t, H, H, H, O], [AC 4040; H, CF ₃ , H, E _{t, O, CH 2 F,} H, H, H, O], [AC4041; H, CF 3, H, Et, O, CHF 2, H, H, H, O], [AC4042; H, CF 3 , H, Et, O, CF 3, H, H, H, O], [AC4043; H, CF 3, H, Et, O, OCH 2 F, H, H, H, O], [AC4044; H , CF ₃ , H, Et, O, OCHF ₂ , H, H, H, O], [AC 4045; H, CF ₃ , H, Et, O, OCF ₃ , H, H, H, O], [AC 4046 H, CF ₃ , H, Et, O, SCH ₂ F, H, H, H, O], [AC 4047; H, CF ₃ , H, Et, O, SCHF ₂ , H, H, H, O] , [AC 4048; H, CF ₃ , H, Et, O, SCF ₃ , H, H, H, O], [AC 4049; H, CF ₃ , H, Et, O, CN, H, H, H, O ], [AC4050; H, CF 3, H, Et, O, NO 2, H, H, H, O], [AC4051; H, CF 3, H, Pr, O, H, H, H, H, O], [AC4052; H, CF 3, H, Pr, O, F, H, H, H, O], [AC4053; H, CF 3, H, Pr, O, Cl, H, H, H, O], [AC4054; H, CF 3, H, Pr, O, Br, H, H, H, O], [AC4055; H, CF 3, H, Pr, O, I, H, H, H, H, CF ₃ , H, Pr, O, Me, H, H, H, O], [AC 4057; H, CF ₃ , H, Pr, O, Et, H, H, H, O], [AC 4056; O], [AC 4058; H, CF ₃ , H, Pr, O, Pr, H, H, H, O], [AC 4059; H, CF ₃ , H, Pr, O, i-Pr, H, H, H, O], [AC 4060; H, CF ₃ , H, Pr, O, CHCHCH ₂ , H, H, H, O], [AC 4061; H, CF ₃ , H, Pr, O, C (CH (CH) _{3) = CH 2, H,} H, H, O], [AC4062; H, CF 3, H, Pr, O, C≡CH, H, H, H, O], [AC4063; H, CF 3, H, Pr, O, C≡CCH ₃ , H, H, H, O], [AC 4064; H, CF ₃ , H, Pr, O, c-Pr, H, H, H, O], [AC 4065; _{H, CF 3, H, Pr} , O, OMe, H, H, H, O], [AC4066; H, CF 3, H, Pr, O, OEt, H, H, H, O] , [AC 4067; H, CF ₃ , H, Pr, O, Oi-Pr, H, H, H, O], [AC 4068; H, CF ₃ , H, Pr, O, S Me, H, H, H, O, [AC 4069; H, CF ₃ , H, Pr, O, SE t, H, H, H, O], [AC 4070; H, CF ₃ , H, Pr, O, CH ₂ F, H, H, H, O], [AC4071; H, CF 3, H, Pr, O, CHF 2, H, H, H, O], [AC4072; H, CF 3, H, Pr, O, CF 3, H, H, H, O], [AC 4073; H, CF ₃ , H, Pr, O, OCH ₂ F, H, H, H, O], [AC 4074; H, CF ₃ , H, Pr, O, OCHF ₂ H, H, H, O], [AC 4075; H, CF ₃ , H, Pr, O, OCF ₃ , H, H, H, O], [AC 4076; H, CF ₃ , H, Pr, O, SCH ₂ F, H, H, H, O], [AC 4077; H, CF ₃ , H, Pr, O, SCHF ₂ , H, H, H, O], [AC 4078; H, CF ₃ , H, Pr , O, SCF ₃ , H, H, H, O, [AC 4079; H, CF ₃ , H, Pr, O, CN, H, H, H, O], [AC 4080; H, CF ₃ , H, _{Pr, O, NO 2, H} , H, H, O], [AC4081; H, CF 3, H, i-Pr, O, H, H, H, H, O], [AC4082; H, CF 3 , H, i-Pr, O , F, H, H, H, O], [AC4083; H, CF 3, H, i-Pr, O, Cl, H, H, H, O], [AC4084; _{H, CF 3, H, i} -Pr, O, Br, H, H, H, O], [AC4085; H, CF 3, H, i-Pr, O, I, H, H, H, O] , [AC 4086; H, CF ₃ , H, i-Pr, O, Me, H, H, H, O],

[AC 4087; H, CF ₃ , H, i-Pr, O, Et, H, H, H, O], [AC 4088; H, CF ₃ , H, i-Pr, O, Pr, H, H, H , O], [AC4089; H , CF 3, H, i-Pr, O, i-Pr, H, H, H, O], [AC4090; H, CF 3, H, i-Pr, O, CH = CH ₂ , H, H, H, O], [AC 4091; H, CF ₃ , H, i-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 4092; _{H, CF 3, H, i} -Pr, O, C≡CH, H, H, H, O], [AC4093; H, CF 3, H, i-Pr, O, C≡CCH 3, H, H , H, O], [AC4094 ; H, CF 3, H, i-Pr, O, c-Pr, H, H, H, O], [AC4095; H, CF 3, H, i-Pr, O , OMe, H, H, H , O], [AC4096; H, CF 3, H, i-Pr, O, OEt, H, H, H, O], [AC4097; H, CF 3, H, i -Pr, O, Oi-Pr, H, H, H, O], [AC 4098; H, CF ₃ , H, i-Pr, O, SMe, H, H, H, O], [AC 4099; H, _{CF 3, H, i-Pr} , O, SEt, H, H, H, O], [AC4100; H, CF 3, H, i-Pr, O, CH 2 F, H, H, H, O] _{, [AC4101; H, CF 3} , H, i-Pr, O, CHF 2, H, H, H, O], [AC4102; H, CF 3, H, i-Pr, O, CF 3, H, H, H, O], [ AC4103; H, CF 3, H, i-Pr, O, OCH 2 F, H, H, H, O], [AC4104; H, CF 3, H, i-Pr, _{O, OCHF 2, H, H} , H, O], [AC4105; H, CF 3, H, i-Pr, O, OCF 3, H, H, H, O], [AC4106; H, CF 3, H, i-Pr, O, SCH ₂ F, H, H, H, O], [AC 4107; H, CF ₃ , H, i-Pr, O, SCHF ₂ , H, H, H, O], [[ _{AC4108; H, CF 3, H} , i-Pr, O, SCF 3, H, H, H, O], [AC4109; H, CF 3, H, i-Pr, O, CN, H, H, H H, CF ₃ , H, i-Pr, O, NO ₂ , H, H, H, O], [AC 4111; H, CF ₃ , H, c-Pr, O, H, H, H, H, O], [ AC4112; H, CF 3, H, c-Pr, O, F, H, H, H, O], [AC4113; H, CF 3, H, c-Pr, O, Cl, H, H, H, O], [AC4114; H, CF 3, H, c-Pr, O, Br, H, H, H, O], [AC4115; H, CF 3, H, c- Pr, O, I, H, H, H, O, [AC 4116; H, CF ₃ , H, c-Pr, O, Me, H, H, O], [AC 4 117; H, CF ₃ , H, c-Pr, O, Et, H, H, H, O], [AC 4118; H, CF ₃ , H, c-Pr, O, Pr, H, H, H, O], [AC 4119; H _{, CF 3, H, c-} Pr, O, i-Pr, H, H, H, O], [AC4120; H, CF 3, H, c-Pr, O, CH = CH 2, H, H, H, O], [AC 4121; H, CF ₃ , H, c-Pr, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 4122; H, CF ₃ , H, c -Pr, O, C≡CH, H, H, H, O], [AC 4123; H, CF ₃ , H, c-Pr, O, C≡CCH ₃ , H, H, H, O], [AC 4124 _{; H, CF 3, H,} c-Pr, O, c-Pr, H, H, H, O], [AC4125; H, CF 3, H, c-Pr, O, OMe, H, H, H , O], [AC4126; H , CF 3, H, c-Pr, O, OEt, H, H, H, O], [AC4127; H, CF 3, H, c-Pr, O, Oi-Pr , H, H, H, O ], [AC4128; H, CF 3, H, c-Pr, O, SMe, H, H, H, O], [AC4129; H, CF 3, H, c-Pr , O, SEt, H, H, H, O], [AC 4130; H, CF ₃ , H, c-Pr, O, CH ₂ F, H, H, O], [AC 4131; H, CF ₃ , H, c-Pr, O , CHF 2, H, H, H, O], [AC4132; H, CF 3, H, c-Pr, O, CF 3, H, H, H, O], [ _{AC4133; H, CF 3, H} , c-Pr, O, OCH 2 F, H, H, H, O], [AC4134; H, CF 3, H, c-Pr, O, OCHF 2, H, H , H, O], [AC4135 ; H, CF 3, H, c-Pr, O, OCF 3, H, H, H, O], [AC4136; H, CF 3, H, c-Pr, O, SCH ₂ F, H, H, H, O] _{, [AC4137; H, CF 3} , H, c-Pr, O, SCHF 2, H, H, H, O], [AC4138; H, CF 3, H, c-Pr, O, SCF 3, H, H, H, O], [ AC4139; H, CF 3, H, c-Pr, O, CN, H, H, H, O], [AC4140; H, CF 3, H, c-Pr, O, _{NO 2, H, H, H} , O], [AC4141; H, CF 3, H, SMe, O, H, H, H, H, O], [AC4142; H, CF 3, H, SMe, O , F, H, H, H , O], [AC4143; H, CF 3, H, SMe, O, Cl, H, H, H, O], [AC4144; H, CF 3, H, SMe, O , Br, H, H, H, O], [AC 4145; H, CF ₃ , H, SMe, O, I, H, H, H, O], [AC 4146; H, CF ₃ , H, SMe, O , Me, H, H, H, O], [AC 4147; H, CF ₃ , H, SMe, O, Et, H, H, H, O], [AC 4148; H, CF ₃ , H, SMe, O , Pr, H, H, H, O], [AC 4149; H, CF ₃ , H, SMe, O, i-Pr, H, H, H, O], [AC 4150; H, CF ₃ , H, SMe _{, O, CH = CH 2,} H, H, H, O], [AC4151; H, CF 3, H, SMe, O, C (CH 3) = CH 2, H, H, H, O], [ _{AC4152; H, CF 3, H} , SMe, O, C≡CH, H, H, H, O], [AC4153; H, CF 3, H, SMe, O, C≡CCH 3, H, H, H , O], [AC4154; H , CF 3, H, SMe, O, c-Pr, H, H, H, O], [AC4155; H, CF 3, H, SMe, O, OMe, H, H , H, O], [AC4156 ; H, CF 3, H, SMe, O, OEt, H, H, H, O], [AC4157; H, CF 3, H, SMe, O, Oi-Pr, H , H, H, O], [AC4158; H, CF 3, H, SMe, O, SMe, H, H, H, O], [AC4159; H, CF 3, H, SMe, O, SEt, H , H, H, O], [AC4160; H, CF 3, H, SMe, O, CH 2 F, H, H, H, O], [AC4161; H, CF 3, H, SMe, O, CHF _{2, H, H, H,} O], [AC4162; H, CF 3, H, SMe, O, CF 3, H, H, H, O ], [AC4163; H, CF 3, H, SMe, O, OCH 2 F, H, H, H, O], [AC4164; H, CF 3, H, SMe, O, OCHF 2, H, H, H, O], [AC4165; H, CF 3, H, SMe, O, OCF 3, H, H, H, O], [AC4166; H, CF 3, H, SMe, O, SCH 2 F, H , H, H, O], [AC4167; H, CF 3, H, SMe, O, SCHF 2, H, H, H, O], [AC4168; H, CF 3, H, SMe, O, SCF 3 , H, H, H, O ], [AC4169; H, CF 3, H, SMe, O, CN, H, H, H, O], [AC4170; H, CF 3, H, SMe, O, NO ₂ , H, H, H, O], [AC 4171; H, CF ₃ , H, OMe, O, H, H, H, H, O], [AC 4172; H, CF ₃ , H, OMe, O, F, H, H, H, O], [AC4173; H, CF 3, H, OMe, O, Cl, H, H, H, O], [AC4174; H, CF 3, H, OMe, O, br, H, H, H, O], [AC4175; H, CF 3, H, OMe, O, I, H, H, H, O], [AC4176; H, CF 3, H, OMe, O, Me, H, H, H, O], [AC4177; H, CF 3, H, OMe, O, Et, H, H, H, O], [AC4178; H, CF 3, H, OMe, O, Pr, H, H, H, O], [AC4179; H, CF 3, H, OMe, O, i-Pr, H, H, H, O], [AC4180; H, CF 3, H, OMe, _{O, CH = CH 2, H} , H, H, O], [AC4181; H, CF 3, H, OMe, O, C (CH 3) = CH 2, H, H, H, O], [AC4182 H, CF ₃ , H, OMe, O, C≡CH, H, H, H, O], [AC4183; H, CF ₃ , H, OMe, O, C≡CCH ₃ , H, H, H, O, [AC 4184; H, CF ₃ , H, OMe, O, c-Pr, H, H, H, O], [AC 4 185; H, CF ₃ , H, OMe, O, OMe, H, H, H H, O], [AC 4186; H, CF ₃ , H, OMe, O, OEt, H, H, H, O],

_{[AC4187; H, CF 3,} H, OMe, O, Oi-Pr, H, H, H, O], [AC4188; H, CF 3, H, OMe, O, SMe, H, H, H, O ], [AC4189; H, CF 3, H, OMe, O, SEt, H, H, H, O], [AC4190; H, CF 3, H, OMe, O, CH 2 F, H, H, H H, CF ₃ , H, OMe, O, CHF ₂ , H, H, H, O], [AC 4192; H, CF ₃ , H, OMe, O, CF ₃ , H, H , H, O], [AC4193 ; H, CF 3, H, OMe, O, OCH 2 F, H, H, H, O], [AC4194; H, CF 3, H, OMe, O, OCHF 2, H, H, H, O] , [AC4195; H, CF 3, H, OMe, O, OCF 3, H, H, H, O], [AC4196; H, CF 3, H, OMe, O, SCH ₂ F, H, H, H, O], [AC 4197; H, CF ₃ , H, OMe, O, SCHF ₂ , H, H, H, O], [AC 4198; H, CF ₃ , H, OMe, O, SCF ₃ , H, H, H, O], [AC 4199; H, CF ₃ , H, OMe, O, CN, H, H, H, O], [AC 4200; H, CF ₃ , H, OMe , O, NO ₂ , H, H, H, O], [AC 4201; H, CF ₃ , H, F, O, H, H, H, H, O], [AC 4202; H, CF ₃ , H, F, O, F, H, H, H, O], [AC 4203; H, CF ₃ , H, F, O, Cl, H, H, H, O], [AC 4204; H, CF ₃ , H, F, O, Br, H, H, H, O], [AC 4205; H, CF ₃ , H, F, O, I, H, H, H, O], [AC 4206; H, CF ₃ , H, F, O, Me, H, H, H, O], [AC 4207; H, CF ₃ , H, F, O, Et, H, H, H, O], [AC 4208; H, CF ₃ , H, F, O, Pr, H, H, H, O, [AC 4209; H, CF ₃ , H, F, O, i-Pr, H, H, H, O], [AC 4210; H, CF ₃ , H, F, O, CH = CH 2, H, H, H, O], [AC4211; H, CF 3, H, F, O, C (CH 3) = CH 2, H, H, H, O ], [AC 4212; H, CF ₃ , H, F, O, C≡CH, H, H, H, O], [AC 4213; H, CF ₃ , H, F, O, C≡CCH ₃ , H, H, H, O], [AC 4214; H, CF ₃ , H, F, O, c-Pr, H, H, H, O], [AC 4215; H, CF ₃ , H, F, O, OMe , H, H, H, O], [AC4216; H, CF 3, H, F, O, OEt, H, H, H, O], [AC4217; H, CF 3 , H, F, O, Oi -Pr, H, H, H, O], [AC4218; H, CF 3, H, F, O, SMe, H, H, H, O], [AC4219; H, _{CF 3, H, F, O} , SEt, H, H, H, O], [AC4220; H, CF 3, H, F, O, CH 2 F, H, H, H, O], [AC4221; _{H, CF 3, H, F} , O, CHF 2, H, H, H, O], [AC4222; H, CF 3, H, F, O, CF 3, H, H, H, O], [ _{AC4223; H, CF 3, H} , F, O, OCH 2 F, H, H, H, O], [AC4224; H, CF 3, H, F, O, OCHF 2, H, H, H, O ], [AC4225; H, CF 3, H, F, O, OCF 3, H, H, H, O], [AC4226; H, CF 3, H, F, O, SCH 2 F, H, H, H, O], [AC4227; H, CF 3, H, F, O, SCHF 2, H, H, H, O], [AC4228; H, CF 3, H, F, O, SCF 3, H, H, H, O], [ AC4229; H, CF 3, H, F, O, CN, H, H, H, O], [AC4230; H, CF 3, H, F, O, NO 2, H , H, H, O], [AC4231; H, CF 3, H, Cl, O, H, H, H, H, O], [AC4232; H, CF 3, H, Cl, O, F, H , H, H, O], [AC4233; H, CF 3, H, Cl, O, Cl, H, H, H, O], [AC4234; H, CF 3, H, Cl, O, Br, H , H, H, O], [AC4235; H, CF 3, H, Cl, O, I, H, H, H, O], [AC4236; H, CF 3, H, Cl, O, Me, H , H, H, O], [AC4237; H, CF 3, H, Cl, O, Et, H, H, H, O], [AC4238; H, CF 3, H, Cl, O, Pr, H , H, H, O], [AC4239; H, CF 3, H, Cl, O, i-Pr, H, H, H, O], [AC4240; H, CF 3, H, Cl, O, CH = CH ₂ , H, H , H, O], [AC4241 ; H, CF 3, H, Cl, O, C (CH 3) = CH 2, H, H, H, O], [AC4242; H, CF 3, H, Cl, O, C≡CH, H, H, H, O], [AC4243; H, CF ₃ , H, Cl, O, C≡CCH ₃ , H, H, H, O], [AC 4244; H, CF ₃ , H, Cl, O, c -Pr, H, H, H, O], [AC4245; H, CF 3, H, Cl, O, OMe, H, H, H, O], [AC4246; H, _{CF 3, H, Cl, O} , OEt, H, H, H, O], [AC4247; H, CF 3, H, Cl, O, Oi-Pr, H, H, H, O], [AC4248; _{H, CF 3, H, Cl} , O, SMe, H, H, H, O], [AC4249; H, CF 3, H, Cl, O, SEt, H, H, H, O], [AC4250; _{H, CF 3, H, Cl} , O, CH 2 F, H, H, H, O], [AC4251; H, CF 3, H, Cl, O, CHF 2, H, H, H, O], _{[AC4252; H, CF 3,} H, Cl, O, CF 3, H, H, H, O], [AC4253; H, CF 3, H, Cl, O, OCH 2 F, H, H, H, O], [AC4254; H, CF 3, H, Cl, O, OCHF 2, H, H, H, O], [AC4255; H, CF 3, H, Cl, O, OCF 3, H, H, H, O], [AC 4 256; H, CF ₃ , H, Cl, O, SCH ₂ F, H, H, H, O], [AC 4 257; H, CF ₃ , H, Cl, O, SCHF ₂ , H , H, H, O], [AC4258; H, CF 3, H, Cl, O, SCF 3, H, H, H, O], [AC4259; H, CF 3, H, Cl, O, CN, H, H, H, O] , [AC4260; H, CF 3, H, Cl, O, NO 2, H, H, H, O], [AC4261; H, CF 3, H, Br, O, H , H, H, H, O ], [AC4262; H, CF 3, H, Br, O, F, H, H, H, O], [AC4263; H, CF 3, H, Br, O, Cl , H, H, H, O ], [AC4264; H, CF 3, H, Br, O, Br, H, H, H, O], [AC4265; H, CF 3, H, Br, O, I , H, H, H, O], [AC 4266; H, CF ₃ , H, Br, O, Me, H, H, H, O], [AC 4 267; H, CF _{3, H, Br, O,} Et, H, H, H, O], [AC4268; H, CF 3, H, Br, O, Pr, H, H, H, O], [AC4269; H, CF _{3, H, Br, O,} i-Pr, H, H, H, O], [AC4270; H, CF 3, H, Br, O, CH = CH 2, H, H, H, O], [ AC 427 1; H, CF ₃ , H, Br, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 427 2; H, CF ₃ , H, Br, O, C≡CH, H , H, H, O], [AC4273; H, CF 3, H, Br, O, C≡CCH 3, H, H, H, O], [AC4274; H, CF 3, H, Br, O, c-Pr, H, H, H, O], [AC 4275; H, CF ₃ , H, Br, O, OMe, H, H, H, O], [AC 4276; H, CF ₃ , H, Br, O, OEt, H, H, H, O], [AC4277; H, CF 3, H, Br, O, Oi-Pr, H, H, H, O], [AC4278; H, CF 3, H, Br, O, SMe, H, H, H, O, [AC 4279; H, CF ₃ , H, Br, O, SE t, H, H, H, O], [AC 4280; H, CF ₃ , H, _{Br, O, CH 2 F,} H, H, H, O], [AC4281; H, CF 3, H, Br, O, CHF 2, H, H, H, O], [AC4282; H, CF 3 , H, Br, O, CF 3, H, H, H, O], [AC4283; H, CF 3, H, Br, O, OCH 2 F, H, H, H, O], [AC4284; H _{, CF 3, H, Br,} O, OCHF 2, H, H, H, O], [AC4285; H, CF 3, H, Br, O, OCF 3, H, H, H, O],

_{[AC4286; H, CF 3,} H, Br, O, SCH 2 F, H, H, H, O], [AC4287; H, CF 3, H, Br, O, SCHF 2, H, H, H, O], [AC 4288; H, CF ₃ , H, Br, O, SCF ₃ , H, H, H, O], [AC 4 289; H, CF ₃ , H, Br, O, CN, H, H, H H, CF ₃ , H, Br, O, NO ₂ , H, H, H, O], [AC 4291; F, H, H, H, H, O, H, H, H, H , O], [AC4292; F, H, H, H, O, F, H, H, O], [AC 4293; F, H, H, H, O, Cl, H, H, H, O ], [AC 4294; F, H, H, H, O, Br, H, H, O], [AC 4295; F, H, H, H, O, I, H, H, H, O], [AC 4296; F, H, H, H, H, O, Me, H, H, H, O], [AC 4297; F, H, H, H, O, Et, H, H, H, O], [AC 4298 F, H, H, H, H, O, Pr, H, H, H, O], [AC 4299; F, H, H, H, O, i-Pr, H, H, H, O], [AC 4300 ; F, H, H, H , O, CH = CH 2, H, H, H, O], [AC4301; F, H, H, H, O, C (CH 3) = CH 2, H, H , H, O], [AC 4302; F, H, H, H, O, C≡CH, H, H, H, O], [AC 4303; F, H, H, H, O, C≡ CCH ₃ , H, H, H, O], [AC 4304; F, H, H, H, O, c-Pr, H, H, H, O], [AC 4305; F, H, H, H, O, OMe, H, H, H, O], [AC 4306; F, H, H, H, O, OEt, H, H, H, O], [AC 4307; F, H, H, H, O, Oi-Pr, H, H, H, O], [AC 4308; F, H, H, H, O, SMe, H, H, H, O], [AC 4309; F, H, H, H, O, SE t, H, H, H, O], [AC 4310; F, H, H, H, O, CH ₂ F, H, H, H, O], [AC 4311; F, H, H, H, O, CHF ₂ , H , H, H, O], [AC4312; F, H, H, H, O, CF 3, H, H, H, O], [AC4313; F, H, H, H, O, OCH 2 F, H, H, H, O], [AC 4314; F, H, H, H, O, OCHF ₂ , H, H, H, O], [AC 4315; F, H, H, H, O, OCF ₃ , H, H, H, O], [AC 4316; F, H, H, H, O, SCH ₂ F, H, H, H, O], [AC 4317; F, H, H, H, O, SCHF ₂ , H, H , H, O], [AC 4318; F, H, H, H, O, SCF ₃ , H, H, H, O], [AC 4319; F, H, H, H, O, CN, H, H, H, H, O], [AC4320; F, H, H, H, O, NO 2, H, H, H, O], [AC4321; F, H, H, Me, O, H, H, H, H , O], [AC4322; F, H, H, Me, O, F, H, H, O], [AC 4323; F, H, H, Me, O, Cl, H, H, H, O ], [AC 4324; F, H, H, Me, O, Br, H, H, O], [AC 4325; F, H, H, Me, O, I, H, H, H, O], [AC 4326; F, H, H, Me, O, Me, H, H, H, O], [AC 4327; F, H, H, Me, O, Et, H, H, H, O], [AC 4328 F, H, H, Me, O, Pr, H, H, H, O], [AC 4329; F, H, H, Me, O, i-Pr, H, H, H, O], [AC 4330] ; F, H, H, Me , O, CH = CH 2, H, H, H, O], [AC4331; F, H, H, Me, O, C (CH 3) = CH 2, H, H , H, O], [AC4332; F, H, H, Me, O, C≡CH, H, H, H, O], [AC 4333; F, H, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC 4334; F, H, H, Me, O, c-Pr, H, H, H, O], [AC 4335; F, H, H, Me, O, OMe, H, H, H, O], [AC 4336; F, H, H, Me, O, OEt, H, H, H, O], [AC 4337; F, H, H, Me, O, Oi-Pr, H, H, H, O], [AC 4338; F, H, H, Me, O, SMe, H, H, H, O], [AC 4339; F, H, H, Me, O, SE t, H, H, H, O], [ AC4340; F, H, H, Me, O, CH 2 F, H, H, H, O], [AC4341; F, H, H, Me, O, CHF 2, H , H, H, O], [AC4342; F, H, H, Me, O, CF 3, H, H, H, O], [AC4343; F, H, H, Me, O, OCH 2 F, H, H, H, O] , [AC4344; F, H, H, Me, O, OCHF 2, H, H, H, O], [AC4345; F, H, H, Me, O, OCF 3 , H, H, H, O], [AC 4346; F, H, H, Me, O, SCH ₂ F, H, H, H, O], [AC 4347; F, H, H, Me, O, SCHF ₂ , H, H, H, O], [AC 4348; F, H, H, Me, O, SCF ₃ , H, H, H, O], [AC 4349; F, H, H, Me, O, CN , H, H, H, O], [AC 4 350; F, H, H, Me, O, NO ₂ , H, H, H, O], [AC 4351; F, Me, H, Me, O, H, H, H, H, O], [AC4352; F, Me, H, Me, O, F, H, H, H, O], [AC4353; F, Me, H, Me, O, Cl, H, H, H, O], [AC 4354; F, Me, H, Me, O, Br, H, H, H, O], [AC 4355; F, Me, H, Me, O, I, H, H, H, O], [AC 4356; F, Me, H, Me, O, Me, H, H, H, O], [AC 4357; F, Me, H, Me, O, Et, H, H, H, H, O], [AC 4358; F, Me, H, Me, O, Pr, H, H, H, O], [AC 4359; F, Me, H, Me, O, i-Pr, H, H, H, O, [AC 4 360; F, Me, H, Me, O, CHCHCH ₂ , H, H, H, O], [AC4361; F, Me, H, Me, O, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC4362; F, Me, H, Me, O, C≡CH, H, H, H, O], [AC4363; F, Me, H, Me, O, C≡CCH ₃ , H, H, H, O], [AC4364; F, Me, H, Me, O, c-Pr, H, H, H, O], [AC 4365; F, Me, H, Me , O, OMe, H, H, H, O], [AC 4366; F, Me, H, Me, O, OEt, H, H, H, O], [AC 4367; F, Me, H, Me, O , Oi-Pr, H, H, H, O], [AC 4368; F, Me, H, Me, O, SMe, H, H, H, O], [AC 4369; F, Me, H, Me, O , SEt, H, H, H, O], [AC 4370; F, Me, H, Me, O, CH ₂ F, H, H, H, O], [AC 4371; F, Me, H, Me, O _{, CHF 2, H, H,} H, O], [AC4372; F, Me, H, Me, O, CF 3, H, H, H, O], [AC4373; F, Me, H, Me, O , OCH ₂ F, H, H, H, O], [AC 4374; F, Me, H, Me, O, OCHF ₂ , H, H, H, O] , [AC4375; F, Me, H, Me, O, OCF 3, H, H, H, O], [AC4376; F, Me, H, Me, O, SCH 2 F H, H, H, O], [AC 4377; F, Me, H, Me, O, SCHF ₂ , H, H, H, O], [AC 4378; F, Me, H, Me, O, SCF ₃ H, H, H, O], [AC 4379; F, Me, H, Me, O, CN, H, H, H, O], [AC 4380; F, Me, H, Me, O, NO ₂ , H, H, H, O], [AC4381; H, H, F, H, O, H, H, H, H, O], [AC4382; H, H, F, H, O, F, H, H, H, O], [AC4383; H, H, F, H, O, Cl, H, H, H, O], [AC 4384; H, H, F, H, O, Br, H, H, H H, O], [AC 4385; H, H, F, H, O, I, H, H, H, O],

[AC 4 386; H, H, F, H, O, Me, H, H, H, O], [AC 4387; H, H, F, H, O, Et, H, H, H, O], [AC 4388 H, H, F, H, H, O, Pr, H, H, H, O], [AC 4389; H, H, F, H, O, i-Pr, H, H, H, O], [AC 4390 ; H, H, F, H , O, CH = CH 2, H, H, H, O], [AC4391; H, H, F, H, O, C (CH 3) = CH 2, H, H , H, O], [AC4392; H, H, F, H, O, C≡CH, H, H, H, O], [AC4393; H, H, F, H, O, C≡ CCH ₃ , H, H, H, O], [AC 4394; H, H, F, H, O, c-Pr, H, H, H, O], [AC 4395; H, H, F, H, O, OMe, H, H, H, O], [AC 4396; H, H, F, H, O, OEt, H, H, H, O], [AC 4397; H, H, F, H, O, Oi-Pr, H, H, H, O], [AC 4398; H, H, F, H, O, SMe, H, H, H, O], [AC 4399; H, H, F, H, O, SE t, H, H, H, O], [AC 4400; H, H, F, H, O, CH ₂ F, H, H, H, O], [AC 4401; H, H, F, H, O, CHF ₂ , H , H, H, O], [AC4402; H, H, F, H, O, CF 3, H, H, H, O], [AC4403; H, H, F, H, O, OCH 2 F, H, H, H, O], [AC 4404; H, H, F, H, O, OCHF ₂ , H, H, H, O], [AC 4405; H, H, F, H, O, OCF ₃ , H, H, H, O], [AC 4406; H, H, F, H, O, SCH ₂ F, H, H, H, O], [AC 4407; H, H, F, H, O, SCHF ₂ , H, H, H, O], [AC 4408; H, H, F, H, O, SCF ₃ , H, H, H, O], [AC 4409; H, H, F, H, O, CN, H, H, H, O], [AC 4410; H, H, F, H, O, NO ₂ , H, H, H, O], [AC 4411; H, H, F, Me, O, H, H H, H, O], [AC 4412; H, H, F, Me, O, F, H, H, H, O], [AC 4413; H, H, F, Me, O, Cl, H, H , H, O], [AC 4414; H, H, F, Me, O, Br, H, H, H, O], [AC 4415; H, H, F, Me, O, I, H, H, H , O], [AC 4416; H, H, F, M e, O, Me, H, H, H, O, [AC 4417; H, H, F, Me, O, Et, H, H, H, O], [AC 4418; H, H, F, Me, O, Pr, H, H, H, O], [AC 4419; H, H, F, Me, O, i-Pr, H, H, H, O], [AC 4420; H, H, F, Me, _{O, CH = CH 2, H} , H, H, O], [AC4421; H, H, F, Me, O, C (CH 3) = CH 2, H, H, H, O], [AC4422; H, H, F, Me, O, C≡CH, H, H, H, O], [AC 4423; H, H, F, Me, O, C≡ CCH ₃ , H, H, H, O], [AC 4424; H, H, F, Me, O, c-Pr, H, H, H, O], [AC 4425; H, H, F, Me, O, OMe, H, H, H, O], [AC 4426; H, H, F, Me, O, OEt, H, H, H, O], [AC 4427; H, H, F, Me, O, Oi-Pr, H, H, H, O], [AC4428; H, H, F, Me, O, SMe, H, H, H, O], [AC 4429; H, H, F, Me, O, SE t, H, H, H, O], [AC 4430 ; H, H, F, Me , O, CH 2 F, H, H, H, O], [AC4431; H, H, F, Me, O, CHF 2, H, H, H, O], [ AC4432; H, H, F, Me, O, CF 3, H, H, H, O], [AC4433; H, H, F, Me, O, OCH 2 F, H, H, H, O], [AC 4434; H, H, F, Me, O, OCHF ₂ , H, H, H, O], [AC 4435; H, H, F, Me, O, OCF ₃ , H, H, H, O], [AC 4436; H, H, F, Me, O, SCH ₂ F, H, H, H, O], [AC 4437; H, H, F, Me, O, SCHF ₂ , H, H, H, O] [AC 4438; H, H, F, Me, O, SCF ₃ , H, H, H, O], [AC 4439; H, H, F, Me, O, CN, H, H, H, O], [AC4440; H, H, F , Me, O, NO 2, H, H, H, O], [AC4441; H, Me, F, Me, O, H, H, H, H, O], [ AC4442; H, Me, F, Me, O, F, H, H, O], [AC4443; H, Me, F, Me, O, Cl, H, H, H, O], [AC4444; H, Me, F, Me, O, Br, H, H, H, O], [AC 4445; H, Me, F, Me, O, I, H, H, H, O], [AC 4446; H, Me, F, Me, O, Me, H, H, H, O], [AC 4447; H, Me, F, Me, O, Et, H, H, H, O], [AC 4448 H, Me, F, Me, O, Pr, H, H, H, O], [AC 4449; H, Me, F, Me, O, i-Pr, H, H, H, O], [AC 4450 H, Me, F, Me, O, CH = CH ₂ , H, H, H, O], [AC4451; H, Me, F, Me, O, C (CH ₃ ) = CH ₂ , H, H H, O], [AC4452; H, Me, F, Me, O, C≡CH, H, H, H, O], [AC4453; H, Me, F, Me, O, C≡CCH ₃ , H, H, H, O], [AC4454; H, Me, F, Me, O, c-Pr, H, H, H, O], [AC 4455; H, Me, F, Me, O, OMe, H, H, H, O], [AC 4456; H, Me, F, Me, O, OEt, H, H, H, O], [AC 4457; H, Me, F, Me, O, Oi-Pr, H, H, H, O], [AC 4458; H, Me, F, Me, O, SMe, H, H, H, O], [AC 4459; H, Me, F, Me, O, SE t, H, H, H, O], [ AC4460; H, Me, F, Me, O, CH 2 F, H, H, H, O], [AC4461; H, Me, F, Me, O, CHF 2, H , H, H, O], [AC4462; H, Me, F, Me, O, CF 3, H, H, H, O], [AC4463; H, Me, F, Me, O, OCH 2 F, H, H, H, O] , [AC4464; H, Me, F, Me, O, OCHF 2, H, H, H, O], [AC4465; H, Me, F, Me, O, OCF 3, H, H, H, O], [AC 4466; H, Me, F, Me, O, SCH ₂ F, H, H, H, O], [AC 4467; H, Me, F, Me, O, SCHF ₂ , H, H, H, O], [AC 4468; H, Me, F, Me, O, SCF ₃ , H, H, H, O], [AC 4469; H, Me, F, Me, O, CN, H, H, H, O], [AC 4470; H, Me, F, Me, O, NO ₂ , H, H, H, O], [AC 4471; H, H, H, H, O, H, F , H, H, O], [AC 4472; H, H, H, H, H, O, F, F, H, H, O], [AC 4473; H, H, H, H, O, Cl, F, H , H, O], [AC 4474; H, H, H, H, O, Br, F, H, H, O] , [AC 4475; H, H, H, H, H, O, I, F, H, O], [AC 4476; H, H, H, H, O, Me, F, H, H, O], [ AC 4477; H, H, H, H, H, O, Et, F, H, H, O], [AC 4478; H, H, H, H, O, Pr, F, H, H, O], [AC 4479; H, H, H, H, O, i-Pr, F, H, H, O], [AC4480; H, H, H, H, O, CH = CH 2, F, H, H, O], [AC 4481; H, H, H, H, H, O, C (CH ₃ ) = CH ₂ , F, H, H, O], [AC 4482; H, H, H, H, O, C≡CH, F, H, H, O], [AC 4483; H, H, H, H, O, C≡CCH ₃ , F, H, H, O], [AC 4484; H, H, H, H, O, c-Pr , F, H, H, O], [AC 4485; H, H, H, H, O, OMe, F, H, H, O],

[AC 4486; H, H, H, H, H, O, OEt, F, H, H, O], [AC 4487; H, H, H, H, O, Oi-Pr, F, H, H, O], [AC 4488; H, H, H, H, H, O, SMe, F, H, H, O], [AC 4489; H, H, H, H, H, O, SE t, F, H, H, O], [AC 4490 ; H, H, H, H , O, CH 2 F, F, H, H, O], [AC4491; H, H, H, H, O, CHF 2, F, H, H, O], [ AC4492; H, H, H, H, O, CF 3, F, H, H, O], [AC4493; H, H, H, H, O, OCH 2 F, F, H, H, O], [AC 4494; H, H, H, H, H, O, OCHF ₂ , F, H, H, O], [AC 4495; H, H, H, H, O, OCF ₃ , F, H, H, O], [AC 4496; H, H, H, H, H, O, SCH ₂ F, F, H, H, O], [AC 4497; H, H, H, H, O, SCHF ₂ , F, H, H, O] , [AC4498; H, H, H, H, O, SCF 3, F, H, H, O], [AC4499; H, H, H, H, O, CN, F, H, H, O], [AC 4500; H, H, H, H, H, O, NO ₂ , F, H, H, O], [AC 4501; H, H, H, Me, O, H, F, H, H, O], [AC AC 4502; H, H, H, Me, O, F, F, H, H, O], [AC 4503; H, H, H, Me, O, Cl, F, H, H, O], [AC 4504; H, H, H, H, Me, O, Br, F, H, H, O], [AC 4505; H, H, H, Me, O, I, F, H, O], [AC 4506; H, H, H, Me, O, Me, F, H, H, O], [AC 4507; H, H, H, Me, O, Et, F, H, H, O], [AC 4508; H, H, H, Me, O, Pr, F, H, H, O], [AC 4509; H, H, H, Me, O, i-Pr, F, H, H, O], [AC 4510; H, H, H, Me, O, CH = CH 2, F, H, H, O], [AC4511; H, H, H, Me, O, C (CH 3) = CH 2, F, H, H, O] , [AC 4512; H, H, H, H, Me, O, C≡CH, F, H, H, O], [AC 4513; H, H, H, Me, O, C≡ CCH ₃ , F, H, H , O], [AC 4514; H, H, H, Me, O, c, Pr, F, H, H, O], [AC 4515; H, H, H, Me, O, OMe, F, H, H , O], [AC 45 16; H, H, H, H, Me, O, OEt, F, H, H, O], [AC 4517; H, H, H, Me, O, Oi-Pr, F, H, H, O], [[ AC 4518; H, H, H, H, Me, O, SMe, F, H, H, O], [AC 4519; H, H, H, Me, O, SE t, F, H, H, O], [AC 4520; H, H, H, Me, O, CH 2 F, F, H, H, O], [AC4521; H, H, H, Me, O, CHF 2, F, H, H, O], [AC4522 ; H, H, H, Me , O, CF 3, F, H, H, O], [AC4523; H, H, H, Me, O, OCH 2 F, F, H, H, O], [ AC 4524; H, H, H, Me, O, OCHF ₂ , F, H, H, O], [AC 4525; H, H, H, Me, O, OCF ₃ , F, H, H, O], [ AC 4526; H, H, H, Me, O, SCH ₂ F, F, H, H, O], [AC 4527; H, H, H, Me, O, SCHF ₂ , F, H, H, O], [AC4528; H, H, H , Me, O, SCF 3, F, H, H, O], [AC4529; H, H, H, Me, O, CN, F, H, H, O], [ AC 4530; H, H, H, Me, O, NO ₂ , F, H, H, O], [AC 4531; H, Me, H, Me, O, H, F, H, H, O], [AC 4532 H, Me, H, Me, O, F, F, H, H, O], [AC4533; H, Me, H, Me, O, Cl, F, H, H, O], [AC 4534; H , Me, H, Me, O, Br, F, H, H, O], [AC 4535; H, Me, H, Me, O, I, F, H, O, [AC 4536; H, Me , H, Me, O, Me, F, H, H, O], [AC 4537; H, Me, H, Me, O, Et, F, H, H, O], [AC 4538; H, Me, H , Me, O, Pr, F, H, H, O], [AC 4539; H, Me, H, Me, O, i-Pr, F, H, H, O], [AC 4540; H, Me, H , Me, O, CH = CH 2, F, H, H, O], [AC4541; H, Me, H, Me, O, C (CH 3) = CH 2, F, H, H, O], [AC4542; H, Me, H, Me, O, C≡CH, F, H, H, O], [AC4543; H, Me, H, Me, O, C≡CCH ₃ , F, H, H, O], [AC 4544; H, Me, H, Me, O, c-Pr, F, H, H, O], [AC 4545; H, Me, H, Me, O, OMe, F, H, H, O], [AC 4546; H, Me, H, Me, O, OEt, F, H, H, O], [AC 4547; H, Me, H, Me, O, Oi-Pr, F, H, H, O], [AC 4548; H, Me, H, Me, O, SMe, F, H, O], [AC 4549; H, Me, H, Me, O, SEt, F, H, H, O], [AC4550; H, Me, H, Me, O, CH 2 F, F, H, H, O], [AC4551; H, Me, H, _{Me, O, CHF 2, F} , H, H, O], [AC4552; H, Me, H, Me, O, CF 3, F, H, H, O], [AC4553; H, Me, H, _{Me, O, OCH 2 F,} F, H, H, O], [AC4554; H, Me, H, Me, O, OCHF 2, F, H, H, O], [AC4555; H, Me, H _{, Me, O, OCF 3,} F, H, H, O], [AC4556; H, Me, H, Me, O, SCH 2 F, F, H, H, O], [AC4557; H, Me, _{H, Me, O, SCHF 2} , F, H, H, O], [AC4558; H, Me, H, Me, O, SCF 3, F, H, H, O], [AC4559; H, Me, H, Me, O, CN, F, H, H, O], [AC 4560; H, Me, H, Me, O, NO ₂ , F, H, H, O], [AC4561; H, H, H , H, O, H, H, H, F, O], [AC4562; H, H, H, H, H, O, F, H, F, O], [AC4563; H, H, H, H] , O, Cl, H, H, F, O], [AC 4564; H, H, H, H, H, O, Br, H, F, O], [AC 4565; H, H, H, H, O , I, H, H, F, O], [AC 4566; H, H, H, H, H, O, Me, H, F, O], [AC 4 567; H, H, H, H, O, Et , H, H, F, O], [AC 4568; H, H, H, H, O, Pr, H, H, F, O], [AC 4569; H, H, H, H, O, i-Pr , H, H, F, O ], [AC4570; H, H, H, H, O, CH = CH 2, H, H, F, O], [AC4571; H, H, H, H, O, _{C (CH 3) = CH 2} , H, H, F, O], [AC4572; H, H, H, H, O, C≡CH, H, H, F, O], [AC4573; H, H , H, H, O, C≡CCH ₃ , H, H, F, O], [AC 4574; H, H, H, H, O, c-Pr, H, H, F, O], [[ AC 4575; H, H, H, H, H, O, OMe, H, H, F, O], [AC 4576; H, H, H, H, O, OEt, H, H, F, O], [AC 4577; H, H, H, H, H, O, Oi-Pr, H, H, F, O], [AC 4578; H, H, H, H, O, SMe, H, F, O], [AC 4579; H, H, H, H, O, SEt, H, H, F, O], [AC4580; H, H, H, H, O, CH 2 F, H, H, F, O], [AC4581; H, H, H, H, O, CHF 2, H, H, F, O], [AC4582; H, H, H, H, O, CF 3, H, H, F, O], [AC4583; H, H, H, H, O, OCH 2 F, H, H, F, O], [AC4584; H, H, H, H, O, OCHF 2, H, H, F, O],

[AC4585; H, H, H , H, O, OCF 3, H, H, F, O], [AC4586; H, H, H, H, O, SCH 2 F, H, H, F, O] , [AC 4587; H, H, H, H, H, O, SCHF ₂ , H, H, F, O], [AC 4588; H, H, H, H, O, SCF ₃ , H, H, F, O] [AC 4589; H, H, H, H, H, O, CN, H, H, F, O], [AC 4590; H, H, H, H, O, NO ₂ , H, H, F, O], [AC 4591; H, H, H, H, Me, O, H, H, F, O], [AC 4592; H, H, H, Me, O, F, H, F, O, [AC 4593] H, H, H, H, Me, O, Cl, H, H, F, O], [AC 4594; H, H, H, Me, O, Br, H, F, O], [AC 4595; H , H, H, Me, O, I, H, H, F, O], [AC 4596; H, H, H, Me, O, Me, H, F, O], [AC 4597; H, H H, Me, O, Et, H, H, F, O], [AC 4598; H, H, H, Me, O, Pr, H, F, O], [AC 4599; H, H, H , Me, O, i-Pr , H, H, F, O], [AC4600; H, H, H, Me, O, CH = CH 2, H, H, F, O], [AC4601; H, H, H, Me, O, C (CH 3) = CH 2, H, H, F, O], [AC4602; H, H, H, Me, O, C≡CH, H, H, F, O H, H, H, Me, O, C≡CCH ₃ , H, H, F, O], [AC 4604; H, H, H, Me, O, c-Pr, H, H, F, O], [AC 4605; H, H, H, Me, O, OMe, H, H, F, O], [AC 4606; H, H, H, Me, O, OEt, H, H, F, O], [AC 4607; H, H, H, Me, O, Oi-Pr, H, H, F, O], [AC 4608; H, H, H, Me, O, SMe, H, H, F, O], [AC 4609; H, H, H, Me, O, SE t, H, F, O], [AC 4610; H, H, H, Me, O, CH ₂ F, H, H, F, O], [AC4611; H, H, H, Me, O, CHF 2, H, H, F, O], [AC4612; H, H, H, Me, O, CF 3, H, H, F, O], [AC 4613; H, H, H, Me, O, OCH ₂ F, H, H, F, O], [AC 4614; H, H, H, Me, O, OCHF ₂ , H, H, F , O], [AC4615; H , H, H, Me, O, OCF 3, H, H, F, O], [AC4616; H, H, H, Me, O, SCH 2 F, H, H, F, O], [AC 4617; H, H, H, Me, O, SCHF ₂ , H, H, F, O], [AC 4618; H, H, H, Me, O, SCF ₃ , H, H, F, O], [AC 4619; H, H, H, Me, O, CN, H, F, O], [AC 4620; H, H, H, Me, O, NO ₂ , H, H, F H, Me, H, Me, H, H, H, F, O], [AC 4622; H, Me, H, Me, O, F, H, H, F, O H, Me, H, Me, O, Cl, H, F, O], [AC 4624; H, Me, H, Me, O, Br, H, H, F, O], [AC 4625; H, Me, H, Me, O, I, H, H, F, O], [AC 4626; H, Me, H, Me, O, Me, H, H, F, O], [AC 4627 H, Me, H, Me, O, Et, H, F, O], [AC 4628; H, Me, H, Me, O, Pr, H, F, O], [AC 4629; H , Me, H, Me, O , i-Pr, H, H, F, O], [AC4630; H, Me, H, Me, O, CH = CH 2, H, H, F, O], [ AC4631; H, Me, H, Me, O, C (CH 3) = CH 2, H, H, F, O], [AC4632; H, Me, H, Me, O, C≡CH, H, H , F, O], [AC 4633; H, Me, H, Me, O, C≡CCH ₃ , H, H, F, O], [AC 4634; H, Me, H, Me, O, c-Pr, H, H, F, O], [AC 4635; H, Me, H, Me, O, OMe, H, H, F, O], [AC 4636; H, Me, H, Me, O, OE t, H, H, F, O], [AC 4637; H, Me, H, Me, O, Oi-Pr, H, H, F, O], [AC 4638; H, Me, H, Me, O, SMe, H, H, F, O], [AC 4639; H, Me, H, Me, O, SE t, H, H, F, O], [AC 4640; H, Me, H, Me, O, CH ₂ F, H, H, F, O], [ AC4641; H, Me, H, Me, O, CHF 2, H, H, F, O], [AC4642; H, Me, H, Me, O, CF 3, H, H, F, O], [ AC4643; H, Me, H, Me, O, OCH 2 F, H, H, F, O] H, Me, H, Me, O, OCHF ₂ , H, H, F, O], [AC 4645; H, Me, H, Me, O, OCF ₃ , H, H, F, O] H, Me, H, Me, O, SCH ₂ F, H, H, F, O], [AC 4647; H, Me, H, Me, O, SCHF ₂ , H, H, F, O H, Me, H, Me, O, SCF ₃ , H, F, O], [AC 4649; H, Me, H, Me, O, CN, H, H, F, O] , [AC 4650; H, Me, H, Me, O, NO ₂ , H, F, O], [AC4651; H, H, H, H, O, H, H, H, F, O], [AC4652; H, H, H, H, H, O, F, H, F, O], [AC4653; H, H, H, H, O, Cl, H, H, F, O], [AC4654 H, H, H, H, H, O, Br, H, H, F, O], [AC 4655; H, H, H, H, O, I, H, F, O], [AC 4656; H , H, H, H, H, O, Me, H, H, F, O], [AC 4657; H, H, H, H, H, O, Et, H, F, O], [AC 4658; H, H , H, H, O, Pr, H, H, F, O], [AC 4659; H, H, H, H, H, O, i-Pr, H, F, O], [AC 4660; H, H , H, H, O, CH = CH 2, H, H, F, O], [AC4661; H, H, H, H, O, C (CH 3) = CH 2, H, H, F, O ], [AC4662; H, H, H, H, H, O, C≡CH, H, H, F, O], [AC4663; H, H, H, H, H, O, C≡ CCH ₃ , H, H, H, H, H, H, H, O, c-Pr, H, H, F, O], [AC 4665; H, H, H, H, O, OMe, H, H, F, O], [AC4664; H, H, H, H, H, O, OEt, H, H, F, O], [AC 4667; H, H, H, H, O, Oi-Pr, H, H, F, O], [AC 4 666; H, H, H, H, H, O, SMe, H, F, O], [AC 4669; H, H, H, H, O, SEt, H, H, F, F, O], [AC 4668; O], [AC4670; H, H, H, H, O, CH 2 F, H, H, F, O], [AC4671; H, H, H, H, O, CHF 2, H, H, F , O], [AC4672; H , H, H, H, O, CF 3, H, H, F, O], [AC4673; H, H, H, H, O, OCH 2 F, H, H, F, O], [AC 46 74; H, H, H, H, O, OCHF 2, H, H, F, O], [AC4675; H, H, H, H, O, OCF 3, H, H, F, O], [ AC 4676; H, H, H, H, H, O, SCH ₂ F, H, H, F, O], [AC 4677; H, H, H, H, O, SCHF ₂ , H, H, F, O], [AC 4678; H, H, H, H, H, O, SCF ₃ , H, H, F, O], [AC 4679; H, H, H, H, O, CN, H, H, F, O], [AC AC 4680; H, H, H, H, H, O, NO ₂ , H, H, F, O], [AC4681; H, H, H, Me, O, H, H, F, O], [AC4682 H, H, H, H, Me, O, F, H, H, F, O], [AC4683; H, H, H, Me, O, Cl, H, F, O], [AC4684; H , H, H, Me, O, Br, H, H, F, O],

[AC 4685; H, H, H, H, Me, O, I, H, F, O], [AC 4686; H, H, H, Me, O, Me, H, F, O], [AC 4687 H, H, H, H, Me, O, Et, H, F, O], [AC 4688; H, H, H, Me, O, Pr, H, F, O], [AC 4689; H , H, H, Me, O , i-Pr, H, H, F, O], [AC4690; H, H, H, Me, O, CH = CH 2, H, H, F, O], [ AC4691; H, H, H, Me, O, C (CH 3) = CH 2, H, H, F, O], [AC4692; H, H, H, Me, O, C≡CH, H, H , F, O], [AC4693; H, H, H, Me, O, C≡CCH ₃ , H, H, F, O], [AC4694; H, H, H, Me, O, c-Pr, H, H, F, O], [AC 4695; H, H, H, Me, O, OMe, H, H, F, O], [AC 4696; H, H, H, Me, O, OE t, H, H, F, O], [AC 4697; H, H, H, Me, O, Oi-Pr, H, H, F, O], [AC 4698; H, H, H, Me, O, SMe, H, H, F, O], [AC 4699; H, H, H, Me, O, SE t, H, H, F, O], [AC 4700; H, H, H, Me, O, CH ₂ F, H, H, F, O], [AC 4701; H, H, H, Me, O, CHF ₂ , H, H, F, O], [AC 4702; H, H, H, Me, O, CF ₃ , H, H, F, O], [AC 4703; H, H, H, Me, O, OCH ₂ F, H, H, F, O], [AC 4704; H, H, H, Me, O, OCHF ₂ , H , H, F, O], [AC4705; H, H, H, Me, O, OCF 3, H, H, F, O], [AC4706; H, H, H, Me, O, SCH 2 F, H, H, F, O], [AC 4707; H, H, H, Me, O, SCHF ₂ , H, H, F, O], [AC 4708; H, H, H, Me, O, SCF ₃ , H, H, F, O], [AC 4709; H, H, H, Me, O, CN, H, H, F, O], [AC 4710; H, H, H, Me, O, NO ₂ , H H, F, O], [AC 4711; H, Me, H, Me, O, H, H, H, F, O], [AC 4712; H, Me, H, Me, O, F, H, H , F, O], [AC 4713; H, Me, H, Me, O, Cl, H, F, O], [AC 4714; H, Me, H, Me, O, Br, H, H, F, O], [AC 4715; H, Me, H, Me, O, I, H, F, O], [AC 4716; H, Me, H, Me, O, H, Me, H, Me, O, Et, H, F, O], [AC 4718; H, Me, H, Me, O, Pr, Me, H, H, F, O], [AC 4717; H, H, F, O], [AC 4719; H, Me, H, Me, O, i-Pr, H, H, F, O], [AC 4720; H, Me, H, Me, O, CH = _{CH 2, H, H, F} , O], [AC4721; H, Me, H, Me, O, C (CH 3) = CH 2, H, H, F, O], [AC4722; H, Me, H, Me, O, C≡CH, H, H, F, O], [AC 4723; H, Me, H, Me, O, C≡CCH ₃ , H, H, F, O], [AC 4724; H , Me, H, Me, O, c-Pr, H, H, F, O], [AC 4725; H, Me, H, Me, O, OMe, H, F, O], [AC 4726; H , Me, H, Me, O, OEt, H, H, F, O], [AC 4727; H, Me, H, Me, O, Oi-Pr, H, H, F, O], [AC 4728; H , Me, H, Me, O, SMe, H, H, F, O], [AC 4729; H, Me, H, Me, O, SE t, H, F, O], [AC 4730; H, Me , H, Me, O, CH 2 F, H, H, F, O], [AC4731; H, Me, H, Me, O, CHF 2, H, H, F, O], [AC4732; H, Me, H, Me, O, CF 3, H, H, F, O], [AC4733; H, Me, H, Me, O, OCH 2 F, H, H, F, O], [AC4734; H , Me, H, Me, O , OCHF 2, H, H, F, O], [AC4735; H, Me, H, Me, O, OCF 3, H, H, F, O], [AC4736; H , Me, H, Me, O, SCH ₂ F, H, H, F, O], [AC 4737; H, Me, H, Me, O, SCHF ₂ , H, H, F, O], [AC 4738; H, Me, H, Me, O, SCF 3, H, H, F, O], [AC4739; H, Me, H, Me, O, CN, H, H, F, O], [AC4740; H , Me, H, Me, O, NO ₂ , H, H, F, O], [AC4741; H, H, H, H, O, H, H, Me, O], [AC4742; H, H, H, H, H, O, F, H, H, Me, O], [AC4743; H, H, H, H, O, Cl, H, H, Me, O], [AC 4744; H, H, H, H, H, O, Br, H, Me, O], [AC 4745; H, H, H, H, O, I, H, H, Me, O], [AC 4746; H, H, H, H, O, Me, H, Me, O], [AC 4747; H, H, H, H, O, Et, H, H, Me, O], [AC 4748; H, H, H, H, H, O, Pr, H, Me, O], [AC 4749; H, H, H, H, O, i-Pr, H, H, Me, O], [AC4750; H, H, H, H, O, CH = CH 2, H, H, Me, O], [AC4751; H, H, H, H _{, O, C (CH 3)} = CH 2, H, H, Me, O], [AC4752; H, H, H, H, O, C≡CH, H, H, Me, O], [AC4753; H, H, H, H, H, O, C≡CCH ₃ , H, H, Me, O], [AC 4754; H, H, H, H, O, c-Pr, H, H, Me, O], [AC4755; H, H, H, H, H, O, OMe, H, H, Me, O], [AC 4756; H, H, H, H, O, OEt, H, Me, O], [AC 4757 H, H, H, H, H, O, Oi-Pr, H, H, Me, O], [AC 4758; H, H, H, H, O, S Me, H, Me, O], [AC 4759 H, H, H, H, H, O, SE t, H, H, Me, O], [AC 4760; H, H, H, H, O, CH ₂ F, H, Me, O], [AC 476 1 ; H, H, H, H , O, CHF 2, H, H, Me, O], [AC4762; H, H, H, H, O, CF 3, H, H, Me, O], [AC4763 H, H, H, H, H, O, OCH ₂ F, H, H, Me, O], [AC 4764; H, H, H, H, O, OCHF ₂ , H, H, Me, O], [, AC4765; H, H, H, H, O, OCF 3, H, H, Me, O], [AC4766; H, H, H, H, O, SCH 2 F, H, H, Me, O], [AC 4767; H, H, H, H, H, O, SCHF ₂ , H, H, Me, O], [AC 4768; H, H, H, H, H, O, SCF ₃ , H, H, Me, O], [AC4769; H, H, H , H, O, CN, H, H, Me, O], [AC4770; H, H, H, H, O, NO 2, H, H, Me, O], [ AC 4771; H, H, H, H, Me, O, H, H, Me, O], [AC 4772; H, H, H, Me, O, F, H, H, Me, O], [AC 4773; H, H, H, H, Me, O, Cl, H, Me, O], [AC 4774; H, H, H, Me, O, Br, H, Me, O], [AC 4775 H, H, H, H, Me, O, I, H, H, Me, O], [AC 4776; H, H, H, Me, O, Me, H, Me, O], [AC 4777; H , H, H, Me, O, Et, H, H, Me, O], [AC 4778; H, H, H, Me, O, Pr, H, Me, O], [AC 4779; H, H , H, Me, O, i -Pr, H, H, Me, O], [AC4780; H, H, H, Me, O, CH = CH 2, H, H, Me, O], [AC4781; H, H, H, Me, O, C (CH 3) = CH 2, H, H, Me, O], [AC4782; H, H, H, Me, O, C≡CH, H, H, Me H, H, H, Me, O, C≡CCH ₃ , H, H, Me, O], [AC 4784; H, H, H, Me, O, c-Pr, H, H, Me, O],

[AC 4785; H, H, H, Me, O, OMe, H, H, Me, O], [AC 4786; H, H, H, Me, O, OE t, H, Me, O], [AC 4787 H, H, H, H, Me, O, Oi-Pr, H, H, Me, O], [AC 4788; H, H, H, Me, O, SMe, H, Me, O], [AC 4789] ; H, H, H, Me , O, SEt, H, H, Me, O], [AC4790; H, H, H, Me, O, CH 2 F, H, H, Me, O], [AC4791 ; H, H, H, Me , O, CHF 2, H, H, Me, O], [AC4792; H, H, H, Me, O, CF 3, H, H, Me, O], [AC4793 ; H, H, H, Me , O, OCH 2 F, H, H, Me, O], [AC4794; H, H, H, Me, O, OCHF 2, H, H, Me, O], [ AC4795; H, H, H, Me, O, OCF 3, H, H, Me, O], [AC4796; H, H, H, Me, O, SCH 2 F, H, H, Me, O], [AC 4 797; H, H, H, Me, O, SCHF ₂ , H, H, Me, O], [AC 4798; H, H, H, Me, O, SCF ₃ , H, H, Me, O], [AC 4799; H, H, H, Me, O, CN, H, H, Me, O], [AC 4800; H, H, H, Me, O, NO ₂ , H, H, Me, O], [AC AC 4801; H, Me, H, Me, O, H, H, Me, O], [AC 4802; H, Me, H, Me, O, F, H, Me, O], [AC 4803; H, Me, H, Me, O, Cl, H, H, Me, O], [AC 4804; H, Me, H, Me, O, Br, H, Me, O], [AC 4805; H, Me, H, Me, O, I, H, H, Me, O], [AC 4806; H, Me, H, Me, O, Me, H, Me, O], [AC 4807; H, Me, H, Me, O, Et, H, Me, O], [AC 4808; H, Me, H, Me, O, Pr, H, Me, O], [AC 4809; H, Me, H, Me, O, i-Pr, H, H, Me, O], [AC 4810; H, Me, H, Me, O, CH = CH ₂ , H, H, Me, O], [AC 4811; H, Me , H, Me, O, C (CH 3) = CH 2, H, H, Me, O], [AC4812; H, Me, H, Me, O, C≡CH, H, H, Me, O] , [AC 4813; H, Me, H, Me, O, C _{CCH 3, H, H, Me} , O], [AC4814; H, Me, H, Me, O, c-Pr, H, H, Me, O], [AC4815; H, Me, H, Me, O , OMe, H, H, Me, O], [AC 4816; H, Me, H, Me, O, OEt, H, H, Me, O], [AC 4817; H, Me, H, Me, O, Oi -Pr, H, H, Me, O], [AC 4818; H, Me, H, Me, O, SMe, H, Me, O], [AC 4819; H, Me, H, Me, O, SEt , H, H, Me, O ], [AC4820; H, Me, H, Me, O, CH 2 F, H, H, Me, O], [AC4821; H, Me, H, Me, O, CHF _{2, H, H, Me,} O], [AC4822; H, Me, H, Me, O, CF 3, H, H, Me, O], [AC4823; H, Me, H, Me, O, OCH ₂ F, H, H, Me, O], [AC 4824; H, Me, H, Me, O, OCHF ₂ , H, H, Me, O], [AC 4825; H, Me, H, Me, O, _{OCF 3, H, H, Me} , O], [AC4826; H, Me, H, Me, O, SCH 2 F, H, H, Me, O], [AC4827; H, Me, H, Me, O , SCHF ₂ , H, H, Me, O], [AC 4828; H, Me, H, Me, O, SCF ₃ , H, H, Me, O], [AC 4829; H, Me, H, Me, O , CN, H, H, Me, O], [AC 4830; H, Me, H, Me, O, NO ₂ , H, H, Me, O], [AC 4831; H, H, H, H, O, H, H, H, Me, O], [AC4832; H, H, H, H, H, O, F, H, Me, O], [AC 4833; H, H, H, H, O, Cl, H, H, Me, O], [AC 4834; H, H, H, H, O, Br, H, Me, O], [AC 4835; H, H, H, H, O, I, H, H, Me, O], [AC 4836; H, H, H, H, H, O, Me, H, Me, O], [AC 4837; H, H, H, H, O, Et, H, H, H, Me, O], [AC 4838; H, H, H, H, H, O, Pr, H, Me, O], [AC 4839; H, H, H, H, O, i-Pr, H, H, Me, O], [AC4840; H, H, H, H, O, CH = CH 2, H, H, Me, O], [AC4841; H, H, H, H, O, C (CH 3) _{= CH 2, H, H,} Me, O], [AC4842; H, H , H, H, O, C≡CH , H, H, Me, O], [AC4843; H, H, H, H, O, C≡CCH 3, H, H, Me, O], [AC4844; H, H, H, H, H, O, c-Pr, H, H, Me, O], [AC 4845; H, H, H, H, O, OMe, H, Me, O], [AC 4846; H, H, H, H, H, O, OEt, H, H, Me, O], [AC 4847; H, H, H, H, O, Oi-Pr, H, H, Me, O], [AC 4848; H, H, H, H, H, O, SMe, H, H, Me, O], [AC 4849; H, H, H, H, O, SE, H, Me, O], [AC 4850; H, H, H, H, O, CH 2 F, H, H, Me, O], [AC4851; H, H, H, H, O, CHF 2, H, H, Me, O], [AC4852; H , H, H, H, O , CF 3, H, H, Me, O], [AC4853; H, H, H, H, O, OCH 2 F, H, H, Me, O], [AC4854; H, H, H, H, O, OCHF 2, H, H, Me, O], [AC4855; H, H, H, H, O, OCF 3, H, H, Me, O], [AC4856; H, H, H, H, H, O, SCH ₂ F, H, H, Me, O], [AC 4857; H, H, H, H, O, SCHF ₂ , H, H, Me, O], [AC 4858 ; H, H, H, H , O, SCF 3, H, H, Me, O], [AC4859; H, H, H, H, O, CN, H, H, Me, O], [AC4860; H, H, H, H, O, NO 2, H, H, Me, O], [AC4861; H, H, H, Me, O, H, H, H, Me, O], [AC4862; H , H, H, Me, O, F, H, H, Me, O], [AC 4863; H, H, H, Me, O, Cl, H, Me, O], [AC 4864; H, H , H, Me, O, Br, H, H, Me, O], [AC 4865; H, H, H, Me, O, I, H, Me, O], [AC 4866; H, H, H , Me, O, Me, H, H, Me, O], [AC 4867; H, H, H, Me, O, Et, H, Me, O], [AC 4868; H, H, H, Me , O, Pr, H, H, Me, O], [AC 4869; H, H, H, Me, O, i-Pr, H, H, Me, O], [AC 4870; H, H, H, Me _{, O, CH = CH 2,} H, H, Me, O], [AC4871; H, H, H, Me, O, C (CH 3) = CH 2, H, H, Me, O], [AC 4872; H, H, H, Me, O, C≡CH, H, H, Me, O], [AC 4873; H, H, H, Me, O, C ≡ _{CCH 3, H, H, Me} , O], [AC4874; H, H, H, Me, O, c-Pr, H, H, Me, O], [AC4875; H, H, H, Me, O , OMe, H, H, Me, O], [AC4876; H, H, H, Me, O, OEt, H, H, Me, O], [AC 4877; H, H, H, Me, O, Oi -Pr, H, H, Me, O], [AC4878; H, H, H, Me, O, SMe, H, Me, O], [AC 4879; H, H, H, Me, O, SEt H, H, Me, O], [AC 4880; H, H, H, Me, O, CH ₂ F, H, H, Me, O], [AC 488 1; H, H, H, Me, O, CHF _{2, H, H, Me,} O], [AC4882; H, H, H, Me, O, CF 3, H, H, Me, O], [AC4883; H, H, H, Me, O, OCH ₂ F, H, H, Me, O],

[AC 4884; H, H, H, Me, O, OCHF ₂ , H, H, Me, O], [AC 4885; H, H, H, Me, O, OCF ₃ , H, H, Me, O], [AC 4886; H, H, H, Me, O, SCH ₂ F, H, H, Me, O], [AC 4887; H, H, H, Me, O, SCHF ₂ , H, H, Me, O] [AC 4 888; H, H, H, Me, O, SCF ₃ , H, H, Me, O], [AC 4889; H, H, H, Me, O, CN, H, H, Me, O], [AC 4890; H, H, H, H, Me, O, NO ₂ , H, H, Me, O], [AC 4891; H, Me, H, Me, O, H, H, H, Me, O], [AC AC 4892; H, Me, H, Me, O, F, H, Me, O], [AC 4893; H, Me, H, Me, O, Cl, H, H, Me, O], [AC 4894; H, Me, H, Me, O, Br, H, H, Me, O], [AC 4895; H, Me, H, Me, O, I, H, Me, O], [AC 4896; H, Me, H, Me, O, Me, H, H, Me, O], [AC 4897; H, Me, H, Me, O, Et, H, Me, O], [AC 4898; H, Me, H, Me, O, Pr, H, H, Me, O], [AC 4899; H, Me, H, Me, O, i-Pr, H, Me, O], [AC 4900; H, Me, H, Me, O, CH = CH 2, H, H, Me, O], [AC4901; H, Me, H, Me, O, C (CH 3) = CH 2, H, H, Me, O] [AC4902; H, Me, H, Me, O, C≡CH, H, H, Me, O], [AC4903; H, Me, H, Me, O, C≡CCH ₃ , H, H, Me , O], [AC 4904; H, Me, H, Me, O, c, Pr, H, H, Me, O], [AC 4905; H, Me, H, Me, O, OMe, H, H, Me , O], [AC 4906; H, Me, H, Me, O, OEt, H, H, Me, O], [AC 4907; H, Me, H, Me, O, Oi-Pr, H, H, Me H, Me, H, Me, O, SMe, H, Me, O], [AC 4909; H, Me, H, Me, O, SEt, H, H, Me, O H, Me, H, Me, O, CH ₂ F, H, H, Me, O], [AC 4911; H, Me, H, Me, O, CHF ₂ , H, H, Me, O], [AC 4912; H, M e, H, Me, O, CF 3, H, H, Me, O], [AC4913; H, Me, H, Me, O, OCH 2 F, H, H, Me, O], [AC4914; H , Me, H, Me, O , OCHF 2, H, H, Me, O], [AC4915; H, Me, H, Me, O, OCF 3, H, H, Me, O], [AC4916; H , Me, H, Me, O, SCH ₂ F, H, H, Me, O], [AC 4917; H, Me, H, Me, O, SCHF ₂ , H, H, Me, O], [AC 4918; H, Me, H, Me, O, SCF 3, H, H, Me, O], [AC4919; H, Me, H, Me, O, CN, H, H, Me, O], [AC4920; H , Me, H, Me, O, NO, ₂ , H, H, Me, O], [AC4921; H, H, H, H, O, H, H, H, S, [AC4922; H, H, H, H, H, O, F, H, H, H, S], [AC 4923; H, H, H, H, H, O, Cl, H, H, S], [AC 4924; H, H, H H, H, O, Br, H, H, H, S], [AC 4925; H, H, H, H, H, O, I, H, H, S, [AC 4926; H, H, H, H, O, Me, H, H, H, S], [AC 4927; H, H, H, H, H, O, Et, H, H, H, S], [AC 4928; H, H, H, H, S O, Pr, H, H, H, S], [AC 4929; H, H, H, H, H, O, i-Pr, H, H, H, S], [AC 4930; H, H, H, H, _{O, CH = CH 2, H} , H, H, S], [AC4931; H, H, H, H, O, C (CH 3) = CH 2, H, H, H, S], [AC4932; H, H, H, H, H, O, C≡CH, H, H, H, S], [AC 4933; H, H, H, H, O, C≡ CCH ₃ , H, H, H, S], [AC 4 934; H, H, H, H, H, O, c-Pr, H, H, H, S], [AC 4935; H, H, H, H, O, OMe, H, H, H, S], [AC 4936; H, H, H, H, H, O, OEt, H, H, H, S], [AC 4937; H, H, H, H, O, Oi-Pr, H, H, H, S], [AC 4938; H, H, H, H, H, O, SMe, H, H, H, S], [AC 4939; H, H, H, H, O, SE, H, H, H, S], [AC 4940 ; H, H, H, H , O, CH 2 F, H, H, H, S], [AC4941; H, H, H, H, O, CHF 2, H, H, H, S], [ AC4 942; H, H, H, H, O, CF 3, H, H, H, S], [AC4943; H, H, H, H, O, OCH 2 F, H, H, H, S], [AC 4944; H, H, H, H, H, O, OCHF ₂ , H, H, H, S], [AC 4945; H, H, H, H, H, O, OCF ₃ , H, H, H, S], [AC 4946; H, H, H, H, H, O, SCH ₂ F, H, H, H, S], [AC 4947; H, H, H, H, O, SCHF ₂ , H, H, H, S] , [AC 4948; H, H, H, H, H, O, SCF ₃ , H, H, H, S], [AC 4949; H, H, H, H, O, CN, H, H, H, S], [AC 4950; H, H, H, H, H, O, NO ₂ , H, H, S], [AC 4951; H, H, H, H, Me, O, H, H, H, S, [, AC4952; H, H, H, Me, O, F, H, H, S], [AC4953; H, H, H, Me, O, Cl, H, H, H, S], [AC 495; H, H, H, H, Me, O, Br, H, H, H, S], [AC 4955; H, H, H, Me, O, I, H, H, S, [AC 4956; H, H, H, Me, O, Me, H, H, H, S], [AC 4957; H, H, H, Me, O, Et, H, H, H, S], [AC 4958; H, H, H, Me, O, Pr, H, H, H, S], [AC 4959; H, H, H, Me, O, i-Pr, H, H, H, S], [AC 4960; H, H, H, Me, O, CH = CH 2, H, H, H, S], [AC4961; H, H, H, Me, O, C (CH 3) = CH 2, H, H, H, S] [AC4962; H, H, H, H, Me, O, C≡CH, H, H, H, S], [AC4963; H, H, H, H, Me, O, C≡ CCH ₃ , H, H, H S, [AC 4964; H, H, H, Me, O, c-Pr, H, H, H, S], [AC 4965; H, H, H, Me, O, OMe, H, H, H , S], [AC 4966; H, H, H, Me, O, OEt, H, H, H, S], [AC 4967; H, H, H, Me, O, Oi-Pr, H, H, H , S], [AC 4968; H, H, H, Me, O, SMe, H, H, H, S], [AC 4969; H, H, H, Me, O, SE t, H, H, H, S ], [AC4970; H, H , H, Me, O, CH 2 F, H, H, H, S], [AC4971; H, H, H, Me, O, CHF 2, H, H, H, S], [AC 4972; H, H, H, Me, O, CF 3, H, H, H, S], [AC4973; H, H, H, Me, O, OCH 2 F, H, H, H, S], [AC 4 974; H, H, H, Me, O, OCHF ₂ , H, H, H, S], [AC 4 975; H, H, H, Me, O, OCF ₃ , H, H, H, S], [AC 4976; H, H, H, H, Me, O, SCH ₂ F, H, H, H, S], [AC 4977; H, H, H, Me, O, SCHF ₂ , H, H, H, S] [AC 4978; H, H, H, Me, O, SCF ₃ , H, H, H, S], [AC 4979; H, H, H, Me, O, CN, H, H, H, S], [AC 4 980; H, H, H, Me, O, NO ₂ , H, H, S], [AC 4981; H, Me, H, Me, O, H, H, H, S, [, AC 4982; H, Me, H, Me, O, F, H, H, S], [AC 4983; H, Me, H, Me, O, Cl, H, H, H, S],

[AC 4984; H, Me, H, Me, O, Br, H, H, S], [AC 4985; H, Me, H, Me, O, I, H, H, S, [AC 4986] H, Me, H, Me, O, Me, H, H, H, S], [AC 4987; H, Me, H, Me, O, Et, H, H, H, S], [AC 4988; H , Me, H, Me, O, Pr, H, H, H, S], [AC 4989; H, Me, H, Me, O, i-Pr, H, H, H, S], [AC 4 990; H , Me, H, Me, O , CH = CH 2, H, H, H, S], [AC4991; H, Me, H, Me, O, C (CH 3) = CH 2, H, H, H S, [AC4992; H, Me, H, Me, O, C≡CH, H, H, H, S], [AC4993; H, Me, H, Me, O, C, CCH ₃ , H, H, H, S], [AC 4994; H, Me, H, Me, O, c-Pr, H, H, H, S], [AC 4995; H, Me, H, Me, O, OMe, H, H, H, S], [AC 4996; H, Me, H, Me, O, OEt, H, H, H, S], [AC 4997; H, Me, H, Me, O, Oi-Pr, H, H, H, S], [AC 4998; H, Me, H, Me, O, SMe, H, H, H, S], [AC 4999; H, Me, H, Me, O, SE t, H, H, H, S], [AC 5000; H, Me, H, Me, O, CH ₂ F, H, H, H, S], [AC 5001; H, Me, H, Me, O, CHF ₂ , H, H , H, S], [AC 5002; H, Me, H, Me, O, CF ₃ , H, H, H, S], [AC 5003; H, Me, H, Me, O, OCH ₂ F, H, H, H, S], [ AC5004; H, Me, H, Me, O, OCHF 2, H, H, H, S], [AC5005; H, Me, H, Me, O, OCF 3, H, H, H, S], [AC 5006; H, Me, H, Me, O, SCH ₂ F, H, H, H, S], [AC 5007; H, Me, H, Me, O, SCHF ₂ , H , H, H, S], [AC 5008; H, Me, H, Me, O, SCF ₃ , H, H, H, S], [AC 5009; H, Me, H, Me, O, CN, H, H, H, S], [AC 5010; H, Me, H, Me, O, NO ₂ , H, H, H, S], [AC 5011; H, H, H, H, O, H, H, H , H, S], [AC 5012; H, H, H, H, O, F, H, H, H , S], [AC 5013; H, H, H, H, O, Cl, H, H, S], [AC 5014; H, H, H, H, O, Br, H, H, H, S , [AC 5015; H, H, H, H, H, O, I, H, H, S], [AC 5016; H, H, H, H, O, Me, H, H, H, S], [AC 50 17; H, H, H, H, H, O, Et, H, H, S], [AC 5018; H, H, H, H, O, Pr, H, H, H, S], [AC 50 19 H, H, H, H, H, O, i-Pr, H, H, H, S], [AC 5020; H, H, H, H, O, CH = CH ₂ , H, H, H, S] , [AC 5021; H, H, H, H, H, O, C (CH ₃ ) = CH ₂ , H, H, H, S], [AC 5022; H, H, H, H, O, C≡CH, H , H, H, S], [AC 5023; H, H, H, H, O, C≡CCH ₃ , H, H, H, S], [AC 5024; H, H, H, H, O, c- Pr, H, H, H, S], [AC 5025; H, H, H, H, O, OMe, H, H, H, S], [AC 5026; H, H, H, H, O, OE t, H, H, H, S], [AC 5027; H, H, H, H, O, Oi-Pr, H, H, H, S], [AC 5028; H, H, H, H, O, SMe, H, H, H, S], [AC 5029; H, H, H, H, O, SE t, H, H, H, S], [AC 5030; H, H, H, H, O, CH ₂ F, H, H, H, S], [AC 5031; H, H, H, H, O, CHF ₂ , H, H, H, S], [AC 5032; H, H, H, H, O, CF ₃ , H, H, H, S], [AC 5033; H, H, H, H, O, OCH ₂ F, H, H, H, S], [AC 5034; H, H, H, H, O, OCHF ₂ , H, H, H, S ], [AC5035; H, H, H, H, O, OCF 3, H, H, H, S], [AC5036; H, H, H, H, O, SCH 2 F, H, H, H, S], [AC 5037; H, H, H, H, H, O, SCHF ₂ , H, H, H, S], [AC 5038; H, H, H, H, O, SCF ₃ , H, H, H, S], [AC 5039; H, H, H, H, O, CN, H, H, H, S], [AC 5040; H, H, H, H, O, NO ₂ , H, H, H, S], [AC 5041; H, H, H, Me, O, H, H, H, H, S], [AC 5042; H, H, H, Me, O, F, H , H, H, S], [AC 5043; H, H, H, Me, O, Cl, H, H, H, S], [AC 5044; H, H, H, Me, O, Br, H, H, H, S], [AC 5045; H, H, H, Me, O, I, H, H, H, S], [AC 5046; H, H, H, Me, O, Me, H, H, H, S], [AC 5047; H, H, H, Me, O, Et, H, H, H, S], [AC 5048; H, H, H, Me, O, Pr, H, H, H, S], [AC 5049; H, H, H, Me, O, i- Pr, H, H, H, S], [AC5050; H, H, H, Me, O, CH = CH 2, H, H, H, S], [AC5051; H, H, H, Me, O _{, C (CH 3) = CH} 2, H, H, H, S], [AC5052; H, H, H, Me, O, C≡CH, H, H, H, S], [AC5053; H, H, H, Me, O, C≡CCH ₃ , H, H, H, S], [AC 5054; H, H, H, Me, O, c-Pr, H, H, H, S], [AC 50 55 H, H, H, H, Me, O, OMe, H, H, H, S], [AC 5056; H, H, H, Me, O, OEt, H, H, H, S], [AC 5057; H , H, H, Me, O, Oi-Pr, H, H, H, S], [AC 5058; H, H, H, Me, O, SMe, H, H, S, [AC 5059; H , H, H, Me, O , SEt, H, H, H, S], [AC5060; H, H, H, Me, O, CH 2 F, H, H, H, S], [AC5061; H , H, H, Me, O , CHF 2, H, H, H, S], [AC5062; H, H, H, Me, O, CF 3, H, H, H, S], [AC5063; H , H, H, Me, O , OCH 2 F, H, H, H, S], [AC5064; H, H, H, Me, O, OCHF 2, H, H, H, S], [AC5065; H, H, H, Me, O, OCF 3, H, H, H, S], [AC5066; H, H, H, Me, O, SCH 2 F, H, H, H, S], [AC5067 H, H, H, H, Me, O, SCHF ₂ , H, H, H, S], [AC 5068; H, H, H, Me, O, SCF ₃ , H, H, H, S], [AC 50 69 ; H, H, H, Me , O, CN, H, H, H, S], [AC5070; H, H, H, Me, O, NO 2, H, H, H, S], [AC5071; H, Me, H, Me, O, H, H, H, H, S], [AC 5072; H, Me, H, Me, O, F, H, H, S, [A H, Me, H, Me, O, Cl, H, H, S], [AC5074; H, Me, H, Me, O, Br, H, H, H, S], [AC 5075; H, Me, H, Me, O, I, H, H, H, S], [AC 5076; H, Me, H, Me, O, Me, H, H, S, [AC 50 77; H, Me, H, Me, O, Et, H, H, H, S], [AC 5078; H, Me, H, Me, O, Pr, H, H, H, S], [AC 5079; H, Me, H, Me, O, i- Pr, H, H, H, S], [AC5080; H, Me, H, Me, O, CH = CH 2, H, H, H, S], [AC5081; H , Me, H, Me, O , C (CH 3) = CH 2, H, H, H, S], [AC5082; H, Me, H, Me, O, C≡CH, H, H, H, S], [AC 5083; H, Me, H, Me, O, C≡CCH ₃ , H, H, H, S],

[AC 5084; H, Me, H, Me, O, c-Pr, H, H, H, S], [AC 5085; H, Me, H, Me, O, OMe, H, H, H, S], [AC 50 86; H, Me, H, Me, O, OEt, H, H, H, S], [AC 5087; H, Me, H, Me, O, Oi-Pr, H, H, H, S], [AC 50 88; H, Me, H, Me, O, SMe, H, H, H, S], [AC 5089; H, Me, H, Me, O, SE t, H, H, H, S], [AC 5090 ; H, Me, H, Me , O, CH 2 F, H, H, H, S], [AC5091; H, Me, H, Me, O, CHF 2, H, H, H, S], [ AC5092; H, Me, H, Me, O, CF 3, H, H, H, S], [AC5093; H, Me, H, Me, O, OCH 2 F, H, H, H, S], [AC 5094; H, Me, H, Me, O, OCHF ₂ , H, H, H, S], [AC 5095; H, Me, H, Me, O, OCF ₃ , H, H, H, S], [AC 5096; H, Me, H, Me, O, SCH ₂ F, H, H, H, S], [AC 5097; H, Me, H, Me, O, SCHF ₂ , H, H, H, S] [AC 50 98; H, Me, H, Me, O, SCF ₃ , H, H, H, S], [AC 5099; H, Me, H, Me, O, CN, H, H, H, S], [AC 5100; H, Me, H, Me, O, NO ₂ , H, H, S], [AC 5101; H, H, H, H, S, H, H, H, O], [AC 5101 AC 5102; H, H, H, H, H, S, F, H, H, O], [AC 5103; H, H, H, H, S, Cl, H, H, H, O], [AC 5104; H, H, H, H, H, S, Br, H, H, H, O], [AC 5105; H, H, H, H, S, I, H, H, O], [AC 5106; H, H, H, H, S, Me, H, H, H, O], [AC 5107; H, H, H, H, S, Et, H, H, O], [AC 5108; H, H, H H, H, S, Pr, H, H, H, O], [AC 5109; H, H, H, H, S, i-Pr, H, H, H, O], [AC 5110; H, H, H H, H, S, CH = CH 2, H, H, H, O], [AC5111; H, H, H, H, S, C (CH 3) = CH 2, H, H, H, O] , [AC 5112; H, H, H, H, S, C, CH, H, H, H, O], [AC 5113; H, H, H, H, S, C, CC _{H 3, H, H, H} , O], [AC5114; H, H, H, H, S, c-Pr, H, H, H, O], [AC5115; H, H, H, H, S , OMe, H, H, H, O], [AC 5116; H, H, H, H, S, OEt, H, H, H, O], [AC 5117; H, H, H, H, S, Oi -Pr, H, H, H, O], [AC5118; H, H, H, H, S, SMe, H, H, H, O], [AC 5119; H, H, H, H, S, SEt , H, H, H, O ], [AC5120; H, H, H, H, S, CH 2 F, H, H, H, O], [AC5121; H, H, H, H, S, CHF _{2, H, H, H,} O], [AC5122; H, H, H, H, S, CF 3, H, H, H, O], [AC5123; H, H, H, H, S, OCH ₂ F, H, H, H, O], [AC 5124; H, H, H, H, S, OCHF ₂ , H, H, H, O], [AC 5 125; H, H, H, H, S, OCF ₃ , H, H, H, O], [AC 5126; H, H, H, H, S, SCH ₂ F, H, H, H, O], [AC 5127; H, H, H, H, S , SCHF ₂ , H, H, H, O], [AC 5128; H, H, H, H, S, SCF ₃ , H, H, H, O], [AC 5129; H, H, H, H, S , CN, H, H, H, O], [AC 5130; H, H, H, H, S, NO ₂ , H, H, H, O], [AC 5131; H, H, H, Me, S, H, H, H, H, O], [AC 5132; H, H, H, Me, S, F, H, H, O], [AC 5133; H, H, H, Me, S, Cl, H, H, H, O], [AC 5134; H, H, H, Me, S, Br, H, H, H, O], [AC 5 135; H, H, H, Me, S, I, H, H, H, O], [AC 5136; H, H, H, Me, S, Me, H, H, H, O], [AC 5137; H, H, H, Me, S, Et, H, H, H, H, O], [AC 5138; H, H, H, Me, S, Pr, H, H, H, O], [AC 5139; H, H, H, Me, S, i-Pr, H, H, H, O], [AC5140; H, H, H, Me, S, CH = CH 2, H, H, H, O], [AC5141; H, H, H, Me, S, C (CH 3) _{= CH 2, H, H,} H, O], [AC5142; H, H, H, Me, S, C≡CH, H, H, H, O], [AC5143; H, H, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 5144; H, H, H, Me, S, c-Pr, H, H, H, O], [AC 5145; H, H, H, Me, S, OMe, H, H, H, O], [AC 5146; H, H, H, Me, S, OEt, H, H, H, O], [AC 5147; H, H, H, Me, S, Oi-Pr, H, H, H, O], [AC 5148; H, H, H, Me, S, SMe, H, H, H, O], [AC 5149; H, H, H, Me, S, SE t, H, H, H, O], [AC 5150; H, H, H, Me, S, CH ₂ F, H, H, H, O], [AC 5151; H, H, H, Me, S, CHF ₂ , H, H , H, O], [AC 5152; H, H, H, Me, S, CF ₃ , H, H, H, O], [AC 5153; H, H, H, Me, S, OCH ₂ F, H, H, H, O], [AC 5154; H, H, H, Me, S, OCHF ₂ , H, H, H, O], [AC 5 155; H, H, H, Me, S, OCF ₃ , H, H, H, O], [AC 5156; H, H, H, Me, S, SCH ₂ F, H, H, H, O], [AC 5 157; H, H, H, Me, S, SCHF ₂ , H , H, H, O], [AC 5158; H, H, H, Me, S, SCF ₃ , H, H, H, O], [AC 5159; H, H, H, Me, S, CN, H, H, H, O], [AC 5160; H, H, H, Me, S, NO ₂ , H, H, H, O], [AC 5161; H, H, H, Et, S, H, H, H , H, O], [AC5162; H, H, H, Et, S, F, H, H, O], [AC 5163; H, H, H, Et, S, Cl, H, H, H H, H, H, Et, S, Br, H, H, O], [AC 5165; H, H, H, Et, S, I, H, H, H, O H, H, H, Et, S, Me, H, H, H, O], [AC 5167; H, H, H, Et, S, Et, H, H, H, O], [AC5168; H, H, H, H, Et, S, Pr, H, H, H, O], [AC 5169; H, H, H, Et, S, i-Pr, H, H, H, O], [AC5170; H, H, H , Et, S, CH = CH 2, H, H, H, O], [AC5171; H, H, H, Et, S, C (CH 3) = CH 2, H H, H, O], [AC 5172; H, H, H, Et, S, C≡CH, H, H, H, O], [AC 5173; H, H, H, Et, S, C _{CCH 3, H, H, H} , O], [AC5174; H, H, H, Et, S, c-Pr, H, H, H, O], [AC5175; H, H, H, Et, S , OMe, H, H, H, O], [AC 5176; H, H, H, Et, S, OEt, H, H, H, O], [AC 5177; H, H, H, Et, S, Oi -Pr, H, H, H, O], [AC5178; H, H, H, Et, S, SMe, H, H, H] O, [AC 5179; H, H, H, Et, S, SEt , H, H, H, O], [AC 5180; H, H, H, Et, S, CH ₂ F, H, H, H, O], [AC 5181; H, H, H, Et, S, CHF _{2, H, H, H,} O], [AC5182; H, H, H, Et, S, CF 3, H, H, H, O],

[AC5183; H, H, H , Et, S, OCH 2 F, H, H, H, O], [AC5184; H, H, H, Et, S, OCHF 2, H, H, H, O] , [AC5185; H, H, H, Et, S, OCF 3, H, H, H, O], [AC5186; H, H, H, Et, S, SCH 2 F, H, H, H, O ], [AC 5187; H, H, H, H, Et, S, SCHF ₂ , H, H, H, O], [AC 5188; H, H, H, Et, S, SCF ₃ , H, H, H, O H, H, H, Et, S, CN, H, H, H, O], [AC 5190; H, H, H, Et, S, NO ₂ , H, H, H, O] [AC5191; H, H, H, H, Pr, S, H, H, H, O], [AC5192; H, H, H, Pr, S, F, H, H, O], [AC5192 AC5193; H, H, H, H, Pr, S, Cl, H, H, H, O], [AC 5194; H, H, H, Pr, S, Br, H, H, H, O], [AC 5195; H, H, H, H, Pr, S, I, H, H, H, O], [AC 5196; H, H, H, Pr, S, Me, H, H, O], [AC 5 197; H, H, H, Pr, S, Et, H, H, H, O], [AC 5198; H, H, H, Pr, S, Pr, H, H, H, O], [AC 5199; H, H, H, Pr, S, i- Pr, H, H, H, O], [AC5200; H, H, H, Pr, S, CH = CH 2, H, H, H, O], [AC5201; H , H, H, Pr, S , C (CH 3) = CH 2, H, H, H, O], [AC5202; H, H, H, Pr, S, C≡CH, H, H, H, O, [AC 5203; H, H, H, H, Pr, S, C≡CCH ₃ , H, H, H, O], [AC 5204; H, H, H, Pr, S, c-Pr, H, H , H, O], [AC 5205; H, H, H, H, Pr, S, OMe, H, H, H, O], [AC 5206; H, H, H, Pr, S, OE t, H, H, H H, H, H, Pr, S, Oi-Pr, H, H, H, O], [AC 5208; H, H, H, Pr, S, SMe, H, H, H] H, H, H, Pr, S, SEt, H, H, H, O], [AC 5210; H, H, H, Pr, S, CH ₂ F, H, H, H , O], [AC5211; H , H, H, Pr, S, CHF 2, H, H, H, O], [AC5212; H, H, H, Pr, S, CF 3 , H, H, H, O ], [AC5213; H, H, H, Pr, S, OCH 2 F, H, H, H, O], [AC5214; H, H, H, Pr, S, OCHF _{2, H, H, H,} O], [AC5215; H, H, H, Pr, S, OCF 3, H, H, H, O], [AC5216; H, H, H, Pr, S, SCH ₂ F, H, H, H, O], [AC 5217; H, H, H, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 5218; H, H, H, Pr, S, SCF ₃ , H, H, H, O], [AC 5219; H, H, H, Pr, S, CN, H, H, H, O], [AC 5220; H, H, H, Pr, S, NO ₂ , H, H, H, O], [AC 5221; H, H, H, i-Pr, S, H, H, H, O], [AC 5222; H, H, H, i-Pr, S, F, H, H, H, O], [AC 5223; H, H, H, i-Pr, S, Cl, H, H, H, O], [AC 5224; H, H, H, i- Pr, S, Br, H, H, H, O], [AC 5225; H, H, H, i-Pr, S, I, H, H, O], [AC 5226; H, H, H, i-Pr, S, Me, H, H, H, O], [AC 5227; H, H, H, i-Pr, S, Et, H, H, O], [AC 5228; H, H, H, i-Pr, S, Pr, H, H, H, O], [AC5229; H, H, H, i-Pr, S, i-Pr, H, H, H, O], [AC 5230; H, H, H, i- Pr, S, CH = CH 2, H, H, H, O], [AC5231; H, H, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC5232; H, H, H, i-Pr, S, C≡CH, H, H, H, O], [AC 5233; H, H, H, i-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 5234; H, H, H, i-Pr, S, c-Pr, H, H, O], [AC 5235; H, H , H, i-Pr, S, OMe, H, H, H, O], [AC 5236; H, H, H, i-Pr, S, OEt, H, H, H, O], [AC 5237; H , H, H, i-Pr, S, Oi-Pr, H, H, H, O], [AC 5238; H, H, H, i-Pr, S, SMe, H, H, H, O], [AC5239; H, H, H , i-Pr, S, SEt, H, H, H, O], [AC5240; H, H, H, i-Pr, S, CH 2 F, H, H, H , O], [AC5241; H , H, H, i-Pr , S, CHF 2, H, H, H, O], [AC5242; H, H, H, i-Pr, S, CF 3, H, H, H, O], [AC5243; H, H, H , i-Pr, S, OCH 2 F, H, H, H, O], [AC5244; H, H, H, i-Pr, S, OCHF 2, H, H, H, O], [AC5245; H, H, H, i-Pr, S, OCF 3, H, H, H, O], [AC5246; H, H, H, i-Pr, S, SCH 2 F , H, H, H, O], [AC 5247; H, H, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 5248; H, H, H, i-Pr, S, SCF ₃ , H, H, H, O], [AC 5249; H, H, H, i-Pr, S, CN, H, H, H, O], [AC 5 250; H, H, H, i -Pr, S, NO ₂ , H, H, H, O], [AC 5251; H, H, H, c-Pr, S, H, H, H, O], [AC 5252; H, H, H, c-Pr, S, F, H, H, H, O], [AC5253; H, H, H, c-Pr, S, Cl, H, H, O], [AC5254; H, H, H, c-Pr, S, Br, H, H, H, O], [AC 5255; H, H, H, c-Pr, S, I, H, H, O], [AC 5 256; H, H, H, c-Pr, S, Me, H, H, H, O], [AC 5257; H, H, H, c-Pr, S, Et, H, H, H, O], [[ AC5258; H, H, H, c-Pr, S, Pr, H, H, H, O], [AC 5259; H, H, H, c-Pr, S, i-Pr, H, H, H, O], [AC5260; H, H, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC5261; H, H, H, c-Pr, S, C (CH _{3) = CH 2, H,} H, H, O], [AC5262; H, H, H, c-Pr, S, C≡CH, H, H, H, O], [AC5263; H, H, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 5264; H, H, H, c-Pr, S, c-Pr, H, H, H, O], [AC5265; H, H, H, c-Pr, S, OMe, H, H, H, O], [AC 5266; H, H, H, c-Pr, S, OEt, H, H, H, O H, H, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 5268; H, H, H, c-Pr, S, SMe, H, H] , H, O], [AC 5269; H, H, H, c-Pr, S, SEt, H, H, H, O], [AC5270; H, H, H, c-Pr, S, CH 2 F, H, H, H, O], [ AC5271; H, H, H, c-Pr, S, CHF 2, H, H, H, O], [AC5272; H, H, H, c-Pr, S, CF 3, H, H, H, O, [AC 5273; H, H, H, c, Pr, S, OCH ₂ F, H, H, H, O], [AC 5274; H, H, H, c, Pr, S, OCHF ₂ , H , H, H, O], [AC5275; H, H, H, c-Pr, S, OCF 3, H, H, H, O], [AC5276; H, H, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 5277; H, H, H, c-Pr, S, SCHF ₂ , H, H, H, O], [AC 5278; H, H, H, c _{-Pr, S, SCF 3, H} , H, H, O], [AC5279; H, H, H, c-Pr, S, CN, H, H, H, O], [AC5280; H, H, H, c-Pr, S, NO 2, H, H, H, O], [AC5281; H, H, H, SMe, S, H, H, H, H, O], [AC5282; H, H , H, SMe, S, F, H, H, H, O],

[AC 5283; H, H, H, SMe, S, Cl, H, H, H, O], [AC 5284; H, H, H, SMe, S, Br, H, H, O], [AC 5285 H, H, H, SMe, S, I, H, H, H, O], [AC5286; H, H, H, SMe, S, Me, H, H, O], [AC 5287; H , H, H, SMe, S, Et, H, H, H, O], [AC5288; H, H, H, SMe, S, Pr, H, H, H, O], [AC 5289; H, H , H, SMe, S, i -Pr, H, H, H, O], [AC5290; H, H, H, SMe, S, CH = CH 2, H, H, H, O], [AC5291; H, H, H, SMe, S, C (CH 3) = CH 2, H, H, H, O], [AC5292; H, H, H, SMe, S, C≡CH, H, H, H , O], [AC 5293; H, H, H, SMe, S, C≡CCH ₃ , H, H, H, O], [AC 5294; H, H, H, SMe, S, c-Pr, H, H, H, O], [AC 5295; H, H, H, SMe, S, OMe, H, H, H, O], [AC 5296; H, H, H, SMe, S, OEt, H, H, H, H, O], [AC 5297; H, H, H, SMe, S, Oi-Pr, H, H, H, O], [AC 5298; H, H, H, SMe, S, SMe, H, H, H, H, O], [AC 5299; H, H, H, SMe, S, SEt, H, H, H, O], [AC 5300; H, H, H, SMe, S, CH ₂ F, H, H, H, O], [AC 5301; H, H, H, S Me, S, CHF ₂ , H, H, H, O], [AC 5302; H, H, H, S Me, S, CF ₃ , H, H, H, O], [AC 5303; H, H, H, SMe, S, OCH ₂ F, H, H, H, O], [AC 5304; H, H, H, SMe, S, OCHF ₂ , H, H , H, O], [AC5305 ; H, H, H, SMe, S, OCF 3, H, H, H, O], [AC5306; H, H, H, SMe, S, SCH 2 F, H, H, H, O], [AC 5307; H, H, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 5308; H, H, H, SMe, S, SCF ₃ , H, H, H, O], [AC 5309; H, H, H, S Me, S, CN, H, H, H, O], [AC 5310; H, H, H, S Me, S, NO ₂ , H, H , H, O], [AC5311; H, H, H, OMe, S, H, H, H, H, O], [AC5312; H, H, H, OMe, S, F, H, H, H, O], [AC5313; H, H, H, OMe, S, Cl, H, H, H, O], [AC5314; H, H, H, OMe, S, Br, H, H, H, O], [AC5315; H, H, H, OMe, S, I, H, H, H, O], [AC5316; H, H, H, OMe, S, Me, H, H, H, O], [AC 5317; H, H, H, OMe, S, Et, H, H, H, H, H, H, OMe, S, Pr, H, H, H, O], [AC5319; H, H, H, OMe, S, i-Pr, H, H, H, O], [AC 5318; O], [AC5320; H, H, H, OMe, S, CH = CH 2, H, H, H, O], [AC5321; H, H, H, OMe, S, C (CH 3) = CH ₂ , H, H, H, O], [AC 5322; H, H, H, OMe, S, C≡CH, H, H, H, O], [AC 5323; H, H, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC5324; H, H, H, OMe, S, c-Pr, H, H, H, O], [AC5325; H, H, H, OMe , S, OMe, H, H, H, O], [AC5326; H, H, H, OMe, S, OEt, H, H, H, O], [AC 5327; H, H, H, OMe, S , Oi-Pr, H, H, H, O], [AC 5328; H, H, H, OMe, S, SMe, H, H, H, O], [AC 5329; H, H, H, OMe, S , SEt, H, H, H, O], [AC 5330; H, H, H, OMe, S, CH ₂ F, H, H, H, O], [AC 5331; H, H, H, OMe, S _{, CHF 2, H, H,} H, O], [AC5332; H, H, H, OMe, S, CF 3, H, H, H, O], [AC5333; H, H, H, OMe, S , OCH ₂ F, H, H, H, O], [AC 5334; H, H, H, OMe, S, OCHF ₂ , H, H, H, O], [AC 5335; H, H, H, OMe, _{S, OCF 3, H, H} , H, O], [AC5336; H, H, H, OMe, S, SCH 2 F, H, H, H, O], [AC5337; H, H, H, OMe , S, SCHF ₂ , H, H, H, O], [AC 5338; H, H, H, OMe, S, SCF ₃ , H, H, H, O], [AC 5339; H, H, H, OMe , S, CN, H, H, H, O], [AC5340; H, H, H, OMe , S, NO ₂ , H, H, H, O], [AC5341; H, H, H, F, S, H, H, H, H, O], [AC5342; H, H, H, F, S, F, H, H, H, O], [AC 5343; H, H, H, F, S, Cl, H, H, O], [AC 5344; H, H, H, F, S, Br, H, H, H, O], [AC 5345; H, H, H, F, S, I, H, H, H, O], [AC 5346; H, H, H, F, S, Me, H, H, H, O], [AC 5347; H, H, H, F, S, Et, H, H, H, O], [AC 5348; H, H, H, F, S, Pr, H, H, H, O], [AC 5349; H, H, H, F, S, i-Pr, H, H, H, O], [AC 5 350; H, H, H, F, S, CH = CH ₂ H, H, H, O], [AC 5351; H, H, H, F, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 5352; H, H, H, F, S, C≡CH, H, H, H, H, O], [AC 5353; H, H, H, F, S, C≡CCH ₃ , H, H, H, O], [AC 5354; H, H , H, F, S, c-Pr, H, H, H, O], [AC 5355; H, H, H, F, S, OMe, H, H, O], [AC 5356; H, H , H, F, S, OEt, H, H, H, O], [AC 5357; H, H, H, H, F, S, Oi-Pr, H, H, H, O], [AC 5358; H, H , H, F, S, SMe, H, H, H, O], [AC 5359; H, H, H, H, F, S, SE t, H, H, H, O], [AC 5360; H, H, H _{, F, S, CH 2 F} , H, H, H, O], [AC5361; H, H, H, F, S, CHF 2, H, H, H, O], [AC5362; H, H, _{H, F, S, CF 3} , H, H, H, O], [AC5363; H, H, H, F, S, OCH 2 F, H, H, H, O], [AC5364; H, H , H, F, S, OCHF ₂ , H, H, H, O], [AC 5365; H, H, H, H, F, S, OCF ₃ , H, H, H, O], [AC 5366; H, H , H, F, S, SCH ₂ F, H, H, H, O], [AC 5367; H, H, H, F, S, SCHF ₂ , H, H, H, O], [AC 5368; H, H, H, F, S, SCF 3, H, H, H, O], [AC5369; H, H, H, F, S, CN, H, H, H, O], [AC5370; H, H , H, F, S, NO ₂ , H, H, H, O], [A H, H, H, H, Cl, S, H, H, H, O], [AC5372; H, H, H, Cl, S, F, H, H, O], [AC 5373; H, H, H, H, Cl, S, Cl, H, H, H, O], [AC5374; H, H, H, Cl, S, Br, H, H, O], [AC 5375; H, H, H, Cl, S, I, H, H, H, O], [AC 5376; H, H, H, Cl, S, Me, H, H, O], [AC 5377; H, H, H, Cl, S, Et, H, H, H, O], [AC 5378; H, H, H, Cl, S, Pr, H, H, H, O], [AC 5379; H, H, H, Cl, S, i-Pr, H, H, H, O], [AC5380; H, H, H, Cl, S, CH = CH 2, H, H, H, O], [AC5381; H, H , H, Cl, S, C (CH 3) = CH 2, H, H, H, O], [AC5382; H, H, H, Cl, S, C≡CH, H, H, H, O] ,

[AC5383; H, H, H, H, Cl, S, C≡CCH ₃ , H, H, H, O], [AC5384; H, H, H, Cl, S, c-Pr, H, H, H, O, [AC5385; H, H, H, H, Cl, S, OMe, H, H, H, O], [AC 5386; H, H, H, Cl, S, OEt, H, H, H, O] [AC 5387; H, H, H, H, Cl, S, Oi-Pr, H, H, H, O], [AC 5388; H, H, H, H, Cl, S, SMe, H, H, H, O] , [AC5389; H, H, H, Cl, S, SEt, H, H, H, O], [AC5390; H, H, H, Cl, S, CH 2 F, H, H, H, O] , [AC5391; H, H, H, Cl, S, CHF 2, H, H, H, O], [AC5392; H, H, H, Cl, S, CF 3, H, H, H, O] , [AC5393; H, H, H, Cl, S, OCH 2 F, H, H, H, O], [AC5394; H, H, H, Cl, S, OCHF 2, H, H, H, O ], [AC5395; H, H , H, Cl, S, OCF 3, H, H, H, O], [AC5396; H, H, H, Cl, S, SCH 2 F, H, H, H, O], [AC5397; H, H, H, Cl, S, SCHF 2, H, H, H, O], [AC5398; H, H, H, Cl, S, SCF 3, H, H, H, O], [AC5399; H, H, H, Cl, S, CN, H, H, H, O], [AC5400; H, H, H, Cl, S, NO 2, H, H, H, O ], [AC5401; H, H, H, H, Br, S, H, H, H, O], [AC 5402; H, H, H, Br, S, F, H, H, H, O], [AC 5403; H, H, H, H, Br, S, Cl, H, H, H, O], [AC 5404; H, H, H, Br, S, Br, H, H, H, O], [AC 5405 H, H, H, H, Br, S, I, H, H, H, O], [AC 5406; H, H, H, Br, S, Me, H, H, O], [AC 5407; H , H, H, Br, S, Et, H, H, H, O], [AC 5408; H, H, H, H, Br, S, Pr, H, H, H, O], [AC 5409; H, H , H, Br, S, i -Pr, H, H, H, O], [AC5410; H, H, H, Br, S, CH = CH 2, H, H, H, O], [AC5411; H, H, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC5412; H, H, H, Br, S, C≡CH H, H, H, O], [AC 5413; H, H, H, Br, S, C≡CCH ₃ , H, H, H, O], [AC 5414; H, H, H, Br, S, c-Pr, H, H, H, O], [AC 5415; H, H, H, Br, S, OMe, H, H, H, O], [AC 5416; H, H, H, Br, S, OEt, H, H, H, O], [AC 5417; H, H, H, Br, S, Oi-Pr, H, H, H, O], [AC 5418; H, H, H, Br, S, SMe, H, H, H, O], [AC 5419; H, H, H, Br, S, SE t, H, H, H, O], [AC 5420; H, H, H, Br, S, CH ₂ F, H, H, H, O], [AC 5421; H, H, H, Br, S, CHF ₂ , H, H, H, O], [AC 5422; H, H, H, Br, S, CF _{3, H, H, H,} O], [AC5423; H, H, H, Br, S, OCH 2 F, H, H, H, O], [AC5424; H, H, H, Br, S, _{OCHF 2, H, H, H} , O], [AC5425; H, H, H, Br, S, OCF 3, H, H, H, O], [AC5426; H, H, H, Br, S, SCH ₂ F, H, H, H, O], [AC 5427; H, H, H, Br, S, SCHF ₂ , H, H, H, O], [AC 5428; H, H, H, Br, S , SCF ₃ , H, H, H, O], [AC 5429; H, H, H, Br, S, CN, H, H, H, O], [AC 5430; H, H, H, Br, S, _{NO 2, H, H, H} , O], [AC5431; H, Me, H, H, S, H, H, H, H, O], [AC5432; H, Me, H, H, S, F , H, H, H, O], [AC5433; H, Me, H, H, S, Cl, H, H, H, O], [AC 5434; H, Me, H, H, S, Br, H , H, H, O], [AC 5435; H, Me, H, H, S, I, H, H, H, O], [AC 5436; H, Me, H, H, S, Me, H, H H, O, [AC5437; H, Me, H, H, S, Et, H, H, H, O], [AC 5438; H, Me, H, H, S, Pr, H, H, H H, Me, H, H, S, i-Pr, H, H, H, O], [AC 5440; H, Me, H, H, S, CH = CH ₂ , H, H, H, O], [ AC5441; H, Me, H, H, S, C (CH 3) = CH 2, H, H, H, O], [AC5442; H, Me, H, H, S, C≡CH, H, H, H, O, [AC5443; H, Me, H, H, S, CSCCH ₃ , H, H, H, O], [AC5444; H, Me , H, H, S, c-Pr, H, H, H, O], [AC 5445; H, Me, H, H, S, OMe, H, H, O], [AC 5446; H, Me , H, H, S, OEt, H, H, H, O], [AC 5447; H, Me, H, H, S, Oi-Pr, H, H, H, O], [AC 5448; H, Me , H, H, S, SMe, H, H, H, O], [AC 5449; H, Me, H, H, S, SE t, H, H, H, O], [AC 5450; H, Me, H _{, H, S, CH 2 F} , H, H, H, O], [AC5451; H, Me, H, H, S, CHF 2, H, H, H, O], [AC5452; H, Me, _{H, H, S, CF 3} , H, H, H, O], [AC5453; H, Me, H, H, S, OCH 2 F, H, H, H, O], [AC5454; H, Me , H, H, S, OCHF 2, H, H, H, O], [AC5455; H, Me, H, H, S, OCF 3, H, H, H, O], [AC5456; H, Me , H, H, S, SCH ₂ F, H, H, H, O], [AC 5457; H, Me, H, H, S, SCHF ₂ , H, H, H, O], [AC 5458; H, Me, H, H, S, SCF 3, H, H, H, O], [AC5459; H, Me, H, H, S, CN, H, H, H, O], [AC5460; H, Me , H, H, S, NO 2, H, H, H, O], [AC5461; H, Me, H, Me, S, H, H, H, H, O], [AC5462; H, Me, H, Me, S, F, H, H, H, O], [AC5463; H, Me, H, Me, S, Cl, H, H, H, O], [AC5464; H, Me, H, Me, S, Br, H, H, H, O], [AC 5465; H, Me, H, Me, S, I, H, H, H, O], [AC 5466; H, Me, H, Me, S, Me, H, H, H, O], [AC 5467; H, Me, H, Me, S, Et, H, H, H, O], [AC 5468; H, Me, H, Me, S, Pr, H, H, H, O], [AC 5469; H, Me, H, Me, S, i-Pr, H, H, H, O], [AC 5470; H, Me, H, Me, S, CH = CH ₂ , H, H, H, O], [AC 5471; H, Me, H, Me, S, C (CH ₃ ) = CH ₂ , H, H , H, O], [AC5472; H, Me, H, Me, S, C, CH, H, H, H, O], [AC5473; H, Me, H, Me, S, CCHCCH ₃ , H, H, H, O], [AC5474; H, Me, H, Me, S, c-Pr, H, H, H, O], [AC 5475; H, Me, H, Me, S, OMe, H, H, H, O], [AC 5476; H, Me, H, Me, S, OEt, H, H, H, O], [AC 5477; H, Me, H, Me, S, Oi-Pr, H, H, H, O], [AC 5478; H, Me, H, Me, S, SMe, H, H, H, O], [AC 5479; H, Me, H, Me, S, SE t, H, H, H, O], [ AC5480; H, Me, H, Me, S, CH 2 F, H, H, H, O], [AC5481; H, Me, H, Me, S, CHF 2, H , H, H, O],

[AC5482; H, Me, H , Me, S, CF 3, H, H, H, O], [AC5483; H, Me, H, Me, S, OCH 2 F, H, H, H, O] , [AC 5484; H, Me, H, Me, S, OCHF ₂ , H, H, H, O], [AC 5485; H, Me, H, Me, S, OCF ₃ , H, H, H, O] H, Me, H, Me, S, SCH ₂ F, H, H, H, O], [AC 5487; H, Me, H, Me, S, SCHF ₂ , H, H, H, O H, Me, H, Me, S, SCF ₃ , H, H, H, O], [AC 5489; H, Me, H, Me, S, CN, H, H, H, O] , [AC5490; H, Me, H, Me, S, NO 2, H, H, H, O], [AC5491; H, Me, H, Et, S, H, H, H, H, O], [AC5492; H, Me, H, Et, S, F, H, H, O], [AC5493; H, Me, H, Et, S, Cl, H, H, H, O], [AC5494 H, Me, H, Et, S, Br, H, H, H, O], [AC5495; H, Me, H, Et, S, I, H, H, H, O], [AC 5496; H , Me, H, Et, S, Me, H, H, H, O], [AC5497; H, Me, H, Et, S, Et, H, H, H, O], [AC 5498; H, Me , H, Et, S, Pr, H, H, H, O], [AC5499; H, Me, H, Et, S, i-Pr, H, H, H, O], [AC 5500; H, Me , H, Et, S, CH = CH 2, H, H, H, O], [AC5501; H, Me, H, Et, S, C (CH 3) = CH 2, H, H, H, O H, Me, H, Et, S, C≡CH, H, H, H, O], [AC5503; H, Me, H, Et, S, C≡CCH ₃ , H, H, H, O], [AC5504; H, Me, H, Et, S, c-Pr, H, H, H, O], [AC 5505; H, Me, H, Et, S, OMe, H, H, H, O], [AC5506; H, Me, H, Et, S, OEt, H, H, H, O], [AC 5507; H, Me, H, Et, S, Oi-Pr, H, H, H, O], [AC 5508; H, Me, H, Et, S, SMe, H, H, H, O], [AC 5509; H, Me, H, Et, S, SE t, H, H, H, O], [AC 5510; H, Me, H, Et, S, CH ₂ F, H, H, H , O], [AC5511; H , Me, H, Et, S, CHF 2, H, H, H, O], [AC5512; H, Me, H, Et, S, CF 3, H, H, H , O], [AC5513; H , Me, H, Et, S, OCH 2 F, H, H, H, O], [AC5514; H, Me, H, Et, S, OCHF 2, H, H, H, O], [AC5515; H, Me, H, Et, S, OCF 3, H, H, H, O], [AC5516; H, Me, H, Et, S, SCH 2 F, H, H , H, O], [AC 5517; H, Me, H, Et, S, SCHF ₂ , H, H, H, O], [AC 5518; H, Me, H, Et, S, SCF ₃ , H, H , H, O], [AC5519; H, Me, H, Et, S, CN, H, H, H, O], [AC 5520; H, Me, H, Et, S, NO ₂ , H, H, H, O], [AC 5521; H, Me, H, Pr, S, H, H, H, O], [AC 5522; H, Me, H, Pr, S, F, H, H, H, H, O], [AC5523; H, Me, H, Pr, S, Cl, H, H, O], [AC5524; H, Me, H, Pr, S, Br, H, H, H, O] , [AC 5525; H, Me, H, Pr, S, I, H, H, O], [AC 5526; H, Me, H, Pr, S, Me, H, H, H, O], [AC 5526; AC5527; H, Me, H, Pr, S, Et, H, H, H, O], [AC5528; H, Me, H, Pr, S, Pr, H, H, H, O], [AC5529; H, Me, H, Pr, S, i-Pr, H, H, H, O], [AC5530; H, Me, H, Pr, S, CH = CH 2, H, H, H, O], [AC5531; H, Me, H , Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC5532; H, Me, H, Pr, S, C≡CH, H, H, H, O], [AC 5533; H, Me, H, Pr, S, C≡CCH ₃ , H, H, H, O], [AC 5534; H, Me, H, Pr, S, c-Pr H, H, H, O], [AC 5535; H, Me, H, Pr, S, OMe, H, H, H, O], [AC 5536; H, Me, H, Pr, S, OE t, H , H, H, O], [AC 5537; H, Me, H, Pr, S, Oi-Pr, H, H, H, O], [AC 5538; H, Me, H, Pr, S, SMe, H , H, H, O], [AC 5539; H, Me, H, Pr, S, SEt, H , H, H, O], [AC5540; H, Me, H, Pr, S, CH 2 F, H, H, H, O], [AC5541; H, Me, H, Pr, S, CHF 2, H, H, H, O] , [AC5542; H, Me, H, Pr, S, CF 3, H, H, H, O], [AC5543; H, Me, H, Pr, S, OCH 2 F H, H, H, O], [AC 5544; H, Me, H, Pr, S, OCHF ₂ , H, H, H, O], [AC 5545; H, Me, H, Pr, S, OCF ₃ H, H, H, O], [AC 5546; H, Me, H, Pr, S, SCH ₂ F, H, H, H, O], [AC 5547; H, Me, H, Pr, S, SCHF _{2, H, H, H,} O], [AC5548; H, Me, H, Pr, S, SCF 3, H, H, H, O], [AC5549; H, Me, H, Pr, S, CN , H, H, H, O ], [AC5550; H, Me, H, Pr, S, NO 2, H, H, H, O], [AC5551; H, Me, H, i-Pr, S, H, H, H, H, O], [AC5552; H, Me, H, i-Pr, S, F, H, H, O], [AC5553; H, Me, H, i-Pr, S, Cl, H, H, H, O], [AC5554; H, Me, H, i-Pr, S, Br, H, H, H, O], [AC5555; H, Me, H, i- Pr, S, I, H, H, H, O], [AC5556; H, Me, H, i-Pr, S, Me, H, H, O], [AC 5557; H, Me, H, i-Pr, S, Et, H, H, H, O], [AC 5558; H, Me, H, i-Pr, S, Pr, H, H, O], [AC 5559; H, Me, H, i-Pr, S, i-Pr, H, H, H, O], [AC5560; H, Me, H, i-Pr, S, CH = CH 2, H, H, H, O], [AC5561; H, Me, H , i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC5562; H, Me, H, i-Pr, S, C≡ CH, H, H, H, O], [AC5563; H, Me, H, i-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 5564; H, Me, H, i -Pr, S, c-Pr, H, H, H, O], [AC 5565; H, Me, H, i-Pr, S, OMe, H, H, O], [AC 5 566; H, Me , H, i-Pr, S, OEt, H, H, H, O], [AC 5567; H, Me, H, i-Pr, S , Oi-Pr, H, H, H, O], [AC 5568; H, Me, H, i-Pr, S, SMe, H, H, H, O], [AC 5569; H, Me, H, i -Pr, S, SEt, H, H, H, O], [AC5570; H, Me, H, i-Pr, S, CH 2 F, H, H, H, O], [AC5571; H, Me , H, i-Pr, S , CHF 2, H, H, H, O], [AC5572; H, Me, H, i-Pr, S, CF 3, H, H, H, O], [AC5573 ; H, Me, H, i -Pr, S, OCH 2 F, H, H, H, O], [AC5574; H, Me, H, i-Pr, S, OCHF 2, H, H, H, O], [AC5575; H, Me, H, i-Pr, S, OCF 3, H, H, H, O], [AC5576; H, Me, H, i-Pr, S, SCH 2 F, H , H, H, O], [AC 5577; H, Me, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 5578; H, Me, H, i-Pr, S, SCF ₃ , H, H, H, O], [AC 5579; H, Me, H, i-Pr, S, CN, H, H, H, O], [AC 5580; H, Me, H, i-Pr , S, NO ₂ , H, H, H, O], [AC5581; H, Me, H, c-Pr, S, H, H, H, H, O],

[AC5582; H, Me, H, c-Pr, S, F, H, H, O], [AC 5583; H, Me, H, c-Pr, S, Cl, H, H, H, O H, Me, H, c-Pr, S, Br, H, H, O], [AC 5585; H, Me, H, c-Pr, S, I, H, H, H] , O], [AC5586; H, Me, H, c-Pr, S, Me, H, H, H, O], [AC5587; H, Me, H, c-Pr, S, Et, H, H , H, O], [AC 5588; H, Me, H, c-Pr, S, Pr, H, H, H, O], [AC 5589; H, Me, H, c-Pr, S, i-Pr , H, H, H, O ], [AC5590; H, Me, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC5591; H, Me, H, c- Pr, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC5592; H, Me, H, c-Pr, S, C≡CH, H, H, H, O], [AC5593; H, Me, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC5594; H, Me, H, c-Pr, S, c-Pr, H, H, H, O], [AC5595; H, Me, H, c-Pr, S, OMe, H, H, H, O], [AC 5596; H, Me, H, c-Pr, S, OE t, H, H, H, O], [AC 5597; H, Me, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 5598; H, Me, H, c-Pr, S, SMe, H, H, H, O], [AC 5599; H, Me, H, c-Pr, S, SE t, H, H, H, O], [AC 5600; H, Me, H, c- _{Pr, S, CH 2 F,} H, H, H, O], [AC5601; H, Me, H, c-Pr, S, CHF 2, H, H, H, O], [AC5602; H, Me , H, c-Pr, S , CF 3, H, H, H, O], [AC5603; H, Me, H, c-Pr, S, OCH 2 F, H, H, H, O], [ AC 5604; H, Me, H, c-Pr, S, OCHF ₂ , H, H, H, O], [AC 5605; H, Me, H, c-Pr, S, OCF ₃ , H, H, H, O, [AC5606; H, Me, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 5607; H, Me, H, c-Pr, S, SCHF ₂ , H , H, H, O], [AC 5608; H, Me, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 5 H, Me, H, c-Pr, S, CN, H, H, H, O], [AC 5610; H, Me, H, c-Pr, S, NO ₂ , H, H, H, O H, Me, H, SMe, S, H, H, H, H, O], [AC5612; H, Me, H, SMe, S, F, H, H, H, O], [AC 5613; H, Me, H, SMe, S, Cl, H, H, H, O], [AC 5614; H, Me, H, SMe, S, Br, H, H, O], [AC 5615 H, Me, H, SMe, S, I, H, H, H, O], [AC 5616; H, Me, H, SMe, S, Me, H, H, O], [AC 5617; H , Me, H, SMe, S, Et, H, H, H, O], [AC 5618; H, Me, H, SMe, S, Pr, H, H, O], [AC 5619; H, Me , H, SMe, S, i -Pr, H, H, H, O], [AC5620; H, Me, H, SMe, S, CH = CH 2, H, H, H, O], [AC5621; H, Me, H, SMe, S, C (CH 3) = CH 2, H, H, H, O], [AC5622; H, Me, H, SMe, S, C≡CH, H, H, H H, Me, H, SMe, S, C≡CCH ₃ , H, H, H, O], [AC 5624; H, Me, H, SMe, S, c-Pr, H, H, H, O], [AC 5625; H, Me, H, SMe, S, OMe, H, H, H, O], [AC 5626; H, Me, H, SMe, S, OEt, H, H, H, H, O], [AC5627; H, Me, H, SMe, S, Oi-Pr, H, H, H, O], [AC5628; H, Me, H, SMe, S, SMe, H, H, H, H, O], [AC 5629; H, Me, H, S Me, S, SE t, H, H, H, O], [AC 5630; H, Me, H, S Me, S, CH ₂ F, H, H, H, O], [AC5631; H, Me, H, SMe, S, CHF 2, H, H, H, O], [AC5632; H, Me, H, SMe, S, CF 3, H, H, H, O], [AC5633; H, Me, H, SMe, S, OCH 2 F, H, H, H, O], [AC5634; H, Me, H, SMe, S, OCHF 2, H, H , H, O], [AC5635 ; H, Me, H, SMe, S, OCF 3, H, H, H, O], [AC5636; H, Me, H, SMe, S, SCH 2 F, H, H, H, O], [AC5637 H, Me, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 5638; H, Me, H, SMe, S, SCF ₃ , H, H, H, O], [AC 5639 H, Me, H, SMe, S, CN, H, H, H, O], [AC 5640; H, Me, H, SMe, S, NO ₂ , H, H, H, O], [AC 564 1; H, Me, H, OMe, S, H, H, H, H, O], [AC5642; H, Me, H, OMe, S, F, H, H, O], [AC5643; H, Me, H, OMe, S, Cl, H, H, H, O], [AC 5644; H, Me, H, OMe, S, Br, H, H, O], [AC 5645; H, Me, H, OMe, S, I, H, H, H, O], [AC 5646; H, Me, H, OMe, S, Me, H, H, O], [AC 5647; H, Me, H, OMe, S, Et, H, H, H, O], [AC 5648; H, Me, H, OMe, S, Pr, H, H, H, O], [AC 5649; H, Me, H, OMe, S, i-Pr, H, H, H, O], [AC5650; H, Me, H, OMe, S, CH = CH 2, H, H, H, O], [AC5651; H, Me, H , OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC5652; H, Me, H, OMe, S, C≡CH, H, H, H, O], [ AC5653; H, Me, H, OMe, S, C≡CCH 3, H, H, H, O], [AC5654; H, Me, H, OMe, S, c-Pr, H, H, H, O H, Me, H, OMe, S, OMe, H, H, H, O], [AC 5656; H, Me, H, OMe, S, OEt, H, H, H, O], [AC5657; H, Me, H, OMe, S, Oi-Pr, H, H, H, O], [AC5658; H, Me, H, OMe, S, SMe, H, H, H, O], [AC 5659; H, Me, H, OMe, S, SEt, H, H, H, O], [AC 5660; H, Me, H, OMe, S, CH ₂ F, H, H, H, O], [AC5661; H, Me, H , OMe, S, CHF 2, H, H, H, O], [AC5662; H, Me, H, OMe, S, CF 3, H, H, H, O], [AC5663; H, Me, H , OMe, S, OCH 2 F, H, H, H, O], [AC5664; H, Me, H, OMe, S, OCHF 2, H, H, H, O] , [AC5665; H, Me , H, OMe, S, OCF 3, H, H, H, O], [AC5666; H, Me, H, OMe, S, SCH 2 F, H, H, H, O], [AC5667; H, Me, H, OMe, S, SCHF 2, H, H, H, O], [AC5668; H, Me, H, OMe, S, SCF 3, H, H, H, O], [AC5669; H, Me, H, OMe, S, CN, H, H, H, O], [AC 5670; H, Me, H, OMe, S, NO ₂ , H, H, H, O], [AC 5671; H, Me , H, F, S, H, H, H, H, O], [AC 5672; H, Me, H, F, S, F, H, H, O], [AC 5673; H, Me, H , F, S, Cl, H, H, H, O], [AC 5674; H, Me, H, F, S, Br, H, H, H, O], [AC 5675; H, Me, H, F , S, I, H, H, H, O], [AC 5 676; H, Me, H, F, S, Me, H, H, H, O], [AC 5677; H, Me, H, F, S , Et, H, H, H, O], [AC5678; H, Me, H, F, S, Pr, H, H, H, O], [AC 5679; H, Me, H, F, S, i -Pr, H, H, H, O], [AC 5680; H, Me, H, F, S, CH = CH ₂ , H, H, H, O], [AC5681; H, Me, H, F, _{S, C (CH 3) =} CH 2, H, H, H, O],

[AC5682; H, Me, H, F, S, C≡CH, H, H, H, O], [AC5683; H, Me, H, F, S, C≡CCH ₃ , H, H, H, O, [AC5684; H, Me, H, F, S, c-Pr, H, H, H, O], [AC 5685; H, Me, H, F, S, OMe, H, H, H, H, Me, H, F, S, OEt, H, H, H, O], [AC5687; H, Me, H, F, S, Oi-Pr, H, H, H, O], [AC 5686; O, [AC 5688; H, Me, H, F, S, SMe, H, H, H, O], [AC 5689; H, Me, H, F, S, SE t, H, H, H, O] , [AC5690; H, Me, H, F, S, CH 2 F, H, H, H, O], [AC5691; H, Me, H, F, S, CHF 2, H, H, H, O ], [AC5692; H, Me , H, F, S, CF 3, H, H, H, O], [AC5693; H, Me, H, F, S, OCH 2 F, H, H, H, O, [AC 5694; H, Me, H, F, S, OCHF ₂ , H, H, H, O], [AC 5695; H, Me, H, F, S, OCF ₃ , H, H, H, H, Me, H, F, S, SCH ₂ F, H, H, H, O], [AC 5697; H, Me, H, F, S, SCHF ₂ , H, H, H] H, Me, H, F, S, SCF ₃ , H, H, H, O], [AC 5699; H, Me, H, F, S, CN, H, H, H, H O], [AC5700; H, Me, H, F, S, NO 2, H, H, H, O], [AC5701; H, Me, H, Cl, S, H, H, H, H, O H, Me, H, Cl, S, F, H, H, O], [AC 5703; H, Me, H, Cl, S, Cl, H, H, H, O], [AC 5704; H, Me, H, Cl, S, Br, H, H, O], [AC 5705; H, Me, H, Cl, S, I, H, H, O], [AC 5706 H, Me, H, Cl, S, Me, H, H, H, O], [AC 5707; H, Me, H, Cl, S, Et, H, H, H, O], [AC 5708; H , Me, H, Cl, S, Pr, H, H, H, O], [AC 5709; H, Me, H, Cl, S, i-Pr, H, H, H, O], [AC 5710; H , Me, H, Cl, S , CH = CH 2, H, H, H, O], [AC5711; H, Me, H, Cl, S, C (C H ₃ ) = CH ₂ , H, H, H, O], [AC 5712; H, Me, H, Cl, S, C≡CH, H, H, H, O], [AC 5713; H, Me, H , Cl, S, C≡CCH ₃ , H, H, H, O], [AC5714; H, Me, H, Cl, S, c-Pr, H, H, O], [AC5715; H, Me, H, Cl, S, OMe, H, H, H, O], [AC5716; H, Me, H, Cl, S, OEt, H, H, H, O], [AC 5717; H, Me, H, Cl, S, Oi-Pr, H, H, H, O], [AC5718; H, Me, H, Cl, S, SMe, H, H, O], [AC5719; H, Me, H, Cl, S, SEt, H, H, H, O], [AC5720; H, Me, H, Cl, S, CH 2 F, H, H, H, O], [AC5721; H, Me, _{H, Cl, S, CHF 2} , H, H, H, O], [AC5722; H, Me, H, Cl, S, CF 3, H, H, H, O], [AC5723; H, Me, _{H, Cl, S, OCH 2} F, H, H, H, O], [AC5724; H, Me, H, Cl, S, OCHF 2, H, H, H, O], [AC5725; H, Me , H, Cl, S, OCF 3, H, H, H, O], [AC5726; H, Me, H, Cl, S, SCH 2 F, H, H, H, O], [AC5727; H, Me, H, Cl, S, SCHF 2, H, H, H, O], [AC5728; H, Me, H, Cl, S, SCF 3, H, H, H, O], [AC5729; H, Me, H, Cl, S, CN, H, H, H, O], [AC5730; H, Me, H, Cl, S, NO 2, H, H, H, O], [AC5731; H, Me , H, Br, S, H, H, H, H, O], [AC5732; H, Me, H, Br, S, F, H, H, H, O], [AC 5733; H, Me, H , Br, S, Cl, H, H, H, O], [AC 5734; H, Me, H, Br, S, Br, H, H, H, O], [AC 5735; H, Me, H, Br] , S, I, H, H, H, O], [AC 5736; H, Me, H, Br, S, Me, H, H, H, O], [AC 5737; H, Me, H, Br, S , Et, H, H, H, O], [AC 5738; H, Me, H, Br, S, Pr, H, H, H, O], [AC 5739; H, Me, H, Br, S, i -Pr, H, H, H, O], [AC 5740; H, Me, H, Br, S, C _{H = CH 2, H, H} , H, O], [AC5741; H, Me, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC5742; H, Me, H, Br, S, C≡CH, H, H, H, O], [AC5743; H, Me, H, Br, S, C≡CCH ₃ , H, H, H, O], [AC 5744 H, Me, H, Br, S, c-Pr, H, H, H, O], [AC5745; H, Me, H, Br, S, OMe, H, H, H, O], [AC5746 H, Me, H, Br, S, OEt, H, H, H, O], [AC 5747; H, Me, H, Br, S, Oi-Pr, H, H, H, O], [AC 5748 H, Me, H, Br, S, SMe, H, H, H, O], [AC 5749; H, Me, H, Br, S, SE, H, H, H, O], [AC 5750; H , Me, H, Br, S , CH 2 F, H, H, H, O], [AC5751; H, Me, H, Br, S, CHF 2, H, H, H, O], [AC5752; H, Me, H, Br, S, CF 3, H, H, H, O], [AC5753; H, Me, H, Br, S, OCH 2 F, H, H, H, O], [AC5754 H, Me, H, Br, S, OCHF ₂ , H, H, H, O], [AC 5755; H, Me, H, Br, S, OCF ₃ , H, H, H, O], [AC 5756 H, Me, H, Br, S, SCH ₂ F, H, H, H, O], [AC 5757; H, Me, H, Br, S, SCHF ₂ , H, H, H, O], [[ AC 5758; H, Me, H, Br, S, SCF ₃ , H, H, H, O], [AC 5759; H, Me, H, Br, S, CN, H, H, H, O], [AC 5760 ; H, Me, H, Br , S, NO 2, H, H, H, O], [AC5761; H, Et, H, H, S, H, H, H, H, O], [AC5762; H, Et, H, H, S, F, H, H, H, O], [AC5763; H, Et, H, H, S, Cl, H, H, O], [AC 5764; H, Et, H, H, S, Br, H, H, H, O], [AC 5765; H, Et, H, H, S, I, H, H, O], [AC 5766; H, Et, H, H, S, Me, H, H, H, O, [AC 5767; H, Et, H, H, S, Et, H, H, H, O], [AC 5768; H, Et, H, H, S, Pr, H, H, H, O], [AC 5769; H, Et, H, H, S, i-Pr , H, H, H, O ], [AC5770; H, Et, H, H, S, CH = CH 2, H, H, H, O], [AC5771; H, Et, H, H, S, _{C (CH 3) = CH 2} , H, H, H, O], [AC5772; H, Et, H, H, S, C≡CH, H, H, H, O], [AC5773; H, Et , H, H, S, C≡CCH ₃ , H, H, H, O], [AC 5774; H, Et, H, H, S, c-Pr, H, H, H, O], [AC 5775; H, Et, H, H, S, OMe, H, H, H, O], [AC5776; H, Et, H, H, S, OEt, H, H, H, O], [AC 5777; H, Et, H, H, S, Oi-Pr, H, H, H, O], [AC 5778; H, Et, H, H, S, SMe, H, H, O], [AC 5779; H, Et, H, H, S, S, SEt, H, H, H, O], [AC 5780; H, Et, H, H, S, CH ₂ F, H, H, H, O],

[AC5781; H, Et, H , H, S, CHF 2, H, H, H, O], [AC5782; H, Et, H, H, S, CF 3, H, H, H, O], [AC5783; H, Et, H , H, S, OCH 2 F, H, H, H, O], [AC5784; H, Et, H, H, S, OCHF 2, H, H, H, O] , [AC5785; H, Et, H, H, S, OCF 3, H, H, H, O], [AC5786; H, Et, H, H, S, SCH 2 F, H, H, H, O H, Et, H, H, S, SCHF ₂ , H, H, H, O], [AC 5788; H, Et, H, H, S, SCF ₃ , H, H, H, O] H, Et, H, H, S, CN, H, H, H, O], [AC 5790; H, Et, H, H, S, NO ₂ , H, H, H, O] [AC5791; H, Et, H, Me, S, H, H, H, O], [AC5792; H, Et, H, Me, S, F, H, H, O], [AC5792; AC5793; H, Et, H, Me, S, Cl, H, H, H, O], [AC5794; H, Et, H, Me, S, Br, H, H, H, O], [AC5795; H, Et, H, Me, S, I, H, H, H, O], [AC5796; H, Et, H, Me, S, Me, H, H, O], [AC5797; H, Et, H, Me, S, Et, H, H, H, O], [AC 5798; H, Et, H, Me, S, Pr, H, H, H, O], [AC 5799; H, Et, H, Me, S, i- Pr, H, H, H, O], [AC5800; H, Et, H, Me, S, CH = CH 2, H, H, H, O], [AC5801; H , Et, H, Me, S , C (CH 3) = CH 2, H, H, H, O], [AC5802; H, Et, H, Me, S, C≡CH, H, H, H, O, [AC5803; H, Et, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 5804; H, Et, H, Me, S, c-Pr, H, H , H, O], [AC 5805; H, Et, H, Me, S, OMe, H, H, H, O], [AC 5806; H, Et, H, Me, S, OEt, H, H, H H, Et, H, Me, S, Oi-Pr, H, H, H, O], [AC 5808; H, Et, H, Me, S, SMe, H, H, H] , O], [AC 5809; H, Et, H, Me, S, SE t, H, H, H, O], [AC 581 0; H, Et, H, Me, S, CH 2 F, H, H, H, O], [AC5811; H, Et, H, Me, S, CHF 2, H, H, H, O], [AC5812; H, Et, H , Me, S, CF 3, H, H, H, O], [AC5813; H, Et, H, Me, S, OCH 2 F, H, H, H, O] , [AC5814; H, Et, H, Me, S, OCHF 2, H, H, H, O], [AC5815; H, Et, H, Me, S, OCF 3, H, H, H, O] [AC 5816; H, Et, H, Me, S, SCH ₂ F, H, H, H, O], [AC 5817; H, Et, H, Me, S, SCHF ₂ , H, H, H, O H, Et, H, Me, S, SCF ₃ , H, H, H, O], [AC 5819; H, Et, H, Me, S, CN, H, H, H, O] [AC 5820; H, Et, H, Me, S, NO ₂ , H, H, O], [AC 5821; H, Et, H, Et, S, H, H, H, H, O], [AC 5822; H, Et, H, Et, S, F, H, H, O], [AC 5823; H, Et, H, Et, S, Cl, H, H, H, O], [AC 5824 H, Et, H, Et, S, Br, H, H, H, O], [AC 5825; H, Et, H, Et, S, I, H, H, H, O], [AC 5826; H , Et, H, Et, S, Me, H, H, H, O], [AC 5827; H, Et, H, Et, S, Et, H, H, H, O], [AC 5828; H, Et , H, Et, S, Pr, H, H, H, O], [AC 5829; H, Et, H, Et, S, i-Pr, H, H, H, O], [AC 5830; H, Et , H, Et, S, CH = CH 2, H, H, H, O], [AC5831; H, Et, H, Et, S, C (CH 3) = CH 2, H, H, H, O H, Et, H, Et, S, C≡CH, H, H, H, O], [AC 5833; H, Et, H, Et, S, C≡CCH ₃ , H, H, H] H, O], [AC 5834; H, Et, H, Et, S, c, Pr, H, H, H, O], [AC 5835; H, Et, H, Et, S, OMe, H, H, H, O], [AC 5836; H, Et, H, Et, S, OEt, H, H, H, O], [AC 5837; H, Et, H, Et, S, Oi-Pr, H, H, H, O], [AC 5838; H, Et, H, Et, S, SMe, H, H, H, O] , [AC 5839; H, Et, H, Et, S, SE t, H, H, H, O], [AC 5840; H, Et, H, Et, S, CH ₂ F, H, H, H, O] , [AC5841; H, Et, H, Et, S, CHF 2, H, H, H, O], [AC5842; H, Et, H, Et, S, CF 3, H, H, H, O] , [AC5843; H, Et, H, Et, S, OCH 2 F, H, H, H, O], [AC5844; H, Et, H, Et, S, OCHF 2, H, H, H, O ], [AC5845; H, Et , H, Et, S, OCF 3, H, H, H, O], [AC5846; H, Et, H, Et, S, SCH 2 F, H, H, H, O], [AC 5847; H, Et, H, Et, S, SCHF ₂ , H, H, H, O], [AC 5848; H, Et, H, Et, S, SCF ₃ , H, H, H, O], [AC 5849; H, Et, H, Et, S, CN, H, H, H, O], [AC 5850; H, Et, H, Et, S, NO ₂ , H, H, H, O ], [AC 5851; H, Et, H, Pr, S, H, H, H, H, O], [AC 5852; H, Et, H, Pr, S, F, H, H, H, O], [AC 5853; H, Et, H, Pr, S, Cl, H, H, H, O], [AC 5854; H, Et, H, Pr, S, Br, H, H, H, O], [AC 5855] H, Et, H, Pr, S, I, H, H, H, O], [AC 5856; H, Et, H, Pr, S, Me, H, H, O], [AC 5857; H , Et, H, Pr, S, Et, H, H, H, O], [AC 5858; H, Et, H, Pr, S, Pr, H, H, H, O], [AC 5859; H, Et , H, Pr, S, i -Pr, H, H, H, O], [AC5860; H, Et, H, Pr, S, CH = CH 2, H, H, H, O], [AC5861; H, Et, H, Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC5862; H, Et, H, Pr, S, C≡CH, H, H, H , O], [AC5863; H , Et, H, Pr, S, C≡CCH 3, H, H, H, O], [AC5864; H, Et, H, Pr, S, c-Pr, H, H, H, O], [AC 5865; H, Et, H, Pr, S, OMe, H, H, H, O], [AC 5866; H, Et, H, Pr, S, OE t, H, H, H, O], [AC5867; H, Et, H, Pr, S, Oi-Pr, H , H, H, O], [AC5868; H, Et, H, Pr, S, SMe, H, H, H, O], [AC 5869; H, Et, H, Pr, S, SEt, H, H , H, O], [AC5870 ; H, Et, H, Pr, S, CH 2 F, H, H, H, O], [AC5871; H, Et, H, Pr, S, CHF 2, H, H, H, O], [ AC5872; H, Et, H, Pr, S, CF 3, H, H, H, O], [AC5873; H, Et, H, Pr, S, OCH 2 F, H , H, H, O], [AC 5874; H, Et, H, Pr, S, OCHF ₂ , H, H, H, O], [AC 5875; H, Et, H, Pr, S, OCF ₃ , H , H, H, O], [AC 5876; H, Et, H, Pr, S, SCH ₂ F, H, H, H, O], [AC 5877; H, Et, H, Pr, S, SCHF ₂ , H, H, H, O] , [AC5878; H, Et, H, Pr, S, SCF 3, H, H, H, O], [AC5879; H, Et, H, Pr, S, CN, H , H, H, O], [AC 5880; H, Et, H, Pr, S, NO ₂ , H, H, H, O],

[AC 5881; H, Et, H, i-Pr, S, H, H, H, H, O], [AC 5882; H, Et, H, i-Pr, S, F, H, H, H, O H, Et, H, i-Pr, S, Cl, H, H, H, O], [AC 5884; H, Et, H, i-Pr, S, Br, H, H, H] , O], [AC 5885; H, Et, H, i-Pr, S, I, H, H, H, O], [AC 5886; H, Et, H, i-Pr, S, Me, H, H , H, O], [AC 5887; H, Et, H, i-Pr, S, Et, H, H, H, O], [AC 5888; H, Et, H, i-Pr, S, Pr, H , H, H, O], [AC 5889; H, Et, H, i-Pr, S, i-Pr, H, H, H, O], [AC 5890; H, Et, H, i-Pr, S , CH = CH ₂ , H, H, H, O], [AC5891; H, Et, H, i-Pr, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC5892 H, Et, H, i-Pr, S, C≡CH, H, H, H, O], [AC5893; H, Et, H, i-Pr, S, C≡CCH ₃ , H, H, H H, O], [AC 5894; H, Et, H, i-Pr, S, c-Pr, H, H, H, O], [AC 5895; H, Et, H, i-Pr, S, OMe, H, H, H, O], [AC 5896; H, Et, H, i-Pr, S, OEt, H, H, H, O], [AC5897; H, Et, H, i-Pr, S, Oi-Pr, H, H, H, O], [AC 5898; H, Et, H, i-Pr, S, SMe, H, H, H, O], [AC 5899; H, Et, H, i- Pr, S, SEt, H, H, H, O], [AC5900; H, Et, H, i-Pr, S, CH 2 F, H, H, H, O], [AC5901; H, Et, H, i-Pr, S, CHF 2, H, H, H, O], [AC5902; H, Et, H, i-Pr, S, CF 3, H, H, H, O], [AC5903; H, Et, H, i- Pr, S, OCH 2 F, H, H, H, O], [AC5904; H, Et, H, i-Pr, S, OCHF 2, H, H, H, O ], [AC5905; H, Et , H, i-Pr, S, OCF 3, H, H, H, O], [AC5906; H, Et, H, i-Pr, S, SCH 2 F, H, H, H, O], [AC 5907; H, Et, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 5908; H , Et, H, i-Pr , S, SCF 3, H, H, H, O], [AC5909; H, Et, H, i-Pr, S, CN, H, H, H, O], [ AC5910; H, Et, H, i-Pr, S, NO 2, H, H, H, O], [AC5911; H, Et, H, c-Pr, S, H, H, H, H, O H, Et, H, c-Pr, S, F, H, H, H, O], [AC 5913; H, Et, H, c-Pr, S, Cl, H, H, H] , O], [AC5914; H, Et, H, c-Pr, S, Br, H, H, H, O], [AC 5915; H, Et, H, c-Pr, S, I, H, H H, O, [AC5916; H, Et, H, c-Pr, S, Me, H, H, H, O], [AC5917; H, Et, H, c-Pr, S, Et, H , H, H, O], [AC5918; H, Et, H, c-Pr, S, Pr, H, H, H, O], [AC5919; H, Et, H, c-Pr, S, i -Pr, H, H, H, O], [AC5920; H, Et, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC5921; H, Et, H, c-Pr, S, C ( CH 3) = CH 2, H, H, H, O], [AC5922; H, Et, H, c-Pr, S, C≡CH, H, H, H, O H, Et, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 5924; H, Et, H, c-Pr, S, c-Pr, H, H, H, O], [AC5925; H, Et, H, c-Pr, S, OMe, H, H, H, O], [AC 5926; H, Et, H, c-Pr, S, OEt, H, H, H, O], [AC 5927; H, Et, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 5928; H, Et, H, c- Pr, S, SMe, H, H, H, O], [AC5929; H, Et, H, c-Pr, S, SEt, H, H, H, O], [AC5930; H, Et, H, _{c-Pr, S, CH 2} F, H, H, H, O], [AC5931; H, Et, H, c-Pr, S, CHF 2, H, H, H, O], [AC5932; H , Et, H, c-Pr , S, CF 3, H, H, H, O], [AC5933; H, Et, H, c-Pr, S, OCH 2 F, H, H, H, O] , [AC5934; H, Et, H, c-Pr, S, OCHF 2, H, H, H, O], [AC5935; H, Et, H, c-Pr, S, OCF _{3, H, H, H,} O], [AC5936; H, Et, H, c-Pr, S, SCH 2 F, H, H, H, O], [AC5937; H, Et, H, c- Pr, S, SCHF ₂ , H, H, H, O], [AC 5938; H, Et, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 5939; H, Et, H, c-Pr, S, CN, H, H, H, O], [AC5940; H, Et, H, c-Pr, S, NO 2, H, H, H, O], [AC5941; H , Et, H, SMe, S, H, H, H, H, O], [AC5942; H, Et, H, SMe, S, F, H, H, O], [AC5943; H, Et , H, SMe, S, Cl, H, H, H, O], [AC 5944; H, Et, H, SMe, S, Br, H, H, O], [AC 5945; H, Et, H , SMe, S, I, H, H, H, O], [AC 5946; H, Et, H, SMe, S, Me, H, H, H, O], [AC 5947; H, Et, H, SMe , S, Et, H, H, H, O], [AC5948; H, Et, H, SMe, S, Pr, H, H, H, O], [AC 5949; H, Et, H, SMe, S , i-Pr, H, H , H, O], [AC5950; H, Et, H, SMe, S, CH = CH 2, H, H, H, O], [AC5951; H, Et, H, _{SMe, S, C (CH 3} ) = CH 2, H, H, H, O], [AC5952; H, Et, H, SMe, S, C≡CH, H, H, H, O], [AC5953 H, Et, H, SMe, S, C≡CCH ₃ , H, H, H, O], [AC5954; H, Et, H, SMe, S, c-Pr, H, H, H, O] H, Et, H, SMe, S, OMe, H, H, H, O], [AC5956; H, Et, H, SMe, S, OEt, H, H, H, O], [AC 5955; AC 5957; H, Et, H, SMe, S, Oi-Pr, H, H, H, O], [AC5958; H, Et, H, SMe, S, SMe, H, H, H, O], [[ AC 5959; H, Et, H, SMe, S, SEt, H, H, H, O], [AC 5960; H, Et, H, SMe, S, CH ₂ F, H, H, H, O], [ AC5961; H, Et, H, SMe, S, CHF 2, H, H, H, O], [AC5962; H, Et, H, SMe, S, CF 3, H, H, H, O], [ AC 5963; H, Et, H, SMe, S, OCH _{2 F, H, H, H} , O], [AC5964; H, Et, H, SMe, S, OCHF 2, H, H, H, O], [AC5965; H, Et, H, SMe, S, _{OCF 3, H, H, H} , O], [AC5966; H, Et, H, SMe, S, SCH 2 F, H, H, H, O], [AC5967; H, Et, H, SMe, S _{, SCHF 2, H, H,} H, O], [AC5968; H, Et, H, SMe, S, SCF 3, H, H, H, O], [AC5969; H, Et, H, SMe, S , CN, H, H, H, O], [AC 5970; H, Et, H, SMe, S, NO ₂ , H, H, H, O], [AC 5971; H, Et, H, OMe, S, H, H, H, H, O], [AC 5972; H, Et, H, OMe, S, F, H, H, H, O], [AC 5973; H, Et, H, OMe, S, Cl, H, H, H, O], [AC 5974; H, Et, H, OMe, S, Br, H, H, H, O], [AC5975; H, Et, H, OMe, S, I, H, H, H, O], [AC5976; H, Et, H, OMe, S, Me, H, H, H, O], [AC 5977; H, Et, H, OMe, S, Et, H, H, H, O], [AC5978; H, Et, H, OMe, S, Pr, H, H, H, O], [AC5979; H, Et, H, OMe, S, i-Pr, H, H, H, O], [AC 5 980; H, Et, H, OMe, S, CH = CH ₂ , H, H, H, O],

[AC5981; H, Et, H , OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC5982; H, Et, H, OMe, S, C≡CH, H, H, H, O], [AC 5983; H, Et, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC 5984; H, Et, H, OMe, S, c-Pr , H, H, H, O], [AC5985; H, Et, H, OMe, S, OMe, H, H, H, O], [AC5986; H, Et, H, OMe, S, OEt, H , H, H, O], [AC5987; H, Et, H, OMe, S, Oi-Pr, H, H, H, O], [AC5988; H, Et, H, OMe, S, SMe, H , H, H, O], [AC 5989; H, Et, H, OMe, S, SE t, H, H, H, O], [AC 5990; H, Et, H, OMe, S, CH ₂ F, H , H, H, O], [AC5991; H, Et, H, OMe, S, CHF 2, H, H, H, O], [AC5992; H, Et, H, OMe, S, CF 3, H , H, H, O], [AC5993; H, Et, H, OMe, S, OCH 2 F, H, H, H, O], [AC5994; H, Et, H, OMe, S, OCHF 2, H, H, H, O] , [AC5995; H, Et, H, OMe, S, OCF 3, H, H, H, O], [AC5996; H, Et, H, OMe, S, SCH 2 F , H, H, H, O], [AC5997; H, Et, H, OMe, S, SCHF ₂ , H, H, H, O], [AC5998; H, Et, H, OMe, S, SCF ₃ , H, H, H, O], [AC 5 999; H, Et, H, OMe, S, CN, H, H, H, O], [AC 6000; H, Et, H, OMe, S, NO ₂ , H, H, H, O], [AC 6001; H, Et, H, F, S, H, H, H, H, O], [AC 6002; H, Et, H, F, S, F, H, H, H, O], [AC 6003; H, Et, H, F, S, Cl, H, H, H, O], [AC 6004; H, Et, H, F, S, Br, H, H, H, O], [AC 6005; H, Et, H, F, S, I, H, H, H, O], [AC 6006; H, Et, H, F, S, Me, H, H, H, H, O], [AC 6007; H, Et, H, F, S, Et, H, H, H, O], [AC 6008; H, Et, H, F, S, Pr, H, H, H, O] , [AC 6009; H, Et, H, F, S, i -Pr, H, H, H, O], [AC6010; H, Et, H, F, S, CH = CH 2, H, H, H, O], [AC6011; H, Et, H, F, _{S, C (CH 3) =} CH 2, H, H, H, O], [AC6012; H, Et, H, F, S, C≡CH, H, H, H, O], [AC6013; H , Et, H, F, S, C≡CCH ₃ , H, H, H, O], [AC 6014; H, Et, H, F, S, c-Pr, H, H, H, O], [[ AC 6015; H, Et, H, F, S, OMe, H, H, H, O], [AC 6016; H, Et, H, F, S, OEt, H, H, H, O], [AC 6017; H, Et, H, F, S, Oi-Pr, H, H, H, O], [AC 6018; H, Et, H, F, S, SMe, H, H, O], [AC 6019; H, Et, H, F, S, SEt, H, H, H, O], [AC 6020; H, Et, H, F, S, CH ₂ F, H, H, H] O, [AC 6021; H, Et, H, F, S, CHF 2, H, H, H, O], [AC6022; H, Et, H, F, S, CF 3, H, H, H, O], [AC6023; H, Et, H, F, S, OCH 2 F, H, H, H, O], [AC6024; H, Et, H, F, S, OCHF 2, H, H, H, O], [AC6025 ; H, Et, H, F , S, OCF 3, H, H, H, O], [AC6026; H, Et, H, F, S, SCH 2 F, H, H, H, O], [ AC 6027; H, Et, H, F, S, SCHF ₂ , H, H, H, O], [AC 6028; H, Et, H, F, S, SCF ₃ , H, H, H, O], [ AC 6029; H, Et, H, F, S, CN, H, H, H, O], [AC 6030; H, Et, H, F, S, NO ₂ , H, H, H, O], [AC6031 H, Et, H, Cl, S, H, H, H, H, O], [AC6032; H, Et, H, Cl, S, F, H, H, O], [AC6033; H , Et, H, Cl, S, Cl, H, H, H, O], [AC 6034; H, Et, H, Cl, S, Br, H, H, O], [AC 6035; H, Et , H, Cl, S, I, H, H, H, O], [AC6036; H, Et, H, Cl, S, Me, H, H, H, O], [AC 6037; H, Et, H , Cl, S, Et, H, H, H, O], [AC 6038; H, Et, H, Cl, S, Pr, H, H, H, O], [A C6039; H, Et, H, Cl, S, i-Pr, H, H, H, O], [AC6040; H, Et, H, Cl, S, CH = CH 2, H, H, H, O ], [AC6041; H, Et , H, Cl, S, C (CH 3) = CH 2, H, H, H, O], [AC6042; H, Et, H, Cl, S, C≡CH, H, H, H, O] , [AC6043; H, Et, H, Cl, S, C≡CCH 3, H, H, H, O], [AC6044; H, Et, H, Cl, S, c -Pr, H, H, H, O], [AC 6045; H, Et, H, Cl, S, OMe, H, H, H, O], [AC 6046; H, Et, H, Cl, S, OEt , H, H, H, O], [AC 6047; H, Et, H, Cl, S, Oi-Pr, H, H, H, O], [AC 6048; H, Et, H, Cl, S, SMe , H, H, H, O], [AC 6049; H, Et, H, Cl, S, SE t, H, H, H, O], [AC 6050; H, Et, H, Cl, S, CH ₂ F , H, H, H, O ], [AC6051; H, Et, H, Cl, S, CHF 2, H, H, H, O], [AC6052; H, Et, H, Cl, S, CF 3 , H, H, H, O ], [AC6053; H, Et, H, Cl, S, OCH 2 F, H, H, H, O], [AC6054; H, Et, H, Cl, S, OCHF _{2, H, H, H,} O], [AC6055; H, Et, H, Cl, S, OCF 3, H, H, H, O], [AC6056; H, Et, H, Cl, S, SCH _{2 F, H, H, H} , O], [AC6057; H, Et, H, Cl, S, SCHF 2, H, H, H, O], [AC6058; H, Et, H, Cl, S, SCF ₃ , H, H, H, O], [AC 6059; H, Et, H, Cl, S, CN, H, H, H, O], [AC 6060; H, Et, H, Cl, S, NO ₂ , H, H, H, O], [AC 6061; H, Et, H, Br, S, H, H, H, H, O], [AC 6062; H, Et, H, Br, S, F, H, H, H, O], [AC 6063; H, Et, H, Br, S, Cl, H, H, H, O], [AC 6064; H, Et, H, Br, S, Br, H, H, H, O], [AC 6065; H, Et, H, Br, S, I, H, H, H, O], [AC 6066; H, Et, H, Br, S, Me, H, H, H, H, O], [AC 6067; H, Et, H, Br, S, Et, H, H , H, O], [AC 6068; H, Et, H, Br, S, Pr, H, H, H, O], [AC 6069; H, Et, H, Br, S, i-Pr, H, H , H, O], [AC6070 ; H, Et, H, Br, S, CH = CH 2, H, H, H, O], [AC6071; H, Et, H, Br, S, C (CH 3 ) = CH ₂ , H, H, H, O], [AC6072; H, Et, H, Br, S, CEtCH, H, H, H, O], [AC 6073; H, Et, H, Br] , S, C≡CCH ₃ , H, H, H, O], [AC 6074; H, Et, H, Br, S, c-Pr, H, H, H, O], [AC 6075; H, Et, H, Br, S, OMe, H, H, H, O], [AC 6076; H, Et, H, Br, S, OEt, H, H, H, O], [AC 6077; H, Et, H, Br, S, Oi-Pr, H, H, H, O, [AC 6078; H, Et, H, Br, S, SMe, H, H, O], [AC 6079; H, Et, H, Br, S, SEt, H, H, H, O],

[AC6080; H, Et, H , Br, S, CH 2 F, H, H, H, O], [AC6081; H, Et, H, Br, S, CHF 2, H, H, H, O] , [AC6082; H, Et, H, Br, S, CF 3, H, H, H, O], [AC6083; H, Et, H, Br, S, OCH 2 F, H, H, H, O ], [AC6084; H, Et , H, Br, S, OCHF 2, H, H, H, O], [AC6085; H, Et, H, Br, S, OCF 3, H, H, H, O H, Et, H, Br, S, SCH ₂ F, H, H, H, O], [AC 6087; H, Et, H, Br, S, SCHF ₂ , H, H, H, O], [AC 6088; H, Et, H, Br, S, SCF ₃ , H, H, H, O], [AC 6089; H, Et, H, Br, S, CN, H, H, H, O ], [AC 6090; H, Et, H, Br, S, NO ₂ , H, H, O], [AC 6091; H, Pr, H, H, S, H, H, H, H, O] [AC6092; H, Pr, H, H, S, F, H, H, O], [AC 6093; H, Pr, H, H, S, Cl, H, H, O], [AC 6093; AC 6094; H, Pr, H, H, S, Br, H, H, O], [AC 6095; H, Pr, H, H, S, I, H, H, O], [AC 6096; H, Pr, H, H, S, Me, H, H, H, O], [AC 6097; H, Pr, H, H, S, Et, H, H, H] O, [AC 6098; H, Pr, H, H, S, Pr, H, H, H, O], [AC 6099; H, Pr, H, H, S, i-Pr, H, H, H, O], [AC 6100; H, Pr, H, H, S, CH = CH 2, H, H, H, O], [AC6101; H, Pr, H, H, S, C (CH 3) = CH 2, H, H, H, O, [AC6102; H, Pr, H, H, S, C≡CH, H, H, H, O], [AC 6103; H, Pr, H, H, S, C≡ CCH ₃ , H, H , H, O], [AC 6104; H, Pr, H, H, S, c-Pr, H, H, H, O], [AC 6105; H, Pr, H, H, S, OMe, H, H , H, O], [AC 6106; H, Pr, H, H, S, OEt, H, H, H, O], [AC 6107; H, Pr, H, H, S, Oi-Pr, H, H , H, O], [AC 6108; H, Pr, H, H, S, SMe, H, H, H, O], [AC 6109; H, P r, H, H, S, SEt, H, H, H, O], [AC6110; H, Pr, H, H, S, CH 2 F, H, H, H, O], [AC6111; H, Pr, H, H, S, CHF 2, H, H, H, O], [AC6112; H, Pr, H, H, S, CF 3, H, H, H, O], [AC6113; H, Pr, H, H, S, OCH 2 F, H, H, H, O], [AC6114; H, Pr, H, H, S, OCHF 2, H, H, H, O], [AC6115; H , Pr, H, H, S , OCF 3, H, H, H, O], [AC6116; H, Pr, H, H, S, SCH 2 F, H, H, H, O], [AC6117; H, Pr, H, H, S, SCHF ₂ , H, H, H, O], [AC 6118; H, Pr, H, H, S, SCF ₃ , H, H, H, O], [AC 6119; H, Pr, H, H, S, CN, H, H, H, O], [AC 6120; H, Pr, H, H, S, NO ₂ , H, H, H, O], [AC 6121; H , Pr, H, Me, S, H, H, H, H, O], [AC 6122; H, Pr, H, Me, S, F, H, H, O], [AC 6123; H, Pr , H, Me, S, Cl, H, H, H, O], [AC 6124; H, Pr, H, Me, S, Br, H, H, H, O], [AC 6 125; H, Pr, H , Me, S, I, H, H, H, O], [AC 6126; H, Pr, H, Me, S, Me, H, H, H, O], [AC 6127; H, Pr, H, Me , S, Et, H, H, H, O, [AC 6128; H, Pr, H, Me, S, Pr, H, H, H, O], [AC 6129; H, Pr, H, Me, S , i-Pr, H, H, H, O], [AC 6130; H, Pr, H, Me, S, CH = CH ₂ , H, H, H, O], [AC 6131; H, Pr, H, _{Me, S, C (CH 3} ) = CH 2, H, H, H, O], [AC6132; H, Pr, H, Me, S, C≡CH, H, H, H, O], [AC6133 H, Pr, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 6134; H, Pr, H, Me, S, c-Pr, H, H, H, O] , [AC 6135; H, Pr, H, Me, S, OMe, H, H, H, O], [AC 6136; H, Pr, H, Me, S, OEt, H, H, H, O], [ AC 6137; H, Pr, H, Me, S, Oi-Pr, H, H, H, O], [AC 6138; H, Pr, H, M e, S, SMe, H, H, H, O], [AC 6139; H, Pr, H, Me, S, SE t, H, H, H, O], [AC 6140; H, Pr, H, Me, _{S, CH 2 F, H,} H, H, O], [AC6141; H, Pr, H, Me, S, CHF 2, H, H, H, O], [AC6142; H, Pr, H, Me _{, S, CF 3, H,} H, H, O], [AC6143; H, Pr, H, Me, S, OCH 2 F, H, H, H, O], [AC6144; H, Pr, H, _{Me, S, OCHF 2, H} , H, H, O], [AC6145; H, Pr, H, Me, S, OCF 3, H, H, H, O], [AC6146; H, Pr, H, Me, S, SCH ₂ F, H, H, H, H, O], [AC 6147; H, Pr, H, Me, S, SCHF ₂ , H, H, H, O], [AC 6148; H, Pr, H , Me, S, SCF ₃ , H, H, H, O], [AC 6149; H, Pr, H, Me, S, CN, H, H, H, O], [AC 6150; H, Pr, H, _{Me, S, NO 2, H} , H, H, O], [AC6151; H, Pr, H, Et, S, H, H, H, H, O], [AC6152; H, Pr, H, Et , S, F, H, H, H, O, [AC6153; H, Pr, H, Et, S, Cl, H, H, H, O], [AC 6154; H, Pr, H, Et, S , Br, H, H, H, O], [AC 6155; H, Pr, H, Et, S, I, H, H, H, O], [AC 6156; H, Pr, H, Et, S, Me H, H, H, O], [AC 6157; H, Pr, H, Et, S, Et, H, H, H, O], [AC 6158; H, Pr, H, Et, S, Pr, H H, H, O], [AC 6159; H, Pr, H, Et, S, i-Pr, H, H, H, O], [AC 6160; H, Pr, H, Et, S, CH = CH _{2, H, H, H,} O], [AC6161; H, Pr, H, Et, S, C (CH 3) = CH 2, H, H, H, O], [AC6162; H, Pr, H , Et, S, C≡CH, H, H, H, O], [AC 6163; H, Pr, H, Et, S, C≡ CCH ₃ , H, H, H, O], [AC 6 164; H, Pr, H, Et, S, c-Pr, H, H, H, O], [AC 6165; H, Pr, H, Et, S, OMe, H, H, O], [AC 6166; H, Pr, H, Et, S, OEt, H, H, H, O], [AC 6167; H, P r, H, Et, S, Oi-Pr, H, H, H, O], [AC 6168; H, Pr, H, Et, S, SMe, H, H, O], [AC 6169; H, Pr, H, Et, S, SEt, H, H, H, O], [AC6170; H, Pr, H, Et, S, CH 2 F, H, H, H, O], [AC6171; H, Pr, H, Et, S, CHF 2, H, H, H, O], [AC6172; H, Pr, H, Et, S, CF 3, H, H, H, O], [AC6173; H, Pr, H, Et, S, OCH 2 F, H, H, H, O], [AC6174; H, Pr, H, Et, S, OCHF 2, H, H, H, O], [AC6175; H , Pr, H, Et, S , OCF 3, H, H, H, O], [AC6176; H, Pr, H, Et, S, SCH 2 F, H, H, H, O], [AC6177; H, Pr, H, Et, S, SCHF ₂ , H, H, H, O], [AC 6178; H, Pr, H, Et, S, SCF ₃ , H, H, H, O], [AC 6179; H, Pr, H, Et, S, CN, H, H, H, O],

[AC 6 180; H, Pr, H, Et, S, NO ₂ , H, H, H, O], [AC 6181; H, Pr, H, Pr, S, H, H, H, O, [, AC 6182; H, Pr, H, Pr, S, F, H, H, O], [AC 6183; H, Pr, H, Pr, S, Cl, H, H, H, O], [AC 6184; H, Pr, H, Pr, S, Br, H, H, H, O], [AC 6185; H, Pr, H, Pr, S, I, H, H, O], [AC 6186; H, Pr, H, Pr, S, Me, H, H, H, O], [AC 6187; H, Pr, H, Pr, S, Et, H, H, H, O], [AC 6188; H, Pr, H, Pr, S, Pr, H, H, H, H, O], [AC 6189; H, Pr, H, Pr, S, i-Pr, H, H, H, O], [AC 6190; H, Pr, H, Pr, S, CH = CH 2, H, H, H, O], [AC6191; H, Pr, H, Pr, S, C (CH 3) = CH 2, H, H, H, O] [AC6192; H, Pr, H, Pr, S, C≡CH, H, H, H, O], [AC 6193; H, Pr, H, Pr, S, C≡CCH ₃ , H, H, H , O], [AC 6194; H, Pr, H, Pr, S, c-Pr, H, H, H, O], [AC 6195; H, Pr, H, Pr, S, OMe, H, H, H H, Pr, H, Pr, S, OEt, H, H, H, O], [AC 6197; H, Pr, H, Pr, S, Oi-Pr, H, H, H , O], [AC 6198; H, Pr, H, Pr, S, SMe, H, H, H, O], [AC 6199; H, Pr, H, Pr, S, SE t, H, H, H, O ], [AC6200; H, Pr , H, Pr, S, CH 2 F, H, H, H, O], [AC6201; H, Pr, H, Pr, S, CHF 2, H, H, H, O], [AC6202; H, Pr, H, Pr, S, CF 3, H, H, H, O], [AC6203; H, Pr, H, Pr, S, OCH 2 F, H, H, H H, Pr, H, Pr, S, OCHF ₂ , H, H, H, O], [AC 6205; H, Pr, H, Pr, S, OCF ₃ , H, H, H , O], [AC 6206; H, Pr, H, Pr, S, SCH ₂ F, H, H, H, O], [AC 6207; H, Pr, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 6208; H, Pr, H, Pr, S, SCF ₃ , H H, H, O], [AC 6209; H, Pr, H, Pr, S, CN, H, H, H, O], [AC 6210; H, Pr, H, Pr, S, NO ₂ , H, H, H, O], [AC6211; H, Pr, H, i-Pr, S, H, H, H, H, O], [AC 6212; H, Pr, H, i-Pr, S, F, H, H, H, O], [AC 6213; H, Pr, H, i-Pr, S, Cl, H, H, H, O], [AC 6214; H, Pr, H, i-Pr, S, Br, H, H, H, O], [AC 6215; H, Pr, H, i-Pr, S, I, H, H, H, O], [AC 6216; H, Pr, H, i-Pr, S, Me, H, H, H, O], [AC 6217; H, Pr, H, i-Pr, S, Et, H, H, H, O], [AC 6218; H, Pr, H, i- Pr, S, Pr, H, H, H, H, O], [AC 6219; H, Pr, H, i-Pr, S, i-Pr, H, H, H, O], [AC 6220; H, Pr, H, i-Pr, S, CH = CH 2, H, H, H, O], [AC6221; H, Pr, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC 6222; H, Pr, H, i-Pr, S, C≡CH, H, H, H, O], [AC 6223; H, Pr, H, i-Pr, S, C ≡ CCH ₃ , H, H, H, O], [AC 6224; H, Pr, H, i-Pr, S, c-Pr, H, H, H, O], [AC 6225; H, Pr, H, i -Pr, S, OMe, H, H, H, O], [AC6226; H, Pr, H, i-Pr, S, OEt, H, H, H, O], [AC 6227; H, Pr, H , i-Pr, S, Oi-Pr, H, H, H, O], [AC 6 228; H, Pr, H, i-Pr, S, SMe, H, H, O], [AC 6229; H , Pr, H, i-Pr, S, SEt, H, H, H, O], [AC 6230; H, Pr, H, i-Pr, S, CH ₂ F, H, H, H, O], [AC6231; H, Pr, H , i-Pr, S, CHF 2, H, H, H, O], [AC6232; H, Pr, H, i-Pr, S, CF 3, H, H, H , O], [AC6233; H , Pr, H, i-Pr, S, OCH 2 F, H, H, H, O], [AC6234; H, Pr, H, i-Pr, S, OCHF 2, H, H, H, O] , [AC6235; H, Pr, H, i-Pr, S, OCF 3, H, H, H, O], [AC6236; H, Pr , H, i-Pr, S, SCH ₂ F, H, H, H, O], [AC 6237; H, Pr, H, i-Pr, S, SCHF ₂ , H, H, H, O], [[ AC6238; H, Pr, H, i-Pr, S, SCF 3, H, H, H, O], [AC6239; H, Pr, H, i-Pr, S, CN, H, H, H, O ], [AC6240; H, Pr , H, i-Pr, S, NO 2, H, H, H, O], [AC6241; H, Pr, H, c-Pr, S, H, H, H, H, O], [AC6242; H, Pr, H, c-Pr, S, F, H, H, H, O], [AC6243; H, Pr, H, c-Pr, S, Cl, H, H, H, O], [AC6244; H, Pr, H, c-Pr, S, Br, H, H, H, O], [AC 6245; H, Pr, H, c-Pr, S, I, H, H, H, O], [AC 6246; H, Pr, H, c-Pr, S, Me, H, H, H, O], [AC 6247; H, Pr, H, c-Pr, S, Et, H, H, H, O], [AC 6248; H, Pr, H, c-Pr, S, Pr, H, H, H, O], [AC 6249; H, Pr, H, c-Pr, S, i-Pr, H, H, H, O], [AC6250; H, Pr, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC6251; H, Pr , H, c-Pr, S , C (CH 3) = CH 2, H, H, H, O], [AC6252; H, Pr, H, c-Pr, S, C≡CH, H, H, H, O], [AC6253; H, Pr, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC6254; H, Pr, H, c-Pr, S, c -Pr, H, H, H, O], [AC 6 255; H, Pr, H, c-Pr, S, OMe, H, H, H, O], [AC 6 256; H, Pr, H, c-Pr , S, OEt, H, H, H, O], [AC 6 257; H, Pr, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 6258; H, Pr, H , c-Pr, S, SMe, H, H, H, O], [AC 6259; H, Pr, H, c-Pr, S, SEt, H, H, H, O], [AC 6260; H, Pr , H, c-Pr, S , CH 2 F, H, H, H, O], [AC6261; H, Pr, H, c-Pr, S, CHF 2, H, H, H, O], [ AC6262; H, Pr, H, c-Pr, S, CF 3, H, H, H, O], [AC6263; H, Pr, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC 6264; H, Pr, H, c-Pr, S, OCHF ₂ , H, H, H, O], [AC 6265; H, Pr, H, c-Pr , S, OCF ₃ , H, H, H, O], [AC 6266; H, Pr, H, c-Pr, S, SCH ₂ F, H, H, O], [AC 6 267; H, Pr, H, c-Pr, S, SCHF 2, H, H, H, O], [AC6268; H, Pr, H, c-Pr, S, SCF 3, H, H, H, O], [AC6269; H, Pr, H, c-Pr, S, CN, H, H, H, O], [AC 6270; H, Pr, H, c-Pr, S, NO ₂ , H, H, H, O], [AC6271; H, Pr, H, SMe, S, H, H, H, O], [AC6272; H, Pr, H, SMe, S, F, H, H, O], [AC6273 H, Pr, H, SMe, S, Cl, H, H, H, O], [AC 6274; H, Pr, H, SMe, S, Br, H, H, O], [AC 6275; H , Pr, H, SMe, S, I, H, H, H, O], [AC 6276; H, Pr, H, SMe, S, Me, H, H, O], [AC 6277; H, Pr , H, SMe, S, Et, H, H, H, O], [AC 6278; H, Pr, H, SMe, S, Pr, H, H, H, O], [AC 6279; H, Pr, H , SMe, S, i-Pr, H, H, H, O],

[AC6280; H, Pr, H , SMe, S, CH = CH 2, H, H, H, O], [AC6281; H, Pr, H, SMe, S, C (CH 3) = CH 2, H H, H, O], [AC6282; H, Pr, H, SMe, S, C≡CH, H, H, H, O], [AC6283; H, Pr, H, SMe, S, C≡ CCH ₃ , H, H, H, O], [AC 6284; H, Pr, H, SMe, S, c-Pr, H, H, H, O], [AC 6285; H, Pr, H, SMe, S, OMe, H, H, H, O], [AC 6286; H, Pr, H, SMe, S, OEt, H, H, H, O], [AC 6287; H, Pr, H, SMe, S, Oi- Pr, H, H, H, O], [AC 6288; H, Pr, H, SMe, S, SMe, H, H, H, O], [AC 6289; H, Pr, H, SMe, S, SEt, H, H, H, O] , [AC6290; H, Pr, H, SMe, S, CH 2 F, H, H, H, O], [AC6291; H, Pr, H, SMe, S, CHF 2 , H, H, H, O ], [AC6292; H, Pr, H, SMe, S, CF 3, H, H, H, O], [AC6293; H, Pr, H, SMe, S, OCH 2 F, H, H, H, O], [AC6294; H, Pr, H, SMe, S, OCHF 2, H, H, H, O], [AC6295; H, Pr, H, SMe, S, OCF _{3, H, H, H,} O], [AC6296; H, Pr, H, SMe, S, SCH 2 F, H, H, H, O], [AC6297; H, Pr, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 6298; H, Pr, H, SMe, S, SCF ₃ , H, H, H, O], [AC 6299; H, Pr, H, SMe, S, CN, H, H, H, O], [AC 6300; H, Pr, H, SMe, S, NO ₂ , H, H, H, O], [AC 6301; H, Pr, H, OMe, S, H H, H, H, O], [AC6302; H, Pr, H, OMe, S, F, H, H, H, O], [AC6303; H, Pr, H, OMe, S, Cl, H] H, H, O], [AC 6304; H, Pr, H, OMe, S, Br, H, H, H, O], [AC 6305; H, Pr, H, OMe, S, I, H, H H, O], [AC 6306; H, Pr, H, OMe, S, Me, H, H, H, O], [AC 6307; H, Pr, H, OMe, S, Et, H, H, H , O H, Pr, H, OMe, S, Pr, H, H, H, O], [AC 6309; H, Pr, H, OMe, S, i-Pr, H, H, H, O] H, Pr, H, OMe, S, CH = CH ₂ , H, H, H, O], [AC 6311; H, Pr, H, OMe, S, C (CH ₃ ) = CH _2] H, H, H, O], [AC 6312; H, Pr, H, OMe, S, C≡CH, H, H, H, O], [AC 6313; H, Pr, H, OMe, S, C ≡ CCH ₃ , H, H, H, O], [AC6314; H, Pr, H, OMe, S, c-Pr, H, H, H, O], [AC 6315; H, Pr, H, OMe, S, OMe, H, H, H, O], [AC6316; H, Pr, H, OMe, S, OEt, H, H, H, O], [AC 6317; H, Pr, H, OMe, S, Oi-Pr, H, H, H, O], [AC 6318; H, Pr, H, OMe, S, SMe, H, H, H, O], [AC 6319; H, Pr, H, OMe, S, SEt, H, H, H, O], [AC6320; H, Pr, H, OMe, S, CH 2 F, H, H, H, O], [AC6321; H, Pr, H, OMe, S, _{CHF 2, H, H, H} , O], [AC6322; H, Pr, H, OMe, S, CF 3, H, H, H, O], [AC6323; H, Pr, H, OMe, S, _{OCH 2 F, H, H,} H, O], [AC6324; H, Pr, H, OMe, S, OCHF 2, H, H, H, O], [AC6325; H, Pr, H, OMe, S _{, OCF 3, H, H,} H, O], [AC6326; H, Pr, H, OMe, S, SCH 2 F, H, H, H, O], [AC6327; H, Pr, H, OMe, _{S, SCHF 2, H, H} , H, O], [AC6328; H, Pr, H, OMe, S, SCF 3, H, H, H, O], [AC6329; H, Pr, H, OMe, S, CN, H, H, H, O], [AC 6330; H, Pr, H, OMe, S, NO ₂ , H, H, H, O], [AC6331; H, Pr, H, F, S , H, H, H, H, O], [AC6332; H, Pr, H, F, S, F, H, H, O], [AC 6333; H, Pr, H, F, S, Cl H, H, H, O], [AC 6334; H, Pr, H, F, S, Br, H, H, H, O], [AC 6335; H, Pr, H, F, S, I, H , H, H, O], [AC 6 H, Pr, H, F, S, Me, H, H, H, O], [AC 6337; H, Pr, H, F, S, Et, H, H, H, O], [AC 6338; H, Pr, H, F, S, Pr, H, H, H, O], [AC6339; H, Pr, H, F, S, i-Pr, H, H, H, O], [AC 6340; H, Pr, H, F, S, CH = CH 2, H, H, H, O], [AC6341; H, Pr, H, F, S, C (CH 3) = CH 2, H, H, H, O], [AC6342; H, Pr, H, F, S, C≡CH, H, H, H, O], [AC6343; H, Pr, H, F, S, C≡ CCH ₃ , H H, H, O], [AC 6344; H, Pr, H, F, S, c-Pr, H, H, H, O], [AC 6345; H, Pr, H, F, S, OMe, H , H, H, O], [AC 6346; H, Pr, H, F, S, OEt, H, H, H, O], [AC 6347; H, Pr, H, F, S, Oi-Pr, H H, H, O], [AC 6348; H, Pr, H, F, S, SMe, H, H, H, O], [AC 6349; H, Pr, H, F, S, SE t, H, H , H, O], [AC6350 ; H, Pr, H, F, S, CH 2 F, H, H, H, O], [AC6351; H, Pr, H, F, S, CHF 2, H, H, H, O], [ AC6352; H, Pr, H, F, S, CF 3, H, H, H, O], [AC6353; H, Pr, H, F, S, OCH 2 F, H H, H, O], [AC 6354; H, Pr, H, F, S, OCHF ₂ , H, H, H, O], [AC 6355; H, Pr, H, F, S, OCF ₃ , H , H, H, O], [AC 6356; H, Pr, H, F, S, SCH ₂ F, H, H, H, O], [AC 6357; H, Pr, H, F, S, SCHF ₂ , H, H, H, O], [AC 6358; H, Pr, H, F, S, SCF ₃ , H, H, H, O], [AC 6359; H, Pr, H, F, S, CN, H , H, H, O], [AC 6360; H, Pr, H, F, S, NO ₂ , H, H, H, O], [AC6361; H, Pr, H, Cl, S, H, H, H, H, H, O], [AC6362; H, Pr, H, Cl, S, F, H, H, H, O], [AC6363; H, Pr, H, Cl, S, Cl, H, H, H, O], [AC 6364; H, Pr, H, Cl, S, Br, H, H, H, O], [AC 6365; H, Pr, H, Cl, S, H, Pr, H, H, H, O, [AC 6366; H, Pr, H, Cl, S, Me, H, H, H, O], [AC 6367; H, Pr, H, Cl, S, Et, H, H, H, O], [AC 6368; H, Pr, H, Cl, S, Pr, H, H, H, O], [AC 6369; H, Pr, H, Cl, S, i-Pr, H, H, H, O] , [AC6370; H, Pr, H, Cl, S, CH = CH 2, H, H, H, O], [AC6371; H, Pr, H, Cl, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC6372; H, Pr, H, Cl, S, C≡CH, H, H, H, O], [AC 6373; H, Pr, _{H, Cl, S, C≡CCH 3} , H, H, H, O], [AC6374; H, Pr, H, Cl, S, c-Pr, H, H, H, O], [AC6375; H , Pr, H, Cl, S, OMe, H, H, H, O], [AC 6376; H, Pr, H, Cl, S, OEt, H, H, H, O], [AC 6377; H, Pr , H, Cl, S, Oi-Pr, H, H, H, O], [AC 6378; H, Pr, H, Cl, S, SMe, H, H, H, O],

[AC 6379; H, Pr, H, Cl, S, SEt, H, H, H, O], [AC 6380; H, Pr, H, Cl, S, CH ₂ F, H, H, H, O], [AC6381; H, Pr, H , Cl, S, CHF 2, H, H, H, O], [AC6382; H, Pr, H, Cl, S, CF 3, H, H, H, O], [AC6383; H, Pr, H , Cl, S, OCH 2 F, H, H, H, O], [AC6384; H, Pr, H, Cl, S, OCHF 2, H, H, H, O] , [AC6385; H, Pr, H, Cl, S, OCF 3, H, H, H, O], [AC6386; H, Pr, H, Cl, S, SCH 2 F, H, H, H, O H, Pr, H, Cl, S, SCHF ₂ , H, H, H, O], [AC 6388; H, Pr, H, Cl, S, SCF ₃ , H, H, H, O] ], [AC 6 389; H, Pr, H, Cl, S, CN, H, H, H, O], [AC 6390; H, Pr, H, Cl, S, NO ₂ , H, H, H, O] [AC6391; H, Pr, H, Br, S, H, H, H, O], [AC6392; H, Pr, H, Br, S, F, H, H, O], [AC6392; AC6393; H, Pr, H, Br, S, Cl, H, H, H, O], [AC6394; H, Pr, H, Br, S, Br, H, H, H, O], [AC6395; H, Pr, H, Br, S, I, H, H, H, O], [AC 6396; H, Pr, H, Br, S, Me, H, H, O], [AC 6397; H, Pr, H, Br, S, Et, H, H, H, O], [AC6398; H, Pr, H, Br, S, Pr, H, H, H, O], [AC 6399; H, Pr, H, Br, S, i- Pr, H, H, H, O], [AC6400; H, Pr, H, Br, S, CH = CH 2, H, H, H, O], [AC6401; H , Pr, H, Br, S , C (CH 3) = CH 2, H, H, H, O], [AC6402; H, Pr, H, Br, S, C≡CH, H, H, H, O], [AC 6403; H, Pr, H, Br, S, C≡CCH ₃ , H, H, H, O], [AC 6404; H, Pr, H, Br, S, c-Pr, H, H , H, O], [AC 6405; H, Pr, H, Br, S, OMe, H, H, H, O], [AC 6406; H, Pr, H, Br, S, OEt, H, H, H , O], [AC 6407; H, Pr, H, Br, S, Oi-Pr, H, H, H, O], [AC 6408; H, Pr, H, Br, S, SMe, H, H, H, O], [AC 6409; H, Pr, H, Br, S, SE t, H, H, H, O], [AC6410; H, Pr, H, Br, S, CH 2 F, H, H, H, O], [AC6411; H, Pr, H, Br, S, CHF 2, H, H , H, O], [AC6412 ; H, Pr, H, Br, S, CF 3, H, H, H, O], [AC6413; H, Pr, H, Br, S, OCH 2 F, H, H, H, O], [AC 6414; H, Pr, H, Br, S, OCHF ₂ , H, H, H, O], [AC 6415; H, Pr, H, Br, S, OCF ₃ , H, H, H, O], [AC 6416; H, Pr, H, Br, S, SCH ₂ F, H, H, H, O], [AC 6417; H, Pr, H, Br, S, SCHF ₂ , H H, H, O], [AC 6418; H, Pr, H, Br, S, SCF ₃ , H, H, H, O], [AC 6419; H, Pr, H, Br, S, CN, H, H, H, O], [AC 6420; H, Pr, H, Br, S, NO ₂ , H, H, H, O], [AC 6421; H, i-Pr, H, H, S, H, H , H, H, O], [AC 6422; H, i-Pr, H, S, F, H, H, H, O], [AC 6423; H, i-Pr, H, H, S, Cl , H, H, H, O], [AC 6424; H, i-Pr, H, H, S, Br, H, H, H, O], [AC 6425; H, i-Pr, H, H, S , I, H, H, H, O], [AC 6426; H, i-Pr, H, H, S, Me, H, H, H, O], [AC 6427; H, i-Pr, H, H , S, Et, H, H, H, O, [AC 6428; H, i-Pr, H, H, S, Pr, H, H, H, O], [AC 6429; H, i-Pr, H , H, S, i-Pr , H, H, H, O], [AC6430; H, i-Pr, H, H, S, CH = CH 2, H, H, H, O], [AC6431; H, i-Pr, H, H, S, C (CH 3) = CH 2, H, H, H, O], [AC6432; H, i-Pr, H, H, S, C≡CH, H , H, H, O], [AC6433; H, i-Pr, H, H, S, C≡CCH 3, H, H, H, O], [AC6434; H, i-Pr, H, H, S, c-Pr, H, H, H, O], [AC 6435; H, i-Pr, H, H, S, OMe, H, H, H, O], [AC 643 6; H, i-Pr, H, H, S, OEt, H, H, H, O], [AC 6437; H, i-Pr, H, H, S, Oi-Pr, H, H, H, O, [AC 6438; H, i-Pr, H, H, S, SMe, H, H, H, O], [AC 6439; H, i-Pr, H, H, S, SE t, H, H, H, O], [AC6440; H, i-Pr, H, H, S, CH 2 F, H, H, H, O], [AC6441; H, i-Pr, H, H, S, CHF 2 , H, H, H, O ], [AC6442; H, i-Pr, H, H, S, CF 3, H, H, H, O], [AC6443; H, i-Pr, H, H, _{S, OCH 2 F, H,} H, H, O], [AC6444; H, i-Pr, H, H, S, OCHF 2, H, H, H, O], [AC6445; H, i-Pr , H, H, S, OCF 3, H, H, H, O], [AC6446; H, i-Pr, H, H, S, SCH 2 F, H, H, H, O], [AC6447; H, i-Pr, H, H, S, SCHF 2, H, H, H, O], [AC6448; H, i-Pr, H, H, S, SCF 3, H, H, H, O] , [AC6449; H, i- Pr, H, H, S, CN, H, H, H, O], [AC6450; H, i-Pr, H, H, S, NO 2, H, H, H , O], [AC6451; H, i-Pr, H, Me, S, H, H, H, H, O], [AC6452; H, i-Pr, H, Me, S, F, H, H , H, O], [AC6453; H, i-Pr, H, Me, S, Cl, H, H, H, O], [AC6454; H, i-Pr, H, Me, S, Br, H , H, H, O], [AC 6455; H, i-Pr, H, Me, S, I, H, H, H, O], [AC 6456; H, i-Pr, H, Me, S, Me , H, H, H, O], [AC 6457; H, i-Pr, H, Me, S, Et, H, H, H, O], [AC 6458; H, i-Pr, H, Me, S , Pr, H, H, H, O], [AC6459; H, i-Pr, H, Me, S, i-Pr, H, H, H, O], [AC 6460; H, i-Pr, H , Me, S, CH = CH 2, H, H, H, O], [AC6461; H, i-Pr, H, Me, S, C (CH 3) = CH 2, H, H, H, O H, i-Pr, H, Me, S, C≡CH, H, H, H, O], [AC 6463; H, i-Pr, H, Me, S, C≡CCH ₃ , H , H, H, O], [AC6464; H, i-Pr, H, Me, S, c-Pr, H, H, H, O], [AC 6465; H, i-Pr, H, Me, S , OMe, H, H, H, O], [AC 6466; H, i-Pr, H, Me, S, OEt, H, H, H, O], [AC 6467; H, i-Pr, H, Me , S, Oi-Pr, H, H, H, O, [AC 6468; H, i-Pr, H, Me, S, SMe, H, H, O], [AC 6469; H, i-Pr , H, Me, S, SEt, H, H, H, O], [AC 6470; H, i-Pr, H, Me, S, CH ₂ F, H, H, O], [AC 6471; H , i-Pr, H, Me , S, CHF 2, H, H, H, O], [AC6472; H, i-Pr, H, Me, S, CF 3, H, H, H, O], [AC 6473; H, i-Pr, H, Me, S, OCH ₂ F, H, H, H, O], [AC 6474; H, i-Pr, H, Me, S, OCHF ₂ , H, H, H, O], [AC6475; H, i-Pr, H, Me, S, OCF 3, H, H, H, O], [AC6476; H, i-Pr, H, Me, S, SCH 2 F , H, H, H, O], [AC 6477; H, i-Pr, H, Me, S, SCHF ₂ , H, H, H, O], [AC 6478; H, i-Pr, H, Me, S, SCF ₃ , H, H, H, O],

[AC 6479; H, i-Pr, H, Me, S, CN, H, H, H, O], [AC 6480; H, i-Pr, H, Me, S, NO ₂ , H, H, H, O], [AC 6481; H, i-Pr, H, Et, S, H, H, H, H, O], [AC 6482; H, i-Pr, H, Et, S, F, H, H, H, O], [AC 6483; H, i-Pr, H, Et, S, Cl, H, H, H, O], [AC 6484; H, i-Pr, H, Et, S, Br, H, H, H, O], [AC 6485; H, i-Pr, H, Et, S, I, H, H, H, O], [AC6486; H, i-Pr, H, Et, S, Me, H, H, H, O], [AC 6487; H, i-Pr, H, Et, S, Et, H, H, H, O], [AC 6488; H, i-Pr, H, Et, S, Pr, H, H, H, O], [AC 6489; H, i-Pr, H, Et, S, i-Pr, H, H, H, O], [AC 6490; H, i-Pr, H, _{Et, S, CH = CH 2} , H, H, H, O], [AC6491; H, i-Pr, H, Et, S, C (CH 3) = CH 2, H, H, H, O] [AC6492; H, i-Pr, H, Et, S, C≡CH, H, H, H, O], [AC6493; H, i-Pr, H, Et, S, C≡CCH ₃ , H , H, H, O], [AC 6494; H, i-Pr, H, Et, S, c, Pr, H, H, H, O], [AC 6495; H, i-Pr, H, Et, S , OMe, H, H, H, O], [AC6496; H, i-Pr, H, Et, S, OEt, H, H, H, O], [AC 6497; H, i-Pr, H, Et , S, Oi-Pr, H, H, H, O, [AC6498; H, i-Pr, H, Et, S, SMe, H, H, O], [AC 6499; H, i-Pr , H, Et, S, SEt , H, H, H, O], [AC6500; H, i-Pr, H, Et, S, CH 2 F, H, H, H, O], [AC6501; H , i-Pr, H, Et , S, CHF 2, H, H, H, O], [AC6502; H, i-Pr, H, Et, S, CF 3, H, H, H, O], [AC6503; H, i-Pr , H, Et, S, OCH 2 F, H, H, H, O], [AC6504; H, i-Pr, H, Et, S, OCHF 2, H, H, H, O], [AC6505; H, i-Pr, H, Et, S, OCF 3, H, H, H, O], [AC6506; H, i-Pr, H , Et, S, SCH ₂ F, H, H, H, O], [AC 6507; H, i-Pr, H, Et, S, SCHF ₂ , H, H, H, O], [AC 6508; H, i-Pr, H, Et, S, SCF 3, H, H, H, O], [AC6509; H, i-Pr, H, Et, S, CN, H, H, H, O], [AC6510 H, i-Pr, H, Et, S, NO ₂ , H, H, H, O], [AC6511; H, i-Pr, H, Pr, S, H, H, H, H, O] [AC 6512; H, i-Pr, H, Pr, S, F, H, H, O], [AC 6513; H, i-Pr, H, Pr, S, Cl, H, H, H, O], [AC 6514; H, i-Pr, H, Pr, S, Br, H, H, H, O], [AC 6515; H, i-Pr, H, Pr, S, I, H, H, H, O], [AC 6516; H, i-Pr, H, Pr, S, Me, H, H, H, O], [AC 6517; H, i-Pr, H, Pr, S, Et, H, H, H, O], [AC 6518; H, i-Pr, H, Pr, S, Pr, H, H, H, O], [AC 6519; H, i-Pr, H, Pr, S, i- Pr, H, H, H, O], [AC6520; H, i-Pr, H, Pr, S, CH = CH 2, H, H, H, O], [AC6521; H, i-Pr, H , Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC6522; H, i-Pr, H, Pr, S, C≡CH, H, H, H, O] , [AC6523; H, i- Pr, H, Pr, S, C≡CCH 3, H, H, H, O], [AC6524; H, i-Pr, H, Pr, S, c-Pr, H , H, H, O], [AC 6525; H, i-Pr, H, Pr, S, OMe, H, H, H, O], [AC 6526; H, i-Pr, H, Pr, S, OEt , H, H, H, O], [AC 6527; H, i-Pr, H, Pr, S, Oi-Pr, H, H, H, O], [AC 6528; H, i-Pr, H, Pr , S, SMe, H, H, H, O, [AC 6529; H, i-Pr, H, Pr, S, SE t, H, H, H, O], [AC 6530; H, i-Pr, H _{, Pr, S, CH 2 F} , H, H, H, O], [AC6531; H, i-Pr, H, Pr, S, CHF 2, H, H, H, O], [AC6532; H, i-Pr, H, Pr, S, CF 3, H, H, H, O], [AC6533; H, i-Pr, H, Pr, S, OCH 2 F, H, H, H, O], [ AC6534; H, i-Pr, H, Pr, S, OCHF 2, H, H, H, O], [AC6535; H, i-Pr, H, Pr, S, OCF ₃ , H, H, H, O], [AC 6536; H, i-Pr, H, Pr, S, SCH ₂ F, H, H, H, O], [AC 6537; H, i-Pr, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 6538; H, i-Pr, H, Pr, S, SCF ₃ , H, H, H, O], [AC 6539; H, i- Pr, H, Pr, S, CN, H, H, H, O], [AC6540; H, i-Pr, H, Pr, S, NO 2, H, H, H, O], [AC6541; H , i-Pr, H, i-Pr, S, H, H, H, H, O], [AC 6542; H, i-Pr, H, i-Pr, S, F, H, H, O, H, i-Pr, H, i-Pr, S, Cl, H, H, H, O], [AC 6544; H, i-Pr, H, i-Pr, S, Br, H] , H, H, O], [AC 6545; H, i-Pr, H, i-Pr, S, I, H, H, H, O], [AC 6546; H, i-Pr, H, i-Pr , S, Me, H, H, H, O], [AC 6547; H, i-Pr, H, i-Pr, S, Et, H, H, H, O], [AC 6548; H, i-Pr , H, i-Pr, S, Pr, H, H, H, O], [AC 6549; H, i-Pr, H, i-Pr, S, i-Pr, H, H, H, O], [AC6550; H, i-Pr , H, i-Pr, S, CH = CH 2, H, H, H, O], [AC6551; H, i-Pr, H, i-Pr, S, C ( CH ₃ ) = CH ₂ , H, H, H, O], [AC6552; H, i-Pr, H, i-Pr, S, C≡CH, H, H, H, O], [AC6553; H , i-Pr, H, i-Pr, S, C≡CCH ₃ , H, H, H, O], [AC6554; H, i-Pr, H, i-Pr, S, c-Pr, H, H, H, O], [AC6555; H, i-Pr, H, i-Pr, S, OMe, H, H, H, O], [AC6556; H, i-Pr, H, i-Pr, S, OEt, H, H, H, O], [AC6557; H, i-Pr, H, i-Pr, S, Oi-Pr, H, H, H, O], [AC6558; H, i- Pr, H, i-Pr, S, SMe, H, H, H, O], [AC6559; H, i-Pr, H, i-Pr, S, SEt, H, H, H, O], [ AC6560 ; H, i-Pr, H , i-Pr, S, CH 2 F, H, H, H, O], [AC6561; H, i-Pr, H, i-Pr, S, CHF 2, H, H, H, O], [ AC6562; H, i-Pr, H, i-Pr, S, CF 3, H, H, H, O], [AC6563; H, i-Pr, H, i-Pr _{, S, OCH 2 F, H} , H, H, O], [AC6564; H, i-Pr, H, i-Pr, S, OCHF 2, H, H, H, O], [AC6565; H, i-Pr, H, i- Pr, S, OCF 3, H, H, H, O], [AC6566; H, i-Pr, H, i-Pr, S, SCH 2 F, H, H, H , O], [AC 6567; H, i-Pr, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 6568; H, i-Pr, H, i-Pr, S, SCF ₃ , H, H, H, O], [AC 6569; H, i-Pr, H, i-Pr, S, CN, H, H, H, O], [AC 6570; H, i-Pr, H , i-Pr, S, NO 2, H, H, H, O], [AC6571; H, i-Pr, H, c-Pr, S, H, H, H, H, O], [AC6572; H, i-Pr, H, c-Pr, S, F, H, H, H, O], [AC 6573; H, i-Pr, H, c-Pr, S, Cl, H, H, H, H, O], [AC6574; H, i-Pr, H, c-Pr, S, Br, H, H, H, O], [AC 6575; H, i-Pr, H, c-Pr, S, I, H, H, H, O], [AC 6576; H, i-Pr, H, c-Pr, S, Me, H, H, H, O], [AC 6577; H, i-Pr, H, c- Pr, S, Et, H, H, H, O, [AC 6578; H, i-Pr, H, c-Pr, S, Pr, H, H, H, O],

[AC 6579; H, i-Pr, H, c-Pr, S, i-Pr, H, H, H, O], [AC 6580; H, i-Pr, H, c-Pr, S, CH = CH _{2, H, H, H,} O], [AC6581; H, i-Pr, H, c-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC6582; H , i-Pr, H, c-Pr, S, C≡CH, H, H, H, O], [AC 6583; H, i-Pr, H, c-Pr, S, C≡ CCH ₃ , H, H, H, O], [AC 6584; H, i-Pr, H, c-Pr, S, c-Pr, H, H, H, O], [AC 6585; H, i-Pr, H, c- Pr, S, OMe, H, H, H, O], [AC 6586; H, i-Pr, H, c-Pr, S, OEt, H, H, H, O], [AC 6587; H, i- Pr, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 6588; H, i-Pr, H, c-Pr, S, SMe, H, H, H, O] H, i-Pr, H, c-Pr, S, SEt, H, H, H, O], [AC 6590; H, i-Pr, H, c-Pr, S, CH ₂ F, H, H, H, O] , [AC6591; H, i-Pr, H, c-Pr, S, CHF 2, H, H, H, O], [AC6592; H, i-Pr, H, c _{-Pr, S, CF 3, H} , H, H, O], [AC6593; H, i-Pr, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC6594; H, i-Pr, H, c-Pr, S, OCHF 2, H, H, H, O], [AC6595; H, i-Pr, H, c-Pr, S, OCF 3, H, H, H, O], [AC 6596; H, i-Pr, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 6597; H, i-Pr, H, c-Pr, S, SCHF ₂ , H, H, H, O], [AC 6598; H, i-Pr, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 6599; H, i- Pr, H, c-Pr, S, CN, H, H, H, O], [AC 6600; H, i-Pr, H, c-Pr, S, NO ₂ , H, H, H, O], [AC6601; H, i-Pr, H, SMe, S, H, H, H, H, O], [AC6602; H, i-Pr, H, SMe, S, F, H, H, H, O H, i-Pr, H, SMe, S, Cl, H, H, H, O], [AC 6604; H, i-Pr, H, SMe, S] , Br, H, H, H, O], [AC 6605; H, i-Pr, H, SMe, S, I, H, H, H, O], [AC 6606; H, i-Pr, H, SMe , S, Me, H, H, H, O], [AC 6607; H, i-Pr, H, SMe, S, Et, H, H, H, O], [AC 6608; H, i-Pr, H , SMe, S, Pr, H, H, H, O], [AC 6609; H, i-Pr, H, SMe, S, i-Pr, H, H, H, O], [AC 6610; H, i -Pr, H, SMe, S, CH = CH 2, H, H, H, O], [AC6611; H, i-Pr, H, SMe, S, C (CH 3) = CH 2, H, H , H, O], [AC6612; H, i-Pr, H, SMe, S, C≡CH, H, H, H, O], [AC6613; H, i-Pr, H, SMe, S, C ≡ CCH ₃ , H, H, H, O], [AC6614; H, i-Pr, H, SMe, S, c-Pr, H, H, H, O], [AC 6615; H, i-Pr, H, SMe, S, OMe, H, H, H, O], [AC 6616; H, i-Pr, H, SMe, S, OEt, H, H, H, O], [AC 6617; H, i- Pr, H, SMe, S, Oi-Pr, H, H, H, O], [AC 6618; H, i-Pr, H, SMe, S, S Me, H, H, O], [AC 6619; H, i-Pr, H, SMe, S, SEt, H, H, H, O], [AC6620; H, i-Pr, H, SMe, S, CH 2 F, H, H, H, O] , [AC6621; H, i- Pr, H, SMe, S, CHF 2, H, H, H, O], [AC6622; H, i-Pr, H, SMe, S, CF 3, H, H, H, O], [AC6623; H, i-Pr, H, SMe, S, OCH 2 F, H, H, H, O], [AC6624; H, i-Pr, H, SMe, S, OCHF 2 , H, H, H, O ], [AC6625; H, i-Pr, H, SMe, S, OCF 3, H, H, H, O], [AC6626; H, i-Pr, H, SMe, _{S, SCH 2 F, H,} H, H, O], [AC6627; H, i-Pr, H, SMe, S, SCHF 2, H, H, H, O], [AC6628; H, i-Pr , H, SMe, S, SCF 3, H, H, H, O], [AC6629; H, i-Pr, H, SMe, S, CN, H, H, H, O], [AC6630; H, i-Pr, H, SMe, S, NO ₂ , H, H, H, O], [AC6631; H, i-Pr, H, OMe, S, H, H, H, H, O], [AC6632; H, i-Pr, H, OMe, S, F, H, H, H, O], [AC6633; H, i-Pr, H, OMe, S, Cl, H, H, H, O], [AC6634; H, i-Pr, H, OMe, S, Br, H, H, H, O], [AC 6635; H, i-Pr, H, OMe, S, I, H, H, H, O], [AC 6636; H, i-Pr, H, OMe, S, Me, H, H, H, O], [AC 6637; H, i-Pr, H, OMe, S, Et, H, H, H, O], [AC 6638; H, i-Pr, H, OMe, S, Pr, H, H, H, O], [AC 6639; H, i-Pr, H, OMe, S, i-Pr, H, H, H, O], [AC 6640; H, i-Pr, H, OMe, S, CH = CH 2, H, H, H, O], [AC6641; H, i-Pr, H, OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC6642; H, i-Pr, H, OMe, S, C, CH, H, H, H, O], [AC6643; H, i-Pr, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC6644; H, i-Pr, H, OMe, S, c-Pr, H, H, H, O], [AC6645; H, i-Pr, H, OMe , S, OMe, H, H, H, O], [AC 6 646; H, i-Pr, H, OMe, S, OEt, H, H, H, O], [AC 6647; H, i-Pr, H , OMe, S, Oi-Pr, H, H, H, O], [AC 6648; H, i-Pr, H, OMe, S, SMe, H, H, H, O], [AC 6649; H, i -Pr, H, OMe, S, SEt, H, H, H, O], [AC6650; H, i-Pr, H, OMe, S, CH 2 F, H, H, H, O], [AC6651 ; H, i-Pr, H , OMe, S, CHF 2, H, H, H, O], [AC6652; H, i-Pr, H, OMe, S, CF 3, H, H, H, O ], [AC6653; H, i -Pr, H, OMe, S, OCH 2 F, H, H, H, O], [AC6654; H, i-Pr, H, OMe, S, OCHF 2, H, H, H, O], [ AC6655; H, i-Pr, H, OMe, S, OCF 3, H, H, H, O], [AC6656; H, i-Pr, H, OMe, S, SCH ₂ F, H, H, H, O], [AC 6657; H, i-Pr, H, _{OMe, S, SCHF 2, H} , H, H, O], [AC6658; H, i-Pr, H, OMe, S, SCF 3, H, H, H, O], [AC6659; H, i- Pr, H, OMe, S, CN, H, H, H, O], [AC 6660; H, i-Pr, H, OMe, S, NO ₂ , H, H, H, O], [AC6661; H , i-Pr, H, F, S, H, H, H, H, O], [AC6662; H, i-Pr, H, F, S, F, H, H, O], [AC6663 H, i-Pr, H, F, S, Cl, H, H, H, O], [AC6664; H, i-Pr, H, F, S, Br, H, H, H, O], [AC6665; H, i-Pr, H, F, S, I, H, H, H, O], [AC 6666; H, i-Pr, H, F, S, Me, H, H, H, O H, i-Pr, H, F, S, Et, H, H, H, O], [AC6668; H, i-Pr, H, F, S, Pr, H, H, H] H, i-Pr, H, F, S, i-Pr, H, H, H, O], [AC 6670; H, i-Pr, H, F, S, CH = CH ₂ , H, H, H, O], [AC 667 1; H, i-Pr, H, F, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 667 2; H, i -Pr, H, F, S, C≡CH, H, H, H, O], [AC6673; H, i-Pr, H, F, S, C≡ CCH ₃ , H, H, H, O] [AC6674; H, i-Pr, H, F, S, c-Pr, H, H, H, O], [AC6675; H, i-Pr, H, F, S, OMe, H, H, H, O], [AC6676; H, i-Pr, H, F, S, OEt, H, H, H, O], [AC 6677; H, i-Pr, H, F, S, Oi-Pr, H, H, H, O],

[AC 6678; H, i-Pr, H, F, S, SMe, H, H, H, O], [AC 6679; H, i-Pr, H, F, S, SE t, H, H, H, O H, i-Pr, H, F, S, CH ₂ F, H, H, H, O], [AC 6681; H, i-Pr, H, F, S, CHF ₂ , H, H, H, O], [ AC6682; H, i-Pr, H, F, S, CF 3, H, H, H, O], [AC6683; H, i-Pr, H, F, S, OCH ₂ F, H, H, H, O], [AC 6684; H, i-Pr, H, F, S, OCHF ₂ , H, H, H, O], [AC 6685; H, i-Pr, H, _{F, S, OCF 3, H} , H, H, O], [AC6686; H, i-Pr, H, F, S, SCH 2 F, H, H, H, O], [AC6687; H, i -Pr, H, F, S, SCHF ₂ , H, H, H, O], [AC 6688; H, i-Pr, H, F, S, SCF ₃ , H, H, H, O], [AC 6689 H, i-Pr, H, F, S, CN, H, H, H, O], [AC 6690; H, i-Pr, H, F, S, NO ₂ , H, H, H, O] [AC6691; H, i-Pr, H, Cl, S, H, H, H, H, O], [AC6692; H, i-Pr, H, Cl, S, F, H, H, H, H, O], [AC6693; H, i-Pr, H, Cl, S, Cl, H, H, H, O], [AC6694; H, i-Pr, H, Cl, S, Br, H, H, H, O], [AC 6695; H, i-Pr, H, Cl, S, I, H, H, H, O], [AC 6696; H, i-Pr, H, Cl, S, Me, H, H, H, O], [AC6697; H, i-Pr, H, Cl, S, Et, H, H, H, O], [AC6698; H, i-Pr, H, Cl, S, Pr, H, H, H, O], [AC 6699; H, i-Pr, H, Cl, S, i-Pr, H, H, H, O], [AC 6700; H, i-Pr, H, Cl, _{S, CH = CH 2, H} , H, H, O], [AC6701; H, i-Pr, H, Cl, S, C (CH 3) = CH 2, H, H, H, O], [ AC 6702; H, i-Pr, H, Cl, S, C≡CH, H, H, H, O], [AC6703; H, i-Pr, H, Cl, S, C≡ CCH ₃ , H, H , H, O], [AC 6704; H, i-Pr, H, Cl, S, c-Pr, H, H, H, O], [AC 6705; H, i-Pr, H, Cl, S, OMe, H, H, H, O], [AC 6706; H, i-Pr, H, Cl, S, OEt, H, H, H, O], [AC 6707; H, i-Pr, H, Cl, S, Oi-Pr, H, H, H, O], [AC 6708; H, i-Pr, H, Cl, S, SMe, H, H, O], [AC 6709; H, i- Pr, H, Cl, S, SEt, H, H, H, O], [AC6710; H, i-Pr, H, Cl, S, CH 2 F, H, H, H, O], [AC6711; H, i-Pr, H, Cl, S, CHF 2, H, H, H, O], [AC6712; H, i-Pr, H, Cl, S, CF 3, H, H, H, O] , [AC6713; H, i- Pr, H, Cl, S, OCH 2 F, H, H, H, O], [AC6714; H, i-Pr, H, Cl, S, OCHF 2, H, H , H, O], [AC6715 ; H, i-Pr, H, Cl, S, OCF 3, H, H, H, O], [AC6716; H, i-Pr, H, Cl, S, SCH 2 F, H, H, H, O], [AC 6717; H, i-Pr, H, Cl, S, SCHF ₂ , H, H, H, O], [AC 6718; H, i-Pr, H, Cl , S, SCF ₃ , H, H, H, O], [AC 6719; H, i-Pr, H, Cl, S, CN, H, H, H, O], [AC 6720; H, i-Pr, _{H, Cl, S, NO 2} , H, H, H, O], [AC6721; H, i-Pr, H, Br, S, H, H, H, H, O], [AC6722; H, i -Pr, H, Br, S, F, H, H, H, O], [AC6723; H, i-Pr, H, Br, S, Cl, H, H, H, O], [AC 6724; H , i-Pr, H, Br, S, Br, H, H, H, O], [AC6725; H, i-Pr, H, Br, S, I, H, H, H, O], [AC 6726 H, i-Pr, H, Br, S, Me, H, H, H, O], [AC 6727; H, i-Pr, H, Br, S, Et, H, H, H, O], [AC 6728; H, i-Pr, H, Br, S, Pr, H, H, H, O], [AC 6729; H, i-Pr, H, Br, S, i-Pr, H, H, H , O], [AC6730; H , i-Pr, H, Br, S, CH = CH 2, H, H, H, O], [AC6731; H, i-Pr, H, Br, S, C ( CH ₃ ) = CH ₂ , H, H, H, O], [AC 6732; H, i-Pr, H, Br, S, C≡CH, H, H, H, O H, i-Pr, H, Br, S, C≡CCH ₃ , H, H, H, O], [AC 6734; H, i-Pr, H, Br, S, c-Pr, H, H, H, O], [AC 6735; H, i-Pr, H, Br, S, OMe, H, H, H, O], [AC 6736; H, i-Pr, H, Br, S, OEt, H, H, H, O], [AC 6737; H, i-Pr, H, Br, S, Oi-Pr, H, H, H, O], [AC 6738; H, i-Pr, H, Br, S, SMe, H, H, H, O, [AC 6739; H, i-Pr, H, Br, S, SE t, H, H, H, O], [AC 6740; H, i-Pr, _{H, Br, S, CH 2} F, H, H, H, O], [AC6741; H, i-Pr, H, Br, S, CHF 2, H, H, H, O], [AC6742; H , i-Pr, H, Br , S, CF 3, H, H, H, O], [AC6743; H, i-Pr, H, Br, S, OCH 2 F, H, H, H, O] , [AC 6744; H, i-Pr, H, Br, S, OCHF ₂ , H, H, H, O], [AC 6745; H, i-Pr, H, Br, S, OCF ₃ , H, H, H, O], [AC 6746; H, i-Pr, H, Br, S, SCH ₂ F, H, H, H, O], [AC 6747; H, i-Pr, H, Br, S, SCHF ₂ , H, H, H, O ], [AC6748; H, i-Pr, H, Br, S, SCF 3, H, H, H, O], [AC6749; H, i-Pr, H, Br, S, CN, H, H, H, O], [AC 6750; H, i-Pr, H, Br, S, NO ₂ , H, H, H, O], [AC 6751; H, c-Pr, H , H, S, H, H, H, H, H, O], [AC6752; H, c-Pr, H, H, S, F, H, H, O], [AC6753; H, c-Pr , H, H, S, Cl, H, H, H, O], [AC 6754; H, c-Pr, H, H, S, Br, H, H, O], [AC 6755; H, c -Pr, H, H, S, I, H, H, H, O], [AC 6756; H, c-Pr, H, H, S, Me, H, H, O], [AC 6757; H , c-Pr, H, H, S, Et, H, H, H, O], [AC 6758; H, c-Pr, H, H, S, Pr, H, H, O], [AC 6759 H, c-Pr, H, H, S, i, Pr, H, H, H, O], [AC 6760; H, c-Pr, H, H, S, CH = CH ₂ , H , H, H, O], [AC6761; H, c-Pr, H, H, S, C (CH 3) = CH 2, H, H, H, O], [AC6762; H, c-Pr, H, H, S, C≡CH, H, H, H, O], [AC6763; H, c-Pr, H, H, S, C≡CCH 3, H, H, H, O], [AC6764 H, c-Pr, H, H, S, c-Pr, H, H, H, O], [AC 6765; H, c-Pr, H, H, S, OMe, H, H, H, O H, c-Pr, H, H, S, OEt, H, H, H, O], [AC 6767; H, c-Pr, H, H, S, Oi-Pr, H, H] , H, O], [AC 6768; H, c-Pr, H, H, S, SMe, H, H, H, O], [AC 6769; H, c-Pr, H, H, S, SEt, H , H, H, O], [AC6770; H, c-Pr, H, H, S, CH 2 F, H, H, H, O], [AC6771; H, c-Pr, H, H, S _{, CHF 2, H, H,} H, O], [AC6772; H, c-Pr, H, H, S, CF 3, H, H, H, O], [AC6773; H, c-Pr, H _{, H, S, OCH 2 F} , H, H, H, O], [AC6774; H, c-Pr, H, H, S, OCHF 2, H, H, H, O], [AC6775; H, c-Pr, H, H, S, OCF 3, H, H, H, O], [AC6776; H, c-Pr, H, H, S, SCH 2 F, H, H, H, O], [AC 6777; H, c-Pr, H, H, S, SCHF ₂ , H, H, H, O],

[AC 6778; H, c-Pr, H, H, S, SCF ₃ , H, H, H, O], [AC 6779; H, c-Pr, H, H, S, CN, H, H, H, O], [AC6780; H, c-Pr, H, H, S, NO 2, H, H, H, O], [AC6781; H, c-Pr, H, Me, S, H, H, H , H, O], [AC6782; H, c-Pr, H, Me, S, F, H, H, H, O], [AC6783; H, c-Pr, H, Me, S, Cl, H , H, H, O], [AC 6784; H, c-Pr, H, Me, S, Br, H, H, H, O], [AC 6785; H, c-Pr, H, Me, S, I , H, H, H, O], [AC 6786; H, c-Pr, H, Me, S, Me, H, H, H, O], [AC 6787; H, c-Pr, H, Me, S , Et, H, H, H, O], [AC 6788; H, c-Pr, H, Me, S, Pr, H, H, H, O], [AC 6789; H, c-Pr, H, Me , S, i-Pr, H , H, H, O], [AC6790; H, c-Pr, H, Me, S, CH = CH 2, H, H, H, O], [AC6791; H, c-Pr, H, Me, S, C (CH 3) = CH 2, H, H, H, O], [AC6792; H, c-Pr, H, Me, S, C≡CH, H, H , H, O], [AC 6793; H, c-Pr, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 6794; H, c-Pr, H, Me, S, c-Pr, H, H, H, O], [AC 6795; H, c-Pr, H, Me, S, OMe, H, H, H, O], [AC 6796; H, c-Pr, H, Me, S, OEt, H, H, H, O], [AC6797; H, c-Pr, H, Me, S, Oi-Pr, H, H, H, O], [AC 6798; H, c- Pr, H, Me, S, SMe, H, H, H, O], [AC 6799; H, c-Pr, H, Me, S, SE t, H, H, O], [AC 6800; H, c-Pr, H, Me, S, CH 2 F, H, H, H, O], [AC6801; H, c-Pr, H, Me, S, CHF 2, H, H, H, O], [AC6802; H, c-Pr , H, Me, S, CF 3, H, H, H, O], [AC6803; H, c-Pr, H, Me, S, OCH 2 F, H, H, H, O], [AC 6804; H, c-Pr, H, Me, S, OCHF ₂ , H, H, H, O], [AC 6805; H, c-Pr, H, Me _{, S, OCF 3, H,} H, H, O], [AC6806; H, c-Pr, H, Me, S, SCH 2 F, H, H, H, O], [AC6807; H, c- Pr, H, Me, S, SCHF ₂ , H, H, H, O], [AC 6808; H, c-Pr, H, Me, S, SCF ₃ , H, H, H, O], [AC 6809; H, c-Pr, H, Me, S, CN, H, H, H, O], [AC6810; H, c-Pr, H, Me, S, NO 2, H, H, H, O], [AC 6811; H, c-Pr, H, Et, S, H, H, H, H, O], [AC 6812; H, c-Pr, H, Et, S, F, H, H, H, O H, c-Pr, H, Et, S, Cl, H, H, H, O], [AC 6814; H, c-Pr, H, Et, S, Br, H, H, H] H, c-Pr, H, Et, S, I, H, H, H, O], [AC 6816; H, c-Pr, H, Et, S, Me, H, H , H, O], [AC 6817; H, c-Pr, H, Et, S, Et, H, H, H, O], [AC 6818; H, c-Pr, H, Et, S, Pr, H , H, H, O], [AC 6819; H, c-Pr, H, Et, S, i-Pr, H, H, H, O], [AC 6820; H, c-Pr, H, Et, S _{, CH = CH 2, H,} H, H, O], [AC6821; H, c-Pr, H, Et, S, C (CH 3) = CH 2, H, H, H, O], [AC6822 H, c-Pr, H, Et, S, C≡CH, H, H, H, O], [AC 6823; H, c-Pr, H, Et, S, C≡CCH ₃ , H, H, H H, O], [AC 6824; H, c-Pr, H, Et, S, c-Pr, H, H, H, O], [AC 6825; H, c-Pr, H, Et, S, OMe, H, H, H, O], [AC 6826; H, c-Pr, H, Et, S, OEt, H, H, H, O], [AC 6827; H, c-Pr, H, Et, S, Oi-Pr, H, H, H, O], [AC 6828; H, c-Pr, H, Et, S, SMe, H, H, H, O], [AC 6829; H, c-Pr, H, Et, S, SEt, H, H, H, O], [AC 6830; H, c-Pr, H, Et, S, CH ₂ F, H, H, O], [AC 6831; H, c- Pr, H, Et, S, CHF 2, H, H, H, O], [AC6832; H, c-Pr, H, Et, S, CF 3, H, H, H, O], [AC6833; H, c-Pr, H, Et, S, OCH 2 F, H, H, H, O], [AC6834; H, c-Pr, H, Et, S, OCHF 2, H , H, H, O], [AC6835; H, c-Pr, H, Et, S, OCF 3, H, H, H, O], [AC6836; H, c-Pr, H, Et, S, SCH ₂ F, H, H, H, H, O], [AC 6837; H, c-Pr, H, Et, S, SCHF ₂ , H, H, H, O], [AC 6838; H, c-Pr, H , Et, S, SCF ₃ , H, H, H, O], [AC 6839; H, c-Pr, H, Et, S, CN, H, H, H, O], [AC 6840; H, c- Pr, H, Et, S, NO 2, H, H, H, O], [AC6841; H, c-Pr, H, Pr, S, H, H, H, H, O], [AC6842; H , c-Pr, H, Pr, S, F, H, H, H, O], [AC6843; H, c-Pr, H, Pr, S, Cl, H, H, H, O], [AC6844 H, c-Pr, H, Pr, S, Br, H, H, H, O], [AC6845; H, c-Pr, H, Pr, S, I, H, H, H, O], [AC 6846; H, c-Pr, H, Pr, S, Me, H, H, H, O], [AC 6847; H, c-Pr, H, Pr, S, Et, H, H, H, O H, c-Pr, H, Pr, S, Pr, H, H, H, O], [AC 6849; H, c-Pr, H, Pr, S, i-Pr, H, H] , H, O], [AC6850 ; H, c-Pr, H, Pr, S, CH = CH 2, H, H, H, O], [AC6851; H, c-Pr, H, Pr, S, _{C (CH 3) = CH 2} , H, H, H, O], [AC6852; H, c-Pr, H, Pr, S, C≡CH, H, H, H, O], [AC6853; H , c-Pr, H, Pr, S, C≡CCH ₃ , H, H, H, O], [AC6854; H, c-Pr, H, Pr, S, c-Pr, H, H, H, H O, [AC 6855; H, c-Pr, H, Pr, S, OMe, H, H, H, O], [AC 6856; H, c-Pr, H, Pr, S, OE t, H, H, H, O], [AC 6857; H, c-Pr, H, Pr, S, Oi-Pr, H, H, H, O], [AC 6858; H, c-Pr, H, Pr, S, SMe, H, H, H, O], [AC 6859; H, c-Pr, H, Pr, S, SE t, H, H, H, O], [AC 6860; H, c-Pr, H, Pr, S, CH 2 F, H, H, H, O], [AC6861; H, c-Pr, H, Pr, S, CHF 2, H, H, H, O], [AC6862; H, c-Pr , H, Pr, S, CF 3, H, H, H, O], [AC6863; H, c-Pr, H, Pr, S, OCH 2 F, H, H, H, O], [AC6864; H, c-Pr, H, Pr, S, OCHF 2, H, H, H, O], [AC6865; H, c-Pr, H, Pr, S, OCF 3, H, H, H, O], [AC 6866; H, c-Pr, H, Pr, S, SCH ₂ F, H, H, H, O], [AC6867; H, c-Pr, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 6868; H, c-Pr, H, Pr, S, SCF ₃ , H, H, H, O], [AC 6869; H, c-Pr, H, Pr, S, CN, H, H, H, H, O], [AC 6870; H, c-Pr, H, Pr, S, NO ₂ , H, H, H, O], [AC 6871; H, c -Pr, H, i-Pr, S, H, H, H, H, O], [AC 6872; H, c-Pr, H, i-Pr, S, F, H, H, O], [AC 6873; H, c-Pr, H, i-Pr, S, Cl, H, H, H, O], [AC 6874; H, c-Pr, H, i-Pr, S, Br, H, H , H, O], [AC 6875; H, c-Pr, H, i-Pr, S, I, H, H, H, O], [AC 6876; H, c-Pr, H, i-Pr, S , Me, H, H, H, O], [AC 6877; H, c-Pr, H, i-Pr, S, Et, H, H, H, O],

[AC 6878; H, c-Pr, H, i-Pr, S, Pr, H, H, H, O], [AC 6879; H, c-Pr, H, i-Pr, S, i-Pr, H , H, H, O], [AC6880; H, c-Pr, H, i-Pr, S, CH = CH 2, H, H, H, O], [AC6881; H, c-Pr, H, i-Pr, S, C ( CH 3) = CH 2, H, H, H, O], [AC6882; H, c-Pr, H, i-Pr, S, C≡CH, H, H, H H, c-Pr, H, i-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 6884; H, c-Pr, H, i-Pr, S, c-Pr, H, H, H, O], [AC 6885; H, c-Pr, H, i-Pr, S, OMe, H, H, H, O], [AC 6886; H, c- Pr, H, i-Pr, S, OEt, H, H, H, O], [AC6887; H, c-Pr, H, i-Pr, S, Oi-Pr, H, H, H, O] , [AC6888; H, c-Pr, H, i-Pr, S, SMe, H, H, H, O], [AC 6889; H, c-Pr, H, i-Pr, S, SEt, H, H, H, O], [ AC6890; H, c-Pr, H, i-Pr, S, CH 2 F, H, H, H, O], [AC6891; H, c-Pr, H, i- _{Pr, S, CHF 2, H} , H, H, O], [AC6892; H, c-Pr, H, i-Pr, S, CF 3, H, H, H, O], [AC6893; H, c-Pr, H, i- Pr, S, OCH 2 F, H, H, H, O], [AC6894; H, c-Pr, H, i-Pr, S, OCHF 2, H, H, H , O], [AC6895; H , c-Pr, H, i-Pr, S, OCF 3, H, H, H, O], [AC6896; H, c-Pr, H, i-Pr, S, SCH ₂ F, H, H, H, O], [AC 6897; H, c-Pr, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 6898; H, c-Pr , H, i-Pr, S , SCF 3, H, H, H, O], [AC6899; H, c-Pr, H, i-Pr, S, CN, H, H, H, O], [ AC6900; H, c-Pr, H, i-Pr, S, NO 2, H, H, H, O], [AC6901; H, c-Pr, H, c-Pr, S, H, H, H , H, O], [AC6902; H, c-Pr, H, c-Pr, S, F, H, H, H, O], [AC 6903; H, c-Pr, H, c- Pr, S, Cl, H, H, H, H, O], [AC 6904; H, c-Pr, H, c-Pr, S, Br, H, H, O], [AC 6905; H, c- Pr, H, c-Pr, S, I, H, H, H, O], [AC 6906; H, c-Pr, H, c-Pr, S, Me, H, H, H, O], [[ AC 6907; H, c-Pr, H, c-Pr, S, Et, H, H, H, O], [AC 6908; H, c-Pr, H, c-Pr, S, Pr, H, H, H, O], [AC 6 909; H, c-Pr, H, c-Pr, S, i-Pr, H, H, H, O], [AC 6910; H, c-Pr, H, c-Pr, _{S, CH = CH 2, H} , H, H, O], [AC6911; H, c-Pr, H, c-Pr, S, C (CH 3) = CH 2, H, H, H, O] H, c-Pr, H, c-Pr, S, C≡CH, H, H, H, O], [AC 6913; H, c-Pr, H, c-Pr, S, CPr _{CCH 3, H, H, H} , O], [AC6914; H, c-Pr, H, c-Pr, S, c-Pr, H, H, H, O], [AC6915; H, c-Pr , H, c-Pr, S, OMe, H, H, H, O], [AC6916; H, c-Pr, H, c-Pr, S, OEt, H, H, H, O], [AC6917 H, c-Pr, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC6918; H, c-Pr, H, c-Pr, S, SMe, H, H , H, O], [AC6919; H, c-Pr, H, c-Pr, S, SEt, H, H, H, O], [AC6920; H, c-Pr, H, c-Pr, S _{, CH 2 F, H, H} , H, O], [AC6921; H, c-Pr, H, c-Pr, S, CHF 2, H, H, H, O], [AC6922; H, c- Pr, H, c-Pr, S, CF 3, H, H, H, O], [AC6923; H, c-Pr, H, c-Pr, S, OCH 2 F, H, H, H, O ], [AC6924; H, c -Pr, H, c-Pr, S, OCHF 2, H, H, H, O], [AC6925; H, c-Pr, H, c-Pr, S, OCF 3 , H, H, H, O], [AC 6926; H, c-Pr, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 6927; H, c-Pr, H , c-Pr, S, SCHF 2, H, H, H, O], [AC6928; H, c-Pr, H, c-Pr, S, SCF 3, H, H, H, O], [AC6 929; H, c-Pr, H, c-Pr, S, CN, H, H, H, O], [AC6930; H, c-Pr, H, c-Pr, S, NO 2, H, H , H, O], [AC6931; H, c-Pr, H, SMe, S, H, H, H, H, O], [AC6932; H, c-Pr, H, SMe, S, F, H , H, H, O], [AC6933; H, c-Pr, H, SMe, S, Cl, H, H, H, O], [AC6934; H, c-Pr, H, SMe, S, Br , H, H, H, O], [AC6935; H, c-Pr, H, SMe, S, I, H, H, H, O], [AC6936; H, c-Pr, H, SMe, S , Me, H, H, H, O], [AC6937; H, c-Pr, H, SMe, S, Et, H, H, H, O], [AC6938; H, c-Pr, H, SMe , S, Pr, H, H, H, O], [AC 6939; H, c-Pr, H, SMe, S, i-Pr, H, H, H, O], [AC6940; H, c-Pr , H, SMe, S, CH = CH 2, H, H, H, O], [AC6941; H, c-Pr, H, SMe, S, C (CH 3) = CH 2, H, H, H H, c-Pr, H, SMe, S, C≡CH, H, H, H, O], [AC6943; H, c-Pr, H, SMe, S, C≡CCH ₃ , H, H, H, O], [AC6944; H, c-Pr, H, SMe, S, c-Pr, H, H, H, O], [AC6945; H, c-Pr, H, SMe, S, OMe, H, H, H, O], [AC6946; H, c-Pr, H, SMe, S, OEt, H, H, H, O], [AC6947; H, c-Pr, H, SMe, S, Oi-Pr, H, H, H, O], [AC6948; H, c-Pr, H, SMe, S, SMe, H, H, O], [AC 6949; H, c-Pr, H, SMe, S, SEt, H, H, H, O], [AC6950; H, c-Pr, H, SMe, S, CH 2 F, H, H, H, O], [ AC6951; H, c-Pr, H, SMe, S, CHF 2, H, H, H, O], [AC6952; H, c-Pr, H, SMe, S, CF 3, H, H, H, O], [AC6953; H, c-Pr, H, SMe, S, OCH 2 F, H, H, H, O], [AC6954; H, c-Pr, H, SMe, S, OCHF 2, H , H, H, O], [AC6955; H, c-Pr, H, SMe, S, OCF ₃ , H, H, H, O], [AC 6956; H, c-Pr, H, SMe, S, SCH ₂ F, H, H, H, O], [AC 6957; H, c-Pr, H, SMe, _{S, SCHF 2, H, H} , H, O], [AC6958; H, c-Pr, H, SMe, S, SCF 3, H, H, H, O], [AC6959; H, c-Pr, H, SMe, S, CN, H, H, H, O], [AC6960; H, c-Pr, H, SMe, S, NO 2, H, H, H, O], [AC6961; H, c -Pr, H, OMe, S, H, H, H, H, O], [AC6962; H, c-Pr, H, OMe, S, F, H, H, O], [AC6963; H , c-Pr, H, OMe, S, Cl, H, H, H, O], [AC6964; H, c-Pr, H, OMe, S, Br, H, H, H, O], [AC6965 H, c-Pr, H, OMe, S, I, H, H, H, O], [AC6966; H, c-Pr, H, OMe, S, Me, H, H, H, O], [AC6967; H, c-Pr, H, OMe, S, Et, H, H, H, O], [AC6968; H, c-Pr, H, OMe, S, Pr, H, H, H, O H, c-Pr, H, OMe, S, i-Pr, H, H, H, O], [AC 6970; H, c-Pr, H, OMe, S, CH = CH ₂ , H, H, H, O] , [AC6971; H, c-Pr, H, OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC6972; H, c-Pr , H, OMe, S, C≡CH, H, H, H, O], [AC6973; H, c-Pr, H, OMe, S, C≡CCH ₃ , H, H, H, O], [, AC 6974; H, c-Pr, H, OMe, S, c-Pr, H, H, H, O], [AC6975; H, c-Pr, H, OMe, S, OMe, H, H, H, O], [AC6976; H, c-Pr, H, OMe, S, OEt, H, H, H, O],

[AC6977; H, c-Pr, H, OMe, S, Oi-Pr, H, H, H, O], [AC 6978; H, c-Pr, H, OMe, S, SMe, H, H, H H, c-Pr, H, OMe, S, SEt, H, H, H, O], [AC 6980; H, c-Pr, H, OMe, S, CH ₂ F, H , H, H, O], [AC6981; H, c-Pr, H, OMe, S, CHF 2, H, H, H, O], [AC6982; H, c-Pr, H, OMe, S, _{CF 3, H, H, H} , O], [AC6983; H, c-Pr, H, OMe, S, OCH 2 F, H, H, H, O], [AC6984; H, c-Pr, H _{, OMe, S, OCHF 2,} H, H, H, O], [AC6985; H, c-Pr, H, OMe, S, OCF 3, H, H, H, O], [AC6986; H, c -Pr, H, OMe, S, SCH ₂ F, H, H, H, O], [AC 6987; H, c-Pr, H, OMe, S, SCHF ₂ , H, H, H, O], [, AC 69 88; H, c-Pr, H, OMe, S, SCF ₃ , H, H, H, O], [AC 6989; H, c-Pr, H, OMe, S, CN, H, H, H, O ], [AC6990; H, c -Pr, H, OMe, S, NO 2, H, H, H, O], [AC6991; H, c-Pr, H, F, S, H, H, H, H, O], [AC 6992; H, c-Pr, H, F, S, F, H, H, H, O], [AC 6993; H, c-Pr, H, F, S, Cl, H, H, H, O], [AC6994; H, c-Pr, H, F, S, Br, H, H, H, O], [AC6995; H, c-Pr, H, F, S, I, H, H, H, O], [AC6996; H, c-Pr, H, F, S, Me, H, H, H, O], [AC6997; H, c-Pr, H, F, S, Et, H, H, H, O], [AC 6998; H, c-Pr, H, F, S, Pr, H, H, H, O], [AC 6999; H, c-Pr, H, F, S, i-Pr, H, H, H, O], [AC7000; H, c-Pr, H, F, S, CH = CH 2, H, H, H, O], [AC7001; H, c -Pr, H, F, S, C (CH 3) = CH 2, H, H, H, O], [AC7002; H, c-Pr, H, F, S, C≡CH, H, H, H, O], [AC 7003; H, c-Pr, H, F, S, C≡CCH ₃ , H, H, H, O], [AC 70 04; H, c-Pr, H, F, S, c-Pr, H, H, H, O], [AC 7005; H, c-Pr, H, F, S, OMe, H, H, H, H H, c-Pr, H, F, S, OEt, H, H, H, O], [AC 7007; H, c-Pr, H, F, S, Oi-Pr, H, O], [AC 7006; H, H, O], [AC 7008; H, c-Pr, H, F, S, S Me, H, H, H, O], [AC 7009; H, c-Pr, H, F, S, SE t, H, H, H, O] , [AC7010; H, c-Pr, H, F, S, CH 2 F, H, H, H, O], [AC7011; H, c-Pr, H, F, _{S, CHF 2, H, H} , H, O], [AC7012; H, c-Pr, H, F, S, CF 3, H, H, H, O], [AC7013; H, c-Pr, _{H, F, S, OCH 2} F, H, H, H, O], [AC7014; H, c-Pr, H, F, S, OCHF 2, H, H, H, O], [AC7015; H , c-Pr, H, F , S, OCF 3, H, H, H, O], [AC7016; H, c-Pr, H, F, S, SCH 2 F, H, H, H, O] , [AC7017; H, c- Pr, H, F, S, SCHF 2, H, H, H, O], [AC7018; H, c-Pr, H, F, S, SCF 3, H, H, H, O], [AC 7019; H, c-Pr, H, F, S, CN, H, H, H, O], [AC 7020; H, c-Pr, H, F, S, NO ₂ , H , H, H, O], [AC7021; H, c-Pr, H, Cl, S, H, H, H, H, O], [AC7022; H, c-Pr, H, Cl, S, F , H, H, H, O], [AC7023; H, c-Pr, H, Cl, S, Cl, H, H, H, O], [AC7024; H, c-Pr, H, Cl, S , Br, H, H, H, O], [AC 7025; H, c-Pr, H, Cl, S, I, H, H, H, O], [AC 7026; H, c-Pr, H, Cl , S, Me, H, H, H, O], [AC 7027; H, c-Pr, H, Cl, S, Et, H, H, H, O], [AC 7028; H, c-Pr, H , Cl, S, Pr, H, H, H, O], [AC 7029; H, c-Pr, H, Cl, S, i-Pr, H, H, H, O], [AC 7030; H, c -Pr, H, Cl, S, CH = CH 2, H, H, H, O], [AC7031; H, c-Pr, H, Cl, S, C (CH 3) = CH 2, H, H , H, O], [A H, c-Pr, H, Cl, S, C≡CH, H, H, H, O], [AC7033; H, c-Pr, H, Cl, S, C≡ CCH ₃ , H, H , H, O], [AC 7034; H, c-Pr, H, Cl, S, c-Pr, H, H, H, O], [AC 7035; H, c-Pr, H, Cl, S, OMe , H, H, H, O], [AC 7036; H, c-Pr, H, Cl, S, OEt, H, H, H, O], [AC 7037; H, c-Pr, H, Cl, S , Oi-Pr, H, H, H, O], [AC 7038; H, c-Pr, H, Cl, S, SMe, H, H, H, O], [AC 7039; H, c-Pr, H , Cl, S, SEt, H , H, H, O], [AC7040; H, c-Pr, H, Cl, S, CH 2 F, H, H, H, O], [AC7041; H, c -Pr, H, Cl, S, CHF 2, H, H, H, O], [AC7042; H, c-Pr, H, Cl, S, CF 3, H, H, H, O], [AC7043 ; H, c-Pr, H , Cl, S, OCH 2 F, H, H, H, O], [AC7044; H, c-Pr, H, Cl, S, OCHF 2, H, H, H, O], [AC7045; H, c-Pr, H, Cl, S, OCF 3, H, H, H, O], [AC7046; H, c-Pr, H, Cl, S, SCH 2 F, H , H, H, O], [AC 7047; H, c-Pr, H, Cl, S, SCHF ₂ , H, H, H, O], [AC 7048; H, c-Pr, H, Cl, S, SCF ₃ , H, H, H, O], [AC 7049; H, c-Pr, H, Cl, S, CN, H, H, H, O], [AC 7050; H, c-Pr, H, Cl , S, NO ₂ , H, H, H, O], [AC7051; H, c-Pr, H, Br, S, H, H, H, H, O], [AC7052; H, c-Pr, H, Br, S, F, H, H, H, O], [AC7053; H, c-Pr, H, Br, S, Cl, H, H, O], [AC7054; H, c- Pr, H, Br, S, Br, H, H, H, O], [AC 7055; H, c-Pr, H, Br, S, I, H, H, O], [AC 7056; H, c-Pr, H, Br, S, Me, H, H, H, O], [AC 7057; H, c-Pr, H, Br, S, Et, H, H, H, O], [AC 7058; H, c-Pr, H, Br, S, Pr, H, H, H, O], [AC 7059; H, c-Pr, H, Br, S, i- Pr, H, H, H, O], [AC7060; H, c-Pr, H, Br, S, CH = CH 2, H, H, H, O], [AC7061; H, c-Pr, H , Br, S, C (CH 3) = CH 2, H, H, H, O], [AC7062; H, c-Pr, H, Br, S, C≡CH, H, H, H, O] , [AC7063; H, c- Pr, H, Br, S, C≡CCH 3, H, H, H, O], [AC7064; H, c-Pr, H, Br, S, c-Pr, H , H, H, O], [AC7065; H, c-Pr, H, Br, S, OMe, H, H, H, O], [AC 7066; H, c-Pr, H, Br, S, OEt , H, H, H, O], [AC 7067; H, c-Pr, H, Br, S, Oi-Pr, H, H, H, O], [AC 7068; H, c-Pr, H, Br , S, SMe, H, H, H, O, [AC 7069; H, c-Pr, H, Br, S, SE t, H, H, H, O], [AC 7070; H, c-Pr, H _{, Br, S, CH 2 F} , H, H, H, O], [AC7071; H, c-Pr, H, Br, S, CHF 2, H, H, H, O], [AC7072; H, c-Pr, H, Br, S, CF 3, H, H, H, O], [AC7073; H, c-Pr, H, Br, S, OCH 2 F, H, H, H, O], [AC7074; H, c-Pr , H, Br, S, OCHF 2, H, H, H, O], [AC7075; H, c-Pr, H, Br, S, OCF 3, H, H, H H, c-Pr, H, Br, S, SCH ₂ F, H, H, H, O],

[AC 7077; H, c-Pr, H, Br, S, SCHF ₂ , H, H, H, O], [AC 7078; H, c-Pr, H, Br, S, SCF ₃ , H, H, H , O], [AC 7079; H, c-Pr, H, Br, S, CN, H, H, H, O], [AC 7080; H, c-Pr, H, Br, S, NO ₂ , H, H, H, O], [AC7081; H, F, H, H, S, H, H, H, H, O], [AC7082; H, F, H, H, S, F, H, H, H, H, O], [AC 708 3; H, F, H, H, S, Cl, H, H, H, O], [AC 7084; H, F, H, H, S, Br, H, H, H, H, O], [AC 7085; H, F, H, H, S, I, H, H, H, O], [AC 7086; H, F, H, H, S, Me, H, H, H, O] , [AC 7087; H, F, H, H, S, Et, H, H, H, O], [AC 7088; H, F, H, H, S, Pr, H, H, H] O, [ AC7089; H, F, H, H, S, i-Pr, H, H, H, O], [AC7090; H, F, H, H, S, CH = CH 2, H, H, H, O ], [AC7091; H, F , H, H, S, C (CH 3) = CH 2, H, H, H, O], [AC7092; H, F, H, H, S, C≡CH, H, H, H, O], [AC 709 3; H, F, H, H, S, C≡CCH ₃ , H, H, H, O], [AC 709 4; H, F, H, H, S, c -Pr, H, H, H, O], [AC 7095; H, F, H, H, S, OMe, H, H, H, O], [AC 7096; H, F, H, H, S, OEt H, H, H, O], [AC 7097; H, F, H, H, S, Oi-Pr, H, H, H, O], [AC 7098; H, F, H, H, S, SMe , H, H, H, O], [AC 7099; H, F, H, H, S, SE t, H, H, H, O], [AC 7100; H, F, H, H, S, CH ₂ F , H, H, H, O], [AC 7101; H, F, H, H, S, CHF ₂ , H, H, H, O], [AC 7102; H, F, H, H, S, CF ₃ , H, H, H, O], [AC 7103; H, F, H, H, S, OCH ₂ F, H, H, H, O], [AC 7104; H, F, H, H, S, OCHF _{2, H, H, H,} O], [AC7105; H, F, H, H, S, OCF 3, H, H, H, O], [AC7106; H, F, H, H, S, SCH ₂ F, H, H, H, O], [AC7 107; H, F, H, H, S, SCHF ₂ , H, H, H, O], [AC 7108; H, F, H, H, S, SCF ₃ , H, H, H, O], [ AC 7109; H, F, H, H, S, CN, H, H, H, O], [AC7110; H, F, H, H, S, NO ₂ , H, H, H, O], [AC 7111 H, F, H, Me, S, H, H, H, H, O], [AC7112; H, F, H, Me, S, F, H, H, O], [AC 7113; H , F, H, Me, S, Cl, H, H, H, O], [AC 7114; H, F, H, Me, S, Br, H, H, O], [AC 7115; H, F , H, Me, S, I, H, H, H, O], [AC 7116; H, F, H, Me, S, Me, H, H, O], [AC 7117; H, F, H , Me, S, Et, H, H, H, O], [AC 7118; H, F, H, Me, S, Pr, H, H, H, O], [AC 7119; H, F, H, Me , S, i-Pr, H , H, H, O], [AC7120; H, F, H, Me, S, CH = CH 2, H, H, H, O], [AC7121; H, F, H, Me, S, C ( CH 3) = CH 2, H, H, H, O], [AC7122; H, F, H, Me, S, C≡CH, H, H, H, O], [AC 7123; H, F, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 7124; H, F, H, Me, S, c-Pr, H, H, H, O], [AC 7125; H, F, H, Me, S, OMe, H, H, H, O], [AC 7126; H, F, H, Me, S, OEt, H, H, H, O] , [AC7127; H, F, H, Me, S, Oi-Pr, H, H, H, O], [AC 7128; H, F, H, Me, S, SMe, H, H, H, O] , [AC7129; H, F, H, Me, S, SEt, H, H, H, O], [AC7130; H, F, H, Me, S, CH 2 F, H, H, H, O] , [AC7131; H, F, H, Me, S, CHF 2, H, H, H, O], [AC7132; H, F, H, Me, S, CF 3, H, H, H, O] H, F, H, Me, S, OCH ₂ F, H, H, H, O], [AC 7134; H, F, H, Me, S, OCHF ₂ , H, H, H, O ], [AC7135; H, F , H, Me, S, OCF 3, H, H, H, O], [AC7136; H, F, H, Me, S, SCH 2 F, H, H, H, O H, F, H, Me, S, SCHF ₂ , H, H, H, O], [AC 7138; H, F, H, Me, S, SCF ₃ , H, H, H, O] H, F, H, Me, S, CN, H, H, H, O], [AC 7140; H, F, H, Me, S, NO ₂ , H, H, H, O] , [AC7141; H, F, H, Et, S, H, H, H, O], [AC7142; H, F, H, Et, S, F, H, H, O], [AC7142; AC7143; H, F, H, Et, S, Cl, H, H, H, O], [AC7144; H, F, H, Et, S, Br, H, H, H, O], [AC7145; H, F, H, Et, S, I, H, H, H, O], [AC 7146; H, F, H, Et, S, Me, H, H, O], [AC 7147; H, F, H, Et, S, Et, H, H, H, O], [AC7148; H, F, H, Et, S, Pr, H, H, O, [AC 7149; H, F, H, Et, S, i- Pr, H, H, H, O], [AC7150; H, F, H, Et, S, CH = CH 2, H, H, H, O], [AC7151; H , F, H, Et, S , C (CH 3) = CH 2, H, H, H, O], [AC7152; H, F, H, Et, S, C≡CH, H, H, H, H, F, H, Et, S, C≡CCH ₃ , H, H, H, O], [AC 7154; H, F, H, Et, S, c-Pr, H, H , H, O], [AC 7 155; H, F, H, Et, S, OMe, H, H, H, O], [AC 7156; H, F, H, Et, S, OE t, H, H, H H, F, H, Et, S, Oi-Pr, H, H, H, O], [AC 7158; H, F, H, Et, S, SMe, H, H, H H, F, H, Et, S, SEt, H, H, H, O], [AC 7160; H, F, H, Et, S, CH ₂ F, H, H, H , O], [AC7161; H , F, H, Et, S, CHF 2, H, H, H, O], [AC7162; H, F, H, Et, S, CF 3, H, H, H , O], [AC7163; H , F, H, Et, S, OCH 2 F, H, H, H, O], [AC7164; H, F, H, Et, S, OCHF 2, H, H, H, O], [AC7165; H, F, H, Et, S, OCF 3, H, H, H, O], [AC7166; H, F, H, Et, S, SCH 2 F, H, H, H, O], [AC 7167; H, F, H, Et, S, SCHF ₂ , H, H, H, O], [AC 7168; H, F, H, Et, S, SCF ₃ , H, H, H, O], [AC7169; H, F, H, Et, S, CN, H, H, H, O], [AC 7170; H, F, H, Et, S, NO ₂ , H, H, H, O], [AC7171; H, F, H, Pr, S, H, H, H, H, O], [AC7172; H, F, H, Pr, S, F, H , H, H, O], [AC7173; H, F, H, Pr, S, Cl, H, H, H, O], [AC7174; H, F, H, Pr, S, Br, H, H , H, O], [AC 7175; H, F, H, Pr, S, I, H, H, H, O], [AC 7176; H, F, H, Pr, S, Me, H, H, H , O],

[AC7177; H, F, H, Pr, S, Et, H, H, H, O], [AC7178; H, F, H, Pr, S, Pr, H, H, H, O], [AC7179 H, F, H, Pr, S, i-Pr, H, H, H, O], [AC 7180; H, F, H, Pr, S, CH = CH ₂ , H, H, H, O] , [AC7181; H, F, H, Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC7182; H, F, H, Pr, S, C≡CH, H , H, H, O], [AC 7183; H, F, H, Pr, S, C≡CCH ₃ , H, H, H, O], [AC 7184; H, F, H, Pr, S, c- Pr, H, H, H, O], [AC 7185; H, F, H, Pr, S, OMe, H, H, H, O], [AC 7186; H, F, H, Pr, S, OE t, H, H, H, O], [AC7187; H, F, H, Pr, S, Oi-Pr, H, H, H, O], [AC 7188; H, F, H, Pr, S, SMe, H, H, H, O], [AC 7189; H, F, H, Pr, S, SE t, H, H, H, O], [AC 7190; H, F, H, Pr, S, CH ₂ F, H, H, H, O] , [AC7191; H, F, H, Pr, S, CHF 2, H, H, H, O], [AC7192; H, F, H, Pr, S, CF 3, H, H, H, O] , [AC7193; H, F, H, Pr, S, OCH 2 F, H, H, H, O], [AC7194; H, F, H, Pr, S, OCHF 2 , H, H, H, O ], [AC7195; H, F, H, Pr, S, OCF 3, H, H, H, O], [AC7196; H, F, H, Pr, S, SCH 2 F, H, H, H, O], [AC7197; H, F, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 7198; H, F, H, Pr, S, SCF ₃ , H, H, H, O], [AC 7199; H, F, H, Pr, S, CN, H, H, H, O], [AC 7200; H, F, H, Pr, S, NO ₂ , H, H, H, O], [AC 7201; H, F, H, i-Pr, S, H, H, H, H, O], [AC 7202; H, F, H, i-Pr, S , F, H, H, H, O], [AC 7203; H, F, H, i-Pr, S, Cl, H, H, H, O], [AC 7204; H, F, H, i-Pr , S, Br, H, H, H, O], [AC 7205; H, F, H, i-Pr, S, I, H, H, O], [AC 7206; H, F , H, i-Pr, S, Me, H, H, H, O], [AC 7207; H, F, H, i-Pr, S, Et, H, H, H] O, [AC 7208; H , F, H, i-Pr, S, Pr, H, H, H, O], [AC 7209; H, F, H, i-Pr, S, i-Pr, H, H, H, O], [AC7210; H, F, H , i-Pr, S, CH = CH 2, H, H, H, O], [AC7211; H, F, H, i-Pr, S, C (CH 3) = _{CH 2, H, H, H} , O], [AC7212; H, F, H, i-Pr, S, C≡CH, H, H, H, O], [AC7213; H, F, H, i -Pr, S, C≡CCH ₃ , H, H, H, O], [AC 7214; H, F, H, i-Pr, S, c-Pr, H, H, H, O], [AC 7215; H, F, H, i-Pr, S, OMe, H, H, H, O], [AC7216; H, F, H, i-Pr, S, OEt, H, H, H, O], [[ AC 7217; H, F, H, i-Pr, S, Oi-Pr, H, H, H, O], [AC 7218; H, F, H, i-Pr, S, SMe, H, H, H, O], [AC7219; H, F, H, i-Pr, S, SEt, H, H, H, O], [AC7220; H, F, H, i-Pr, S, CH 2 F, H, H, H, O], [ AC7221; H, F, H, i-Pr, S, CHF 2, H, H, H, O], [AC7222; H, F, H, i-Pr, S, CF _{3, H, H, H,} O], [AC7223; H, F, H, i-Pr, S, OCH 2 F, H, H, H, O], [AC7224; H, F, H, i- _{Pr, S, OCHF 2, H} , H, H, O], [AC7225; H, F, H, i-Pr, S, OCF 3, H, H, H, O], [AC7226; H, F, H, i-Pr, S, SCH ₂ F, H, H, H, O], [AC 7227; H, F, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 7228 ; H, F, H, i -Pr, S, SCF 3, H, H, H, O], [AC7229; H, F, H, i-Pr, S, CN, H, H, H, O] , [AC7230; H, F, H, i-Pr, S, NO 2, H, H, H, O], [AC7231; H, F, H, c-Pr, S, H, H, H, H H, F, H, c-Pr, S, F, H, H, H, O], [AC7233; H, F, H, c-Pr, S, Cl, H, H] , H, O], [AC 723 4; H, F, H, c-Pr, S, Br, H, H, H, O], [AC 7235; H, F, H, c-Pr, S, I, H, H, H, O] H, F, H, c-Pr, S, Me, H, H, H, O], [AC 7237; H, F, H, c-Pr, S, Et, H, H, H, O, [AC 7238; H, F, H, c-Pr, S, Pr, H, H, H, O], [AC 7239; H, F, H, c-Pr, S, i-Pr, H, H, H, O], [ AC7240; H, F, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC7241; H, F, H, c-Pr, S , C (CH ₃ ) = CH ₂ , H, H, H, O], [AC7242; H, F, H, c-Pr, S, C≡CH, H, H, H, O], [AC7243; H, F, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC7244; H, F, H, c-Pr, S, c-Pr, H, H, H , O], [AC7245; H, F, H, c-Pr, S, OMe, H, H, H, O], [AC7246; H, F, H, c-Pr, S, OEt, H, H , H, O], [AC7247; H, F, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 7248; H, F, H, c-Pr, S, SMe , H, H, H, O], [AC 7249; H, F, H, c-Pr, S, SE t, H, H, H, O], [AC 7250; H, F, H, c-Pr, S _{, CH 2 F, H, H} , H, O], [AC7251; H, F, H, c-Pr, S, CHF 2, H, H, H, O], [AC7252; H, F, H, _{c-Pr, S, CF 3} , H, H, H, O], [AC7253; H, F, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC7254; H , F, H, c-Pr , S, OCHF 2, H, H, H, O], [AC7255; H, F, H, c-Pr, S, OCF 3, H, H, H, O], [AC 7256; H, F, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 7257; H, F, H, c-Pr, S, SCHF ₂ , H, H, H, O], [AC 7258; H, F, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 7259; H, F, H, c-Pr, S, CN, H , H, H, O], [AC7260; H, F, H, c-Pr, S, NO 2, H, H, H, O], [AC7261; H, F, H, SMe, S, H, H, H, H, O], [A H, F, H, SMe, S, F, H, H, H, O], [AC 7263; H, F, H, SMe, S, Cl, H, H, H, O], [AC 7264; H, F, H, SMe, S, Br, H, H, H, O], [AC7265; H, F, H, SMe, S, I, H, H, O], [AC7266; H, F, H, SMe, S, Me, H, H, H, O], [AC 7267; H, F, H, SMe, S, Et, H, H, O], [AC 7268; H, F, H, SMe, S, Pr, H, H, H, O], [AC 7269; H, F, H, SMe, S, i-Pr, H, H, H, O], [AC 7270; H, F, H, SMe, S, CH = CH 2, H, H, H, O], [AC7271; H, F, H, SMe, S, C (CH 3) = CH 2, H, H, H, O] , [AC7272; H, F, H, SMe, S, C≡CH, H, H, H, O], [AC7273; H, F, H, SMe, S, C≡ CCH ₃ , H, H, H H, F, H, SMe, S, c-Pr, H, H, H, O], [AC7275; H, F, H, SMe, S, OMe, H, H, H , O],

[AC 7276; H, F, H, SMe, S, OEt, H, H, H, O], [AC 7277; H, F, H, SMe, S, Oi-Pr, H, H, H, O], [AC 7278; H, F, H, SMe, S, SMe, H, H, H, O], [AC 7279; H, F, H, SMe, S, SE t, H, H, H, O], [AC 7280 ; H, F, H, SMe , S, CH 2 F, H, H, H, O], [AC7281; H, F, H, SMe, S, CHF 2, H, H, H, O], [ AC7282; H, F, H, SMe, S, CF 3, H, H, H, O], [AC7283; H, F, H, SMe, S, OCH 2 F, H, H, H, O], [AC7284; H, F, H , SMe, S, OCHF 2, H, H, H, O], [AC7285; H, F, H, SMe, S, OCF 3, H, H, H, O], [AC 7286; H, F, H, SMe, S, SCH ₂ F, H, H, H, O], [AC 7287; H, F, H, SMe, S, SCHF ₂ , H, H, H, O] , [AC7288; H, F, H, SMe, S, SCF 3, H, H, H, O], [AC7289; H, F, H, SMe, S, CN, H, H, H, O], [AC7290; H, F, H , SMe, S, NO 2, H, H, H, O], [AC7291; H, F, H, OMe, S, H, H, H, H, O], [ AC7292; H, F, H, OMe, S, F, H, H, O], [AC7293; H, F, H, OMe, S, Cl, H, H, H, O], [AC7294; H, F, H, OMe, S, Br, H, H, H, O], [AC7295; H, F, H, OMe, S, I, H, H, O], [AC 7296; H, F, H, OMe, S, Me, H, H, H, O], [AC 7297; H, F, H, OMe, S, Et, H, H, H, O], [AC 7298; H, F, H, OMe, S, Pr, H, H, H, O], [AC 7299; H, F, H, OMe, S, i-Pr, H, H, H, O], [AC 7300; H, F, H, OMe, S, CH = CH 2, H, H, H, O], [AC7301; H, F, H, OMe, S, C (CH 3) = CH 2, H, H, H, O] H, F, H, OMe, S, C≡CH, H, H, H, O], [AC 7303; H, F, H, OMe, S, C≡ CCH ₃ , H, H, H , O], [AC 7304; H, F, H, OMe, S, c-Pr, H, H, H, O], [AC 7305; H, F, H, OMe, S, OMe, H, H, H, O], [AC 7306; H, F, H, OMe, S, OE t, H, H, H, H, O], [AC 7307; H, F, H, OMe, S, Oi-Pr, H, H, H, O], [AC 7308; H, F, H, OMe, S, SMe, H, H, H, H, O], [AC 7309; H, F, H, OMe, S, SE t, H, H, H, O], [AC 7310; H, F, H, OMe, S, CH ₂ F, H, H, H, O], [AC7311; H, F, H, OMe, S, CHF 2, H, H, H, O], [AC7312; H, F, H, OMe, S, CF 3, H, H, H, O], [AC7313; H, F, H, OMe, S, OCH 2 F, H, H, H, O], [AC7314; H, F, H, OMe, S, OCHF 2, H, H , H, O], [AC7315 ; H, F, H, OMe, S, OCF 3, H, H, H, O], [AC7316; H, F, H, OMe, S, SCH 2 F, H, H, H, O], [AC 7317; H, F, H, OMe, S, SCHF ₂ , H, H, H, O], [AC 7318; H, F, H, OMe, S, SCF ₃ , H, H, H, O], [AC7319; H, F, H, OMe, S, CN, H, H, H, O], [AC 7320; H, F, H, OMe, S, NO ₂ , H, H , H, O], [AC7321; H, F, H, F, S, H, H, H, H, O], [AC7322; H, F, H, F, S, F, H, H, H H, F, H, F, S, Cl, H, H, O], [AC7324; H, F, H, F, S, Br, H, H, H, O] H, F, H, F, S, I, H, H, H, O], [AC 7326; H, F, H, F, S, Me, H, H, H, O], [AC 7327; H, F, H, F, S, Et, H, H, H, O], [AC 7328; H, F, H, F, S, Pr, H, H, O], [AC 7329 ; H, F, H, F , S, i-Pr, H, H, H, O], [AC7330; H, F, H, F, S, CH = CH 2, H, H, H, O] , [AC7331; H, F, H, F, S, C (CH 3) = CH 2, H, H, H, O], [AC7332; H, F, H, F, S, C≡CH, H , H, H, O], [AC7333; H, F, H, F, S, C≡CCH ₃ , H, H, H, O], [AC7334; H, F, H , F, S, c-Pr, H, H, H, O], [AC7335; H, F, H, F, S, OMe, H, H, O], [AC 7336; H, F, H , F, S, OEt, H, H, H, O], [AC 7337; H, F, H, F, S, Oi-Pr, H, H, H, O], [AC 7338; H, F, H , F, S, SMe, H, H, H, O], [AC 7339; H, F, H, F, S, SE t, H, H, H, O], [AC 7340; H, F, H, F _{, S, CH 2 F, H} , H, H, O], [AC7341; H, F, H, F, S, CHF 2, H, H, H, O], [AC7342; H, F, H, _{F, S, CF 3, H} , H, H, O], [AC7343; H, F, H, F, S, OCH 2 F, H, H, H, O], [AC7344; H, F, H _{, F, S, OCHF 2,} H, H, H, O], [AC7345; H, F, H, F, S, OCF 3, H, H, H, O], [AC7346; H, F, H , F, S, SCH ₂ F, H, H, H, O, [AC 7347; H, F, H, F, S, SCHF ₂ , H, H, H, O], [AC 7348; H, F, _{H, F, S, SCF 3} , H, H, H, O], [AC7349; H, F, H, F, S, CN, H, H, H, O], [AC7350; H, F, H , F, S, NO ₂ , H, H, H, O], [AC 7351; H, F, H, Cl, S, H, H, H, H, O], [AC 7352; H, F, H, Cl, S, F, H, H, H, O], [AC7353; H, F, H, Cl, S, Cl, H, H, H, O], [AC7354; H, F, H, Cl, S, Br, H, H, H, O], [AC7355; H, F, H, Cl, S, I, H, H, O], [AC 7356; H, F, H, Cl, S, Me, H, H, H, O], [AC 7357; H, F, H, Cl, S, Et, H, H, H, O], [AC 7358; H, F, H, Cl, S, Pr, H, H, H, O], [AC 7359; H, F, H, Cl, S, i-Pr, H, H, H, O], [AC 7360; H, F, H, Cl, S, CH = _{CH 2, H, H, H} , O], [AC7361; H, F, H, Cl, S, C (CH 3) = CH 2, H, H, H, O], [AC7362; H, F, H, Cl, S, C≡CH, H, H, H, O], [AC7363; H, F, H, Cl, S, C≡CCH 3, H, H, H, O], [AC7364; H , F, H, Cl, S, c -Pr, H, H, H, O], [AC7365; H, F, H, Cl, S, OMe, H, H, H, O], [AC 7366; H, F, H, Cl, S, OEt , H, H, H, O], [AC 7367; H, F, H, Cl, S, Oi-Pr, H, H, H, O], [AC 7368; H, F, H, Cl, S, SMe H, H, H, O], [AC 7369; H, F, H, Cl, S, SE t, H, H, H, O], [AC 7370; H, F, H, Cl, S, CH ₂ F , H, H, H, O], [AC 7371; H, F, H, Cl, S, CHF ₂ , H, H, H, O], [AC 7372; H, F, H, Cl, S, CF ₃ , H, H, H, O], [AC 7373; H, F, H, Cl, S, OCH ₂ F, H, H, H, O], [AC 7374; H, F, H, Cl, S, OCHF _{2, H, H, H,} O], [AC7375; H, F, H, Cl, S, OCF 3, H, H, H, O],

[AC 7376; H, F, H, Cl, S, SCH ₂ F, H, H, H, O], [AC 7377; H, F, H, Cl, S, SCHF ₂ , H, H, H, O] [AC 7378; H, F, H, Cl, S, SCF ₃ , H, H, H, O], [AC 7379; H, F, H, Cl, S, CN, H, H, H, O], [AC7380; H, F, H , Cl, S, NO 2, H, H, H, O], [AC7381; H, F, H, Br, S, H, H, H, H, O], [ AC7382; H, F, H, Br, S, F, H, H, O], [AC7383; H, F, H, Br, S, Cl, H, H, H, O], [AC7384; H, F, H, Br, S, Br, H, H, H, O], [AC 7385; H, F, H, Br, S, I, H, H, O], [AC 7386; H, F, H, Br, S, Me, H, H, H, O], [AC 7387; H, F, H, Br, S, Et, H, H, O], [AC 7388; H, F, H, Br, S, Pr, H, H, H, O], [AC 7389; H, F, H, Br, S, i-Pr, H, H, H, O], [AC 7390; H, F, H, Br, S, CH = CH 2, H, H, H, O], [AC7391; H, F, H, Br, S, C (CH 3) = CH 2, H, H, H, O] , [AC 7392; H, F, H, Br, S, C, CH, H, H, H, O], [AC 7393; H, F, H, Br, S, C≡ CCH ₃ , H, H, H , O], [AC 7394; H, F, H, Br, S, c-Pr, H, H, H, O], [AC 7395; H, F, H, Br, S, OMe, H, H, H H, F, H, Br, S, OEt, H, H, H, O], [AC 7397; H, F, H, Br, S, Oi-Pr, H, H, H H, F, H, Br, S, SMe, H, H, H, O], [AC 7399; H, F, H, Br, S, SE t, H, H, H, O ], [AC7400; H, F , H, Br, S, CH 2 F, H, H, H, O], [AC7401; H, F, H, Br, S, CHF 2, H, H, H, O], [AC7402; H, F, H, Br, S, CF 3, H, H, H, O], [AC7403; H, F, H, Br, S, OCH 2 F, H, H, H , O], [AC7404; H , F, H, Br, S, OCHF 2, H, H, H, O], [AC7405; H, F, H, Br, S, OCF 3 H, H, H, O], [AC 7406; H, F, H, Br, S, SCH ₂ F, H, H, H, O], [AC 7407; H, F, H, Br, S, SCHF ₂ , H, H, H, O], [AC 7408; H, F, H, Br, S, SCF ₃ , H, H, H, O], [AC 7409; H, F, H, Br, S, CN H, H, H, O], [AC 7410; H, F, H, Br, S, NO ₂ , H, H, H, O], [AC 7411; H, Cl, H, H, S, H, H, H, H, O], [AC 7412; H, Cl, H, H, S, F, H, H, H, O], [AC 7413; H, Cl, H, H, S, Cl, H, H, H, O], [AC 7414; H, Cl, H, H, S, Br, H, H, H, O], [AC 7415; H, Cl, H, H, S, I, H, H, H, O], [AC 7416; H, Cl, H, H, S, Me, H, H, H, O], [AC 7417; H, Cl, H, H, S, Et, H, H, H, H, H, Cl, H, H, S, Pr, H, H, H, O], [AC 7419; H, Cl, H, H, S, i-Pr, H, H, H, O], [AC 7418; O], [AC7420; H, Cl, H, H, S, CH = CH 2, H, H, H, O], [AC7421; H, Cl, H, H, S, C (CH 3) = CH ₂ , H, H, H, O], [AC 7422; H, Cl, H, H, S, C3CH, H, H, H, O], [AC 7243; H, Cl, H, H, S, C≡CCH ₃ , H, H, H, O], [AC7424; H, Cl, H, H, S, c-Pr, H, H, H, O], [AC 7425; H, Cl, H, H , S, OMe, H, H, H, O], [AC 7426; H, Cl, H, H, S, OEt, H, H, H, O], [AC 7427; H, Cl, H, H, S , Oi-Pr, H, H, H, O], [AC 7428; H, Cl, H, H, S, SMe, H, H, H, O], [AC 7429; H, Cl, H, H, S , SEt, H, H, H, O], [AC 7430; H, Cl, H, H, S, CH ₂ F, H, H, H, O], [AC 743 1; H, Cl, H, H, S _{, CHF 2, H, H,} H, O], [AC7432; H, Cl, H, H, S, CF 3, H, H, H, O], [AC7433; H, Cl, H, H, S OCH ₂ F, H, H, H, O, [AC 743 4; H, Cl, H, H, S, OCHF ₂ , H, H, H, O], [AC 7435; H, Cl, H, _{H, S, OCF 3, H} , H, H, O], [AC7436; H, Cl, H, H, S, SCH 2 F, H, H, H, O], [AC7437; H, Cl, H _{, H, S, SCHF 2,} H, H, H, O], [AC7438; H, Cl, H, H, S, SCF 3, H, H, H, O], [AC7439; H, Cl, H , H, S, CN, H, H, H, O], [AC 7440; H, Cl, H, H, S, NO ₂ , H, H, H, O], [AC7441; H, Cl, H, Me, S, H, H, H, H, H, O], [AC7442; H, Cl, H, Me, S, F, H, H, H, O], [AC7443; H, Cl, H, Me, S, Cl, H, H, H, O], [AC7444; H, Cl, H, Me, S, Br, H, H, H, O], [AC 7445; H, Cl, H, Me, S, H, Cl, H, Me, S, Me, H, H, H, O], [AC 7447; H, Cl, H, Me, S, Et, I, H, H, H, O], [AC 7446; H, H, H, O], [AC 7 448; H, Cl, H, Me, S, Pr, H, H, H, O], [AC 7449; H, Cl, H, Me, S, i-Pr, H, H, H, O] , [AC7450; H, Cl, H, Me, S, CH = CH 2, H, H, H, O], [AC7451; H, Cl, H, Me, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC7452; H, Cl, H, Me, S, C≡CH, H, H, H, O], [AC7453; H, Cl, _{H, Me, S, C≡CCH 3} , H, H, H, O], [AC7454; H, Cl, H, Me, S, c-Pr, H, H, H, O], [AC7455; H , Cl, H, Me, S, OMe, H, H, H, O], [AC 7456; H, Cl, H, Me, S, OEt, H, H, H, O], [AC 7457; H, Cl , H, Me, S, Oi-Pr, H, H, H, O], [AC 7458; H, Cl, H, Me, S, SMe, H, H, O], [AC 7459; H, Cl , H, Me, S, SEt , H, H, H, O], [AC7460; H, Cl, H, Me, S, CH 2 F, H, H, H, O], [AC7461; H, Cl , H, Me, S, CHF 2, H, H, H, O], [AC7462; H, Cl, H, Me, S, CF 3, H, H, H, O], [AC7463; H, Cl , H, Me, S, OCH ₂ F, H, H, H, O], [AC7464; H, Cl, H, Me, _{S, OCHF 2, H, H} , H, O], [AC7465; H, Cl, H, Me, S, OCF 3, H, H, H, O], [AC7466; H, Cl, H, Me, S, SCH ₂ F, H, H, H, O], [AC 7467; H, Cl, H, Me, S, SCHF ₂ , H, H, H, O], [AC 7468; H, Cl, H, Me , S, SCF ₃ , H, H, H, O], [AC 7469; H, Cl, H, Me, S, CN, H, H, H, O], [AC 7470; H, Cl, H, Me, _{S, NO 2, H, H} , H, O], [AC7471; H, Cl, H, Et, S, H, H, H, H, O], [AC7472; H, Cl, H, Et, S , F, H, H, H, O], [AC7473; H, Cl, H, Et, S, Cl, H, H, H, O], [AC 7474; H, Cl, H, Et, S, Br , H, H, H, O], [AC 7475; H, Cl, H, Et, S, I, H, H, H, O],

[AC 7476; H, Cl, H, Et, S, Me, H, H, H, O], [AC 7477; H, Cl, H, Et, S, Et, H, H, H, O], [AC 7478 H, Cl, H, Et, S, Pr, H, H, H, O], [AC 7479; H, Cl, H, Et, S, i-Pr, H, H, H, O], [AC 7480 ; H, Cl, H, Et , S, CH = CH 2, H, H, H, O], [AC7481; H, Cl, H, Et, S, C (CH 3) = CH 2, H, H , H, O], [AC 7482; H, Cl, H, Et, S, C≡CH, H, H, H, O], [AC 7483; H, Cl, H, Et, S, C≡ CCH ₃ , H, H, H, O], [AC 7484; H, Cl, H, Et, S, c-Pr, H, H, H, O], [AC 7485; H, Cl, H, Et, S, OMe, H, H, H, O], [AC 7486; H, Cl, H, Et, S, OEt, H, H, H, O], [AC 7487; H, Cl, H, Et, S, Oi-Pr, H, H, H, O], [AC 7488; H, Cl, H, Et, S, SMe, H, H, H, O], [AC 7489; H, Cl, H, Et, S, SE t, H, H, H, O], [ AC7490; H, Cl, H, Et, S, CH 2 F, H, H, H, O], [AC7491; H, Cl, H, Et, S, CHF 2, H , H, H, O], [AC7492; H, Cl, H, Et, S, CF 3, H, H, H, O], [AC7493; H, Cl, H, Et, S, OCH 2 F, H, H, H, O] , [AC7494; H, Cl, H, Et, S, OCHF 2, H, H, H, O], [AC7495; H, Cl, H, Et, S, OCF 3, H, H, H, O], [AC 7496; H, Cl, H, Et, S, SCH ₂ F, H, H, H, O], [AC 7497; H, Cl, H, Et, S, SCHF ₂ , H, H, H, O ], [AC7498; H, Cl, H, Et, S, SCF 3, H, H, H, O], [AC7499; H, Cl, H, Et, S, CN, H, H, H, O] , [AC7500; H, Cl, H, Et, S, NO 2, H, H, H, O], [AC7501; H, Cl, H, Pr, S, H, H , H, H, O], [AC 7502; H, Cl, H, Pr, S, F, H, H, H, O], [AC 7503; H, Cl, H, Pr, S, Cl, H, H , H, O], [AC 7504; H, Cl, H, Pr, S, Br, H, H, H, O], [AC 7505; H, Cl, H, Pr, S, I, H, H, H, O], [AC 7506; H, Cl, H, Pr, S, Me, H, H, H, O], [AC 7507; H, Cl, H, Pr, S, Et, H, H, H, O], [AC 7508; H, Cl, H, Pr, S, Pr, H, H, H, O], [AC7509; H, Cl, H, Pr, S, i-Pr, H, H, H, O], [AC7510; H, Cl, H, Pr, S, CH = CH 2, H H, H, O], [AC 7511; H, Cl, H, Pr, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 7512; H, Cl, H, Pr, S, C≡CH, H, H, H, O, [AC 7513; H, Cl, H, Pr, S, C≡CCH ₃ , H, H, H, O], [AC 7514; H, Cl, H , Pr, S, c-Pr, H, H, H, O], [AC 7515; H, Cl, H, Pr, S, OMe, H, H, O], [AC 7516; H, Cl, H , Pr, S, OEt, H, H, H, O], [AC 7517; H, Cl, H, Pr, S, Oi-Pr, H, H, H, O], [AC 7518; H, Cl, H , Pr, S, SMe, H, H, H, O], [AC 7519; H, Cl, H, Pr, S, SE t, H, H, H, O], [AC 7520; H, Cl, H, Pr , S, CH ₂ F, H, H, H, O], [AC 7521; H, Cl, H, Pr, S, CHF ₂ , H, H, H, O], [AC 7522; H, Cl, H, _{Pr, S, CF 3, H} , H, H, O], [AC7523; H, Cl, H, Pr, S, OCH 2 F, H, H, H, O], [AC7524; H, Cl, H , Pr, S, OCHF ₂ , H, H, H, O], [AC 7525; H, Cl, H, Pr, S, OCF ₃ , H, H, H, O], [AC 7526; H, Cl, H , Pr, S, SCH ₂ F, H, H, H, O], [AC 7527; H, Cl, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 7528; H, Cl, _{H, Pr, S, SCF 3} , H, H, H, O], [AC7529; H, Cl, H, Pr, S, CN, H, H, H, O], [AC7530; H, Cl, H , Pr, S, NO ₂ , H, H, H, O], [AC 7531; H, Cl, H, i-Pr, S, H, H, H, O], [AC 7532; H, Cl, H, i-Pr, S, F, H, H, H, O], [AC 7533; H, C l, H, i-Pr, S, Cl, H, H, H, O], [AC7534; H, Cl, H, i-Pr, S, Br, H, H, O], [AC 7535; H, Cl, H, i-Pr, S, I, H, H, H, O], [AC 7536; H, Cl, H, i-Pr, S, Me, H, H, H, O], [[ AC 7537; H, Cl, H, i-Pr, S, Et, H, H, H, O], [AC 7538; H, Cl, H, i-Pr, S, Pr, H, H, H, O] , [AC7539; H, Cl, H, i-Pr, S, i-Pr, H, H, H, O], [AC7540; H, Cl, H, i-Pr, S, CH = CH 2, H , H, H, O], [AC7541; H, Cl, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC7542; H, Cl, H, i-Pr, S, C≡CH, H, H, H, O], [AC7543; H, Cl, H, i-Pr, S, C≡CCH 3, H, H, H, O], [AC7544 H, Cl, H, i-Pr, S, c-Pr, H, H, H, O], [AC7545; H, Cl, H, i-Pr, S, OMe, H, H, H, O H, Cl, H, i-Pr, S, OEt, H, H, H, O], [AC 7547; H, Cl, H, i-Pr, S, Oi-Pr, H, H] , H, O], [AC7548; H, Cl, H, i-Pr, S, SMe, H, H, H, O], [AC7549; H, Cl, H, i-Pr, S, SEt, H , H, H, O], [AC7550; H, Cl, H, i-Pr, S, CH 2 F, H, H, H, O], [AC7551; H, Cl, H, i-Pr, S _{, CHF 2, H, H,} H, O], [AC7552; H, Cl, H, i-Pr, S, CF 3, H, H, H, O], [AC7553; H, Cl, H, i _{-Pr, S, OCH 2 F,} H, H, H, O], [AC7554; H, Cl, H, i-Pr, S, OCHF 2, H, H, H, O], [AC7555; H, Cl, H, i-Pr, S, OCF 3, H, H, H, O], [AC7556; H, Cl, H, i-Pr, S, SCH 2 F, H, H, H, O], [AC7557; H, Cl, H , i-Pr, S, SCHF 2, H, H, H, O], [AC7558; H, Cl, H, i-Pr, S, SCF 3, H, H, H , O], [AC7559; H, Cl, H, i-Pr, S, CN, H, H, H, O], [AC 7560; H, Cl, H , i-Pr, S, NO ₂ , H, H, H, O], [AC7561; H, Cl, H, c-Pr, S, H, H, H, O], [AC7562; H, Cl, H, c-Pr, S, F, H, H, H, O], [AC7563; H, Cl, H, c-Pr, S, Cl, H, H, H, O], [AC7564; H, Cl, H, c-Pr, S, Br, H, H, H, O], [AC7565; H, Cl, H, c-Pr, S, I, H, H, H] O, [, AC 7566; H, Cl, H, c-Pr, S, Me, H, H, H, O], [AC 7567; H, Cl, H, c-Pr, S, Et, H, H, H, O] [AC 7568; H, Cl, H, c-Pr, S, Pr, H, H, H, O], [AC 7569; H, Cl, H, c-Pr, S, i-Pr, H, H, H, O], [AC7570; H, Cl, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC7571; H, Cl, H, c-Pr, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 7572; H, Cl, H, c-Pr, S, C≡CH, H, H, H, O], [AC 7573; H, Cl, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 7574; H, Cl, H, c-Pr, S, c-Pr, H, H, H, O ],

[AC7575; H, Cl, H, c-Pr, S, OMe, H, H, H, O], [AC 7576; H, Cl, H, c-Pr, S, OEt, H, H, H, O H, Cl, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 7578; H, Cl, H, c-Pr, S, SMe, H, H] , H, O], [AC 7579; H, Cl, H, c-Pr, S, SE t, H, H, H, O], [AC 7580; H, Cl, H, c-Pr, S, CH ₂ F , H, H, H, O ], [AC7581; H, Cl, H, c-Pr, S, CHF 2, H, H, H, O], [AC7582; H, Cl, H, c-Pr, _{S, CF 3, H, H} , H, O], [AC7583; H, Cl, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC7584; H, Cl, H , c-Pr, S, OCHF ₂ , H, H, H, O], [AC 7585; H, Cl, H, c-Pr, S, OCF ₃ , H, H, H] O, [AC 7586; H , Cl, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 7587; H, Cl, H, c-Pr, S, SCHF ₂ , H, H, H, O] , [AC7588; H, Cl, H, c-Pr, S, SCF 3, H, H, H, O], [AC7589; H, Cl, H, c-Pr, S, CN, H, H, H , O], [AC7590; H , Cl, H, c-Pr, S, NO 2, H, H, H, O], [AC7591; H, Cl, H, SMe, S, H, H, H, H, O], [AC7592; H, Cl, H, SMe, S, F, H, H, H, O], [AC7593; H, Cl, H, SMe, S, Cl, H, H, H, O], [AC7594; H, Cl, H, SMe, S, Br, H, H, O], [AC7595; H, Cl, H, SMe, S, I, H, H, H, O] , [AC7596; H, Cl, H, SMe, S, Me, H, H, H, O], [AC 7597; H, Cl, H, SMe, S, Et, H, H, H, O], [AC7597; AC 7598; H, Cl, H, SMe, S, Pr, H, H, H, O], [AC 7599; H, Cl, H, SMe, S, i-Pr, H, H, H, O], [ AC7600; H, Cl, H, SMe, S, CH = CH 2, H, H, H, O], [AC7601; H, Cl, H, SMe, S, C (CH 3) = CH 2, H, H, H, O], [AC7602; H, Cl, H, SMe, S, C≡CH , H, H, H, O ], [AC7603; H, Cl, H, SMe, S, C≡CCH 3, H, H, H, O], [AC7604; H, Cl, H, SMe, S, c-Pr, H, H, H, O], [AC7605; H, Cl, H, SMe, S, OMe, H, H, H, O], [AC 7606; H, Cl, H, SMe, S, H, Cl, H, SMe, S, Oi-Pr, H, H, H, O], [AC 7608; H, Cl, H, SMe, S, OETt, H, H, H, O], [AC 7607; SMe, H, H, H, O], [AC 7609; H, Cl, H, SMe, S, SEt, H, H, H, O], [AC 7610; H, Cl, H, SMe, S, CH ₂ F, H, H, H, O], [AC7611; H, Cl, H, SMe, S, CHF 2, H, H, H, O], [AC7612; H, Cl, H, SMe, S, CF _{3, H, H, H,} O], [AC7613; H, Cl, H, SMe, S, OCH 2 F, H, H, H, O], [AC7614; H, Cl, H, SMe, S, _{OCHF 2, H, H, H} , O], [AC7615; H, Cl, H, SMe, S, OCF 3, H, H, H, O], [AC7616; H, Cl, H, SMe, S, SCH ₂ F, H, H, H, O], [AC 7617; H, Cl, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 7618; H, Cl, H, SMe, S , SCF ₃ , H, H, H, O], [AC 7619; H, Cl, H, SMe, S, CN, H, H, H, O], [AC 7620; H, Cl, H, SMe, S, _{NO 2, H, H, H} , O], [AC7621; H, Cl, H, OMe, S, H, H, H, H, O], [AC7622; H, Cl, H, OMe, S, F H, H, H, O], [AC7623; H, Cl, H, OMe, S, Cl, H, H, H, O], [AC7624; H, Cl, H, OMe, S, Br, H H, H, O], [AC 7625; H, Cl, H, OMe, S, I, H, H, H, O], [AC 7626; H, Cl, H, OMe, S, Me, H, H , H, O], [AC 7627; H, Cl, H, OMe, S, Et, H, H, H, O], [AC 7628; H, Cl, H, OMe, S, Pr, H, H, H H, Cl, H, OMe, S, i-Pr, H, H, H, O], [AC 7630; H, Cl, H, OMe, S, CH = CH ₂ , H, H, H, O], [A C7631; H, Cl, H, OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC7632; H, Cl, H, OMe, S, C≡CH, H, H , H, O], [AC7633; H, Cl, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC7634; H, Cl, H, OMe, S, c-Pr, H, H, H, O], [AC 7635; H, Cl, H, OMe, S, OMe, H, H, H, O], [AC 7636; H, Cl, H, OMe, S, OE t, H, H, H, O], [AC 7637; H, Cl, H, OMe, S, Oi-Pr, H, H, H, O], [AC 7638; H, Cl, H, OMe, S, SMe, H, H, H, O], [AC 7639; H, Cl, H, OMe, S, SE t, H, H, H, O], [AC 7640; H, Cl, H, OMe, S, CH ₂ F, H, H, H, O], [ AC7641; H, Cl, H, OMe, S, CHF 2, H, H, H, O], [AC7642; H, Cl, H, OMe, S, CF 3, H, H, H, O], [ AC7643; H, Cl, H, OMe, S, OCH 2 F, H, H, H, O], [AC7644; H, Cl, H, OMe, S, OCHF 2, H , H, H, O], [AC7645; H, Cl, H, OMe, S, OCF 3, H, H, H, O], [AC7646; H, Cl, H, OMe, S, SCH 2 F, H, H, H, O], [AC7647; H, Cl, H, OMe, S, SCHF ₂ , H, H, H, O], [AC 7648; H, Cl, H, OMe, S, SCF ₃ , H, H, H, O], [AC 7649; H, Cl, H, OMe, S, CN, H, H, H, O], [AC7650; H, Cl, H, OMe, S, NO ₂ , H , H, H, O], [AC7651; H, Cl, H, F, S, H, H, H, H, O], [AC7652; H, Cl, H, F, S, F, H, H , H, O], [AC7653; H, Cl, H, F, S, Cl, H, H, H, O], [AC7654; H, Cl, H, F, S, Br, H, H, H H, Cl, H, F, S, I, H, H, H, O], [AC 7656; H, Cl, H, F, S, Me, H, H, H, O H, Cl, H, F, S, Et, H, H, H, O], [AC 7658; H, Cl, H, F, S, Pr, H, H, H, O], [AC 7659; H, Cl, H, F, S, iP r, H, H, H, O], [AC7660; H, Cl, H, F, S, CH = CH 2, H, H, H, O], [AC7661; H, Cl, H, F, S , C (CH ₃ ) = CH ₂ , H, H, H, O], [AC7662; H, Cl, H, F, S, C≡CH, H, H, H, O], [AC7663; H, Cl, H, F, S, C≡CCH ₃ , H, H, H, O], [AC7664; H, Cl, H, F, S, c-Pr, H, H, H, O], [AC7665 H, Cl, H, F, S, OMe, H, H, H, O], [AC 7666; H, Cl, H, F, S, OEt, H, H, H, O], [AC7667; H , Cl, H, F, S, Oi-Pr, H, H, H, O], [AC7668; H, Cl, H, F, S, SMe, H, H, O], [AC 7669; H , Cl, H, F, S , SEt, H, H, H, O], [AC7670; H, Cl, H, F, S, CH 2 F, H, H, H, O], [AC7671; H , Cl, H, F, S , CHF 2, H, H, H, O], [AC7672; H, Cl, H, F, S, CF 3, H, H, H, O], [AC7673; H , Cl, H, F, S , OCH 2 F, H, H, H, O], [AC7674; H, Cl, H, F, S, OCHF 2, H, H, H, O],

[AC7675; H, Cl, H , F, S, OCF 3, H, H, H, O], [AC7676; H, Cl, H, F, S, SCH 2 F, H, H, H, O] , [AC 7677; H, Cl, H, F, S, SCHF ₂ , H, H, H, O], [AC 7678; H, Cl, H, F, S, SCF ₃ , H, H, H, O] [AC 7679; H, Cl, H, F, S, CN, H, H, H, O], [AC 7680; H, Cl, H, F, S, NO ₂ , H, H, H, O], [AC7681; H, Cl, H, Cl, S, H, H, H, O], [AC7682; H, Cl, H, Cl, S, F, H, H, O], [AC7683 H, Cl, H, Cl, S, Cl, H, H, H, O], [AC7684; H, Cl, H, Cl, S, Br, H, H, O], [AC7685; H , Cl, H, Cl, S, I, H, H, H, O], [AC7686; H, Cl, H, Cl, S, Me, H, H, O], [AC7687; H, Cl H, Cl, S, Et, H, H, H, O], [AC 7688; H, Cl, H, Cl, S, Pr, H, H, H, O], [AC 7689; H, Cl, H , Cl, S, i-Pr , H, H, H, O], [AC7690; H, Cl, H, Cl, S, CH = CH 2, H, H, H, O], [AC7691; H, Cl, H, Cl, S, C (CH 3) = CH 2, H, H, H, O], [AC7692; H, Cl, H, Cl, S, C≡CH, H, H, H, O H, Cl, H, Cl, S, C≡CCH ₃ , H, H, H, O], [AC 7694; H, Cl, H, Cl, S, c-Pr, H, H, H, O], [AC7695; H, Cl, H, Cl, S, OMe, H, H, H, O], [AC7696; H, Cl, H, Cl, S, OEt, H, H, H, H, Cl, H, Cl, S, Oi-Pr, H, H, H, O], [AC 7698; H, Cl, H, Cl, S, SMe, H, H, H, O], [AC 7697; H, Cl, H, Cl, S, SEt, H, H, H, O], [AC 7700; H, Cl, H, Cl, S, CH ₂ F, H, H, H, O], [AC 7699; O], [AC7701; H, Cl, H, Cl, S, CHF 2, H, H, H, O], [AC7702; H, Cl, H, Cl, S, CF 3, H, H, H, O], [AC 7703; H, Cl, H, Cl, S, OCH ₂ F, H, H, H, O], [AC 7704; H, Cl, H, Cl, S, OCHF 2, H, H, H, O], [AC7705; H, Cl, H, Cl, S, OCF 3, H, H, H, O], [ AC 7706; H, Cl, H, Cl, S, SCH ₂ F, H, H, H, O], [AC 7707; H, Cl, H, Cl, S, SCHF ₂ , H, H, H, O], [AC7708; H, Cl, H , Cl, S, SCF 3, H, H, H, O], [AC7709; H, Cl, H, Cl, S, CN, H, H, H, O], [ AC 7710; H, Cl, H, Cl, S, NO ₂ , H, H, H, O], [AC 7711; H, Cl, H, Br, S, H, H, H, H, O], [AC 7712 H, Cl, H, Br, S, F, H, H, H, O], [AC 7713; H, Cl, H, Br, S, Cl, H, H, H, O], [AC 7714; H , Cl, H, Br, S, Br, H, H, H, O], [AC 7715; H, Cl, H, Br, S, I, H, H, O], [AC 7716; H, Cl , H, Br, S, Me, H, H, H, O], [AC 7717; H, Cl, H, Br, S, Et, H, H, H, O], [AC 7718; H, Cl, H , Br, S, Pr, H, H, H, O], [AC 7719; H, Cl, H, Br, S, i-Pr, H, H, H, O], [AC 7720; H, Cl, H , Br, S, CH = CH 2, H, H, H, O], [AC7721; H, Cl, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC 7222; H, Cl, H, Br, S, C≡CH, H, H, H, O], [AC 7723; H, Cl, H, Br, S, C≡ CCH ₃ , H, H, H, O], [AC 7724; H, Cl, H, Br, S, c-Pr, H, H, H, O], [AC 7725; H, Cl, H, Br, S, OMe, H, H, H, H, Cl, H, Br, S, OEt, H, H, H, O], [AC 7727; H, Cl, H, Br, S, Oi-Pr, H, H, H, O], [AC 7726; O, [AC 7728; H, Cl, H, Br, S, SMe, H, H, H, O], [AC 7729; H, Cl, H, Br, S, SE t, H, H, H, O] , [AC7730; H, Cl, H, Br, S, CH 2 F, H, H, H, O], [AC7731; H, Cl, H, Br, S, CHF 2, H, H, H, O ], [AC7732; H, Cl , H, Br, S, CF 3, H, H, H, O], [AC7733; H, Cl, H , Br, S, OCH 2 F, H, H, H, O], [AC7734; H, Cl, H, Br, S, OCHF 2, H, H, H, O] , [AC7735; H, Cl, H, Br, S, OCF 3, H, H, H, O], [AC7736; H, Cl, H, Br, S, SCH 2 F, H, H, H, O H, Cl, H, Br, S, SCHF ₂ , H, H, H, O], [AC 7738; H, Cl, H, Br, S, SCF ₃ , H, H, H, O] H, Cl, H, Br, S, CN, H, H, H, O], [AC 7740; H, Cl, H, Br, S, NO ₂ , H, H, H, O] [AC7741; H, Br, H, H, S, H, H, H, H, O], [AC7742; H, Br, H, H, S, F, H, H, H, O], [AC7741; AC7743; H, Br, H, H, S, Cl, H, H, H, O], [AC7744; H, Br, H, H, S, Br, H, H, H, O], [AC7745; H, Br, H, H, S, I, H, H, H, O], [AC7746; H, Br, H, H, S, Me, H, H, O], [AC 7747; H, Br, H, H, S, Et, H, H, H, O], [AC 7748; H, Br, H, H, S, Pr, H, H, O, [AC 7749; H, Br, H, H, S, i- Pr, H, H, H, O], [AC7750; H, Br, H, H, S, CH = CH 2, H, H, H, O], [AC7751; H , Br, H, H, S , C (CH 3) = CH 2, H, H, H, O], [AC7752; H, Br, H, H, S, C≡CH, H, H, H, O, [AC7753; H, Br, H, H, S, C≡CCH ₃ , H, H, H, O], [AC7754; H, Br, H, H, S, c-Pr, H, H , H, O], [AC7755; H, Br, H, H, S, OMe, H, H, H, O], [AC 7756; H, Br, H, H, S, OEt, H, H, H H, Br, H, H, S, Oi-Pr, H, H, H, O], [AC 7758; H, Br, H, H, S, SMe, H, H, H , O], [AC7759; H , Br, H, H, S, SEt, H, H, H, O], [AC7760; H, Br, H, H, S, CH 2 F, H, H, H , O], [AC7761; H , Br, H, H, S, CHF 2, H, H, H, O], [AC7762; H, Br, H, H _{, S, CF 3, H,} H, H, O], [AC7763; H, Br, H, H, S, OCH 2 F, H, H, H, O], [AC7764; H, Br, H, _{H, S, OCHF 2, H} , H, H, O], [AC7765; H, Br, H, H, S, OCF 3, H, H, H, O], [AC7766; H, Br, H, H, S, SCH ₂ F, H, H, H, H, O], [AC 7767; H, Br, H, H, S, SCHF ₂ , H, H, H, O], [AC 7768; H, Br, H _{, H, S, SCF 3,} H, H, H, O], [AC7769; H, Br, H, H, S, CN, H, H, H, O], [AC7770; H, Br, H, _{H, S, NO 2, H} , H, H, O], [AC7771; H, Br, H, Me, S, H, H, H, H, O], [AC7772; H, Br, H, Me , S, F, H, H, H, O], [AC7773; H, Br, H, Me, S, Cl, H, H, H, O], [AC7774; H, Br, H, Me, S , Br, H, H, H, O],

[AC7775; H, Br, H, Me, S, I, H, H, O], [AC7776; H, Br, H, Me, S, Me, H, H, H, O], [AC 7777 H, Br, H, Me, S, Et, H, H, O], [AC7778; H, Br, H, Me, S, Pr, H, H, O], [AC7779; H , Br, H, Me, S , i-Pr, H, H, H, O], [AC7780; H, Br, H, Me, S, CH = CH 2, H, H, H, O], [ AC7781; H, Br, H, Me, S, C (CH 3) = CH 2, H, H, H, O], [AC7782; H, Br, H, Me, S, C≡CH, H, H H, O], [AC 7783; H, Br, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 7784; H, Br, H, Me, S, c-Pr, H, H, H, O], [AC 7785; H, Br, H, Me, S, OMe, H, H, H, O], [AC 7786; H, Br, H, Me, S, OE t, H, H, H, O], [AC 7787; H, Br, H, Me, S, Oi-Pr, H, H, H, O], [AC 7788; H, Br, H, Me, S, S Me, H, H, H, O], [AC 7789; H, Br, H, Me, S, SE t, H, H, H, O], [AC 7790; H, Br, H, Me, S, CH ₂ F, H, H, H, O], [ AC7791; H, Br, H, Me, S, CHF 2, H, H, H, O], [AC7792; H, Br, H, Me, S, CF 3, H, H, H, O], [ AC7793; H, Br, H, Me, S, OCH 2 F, H, H, H, O], [AC7794; H, Br, H, Me, S, OCHF 2, H , H, H, O], [AC7795; H, Br, H, Me, S, OCF 3, H, H, H, O], [AC7796; H, Br, H, Me, S, SCH 2 F, H, H, H, O], [AC 7797; H, Br, H, Me, S, SCHF ₂ , H, H, H, O], [AC 7798; H, Br, H, Me, S, SCF ₃ , H, H, H, O], [AC 7799; H, Br, H, Me, S, CN, H, H, H, O], [AC 7800; H, Br, H, Me, S, NO ₂ , H , H, H, O], [AC7801; H, Br, H, Et, S, H, H, H, H, O], [AC7802; H, Br, H, Et, S, F, H, H , H, O], [AC 7803; H, Br, H, Et, S, Cl, H H, H, O], [AC 7804; H, Br, H, Et, S, Br, H, H, H, O], [AC 7805; H, Br, H, Et, S, I, H, H H, O], [AC 7806; H, Br, H, Et, S, Me, H, H, H, O], [AC 7807; H, Br, H, Et, S, Et, H, H, H H, Br, H, Et, S, Pr, H, H, H, O], [AC 7809; H, Br, H, Et, S, i-Pr, H, H, H , O], [AC7810; H , Br, H, Et, S, CH = CH 2, H, H, H, O], [AC7811; H, Br, H, Et, S, C (CH 3) = _{CH 2, H, H, H} , O], [AC7812; H, Br, H, Et, S, C≡CH, H, H, H, O], [AC7813; H, Br, H, Et, S _{, C≡CCH 3, H, H,} H, O], [AC7814; H, Br, H, Et, S, c-Pr, H, H, H, O], [AC7815; H, Br, H, Et, S, OMe, H, H, H, O], [AC 7816; H, Br, H, Et, S, OEt, H, H, H, O], [AC 7817; H, Br, H, Et, S, Oi-Pr, H, H, H, O], [AC 7818; H, Br, H, Et, S, SMe, H, H, H, O], [AC 7819; H, Br, H, Et, S, SEt, H, H, H, O], [AC 7820; H, Br, H, Et, S, CH ₂ F, H, H, H, O], [AC 7821; H, Br, H, Et, _{S, CHF 2, H, H} , H, O], [AC7822; H, Br, H, Et, S, CF 3, H, H, H, O], [AC7823; H, Br, H, Et, _{S, OCH 2 F, H,} H, H, O], [AC7824; H, Br, H, Et, S, OCHF 2, H, H, H, O], [AC7825; H, Br, H, Et _{, S, OCF 3, H,} H, H, O], [AC7826; H, Br, H, Et, S, SCH 2 F, H, H, H, O], [AC7827; H, Br, H, _{Et, S, SCHF 2, H} , H, H, O], [AC7828; H, Br, H, Et, S, SCF 3, H, H, H, O], [AC7829; H, Br, H, Et, S, CN, H, H, H, H, O], [AC7830; H, Br, H, Et, S, NO ₂ , H, H, H, O], [AC 7831; H, Br, H, Pr , S, H, H, H, H, O], [AC7832; H, Br, H, Pr, S, F, H, H, H, O, [AC7833; H, Br, H, Pr, S, Cl, H, H, H, O], [AC 7834; H, Br, H, Pr, S, Br, H, H, H, O], [AC 7835; H, Br, H, Pr, S, I, H, H, O], [AC 7836; H, Br, H, Pr, S, Me, H, H, H, O], [AC 7837; H, Br, H, Pr, S, Et, H, H, H, O], [AC 7838; H, Br, H, Pr, S, Pr, H, H, H, O], [AC 7839; H, Br, H, Pr, S, i-Pr, H, H, H, O], [AC 7840; H, Br, H, Pr, S, CH = _{CH 2, H, H, H} , O], [AC7841; H, Br, H, Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC7842; H, Br, H, Pr, S, C≡CH, H, H, H, O], [AC7843; H, Br, H, Pr, S, C≡CCH 3, H, H, H, O], [AC7844; H , Br, H, Pr, S, c-Pr, H, H, H, O], [AC 7845; H, Br, H, Pr, S, OMe, H, H, O], [AC 7846; H , Br, H, Pr, S, OEt, H, H, H, O], [AC7847; H, Br, H, Pr, S, Oi-Pr, H, H, H, O], [AC 7848; H , Br, H, Pr, S, SMe, H, H, H, O], [AC 7849; H, Br, H, Pr, S, SE t, H, H, H, O], [AC 7850; H, Br , H, Pr, S, CH 2 F, H, H, H, O], [AC7851; H, Br, H, Pr, S, CHF 2, H, H, H, O], [AC7852; H, Br, H, Pr, S, CF 3, H, H, H, O], [AC7853; H, Br, H, Pr, S, OCH 2 F, H, H, H, O], [AC7854; H , Br, H, Pr, S , OCHF 2, H, H, H, O], [AC7855; H, Br, H, Pr, S, OCF 3, H, H, H, O], [AC7856; H , Br, H, Pr, S, SCH ₂ F, H, H, H, O], [AC7857; H, Br, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 7858; H, Br, H, Pr, S, SCF 3, H, H, H, O], [AC7859; H, Br, H, Pr, S, CN, H, H, H, O], [AC7860; H , Br, H, Pr, S , NO 2, H, H, H, O], [AC786 1; H, Br, H, i-Pr, S, H, H, H, H, O], [AC7862; H, Br, H, i-Pr, S, F, H, H, H, O] [AC7863; H, Br, H, i-Pr, S, Cl, H, H, H, O], [AC7864; H, Br, H, i-Pr, S, Br, H, H, H, O], [AC7865; H, Br, H, i-Pr, S, I, H, H, O], [AC 7866; H, Br, H, i-Pr, S, Me, H, H, H, O], [AC7867; H, Br, H, i-Pr, S, Et, H, H, H, O], [AC 7868; H, Br, H, i-Pr, S, Pr, H, H, H, O], [AC 7869; H, Br, H, i-Pr, S, i-Pr, H, H, H, O], [AC 7870; H, Br, H, i-Pr, S, _{CH = CH 2, H, H} , H, O], [AC7871; H, Br, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC7872; H, Br, H, i-Pr, S, C≡CH, H, H, H, O], [AC 7873; H, Br, H, i-Pr, S, C≡CCH ₃ , H, H, H , O],

[AC 7874; H, Br, H, i-Pr, S, c-Pr, H, H, H, O], [AC 7875; H, Br, H, i-Pr, S, OMe, H, H, H H, Br, H, i-Pr, S, OEt, H, H, H, O], [AC 7877; H, Br, H, i-Pr, S, Oi-Pr, H H, H, O], [AC7878; H, Br, H, i-Pr, S, SMe, H, H, H, O], [AC7879; H, Br, H, i-Pr, S, SEt , H, H, H, O ], [AC7880; H, Br, H, i-Pr, S, CH 2 F, H, H, H, O], [AC7881; H, Br, H, i-Pr _{, S, CHF 2, H,} H, H, O], [AC7882; H, Br, H, i-Pr, S, CF 3, H, H, H, O], [AC7883; H, Br, H , i-Pr, S, OCH ₂ F, H, H, H, O], [AC 7884; H, Br, H, i-Pr, S, OCHF ₂ , H, H, H, O], [AC 7885; H, Br, H, i- Pr, S, OCF 3, H, H, H, O], [AC7886; H, Br, H, i-Pr, S, SCH 2 F, H, H, H, O H, Br, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 7888; H, Br, H, i-Pr, S, SCF ₃ , H, H] H, O], [AC7889; H, Br, H, i-Pr, S, CN, H, H, H, O], [AC7890; H, Br, H, i-Pr, S, NO ₂ , H, H, H, O], [AC 7891; H, Br, H, c-Pr, S, H, H, H, H, O], [AC 7892; H, Br, H, c-Pr, S, F, H, H, H, O], [AC 7893; H, Br, H, c-Pr, S, Cl, H, H, H, O], [AC 7894; H, Br, H, c-Pr, S, Br, H, H, H, O], [AC 7895; H, Br, H, c-Pr, S, I, H, H, H, O], [AC 7896; H, Br, H, c- Pr, S, Me, H, H, H, O], [AC 7897; H, Br, H, c-Pr, S, Et, H, H, H, O], [AC 7898; H, Br, H, c-Pr, S, Pr, H, H, H, O, [AC 7899; H, Br, H, c-Pr, S, i-Pr, H, H, O], [AC 7900; H, Br, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC7901; H, Br, H, c-Pr, S, C (CH _{3) = CH 2, H,} H, H, O], [AC7902; H, Br, H, c-Pr, S, C≡CH, H, H, H, O], [AC7903; H, Br, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC7904; H, Br, H, c-Pr, S, c-Pr, H, H, H, O], [AC 7905; H, Br, H, c-Pr, S, OMe, H, H, H, O], [AC 7906; H, Br, H, c-Pr, S, OEt, H, H, H, O H, Br, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 7908; H, Br, H, c-Pr, S, SMe, H, H] , H, O], [AC 7909; H, Br, H, c-Pr, S, SEt, H, H, H, O], [AC 7910; H, Br, H, c-Pr, S, CH ₂ F , H, H, H, O ], [AC7911; H, Br, H, c-Pr, S, CHF 2, H, H, H, O], [AC7912; H, Br, H, c-Pr, _{S, CF 3, H, H} , H, O], [AC7913; H, Br, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC7914; H, Br, H , c-Pr, S, OCHF 2, H, H, H, O], [AC7915; H, Br, H, c-Pr, S, OCF 3, H, H, H, O], [AC7916; H , Br, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC7917; H, Br, H, c-Pr, S, SCHF ₂ , H, H, H, O] , [AC7918; H, Br, H, c-Pr, S, SCF 3, H, H, H, O], [AC7919; H, Br, H, c-Pr, S, CN, H, H, H , O], [AC7920; H , Br, H, c-Pr, S, NO 2, H, H, H, O], [AC7921; H, Br, H, SMe, S, H, H, H, H, O], [AC7922; H, Br, H, SMe, S, F, H, H, H, O], [AC7923; H, Br, H, SMe, S, Cl, H, H, H, O], [AC7924; H, Br, H, SMe, S, Br, H, H, H, O], [AC7925; H, Br, H, SMe, S, I, H, H, H, O] , [AC7926; H, Br, H, SMe, S, Me, H, H, H, O], [AC7927; H, Br, H, SMe, S, Et, H, H, H, O], [AC7927; AC7928; H, Br, H, SMe, S, Pr, H, H, H, O], [AC7929; H, Br, H, SMe, S, i-Pr, H, H, H, O], [AC7930; H, Br, H, SMe, S, CH = CH 2, H, H, H, O], [AC7931 ; H, Br, H, SMe , S, C (CH 3) = CH 2, H, H, H, O], [AC7932; H, Br, H, SMe, S, C≡CH, H, H, H, O], [AC7933; H, Br, H, SMe, S, C≡CCH ₃ , H, H, H, O], [AC7934; H, Br, H, SMe, S, c-Pr, H , H, H, O], [AC7935; H, Br, H, SMe, S, OMe, H, H, H, O], [AC7936; H, Br, H, SMe, S, OEt, H, H , H, O], [AC7937; H, Br, H, SMe, S, Oi-Pr, H, H, H, O], [AC7938; H, Br, H, SMe, S, SMe, H, H , H, O], [AC 7939; H, Br, H, SMe, S, SEt, H, H, H, O], [AC7940; H, Br, H, SMe, S, CH ₂ F, H, H , H, O], [AC7941 ; H, Br, H, SMe, S, CHF 2, H, H, H, O], [AC7942; H, Br, H, SMe, S, CF 3, H, H , H, O], [AC 794 3; H, Br, H, S Me, S, OCH ₂ F, H, H, H, O], [AC 7944; H, Br, H, S Me, S, OC H ₂ , H, H, H, O], [ AC7945; H, Br, H, SMe, S, OCF 3, H, H, H, O], [AC7946; H, Br, H, SMe, S, SCH 2 F, H H, H, O], [AC7947; H, Br, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 7948; H, Br, H, SMe, S, SCF ₃ , H , H, H, O], [AC7949; H, Br, H, SMe, S, CN, H, H, H, O], [AC7950; H, Br, H, SMe, S, NO 2, H, H, H, O], [AC 7951; H, Br, H, OMe, S, H, H, H, H, O], [AC 7952; H, Br, H, OMe, S, F, H, H, H, O], [AC7953; H, Br, H, OMe, S, Cl, H, H, H, O], [AC 7954; H, Br, H, OMe, S, Br, H, H, H, O], [AC7955; H, Br, H, OMe, S, I, H, H, H, O], [AC 7956; H, Br, H, OMe, S, Me, H, H, H, O] , [AC795 7; H, Br, H, OMe, S, Et, H, H, H, O], [AC7958; H, Br, H, OMe, S, Pr, H, H, H, O], [AC7959; H, Br, H, OMe, S, i-Pr, H, H, H, O], [AC7960; H, Br, H, OMe, S, CH = CH 2, H, H, H, O], [AC7961; H, Br, H , OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC7962; H, Br, H, OMe, S, C≡CH, H, H, H, O], [AC 7963; H, Br, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC 7964; H, Br, H, OMe, S, c-Pr H, H, H, O], [AC7965; H, Br, H, OMe, S, OMe, H, H, H, O], [AC 7966; H, Br, H, OMe, S, OEt, H , H, H, O], [AC 7967; H, Br, H, OMe, S, Oi-Pr, H, H, H, O], [AC 7968; H, Br, H, OMe, S, SMe, H , H, H, O], [AC 7969; H, Br, H, OMe, S, SE t, H, H, H, O], [AC 7970; H, Br, H, OMe, S, CH ₂ F, H , H, H, O], [AC7971; H, Br, H, OMe, S, CHF 2, H, H, H, O], [AC7972; H, Br, H, OMe, S, CF 3, H , H, H, O], [AC7973; H, Br, H, OMe, S, OCH 2 F, H, H, H, O],

[AC7974; H, Br, H , OMe, S, OCHF 2, H, H, H, O], [AC7975; H, Br, H, OMe, S, OCF 3, H, H, H, O], [AC7976; H, Br, H, OMe, S, SCH ₂ F, H, H, H, O], [AC 7977; H, Br, H, OMe, S, SCHF ₂ , H, H, H, O] , [AC7978; H, Br, H, OMe, S, SCF 3, H, H, H, O], [AC7979; H, Br, H, OMe, S, CN, H, H, H, O], [AC 7980; H, Br, H, OMe, S, NO ₂ , H, H, H, O], [AC 7981; H, Br, H, F, S, H, H, H, O], [AC 7980; AC 7982; H, Br, H, F, S, F, H, H, O], [AC 7983; H, Br, H, F, S, Cl, H, H, H, O], [AC 7984; H, Br, H, F, S, Br, H, H, H, O], [AC 7985; H, Br, H, F, S, I, H, H, O], [AC 7986; H, Br, H, F, S, Me, H, H, H, O], [AC 7987; H, Br, H, F, S, Et, H, H, O], [AC 7988; H, Br, H, F, S, Pr, H, H, H, O, [AC 7989; H, Br, H, F, S, i-Pr, H, H, H, O], [AC7990; H, Br, H, F, S, CH = CH 2, H, H, H, O], [AC7991; H, Br, H, F, S, C (CH 3) = CH 2, H, H, H, O] , [AC7992; H, Br, H, F, S, C≡CH, H, H, H, O], [AC7993; H, Br, H, F, S, C≡ CCH ₃ , H, H, H H, Br, H, F, S, c-Pr, H, H, H, O], [AC7995; H, Br, H, F, S, OMe, H, H, H H, Br, H, F, S, OEt, H, H, H, O], [AC7997; H, Br, H, F, S, Oi-Pr, H, H, H H, Br, H, F, S, SMe, H, H, H, O], [AC 7999; H, Br, H, F, S, SE t, H, H, H, O ], [AC8000; H, Br , H, F, S, CH 2 F, H, H, H, O], [AC8001; H, Br, H, F, S, CHF 2, H, H, H, O], [AC 8002; H, Br, H, F, S, CF ₃ , H, H, H, O], [AC 8003; H, Br , H, F, S, OCH 2 F, H, H, H, O], [AC8004; H, Br, H, F, S, OCHF 2, H, H, H, O], [AC8005; H, Br, H, F, S, OCF 3, H, H, H, O], [AC8006; H, Br, H, F, S, SCH 2 F, H, H, H, O], [AC8007; H , Br, H, F, S, SCHF ₂ , H, H, H, O], [AC 8008; H, Br, H, F, S, SCF ₃ , H, H, O], [AC 8009; H , Br, H, F, S, CN, H, H, H, O], [AC 8010; H, Br, H, F, S, NO ₂ , H, H, H, O], [AC 8011; H, Br, H, Cl, S, H, H, H, H, O], [AC8012; H, Br, H, Cl, S, F, H, H, O], [AC8013; H, Br, H, Cl, S, Cl, H, H, H, O, [AC 8014; H, Br, H, Cl, S, Br, H, H, H, O], [AC 8015; H, Br, H, Cl, S, I, H, H, H, O], [AC 8016; H, Br, H, Cl, S, Me, H, H, H, O], [AC 8017; H, Br, H, Cl, S, Et, H, H, H, O], [AC 8018; H, Br, H, Cl, S, Pr, H, H, H, O], [AC 8019; H, Br, H, Cl, S, i-Pr, H, H, H, O], [AC8020; H, Br, H, Cl, S, CH = CH 2, H, H, H, O], [AC8021; H, Br, H, Cl _{, S, C (CH 3)} = CH 2, H, H, H, O], [AC8022; H, Br, H, Cl, S, C≡CH, H, H, H, O], [AC8023; H, Br, H, Cl, S, C≡CCH 3, H, H, H, O], [AC8024; H, Br, H, Cl, S, c-Pr, H, H, H, O], [AC 8025; H, Br, H, Cl, S, OMe, H, H, H, O], [AC 8026; H, Br, H, Cl, S, OEt, H, H, H, O], [AC 8027 H, Br, H, Cl, S, Oi-Pr, H, H, H, O], [AC 8028; H, Br, H, Cl, S, SMe, H, H, H, O], [AC 8029 H, Br, H, Cl, S, SEt, H, H, H, O], [AC 8030; H, Br, H, Cl, S, CH ₂ F, H, H, H, O], [AC 803 1 ; H, Br, H, Cl , S, CHF 2, H, H, H, O], [AC8032; H, Br, H, _{Cl, S, CF 3, H} , H, H, O], [AC8033; H, Br, H, Cl, S, OCH 2 F, H, H, H, O], [AC8034; H, Br, H _{, Cl, S, OCHF 2,} H, H, H, O], [AC8035; H, Br, H, Cl, S, OCF 3, H, H, H, O], [AC8036; H, Br, H , Cl, S, SCH ₂ F, H, H, H, O, [AC 8037; H, Br, H, Cl, S, SCHF ₂ , H, H, H, O], [AC 8038; H, Br, _{H, Cl, S, SCF 3} , H, H, H, O], [AC8039; H, Br, H, Cl, S, CN, H, H, H, O], [AC8040; H, Br, H _{, Cl, S, NO 2,} H, H, H, O], [AC8041; H, Br, H, Br, S, H, H, H, H, O], [AC8042; H, Br, H, Br, S, F, H, H, H, O], [AC 8043; H, Br, H, Br, S, Cl, H, H, H, O], [AC 8044; H, Br, H, Br, S, Br, H, H, H, O], [AC 8045; H, Br, H, Br, S, I, H, H, H, O], [AC 8046; H, Br, H, Br, S, Me, H, H, H, O], [AC 8047; H, Br, H, Br, S, Et, H, H, H, O], [AC 8048; H, Br, H, Br, S, Pr, H, H, H, O], [AC 8049; H, Br, H, Br, S, i-Pr, H, H, H, O], [AC 8050; H, Br, H, Br, S, CH = _{CH 2, H, H, H} , O], [AC8051; H, Br, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC8052; H, Br, H, Br, S, C≡CH, H, H, H, O], [AC 8053; H, Br, H, Br, S, C≡CCH ₃ , H, H, H, O], [AC8054; H , Br, H, Br, S, c-Pr, H, H, H, O], [AC 8055; H, Br, H, Br, S, OMe, H, H, H, O], [AC 8056; H , Br, H, Br, S, OEt, H, H, H, O], [AC 8057; H, Br, H, Br, S, Oi-Pr, H, H, H, O], [AC 8058; H , Br, H, Br, S, SMe, H, H, H, O], [AC 8059; H, Br, H, Br, S, SE, H, H, H, O], [AC 8060; H, Br , H, Br, S, CH 2 F, H, H, H, O], [AC8061; H, B r, H, Br, S, CHF 2, H, H, H, O], [AC8062; H, Br, H, Br, S, CF 3, H, H, H, O], [AC8063; H, Br, H, Br, S, OCH 2 F, H, H, H, O], [AC8064; H, Br, H, Br, S, OCHF 2, H, H, H, O], [AC8065; H , Br, H, Br, S , OCF 3, H, H, H, O], [AC8066; H, Br, H, Br, S, SCH 2 F, H, H, H, O], [AC8067; H, Br, H, Br, S, SCHF 2, H, H, H, O], [AC8068; H, Br, H, Br, S, SCF 3, H, H, H, O], [AC8069; H, Br, H, Br, S, CN, H, H, H, O], [AC 8070; H, Br, H, Br, S, NO ₂ , H, H, H, O], [AC 807 1; H , OMe, H, H, S, H, H, H, H, O], [AC8072; H, OMe, H, H, S, F, H, H, O], [AC8073; H, OMe , H, H, S, Cl, H, H, H, O],

[AC 8074; H, OMe, H, H, S, Br, H, H, H, O], [AC 8075; H, OMe, H, H, S, I, H, H, O], [AC 8076 H, OMe, H, H, S, Me, H, H, H, O], [AC 8077; H, OMe, H, H, S, Et, H, H, O], [AC 8078; H , OMe, H, H, S, Pr, H, H, H, O], [AC 8079; H, OMe, H, H, S, i-Pr, H, H, H, O], [AC 8080; H , OMe, H, H, S , CH = CH 2, H, H, H, O], [AC8081; H, OMe, H, H, S, C (CH 3) = CH 2, H, H, H H, OMe, H, S, C≡CH, H, H, H, O], [AC8083; H, OMe, H, H, S, C≡CCH ₃ , H, H, H, O], [AC8084; H, OMe, H, S, c-Pr, H, H, H, O], [AC8085; H, OMe, H, S, OMe, H, H, H, O], [AC8086; H, OMe, H, S, OEt, H, H, H, O], [AC 8087; H, OMe, H, H, S, Oi-Pr, H, H, H, O], [AC 8088; H, OMe, H, S, SMe, H, H, H, O], [AC 8089; H, OMe, H, H, S, SE t, H, H, H, H, O], [AC8090; H, OMe, H, H, S, CH 2 F, H, H, H, O], [AC8091; H, OMe, H, H, S, CHF 2, H, H , H, O], [AC8092 ; H, OMe, H, H, S, CF 3, H, H, H, O], [AC8093; H, OMe, H, H, S, OCH 2 F, H, H, H, O], [ AC8094; H, OMe, H, H, S, OCHF 2, H, H, H, O], [AC8095; H, OMe, H, H, S, OCF 3, H, H, H, O], [AC 8096; H, OMe, H, H, S, SCH ₂ F, H, H, H, O], [AC 8097; H, OMe, H, H, S, SCHF ₂ , H , H, H, O], [AC 8098; H, OMe, H, H, S, SCF ₃ , H, H, H, O], [AC 8099; H, OMe, H, H, S, CN, H, H, H, O], [AC 8100; H, OMe, H, H, S, NO ₂ , H, H, H, O], [AC 8101; H, OMe, H, Me, S, H, H, H , H, O], [AC 8102; H, OMe, H, Me, S, F , H, H, H, O], [AC 8103; H, OMe, H, Me, S, Cl, H, H, H, O], [AC 8104; H, OMe, H, Me, S, Br, H , H, H, O], [AC 8105; H, OMe, H, Me, S, I, H, H, H, O], [AC 8106; H, OMe, H, Me, S, Me, H, H H, O], [AC 8107; H, OMe, H, Me, S, Et, H, H, H, O], [AC 8108; H, OMe, H, Me, S, Pr, H, H, H , O], [AC 8109; H, OMe, H, Me, S, i-Pr, H, H, H, O], [AC 8110; H, OMe, H, Me, S, CH = CH ₂ , H, H, H, O], [ AC8111; H, OMe, H, Me, S, C (CH 3) = CH 2, H, H, H, O], [AC8112; H, OMe, H, Me, S , COMCH, H, H, H, O, [AC 8113; H, OMe, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 8114; H, OMe, H, Me, S, c-Pr, H, H, H, H, O], [AC 8115; H, OMe, H, Me, S, OMe, H, H, H, O], [AC 8116; H, OMe, H, Me, S, OEt, H, H, H, O], [AC 8117; H, OMe, H, Me, S, Oi-Pr, H, H, H, O], [AC 8118; H, OMe, H, Me, S, SMe, H, H, H, O], [AC 8119; H, OMe, H, Me, S, SE t, H, H, H, O], [AC 8120; H, OMe, H, Me, _{S, CH 2 F, H,} H, H, O], [AC8121; H, OMe, H, Me, S, CHF 2, H, H, H, O], [AC8122; H, OMe, H, Me _{, S, CF 3, H,} H, H, O], [AC8123; H, OMe, H, Me, S, OCH 2 F, H, H, H, O], [AC8124; H, OMe, H, _{Me, S, OCHF 2, H} , H, H, O], [AC8125; H, OMe, H, Me, S, OCF 3, H, H, H, O], [AC8126; H, OMe, H, _{Me, S, SCH 2 F,} H, H, H, O], [AC8127; H, OMe, H, Me, S, SCHF 2, H, H, H, O], [AC8128; H, OMe, H _{, Me, S, SCF 3,} H, H, H, O], [AC8129; H, OMe, H, Me, S, CN, H, H, H, O], [AC8130; H, OMe, H, Me, S , NO ₂ , H, H, H, O], [AC8131; H, OMe, H, Et, S, H, H, H, H, O], [AC8132; H, OMe, H, Et, S, H, OMe, H, Et, S, Cl, H, H, O], [AC 8134; H, OMe, H, Et, S, Br, F, H, H, H, O], [AC 8133; H, H, H, O], [AC 8135; H, OMe, H, Et, S, I, H, H, H, O], [AC 8136; H, OMe, H, Et, S, Me, H, H, H, O], [AC 8137; H, OMe, H, Et, S, Et, H, H, H, O], [AC 8138; H, OMe, H, Et, S, Pr, H, H, H, O], [AC 8139; H, OMe, H, Et, S, i-Pr, H, H, H, O], [AC 8140; H, OMe, H, Et, S, CH = CH ₂ , H , H, H, O], [AC8141; H, OMe, H, Et, S, C (CH 3) = CH 2, H, H, H, O], [AC8142; H, OMe, H, Et, S, C≡CH, H, H, H, H, O], [AC 8143; H, OMe, H, Et, S, C≡CCH ₃ , H, H, H, O], [AC 8144; H, OMe, H , Et, S, c-Pr, H, H, H, O], [AC 8145; H, OMe, H, Et, S, OMe, H, H, H, O], [AC 8146; H, OMe, H , Et, S, OEt, H, H, H, O], [AC 8147; H, OMe, H, Et, S, Oi-Pr, H, H, H, O], [AC 8148; H, OMe, H , Et, S, SMe, H, H, H, O], [AC 8149; H, OMe, H, Et, S, SE t, H, H, H, O], [AC 8150; H, OMe, H, Et _{, S, CH 2 F, H} , H, H, O], [AC8151; H, OMe, H, Et, S, CHF 2, H, H, H, O], [AC8152; H, OMe, H, _{Et, S, CF 3, H} , H, H, O], [AC8153; H, OMe, H, Et, S, OCH 2 F, H, H, H, O], [AC8154; H, OMe, H _{, Et, S, OCHF 2,} H, H, H, O], [AC8155; H, OMe, H, Et, S, OCF 3, H, H, H, O], [AC8156; H, OMe, H , Et, S, SCH ₂ F, H, H, H, O], [AC 8157; H, OMe, H, Et, S, SCHF ₂ , H, H, H, O], [AC 8158; H, OMe, H, Et, S , SCF ₃ , H, H, H, O], [AC8159; H, OMe, H, Et, S, CN, H, H, H, O], [AC 8160; H, OMe, H, Et, S, _{NO 2, H, H, H} , O], [AC8161; H, OMe, H, Pr, S, H, H, H, H, O], [AC8162; H, OMe, H, Pr, S, F , H, H, H, O], [AC8163; H, OMe, H, Pr, S, Cl, H, H, H, O], [AC 8164; H, OMe, H, Pr, S, Br, H H, H, O], [AC8165; H, OMe, H, Pr, S, I, H, H, H, O], [AC 8166; H, OMe, H, Pr, S, Me, H, H H, O], [AC 8167; H, OMe, H, Pr, S, Et, H, H, H, O], [AC 8168; H, OMe, H, Pr, S, Pr, H, H, H H, OMe, H, Pr, S, i-Pr, H, H, H, O], [AC 8170; H, OMe, H, Pr, S, CH = CH ₂ , H, H, H, O], [ AC8171; H, OMe, H, Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC8172; H, OMe, H, Pr, S , C≡CH, H, H, H, O],

[AC8173; H, OMe, H, Pr, S, C≡CCH ₃ , H, H, H, O], [AC 8174; H, OMe, H, Pr, S, c-Pr, H, H, H, O, [AC 8175; H, OMe, H, Pr, S, OMe, H, H, H, O], [AC 8176; H, OMe, H, Pr, S, OE t, H, H, H, O] [AC 8177; H, OMe, H, Pr, S, Oi-Pr, H, H, H, O], [AC 8178; H, OMe, H, Pr, S, SMe, H, H, H, O] [AC 8179; H, OMe, H, Pr, S, SEt, H, H, H, O], [AC 8180; H, OMe, H, Pr, S, CH ₂ F, H, H, H, O] , [AC8181; H, OMe, H, Pr, S, CHF 2, H, H, H, O], [AC8182; H, OMe, H, Pr, S, CF 3, H, H, H, O] , [AC8183; H, OMe, H, Pr, S, OCH 2 F, H, H, H, O], [AC8184; H, OMe, H, Pr, S, OCHF 2, H, H, H, O ], [AC8185; H, OMe , H, Pr, S, OCF 3, H, H, H, O], [AC8186; H, OMe, H, Pr, S, SCH 2 F, H, H, H, O, [AC 8187; H, OMe, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 8188; H, OMe, H, Pr, S, SCF ₃ , H, H, H, O, [AC 8189; H, OMe, H, Pr, S, CN, H, H, H, O], [AC 8190; H, OMe, H, Pr, S, NO ₂ , H, H, H, O H, OMe, H, i-Pr, S, H, H, H, O], [AC8192; H, OMe, H, i-Pr, S, F, H, H, H] , O], [AC 8193; H, OMe, H, i-Pr, S, Cl, H, H, H, O], [AC 8194; H, OMe, H, i-Pr, S, Br, H, H H, O], [AC 8195; H, OMe, H, i-Pr, S, I, H, H, H, O], [AC 8196; H, OMe, H, i-Pr, S, Me, H H, H, O], [AC 8197; H, OMe, H, i-Pr, S, Et, H, H, H, O], [AC 8198; H, OMe, H, i-Pr, S, Pr H, H, H, O], [AC 8199; H, OMe, H, i-Pr, S, i-Pr, H, H, H, O], [AC 8200; H, OMe, H, i-Pr , S, CH = CH ₂ , H , H, H, O], [AC8201; H, OMe, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC8202; H, OMe, H, i-Pr, S, C≡CH, H, H, H, O], [AC 8203; H, OMe, H, i-Pr, S, C≡ CCH ₃ , H, H, H, O], [AC 8204 H, OMe, H, i-Pr, S, c-Pr, H, H, H, O], [AC 8205; H, OMe, H, i-Pr, S, OMe, H, H, H, O H, OMe, H, i-Pr, S, OEt, H, H, H, O], [AC 8207; H, OMe, H, i-Pr, S, Oi-Pr, H, H] , H, O], [AC 8208; H, OMe, H, i-Pr, S, SMe, H, H, H, O], [AC 8209; H, OMe, H, i-Pr, S, SEt, H , H, H, O], [AC8210; H, OMe, H, i-Pr, S, CH 2 F, H, H, H, O], [AC8211; H, OMe, H, i-Pr, S , CHF ₂ , H, H, H, O], [AC 8212; H, OMe, H, i-Pr, S, CF ₃ , H, H, O], [AC 8213; H, OMe, H, i _{-Pr, S, OCH 2 F,} H, H, H, O], [AC8214; H, OMe, H, i-Pr, S, OCHF 2, H, H, H, O], [AC8215; H, OMe, H, i-Pr, S, OCF 3, H, H, H, O], [AC8216; H, OMe, H, i-Pr, S, SCH 2 F, H, H, H, O], [AC 8217; H, OMe, H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 8218; H, OMe, H, i-Pr, S, SCF ₃ , H, H, H H, OMe, H, i-Pr, S, CN, H, H, H, O], [AC 8220; H, OMe, H, i-Pr, S, NO ₂ , H, H, H, O], [AC8221; H, OMe, H, c-Pr, S, H, H, H, H, O], [AC8222; H, OMe, H, c-Pr, S, F, H, H, H, O], [AC8223; H, OMe, H, c-Pr, S, Cl, H, H, H] O, [AC8224; H, OMe, H, c-Pr, S, Br, H, H, H, O], [AC 8225; H, OMe, H, c-Pr, S, I, H, H, H, O], [AC 8226; H, OMe, H, c-Pr, S, Me, H, H, H, O], [AC 8227; H, OMe, H, c-Pr, S, Et, H, H, H, O], [AC 8228; H, OMe, H, c-Pr, S, Pr, H, H, H, O], [AC 8229; H, OMe, H, c- Pr, S, i-Pr, H, H, H, O], [AC8230; H, OMe, H, c-Pr, S, CH = CH 2, H, H, H , O], [AC8231; H , OMe, H, c-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC8232; H, OMe, H, c-Pr, S, C≡CH, H, H, H, O], [AC8233; H, OMe, H, c-Pr, S, C≡CCH ₃ , H, H, H, O], [AC8234; H, OMe , H, c-Pr, S, c-Pr, H, H, H, O], [AC 8235; H, OMe, H, c-Pr, S, OMe, H, H, H, O], [AC 8236 H, OMe, H, c-Pr, S, OEt, H, H, H, O], [AC 8237; H, OMe, H, c-Pr, S, Oi-Pr, H, H, H, O H, OMe, H, c-Pr, S, SMe, H, H, H, O], [AC 8239; H, OMe, H, c-Pr, S, SEt, H, H, H] , O], [AC8240; H , OMe, H, c-Pr, S, CH 2 F, H, H, H, O], [AC8241; H, OMe, H, c-Pr, S, CHF 2, H, H, H, O] , [AC8242; H, OMe, H, c-Pr, S, CF 3, H, H, H, O], [AC8243; H, OMe, H, c-Pr, S , OCH ₂ F, H, H, H, O], [AC8244; H, OMe, H, c-Pr, S, OCHF ₂ , H, H, H, O], [AC8245; H, OMe, H, _{c-Pr, S, OCF 3} , H, H, H, O], [AC8246; H, OMe, H, c-Pr, S, SCH 2 F, H, H, H, O], [AC8247; H , OMe, H, c-Pr, S, SCHF ₂ , H, H, H, O], [AC 8248; H, OMe, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 8249; H, OMe, H, c-Pr, S, CN, H, H, H, O], [AC 8250; H, OMe, H, c-Pr, S, NO ₂ , H, H, H, O], [AC 8251; H, OMe, H, SMe, S, H, H, H, H, O], [AC 8252; H, OMe, H, SMe, S, F, H, H, H, O] , [AC 8253; H, OMe, H, SMe, S , Cl, H, H, H, O], [AC 8254; H, OMe, H, SMe, S, Br, H, H, H, O], [AC 8255; H, OMe, H, SMe, S, I H, H, H, O], [AC 8256; H, OMe, H, SMe, S, Me, H, H, H, O], [AC 8257; H, OMe, H, SMe, S, Et, H , H, H, O], [AC8258; H, OMe, H, SMe, S, Pr, H, H, H, O], [AC 8259; H, OMe, H, SMe, S, i-Pr, H H, H, O], [AC 8260; H, OMe, H, SMe, S, CH = CH ₂ , H, H, H, O], [AC 8261; H, OMe, H, SMe, S, C ( CH ₃ ) = CH ₂ , H, H, H, O], [AC 8262; H, OMe, H, SMe, S, C≡CH, H, H, H, O], [AC 8263; H, OMe, H , SMe, S, C≡CCH ₃ , H, H, H, O], [AC 8 264; H, OMe, H, SMe, S, c-Pr, H, H, H, O], [AC 8 265; H, OMe, H, SMe, S, OMe, H, H, H, O], [AC 8266; H, OMe, H, SMe, S, OEt, H, H, H, O], [AC 8267; H, OMe, H, SMe, S, Oi-Pr, H, H, H, O], [AC 8268; H, OMe, H, SMe, S, SMe, H, H, H, O], [AC 8269; H, OMe, H, SMe, S, SEt, H, H, H, O], [AC8270; H, OMe, H, SMe, S, CH 2 F, H, H, H, O], [AC8271; H, OMe, _{H, SMe, S, CHF 2} , H, H, H, O], [AC8272; H, OMe, H, SMe, S, CF 3, H, H, H, O],

[AC8273; H, OMe, H , SMe, S, OCH 2 F, H, H, H, O], [AC8274; H, OMe, H, SMe, S, OCHF 2, H, H, H, O] , [AC8275; H, OMe, H, SMe, S, OCF 3, H, H, H, O], [AC8276; H, OMe, H, SMe, S, SCH 2 F, H, H, H, O H, OMe, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 8278; H, OMe, H, SMe, S, SCF ₃ , H, H, H, O] H, OMe, H, SMe, S, CN, H, H, H, O], [AC 8280; H, OMe, H, SMe, S, NO ₂ , H, H, H, O] [AC8281; H, OMe, H, OMe, S, H, H, H, H, O], [AC8282; H, OMe, H, OMe, S, F, H, H, H, O], [AC8282; AC 8283; H, OMe, H, OMe, S, Cl, H, H, H, O], [AC 8284; H, OMe, H, OMe, S, Br, H, H, O], [AC 8285; H, OMe, H, OMe, S, I, H, H, H, O], [AC 8286; H, OMe, H, OMe, S, Me, H, H, O], [AC 8287; H, OMe, H, OMe, S, Et, H, H, H, O], [AC 8288; H, OMe, H, OMe, S, Pr, H, H, H, O], [AC 8289; H, OMe, H, OMe, S, i-Pr, H, H, H, O], [AC 8290; H, OMe, H, OMe, S, CH = CH ₂ , H, H, H, O], [AC 8291; H , OMe, H, OMe, S , C (CH 3) = CH 2, H, H, H, O], [AC8292; H, OMe, H, OMe, S, C≡CH, H, H, H, O, [AC 8293; H, OMe, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC 8294; H, OMe, H, OMe, S, c-Pr, H, H H, O], [AC 8295; H, OMe, H, OMe, S, OMe, H, H, H, O], [AC 8296; H, OMe, H, OMe, S, OEt, H, H, H , O], [AC 8297; H, OMe, H, OMe, S, Oi-Pr, H, H, H, O], [AC 8298; H, OMe, H, OMe, S, SMe, H, H, H , O], [AC 8299; H, OMe, H, OMe, S, SE t, H, H, H, O], [AC 8300; H, OMe , H, OMe, S, CH 2 F, H, H, H, O], [AC8301; H, OMe, H, OMe, S, CHF 2, H, H, H, O], [AC8302; H, OMe, H, OMe, S, CF 3, H, H, H, O], [AC8303; H, OMe, H, OMe, S, OCH 2 F, H, H, H, O], [AC8304; H , OMe, H, OMe, S , OCHF 2, H, H, H, O], [AC8305; H, OMe, H, OMe, S, OCF 3, H, H, H, O], [AC8306; H , OMe, H, OMe, S, SCH ₂ F, H, H, H, O], [AC 8307; H, OMe, H, OMe, S, SCHF ₂ , H, H, H, O], [AC 8308; H, OMe, H, OMe, S, SCF 3, H, H, H, O], [AC8309; H, OMe, H, OMe, S, CN, H, H, H, O], [AC8310; H , OMe, H, OMe, S, NO ₂ , H, H, H, O], [AC 8311; H, OMe, H, F, S, H, H, H, O], [AC 8312; H, OMe, H, F, S, F, H, H, H, O], [AC 8313; H, OMe, H, F, S, Cl, H, H, O], [AC 8314; H, OMe, H, F, S, Br, H, H, H, O], [AC8315; H, OMe, H, F, S, I, H, H, O], [AC 8316; H, OMe, H, F, S, Me, H, H, H, O], [AC 8317; H, OMe, H, F, S, Et, H, H, H, O], [AC 8318; H, OMe, H, F, S, Pr, H, H, H, O], [AC 8319; H, OMe, H, F, S, i-Pr, H, H, H, O], [AC 8320; H, OMe, H, F, _{S, CH = CH 2, H} , H, H, O], [AC8321; H, OMe, H, F, S, C (CH 3) = CH 2, H, H, H, O], [AC8322; H, OMe, H, F, S, C≡CH, H, H, H, O], [AC 8323; H, OMe, H, F, S, C≡ CCH ₃ , H, H, H, O], [AC 8324; H, OMe, H, F, S, c-Pr, H, H, H, O], [AC 8325; H, OMe, H, F, S, OMe, H, H, H, O], [AC 83 26; H, OMe, H, F, S, OEt, H, H, H, O], [AC 8327; H, OMe, H, F, S, Oi-Pr, H, H, H, O], [AC 8328; H, OMe, H, F , S, SMe, H, H, H, O], [AC 8329; H, OMe, H, F, S, SE t, H, H, H, O], [AC 8330; H, OMe, H, F, S _{, CH 2 F, H, H} , H, O], [AC8331; H, OMe, H, F, S, CHF 2, H, H, H, O], [AC8332; H, OMe, H, F, _{S, CF 3, H, H} , H, O], [AC8333; H, OMe, H, F, S, OCH 2 F, H, H, H, O], [AC8334; H, OMe, H, F , S, OCHF ₂ , H, H, H, O], [AC 8335; H, OMe, H, F, S, OCF ₃ , H, H, O], [AC 8336; H, OMe, H, F , S, SCH ₂ F, H, H, H, O], [AC 8337; H, OMe, H, F, S, SCHF ₂ , H, H, H, O], [AC 8338; H, OMe, H, _{F, S, SCF 3, H} , H, H, O], [AC8339; H, OMe, H, F, S, CN, H, H, H, O], [AC8340; H, OMe, H, F , S, NO ₂ , H, H, H, O], [AC8341; H, OMe, H, Cl, S, H, H, H, H, O], [AC8342; H, OMe, H, Cl, S, F, H, H, H, O], [AC8343; H, OMe, H, Cl, S, Cl, H, H, H, O], [AC 8344; H, OMe, H, Cl, S, Br, H, H, H, O], [AC 8345; H, OMe, H, Cl, S, I, H, H, H, O], [AC 8346; H, OMe, H, Cl, S, Me, H, H, H, O], [AC 8347; H, OMe, H, Cl, S, Et, H, H, H, O], [AC 8348; H, OMe, H, Cl, S, Pr, H, H, H, O], [AC 8349; H, OMe, H, Cl, S, i-Pr, H, H, H, O], [AC 8350; H, OMe, H, Cl, S, CH = CH ₂ , H, H, H, O], [AC 8351; H, OMe, H, Cl, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 8352; H, OMe, H, Cl, S, C≡CH, H, H, H, O], [AC8353; H, OMe, H, Cl, S, C≡CCH 3, H, H, H, O], [AC8354; H, OMe , H, Cl, S, c-Pr, H, H, H, O], [AC 8355; H, OMe, H, Cl, S, OMe, H, H, H, O], [AC 8356; H, OMe , H, Cl, S, OEt, H, H, H H, OMe, H, Cl, S, Oi-Pr, H, H, H, O], [AC 8358; H, OMe, H, Cl, S, SMe, H, H, H H, OMe, H, Cl, S, SEt, H, H, H, O], [AC 8360; H, OMe, H, Cl, S, CH ₂ F, H, H, H , O], [AC8361; H , OMe, H, Cl, S, CHF 2, H, H, H, O], [AC8362; H, OMe, H, Cl, S, CF 3, H, H, H , O], [AC8363; H , OMe, H, Cl, S, OCH 2 F, H, H, H, O], [AC8364; H, OMe, H, Cl, S, OCHF 2, H, H, H, O], [AC8365; H, OMe, H, Cl, S, OCF 3, H, H, H, O], [AC8366; H, OMe, H, Cl, S, SCH 2 F, H, H , H, O], [AC 8367; H, OMe, H, Cl, S, SCHF ₂ , H, H, H, O], [AC 8368; H, OMe, H, Cl, S, SCF ₃ , H, H H, O], [AC 8369; H, OMe, H, Cl, S, CN, H, H, H, O], [AC 8370; H, OMe, H, Cl, S, NO ₂ , H, H, H, O], [AC 8371; H, OMe, H, Br, S, H, H, H, H, O], [AC 8372; H, OMe, H, Br, S, F, H, H, H, O],

[AC 8373; H, OMe, H, Br, S, Cl, H, H, H, O], [AC 8374; H, OMe, H, Br, S, Br, H, H, H, O], [AC 8375 H, OMe, H, Br, S, I, H, H, H, O], [AC 8376; H, OMe, H, Br, S, Me, H, H, H, O], [AC 8377; H , OMe, H, Br, S, Et, H, H, H, O], [AC 8378; H, OMe, H, Br, S, Pr, H, H, H, O], [AC 8379; H, OMe , H, Br, S, i -Pr, H, H, H, O], [AC8380; H, OMe, H, Br, S, CH = CH 2, H, H, H, O], [AC8381; H, OMe, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC8382; H, OMe, H, Br, S, C≡CH, H, H, H , O], [AC8383; H, OMe, H, Br, S, C≡CCH ₃ , H, H, H, O], [AC8384; H, OMe, H, Br, S, c-Pr, H, H, H, O], [AC 8385; H, OMe, H, Br, S, OMe, H, H, H, O], [AC 8386; H, OMe, H, Br, S, OE t, H, H, H, H, O], [AC 8387; H, OMe, H, Br, S, Oi-Pr, H, H, H, O], [AC 8388; H, OMe, H, Br, S, SMe, H, H, H, H, O], [AC 8389; H, OMe, H, Br, S, SEt, H, H, H, O], [AC 8390; H, OMe, H, Br, S, CH ₂ F, H, H, H, O], [AC 8391; H, OMe, H, Br, S, CHF ₂ , H, H, H, O], [AC 8392; H, OMe, H, Br, S, CF ₃ , H, H, H, O], [AC 8393; H, OMe, H, Br, S, OCH ₂ F, H, H, H, O], [AC 8394; H, OMe, H, Br, S, OCF ₂ , H, H , H, O], [AC8395 ; H, OMe, H, Br, S, OCF 3, H, H, H, O], [AC8396; H, OMe, H, Br, S, SCH 2 F, H, H, H, O], [AC 8397; H, OMe, H, Br, S, SCHF ₂ , H, H, H, O], [AC 8398; H, OMe, H, Br, S, SCF ₃ , H, H, H, O], [AC 8399; H, OMe, H, Br, S, CN, H, H, H, O], [AC 8400; H, OMe, H, Br, S, NO ₂ , H, H , H, O], [AC8401; H, OEt, H, H, S, H, H, H, H, O], [AC8402; H, OEt, H, H, S, F, H, H, H] , O], [AC 8403; H, OEt, H, H, S, Cl, H, H, H] O, [AC 8404; H, OEt, H, H, S, Br, H, H, H, O , [AC 8405; H, OEt, H, H, S, I, H, H, H, O], [AC 8406; H, OEt, H, H, S, Me, H, H, H, O], [AC 8407; H, OEt, H, H, S, Et, H, H, H, O], [AC 8408; H, OEt, H, H, S, Pr, H, H, H, O], [AC 8409 ; H, OEt, H, H , S, i-Pr, H, H, H, O], [AC8410; H, OEt, H, H, S, CH = CH 2, H, H, H, O] , [AC8411; H, OEt, H, H, S, C (CH 3) = CH 2, H, H, H, O], [AC8412; H, OEt, H, H, S, C≡CH, H , H, H, O], [AC 8413; H, OEt, H, H, S, C≡CCH ₃ , H, H, H, O], [AC 8414; H, OE t, H, H, S, c- Pr, H, H, H, O], [AC 8415; H, OEt, H, H, S, OMe, H, H, H, O], [AC 8416; H, OE t, H, H, S, OE t, H, H, H, O], [AC 8417; H, OEt, H, H, S, Oi-Pr, H, H, H, O], [AC 8418; H, OEt, H, H, S, SMe, H, H, H, O], [AC 8419; H, OEt, H, H, S, SE t, H, H, H, O], [AC 8420; H, OE t, H, H, S, CH ₂ F, H, H, H, O] , [AC8421; H, OEt, H, H, S, CHF 2, H, H, H, O], [AC8422; H, OEt, H, H, S, CF 3, H, H, H, O] , [AC8423; H, OEt, H, H, S, OCH 2 F, H, H, H, O], [AC8424; H, OEt, H, H, S, OCHF 2 , H, H, H, O ], [AC8425; H, OEt, H, H, S, OCF 3, H, H, H, O], [AC8426; H, OEt, H, H, S, SCH 2 F, H, H, H, O], [AC 8427; H, OEt, H, H, S, SCHF ₂ , H, H, H, O], [AC 8428; H, OE t, H, H, S, SCF ₃ , H, H, H, O], [AC 8429; H, OEt, H, H, S, C N, H, H, H, O], [AC 8430; H, OEt, H, H, S, NO ₂ , H, H, H, O], [AC8431; H, OE t, H, Me, S, H] , H, H, H, O], [AC8432; H, OEt, H, Me, S, F, H, H, H, O], [AC8433; H, OEt, H, Me, S, Cl, H] H, H, O], [AC8434; H, OEt, H, Me, S, Br, H, H, H, O], [AC 8435; H, OEt, H, Me, S, I, H, H , H, O], [AC 8436; H, OEt, H, Me, S, Me, H, H, H, O], [AC 8437; H, OE t, H, Me, S, Et, H, H, H , O], [AC 8438; H, OEt, H, Me, S, Pr, H, H, H, O], [AC 8439; H, OEt, H, Me, S, i-Pr, H, H, H , O], [AC8440; H , OEt, H, Me, S, CH = CH 2, H, H, H, O], [AC8441; H, OEt, H, Me, S, C (CH 3) = _{CH 2, H, H, H} , O], [AC8442; H, OEt, H, Me, S, C≡CH, H, H, H, O], [AC8443; H, OEt, H, Me, S , C≡CCH ₃ , H, H, H, O], [AC 8444; H, OEt, H, Me, S, c-Pr, H, H, H, O], [AC 8445; H, OE t, H, Me, S, OMe, H, H, H, O], [AC 8446; H, OEt, H, Me, S, OEt, H, H, H, O], [AC 8447; H, OEt, H, Me, S, Oi-Pr, H, H, H, O], [AC8448; H, OEt, H, Me, S, SMe, H, H, H, O], [AC 8449; H, OEt, H, Me, S, SEt, H, H, H, O], [AC8450; H, OEt, H, Me, S, CH 2 F, H, H, H, O], [AC8451; H, OEt, H, Me, _{S, CHF 2, H, H} , H, O], [AC8452; H, OEt, H, Me, S, CF 3, H, H, H, O], [AC8453; H, OEt, H, Me, _{S, OCH 2 F, H,} H, H, O], [AC8454; H, OEt, H, Me, S, OCHF 2, H, H, H, O], [AC8455; H, OEt, H, Me , S, OCF ₃ , H, H, H, O], [AC 8456; H, OEt, H, Me, S, SCH ₂ F, H, H, H, O], [AC 8457; H, OE t, H, Me, S, SCHF ₂ H, H, H, O], [AC 8458; H, OEt, H, Me, S, SCF ₃ , H, H, H, O], [AC 8459; H, OE t, H, Me, S, CN, H, H, H, O], [AC 8460; H, OEt, H, Me, S, NO ₂ , H, H, H, O], [AC 8461; H, OE t, H, Et, S, H, H , H, H, O], [AC8462; H, OEt, H, Et, S, F, H, H, H, O], [AC8463; H, OEt, H, Et, S, Cl, H, H H, O], [AC 8464; H, OEt, H, Et, S, Br, H, H, H, O], [AC 8465; H, OEt, H, Et, S, I, H, H, H H, OEt, H, Et, S, Me, H, H, H, O], [AC 8467; H, OEt, H, Et, S, Et, H, H, H, O H, OEt, H, Et, S, Pr, H, H, H, O], [AC 8469; H, OEt, H, Et, S, i-Pr, H, H, H, O] ], [AC8470; H, OEt , H, Et, S, CH = CH 2, H, H, H, O], [AC8471; H, OEt, H, Et, S, C (CH 3) = CH 2 , H, H, H, O],

[AC 8472; H, OEt, H, Et, S, CHCH, H, H, H, O], [AC 8473; H, OEt, H, Et, S, C≡CCH ₃ , H, H, H, O, [AC 8474; H, OEt, H, Et, S, c-Pr, H, H, H, O], [AC 8475; H, OEt, H, Et, S, OMe, H, H, H, O], [AC 8476; H, OEt, H, Et, S, OEt, H, H, H, O], [AC 8477; H, OEt, H, Et, S, Oi-Pr, H, H, H, H, O, [AC 8478; H, OEt, H, Et, S, SMe, H, H, H, O], [AC 8479; H, OEt, H, Et, S, SE t, H, H, H, O] , [AC8480; H, OEt, H, Et, S, CH 2 F, H, H, H, O], [AC8481; H, OEt, H, Et, S, CHF 2, H, H, H, O ], [AC8482; H, OEt , H, Et, S, CF 3, H, H, H, O], [AC8483; H, OEt, H, Et, S, OCH 2 F, H, H, H, O], [AC 8484; H, OEt, H, Et, S, OCHF ₂ , H, H, H, O], [AC 8485; H, OEt, H, Et, S, OCF ₃ , H, H, H, H, H, OEt, H, Et, S, SCH ₂ F, H, H, H, O], [AC 8487; H, OEt, H, Et, S, SCHF ₂ , H, H, H] , O], [AC8488; H , OEt, H, Et, S, SCF 3, H, H, H, O], [AC8489; H, OEt, H, Et, S, CN, H, H, H, O, [AC 8490; H, OEt, H, Et, S, NO ₂ , H, H, O], [AC 8491; H, OEt, H, Pr, S, H, H, H, H, O H, OEt, H, Pr, S, F, H, H, O], [AC8493; H, OEt, H, Pr, S, Cl, H, H, H, O], [AC 8494; H, OEt, H, Pr, S, Br, H, H, H, O], [AC 8495; H, OEt, H, Pr, S, I, H, H, H, O], [AC 8496 H, OEt, H, Pr, S, Me, H, H, H, O], [AC 8497; H, OEt, H, Pr, S, Et, H, H, H, O], [AC 8498; H , OEt, H, Pr, S, Pr, H, H, H, O], [AC 8499; H, OEt, H, Pr, S, i-Pr, H, H, H, O], [AC 8500; H , OEt, H, Pr, S, CH = CH 2, H, H, H, O], [AC8501; H, OEt, H, Pr, S, C (CH 3) = CH 2, H, H, H, O] H, OEt, H, Pr, S, C≡CH, H, H, H, O], [AC8503; H, OEt, H, Pr, S, C≡CCH ₃ , H, H, H , O], [AC8504; H, OEt, H, Pr, S, c-Pr, H, H, H, O], [AC8505; H, OEt, H, Pr, S, OMe, H, H, H] , O], [AC8506; H, OEt, H, Pr, S, OEt, H, H, H, O], [AC 8507; H, OEt, H, Pr, S, Oi-Pr, H, H, H H, OEt, H, Pr, S, SMe, H, H, H, O], [AC 8509; H, OEt, H, Pr, S, SEt, H, H, H, O ], [AC8510; H, OEt , H, Pr, S, CH 2 F, H, H, H, O], [AC8511; H, OEt, H, Pr, S, CHF 2, H, H, H, O], [AC8512; H, OEt, H, Pr, S, CF 3, H, H, H, O], [AC8513; H, OEt, H, Pr, S, OCH 2 F, H, H, H , O], [AC 8514; H, OEt, H, Pr, S, OCHF ₂ , H, H, H, O], [AC 8515; H, OE t, H, Pr, S, OCF ₃ , H, H, H , O], [AC 8516; H, OEt, H, Pr, S, SCH ₂ F, H, H, H, O], [AC 8517; H, OE t, H, Pr, S, SCHF ₂ , H, H, H, O], [AC 8518; H, OEt, H, Pr, S, SCF ₃ , H, H, H, O], [AC 8519; H, OE t, H, Pr, S, CN, H, H, H , O], [AC 8520; H, OEt, H, Pr, S, NO ₂ , H, H, H, O], [AC 8521; H, OE t, H, i-Pr, S, H, H, H, H, O], [AC 8522; H, OEt, H, i-Pr, S, F, H, H, H, O], [AC 8523; H, OE t, H, i-Pr, S, Cl, H, H, H, O], [AC 8524; H, OEt, H, i-Pr, S, Br, H, H, H, O], [AC 8525; H, OE t, H, i-Pr, S, I, H, H, H, O], [AC 8526; H, OEt, H, i-Pr, S, Me, H, H, H, O], [AC 8527; H, OE t, H, i-Pr, S, Et, H, H, H, O H, OEt, H, i-Pr, S, Pr, H, H, H, O], [AC8529; H, OEt, H, i-Pr, S, i-Pr, H, H] , H, O], [AC8530 ; H, OEt, H, i-Pr, S, CH = CH 2, H, H, H, O], [AC8531; H, OEt, H, i-Pr, S, _{C (CH 3) = CH 2} , H, H, H, O], [AC8532; H, OEt, H, i-Pr, S, C≡CH, H, H, H, O], [AC8533; H , OEt, H, i-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 8534; H, OEt, H, i-Pr, S, c-Pr, H, H, H, O], [AC 8535; H, OEt, H, i-Pr, S, OMe, H, H, H, O], [AC 8536; H, OEt, H, i-Pr, S, OEt, H, H, H, H, O], [AC 8537; H, OEt, H, i-Pr, S, Oi-Pr, H, H, H, O], [AC 8538; H, OEt, H, i-Pr, S, SMe, H, H, H, O], [AC 8539; H, OEt, H, i-Pr, S, SE t, H, H, H, O], [AC 8540; H, OE t, H, i-Pr, S, _{CH 2 F, H, H,} H, O], [AC8541; H, OEt, H, i-Pr, S, CHF 2, H, H, H, O], [AC8542; H, OEt, H, i _{-Pr, S, CF 3, H} , H, H, O], [AC8543; H, OEt, H, i-Pr, S, OCH 2 F, H, H, H, O], [AC8544; H, OEt, H, i-Pr, S, OCHF 2, H, H, H, O], [AC8545; H, OEt, H, i-Pr, S, OCF 3, H, H, H, O], [ AC 8546; H, OEt, H, i-Pr, S, SCH ₂ F, H, H, H, O], [AC 8547; H, OEt, H, i-Pr, S, SCHF ₂ , H, H, H , O], [AC8548; H , OEt, H, i-Pr, S, SCF 3, H, H, H, O], [AC8549; H, OEt, H, i-Pr, S, CN, H, H, H, O], [ AC8550; H, OEt, H, i-Pr, S, NO 2, H, H, H, O], [AC8551; H, OEt, H, c-Pr, S, H H, H, H, O], [AC8552; H, OEt, H, c-Pr, S, F, H, H, H] O, [AC8553; H, OEt, H, c-Pr, S , Cl, H, H, H, O], [AC8554 H, OEt, H, c-Pr, S, Br, H, H, H, O], [AC 8555; H, OEt, H, c-Pr, S, I, H, H, O], [AC 8556; H, OEt, H, c-Pr, S, Me, H, H, H, O], [AC 8557; H, OEt, H, c-Pr, S, Et, H, H, H, O H, OEt, H, c-Pr, S, Pr, H, H, H, O], [AC 8559; H, OEt, H, c-Pr, S, i-Pr, H, H] , H, O], [AC8560 ; H, OEt, H, c-Pr, S, CH = CH 2, H, H, H, O], [AC8561; H, OEt, H, c-Pr, S, _{C (CH 3) = CH 2} , H, H, H, O], [AC8562; H, OEt, H, c-Pr, S, C≡CH, H, H, H, O], [AC8563; H , OEt, H, c-Pr , S, C≡CCH 3, H, H, H, O], [AC8564; H, OEt, H, c-Pr, S, c-Pr, H, H, H, O], [AC 8565; H, OEt, H, c-Pr, S, OMe, H, H, H, O], [AC 8566; H, OEt, H, c-Pr, S, OEt, H, H, H, H, O], [AC 8567; H, OEt, H, c-Pr, S, Oi-Pr, H, H, H, O], [AC 8568; H, OEt, H, c-Pr, S, SMe, H, H, H, O], [AC 8569; H, OEt, H, c-Pr, S, SE t, H, H, H, O], [AC 8570; H, OE t, H, c-Pr, S, _{CH 2 F, H, H,} H, O], [AC8571; H, OEt, H, c-Pr, S, CHF 2, H, H, H, O],

[AC8572; H, OEt, H , c-Pr, S, CF 3, H, H, H, O], [AC8573; H, OEt, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC8574; H, OEt, H, c-Pr, S, OCHF 2, H, H, H, O], [AC8575; H, OEt, H, c-Pr, S, OCF 3, H, H, H, O], [AC 8576; H, OEt, H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC 8577; H, OE t, H, c-Pr, S, SCHF ₂ , H, H, H, O], [AC 8578; H, OEt, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 8579; H, OE t, H, c-Pr, S, CN, H, H, H, O, [AC 8580; H, OEt, H, c-Pr, S, NO ₂ , H, H, H, O], [AC 858 1; H, OE t , H, SMe, S, H, H, H, H, O], [AC8582; H, OEt, H, SMe, S, F, H, H, O], [AC8583; H, OEt, H , SMe, S, Cl, H, H, H, O], [AC 8584; H, OEt, H, SMe, S, Br, H, H, O], [AC 8585; H, OEt, H, SMe , S, I, H, H, H, O], [AC 8586; H, OEt, H, SMe, S, Me, H, H, H, O], [AC 8587; H, OE t, H, SMe, S , Et, H, H, H, O], [AC 8588; H, OEt, H, SMe, S, Pr, H, H, H, O], [AC 8589; H, OE t, H, SMe, S, i, -Pr, H, H, H, O], [AC8590; H, OEt, H, SMe, S, CH = CH 2, H, H, H, O], [AC8591; H, OEt, H, SMe, _{S, C (CH 3) =} CH 2, H, H, H, O], [AC8592; H, OEt, H, SMe, S, C≡CH, H, H, H, O], [AC8593; H , OEt, H, SMe, S, C≡CCH ₃ , H, H, H, O], [AC 8594; H, OEt, H, SMe, S, c-Pr, H, H, H, O], [[ AC 8595; H, OEt, H, SMe, S, OMe, H, H, H, O], [AC 8596; H, OEt, H, SMe, S, OEt, H, H, H, O], [AC 8597; H, OEt, H, SMe, S, Oi-Pr, H, H, H, O], [AC 8598; H, OEt, H, SMe, S, SMe, H, H, H, O], [A H, OEt, H, SMe, S, SEt, H, H, H, O], [AC 8600; H, OEt, H, SMe, S, CH ₂ F, H, H, H, O], [C 8 599; AC8601; H, OEt, H, SMe, S, CHF 2, H, H, H, O], [AC8602; H, OEt, H, SMe, S, CF 3, H, H, H, O], [ AC8603; H, OEt, H, SMe, S, OCH 2 F, H, H, H, O], [AC8604; H, OEt, H, SMe, S, OCHF 2, H, H, H, O], [AC8605; H, OEt, H , SMe, S, OCF 3, H, H, H, O], [AC8606; H, OEt, H, SMe, S, SCH 2 F, H, H, H, O] , [AC 8607; H, OEt, H, SMe, S, SCHF ₂ , H, H, H, O], [AC 8608; H, OEt, H, SMe, S, SCF ₃ , H, H, H, O] [AC 8609; H, OEt, H, SMe, S, CN, H, H, H, O], [AC 8610; H, OEt, H, SMe, S, NO ₂ , H, H, H, O], [AC8611; H, OEt, H, OMe, S, H, H, H, H, O], [AC8612; H, OEt, H, OMe, S, F, H, H, H, O], [AC8613 H, OEt, H, OMe, S, Cl, H, H, H, O], [AC8614; H, OEt, H, OMe, S, Br, H, H, H, O], [AC8615; H , OEt, H, OMe, S, I, H, H, H, O], [AC8616; H, OEt, H, OMe, S, Me, H, H, H, O], [AC8617; H, OEt , H, OMe, S, Et, H, H, H, O], [AC8618; H, OEt, H, OMe, S, Pr, H, H, H, O], [AC8619; H, OEt, H , OMe, S, i-Pr , H, H, H, O], [AC8620; H, OEt, H, OMe, S, CH = CH 2, H, H, H, O], [AC8621; H, OEt, H, OMe, S, C (CH 3) = CH 2, H, H, H, O], [AC8622; H, OEt, H, OMe, S, C≡CH, H, H, H, O ], [AC8623; H, OEt , H, OMe, S, C≡CCH 3, H, H, H, O], [AC8624; H, OEt, H, OMe, S, c-Pr, H, H, H, O], [AC8625; H, OEt, H, OMe, S, OMe, H, H, H, O], [AC 8626; H , OEt, H, OMe, S, OEt, H, H, H, O], [AC8627; H, OEt, H, OMe, S, Oi-Pr, H, H, H, O], [AC8628; H , OEt, H, OMe, S, SMe, H, H, H, O], [AC8629; H, OEt, H, OMe, S, SEt, H, H, H, O], [AC8630; H, OEt , H, OMe, S, CH 2 F, H, H, H, O], [AC8631; H, OEt, H, OMe, S, CHF 2, H, H, H, O], [AC8632; H, OEt, H, OMe, S, CF 3, H, H, H, O], [AC8633; H, OEt, H, OMe, S, OCH 2 F, H, H, H, O], [AC8634; H , OEt, H, OMe, S , OCHF 2, H, H, H, O], [AC8635; H, OEt, H, OMe, S, OCF 3, H, H, H, O], [AC8636; H , OEt, H, OMe, S, SCH ₂ F, H, H, H, O], [AC 8637; H, OE t, H, OMe, S, SCHF ₂ , H, H, H, O], [AC 8638; H, OEt, H, OMe, S, SCF 3, H, H, H, O], [AC8639; H, OEt, H, OMe, S, CN, H, H, H, O], [AC8640; H , OEt, H, OMe, S , NO 2, H, H, H, O], [AC8641; H, OEt, H, F, S, H, H, H, H, O], [AC8642; H, OEt, H, F, S, F, H, H, H, O], [AC8643; H, OEt, H, F, S, Cl, H, H, O], [AC8644; H, OEt, H, F, S, Br, H, H, H, O], [AC8645; H, OEt, H, F, S, I, H, H, H, O], [AC 8646; H, OEt, H, F, S, Me, H, H, H, O], [AC 8647; H, OEt, H, F, S, Et, H, H, H, O], [AC 8648; H, OE t, H, F, S, Pr, H, H, H, O], [AC8649; H, OEt, H, F, S, i-Pr, H, H, H, O], [AC8650; H, OEt, H, F, _{S, CH = CH 2, H} , H, H, O], [AC8651; H, OEt, H, F, S, C (CH 3) = CH 2, H, H, H, O], [AC8652; H, OEt, H, F, S, C≡CH, H, H, H, O], [AC8653; H, OEt, H, F, S, C≡ CCH ₃ , H, H, H, O], [AC865 4; H, OEt, H, F, S, c-Pr, H, H, H, O], [AC8655; H, OEt, H, F, S, OMe, H, H, H, O], [[ AC 8656; H, OEt, H, F, S, OEt, H, H, H, O], [AC8657; H, OEt, H, F, S, Oi-Pr, H, H, H, O], [ AC 8658; H, OEt, H, F, S, SMe, H, H, H, O], [AC 8659; H, OEt, H, F, S, SE t, H, H, H, O], [AC 8660; H, OEt, H, F, S, CH 2 F, H, H, H, O], [AC8661; H, OEt, H, F, S, CHF 2, H, H, H, O], [AC8662 ; H, OEt, H, F , S, CF 3, H, H, H, O], [AC8663; H, OEt, H, F, S, OCH 2 F, H, H, H, O], [ AC8664; H, OEt, H, F, S, OCHF 2, H, H, H, O], [AC8665; H, OEt, H, F, S, OCF 3, H, H, H, O], [ AC 8666; H, OEt, H, F, S, SCH ₂ F, H, H, H, O], [AC 8667; H, OEt, H, F, S, SCHF ₂ , H, H, H, O], [AC8668; H, OEt, H , F, S, SCF 3, H, H, H, O], [AC8669; H, OEt, H, F, S, CN, H, H, H, O], [ AC8670; H, OEt, H, F, S, NO 2, H, H, H, O], [AC8671; H, OEt, H, Cl, S, H, H, H, H, O],

[AC8672; H, OEt, H, Cl, S, F, H, H, O], [AC8673; H, OEt, H, Cl, S, Cl, H, H, H, O], [AC 8674 H, OEt, H, Cl, S, Br, H, H, O], [AC8675; H, OEt, H, Cl, S, I, H, H, O], [AC8676; H , OEt, H, Cl, S, Me, H, H, H, O], [AC 8677; H, OEt, H, Cl, S, Et, H, H, H, O], [AC 8678; H, OEt , H, Cl, S, Pr, H, H, H, O], [AC 8679; H, OEt, H, Cl, S, i-Pr, H, H, H, O], [AC 8680; H, OEt , H, Cl, S, CH = CH 2, H, H, H, O], [AC8681; H, OEt, H, Cl, S, C (CH 3) = CH 2, H, H, H, O H, OEt, H, Cl, S, C≡CH, H, H, H, O], [AC8683; H, OEt, H, Cl, S, C≡CCH ₃ , H, H, H] H, O], [AC8684; H, OEt, H, Cl, S, c-Pr, H, H, H, O], [AC8685; H, OEt, H, Cl, S, OMe, H, H, H H, O], [AC8686; H, OEt, H, Cl, S, OEt, H, H, H, O], [AC8687; H, OEt, H, Cl, S, Oi-Pr, H, H, H, H, O], [AC8688; H, OEt, H, Cl, S, SMe, H, H, H, O], [AC8689; H, OEt, H, Cl, S, SEt, H, H, H, H, O], [AC8690; H, OEt, H, Cl, S, CH 2 F, H, H, H, O], [AC8691; H, OEt, H, Cl, S, CHF 2, H, H, H , O], [AC8692; H , OEt, H, Cl, S, CF 3, H, H, H, O], [AC8693; H, OEt, H, Cl, S, OCH 2 F, H, H, H, O], [AC8694; H, OEt, H, Cl, S, OCHF 2, H, H, H, O], [AC8695; H, OEt, H, Cl, S, OCF 3, H, H, H, O], [AC 8696; H, OEt, H, Cl, S, SCH ₂ F, H, H, H, O], [AC 8697; H, OE t, H, Cl, S, SCHF ₂ , H, H , H, O], [AC 86 98; H, OEt, H, Cl, S, SCF ₃ , H, H, H, O], [AC 8699; H, OE t, H, Cl, S, CN, H, H, H, O ], [AC8700; H, OEt , H, Cl, S, NO 2, H, H, H, O], [AC8701; H, OEt, H, Br, S, H, H, H, H, O] H, OEt, H, Br, S, F, H, H, O], [AC 8703; H, OEt, H, Br, S, Cl, H, H, H, O], [AC 8702; AC 8704; H, OEt, H, Br, S, Br, H, H, H, O], [AC 8705; H, OEt, H, Br, S, I, H, H, H, O], [AC 8706; H, OEt, H, Br, S, Me, H, H, H, O], [AC 8707; H, OEt, H, Br, S, Et, H, H, H, O], [AC 8708; H, OEt, H, Br, S, Pr, H, H, H, O], [AC 8709; H, OEt, H, Br, S, i-Pr, H, H, H, O], [AC 8710; H, OEt, H, Br, S, CH = CH 2, H, H, H, O], [AC8711; H, OEt, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC 8712; H, OEt, H, Br, S, C≡CH, H, H, H, O], [AC 8713; H, OEt, H, Br, S, C≡ CCH ₃ , H, H , H, O], [AC 8714; H, OEt, H, Br, S, c-Pr, H, H, H, O], [AC 8715; H, OE t, H, Br, S, OMe, H, H , H, O], [AC8716; H, OEt, H, Br, S, OEt, H, H, H, O], [AC 8717; H, OEt, H, Br, S, Oi-Pr, H, H , H, O], [AC 8718; H, OEt, H, Br, S, SMe, H, H, H, O], [AC 8719; H, OEt, H, Br, S, SE t, H, H, H , O], [AC8720; H , OEt, H, Br, S, CH 2 F, H, H, H, O], [AC8721; H, OEt, H, Br, S, CHF 2, H, H, H, O], [AC8722; H, OEt, H, Br, S, CF 3, H, H, H, O], [AC8723; H, OEt, H, Br, S, OCH 2 F, H, H , H, O], [AC 8724; H, OEt, H, Br, S, OCHF ₂ , H, H, H, O], [AC 8725; H, OE t, H, Br, S, OCF ₃ , H, H , H, O], [AC 8726; H, OEt, H, Br, S, SCH ₂ F, H, H, H, O], [AC 8727; H, OE t, H, Br, S, SCHF ₂ , H, H, H, O ], [AC8728; H, OEt , H, Br, S, SCF 3, H, H, H, O], [AC8729; H, OEt, H, Br, S, CN, H, H, H, O] H, OEt, H, Br, S, NO ₂ , H, H, O], [AC 8731; H, CHF ₂ , H, H, S, H, H, H, H, O] _{, [AC8732; H, CHF 2} , H, H, S, F, H, H, H, O], [AC8733; H, CHF 2, H, H, S, Cl, H, H, H, O] , [AC 8734; H, CHF ₂ , H, H, S, Br, H, H, H, O], [AC 87 35; H, CHF ₂ , H, H, S, I, H, H, H, O] _{, [AC8736; H, CHF 2} , H, H, S, Me, H, H, H, O], [AC8737; H, CHF 2, H, H, S, Et, H, H, H, O] _{, [AC8738; H, CHF 2} , H, H, S, Pr, H, H, H, O], [AC8739; H, CHF 2, H, H, S, i-Pr, H, H, H, O], [AC8740; H, CHF 2, H, H, S, CH = CH 2, H, H, H, O], [AC8741; H, CHF 2, H, H, S, C (CH 3) = CH ₂ , H, H, H, O], [AC8742; H, CHF ₂ , H, H, S, C≡CH, H, H, H, O], [AC8743; H, CHF ₂ , H, _{H, S, C≡CCH 3, H} , H, H, O], [AC8744; H, CHF 2, H, H, S, c-Pr, H, H, H, O], [AC8745; H, _{CHF 2, H, H, S} , OMe, H, H, H, O], [AC8746; H, CHF 2, H, H, S, OEt, H, H, H, O], [AC8747; H, _{CHF 2, H, H, S} , Oi-Pr, H, H, H, O], [AC8748; H, CHF 2, H, H, S, SMe, H, H, H, O], [AC8749; _{H, CHF 2, H, H} , S, SEt, H, H, H, O], [AC8750; H, CHF 2, H, H, S, CH 2 F, H, H, H, O], [ _{AC8751; H, CHF 2, H} , H, S, CHF 2, H, H, H, O], [AC8752; H, CHF 2, H, H, S, CF 3, H, H, H, O] _{, [AC8753; H, CHF 2} , H, H, S, OCH 2 F, H, H, H, O], [AC8754; H, CHF 2, H, H, S, OCHF 2, H, H, H, O], [ AC8755; H, CHF 2, H, H, S, OCF 3, H, H, H, O], [AC8756; H, CHF 2, H, H, S, SCH 2 F , H, H, H, O ], [AC8757; H, CHF 2, H, H, S, SCHF 2, H, H, H, O], [AC8758; H, CHF 2, H, H, S, SCF ₃ , H, H, H, O], [AC 8759; H, CHF ₂ , H, H, S, CN, H, H, H, O], [AC 8760; H, CHF ₂ , H, H, S _{, NO 2, H, H,} H, O], [AC8761; H, CHF 2, H, Me, S, H, H, H, H, O], [AC8762; H, CHF 2, H, Me, S, F, H, H, H, O], [AC8763; H, CHF 2, H, Me, S, Cl, H, H, H, O], [AC8764; H, CHF 2, H, Me, S, Br, H, H, H, O], [AC8765; H, CHF 2, H, Me, S, I, H, H, H, O], [AC8766; H, CHF 2, H, Me, S, Me, H, H, H, O], [AC 8767; H, CHF ₂ , H, Me, S, Et, H, H, H, O], [AC 8768; H, CHF ₂ , H, Me, S, Pr, H, H, H, O], [AC 8769; H, CHF ₂ , H, Me, S, i-Pr, H, H, H, O], [AC 8770; H, CHF ₂ , H, Me, S, CH = CH ₂ , H, H, H, O],

_{[AC8771; H, CHF 2,} H, Me, S, C (CH 3) = CH 2, H, H, H, O], [AC8772; H, CHF 2, H, Me, S, C≡CH, H, H, H, O] , [AC8773; H, CHF 2, H, Me, S, C≡CCH 3, H, H, H, O], [AC8774; H, CHF 2, H, Me, S , c-Pr, H, H , H, O], [AC8775; H, CHF 2, H, Me, S, OMe, H, H, H, O], [AC8776; H, CHF 2, H, Me , S, OEt, H, H , H, O], [AC8777; H, CHF 2, H, Me, S, Oi-Pr, H, H, H, O], [AC8778; H, CHF 2, H , Me, S, SMe, H, H, H, O], [AC 8779; H, CHF ₂ , H, Me, S, SE t, H, H, H, O], [AC 8780; H, CHF ₂ , H _{, Me, S, CH 2 F} , H, H, H, O], [AC8781; H, CHF 2, H, Me, S, CHF 2, H, H, H, O], [AC8782; H, CHF _{2, H, Me, S,} CF 3, H, H, H, O], [AC8783; H, CHF 2, H, Me, S, OCH 2 F, H, H, H, O], [AC8784; _{H, CHF 2, H, Me} , S, OCHF 2, H, H, H, O], [AC8785; H, CHF 2, H, Me, S, OCF 3, H, H, H, O], [ _{AC8786; H, CHF 2, H} , Me, S, SCH 2 F, H, H, H, O], [AC8787; H, CHF 2, H, Me, S, SCHF 2, H, H, H, O H, CHF ₂ , H, Me, S, SCF ₃ , H, H, H, O], [AC 8789; H, CHF ₂ , H, Me, S, CN, H, H, H, H] O], [AC8790; H, CHF 2, H, Me, S, NO 2, H, H, H, O], [AC8791; H, CHF 2, H, Et, S, H, H, H, H , O], [AC8792; H , CHF 2, H, Et, S, F, H, H, H, O], [AC8793; H, CHF 2, H, Et, S, Cl, H, H, H , O], [AC8794; H , CHF 2, H, Et, S, Br, H, H, H, O], [AC8795; H, CHF 2, H, Et, S, I, H, H, H , O], [AC8796; H , CHF 2, H, Et, S, Me, H , H, H, O], [AC8797; H, CHF 2, H, Et, S, Et, H, H, H, O], [AC8798; H, CHF 2, H, Et, S, Pr, H , H, H, O], [AC8799; H, CHF 2, H, Et, S, i-Pr, H, H, H, O], [AC8800; H, CHF 2, H, Et, S, CH _{= CH 2, H, H,} H, O], [AC8801; H, CHF 2, H, Et, S, C (CH 3) = CH 2, H, H, H, O], [AC8802; H, _{CHF 2, H, Et, S} , C≡CH, H, H, H, O], [AC8803; H, CHF 2, H, Et, S, C≡CCH 3, H, H, H, O], _{[AC8804; H, CHF 2,} H, Et, S, c-Pr, H, H, H, O], [AC8805; H, CHF 2, H, Et, S, OMe, H, H, H, O ], [AC8806; H, CHF 2, H, Et, S, OEt, H, H, H, O], [AC8807; H, CHF 2, H, Et, S, Oi-Pr, H, H, H , O], [AC8808; H , CHF 2, H, Et, S, SMe, H, H, H, O], [AC8809; H, CHF 2, H, Et, S, SEt, H, H, H , O], [AC8810; H , CHF 2, H, Et, S, CH 2 F, H, H, H, O], [AC8811; H, CHF 2, H, Et, S, CHF 2, H, H, H, O], [ AC8812; H, CHF 2, H, Et, S, CF 3, H, H, H, O], [AC8813; H, CHF 2, H, Et, S, OCH 2 F , H, H, H, O ], [AC8814; H, CHF 2, H, Et, S, OCHF 2, H, H, H, O], [AC8815; H, CHF 2, H, Et, S, OCF ₃ , H, H, H, O], [AC 8816; H, CHF ₂ , H, Et, S, SCH ₂ F, H, H, H, O], [AC 8817; H, CHF ₂ , H, Et , S, SCHF ₂ , H, H, H, O], [AC 8818; H, CHF ₂ , H, Et, S, SCF ₃ , H, H, H, O], [AC 8819; H, CHF ₂ , H , Et, S, CN, H , H, H, O], [AC8820; H, CHF 2, H, Et, S, NO 2, H, H, H, O], [AC8821; H, CHF 2, H, Pr, S, H, H, H, H, O], [AC8822; H, _{CHF 2, H, Pr, S} , F, H, H, H, O], [AC8823; H, CHF 2, H, Pr, S, Cl, H, H, H, O], [AC8824; H, CHF ₂ , H, Pr, S, Br, H, H, H, O], [AC 8825; H, CHF ₂ , H, Pr, S, I, H, H, O, [AC 8826; H, _{CHF 2, H, Pr, S} , Me, H, H, H, O], [AC8827; H, CHF 2, H, Pr, S, Et, H, H, H, O], [AC8828; H, _{CHF 2, H, Pr, S} , Pr, H, H, H, O], [AC8829; H, CHF 2, H, Pr, S, i-Pr, H, H, H, O], [AC8830; _{H, CHF 2, H, Pr} , S, CH = CH 2, H, H, H, O], [AC8831; H, CHF 2, H, Pr, S, C (CH 3) = CH 2, H, H, H, O], [ AC8832; H, CHF 2, H, Pr, S, C≡CH, H, H, H, O], [AC8833; H, CHF 2, H, Pr, S, C≡ CCH ₃ , H, H, H, O], [AC 8834; H, CHF ₂ , H, Pr, S, c-Pr, H, H, H, O], [AC 8835; H, CHF ₂ , H, Pr , S, OMe, H, H , H, O], [AC8836; H, CHF 2, H, Pr, S, OEt, H, H, H, O], [AC8837; H, CHF 2, H, Pr , S, Oi-Pr, H , H, H, O], [AC8838; H, CHF 2, H, Pr, S, SMe, H, H, H, O], [AC8839; H, CHF 2, H , Pr, S, SEt, H, H, H, O], [AC 8840; H, CHF ₂ , H, Pr, S, CH ₂ F, H, H, O], [AC 884 1; H, CHF ₂ , H, Pr, S, CHF 2, H, H, H, O], [AC8842; H, CHF 2, H, Pr, S, CF 3, H, H, H, O], [AC8843; H, _{CHF 2, H, Pr, S} , OCH 2 F, H, H, H, O], [AC8844; H, CHF 2, H, Pr, S, OCHF 2, H, H, H, O], [AC8845 H, CHF ₂ , H, Pr, S, OCF ₃ , H, H, H, O], [AC8846; H, CHF ₂ , H, Pr, S, SCH ₂ F, H, H, H, O] _{, [AC8847; H, CHF 2} , H, Pr, S, SCHF 2, H, H, H, O], _{[AC8848; H, CHF 2,} H, Pr, S, SCF 3, H, H, H, O], [AC8849; H, CHF 2, H, Pr, S, CN, H, H, H, O] _{, [AC8850; H, CHF 2} , H, Pr, S, NO 2, H, H, H, O], [AC8851; H, CHF 2, H, i-Pr, S, H, H, H, H , O], [AC8852; H , CHF 2, H, i-Pr, S, F, H, H, H, O], [AC8853; H, CHF 2, H, i-Pr, S, Cl, H , H, H, O], [AC8854; H, CHF 2, H, i-Pr, S, Br, H, H, H, O], [AC8855; H, CHF 2, H, i-Pr, S , I, H, H, H , O], [AC8856; H, CHF 2, H, i-Pr, S, Me, H, H, H, O], [AC8857; H, CHF 2, H, i -Pr, S, Et, H, H, H, O], [AC 8858; H, CHF ₂ , H, i-Pr, S, Pr, H, H, H, O], [AC 8859; H, CHF ₂ , H, i-Pr, S , i-Pr, H, H, H, O], [AC8860; H, CHF 2, H, i-Pr, S, CH = CH 2, H, H, H, O ], [AC8861; H, CHF 2, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC8862; H, CHF 2, H, i-Pr, S, C≡CH, H, H, H, O, [AC 8863; H, CHF ₂ , H, i-Pr, S, C≡CCH ₃ , H, H, H, O], [AC 8864; H, _{CHF 2, H, i-Pr} , S, c-Pr, H, H, H, O], [AC8865; H, CHF 2, H, i-Pr, S, OMe, H, H, H, O] _{, [AC8866; H, CHF 2} , H, i-Pr, S, OEt, H, H, H, O], [AC8867; H, CHF 2, H, i-Pr, S, Oi-Pr, H, H, H, O], [ AC8868; H, CHF 2, H, i-Pr, S, SMe, H, H, H, O], [AC8869; H, CHF 2, H, i-Pr, S, SEt, H, H, H, O], [AC 8870; H, CHF ₂ , H, i-Pr, S, CH ₂ F, H, H, H, O],

[AC 8871; H, CHF ₂ , H, i-Pr, S, CHF ₂ , H, H, H, O], [AC 8872; H, CHF ₂ , H, i-Pr, S, CF ₃ , H, H , H, O], [AC 8873; H, CHF ₂ , H, i-Pr, S, OCH ₂ F, H, H, H, O], [AC 8874; H, CHF ₂ , H, i-Pr, S , OCHF ₂ , H, H, H, O], [AC 8875; H, CHF ₂ , H, i-Pr, S, OCF ₃ , H, H, H, O], [AC 8876; H, CHF ₂ , H , i-Pr, S, SCH ₂ F, H, H, H, O], [AC 8877; H, CHF ₂ , H, i-Pr, S, SCHF ₂ , H, H, H, O], [AC 8878 H, CHF ₂ , H, i-Pr, S, SCF ₃ , H, H, H, O], [AC 8879; H, CHF ₂ , H, i-Pr, S, CN, H, H, H, H O], [AC 8880; H, CHF ₂ , H, i-Pr, S, NO ₂ , H, H, H, O], [AC 888 1; H, CHF ₂ , H, c-Pr, S, H, H , H, H, O], [AC8882; H, CHF 2, H, c-Pr, S, F, H, H, H, O], [AC8883; H, CHF 2, H, c-Pr, S , Cl, H, H, H , O], [AC8884; H, CHF 2, H, c-Pr, S, Br, H, H, H, O], [AC8885; H, CHF 2, H, c -Pr, S, I, H, H, H, O], [AC 8886; H, CHF ₂ , H, c-Pr, S, Me, H, H, O], [AC 8887; H, CHF ₂ , H, c-Pr, S , Et, H, H, H, O], [AC8888; H, CHF 2, H, c-Pr, S, Pr, H, H, H, O], [AC8889; _{H, CHF 2, H, c} -Pr, S, i-Pr, H, H, H, O], [AC8890; H, CHF 2, H, c-Pr, S, CH = CH 2, H, H , H, O], [AC8891 ; H, CHF 2, H, c-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC8892; H, CHF 2, H, c-Pr, S, C≡CH, H, H, H, O], [AC 8893; H, CHF ₂ , H, c-Pr, S, C≡ CCH ₃ , H, H, H, O], [[ _{AC8894; H, CHF 2, H} , c-Pr, S, c-Pr, H, H, H, O], [AC8895; H, CHF 2, H, c-Pr, S, OMe, H, H, H, O], [AC8896; H, CHF 2, H, c-Pr, S, OEt, H, H, H, O], [AC8897; H, CHF _{2, H, c-Pr,} S, Oi-Pr, H, H, H, O], [AC8898; H, CHF 2, H, c-Pr, S, SMe, H, H, H, O], _{[AC8899; H, CHF 2,} H, c-Pr, S, SEt, H, H, H, O], [AC8900; H, CHF 2, H, c-Pr, S, CH 2 F, H, H , H, O], [AC8901 ; H, CHF 2, H, c-Pr, S, CHF 2, H, H, H, O], [AC8902; H, CHF 2, H, c-Pr, S, _{CF 3, H, H, H} , O], [AC8903; H, CHF 2, H, c-Pr, S, OCH 2 F, H, H, H, O], [AC8904; H, CHF 2, H , c-Pr, S, OCHF 2, H, H, H, O], [AC8905; H, CHF 2, H, c-Pr, S, OCF 3, H, H, H, O], [AC8906; _{H, CHF 2, H, c} -Pr, S, SCH 2 F, H, H, H, O], [AC8907; H, CHF 2, H, c-Pr, S, SCHF 2, H, H, H , O], [AC8908; H , CHF 2, H, c-Pr, S, SCF 3, H, H, H, O], [AC8909; H, CHF 2, H, c-Pr, S, CN, H, H, H, O] , [AC8910; H, CHF 2, H, c-Pr, S, NO 2, H, H, H, O], [AC8911; H, CHF 2, H, SMe, S , H, H, H, H , O], [AC8912; H, CHF 2, H, SMe, S, F, H, H, H, O], [AC8913; H, CHF 2, H, SMe, S , Cl, H, H, H , O], [AC8914; H, CHF 2, H, SMe, S, Br, H, H, H, O], [AC8915; H, CHF 2, H, SMe, S , I, H, H, H , O], [AC8916; H, CHF 2, H, SMe, S, Me, H, H, H, O], [AC8917; H, CHF 2, H, SMe, S , Et, H, H, H , O], [AC8918; H, CHF 2, H, SMe, S, Pr, H, H, H, O], [AC8919; H, CHF 2, H, SMe, S , i-Pr, H, H , H, O], [AC8920; H, CHF 2, H, SMe, S, CH = CH _{2, H, H, H,} O], [AC8921; H, CHF 2, H, SMe, S, C (CH 3) = CH 2, H, H, H, O], [AC8922; H, CHF 2 , H, SMe, S, C≡CH, H, H, H, O], [AC 8923; H, CHF ₂ , H, SMe, S, C≡ CCH ₃ , H, H, H, O], [AC 8924 _{; H, CHF 2, H,} SMe, S, c-Pr, H, H, H, O], [AC8925; H, CHF 2, H, SMe, S, OMe, H, H, H, O], _{[AC8926; H, CHF 2,} H, SMe, S, OEt, H, H, H, O], [AC8927; H, CHF 2, H, SMe, S, Oi-Pr, H, H, H, O ], [AC8928; H, CHF 2, H, SMe, S, SMe, H, H, H, O], [AC8929; H, CHF 2, H, SMe, S, SEt, H, H, H, O ], [AC8930; H, CHF 2, H, SMe, S, CH 2 F, H, H, H, O], [AC8931; H, CHF 2, H, SMe, S, CHF 2, H, H, H, O], [AC8932; H, CHF 2, H, SMe, S, CF 3, H, H, H, O], [AC8933; H, CHF 2, H, SMe, S, OCH 2 F, H , H, H, O], [AC8934; H, CHF 2, H, SMe, S, OCHF 2, H, H, H, O], [AC8935; H, CHF 2, H, SMe, S, OCF 3 , H, H, H, O ], [AC8936; H, CHF 2, H, SMe, S, SCH 2 F, H, H, H, O], [AC8937; H, CHF 2, H, SMe, S _{, SCHF 2, H, H,} H, O], [AC8938; H, CHF 2, H, SMe, S, SCF 3, H, H, H, O], [AC8939; H, CHF 2, H, SMe , S, CN, H, H , H, O], [AC8940; H, CHF 2, H, SMe, S, NO 2, H, H, H, O], [AC8941; H, CHF 2, H, OMe, S, H, H, H, H, O], [AC8942; H, CHF 2, H, OMe, S, F, H, H, H, O], [AC8943; H, CHF 2, H, OMe, S, Cl, H, H, H, O], [AC8944; H, CHF 2, H, OMe, S, Br, H, H, H, O], [AC8945; H, CHF 2, H, OMe, S, I , H, H, H, O ], [AC8946; H, CHF 2, H, OMe, S, Me, H, H, H, O], [AC8947; H, CHF 2, H, OMe, S, Et H, H, H, O], [AC 8948; H, CHF ₂ , H, OMe, S, Pr, H, H, H, O], [AC 8949; H, CHF ₂ , H, OMe, S, i -Pr, H, H, H, O], [AC 8950; H, CHF ₂ , H, OMe, S, CH = CH ₂ , H, H, H, O], [AC 8951; H, CHF ₂ , H, _{OMe, S, C (CH 3} ) = CH 2, H, H, H, O], [AC8952; H, CHF 2, H, OMe, S, C≡CH, H, H, H, O], [ _{AC8953; H, CHF 2, H} , OMe, S, C≡CCH 3, H, H, H, O], [AC8954; H, CHF 2, H, OMe, S, c-Pr, H, H, H , O], [AC8955; H , CHF 2, H, OMe, S, OMe, H, H, H, O], [AC8956; H, CHF 2, H, OMe, S, OEt, H, H, H , O], [AC8957; H , CHF 2, H, OMe, S, Oi-Pr, H, H, H, O], [AC8958; H, CHF 2, H, OMe, S, SMe, H, H , H, O], [AC 8959; H, CHF ₂ , H, OMe, S, SE t, H, H, H, O], [AC 8960; H, CHF ₂ , H, OMe, S, CH ₂ F, H , H, H, O], [AC8961; H, CHF 2, H, OMe, S, CHF 2, H, H, H, O], [AC8962; H, CHF 2, H, OMe, S, CF 3 , H, H, H, O ], [AC8963; H, CHF 2, H, OMe, S, OCH 2 F, H, H, H, O], [AC8964; H, CHF 2, H, OMe, S _{, OCHF 2, H, H,} H, O], [AC8965; H, CHF 2, H, OMe, S, OCF 3, H, H, H, O], [AC8966; H, CHF 2, H, OMe , S, SCH ₂ F, H, H, H, O], [AC 8967; H, CHF ₂ , H, OMe, S, SCHF ₂ , H, H, H, O], [AC 8968; H, CHF ₂ , _{H, OMe, S, SCF 3} , H, H, H, O], [AC8969; H, CHF 2, H, OMe, S, CN, H, H, H, O], [AC8970; H, CHF 2 , H, OMe , S, NO ₂ , H, H, H, O],

_{[AC8971; H, CHF 2,} H, F, S, H, H, H, H, O], [AC8972; H, CHF 2, H, F, S, F, H, H, H, O], _{[AC8973; H, CHF 2,} H, F, S, Cl, H, H, H, O], [AC8974; H, CHF 2, H, F, S, Br, H, H, H, O], _{[AC8975; H, CHF 2,} H, F, S, I, H, H, H, O], [AC8976; H, CHF 2, H, F, S, Me, H, H, H, O], _{[AC8977; H, CHF 2,} H, F, S, Et, H, H, H, O], [AC8978; H, CHF 2, H, F, S, Pr, H, H, H, O], _{[AC8979; H, CHF 2,} H, F, S, i-Pr, H, H, H, O], [AC8980; H, CHF 2, H, F, S, CH = CH 2, H, H, H, O], [AC8981; H, CHF 2, H, F, S, C (CH 3) = CH 2, H, H, H, O], [AC8982; H, CHF 2, H, F, S , C≡CH, H, H, H, O], [AC 8983; H, CHF ₂ , H, F, S, C≡ CCH ₃ , H, H, H, O], [AC 8984; H, CHF ₂ , H, F, S, c- Pr, H, H, H, O], [AC8985; H, CHF 2, H, F, S, OMe, H, H, H, O], [AC8986; H, CHF ₂ , H, F, S, OEt, H, H, H, O], [AC 8987; H, CHF ₂ , H, F, S, Oi-Pr, H, H, H, O], [AC 8988; H _{, CHF 2, H, F,} S, SMe, H, H, H, O], [AC8989; H, CHF 2, H, F, S, SEt, H, H, H, O], [AC8990; H , CHF ₂ , H, F, S, CH ₂ F, H, H, H, O], [AC8991; H, CHF ₂ , H, F, S, CHF ₂ , H, H, H, O], [[ _{AC8992; H, CHF 2, H} , F, S, CF 3, H, H, H, O], [AC8993; H, CHF 2, H, F, S, OCH 2 F, H, H, H, O ], [AC8994; H, CHF 2, H, F, S, OCHF 2, H, H, H, O], [AC8995; H, CHF 2, H, F, S, OCF 3, H, H, H , O], [AC8996; H , CHF 2, H, F, S, SCH 2 F, H, H, H, O], [AC8997; H, CHF 2, H, F, S , SCHF ₂ , H, H, H, O], [AC 8998; H, CHF ₂ , H, F, S, SCF ₃ , H, H, H, O], [AC 8999; H, CHF ₂ , H, F , S, CN, H, H, H, O], [AC 9000; H, CHF ₂ , H, F, S, NO ₂ , H, H, H, O], [AC 9001; H, CHF ₂ , H, O, Cl, S, H, H, H, H, O], [AC9002; H, CHF 2, H, Cl, S, F, H, H, H, O], [AC9003; H, CHF 2, H, Cl, S, Cl, H, H, H, O], [AC9004; H, CHF 2, H, Cl, S, Br, H, H, H, O], [AC9005; H, CHF 2, H, Cl, S, I, H, H, H, O], [AC9006; H, CHF 2, H, Cl, S, Me, H, H, H, O], [AC9007; H, CHF 2, H, Cl, S, Et, H, H, H, O], [AC9008; H, CHF 2, H, Cl, S, Pr, H, H, H, O], [AC9009; H, CHF 2, H, Cl, S, i-Pr, H, H, H, O], [AC9010; H, CHF 2, H, Cl, S, CH = CH 2, H, H, H, O], [AC9011; H, _{CHF 2, H, Cl, S} , C (CH 3) = CH 2, H, H, H, O], [AC9012; H, CHF 2, H, Cl, S, C≡CH, H, H, H , O], [AC9013; H , CHF 2, H, Cl, S, C≡CCH 3, H, H, H, O], [AC9014; H, CHF 2, H, Cl, S, c-Pr, H, H, H, O] , [AC9015; H, CHF 2, H, Cl, S, OMe, H, H, H, O], [AC9016; H, CHF 2, H, Cl, S, OEt, H, H, H, O] , [AC9017; H, CHF 2, H, Cl, S, Oi-Pr, H, H, H, O], [AC9018; H, CHF 2, H, Cl, S, SMe, H, H, H, O], [AC9019; H, CHF 2, H, Cl, S, SEt, H, H, H, O], [AC9020; H, CHF 2, H, Cl, S, _{CH 2 F, H, H,} H, O], [AC9021; H, CHF 2, H, Cl, S, CHF 2, H, H, H, O], [AC9022; H, CHF 2, H, Cl , S, CF ₃ , H, H, H, O], [AC 9023; H, CHF ₂ , H, Cl, S, OCH ₂ F, H, H, H, O], [AC9024; H, CHF 2, H, Cl, S, OCHF 2, H, H, H, O], [AC9025; H, CHF 2, H, Cl, S , OCF ₃ , H, H, H, O], [AC 9026; H, CHF ₂ , H, Cl, S, SCH ₂ F, H, H, H, O], [AC 9027; H, CHF ₂ , H, H, _{Cl, S, SCHF 2, H} , H, H, O], [AC9028; H, CHF 2, H, Cl, S, SCF 3, H, H, H, O], [AC9029; H, CHF 2, H, Cl, S, CN, H, H, H, O], [AC9030; H, CHF 2, H, Cl, S, NO 2, H, H, H, O], [AC9031; H, CHF 2 , H, Br, S, H , H, H, H, O], [AC9032; H, CHF 2, H, Br, S, F, H, H, H, O], [AC9033; H, CHF 2 , H, Br, S, Cl, H, H, H, O], [AC 9034; H, CHF ₂ , H, Br, S, Br, H, H, H, O], [AC 9035; H, CHF ₂ , H, Br, S, I , H, H, H, O], [AC9036; H, CHF 2, H, Br, S, Me, H, H, H, O], [AC9037; H, CHF 2 , H, Br, S, Et, H, H, H, O], [AC 9038; H, CHF ₂ , H, Br, S, Pr, H, H, H, O], [AC 9039; H, CHF ₂ , H, Br, S, i -Pr, H, H, H, O], [AC9040; H, CHF 2, H, Br, S, CH = CH 2, H, H, H, O], [AC9041 _{; H, CHF 2, H,} Br, S, C (CH 3) = CH 2, H, H, H, O], [AC9042; H, CHF 2, H, Br, S, C≡CH, H, H, H, O], [ AC9043; H, CHF 2, H, Br, S, C≡CCH 3, H, H, H, O], [AC9044; H, CHF 2, H, Br, S, c -Pr, H, H, H, O], [AC9045; H, CHF 2, H, Br, S, OMe, H, H, H, O], [AC9046; H, CHF 2, H, Br, S , OEt, H, H, H, O], [AC 9047; H, CHF ₂ , H, Br, S, Oi-Pr, H, H, H, O], [AC 9048; H, CHF ₂ , H, Br , S, SMe, H, H, H, O], [AC 9049; H, CHF ₂ , H, Br, S, S Et, H, H, H, O], [AC9050; H, CHF 2, H, Br, S, CH 2 F, H, H, H, O], [AC9051; H, CHF 2, H, Br, _{S, CHF 2, H, H} , H, O], [AC9052; H, CHF 2, H, Br, S, CF 3, H, H, H, O], [AC9053; H, CHF 2, H, _{Br, S, OCH 2 F,} H, H, H, O], [AC9054; H, CHF 2, H, Br, S, OCHF 2, H, H, H, O], [AC9055; H, CHF 2 , H, Br, S, OCF 3, H, H, H, O], [AC9056; H, CHF 2, H, Br, S, SCH 2 F, H, H, H, O], [AC9057; H , CHF ₂ , H, Br, S, SCHF ₂ , H, H, H, O], [AC 9058; H, CHF ₂ , H, Br, S, SCF ₃ , H, H, H, O], [AC 9059 H, CHF ₂ , H, Br, S, CN, H, H, H, O], [AC 9060; H, CHF ₂ , H, Br, S, NO ₂ , H, H, H, O], [, _{AC9061; H, CF 3, H} , H, S, H, H, H, H, O], [AC9062; H, CF 3, H, H, S, F, H, H, H, O], [ _{AC9063; H, CF 3, H} , H, S, Cl, H, H, H, O], [AC9064; H, CF 3, H, H, S, Br, H, H, H, O], [ _{AC9065; H, CF 3, H} , H, S, I, H, H, H, O], [AC9066; H, CF 3, H, H, S, Me, H, H, H, O], [ _{AC9067; H, CF 3, H} , H, S, Et, H, H, H, O], [AC9068; H, CF 3, H, H, S, Pr, H, H, H, O], [ AC 9069; H, CF ₃ , H, H, S, i-Pr, H, H, H, O],

_{[AC9070; H, CF 3,} H, H, S, CH = CH 2, H, H, H, O], [AC9071; H, CF 3, H, H, S, C (CH 3) = CH 2 , H, H, H, O ], [AC9072; H, CF 3, H, H, S, C≡CH, H, H, H, O], [AC9073; H, CF 3, H, H, S , CCFCCH ₃ , H, H, H, O], [AC 9074; H, CF ₃ , H, H, S, c-Pr, H, H, H, O], [AC 9075; H, CF ₃ , H, H, S, OMe, H, H, H, O], [AC 9076; H, CF ₃ , H, H, S, OE t, H, H, H, O], [AC 9077; H, CF ₃ , H, H, S, Oi- Pr, H, H, H, O], [AC9078; H, CF 3, H, H, S, SMe, H, H, H, O], [AC9079; H, CF ₃ , H, H, H, S, SEt, H, H, H, O], [AC 9080; H, CF ₃ , H, H, S, CH ₂ F, H, H, O], [AC9081; H , CF ₃ , H, H, S, CHF ₂ , H, H, H, O], [AC 908 2; H, CF ₃ , H, H, S, CF ₃ , H, H, O], [AC 9083 _{; H, CF 3, H,} H, S, OCH 2 F, H, H, H, O], [AC9084; H, CF 3, H, H, S, OCHF 2, H, H, H, O] , [AC 9085; H, CF ₃ , H, H, S, OCF ₃ , H, H, H, O], [AC 9086; H, CF ₃ , H, H, S, SCH ₂ F, H, H, H H, CF ₃ , H, H, S, SCHF ₂ , H, H, H, O], [AC 9088; H, CF ₃ , H, H, S, SCF ₃ , H, H , H, O], [AC9089 ; H, CF 3, H, H, S, CN, H, H, H, O], [AC9090; H, CF 3, H, H, S, NO 2, H, H, H, O], [ AC9091; H, CF 3, H, Me, S, H, H, H, H, O], [AC9092; H, CF 3, H, Me, S, F, H, H, H, O], [ AC9093; H, CF 3, H, Me, S, Cl, H, H, H, O], [AC9094; H, CF 3, H, Me, S, Br, H, H, H, O], [ AC9095; H, CF 3, H, Me, S, I, H, H, H, O], [AC9096; H, CF 3, H, Me, S, Me, H, H, H, O ], [AC9097; H, CF 3, H, Me, S, Et, H, H, H, O], [AC9098; H, CF 3, H, Me, S, Pr, H, H, H, O H, CF ₃ , H, Me, S, i-Pr, H, H, H, O], [AC 9100; H, CF ₃ , H, Me, S, CH = CH ₂ , H, H, H, O], [AC 9101; H, CF ₃ , H, Me, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC 9102; H, CF ₃ , H, Me , S, C≡CH, H, H, H, O, [AC 9103; H, CF ₃ , H, Me, S, C≡CCH ₃ , H, H, H, O], [AC 9104; H, CF _{3, H, Me, S,} c-Pr, H, H, H, O], [AC9105; H, CF 3, H, Me, S, OMe, H, H, H, O], [AC9106; H , CF ₃ , H, Me, S, OEt, H, H, H, O], [AC 9107; H, CF ₃ , H, Me, S, Oi-Pr, H, H, H, O], [AC 9108 H, CF ₃ , H, Me, S, SMe, H, H, H, O], [AC 9109; H, CF ₃ , H, Me, S, SE t, H, H, H, O], [AC 9110 _{; H, CF 3, H,} Me, S, CH 2 F, H, H, H, O], [AC9111; H, CF 3, H, Me, S, CHF 2, H, H, H, O] _{, [AC9112; H, CF 3} , H, Me, S, CF 3, H, H, H, O], [AC9113; H, CF 3, H, Me, S, OCH 2 F, H, H, H , O], [AC 9114; H, CF ₃ , H, Me, S, OCHF ₂ , H, H, H, O], [AC 9115; H, CF ₃ , H, Me, S, OCF ₃ , H, H , H, O], [AC 9116; H, CF ₃ , H, Me, S, SCH ₂ F, H, H, H, O], [AC 9117; H, CF ₃ , H, Me, S, SCHF ₂ , H, H, H, O], [AC 9118; H, CF ₃ , H, Me, S, SCF ₃ , H, H, H, O], [AC 9119; H, CF ₃ , H, Me, S, CN , H, H, H, O ], [AC9120; H, CF 3, H, Me, S, NO 2, H, H, H, O], [AC9121; H, CF 3, H, Et, S, H, H, H, H, O], [AC9122; H, CF 3, H, Et, S, F, H, H, H, O], [AC9123 H, CF ₃ , H, Et, S, Cl, H, H, H, O], [AC9124; H, CF ₃ , H, Et, S, Br, H, H, H, O], [AC 9125 H, CF ₃ , H, Et, S, I, H, H, H, O], [AC 9126; H, CF ₃ , H, Et, S, Me, H, H, H, O], [AC 9127 H, CF ₃ , H, Et, S, Et, H, H, O], [AC 9128; H, CF ₃ , H, Et, S, Pr, H, H, H, O], [AC 9129 H, CF ₃ , H, Et, S, i-Pr, H, H, H, O], [AC 9130; H, CF ₃ , H, Et, S, CH = CH ₂ , H, H, H, H O], [AC9131; H, CF 3, H, Et, S, C (CH 3) = CH 2, H, H, H, O], [AC9132; H, CF 3, H, Et, S, C ≡CH, H, H, H, O], [AC9133; H, CF ₃ , H, Et, S, C≡CCH ₃ , H, H, H, O], [AC9134; H, CF ₃ , H, Et, S, c-Pr, H, H, H, H, O], [AC 9135; H, CF ₃ , H, Et, S, OMe, H, H, H, O], [AC 9136; H, CF ₃ , H, Et, S, OEt, H, H, H, O], [AC 9137; H, CF ₃ , H, Et, S, Oi-Pr, H, H, H, O], [AC 9138; H, CF ₃ , H, Et, S, SMe, H, H, H, O], [AC 9139; H, CF ₃ , H, Et, S, SE t, H, H, H, O], [AC 9140; H, CF _{3, H, Et, S,} CH 2 F, H, H, H, O], [AC9141; H, CF 3, H, Et, S, CHF 2, H, H, H, O], [AC9142; _{H, CF 3, H, Et} , S, CF 3, H, H, H, O], [AC9143; H, CF 3, H, Et, S, OCH 2 F, H, H, H, O], _{[AC9144; H, CF 3,} H, Et, S, OCHF 2, H, H, H, O], [AC9145; H, CF 3, H, Et, S, OCF 3, H, H, H, O H, CF ₃ , H, Et, S, SCH ₂ F, H, H, H, O], [AC 9147; H, CF ₃ , H, Et, S, SCHF ₂ , H, H, H] H, O], [AC 9148; H, CF ₃ , H, Et, S, SCF ₃ , H, H, H, O], [AC 9149; H, CF ₃ , H, H, Et, S, CN, H, H, H, O], [AC9150; H, CF 3, H, Et, S, NO 2, H, H, H, O], [AC9151; H, CF 3, H , Pr, S, H, H , H, H, O], [AC9152; H, CF 3, H, Pr, S, F, H, H, H, O], [AC9153; H, CF 3, H , Pr, S, Cl, H , H, H, O], [AC9154; H, CF 3, H, Pr, S, Br, H, H, H, O], [AC9155; H, CF 3, H , Pr, S, I, H, H, H, O], [AC 9156; H, CF ₃ , H, Pr, S, Me, H, H, H, O], [AC 9157; H, CF ₃ , H , Pr, S, Et, H , H, H, O], [AC9158; H, CF 3, H, Pr, S, Pr, H, H, H, O], [AC9159; H, CF 3, H , Pr, S, i-Pr , H, H, H, O], [AC9160; H, CF 3, H, Pr, S, CH = CH 2, H, H, H, O], [AC9161; H , CF ₃ , H, Pr, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AC9162; H, CF ₃ , H, Pr, S, C≡CH, H, H, H H, O], [AC9163; H, CF 3, H, Pr, S, C≡CCH 3, H, H, H, O], [AC9164; H, CF 3, H, Pr, S, c-Pr , H, H, H, O ], [AC9165; H, CF 3, H, Pr, S, OMe, H, H, H, O], [AC9166; H, CF 3, H, Pr, S, OEt , H, H, H, O], [AC 9167; H, CF ₃ , H, Pr, S, Oi-Pr, H, H, H, O], [AC 9168; H, CF ₃ , H, Pr, S , SMe, H, H, H, O], [AC9169; H, CF ₃ , H, Pr, S, SEt, H, H, H, O],

_{[AC9170; H, CF 3,} H, Pr, S, CH 2 F, H, H, H, O], [AC9171; H, CF 3, H, Pr, S, CHF 2, H, H, H, O], [AC9172; H, CF 3, H, Pr, S, CF 3, H, H, H, O], [AC9173; H, CF 3, H, Pr, S, OCH 2 F, H, H , H, O], [AC9174 ; H, CF 3, H, Pr, S, OCHF 2, H, H, H, O], [AC9175; H, CF 3, H, Pr, S, OCF 3, H , H, H, O], [AC 9176; H, CF ₃ , H, Pr, S, SCH ₂ F, H, H, H, O], [AC 9177; H, CF ₃ , H, Pr, S, SCHF ₂ , H, H, H, O], [AC 9178; H, CF ₃ , H, Pr, S, SCF ₃ , H, H, H, O], [AC 9179; H, CF ₃ , H, Pr, S , CN, H, H, H , O], [AC9180; H, CF 3, H, Pr, S, NO 2, H, H, H, O], [AC9181; H, CF 3, H, i- Pr, S, H, H, H, H, O], [AC9182; H, CF 3, H, i-Pr, S, F, H, H, H, O], [AC9183; H, CF 3, H, i-Pr, S, Cl, H, H, H, O], [AC9184; H, CF 3, H, i-Pr, S, Br, H, H, H, O], [AC9185; H _{, CF 3, H, i-} Pr, S, I, H, H, H, O], [AC9186; H, CF 3, H, i-Pr, S, Me, H, H, H, O], _{[AC9187; H, CF 3,} H, i-Pr, S, Et, H, H, H, O], [AC9188; H, CF 3, H, i-Pr, S, Pr, H, H, H , O], [AC9189; H , CF 3, H, i-Pr, S, i-Pr, H, H, H, O], [AC9190; H, CF 3, H, i-Pr, S, CH _{= CH 2, H, H,} H, O], [AC9191; H, CF 3, H, i-Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC9192; _{H, CF 3, H, i} -Pr, S, C≡CH, H, H, H, O], [AC9193; H, CF 3, H, i-Pr, S, C≡CCH 3, H, H , H, O], [AC9194 ; H, CF 3, H, i-Pr, S, c-Pr, H, H, H, O], [AC9195; H, CF 3, H, i-Pr, S , OMe, H, H, H, O], [AC 9196; H, CF ₃ , H, i-Pr, S, OEt, H, H, H, O], [AC9197; H, CF ₃ , H, i -Pr, S, Oi-Pr, H, H, H, O], [AC9198; H, CF 3, H, i-Pr, S, SMe, H, H, H, O], [AC9199; H, _{CF 3, H, i-Pr} , S, SEt, H, H, H, O], [AC9200; H, CF 3, H, i-Pr, S, CH 2 F, H, H, H, O] _{, [AC9201; H, CF 3} , H, i-Pr, S, CHF 2, H, H, H, O], [AC9202; H, CF 3, H, i-Pr, S, CF 3, H, H, H, O], [ AC9203; H, CF 3, H, i-Pr, S, OCH 2 F, H, H, H, O], [AC9204; H, CF 3, H, i-Pr, S, OCHF ₂ , H, H, H, O], [AC 9205; H, CF ₃ , H, i-Pr, S, OCF ₃ , H, H, H, O], [AC 9206; H, CF ₃ , H, i-Pr, S, SCH ₂ F, H, H, H, O], [AC 9207; H, CF ₃ , H, i-Pr, S, SCHF ₂ , H, H, H, O], [[ AC 9208; H, CF ₃ , H, i-Pr, S, SCF ₃ , H, H, H, O], [AC 9209; H, CF ₃ , H, i-Pr, S, CN, H, H, H , O], [AC9210; H , CF 3, H, i-Pr, S, NO 2, H, H, H, O], [AC9211; H, CF 3, H, c-Pr, S, H, H, H, H, O] , [AC9212; H, CF 3, H, c-Pr, S, F, H, H, H, O], [AC9213; H, CF 3, H, c-Pr, S, Cl, H, H, H, O], [AC 9214; H, CF ₃ , H, c-Pr, S, Br, H, H, H, O], [AC 9215; H, CF ₃ , H, c-Pr, S, I, H, H, H, O], [AC9216; H, CF 3, H, c-Pr, S, Me, H, H, H, O], [AC9217; H, CF ₃ , H, c-Pr, S, Et, H, H, H, O], [AC 9218; H, CF ₃ , H, c-Pr, S, Pr, H, H, H, O], [AC 9219 H, CF ₃ , H, c-Pr, S, i-Pr, H, H, H, O], [AC9220; H, CF ₃ , H, c-Pr, S, CH 2CH ₂ , H, H, H, H, O], [AC9221; _{H, CF 3, H, c} -Pr, S, C (CH 3) = CH 2, H, H, H, O], [AC9222; H, CF 3, H, c-Pr, S, C≡CH , H, H, H, O ], [AC9223; H, CF 3, H, c-Pr, S, C≡CCH 3, H, H, H, O], [AC9224; H, CF 3, H, c-Pr, S, c- Pr, H, H, H, O], [AC9225; H, CF 3, H, c-Pr, S, OMe, H, H, H, O], [AC9226; H _{, CF 3, H, c-} Pr, S, OEt, H, H, H, O], [AC9227; H, CF 3, H, c-Pr, S, Oi-Pr, H, H, H, O ], [AC9228; H, CF 3, H, c-Pr, S, SMe, H, H, H, O], [AC9229; H, CF 3, H, c-Pr, S, SEt, H, H , H, O], [AC9230 ; H, CF 3, H, c-Pr, S, CH 2 F, H, H, H, O], [AC9231; H, CF 3, H, c-Pr, S _{, CHF 2, H, H,} H, O], [AC9232; H, CF 3, H, c-Pr, S, CF 3, H, H, H, O], [AC9233; H, CF 3, H , c-Pr, S, OCH 2 F, H, H, H, O], [AC9234; H, CF 3, H, c-Pr, S, OCHF 2, H, H, H, O], [AC9235 H, CF ₃ , H, c-Pr, S, OCF ₃ , H, H, H, O], [AC 9236; H, CF ₃ , H, c-Pr, S, SCH ₂ F, H, H, H, O], [AC9237; H, CF 3, H, c-Pr, S, SCHF 2, H, H, H, O], [AC9238; H, CF 3, H, c-Pr, S, SCF ₃ , H, H, H, O], [AC 9239; H, CF ₃ , H, c-Pr, S, CN, H, H, H, O], [AC 9240; H, CF ₃ , H, c- _{Pr, S, NO 2, H} , H, H, O], [AC9241; H, CF 3, H, SMe, S, H, H, H, H, O], [AC9242; H, CF 3, H , SMe, S, F, H , H, H, O], [AC9243; H, CF 3, H, SMe, S, Cl, H, H, H, O], [AC9244; H, CF 3, H , SMe, S, Br, H , H, H, O], [AC9245; H, CF 3, H, SMe, S, I, H, H, H, O], [AC9246; H, CF 3, H, SMe, S, Me, H, H, H, O], [AC9247; H, CF 3, H, SMe, S, Et, H, H, H, O], [AC9248; H, CF 3, H, SMe, S, Pr, H, H, H, O], [AC 9249; H, CF ₃ , H, SMe, S, i-Pr, H, H, H, O], [AC 9250; H, CF _{3, H, SMe, S,} CH = CH 2, H, H, H, O], [AC9251; H, CF 3, H, SMe, S, C (CH 3) = CH 2, H, H, H , O], [AC9252; H , CF 3, H, SMe, S, C≡CH, H, H, H, O], [AC9253; H, CF 3, H, SMe, S, C≡CCH 3, H, H, H, O] , [AC9254; H, CF 3, H, SMe, S, c-Pr, H, H, H, O], [AC9255; H, CF 3, H, SMe, S, OMe, H, H, H, O], [AC9256; H, CF 3, H, SMe, S, OEt, H, H, H, O], [AC9257; H, CF 3, H, SMe, S, Oi-Pr, H, H, H, O], [AC9258; H, CF 3, H, SMe, S, SMe, H, H, H, O], [AC9259; H, CF 3, H, SMe, S, SEt, H, H, H, O], [AC9260; H, CF 3, H, SMe, S, CH 2 F, H, H, H, O], [AC9261; H, CF 3, H, _{SMe, S, CHF 2, H} , H, H, O], [AC9262; H, CF 3, H, SMe, S, CF 3, H, H, H, O], [AC9263; H, CF 3, _{H, SMe, S, OCH 2} F, H, H, H, O], [AC9264; H, CF 3, H, SMe, S, OCHF 2, H, H, H, O], [AC9265; H, _{CF 3, H, SMe, S} , OCF 3, H, H, H, O], [AC9266; H, CF 3, H, SMe, S, SCH 2 F, H, H, H, O], [AC9267 _{; H, CF 3, H,} SMe, S, SCHF 2, H, H, H, O], [AC9268; H, CF 3, H, SMe, S, SCF 3, H, H, H, O], _{[AC9269; H, CF 3,} H, SMe, S, CN, H, H, H, O],

_{[AC9270; H, CF 3,} H, SMe, S, NO 2, H, H, H, O], [AC9271; H, CF 3, H, OMe, S, H, H, H, H, O] [AC 927 2; H, CF ₃ , H, OMe, S, F, H, H, H, O], [AC 927 ₃ ; H, CF ₃ , H, OMe, S, Cl, H, H, H, O] [AC 9274; H, CF ₃ , H, OMe, S, Br, H, H, O], [AC 9275; H, CF ₃ , H, OMe, S, I, H, H, H, O] _{, [AC9276; H, CF 3} , H, OMe, S, Me, H, H, H, O], [AC9277; H, CF 3, H, OMe, S, Et, H, H, H, O] _{, [AC9278; H, CF 3} , H, OMe, S, Pr, H, H, H, O], [AC9279; H, CF 3, H, OMe, S, i-Pr, H, H, H, O], [AC9280; H, CF 3, H, OMe, S, CH = CH 2, H, H, H, O], [AC9281; H, CF 3, H, OMe, S, C (CH 3) _{= CH 2, H, H,} H, O], [AC9282; H, CF 3, H, OMe, S, C≡CH, H, H, H, O], [AC9283; H, CF 3, H, OMe, S, C≡CCH ₃ , H, H, H, O], [AC9284; H, CF ₃ , H, OMe, S, c-Pr, H, H, H, O], [AC9285; H, _{CF 3, H, OMe, S} , OMe, H, H, H, O], [AC9286; H, CF 3, H, OMe, S, OEt, H, H, H, O], [AC9287; H, _{CF 3, H, OMe, S} , Oi-Pr, H, H, H, O], [AC9288; H, CF 3, H, OMe, S, SMe, H, H, H, O], [AC9289; _{H, CF 3, H, OMe} , S, SEt, H, H, H, O], [AC9290; H, CF 3, H, OMe, S, CH 2 F, H, H, H, O], [ _{AC9291; H, CF 3, H} , OMe, S, CHF 2, H, H, H, O], [AC9292; H, CF 3, H, OMe, S, CF 3, H, H, H, O] _{, [AC9293; H, CF 3} , H, OMe, S, OCH 2 F, H, H, H, O], [AC9294; H, CF 3, H, OMe, S, OCHF 2, H, H, H , O], [AC9295; H , CF 3, H, OMe, S, OCF 3, H, H, H, O ], [AC9296; H, CF 3, H, OMe, S, SCH 2 F, H, H, H, O], [AC9297; H, CF 3, H, OMe, S, SCHF 2, H, H, H, O], [AC9298; H, CF 3, H, OMe, S, SCF 3, H, H, H, O], [AC9299; H, CF 3, H, OMe, S, CN, H, H , H, O], [AC9300 ; H, CF 3, H, OMe, S, NO 2, H, H, H, O], [AC9301; H, CF 3, H, F, S, H, H, H, H, O], [ AC9302; H, CF 3, H, F, S, F, H, H, H, O], [AC9303; H, CF 3, H, F, S, Cl, H, H, H, O], [ AC9304; H, CF 3, H, F, S, Br, H, H, H, O], [AC9305; H, CF 3, H, F, S, I, H, H, H, O], [ AC9306; H, CF 3, H, F, S, Me, H, H, H, O], [AC9307; H, CF 3, H, F, S, Et, H, H, H, O], [AC 9308; H, CF ₃ , H, F, S, Pr, H, H, H, O], [AC 9309; H, CF ₃ , H, F, S, i-Pr, H, H, H, O] , [AC9310; H, CF 3, H, F, S, CH = CH 2, H, H, H, O], [AC9311; H, CF 3, H, F, S _{, C (CH 3) = CH} 2, H, H, H, O], [AC9312; H, CF 3, H, F, S, C≡CH, H, H, H, O], [AC9313; H , CF ₃ , H, F, S, C≡CCH ₃ , H, H, H, O], [AC 9314; H, CF ₃ , H, F, S, c-Pr, H, H, H, O] _{, [AC9315; H, CF 3} , H, F, S, OMe, H, H, H, O], [AC9316; H, CF 3, H, F, S, OEt, H, H, H, O] _{, [AC9317; H, CF 3} , H, F, S, Oi-Pr, H, H, H, O], [AC9318; H, CF 3, H, F, S, SMe, H, H, H, O], [AC9319; H, CF 3, H, F, S, SEt, H, H, H, O], [AC9320; H, CF 3, H, F, S, CH 2 F, H, H, H, O], [AC9321; H, CF 3, H, F, S, CHF 2, H, H, H, O], [AC9322; H, CF 3, H, F, S, CF 3, H, H, H, O], [AC9 _{323; H, CF 3, H} , F, S, OCH 2 F, H, H, H, O], [AC9324; H, CF 3, H, F, S, OCHF 2, H, H, H, O H, CF ₃ , H, F, S, OCF ₃ , H, H, H, O], [AC 9326; H, CF ₃ , H, F, S, SCH ₂ F, H, H, H, O], [AC9327; H, CF 3, H, F, S, SCHF 2, H, H, H, O], [AC9328; H, CF 3, H, F, S, SCF 3, H, H, H, O], [ AC9329; H, CF 3, H, F, S, CN, H, H, H, O], [AC9330; H, CF 3, H, F, S, NO 2, H , H, H, O], [AC9331; H, CF 3, H, Cl, S, H, H, H, H, O], [AC9332; H, CF 3, H, Cl, S, F, H , H, H, O], [AC9333; H, CF 3, H, Cl, S, Cl, H, H, H, O], [AC9334; H, CF 3, H, Cl, S, Br, H , H, H, O], [AC9335; H, CF 3, H, Cl, S, I, H, H, H, O], [AC9336; H, CF 3, H, Cl, S, Me, H , H, H, O], [AC9337; H, CF 3, H, Cl, S, Et, H, H, H, O], [AC9338; H, CF 3, H, Cl, S, Pr, H , H, H, O], [AC9339; H, CF 3, H, Cl, S, i-Pr, H, H, H, O], [AC9340; H, CF 3, H, Cl, S, CH _{= CH 2, H, H,} H, O], [AC9341; H, CF 3, H, Cl, S, C (CH 3) = CH 2, H, H, H, O], [AC9342; H, _{CF 3, H, Cl, S} , C≡CH, H, H, H, O], [AC9343; H, CF 3, H, Cl, S, C≡CCH 3, H, H, H, O], [AC 9344; H, CF ₃ , H, Cl, S, c-Pr, H, H, H, O], [AC 9345; H, CF ₃ , H, Cl, S, OMe, H, H, H, O ], [AC9346; H, CF 3, H, Cl, S, OEt, H, H, H, O], [AC9347; H, CF 3, H, Cl, S, Oi-Pr, H, H, H , O], [AC9348; H , CF 3, H, Cl, S, SMe, H, H, H, O], [AC9349; H, CF 3, H, Cl, S, SEt, H, H, H , O ], [AC9350; H, CF 3, H, Cl, S, CH 2 F, H, H, H, O], [AC9351; H, CF 3, H, Cl, S, CHF 2, H, H, H, O], [AC9352; H, CF 3, H, Cl, S, CF 3, H, H, H, O], [AC9353; H, CF 3, H, Cl, S, OCH 2 F, H , H, H, O], [AC9354; H, CF 3, H, Cl, S, OCHF 2, H, H, H, O], [AC9355; H, CF 3, H, Cl, S, OCF 3 , H, H, H, O], [AC 9356; H, CF ₃ , H, Cl, S, SCH ₂ F, H, H, H, O], [AC 9357; H, CF ₃ , H, Cl, S , SCHF ₂ , H, H, H, O], [AC 9358; H, CF ₃ , H, Cl, S, SCF ₃ , H, H, H, O], [AC 9359; H, CF ₃ , H, Cl , S, CN, H, H, H, O], [AC 9360; H, CF ₃ , H, Cl, S, NO ₂ , H, H, H, O], [AC 9361; H, CF ₃ , H, Br, S, H, H, H, H, O], [AC9362; H, CF 3, H, Br, S, F, H, H, H, O], [AC9363; H, CF 3, H, Br, S, Cl, H, H, H, O], [AC 9364; H, CF ₃ , H, Br, S, Br, H, H, H, O], [AC 9365; H, CF ₃ , H, Br, S, I, H, H, H, O], [AC9366; H, CF 3, H, Br, S, Me, H, H, H, O], [AC9367; H, CF 3, H, Br, S, Et, H, H, H, O], [AC9368; H, CF 3, H, Br, S, Pr, H, H, H, O],

_{[AC9369; H, CF 3,} H, Br, S, i-Pr, H, H, H, O], [AC9370; H, CF 3, H, Br, S, CH = CH 2, H, H, H, O], [AC9371; H, CF 3, H, Br, S, C (CH 3) = CH 2, H, H, H, O], [AC9372; H, CF 3, H, Br, S , C≡CH, H, H, H, O], [AC9373; H, CF ₃ , H, Br, S, C≡CCH ₃ , H, H, H, O], [AC 9374; H, CF ₃ , H, Br, S, c- Pr, H, H, H, O], [AC9375; H, CF 3, H, Br, S, OMe, H, H, H, O], [AC9376; H, CF _{3, H, Br, S,} OEt, H, H, H, O], [AC9377; H, CF 3, H, Br, S, Oi-Pr, H, H, H, O], [AC9378; H _{, CF 3, H, Br,} S, SMe, H, H, H, O], [AC9379; H, CF 3, H, Br, S, SEt, H, H, H, O], [AC9380; H , CF ₃ , H, Br, S, CH ₂ F, H, H, H, O], [AC 9381; H, CF ₃ , H, Br, S, CHF ₂ , H, H, H, O], [[ AC 9382; H, CF ₃ , H, Br, S, CF ₃ , H, H, H, O], [AC 9383; H, CF ₃ , H, Br, S, OCH ₂ F, H, H, H, O H, CF ₃ , H, Br, S, OCHF ₂ , H, H, H, O], [AC 9385; H, CF ₃ , H, Br, S, OCF ₃ , H, H, H] , O], [AC9386; H , CF 3, H, Br, S, SCH 2 F, H, H, H, O], [AC9387; H, CF 3, H, Br, S, SCHF 2, H, H, H, O], [ AC9388; H, CF 3, H, Br, S, SCF 3, H, H, H, O], [AC9389; H, CF 3, H, Br, S, CN, H , H, H, O], [AC9390; H, CF 3, H, Br, S, NO 2, H, H, H, O], [AC9391; F, H, H, H, S, H, H , H, H, O], [AC9392; F, H, H, H, S, F, H, H, H, O], [AC9393; F, H, H, H, S, Cl, H, H , H, O], [AC9394; F, H, H, H, S, Br, H, H, H, O], [AC9395; F, H, H, H, S, I, H, H, H , O], [AC9396; F, H, H, H, H, S, Me, H, H, H, O], [AC9397; F, H, H, H, S, Et, H, H, H, O], [AC9398 F, H, H, H, H, S, Pr, H, H, H, O], [AC9399; F, H, H, H, S, i-Pr, H, H, H, O], [AC 9400 ; F, H, H, H , S, CH = CH 2, H, H, H, O], [AC9401; F, H, H, H, S, C (CH 3) = CH 2, H, H , H, O], [AC9402; F, H, H, H, S, C≡CH, H, H, H, O], [AC9403; F, H, H, H, S, C≡ CCH ₃ , H, H, H, O], [AC 9404; F, H, H, H, S, c-Pr, H, H, H, O], [AC 9405; F, H, H, H, S, OMe, H, H, H, O], [AC 9406; F, H, H, H, S, OEt, H, H, H, O], [AC 9407; F, H, H, H, S, Oi-Pr, H, H, H, O], [AC 9408; F, H, H, H, S, S Me, H, H, H, O], [AC 9409; F, H, H, H, S, SE t, H, H, H, O], [AC 9410; F, H, H, H, S, CH ₂ F, H, H, H, O], [AC 9411; F, H, H, H, S, CHF ₂ , H , H, H, O], [AC9412; F, H, H, H, S, CF 3, H, H, H, O], [AC9413; F, H, H, H, S, OCH 2 F, H, H, H, O], [AC 9414; F, H, H, H, S, OCHF ₂ , H, H, H, O], [AC 9415; F, H, H, H, S, OCF ₃ , H, H, H, O], [AC 9416; F, H, H, H, S, SCH ₂ F, H, H, H, O], [AC 9417; F, H, H, H, S, SCHF ₂ , H, H, H, O ], [AC9418; F, H, H, H, S, SCF 3, H, H, H, O], [AC9419; F, H, H, H, S, CN, H, H, H, O] , [AC9420; F, H, H, H, S, NO 2, H, H, H, O], [AC9421; F, H, H, Me, S, H, H , H, H, O], [AC9422; F, H, H, Me, S, F, H, H, H, O], [AC 9423; F, H, H, Me, S, Cl, H, H , H, O], [AC9424; F, H, H, Me, S, Br, H, H, H, O], [AC 9425; F, H, H, Me, S, I, H, H, H , O], [AC 9426; F, H, H, M e, S, Me, H, H, H, O], [AC 9427; F, H, H, Me, S, Et, H, H, H, O], [AC 9428; F, H, H, Me, S, Pr, H, H, H, O], [AC9429; F, H, H, Me, S, i-Pr, H, H, H, O], [AC9430; F, H, H, Me, _{S, CH = CH 2, H} , H, H, O], [AC9431; F, H, H, Me, S, C (CH 3) = CH 2, H, H, H, O], [AC9432; F, H, H, Me, S, C≡CH, H, H, H, O], [AC 9433; F, H, H, Me, S, C≡ CCH ₃ , H, H, H, O], [AC9434; F, H, H, Me, S, c-Pr, H, H, H, O], [AC 9435; F, H, H, Me, S, OMe, H, H, H, O], [AC9436; F, H, H, Me, S, OEt, H, H, H, O], [AC 9437; F, H, H, Me, S, Oi-Pr, H, H, H, O], [AC9438; F, H, H, Me, S, SMe, H, H, H, O], [AC9439; F, H, H, Me, S, SE t, H, H, H, O], [AC9440 ; F, H, H, Me , S, CH 2 F, H, H, H, O], [AC9441; F, H, H, Me, S, CHF 2, H, H, H, O], [ AC9442; F, H, H, Me, S, CF 3, H, H, H, O], [AC9443; F, H, H, Me, S, OCH 2 F, H, H, H, O], [AC 9444; F, H, H, Me, S, OCHF ₂ , H, H, H, O], [AC 9445; F, H, H, Me, S, OCF ₃ , H, H, H, O], [AC 9446; F, H, H, Me, S, SCH ₂ F, H, H, H, O], [AC 9447; F, H, H, Me, S, SCHF ₂ , H, H, H, O] , [AC 9448; F, H, H, Me, S, SCF ₃ , H, H, H, O], [AC 9449; F, H, H, Me, S, CN, H, H, H, O], [AC 9450; F, H, H, Me, S, NO ₂ , H, H, H, O], [AC 9451; F, Me, H, Me, S, H, H, H, O], [AC AC9452; F, Me, H, Me, S, F, H, H, O], [AC9453; F, Me, H, Me, S, Cl, H, H, H, O], [AC9454; F, Me, H, Me, S, Br, H, H, H, O], [AC9455; F, Me, H, Me, S, I, H, H, O], [AC 9456; F, Me, H, Me, S, Me, H, H, H, O], [AC 9457; F, Me, H, Me, S, Et, H, H, H, O], [AC 9458 F, Me, H, Me, S, Pr, H, H, H, O], [AC 9459; F, Me, H, Me, S, i-Pr, H, H, H, O], [AC 9460] F, Me, H, Me, S, CH = CH ₂ , H, H, H, O], [AC9461; F, Me, H, Me, S, C (CH ₃ ) = CH ₂ , H, H , H, O], [AC9462; F, Me, H, Me, S, C≡CH, H, H, H, O], [AC9463; F, Me, H, Me, S, C≡CCH ₃ , H, H, H, O], [AC9464; F, Me, H, Me, S, c-Pr, H, H, H, O], [AC9465; F, Me, H, Me, S, OMe, H, H, H, O], [AC 9466; F, Me, H, Me, S, OEt, H, H, H, O], [AC 9467; F, Me, H, Me, S, Oi-Pr, H, H, H, O], [AC 9468; F, Me, H, Me, S, SMe, H, H, H, O],

[AC9469; F, Me, H , Me, S, SEt, H, H, H, O], [AC9470; F, Me, H, Me, S, CH 2 F, H, H, H, O], [AC9471; F, Me, H , Me, S, CHF 2, H, H, H, O], [AC9472; F, Me, H, Me, S, CF 3, H, H, H, O], [AC 9473; F, Me, H, Me, S, OCH ₂ F, H, H, H, O], [AC 9474; F, Me, H, Me, S, OCHF ₂ , H, H, H, O] , [AC9475; F, Me, H, Me, S, OCF 3, H, H, H, O], [AC9476; F, Me, H, Me, S, SCH 2 F, H, H, H, O F, Me, H, Me, S, SCHF ₂ , H, H, H, O], [AC 9478; F, Me, H, Me, S, SCF ₃ , H, H, H, O] F, Me, H, Me, S, CN, H, H, H, O], [AC 9480; F, Me, H, Me, S, NO ₂ , H, H, H, O] [AC9481; H, H, F, H, S, H, H, H, O], [AC9482; H, H, F, H, S, F, H, H, O], [AC9482; AC 9483; H, H, F, H, S, Cl, H, H, H, O], [AC9484; H, H, F, H, S, Br, H, H, O], [AC 9485; H, H, F, H, S, I, H, H, H, O], [AC9486; H, H, F, H, S, Me, H, H, O], [AC 9487; H, H, F, H, S, Et, H, H, H, O], [AC 9488; H, H, F, H, S, Pr, H, H, O], [AC 9489; H, H, F, H, S, i- Pr, H, H, H, O], [AC9490; H, H, F, H, S, CH = CH 2, H, H, H, O], [AC9491; H , H, F, H, S , C (CH 3) = CH 2, H, H, H, O], [AC9492; H, H, F, H, S, C≡CH, H, H, H, O], [AC9493; H, H, F, H, S, C≡CCH ₃ , H, H, H, O], [AC9494; H, H, F, H, S, c-Pr, H, H , H, O], [AC 9495; H, H, F, H, S, OMe, H, H, H, O], [AC 9496; H, H, F, H, S, OE t, H, H, H H, H, F, H, S, Oi-Pr, H, H, H, O], [AC 9498; H, H, F, H, S, SMe, H, H, H , O], [AC9499; H, H, F, H, S, SEt, H, H, H, O], [AC 9500; H, H, F, H, S, CH ₂ F, H, H, H , O], [AC9501; H , H, F, H, S, CHF 2, H, H, H, O], [AC9502; H, H, F, H, S, CF 3, H, H, H , O], [AC9503; H , H, F, H, S, OCH 2 F, H, H, H, O], [AC9504; H, H, F, H, S, OCHF 2, H, H, H, O], [AC9505; H, H, F, H, S, OCF 3, H, H, H, O], [AC9506; H, H, F, H, S, SCH 2 F, H, H , H, O], [AC9507 ; H, H, F, H, S, SCHF 2, H, H, H, O], [AC9508; H, H, F, H, S, SCF 3, H, H , H, O], [AC 9509; H, H, F, H, S, CN, H, H, H, O], [AC 9510; H, H, F, H, S, NO ₂ , H, H, H, O], [AC 9511; H, H, F, Me, S, H, H, H, O], [AC 9512; H, H, F, Me, S, F, H, H, H, H, O], [AC9513; H, H, F, Me, S, Cl, H, H, O], [AC 9514; H, H, F, Me, S, Br, H, H, H, O] , [AC9515; H, H, F, Me, S, I, H, H, O], [AC 9516; H, H, F, Me, S, Me, H, H, H, O], [AC 9516; AC 9517; H, H, F, Me, S, Et, H, H, H, O], [AC 9518; H, H, F, Me, S, Pr, H, H, H, O], [AC 9519; H, H, F, Me, S, i-Pr, H, H, H, O], [AC9520; H, H, F, Me, S, CH = CH 2, H, H, H, O], [AC9521; H, H, F , Me, S, C (CH 3) = CH 2, H, H, H, O], [AC9522; H, H, F, Me, S, C≡CH, H, H, H, O], [AC 9523; H, H, F, Me, S, C≡CCH ₃ , H, H, H, O], [AC 9524; H, H, F, Me, S, c-Pr , H, H, H, O], [AC9525; H, H, F, Me, S, OMe, H, H, H, O], [AC9526; H, H, F, Me, S, OEt, H , H, H, O], [AC9527; H, H, F, Me, S, Oi-Pr, H, H, H, O], [AC 9528; H, H, F, Me, S, SMe, H , H, H, O ], [AC9529; H, H , F, Me, S, SEt, H, H, H, O], [AC9530; H, H, F, Me, S, CH 2 F, H, H, H, O ], [AC9531; H, H , F, Me, S, CHF 2, H, H, H, O], [AC9532; H, H, F, Me, S, CF 3, H, H, H, O ], [AC9533; H, H , F, Me, S, OCH 2 F, H, H, H, O], [AC9534; H, H, F, Me, S, OCHF 2, H, H, H, O], [AC9535; H, H, F, Me, S, OCF 3, H, H, H, O], [AC9536; H, H, F, Me, S, SCH 2 F, H, H, H H, H, F, Me, S, SCHF ₂ , H, H, H, O], [AC 9538; H, H, F, Me, S, SCF ₃ , H, H, H H, H, F, Me, S, CN, H, H, H, O], [AC 9540; H, H, F, Me, S, NO ₂ , H, H, H, H O], [AC 9541; H, Me, F, Me, S, H, H, H, O], [AC 9542; H, Me, F, Me, S, F, H, H, H, O] [AC 9543; H, Me, F, Me, S, Cl, H, H, H, O], [AC 9544; H, Me, F, Me, S, Br, H, H, H, O], [AC 9544; AC 9545; H, Me, F, Me, S, I, H, H, O], [AC 9546; H, Me, F, Me, S, Me, H, H, H, O], [AC 9547; H, Me, F, Me, S, Et, H, H, H, O], [AC9548; H, Me, F, Me, S, Pr, H, H, O], [AC9549; H, Me, F, Me, S, i-Pr, H, H, H, O], [AC9550; H, Me, F, Me, S, CH = CH 2, H, H, H, O], [AC9551 ; H, Me, F, Me , S, C (CH 3) = CH 2, H, H, H, O], [AC9552; H, Me, F, Me, S, C≡CH, H, H, H, O], [AC9553; H, Me, F, Me, S, C≡CCH ₃ , H, H, H, O], [AC9554; H, Me, F, Me, S, c-Pr, H H, H, O], [AC 9555; H, Me, F, Me, S, OMe, H, H, H, O], [AC 9556; H, Me, F, Me, S, OE t, H, H , H, O], [AC9557; H, Me, F, Me, S, Oi-Pr, H, H, H, O], [AC 9558; H, Me, F, Me, S, SMe, H, H, H, O], [AC9559; H, Me, F, Me, S, SE t, H, H, H, O], [AC9560; H, Me, F, Me, S, CH 2 F, H, H, H, O], [AC9561; H, Me, F, Me, S, CHF 2, H, H, H, O], [AC9562 H, Me, F, Me, S, CF ₃ , H, H, H, O], [AC 9563; H, Me, F, Me, S, OCH ₂ F, H, H, H, O], [[ AC 9564; H, Me, F, Me, S, OCHF ₂ , H, H, H, O], [AC 9565; H, Me, F, Me, S, OCF ₃ , H, H, H, O], [, AC 9566; H, Me, F, Me, S, SCH ₂ F, H, H, H, O], [AC 9567; H, Me, F, Me, S, SCHF ₂ , H, H, H, O], [AC9568; H, Me, F , Me, S, SCF 3, H, H, H, O],

[AC9569; H, Me, F , Me, S, CN, H, H, H, O], [AC9570; H, Me, F, Me, S, NO 2, H, H, H, O], [ AC9571; H, H, H, H, H, S, H, F, H, H, O], [AC9572; H, H, H, H, S, F, H, H, O], [AC9573; H, H, H, H, H, S, Cl, F, H, H, O], [AC9574; H, H, H, H, S, Br, F, H, O], [AC9575; H, H, H, H, H, S, I, F, H, H, O], [AC9576; H, H, H, H, S, Me, F, H, O], [AC 9577; H, H, H, H, S, Et, F, H, H, O], [AC9578; H, H, H, H, S, Pr, F, H, H, O], [AC 9579; H, H, H, H, S, i-Pr, F, H, H, O], [AC9580; H, H, H, H, S, CH = CH 2, F, H, H, O], [AC9581; H, H , H, H, S, C (CH 3) = CH 2, F, H, H, O], [AC9582; H, H, H, H, S, C≡CH, F, H, H, O] , [AC9583; H, H, H, H, H, S, C≡CCH ₃ , F, H, H, O], [AC 9584; H, H, H, H, S, c-Pr, F, H, H H, H, H, H, S, OMe, F, H, H, O], [AC 9586; H, H, H, H, S, OEt, F, H, H, O H, H, H, H, H, S, Oi-Pr, F, H, H, O], [AC 9588; H, H, H, H, S, SMe, F, H, H, O] H, H, H, H, H, S, SE t, F, H, H, O], [AC 9590; H, H, H, H, S, CH ₂ F, F, H, H, O] ], [AC9591; H, H , H, H, S, CHF 2, F, H, H, O], [AC9592; H, H, H, H, S, CF 3, F, H, H, O ], [AC9593; H, H , H, H, S, OCH 2 F, F, H, H, O], [AC9594; H, H, H, H, S, OCHF 2, F, H, H, O], [AC9595; H, H, H, H, S, OCF 3, F, H, H, O], [AC9596; H, H, H, H, S, SCH 2 F, F, H, H , O], [AC9597; H, H, H, H, S, SCHF ₂ , F, H, H, O], [AC 9598; H, H, H, H, S, SCF ₃ , F, H, H , O], [AC9599; H, H, H, H, S, CN, F, H, H, O], [AC 9600; H, H, H, H, S, NO ₂ , F, H, H, O], [AC9601; H, H, H, Me, S , H, F, H, H, O], [AC9602; H, H, H, Me, S, F, H, H, O], [AC9603; H, H, H, Me, S, Cl , F, H, H, O], [AC9604; H, H, H, Me, S, Br, F, H, H, O], [AC9605; H, H, H, Me, S, I, F , H, H, O], [AC9606; H, H, H, Me, S, Me, F, H, H, O], [AC 9607; H, H, H, Me, S, Et, F, H , H, O], [AC9608; H, H, H, Me, S, Pr, F, H, H, O], [AC 9609; H, H, H, Me, S, i-Pr, F, H , H, O], [AC9610 ; H, H, H, Me, S, CH = CH 2, F, H, H, O], [AC9611; H, H, H, Me, S, C (CH 3 ) = CH ₂ , F, H, H, O], [AC 9612; H, H, H, Me, S, C≡CH, F, H, H, O], [AC 9613; H, H, H, Me , S, C≡CCH ₃ , F, H, H, O], [AC 9614; H, H, H, Me, S, c-Pr, F, H, H, O], [AC 9615; H, H, H, Me, S, OMe, F, H, H, O], [AC9616; H, H, H, Me, S, OEt, F, H, H, O], [AC9617; H, H, H, Me, S, Oi-Pr, F, H, H, O], [AC9618; H, H, H, Me, S, SMe, F, H, O], [AC9619; H, H, H, Me, S, SEt, F, H, H, O], [AC9620; H, H, H, Me, S, CH 2 F, F, H, H, O], [AC9621; H, H, H, _{Me, S, CHF 2, F} , H, H, O], [AC9622; H, H, H, Me, S, CF 3, F, H, H, O], [AC9623; H, H, H, _{Me, S, OCH 2 F,} F, H, H, O], [AC9624; H, H, H, Me, S, OCHF 2, F, H, H, O], [AC9625; H, H, H _{, Me, S, OCF 3,} F, H, H, O], [AC9626; H, H, H, Me, S, SCH 2 F, F, H, H, O], [AC9627; H, H, _{H, Me, S, SCHF 2} , F, H, H, O], [AC9628; H, H, H, Me, S, SCF 3, F, H, H, O], [AC9629; H, H, H, Me, S, CN, F, H, H, O], [AC9630; H, H, H, Me, S, NO 2, F, H, H, O], [AC9631; H , Me, H, Me, S, H, F, H, H, O], [AC9632; H, Me, H, Me, S, F, H, H, O], [AC9633; H, Me , H, Me, S, Cl, F, H, H, O], [AC9634; H, Me, H, Me, S, Br, F, H, H, O], [AC9635; H, Me, H] , Me, S, I, F, H, H, O], [AC 9636; H, Me, H, Me, S, Me, F, H, H, O], [AC 9637; H, Me, H, Me , S, Et, F, H, H, O], [AC 9638; H, Me, H, Me, S, Pr, F, H, H, O], [AC 9639; H, Me, H, Me, S , i-Pr, F, H , H, O], [AC9640; H, Me, H, Me, S, CH = CH 2, F, H, H, O], [AC9641; H, Me, H, _{Me, S, C (CH 3} ) = CH 2, F, H, H, O], [AC9642; H, Me, H, Me, S, C≡CH, F, H, H, O], [AC9643 H, Me, H, Me, S, C≡CCH ₃ , F, H, H, O], [AC9644; H, Me, H, Me, S, c-Pr, F, H, H, O] H, Me, H, Me, S, OMe, F, H, H, O], [AC 9646; H, Me, H, Me, S, OEt, F, H, H, O], [AC 9645; AC, 947; H, Me, H, Me, S, Oi-Pr, F, H, H, O], [AC9648; H, Me, H, Me, S, SMe, F, H, H, O], [ AC9649; H, Me, H, Me, S, SEt, F, H, H, O], [AC9650; H, Me, H, Me, S, CH 2 F, F, H, H, O], [ AC9651; H, Me, H, Me, S, CHF 2, F, H, H, O], [AC9652; H, Me, H, Me, S, CF 3, F, H, H, O], [ AC9653; H, Me, H, Me, S, OCH 2 F, F, H, H, O], [AC9654; H, Me, H, Me, S, OCHF 2, F, H, H, O], [AC9655; H, Me, H , Me, S, OCF 3, F, H, H, O], [AC9656; H, Me, H, Me, S, SCH 2 F, F, H, H, O] , [AC 9657; H, Me, H, Me, S, SCHF ₂ , F, H, H, O], [AC 965 8; H, Me, H, Me, S, SCF 3, F, H, H, O], [AC9659; H, Me, H, Me, S, CN, F, H, H, O], [AC9660 ; H, Me, H, Me , S, NO 2, F, H, H, O], [AC9661; H, H, H, H, S, H, H, H, F, O], [AC9662; H, H, H, H, H, S, F, H, H, F, O], [AC9663; H, H, H, H, S, Cl, H, F, O], [AC 9664; H, H, H, H, H, S, Br, H, H, F, O], [AC 9665; H, H, H, H, S, I, H, F, O], [AC 9666; H, H, H, H, S, Me, H, H, F, O], [AC 9667; H, H, H, H, S, Et, H, H, F, O],

[AC 9668; H, H, H, H, H, S, Pr, H, H, F, O], [AC 9669; H, H, H, H, S, i-Pr, H, H, F, O], [AC9670; H, H, H , H, S, CH = CH 2, H, H, F, O], [AC9671; H, H, H, H, S, C (CH 3) = CH 2, H H, H, H, H, H, S, CHCH, H, H, F, O], [AC 9673; H, H, H, H, S, C≡ CCH ₃ , H, H, F, O], [AC9674; H, H, H, H, S, c, Pr, H, H, F, O], [AC 9675; H, H, H, H, S, OMe, H, H, F, O], [AC 9676; H, H, H, H, S, OEt, H, H, F, O], [AC 9677; H, H, H, H, S, Oi- Pr, H, H, F, O], [AC 9678; H, H, H, H, S, S Me, H, F, O], [AC 9679; H, H, H, H, S, SE t, H, H, F, O] , [AC9680; H, H, H, H, S, CH 2 F, H, H, F, O], [AC9681; H, H, H, H, S, CHF 2 , H, H, F, O ], [AC9682; H, H, H, H, S, CF 3, H, H, F, O], [AC9683; H, H, H, H, S, OCH 2 F, H, H, F, O], [AC9684; H, H, H, H, S, OCHF 2, H, H, F, O], [AC9685; H, H, H, H, S, OCF ₃ , H, H, F, O], [AC9686; H, H, H, H, S, SCH ₂ F, H, H, F, O], [AC9687; H, H, H, H, S, _{SCHF 2, H, H, F} , O], [AC9688; H, H, H, H, S, SCF 3, H, H, F, O], [AC9689; H, H, H, H, S, CN, H, H, F, O], [AC 9690; H, H, H, H, S, NO ₂ , H, H, F, O], [AC 9691; H, H, H, Me, S, H H, H, F, O], [AC 9692; H, H, H, Me, S, F, H, F, O], [AC 9693; H, H, H, Me, S, Cl, H , H, F, O], [AC9694; H, H, H, Me, S, Br, H, F, O], [AC9695; H, H, H, Me, S, I, H, H , F, O], [AC9696; H, H, H, Me, S, Me, H, F, O], [AC9697; H, H, H, Me, S, Et, H, H, F , O], [AC9698; H, H, H , Me, S, Pr, H, H, F, O], [AC 9699; H, H, H, Me, S, i-Pr, H, F, O], [AC 9700; H, H, H , Me, S, CH = CH 2, H, H, F, O], [AC9701; H, H, H, Me, S, C (CH 3) = CH 2, H, H, F, O], [AC9702; H, H, H, H, Me, S, C≡CH, H, H, F, O], [AC 9703; H, H, H, Me, S, C≡CCH ₃ , H, H, F, O, [AC 9704; H, H, H, Me, S, c-Pr, H, F, O], [AC 9705; H, H, H, Me, S, OMe, H, H, F, O, [AC 9706; H, H, H, Me, S, OEt, H, H, F, O], [AC 9707; H, H, H, Me, S, Oi-Pr, H, H, F, O, [AC9708; H, H, H, Me, S, SMe, H, F, O], [AC 9709; H, H, H, Me, S, SEt, H, H, F, O] , [AC9710; H, H, H, Me, S, CH 2 F, H, H, F, O], [AC9711; H, H, H, Me, S, CHF 2, H, H, F, O ], [AC9712; H, H , H, Me, S, CF 3, H, H, F, O], [AC9713; H, H, H, Me, S, OCH 2 F, H, H, F, O, [AC9714; H, H, H, Me, S, OCHF ₂ , H, H, F, O], [AC 9715; H, H, H, Me, S, OCF ₃ , H, H, F, O], [AC9716; H, H, H, Me, S, SCH 2 F, H, H, F, O], [AC9717; H, H, H, Me, S, SCHF 2, H, H, F , O], [AC9718; H , H, H, Me, S, SCF 3, H, H, F, O], [AC9719; H, H, H, Me, S, CN, H, H, F, O, [AC9720; H, H, H, Me, S, NO ₂ , H, F, O], [AC9721; H, Me, H, Me, S, H, H, F, O H, Me, H, Me, S, F, H, F, O], [AC 9723; H, Me, H, Me, S, Cl, H, F, O], [AC9724; H, Me, H, Me, S, Br, H, F, O], [AC9725; H, Me, H, Me, S, I, H, F, O], [AC9726 H, Me, H, Me, S, Me, H, H, F, O], [AC 9727; H, Me, H, Me, S, Et, H, H, F H, Me, H, Me, S, Pr, H, F, O], [AC 9729; H, Me, H, Me, S, i-Pr, H, H, F , O], [AC9730; H , Me, H, Me, S, CH = CH 2, H, H, F, O], [AC9731; H, Me, H, Me, S, C (CH 3) = _{CH 2, H, H, F} , O], [AC9732; H, Me, H, Me, S, C≡CH, H, H, F, O], [AC9733; H, Me, H, Me, S H, Me, H, Me, S, c-Pr, H, H, F, O], [AC9735; H, Me, H, C, CCHCCH ₃ , H, H, F, O], [AC 9734; Me, S, OMe, H, H, F, O], [AC 9736; H, Me, H, Me, S, OEt, H, H, F, O], [AC 9737; H, Me, H, Me, S, Oi-Pr, H, H, F, O], [AC 9738; H, Me, H, Me, S, SMe, H, F, O], [AC 9739; H, Me, H, Me, S, SEt, H, H, F, O], [AC9740; H, Me, H, Me, S, CH 2 F, H, H, F, O], [AC9741; H, Me, H, Me, _{S, CHF 2, H, H} , F, O], [AC9742; H, Me, H, Me, S, CF 3, H, H, F, O], [AC9743; H, Me, H, Me, _{S, OCH 2 F, H,} H, F, O], [AC9744; H, Me, H, Me, S, OCHF 2, H, H, F, O], [AC9745; H, Me, H, Me _{, S, OCF 3, H,} H, F, O], [AC9746; H, Me, H, Me, S, SCH 2 F, H, H, F, O], [AC9747; H, Me, H, _{Me, S, SCHF 2, H} , H, F, O], [AC9748; H, Me, H, Me, S, SCF 3, H, H, F, O], [AC9749; H, Me, H, Me, S, CN, H, H, F, O], [AC 9750; H, Me, H, Me, S, NO ₂ , H, H, F, O], [AC 9751; H, H, H, H , S, H, H, H, F, O], [AC9752; H, H, H, H, S, F, H, F, O], [AC9753; H, H, H, H, S , Cl, H, H, F, O], [AC 9754; H, H, H, H, S, Br, H, F, O], [AC 9755; H, H, H, H, S, I , H, H, F, O], [AC 9756; H, H, H, H, S, Me, H, H, F, O], [AC9757; H, H, H, H, H, S, Et, H, H, F, O], [AC9758; H, H, H, H, S, Pr, H, F, O], [AC9759 ; H, H, H, H , S, i-Pr, H, H, F, O], [AC9760; H, H, H, H, S, CH = CH 2, H, H, F, O] , [AC9761; H, H, H, H, S, C (CH 3) = CH 2, H, H, F, O], [AC9762; H, H, H, H, S, C≡CH, H H, H, H, H, S, C≡CCH ₃ , H, H, F, O], [AC 9764; H, H, H, H, S, c- Pr, H, H, F, O], [AC 9765; H, H, H, H, S, OMe, H, H, F, O], [AC 9766; H, H, H, H, S, OE t, H, H, F, O], [AC9767; H, H, H, H, S, Oi-Pr, H, H, F, O],

[AC 9768; H, H, H, H, H, S, SMe, H, H, F, O], [AC 9769; H, H, H, H, S, SE t, H, H, F, O], [AC 9770 ; H, H, H, H , S, CH 2 F, H, H, F, O], [AC9771; H, H, H, H, S, CHF 2, H, H, F, O], [ AC9772; H, H, H, H, S, CF 3, H, H, F, O], [AC9773; H, H, H, H, S, OCH 2 F, H, H, F, O], [AC 9774; H, H, H, H, H, S, OCHF ₂ , H, H, F, O], [AC 9775; H, H, H, H, S, OCF ₃ , H, H, F, O], [AC 9776; H, H, H, H, H, S, SCH ₂ F, H, H, F, O], [AC 9777; H, H, H, H, S, SCHF ₂ , H, H, F, O] , [AC9778; H, H, H, H, S, SCF 3, H, H, F, O], [AC9779; H, H, H, H, S, CN, H, H, F, O], [AC 9780; H, H, H, H, H, S, NO ₂ , H, H, F, O], [AC 9781; H, H, H, Me, S, H, H, F, O], [AC AC 9782; H, H, H, H, Me, S, F, H, F, O], [AC 9783; H, H, H, Me, S, Cl, H, F, O], [AC 9784; H, H, H, H, Me, S, Br, H, H, F, O], [AC9785; H, H, H, Me, S, I, H, F, O], [AC9786; H, H, H, Me, S, Me, H, H, F, O], [AC9787; H, H, H, Me, S, Et, H, F, O], [AC 9788; H, H, H, Me, S, Pr, H, H, F, O], [AC 9789; H, H, H, Me, S, i-Pr, H, F, O], [AC 9790; H, H, H, Me, S, CH = CH 2, H, H, F, O], [AC9791; H, H, H, Me, S, C (CH 3) = CH 2, H, H, F, O] H, H, H, Me, S, C≡CH, H, H, F, O], [AC 9793; H, H, H, Me, S, C≡ CCH ₃ , H, H, F , O], [AC 9794; H, H, H, Me, S, c-Pr, H, H, F, O], [AC 9795; H, H, H, Me, S, OMe, H, H, F H, H, H, Me, S, OEt, H, H, F, O], [AC9797; H, H, H, Me, S, Oi-Pr, H, H, F , O], [AC 9798; H, H, H, H, Me, S, SMe, H, H, F, O], [AC 9799; H, H, H, Me, S, SE t, H, H, F, O], [AC 9800; H, H, H, Me, S, CH 2 F, H, H, F, O], [AC9801; H, H, H, Me, S, CHF 2, H, H, F, O], [AC9802 ; H, H, H, Me , S, CF 3, H, H, F, O], [AC9803; H, H, H, Me, S, OCH 2 F, H, H, F, O], [ AC9804; H, H, H, Me, S, OCHF 2, H, H, F, O], [AC9805; H, H, H, Me, S, OCF 3, H, H, F, O], [ AC 9806; H, H, H, H, Me, S, SCH ₂ F, H, H, F, O], [AC 9807; H, H, H, Me, S, SCHF ₂ , H, H, F, O], [AC9808; H, H, H , Me, S, SCF 3, H, H, F, O], [AC9809; H, H, H, Me, S, CN, H, H, F, O], [ AC 9810; H, H, H, H, Me, S, NO ₂ , H, H, F, O], [AC 9811; H, Me, H, Me, S, H, H, F, O], [AC 9812 H, Me, H, Me, S, F, H, H, F, O], [AC 9813; H, Me, H, Me, S, Cl, H, F, O], [AC 9814; H , Me, H, Me, S, Br, H, H, F, O], [AC 9815; H, Me, H, Me, S, I, H, F, O], [AC 9816; H, Me , H, Me, S, Me, H, H, F, O], [AC 9817; H, Me, H, Me, S, Et, H, F, O], [AC 9818; H, Me, H , Me, S, Pr, H, H, F, O], [AC 9819; H, Me, H, Me, S, i-Pr, H, H, F, O], [AC 9820; H, Me, H , Me, S, CH = CH 2, H, H, F, O], [AC9821; H, Me, H, Me, S, C (CH 3) = CH 2, H, H, F, O], [AC 9822; H, Me, H, Me, S, C≡CH, H, H, F, O], [AC 9823; H, Me, H, Me, S, C≡CCH ₃ , H, H, F, H, Me, H, Me, S, c-Pr, H, F, O], [AC 9825; H, Me, H, Me, S, OMe, H, H, F, O], [AC 9824; O], [AC 9826; H, Me, H, Me, S, OEt, H, H, F, O], [AC 9827; H, M e, H, Me, S, Oi-Pr, H, H, F, O], [AC 9828; H, Me, H, Me, S, S Me, H, F, O], [AC 9829; H, Me, H, Me, S, SEt, H, H, F, O], [AC9830; H, Me, H, Me, S, CH 2 F, H, H, F, O], [AC9831; H, Me, H, Me, S, CHF 2, H, H, F, O], [AC9832; H, Me, H, Me, S, CF 3, H, H, F, O], [AC9833; H, Me, H, Me, S, OCH 2 F, H, H, F, O], [AC9834; H, Me, H, Me, S, OCHF 2, H, H, F, O], [AC9835; H , Me, H, Me, S , OCF 3, H, H, F, O], [AC9836; H, Me, H, Me, S, SCH 2 F, H, H, F, O], [AC9837; H, Me, H, Me, S, SCHF ₂ , H, H, F, O], [AC 9838; H, Me, H, Me, S, SCF ₃ , H, H, F, O], [AC 9839; H, Me, H, Me, S, CN, H, H, F, O], [AC 9840; H, Me, H, Me, S, NO ₂ , H, H, F, O], [AC 9841; H , H, H, H, S, H, H, H, Me, O], [AC 9842; H, H, H, H, S, F, H, Me, O], [AC 9843; H, H , H, H, S, Cl, H, H, Me, O], [AC 9844; H, H, H, H, S, Br, H, Me, O], [AC 9845; H, H, H , H, S, I, H, H, Me, O], [AC 9846; H, H, H, H, S, Me, H, Me, O], [AC 9847; H, H, H, H , S, Et, H, H, Me, O], [AC 9848; H, H, H, H, S, Pr, H, Me, O], [AC 9849; H, H, H, H, S , i-Pr, H, H, Me, O], [AC 9850; H, H, H, H, S, CH = CH ₂ , H, H, Me, O], [AC 9851; H, H, H, H, S, C (CH ₃ ) = CH ₂ , H, H, Me, O], [AC 9852; H, H, H, H, S, C≡CH, H, H, Me, O], [AC 9853 H, H, H, H, H, S, C≡CCH ₃ , H, H, Me, O], [AC 9854; H, H, H, H, S, c-Pr, H, H, Me, O] , [AC 9855; H, H, H, H, S, OMe, H, H, Me, O], [AC 9856; H, H, H, H, S, O Et, H, H, Me, O], [AC 9857; H, H, H, H, S, Oi-Pr, H, H, Me, O], [AC 9858; H, H, H, H, S, SMe, H, H, Me, O], [AC 9859; H, H, H, H, S, SE t, H, H, Me, O], [AC 9860; H, H, H, H, S, CH ₂ F, H, H, Me, O], [AC 9861; H, H, H, H, S, CHF ₂ , H, H, Me, O], [AC 9862; H, H, H, H, S, CF _{3, H, H, Me,} O], [AC9863; H, H, H, H, S, OCH 2 F, H, H, Me, O], [AC9864; H, H, H, H, S, _{OCHF 2, H, H, Me} , O], [AC9865; H, H, H, H, S, OCF 3, H, H, Me, O], [AC9866; H, H, H, H, S, SCH ₂ F, H, H, Me, O], [AC 9867; H, H, H, H, S, SCHF ₂ , H, H, Me, O],

[AC9868; H, H, H , H, S, SCF 3, H, H, Me, O], [AC9869; H, H, H, H, S, CN, H, H, Me, O], [ AC9870; H, H, H, H, S, NO 2, H, H, Me, O], [AC9871; H, H, H, Me, S, H, H, H, Me, O], [AC9872 H, H, H, H, Me, S, F, H, H, Me, O], [AC 9873; H, H, H, Me, S, Cl, H, Me, O], [AC 9874; H , H, H, Me, S, Br, H, H, Me, O], [AC9875; H, H, H, Me, S, I, H, Me, O], [AC 9876; H, H , H, Me, S, Me, H, H, Me, O], [AC 9877; H, H, H, Me, S, Et, H, Me, O], [AC 9878; H, H, H , Me, S, Pr, H, H, Me, O], [AC 9879; H, H, H, Me, S, i-Pr, H, H, Me, O], [AC 9880; H, H, H , Me, S, CH = CH 2, H, H, Me, O], [AC9881; H, H, H, Me, S, C (CH 3) = CH 2, H, H, Me, O], [AC 9882; H, H, H, H, Me, S, CHCH, H, H, Me, O], [AC 9883; H, H, H, Me, S, C≡ CCH ₃ , H, H, Me, H, H, H, Me, S, c-Pr, H, Me, O], [AC 9885; H, H, H, Me, S, OMe, H, H, Me, O], [AC 9884; O, [AC 9886; H, H, H, Me, S, OEt, H, H, Me, O], [AC 9887; H, H, H, Me, S, Oi-Pr, H, H, Me, O, [AC 9888; H, H, H, Me, S, SMe, H, Me, O], [AC 9889; H, H, H, Me, S, SE t, H, H, Me, O] , [AC9890; H, H, H, Me, S, CH 2 F, H, H, Me, O], [AC9891; H, H, H, Me, S, CHF 2, H, H, Me, O ], [AC9892; H, H , H, Me, S, CF 3, H, H, Me, O], [AC9893; H, H, H, Me, S, OCH 2 F, H, H, Me, O, [AC 9894; H, H, H, Me, S, OCHF ₂ , H, H, Me, O], [AC 9895; H, H, H, Me, S, OCF ₃ , H, H, Me, O], [AC 9896; H, H, H, Me, S, SCH ₂ F, H, H, Me, O], [AC9897; H, H, H, Me, S, SCHF ₂ , H, H, Me, O], [AC 9898; H, H, H, Me, S, SCF ₃ , H, H, Me, O], [AC9899; H, H, H , Me, S, CN, H, H, Me, O], [AC9900; H, H, H, Me, S, NO 2, H, H, Me, O], [ AC9901; H, Me, H, Me, S, H, H, Me, O], [AC9902; H, Me, H, Me, S, F, H, Me, O], [AC9903; H, Me, H, Me, S, Cl, H, H, Me, O], [AC9904; H, Me, H, Me, S, Br, H, Me, O], [AC9905; H, Me, H, Me, S, I, H, H, Me, O], [AC9906; H, Me, H, Me, S, Me, H, Me, O], [AC9907; H, Me, H, Me, S, Et, H, H, Me, O], [AC9908; H, Me, H, Me, S, Pr, H, Me, O], [AC 9909; H, Me, H, Me, S, i-Pr, H, H, Me, O], [AC9910; H, Me, H, Me, S, CH = CH 2, H, H, Me, O], [AC9911; H, Me , H, Me, S, C (CH 3) = CH 2, H, H, Me, O], [AC9912; H, Me, H, Me, S, C≡CH, H, H, Me, O] , [AC 9913; H, Me, H, Me, S, C≡CCH ₃ , H, H, Me, O], [AC 9914; H, Me, H, Me, S, c-Pr, H, H, Me H, Me, H, Me, S, OMe, H, Me, O], [AC 9916; H, Me, H, Me, S, OEt, H, H, Me, O H, Me, H, Me, S, Oi-Pr, H, H, Me, O], [AC 9918; H, Me, H, Me, S, SMe, H, H, Me, O] ], [AC9919; H, Me , H, Me, S, SEt, H, H, Me, O], [AC9920; H, Me, H, Me, S, CH 2 F, H, H, Me, O ], [AC9921; H, Me , H, Me, S, CHF 2, H, H, Me, O], [AC9922; H, Me, H, Me, S, CF 3, H, H, Me, O ], [AC9923; H, Me , H, Me, S, OCH 2 F, H, H, Me, O], [AC9924; H, Me, H, Me, S, OCHF 2, H, H, Me, O], [AC 9925; H , Me, H, Me, S , OCF 3, H, H, Me, O], [AC9926; H, Me, H, Me, S, SCH 2 F, H, H, Me, O], [AC9927; H, Me, H, Me, S, SCHF 2, H, H, Me, O], [AC9928; H, Me, H, Me, S, SCF 3, H, H, Me, O], [AC9929; H, Me, H, Me, S, CN, H, H, Me, O], [AC9930; H, Me, H, Me, S, NO 2, H, H, Me, O], [AC9931; H , H, H, H, S, H, H, H, Me, O], [AC 9932; H, H, H, H, S, F, H, Me, O], [AC 9933; H, H , H, H, S, Cl, H, H, Me, O], [AC9934; H, H, H, H, S, Br, H, Me, O], [AC9935; H, H, H] , H, S, I, H, H, Me, O], [AC9936; H, H, H, H, S, Me, H, Me, O], [AC9937; H, H, H, H] , S, Et, H, H, Me, O], [AC 9938; H, H, H, H, S, Pr, H, Me, O], [AC 9939; H, H, H, H, S , i-Pr, H, H , Me, O], [AC9940; H, H, H, H, S, CH = CH 2, H, H, Me, O], [AC9941; H, H, H, _{H, S, C (CH 3} ) = CH 2, H, H, Me, O], [AC9942; H, H, H, H, S, C≡CH, H, H, Me, O], [AC9943 H, H, H, H, H, S, C≡CCH ₃ , H, H, Me, O], [AC 9944; H, H, H, H, S, c-Pr, H, H, Me, O] [AC9945; H, H, H, H, H, S, OMe, H, H, Me, O], [AC9946; H, H, H, H, S, OEt, H, H, Me, O], [, AC 99 47; H, H, H, H, H, S, Oi-Pr, H, H, Me, O], [AC 9948; H, H, H, H, S, S Me, H, Me, O], [ AC 9949; H, H, H, H, H, S, SEt, H, H, Me, O], [AC9950; H, H, H, H, S, CH ₂ F, H, Me, O], [, AC9951; H, H, H, H, S, CHF 2, H, H, Me, O], [AC9952; H, H, H, H, S, CF 3, H, H, Me, O], [ AC 9953; H, H, H, H, S, OCH ₂ F, H, H, Me, O], [AC 9954; H, H, H, H, S, OCHF _{2, H, H, Me,} O], [AC9955; H, H, H, H, S, OCF 3, H, H, Me, O], [AC9956; H, H, H, H, S, SCH ₂ F, H, H, Me, O], [AC9957; H, H, H, H, S, SCHF ₂ , H, H, Me, O], [AC 9958; H, H, H, H, S, SCF ₃ , H, H, Me, O], [AC 9959; H, H, H, H, S, CN, H, H, Me, O], [AC 9960; H, H, H, H, S, NO ₂ , H, H, Me, O], [AC9961; H, H, H, Me, S, H, H, H, Me, O], [AC 9962; H, H, H, Me, S, F, H, H, Me, O], [AC9963; H, H, H, Me, S, Cl, H, H, Me, O], [AC9964; H, H, H, Me, S, Br, H, H, Me, O], [AC9965; H, H, H, Me, S, I, H, Me, O], [AC 9966; H, H, H, Me, S, Me, H, H, H, Me, O],

[AC9967; H, H, H, H, Me, S, Et, H, H, Me, O], [AC9968; H, H, H, Me, S, Pr, H, Me, O], [AC9969 ; H, H, H, Me , S, i-Pr, H, H, Me, O], [AC9970; H, H, H, Me, S, CH = CH 2, H, H, Me, O] , [AC9971; H, H, H, Me, S, C (CH 3) = CH 2, H, H, Me, O], [AC9972; H, H, H, Me, S, C≡CH, H , H, Me, O], [AC 9973; H, H, H, Me, S, C≡CCH ₃ , H, H, Me, O], [AC 9974; H, H, H, Me, S, c- Pr, H, H, Me, O], [AC9975; H, H, H, Me, S, OMe, H, H, Me, O], [AC9976; H, H, H, Me, S, OEt, H, H, Me, O], [AC9977; H, H, H, Me, S, Oi-Pr, H, H, Me, O], [AC9978; H, H, H, Me, S, SMe, H, H, Me, O], [AC 9979; H, H, H, Me, S, SE t, H, H, Me, O], [AC 9980; H, H, H, Me, S, CH ₂ F, H, H, Me, O], [AC 9981; H, H, H, Me, S, CHF ₂ , H, H, Me, O], [AC 9982; H, H, H, Me, S, CF ₃ , H, H, Me, O], [AC 9983; H, H, H, Me, S, OCH ₂ F, H, H, Me, O], [AC 9984; H, H, H, Me, S, OCHF ₂ , H, H, Me, O ], [AC9985; H, H, H, Me, S, OCF 3, H, H, Me, O], [AC9986; H, H, H, Me, S, SCH 2 F, H, H, Me, O], [AC 9987; H, H, H, Me, S, SCHF ₂ , H, H, Me, O], [AC 9988; H, H, H, Me, S, SCF ₃ , H, H, Me, O], [AC 9989; H, H, H, Me, S, CN, H, H, Me, O], [AC 9990; H, H, H, Me, S, NO ₂ , H, H, Me, O], [AC 999 1; H, Me, H, Me, S, H, H, H, Me, O], [AC 999 2; H, Me, H, Me, S, F, H , H, Me, O], [AC9993; H, Me, H, Me, S, Cl, H, H, Me, O], [AC9994; H, Me, H, Me, S, Br, H, H , Me, O], [AC9995; H, Me, H, Me, S , I, H, H, Me, O], [AC9996; H, Me, H, Me, S, Me, H, H, Me, O], [AC 9997; H, Me, H, Me, S, Et , H, H, Me, O], [AC 9998; H, Me, H, Me, S, Pr, H, H, Me, O], [AC 9999; H, Me, H, Me, S, i-Pr , H, H, Me, O ], [AC10000; H, Me, H, Me, S, CH = CH 2, H, H, Me, O], [AC10001; H, Me, H, Me, S, _{C (CH 3) = CH 2} , H, H, Me, O], [AC10002; H, Me, H, Me, S, C≡CH, H, H, Me, O], [AC10003; H, Me , H, Me, S, C≡CCH ₃ , H, H, Me, O], [AC 10004; H, Me, H, Me, S, c-Pr, H, H, Me, O], [AC 1 0005; H, Me, H, Me, S, OMe, H, H, Me, O], [AC 10006; H, Me, H, Me, S, OEt, H, Me, O], [AC 1 0007; H, Me, H, Me, S, Oi-Pr, H, H, Me, O], [AC10008; H, Me, H, Me, S, SMe, H, Me, O], [AC 1 0009; H, Me, H, Me, S, SEt, H, H, Me, O], [AC 10010; H, Me, H, Me, S, CH ₂ F, H, Me, O], [AC 100 11; H, Me, H, Me, S, CHF 2, H, H, Me, O], [AC10012; H, Me, H, Me, S, CF 3, H, H, Me, O], [AC10013; H, Me, H, Me, S, OCH 2 F, H, H, Me, O], [AC10014; H, Me, H, Me, S, OCHF 2, H, H, Me, O], [AC10015; H , Me, H, Me, S , OCF 3, H, H, Me, O], [AC10016; H, Me, H, Me, S, SCH 2 F, H, H, Me, O], [AC10017; H, Me, H, Me, S, SCHF 2, H, H, Me, O], [AC10018; H, Me, H, Me, S, SCF 3, H, H, Me, O], [AC10019; H, Me, H, Me, S, CN, H, H, Me, O], [AC10020; H, Me, H, Me, S, NO 2, H, H, Me, O], [AC10021; H , H, H, H, S, H, H, H, H, S], [AC 10022; H, H, H, H, S, F, H, H, H, S H, H, H, H, H, S, Cl, H, H, H, S], [AC 10024; H, H, H, H, S, Br, H, H, H, S], [AC1 0025; H, H, H, H, S, I, H, H, S], [AC 1 0026; H, H, H, H, S, Me, H, H, H, S], [AC 1 0027 H, H, H, H, H, S, Et, H, H, H, S], [AC10028; H, H, H, H, S, Pr, H, H, S, [AC10029; H , H, H, H, S , i-Pr, H, H, H, S], [AC10030; H, H, H, H, S, CH = CH 2, H, H, H, S], [ AC10031; H, H, H, H, S, C (CH 3) = CH 2, H, H, H, S], [AC10032; H, H, H, H, S, C≡CH, H, H , H, S], [AC1 0033; H, H, H, H, S, C≡CCH ₃ , H, H, H, S], [AC 1 0034; H, H, H, H, S, c-Pr, H, H, H, S], [AC1 0035; H, H, H, H, S, OMe, H, H, H, S], [AC 10036; H, H, H, H, S, OE t, H, H, H, S], [AC 1 0037; H, H, H, H, S, Oi-Pr, H, H, H, S], [AC 1 0038; H, H, H, H, S, S Me, H, H, H, S], [AC 1 0039; H, H, H, H, S, SE t, H, H, H, S], [AC 1 040; H, H, H, H, S, CH ₂ F, H, H, H, S], [ AC10041; H, H, H, H, S, CHF 2, H, H, H, S], [AC10042; H, H, H, H, S, CF 3, H, H, H, S], [ AC10043; H, H, H, H, S, OCH 2 F, H, H, H, S], [AC10044; H, H, H, H, S, OCHF 2, H , H, H, S], [AC10045; H, H, H, H, S, OCF 3, H, H, H, S], [AC10046; H, H, H, H, S, SCH 2 F, H, H, H, S], [AC 10047; H, H, H, H, S, SCHF ₂ , H, H, H, S], [AC 10048; H, H, H, H, S, SCF ₃ , H, H, H, S], [AC 10049; H, H, H, H, S, CN, H, H, H, S], [AC 10050; H, H, H, H, S, NO ₂ , H , H, H, S], [AC10051; H, H, H, Me, S, H, H, H, H, S], [AC 10052; H, H, H, Me , S, F, H, H, H, S], [AC 10053; H, H, H, Me, S, Cl, H, H, H, S], [AC 10054; H, H, H, Me, S , Br, H, H, H, S], [AC10055; H, H, H, Me, S, I, H, H, H, S], [AC 10056; H, H, H, Me, S, Me H, H, H, S], [AC 10057; H, H, H, Me, S, Et, H, H, H, S], [AC 10058; H, H, H, Me, S, Pr, H , H, H, S], [AC 1 0059; H, H, H, Me, S, i-Pr, H, H, H, S], [AC 1 060; H, H, H, Me, S, CH = CH ₂ , H, H, H, S], [AC 10061; H, H, H, Me, S, C (CH ₃ ) = CH ₂ , H, H, H, S], [AC 10062; H, H, H , Me, S, C≡CH, H, H, H, S], [AC10063; H, H, H, Me, S, C≡CCH ₃ , H, H, H, S], [AC10064; H, H, H, Me, S, c-Pr, H, H, H, S], [AC10065; H, H, H, Me, S, OMe, H, H, S, [AC10066; H, H, H, Me, S, OEt, H, H, H, S],

[AC10067; H, H, H, Me, S, Oi-Pr, H, H, H, S], [AC 10068; H, H, H, Me, S, SMe, H, H, H, S], [AC10069; H, H, H , Me, S, SEt, H, H, H, S], [AC10070; H, H, H, Me, S, CH 2 F, H, H, H, S], [AC10071; H, H, H , Me, S, CHF 2, H, H, H, S], [AC10072; H, H, H, Me, S, CF 3, H, H, H, S], [AC10073; H, H, H , Me, S, OCH 2 F, H, H, H, S], [AC10074; H, H, H, Me, S, OCHF 2, H, H, H, S] , [AC10075; H, H, H, Me, S, OCF 3, H, H, H, S], [AC10076; H, H, H, Me, S, SCH 2 F, H, H, H, S H, H, H, H, Me, S, SCHF ₂ , H, H, H, S], [AC 10078; H, H, H, Me, S, SCF ₃ , H, H, H, S H, H, H, Me, S, CN, H, H, H, S], [AC 10080; H, H, H, Me, S, NO ₂ , H, H, H, S] , [AC10081; H, Me, H, Me, S, H, H, H, S], [AC 10082; H, Me, H, Me, S, F, H, H, S, [, AC10083; H, Me, H, Me, S, Cl, H, H, S], [AC10084; H, Me, H, Me, S, Br, H, H, H, S], [AC10085; H, Me, H, Me, S, I, H, H, H, S], [AC10086; H, Me, H, Me, S, Me, H, H, S, [AC10087; H, Me, H, Me, S, Et, H, H, H, S], [AC 10088; H, Me, H, Me, S, Pr, H, H, S, [AC 10089; H, Me, H, Me, S, i- Pr, H, H, H, S], [AC10090; H, Me, H, Me, S, CH = CH 2, H, H, H, S], [AC10091; H , Me, H, Me, S , C (CH 3) = CH 2, H, H, H, S], [AC10092; H, Me, H, Me, S, C≡CH, H, H, H, S, [AC10093; H, Me, H, Me, S, C≡CCH ₃ , H, H, H, S], [AC10094; H, Me, H, Me, S, c-Pr, H, H , H, S], [AC 10095; H, M e, H, Me, S, OMe, H, H, H, S], [AC10096; H, Me, H, Me, S, OEt, H, H, H, S], [AC10097; H, Me, H, Me, S, Oi-Pr, H, H, H, S], [AC10098; H, Me, H, Me, S, SMe, H, H, S, [AC10099; H, Me, H, Me, S, SEt, H, H, H, S], [AC 10 100; H, Me, H, Me, S, CH ₂ F, H, H, S, [AC 10 101; H, Me, _{H, Me, S, CHF 2} , H, H, H, S], [AC10102; H, Me, H, Me, S, CF 3, H, H, H, S], [AC10103; H, Me, _{H, Me, S, OCH 2} F, H, H, H, S], [AC10104; H, Me, H, Me, S, OCHF 2, H, H, H, S], [AC10105; H, Me , H, Me, S, OCF 3, H, H, H, S], [AC10106; H, Me, H, Me, S, SCH 2 F, H, H, H, S], [AC10107; H, Me, H, Me, S, SCHF ₂ , H, H, H, S], [AC 10108; H, Me, H, Me, S, SCF ₃ , H, H, H, S], [AC 10109; H, Me, H, Me, S, CN, H, H, H, S], [AC 10110; H, Me, H, Me, S, NO ₂ , H, H, H, S], [AC 10 111; H, H , H, H, S, H, H, H, H, S], [AC 10112; H, H, H, H, S, F, H, H, S], [AC 10 113; H, H, H , H, S, Cl, H, H, H, S], [AC 10114; H, H, H, H, S, Br, H, H, H, S], [AC 10 115; H, H, H, H , S, I, H, H, H, S], [AC 10 116; H, H, H, H, S, Me, H, H, H, S], [AC 10117; H, H, H, H, S , Et, H, H, H, S], [AC10118; H, H, H, H, S, Pr, H, H, H, S], [AC 10119; H, H, H, H, S, i -Pr, H, H, H, S], [AC10120; H, H, H, H, S, CH = CH 2, H, H, H, S], [AC10121; H, H, H, H, S, C (CH ₃ ) = CH ₂ , H, H, H, S], [AC 10122; H, H, H, H, S, C≡CH, H, H, H, S], [AC 10123; H , H, H, H, S, C≡CCH ₃ , H, H, H, S], [AC H, H, H, H, H, S, c-Pr, H, H, H, S], [AC 10 125; H, H, H, H, S, OMe, H, H, H, S], [ AC 10 126; H, H, H, H, S, OEt, H, H, H, S], [AC10127; H, H, H, H, S, Oi-Pr, H, H, H, S], [ AC 10 128; H, H, H, H, H, S, SMe, H, H, H, S], [AC10129; H, H, H, H, S, SE t, H, H, H, S], [AC 10130; H, H, H, H, S, CH 2 F, H, H, H, S], [AC10131; H, H, H, H, S, CHF 2, H, H, H, S], [AC10132 H, H, H, H, H, S, CF ₃ , H, H, H, S], [AC 10133; H, H, H, H, S, OCH ₂ F, H, H, H, S], [, AC 10 134; H, H, H, H, H, S, OCHF ₂ , H, H, H, S], [AC 10 135; H, H, H, H, S, OCF ₃ , H, H, H, S], [ AC 10136; H, H, H, H, H, S, SCH ₂ F, H, H, H, S], [AC 10137; H, H, H, H, S, SCHF ₂ , H, H, H, S], [AC10138; H, H, H , H, S, SCF 3, H, H, H, S], [AC10139; H, H, H, H, S, CN, H, H, H, S], [ AC 10 140; H, H, H, H, H, S, NO ₂ , H, H, H, S], [AC10141; H, H, H, Me, S, H, H, H, S,] [AC 10142 H, H, H, H, Me, S, F, H, H, S], [AC10143; H, H, H, Me, S, Cl, H, H, H, S], [AC 10144; H , H, H, Me, S, Br, H, H, H, S], [AC10145; H, H, H, Me, S, I, H, H, S], [AC 10146; H, H , H, Me, S, Me, H, H, H, S], [AC10147; H, H, H, Me, S, Et, H, H, H, S], [AC10148; H, H, H , Me, S, Pr, H, H, H, S], [AC10149; H, H, H, Me, S, i-Pr, H, H, H, S], [AC 10150; H, H, H , Me, S, CH = CH 2, H, H, H, S], [AC10151; H, H, H, Me, S, C (CH 3) = CH 2, H, H, H, S], [AC 10 152; H, H, H, Me, S, C≡CH, H, H, H, S], [AC 10153; H, H, H, Me, S, C≡CCH ₃ , H, H, H, S], [AC10154; H, H, H, Me, S, c-Pr, H, H, H, S], [AC 10155; H, H, H, Me , S, OMe, H, H, H, S], [AC10156; H, H, H, Me, S, OEt, H, H, H, S], [AC10157; H, H, H, Me, S , Oi-Pr, H, H, H, S], [AC10158; H, H, H, Me, S, SMe, H, H, H, S], [AC10159; H, H, H, Me, S , SEt, H, H, H, S], [AC 10 160; H, H, H, Me, S, CH ₂ F, H, H, H, S], [AC 10 161; H, H, H, Me, S , CHF ₂ , H, H, H, S], [AC 10 162; H, H, H, Me, S, CF ₃ , H, H, H, S], [AC 10 163; H, H, H, Me, S OCH ₂ F, H, H, H, S], [AC10164; H, H, H, Me, S, OCHF ₂ , H, H, H, S], [AC 1 0165; H, H, H, Me, S, OCF ₃ , H, H, H, S], [AC10166; H, H, H, Me, S, SCH ₂ F, H, H, H, S],

[AC10167; H, H, H, Me, S, SCHF ₂ , H, H, H, S], [AC 10 168; H, H, H, Me, S, SCF ₃ , H, H, H, S], [AC10169; H, H, H , Me, S, CN, H, H, H, S], [AC10170; H, H, H, Me, S, NO 2, H, H, H, S], [ AC 10171; H, Me, H, Me, S, H, H, H, S], [AC 10172; H, Me, H, Me, S, F, H, H, S], [AC 10173; H, Me, H, Me, S, Cl, H, H, H, S], [AC10174; H, Me, H, Me, S, Br, H, H, S], [AC10175; H, Me, H, Me, S, I, H, H, H, S], [AC 10176; H, Me, H, Me, S, Me, H, H, S, [AC 10177; H, Me, H, Me, S, Et, H, H, H, S], [AC 10178; H, Me, H, Me, S, Pr, H, H, H, S], [AC 10179; H, Me, H, Me, S, i-Pr, H, H, H, S], [AC10180; H, Me, H, Me, S, CH = CH 2, H, H, H, S], [AC10181; H, Me , H, Me, S, C (CH 3) = CH 2, H, H, H, S], [AC10182; H, Me, H, Me, S, C≡CH, H, H, H, S] H, Me, H, Me, S, C≡CCH ₃ , H, H, H, S], [AC 10184; H, Me, H, Me, S, c-Pr, H, H, H H, Me, H, Me, S, OMe, H, H, H, S], [AC 10186; H, Me, H, Me, S, OEt, H, H, H, S H, Me, H, Me, S, Oi-Pr, H, H, H, S], [AC 10188; H, Me, H, Me, S, SMe, H, H, H, S] ], [AC10189; H, Me , H, Me, S, SEt, H, H, H, S], [AC10190; H, Me, H, Me, S, CH 2 F, H, H, H, S H, Me, H, Me, S, CHF ₂ , H, H, H, S], [AC 10 192; H, Me, H, Me, S, CF ₃ , H, H, H, S H, Me, H, Me, S, OCH ₂ F, H, H, H, S], [AC 10 194; H, Me, H, Me, S, OCHF ₂ , H, H, H, S], [AC10195; H, Me, H, Me, S, OCF 3, H, H, H, S], [AC10196; H, Me, H, Me, S, SCH 2 F, H, H, H, S], [AC10197 H, Me, H, Me, S, SCHF ₂ , H, H, H, S], [AC10198; H, Me, H, Me, S, SCF ₃ , H, H, H, S], [AC10199 H, Me, H, Me, S, CN, H, H, H, S], [AC 10 200; H, Me, H, Me, S, NO ₂ , H, H, H, S].

[Substituent number (MC2); E ¹⁰³ ], [BC1; pyrazol-1-yl], [BC2; 4-fluoro-pyrazol-1-yl], [BC3; 4-chloro-pyrazol-1-yl], [BC4; 4-bromo-pyrazol-1-yl], [BC5; 4-methyl-pyrazol-1-yl], [BC6; 4-ethyl-pyrazol-1-yl], [BC7; 4-propyl-pyrazole -4-yl], [BC8; 4-isopropyl-pyrazol-1-yl], [BC9; 4-cyclopropyl-pyrazol-1-yl], [BC10; 4-difluoromethyl-pyrazol-1-yl], [BC11; 4-cyano-pyrazol-1-yl], [BC12; 4-ethynyl-pyrazol-1-yl], [BC13; 4- (1-propynyl) -pyrazol-1-yl], [BC14; -Methyl-pyrazol-1-yl], [BC15; 4-fluoro-5-methyl-pyrazol-1-yl], [BC16; 4-chloro-5-methyl-pyrazol-1-yl], [BC17; 4 -Bromo-5-methyl-pyrazol-1-yl], [BC 18; 4, 5-dimethyl-pyrazol-1-yl], [BC 19; 4-ethyl-5-methyl-pyrazol-1-yl], [BC 20 5-methyl-4-propyl-pi; Razol-1-yl], [BC 21; 4-isopropyl-5-methyl-pyrazol-1-yl], [BC 22; 4-cyclopropyl-5-methyl-pyrazol-1-yl], [BC 23; 4-difluoro Methyl-5-methyl-pyrazol-1-yl], [BC24; 4-cyano-5-methyl-pyrazol-1-yl], [BC25; 4-ethynyl-5-methyl-pyrazol-1-yl], BC26; 5-methyl-4- (1-propynyl) -pyrazol-1-yl], [BC27; 5-ethyl-pyrazol-1-yl], [BC28; 4-fluoro-5-ethyl-pyrazole-1-l 4-chloro-5-ethyl-pyrazol-1-yl], [BC30; 4-bromo-5-ethyl-pyrazol-1-yl], [BC 31; 5-ethyl-4-methyl- Pyrazol-1-yl], [BC32; 4,5-diethyl-pyrazol-1-yl], [BC33; 4,5,6,7-tetrahydro-indazol-1-yl], [BC34; 3-methyl- 4,5,6,7-Tetrahydro-indazol-1-yl], [BC35; 4,5,6,7-Tetrahydro-indazol-2-yl], [BC36; 3-Methyl-4,5,6, 7-Tetrahydro-indazol-2-yl], [BC37; 4,5-dihydro-1H, 6H-cyclopenta [d] pyrazol-1-yl], [BC38; 3-methyl-4,5,6,7-tetrahydro-indazol-2-yl], [BC39 3-methyl-pyrazol-1-yl], [BC40; 4-fluoro-3-methyl-pyrazol-1-yl], [BC41; 4-chloro-3-methyl-pyrazol-1-yl], [BC42 4-bromo-3-methyl-pyrazol-1-yl], [BC 43; 3,4-dimethyl-pyrazol-1-yl], [BC 44; 4-ethyl-3-methyl-pyrazol-1-yl], [BC45; 4-propyl-3-methyl-pyrazol-1-yl], [BC46; 4-isopropyl-3-methyl-pyrazol-1-yl], [BC47; 4-cyclopropyl-3-methyl-pyrazole- 1-yl], [BC48; 4-difluoromethyl-3-methyl-pyrazol-1-yl], [BC49; 3-methyl-4-trifluoromethyl-pyrazol-1-yl], [BC50; 4-cyano -3-Methyl-pyrazol-1-yl], [BC 51; 4-ethynyl-3-methyl-pyrazol-1-yl], [BC 52; 3-methyl-4- (1-propynyl) -pyrazol-1-yl ], [BC53; 3,5-Dimethyl-pyrazol-1-yl], [BC54; 4-fluoro-3,5-dimethyl-pyrazol-1-yl], [BC55; 4-chloro-3,5-dimethyl-pyrazole-1-] 4-bromo-3,5-dimethyl-pyrazol-1-yl], [BC 57; 3,4,5-trimethyl-pyrazol-1-yl], [BC 58; 4-ethyl-3, 5-dimethyl-pyrazol-1-yl], [BC59; 3,5-dimethyl-4-propyl-pyrazol-1-yl], [BC60; 3,5-dimethyl-4-isopropyl-pyrazol-1-yl] , [BC61; 3,5-dimethyl-4-cyclopropyl-pyrazol-1-yl], [BC62; 4-difluoromethyl-3,5-dimethyl-pyrazol-1-yl], [BC63; 4-cyano- 3,5-Dimethyl-pyrazol-1-yl], [BC 64; 4-ethynyl-3,5-dimethyl-pyrazol-1-yl], [BC 65; 3,5-dimethyl-4- (1-propynyl)- Pyrazol-1-yl], [BC 66; 5-ethyl-3-methyl-pyrazol-1-yl], [BC 67; 5-ethyl-4-fluoro-3-methyl-pyrazol-1-yl], [BC 68; 4-chloro-5-ethyl-3-methyl-pyra -1-yl], [BC69; 4-bromo-5-ethyl-3-methyl-pyrazol-1-yl], [BC70; 3,4-dimethyl-5-ethyl-pyrazol-1-yl], [BC71; 4,5-diethyl-3-methyl-pyrazol-1-yl], [BC72; 5-ethyl-4-propyl-3-methyl-pyrazol-1-yl], [BC73; 5-ethyl-4 -Isopropyl-3-methyl-pyrazol-1-yl], [BC 74; 5-ethyl-4-cyclopropyl-3-methyl-pyrazol-1-yl], [BC 75; 5-ethyl-4-difluoromethyl-3 -Methyl-pyrazol-1-yl], [BC 76; 4-cyano-5-ethyl-3-methyl-pyrazol-1-yl], [BC 77; 5-ethyl-4-ethynyl-3-methyl-pyrazole-1 -Yl], [BC 78; 5-ethyl-3-methyl-4- (1-propynyl) -pyrazol-1-yl], [BC 79; 3,5-dimethyl-4-methoxy-pyrazol-1-yl], [BC 80; 4-ethoxy-3,5-dimethyl-pyrazol-1-yl], [BC 81; 3,5-dimethyl-4- (2-propynyloxy) -pyrazol-1-yl], [BC 82; 5-dimethyl-4-trifluoromethyl-pi Razol-1-yl], [BC 83; 3-ethyl-pyrazol-1-yl], [BC 84; 4-fluoro-3-ethyl-pyrazol-1-yl], [BC 85; 4-chloro-3-ethyl- Pyrazol-1-yl], [BC 86; 4-bromo-3-ethyl-pyrazol-1-yl], [BC 87; 3-ethyl-4-methyl-pyrazol-1-yl], [BC 88; Diethyl-pyrazol-1-yl], [BC 89; 3-ethyl-4-propyl-pyrazol-1-yl], [BC 90; 3-ethyl-4-isopropyl-pyrazol-1-yl], [BC 91; Cyclopropyl-3-ethyl-pyrazol-1-yl], [BC 92; 3-ethyl-4-difluoromethyl-pyrazol-1-yl], [BC 93; 4-cyano-3-ethyl-pyrazol-1-yl] , [BC94; 3-ethyl-4-ethynyl-pyrazol-1-yl], [BC95; 3-ethyl-4- (1-propynyl) -pyrazol-1-yl], [BC96; 3-ethyl-5- Methyl-pyrazol-1-yl], [BC97; 3-ethyl-4-fluoro-5-methyl-pyrazol-1-yl], [BC 98; 4-chloro-3-ethyl-5-methyl-pyrazole-1-l Y], [BC99; 4-bromo- 3-ethyl-5-methyl-pyrazol-1-yl], [BC100; 3-ethyl-4,5-dimethyl-pyrazol-1-yl],

[BC101; 3,4-diethyl-5-methyl-pyrazol-1-yl], [BC 102; 3-ethyl-5-methyl-4- (1-propynyl) -pyrazol-1-yl], [BC 103; 3 -Ethyl-4-isopropyl-5-methyl-pyrazol-1-yl], [BC104; 4-difluoromethyl-3-ethyl-5-methyl-pyrazol-1-yl], [BC105; 3-ethyl-5- Methyl-4-trifluoromethyl-pyrazol-1-yl], [BC106; 3-ethyl-4-ethynyl-5-methyl-pyrazol-1-yl], [BC107; 3-ethyl-5-methyl-4- (1-propynyl) -pyrazol-1-yl], [BC108; 3-cyclopropyl-pyrazol-1-yl], [BC109; 3-cyclopropyl-4-fluoro-pyrazol-1-yl], [BC110; 4-chloro-3-cyclopropyl-pyrazol-1-yl], [BC 111; 4-bromo-3-cyclopropyl-pyrazol-1-yl], [BC 112; 3-cyclopropyl-4-methyl-pyrazole-1 -Yl], [BC113; 3-cyclopropyl-4-ethyl-pyrazol-1-yl], [BC114; 3-cyclopropyl-4-propyl-pyra -L-yl], [BC115; 3,5-dimethyl-4- (2-propynyloxy) -pyrazol-1-yl], [BC116; 3,5-dimethyl-4- (2-butynyloxy)- Pyrazol-1-yl], [BC117; 3-cyclopropyl-4-isopropyl-pyrazol-1-yl], [BC118; 3,5-dicyclopropyl-pyrazol-1-yl], [BC119; 3-cyclo Propyl-4-difluoromethyl-pyrazol-1-yl], [BC120; 3-cyclopropyl-4-trifluoromethyl-pyrazol-1-yl], [BC121; 3-cyclopropyl-4-ethynyl-pyrazole-1 -Yl], [BC122; 3-cyclopropyl-4- (1-propynyl) -pyrazol-1-yl], [BC123; 3-cyclopropyl-5-methyl-pyrazol-1-yl], [BC124; 3 -Cyclopropyl-4-fluoro-5-methyl-pyrazol-1-yl], [BC 125; 4-chloro-3-cyclopropyl-5-methyl-pyrazol-1-yl], [BC 126; 4-bromo-3 -Cyclopropyl-5-methyl-pyrazol-1-yl], [BC127; 3-cyclopropyl-4,5-dimethy] -Pyrazol-1-yl], [BC128; 3-cyclopropyl-4-ethyl-5-methyl-pyrazol-1-yl], [BC129; 3-cyclopropyl-4-propyl-5-methyl-pyrazole-1 -Yl], [BC130; 3-cyclopropyl-4-isopropyl-5-methyl-pyrazol-1-yl], [BC131; 3,5-dicyclopropyl-4-methyl-pyrazol-1-yl], [BC BC 132; 3-Cyclopropyl-4-difluoromethyl-5-methyl-pyrazol-1-yl], [BC 133; 3-cyclopropyl-4-trifluoromethyl-5-methyl-pyrazol-1-yl], [BC 134 3-Cyclopropyl-4-ethynyl-5-methyl-pyrazol-1-yl], [BC 135; 3-cyclopropyl-4- (1-propynyl) -5-methyl-pyrazol-1-yl], [BC 136 3-difluoromethyl-pyrazol-1-yl], [BC 137; 3-difluoromethyl-4-methyl-pyrazol-1-yl], [BC 138; 3-difluoromethyl-4-ethyl-pyrazol-1-yl] , [BC139; 3-difluoromethyl-4-propyl-pyrazole-1- [BC140; 3-difluoromethyl-4-isopropyl-pyrazol-1-yl], [BC141; 3-difluoromethyl-4-cyclopropyl-pyrazol-1-yl], [BC142; 3-difluoromethyl- 4-ethynyl-pyrazol-1-yl], [BC 143; 3-difluoromethyl-4- (1-propynyl) -pyrazol-1-yl], [BC 144; 3-difluoromethyl-4-isobutyl-pyrazole-1-l , [BC145; 3-difluoromethyl-4-fluoro-pyrazol-1-yl], [BC146; 4-chloro-3-difluoromethyl-pyrazol-1-yl], [BC147; 4-bromo-3- Difluoromethyl-pyrazol-1-yl], [BC 148; 3-trifluoromethyl-pyrazol-1-yl], [BC 149; 4-fluoro-3-trifluoromethyl-pyrazol-1-yl], [BC 150; 4 4-Chloro-3-trifluoromethyl-pyrazol-1-yl], [BC 151; 4-bromo-3-trifluoromethyl-pyrazol-1-yl], [BC 152; 4-methyl-3-trifluoromethyl-pyrazole -1-yl], [BC 153; 4- Ethyl-3-trifluoromethyl-pyrazol-1-yl], [BC 154; 4-propyl-3-trifluoromethyl-pyrazol-1-yl], [BC 155; 4-isopropyl-3-trifluoromethyl-pyrazole- 1-yl], [BC156; 4-cyclopropyl-3-trifluoromethyl-pyrazol-1-yl], [BC157; 4-difluoromethyl-3-trifluoromethyl-pyrazol-1-yl], [BC158; 3,4-bis-trifluoromethyl-pyrazol-1-yl], [BC 159; 4-ethynyl-3-trifluoromethyl-pyrazol-1-yl], [BC 160; 4- (1-propynyl) -3-] Trifluoromethyl-pyrazol-1-yl], [BC161; 3,5-dimethyl-4-trifluoromethyl-pyrazol-1-yl], [BC162; 3-propyl-pyrazol-1-yl], [BC163; 3-propyl-4-methyl-pyrazol-1-yl], [BC 164; 3-propyl-4,5-dimethyl-pyrazol-1-yl], [BC 165; 3-isopropyl-pyrazol-1-yl], BC 166; 3-isopropyl-4-methyl-pyrazo -1-yl], [BC 167; 3-isopropyl-4,5-dimethyl-pyrazol-1-yl], [BC 168; 3-tert-butyl-pyrazol-1-yl], [BC 169; 4-methyl-3 -tert-Butyl-pyrazol-1-yl], [BC170; 4,5-dimethyl-3-tert-butyl-pyrazol-1-yl], [BC171; 5-methyl-3-propyl-pyrazol-1-yl] ], [BC172; 3-isopropyl-5-methyl-pyrazol-1-yl], [BC173; 5-methyl-3-tert-butyl-pyrazol-1-yl], [BC 174; 3-ethyl-4-methoxy -5-Methyl-pyrazol-1-yl], [BC 175; 1-methyl-1H-pyrazol-3-yl], [BC 176; 1-ethyl-1H-pyrazol-3-yl], [BC 177; 1-isopropyl] -1H-pyrazol-3-yl], [BC 178; 1- (2, 2-difluoroethyl) -1 H-pyrazol-3-yl], [BC 179; 1- (2-propynyl) -1 H-pyrazole-3- 3 1- (2-butynyl) -1H-pyrazol-3-yl], [BC181; 1-cyclopropylmethyl-1H-pyrazol-3-yl], [BC 182; 1- (2,2 , 2-Trifluoroethyl) -1H-pyrazo 1-propyl-1H-pyrazol-3-yl], [BC184; 1-butyl-1H-pyrazol-3-yl], [BC185; 1-isobutyl-1H-pyrazole] -3-yl], [BC 186; 1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC 187; 1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC188; 1,4-dimethyl-1H-pyrazol-3-yl], [BC189; 1-ethyl-4-methyl-1H-pyrazol-3-yl], [BC190; 1-isopropyl-4-methyl-1H -Pyrazol-3-yl], [BC191; 1- (2,2-difluoroethyl) -4-methyl-1H-pyrazol-3-yl], [BC192; 1- (2-propynyl) -4-methyl- 1H-pyrazol-3-yl], [BC193; 1- (2-butynyl) -4-methyl-1H-pyrazol-3-yl], [BC194; 1-cyclopropylmethyl-4-methyl-1H-pyrazole- 3-yl], [BC195; 1- (2,2,2-trifluoroethyl) -4-methyl-1H-pyrazol-3-yl], [BC196; 4-methyl-1-propyl-1H-pyrazole- 3-yl], [BC 197; 1-butyl-4-methyl-1H-pyrazol-3-yl], [BC 198; 1-i Butyl-4-methyl-1H-pyrazol-3-yl], [BC199; 1- (3-methyl-butyl) -4-methyl-1H-pyrazol-3-yl], [BC200; 1- (4-methyl) -Pentyl) -4-methyl-1H-pyrazol-3-yl],

[BC201; 5-ethyl-1-methyl-1H-pyrazol-3-yl], [BC202; 4-ethyl-1-isopropyl-1H-pyrazol-3-yl], [BC203; 4-ethyl-1- ( 2,2-Difluoroethyl) -1H-pyrazol-3-yl], [BC 204; 4-ethyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC205; 1- (2-butynyl) ) 4-Ethyl-1H-pyrazol-3-yl], [BC206; 4-ethyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC207; Ethyl-1- (2,2-difluoroethyl) -1H-pyrazol-3-yl], [BC208; 4-ethyl-1-propyl-1H-pyrazol-3-yl], [BC209; 1-butyl-4 -Ethyl-1H-pyrazol-3-yl], [BC210; 4-ethyl-1-isobutyl-1H-pyrazol-3-yl], [BC211; 4-ethyl-1- (3-methyl-butyl) -1H 4-Pyrazol-3-yl], [BC 212; 4-ethyl-1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 213; 4-fluoro-1-methyl-1H-pyrazole-3 -Yl], [BC214; 1-ethyl-4-fluoro-1H-pyrazol-3-yl], [BC215; 4-fluo -1-isopropyl-1H-pyrazol-3-yl], [BC 216; 4-fluoro-1- (2,2-difluoroethyl) -1H-pyrazol-3-yl], [BC 217; (2-propynyl) -1H-pyrazol-3-yl], [BC 218; 1- (2-butynyl) -4-fluoro-1H-pyrazol-3-yl], [BC 219; 1-cyclopropylmethyl-4- Fluoro-1 H-pyrazol-3-yl], [BC 220; 4-fluoro-1- (2,2,2-trifluoroethyl) -1 H-pyrazol-3-yl], [BC 221; 4-fluoro-1- Propyl-1H-pyrazol-3-yl], [BC222; 1-butyl-4-fluoro-1H-pyrazol-3-yl], [BC223; 4-fluoro-1-isobutyl-1H-pyrazol-3-yl] , [BC224; 4-fluoro-1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC225; 4-fluoro-1- (4-methyl-pentyl) -1H-pyrazole-3- 3 4-chloro-1-methyl-1H-pyrazol-3-yl], [BC227; 4-chloro-1-ethyl-1H-pyrazol-3-yl], [BC228; 4-chloro- 1-isopropyl-1H-pyrazol-3-yl], [BC2 29; 4-chloro-1-cyclopropylmethyl-1H-pyrazol-3-yl], [BC 230; 4-chloro-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl] , [BC231; 4-chloro-1-propyl-1H-pyrazol-3-yl], [BC232; 1-butyl-4-chloro-1H-pyrazol-3-yl], [BC233; Isobutyl-1H-pyrazol-3-yl], [BC234; 4-chloro-1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC235; 4-chloro-1- (4-methyl) -Pentyl) -1H-pyrazol-3-yl], [BC 236; 1,4-diethyl-1H-pyrazol-3yl], [BC 237; 4-bromo-1-methyl-1H-pyrazol-3-yl], [BC238; 4-bromo-1-ethyl-1H-pyrazol-3-yl], [BC239; 4-bromo-1-isopropyl-1H-pyrazol-3-yl], [BC240; 4-bromo-1- ( 2,2-Difluoroethyl) -1H-pyrazol-3-yl], [BC 241; 4-bromo-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 242; 4-bromo-1- (2-butynyl) -1H-pyrazol-3-yl], [BC 243; 4-bromo-1-cyclopro Rumethyl-1H-pyrazol-3-yl], [BC244; 4-bromo-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC245; 4-bromo-1- Propyl-1H-pyrazol-3-yl], [BC 246; 4-bromo-1-butyl-1H-pyrazol-3-yl], [BC 247; 4-bromo-1-isobutyl-1H-pyrazol-3-yl] , [BC248; 4-bromo-1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC249; 4-bromo-1- (4-methyl-pentyl) -1H-pyrazole-3- 3 , [BC250; 1,5-dimethyl-1H-pyrazol-3-yl], [BC251; 1-ethyl-5-methyl-1H-pyrazol-3-yl], [BC252; 1-isopropyl-5-one] Methyl-1H-pyrazol-3-yl], [BC 253; 1- (2,2-difluoroethyl) -5-methyl-1H-pyrazol-3-yl], [BC254; 5-methyl-1- (2-) Propynyl) -1H-pyrazol-3-yl], [BC 255; 1- (2-butynyl) -5-methyl-1H-pyrazol-3-yl], [BC 256; 1-cyclopropylmethyl-5-methyl-1H -Pyrazol-3-yl], [BC 257; 5-methyl-1- (2,2,2-trifluoroe) Le) -1H-pyrazol-3-yl], [BC258; 5-methyl-1-propyl-1H-pyrazol-3-yl], [BC259; 1-butyl-5-methyl-1H-pyrazol-3-yl ], [BC260; 1-isobutyl-5-methyl-1H-pyrazol-3-yl], [BC261; 1- (3-methyl-butyl) -5-methyl-1H-pyrazol-3-yl], [BC262] 1- (4-Methyl-pentyl) -5-methyl-1H-pyrazol-3-yl], [BC263; 1,4,5-trimethyl-1H-pyrazol-3-yl], [BC264; 1-ethyl -4,5-Dimethyl-1H-pyrazol-3-yl], [BC 265; 4,5-Dimethyl-1-isopropyl-1H-pyrazol-3-yl], [BC 266; 1- (2,2-difluoroethyl) ) -4,5-Dimethyl-1H-pyrazol-3-yl], [BC 267; 4,5-Dimethyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 268; 1- (2) -Butynyl) -4,5-dimethyl-1H-pyrazol-3-yl], [BC 269; 1-cyclopropylmethyl-4,5-dimethyl-1H-pyrazol-3-yl], [BC 270; 4,5- Dimethyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 271; 4,5-dime 1-Butyl-4,5-dimethyl-1H-pyrazol-3-yl], [BC 273; 4,5-dimethyl-1-isobutyl- 1 H-Pyrazol-3-yl], [BC 274; 4, 5-dimethyl-1- (3-methyl-butyl) -1 H-pyrazol-3-yl], [BC 275; 4, 5-dimethyl-1- (4) -Methyl-pentyl) -1H-pyrazol-3-yl], [BC 276; 4-ethyl-1,5-dimethyl-1H-pyrazol-3-yl], [BC 277; 1,4-diethyl-5-methyl- 1H-pyrazol-3-yl], [BC 278; 1-isopropyl-4-ethyl-5-methyl-1H-pyrazol-3-yl], [BC 279; 4-ethyl-1- (2, 2-difluoroethyl) -5-methyl-1H-pyrazol-3-yl], [BC 280; 4-ethyl-5-methyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 281; 1- (2-) Butynyl (4-ethyl-5-methyl-1H-pyrazol-3-yl), [BC282; 1-cyclopropylmethyl-4-ethyl-5-methyl-1H-pyrazol-3-yl], [BC 283; 4- Ethyl-1- (2,2,2-trifluoroethyl) -5-methyl-1H-pyrazole-3-yl [BC284; 4-ethyl-1-propyl-5-methyl-1H-pyrazol-3-yl], [BC285; 1-butyl-4-ethyl-5-methyl-1H-pyrazol-3-yl] , [BC 286; 4-ethyl-1-isobutyl-5-methyl-1H-pyrazol-3-yl], [BC 287; 4-ethyl-1- (3-methyl-butyl) -5-methyl-1H-pyrazole- 3-yl], [BC288; 4-ethyl-1- (4-methyl-pentyl) -5-methyl-1H-pyrazol-3-yl], [BC 289; 4-fluoro-1,5-dimethyl-1H- 1-ethyl-4-fluoro-5-methyl-1H-pyrazol-3-yl], [BC 291; 4-fluoro-1-isopropyl-5-methyl-1H-pyrazole- 3-yl], [BC292; 1- (2,2-difluoroethyl) -4-fluoro-5-methyl-1 H-pyrazol-3-yl], [BC293; 4-fluoro-5-methyl-1- ( 2-propynyl) -1H-pyrazol-3-yl], [BC 294; 1- (2-butynyl) -4-fluoro-5-methyl-1 H-pyrazol-3-yl], [BC 295; 1-cyclopropylmethyl -4-Fluoro-5-methyl-1H-pyrazol-3-yl], [BC 296; 1- (2,2,2-trifluoroethyl) -4-fluoro-5-methyl-1H-pyrazol-3-yl], [BC 297; 1-propyl-4-fluoro-5-methyl-1H-pyrazole-3- 1-Butyl-4-fluoro-5-methyl-1H-pyrazol-3-yl], [BC 299; 1-isobutyl-4-fluoro-5-methyl-1H-pyrazol-3-yl] [BC 300; 4-fluoro-1- (3-methyl-butyl) -5-methyl-1H-pyrazol-3-yl],

[BC301; 4-fluoro-1- (4-methyl-pentyl) -5-methyl-1H-pyrazol-3-yl], [BC 302; 4-chloro-1,5-dimethyl-1H-pyrazol-3-yl ], [BC303; 4-chloro-1-ethyl-5-methyl-1H-pyrazol-3-yl], [BC304; 4-chloro-1-isopropyl-5-methyl-1H-pyrazol-3-yl], [BC 305; 4-chloro-1- (2,2-difluoroethyl) -5-methyl-1H-pyrazol-3-yl], [BC 306; 4-chloro-5-methyl-1- (2-propynyl)- 1H-pyrazol-3-yl], [BC 307; 1- (2-butynyl) -4-chloro-5-methyl-1H-pyrazol-3-yl], [BC 308; 4-chloro-1-cyclopropylmethyl- 5-methyl-1H-pyrazol-3-yl], [BC 309; 4-chloro-1- (2,2,2-trifluoroethyl) -5-methyl-1H-pyrazol-3-yl], [BC310; 4-chloro-5-methyl-1-propyl-1H-pyrazol-3-yl], [BC311; 1-butyl-4-chloro-5-methyl-1H-pyrazol-3-yl], [BC312; 4- Chloro-1-isobutyl-5-methyl-1H-pyrazol-3-yl], [BC313; 4-chloro-1 -(3-Methyl-butyl) -5-methyl-1H-pyrazol-3-yl], [BC 314; 4-chloro-1- (4-methyl-pentyl) -5-methyl-1H-pyrazol-3-yl ], [BC315; 4-bromo-1,5-dimethyl-1H-pyrazol-3-yl], [BC316; 4-bromo-1-ethyl-5-methyl-1H-pyrazol-3-yl], [BC317] 4-bromo-1-isopropyl-5-methyl-1H-pyrazol-3-yl], [BC 318; 4-bromo-1- (2,2-difluoroethyl) -5-methyl-1H-pyrazole-3- 4-bromo-5-methyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC320; 4-bromo-1- (2-butynyl) -5-methyl- 1 H-pyrazol-3-yl], [BC 321; 4-bromo-1-cyclopropylmethyl-5-methyl-1 H-pyrazol-3-yl], [BC 322; 4-bromo-5-methyl-1- (2) , 2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC323; 4-bromo-5-methyl-1-propyl-1H-pyrazol-3-yl], [BC324; 4-bromo- 1-Butyl-5-methyl-1H-pyrazol-3-yl], [BC 325; 4-bromo-1-isobutyl] -5-methyl-1H-pyrazol-3-yl], [BC 326; 4-bromo-1- (3-methyl-butyl) -5-methyl-1H-pyrazol-3-yl], [BC 327; 4-bromo -1- (4-Methyl-pentyl) -5-methyl-1H-pyrazol-3-yl], [BC 328; 5-ethyl-1-methyl-1H-pyrazol-3-yl], [BC 329; -Diethyl-1H-pyrazol-3-yl], [BC330; 5-ethyl-1-isopropyl-1H-pyrazol-3-yl], [BC331; 5-ethyl-1- (2,2-difluoroethyl)- 1H-pyrazol-3-yl], [BC332; 5-ethyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC333; 1- (2-butynyl) -5-ethyl-1H- Pyrazol-3-yl], [BC 334; 1-cyclopropylmethyl-5-ethyl-1H-pyrazol-3-yl], [BC 335; 1- (2,2,2-trifluoroethyl) -5-ethyl- 1H-pyrazol-3-yl], [BC 336; 5-ethyl-1-propyl-1H-pyrazol-3-yl], [BC 337; 1-butyl-5-ethyl-1H-pyrazol-3-yl], [BC BC 338; 5-ethyl-1-isobutyl-1H-pyrazol-3-yl], [BC 339; 5-ethyl-1- (3-) -Butyl) -1H-pyrazol-3-yl], [BC 340; 5-ethyl-1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 341; 5-ethyl-1,4 -Dimethyl-1H-pyrazol-3-yl], [BC 342; 1, 5-diethyl-4-methyl-1H-pyrazol-3-yl], [BC 343; 5-ethyl-1-isopropyl-4-methyl-1 H -Pyrazol-3-yl], [BC 344; 5-ethyl-1- (2,2-difluoroethyl) -4-methyl-1 H-pyrazol-3-yl], [BC 345; 5-ethyl-1- (2) -Propynyl) -4-methyl-1H-pyrazol-3-yl], [BC 346; 1- (2-butynyl) -5-ethyl-4-methyl-1 H-pyrazol-3-yl], [BC 347; 1- Cyclopropylmethyl-5-ethyl-4-methyl-1H-pyrazol-3-yl], [BC 348; 5-ethyl-4-methyl-1- (2,2,2-trifluoroethyl) -1H-pyrazole- 3-yl], [BC 349; 5-ethyl-4-methyl-1-propyl-1H-pyrazol-3-yl], [BC 350; 1-butyl-5-ethyl-4-methyl-1H-pyrazole-3- 3 , [BC 351; 5-ethyl-1-isobutyl-4-methyl-1H-pyrazole-3- 3 [BC352; 5-ethyl-1- (3-methyl-butyl) -4-methyl-1H-pyrazol-3-yl], [BC 353; 5-ethyl-1- (4-methyl-pentyl)- 4-Methyl-1H-pyrazol-3-yl], [BC 354; 4,5-diethyl-1-methyl-1H-pyrazol-3-yl], [BC 355; 1,4,5-triethyl-1H-pyrazole- 3-yl], [BC 356; 4,5-diethyl-1-isopropyl-1H-pyrazol-3-yl], [BC 357; 4,5-diethyl-1- (2,2-difluoroethyl) -1H-pyrazole -4-yl], [BC 358; 4,5-diethyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 359; 1- (2-butynyl) -4,5-diethyl-1H -Pyrazol-3-yl], [BC 360; 1-cyclopropylmethyl-4,5-diethyl-1H-pyrazol-3-yl], [BC 361; 4,5-diethyl-1- (2,2,2-) Trifluoroethyl) -1H-pyrazol-3-yl], [BC 362; 4,5-diethyl-1-propyl-1H-pyrazol-3-yl], [BC 363; 1-butyl-4,5-diethyl-1H -Pyrazol-3-yl], [BC 364; 4,5-diethyl-1-pentyl-1H-pyrazol-3-yl], [BC 365; 4,5- Diethyl-1-isobutyl-1H-pyrazol-3-yl], [BC 366; 4,5-diethyl-1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC 367; 4,5- Diethyl-1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 368; 5-ethyl-4-fluoro-1-methyl-1H-pyrazol-3-yl], [BC 369; 1, 5-diethyl-4-fluoro-1H-pyrazol-3-yl], [BC 370; 5-ethyl-4-fluoro-1-isopropyl-1H-pyrazol-3-yl], [BC 371; 1- (2, 2 -Difluoroethyl) -5-ethyl-4-fluoro-1H-pyrazol-3-yl], [BC 372; 5-ethyl-4-fluoro-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 373; 1- (2-butynyl) -5-ethyl-4-fluoro-1H-pyrazol-3-yl], [BC 374; 1-cyclopropylmethyl-5-ethyl-4-fluoro-1H-pyrazole-3 -Yl], [BC 375; 5-ethyl-4-fluoro-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 376; 5-ethyl-4-fluoro-1 -Propyl-1H-pyrazol-3-yl], [BC 377; 1- 5-ethyl-4-fluoro-1H-pyrazol-3-yl], [BC 378; 5-ethyl-4-fluoro-1-pentyl-1H-pyrazol-3-yl], [BC 379; 5-ethyl- 4-Fluoro-1-isobutyl-1H-pyrazol-3-yl], [BC 380; 5-ethyl-4-fluoro- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC 381; 5- Ethyl-4-fluoro- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 382; 4-bromo-5-ethyl-1-methyl-1 H-pyrazol-3-yl], [BC 383; 4-bromo-5-ethyl-1-ethyl-1H-pyrazol-3-yl], [BC 384; 4-bromo-5-ethyl-1-isopropyl-1H-pyrazol-3-yl], [BC 385; 4- Bromo-1- (2,2-difluoroethyl) -5-ethyl-1H-pyrazol-3-yl], [BC 386; 4-bromo-5-ethyl-1- (2-propynyl) -1H-pyrazole-3 -Yl], [BC 387; 4-bromo-1- (2-butynyl) -5-ethyl-1H-pyrazol-3-yl], [BC 388; 4-bromo-1-cyclopropylmethyl-5-ethyl-1H -Pyrazol-3-yl], [BC 389; 4-bromo-1-5-ethy -(2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC390; 4-bromo-5-ethyl-1-propyl-1H-pyrazol-3-yl], [BC 391; 4 4-Bromo-1-butyl-5-ethyl-1H-pyrazol-3-yl], [BC 392; 4-bromo-5-ethyl-1-pentyl-1H-pyrazol-3-yl], [BC 393; 4-bromo -5-ethyl-1-isobutyl-1H-pyrazol-3-yl], [BC 394; 4-bromo-5-ethyl- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC 395; 4 -Bromo-5-ethyl- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 396; 5-cyclopropyl-1-methyl-1 H-pyrazol-3-yl], [BC 397; 5- Cyclopropyl-1-ethyl-1H-pyrazol-3-yl], [BC 398; 5-cyclopropyl-1-isopropyl-1H-pyrazol-3-yl], [BC 399; 5-cyclopropyl-1- (2, 2-Difluoroethyl) -1H-pyrazol-3-yl], [BC400; 5-cyclopropyl-1- (2-propynyl) -1H-pyrazol-3-yl],

[BC401; 1- (2-butynyl) -5-cyclopropyl-1H-pyrazol-3-yl], [BC402; 1-cyclopropylmethyl-5-cyclopropyl-1H-pyrazol-3-yl], [BC403 5-Cyclopropyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 404; 5-cyclopropyl-1-propyl-1H-pyrazol-3-yl], [BC405; 1-butyl-5-cyclopropyl-1H-pyrazol-3-yl], [BC406; 5-cyclopropyl-1-pentyl-1H-pyrazol-3-yl], [BC407; 5-cyclopropyl- 1-isobutyl-1H-pyrazol-3-yl], [BC408; 5-cyclopropyl-1- (3-methylbutyl) -1H-pyrazol-3-yl], [BC409; 5-cyclopropyl-1- (4) -Methylpentyl) -1H-pyrazol-3-yl], [BC410; 5-cyclopropyl-1,4-dimethyl-1H-pyrazol-3-yl], [BC411; 5-cyclopropyl-1-ethyl-4 -Methyl-1H-pyrazol-3-yl], [BC 412; 5-cyclopropyl-1-isopropyl-4-methyl-1H-pyrazol-3-yl], [BC 413; 5-cyclopropyl-1- (2,2-difluoroethyl) -4-methyl-1H-pyrazol-3-yl], [BC 414; 5-cyclopropyl-4-methyl-1- (2-propynyl) -1H-Pyrazol-3-yl], [BC 415; 1- (2-butynyl) -5-cyclopropyl-4-methyl-1H-pyrazol-3-yl], [BC 416; 1-cyclopropylmethyl-5-l Cyclopropyl-4-methyl-1H-pyrazol-3-yl], [BC 417; 5-cyclopropyl-1- (2,2,2-trifluoroethyl) -4-methyl-1H-pyrazol-3-yl] , [BC418; 5-cyclopropyl-4-methyl-1-propyl-1H-pyrazol-3-yl], [BC419; 1-butyl-5-cyclopropyl-4-methyl-1H-pyrazol-3-yl] [BC 420; 5-cyclopropyl-4-methyl-1-pentyl-1H-pyrazol-3-yl], [BC 421; 5-cyclopropyl-1-isobutyl-4-methyl-1H-pyrazol-3-yl] , [BC 422; 5-cyclopropyl-4-methyl-1- (3-methyl-butyl) -1 H-pyrazol-3-yl], [BC 423; 5-cyclopropyl-4-methyl-1- (4-methyl). Le-pentyl) -1H-pyrazol-3-yl], [BC 424; 5-cyclopropyl-4-fluoro-1-methyl-1H-pyrazol-3-yl], [BC 425; 5-cyclopropyl-4-fluoro] -1-ethyl-1H-pyrazol-3-yl], [BC 426; 5-cyclopropyl-4-fluoro-1-isopropyl-1H-pyrazol-3-yl], [BC 427; 5-cyclopropyl-4-fluoro] -1- (2,2-difluoroethyl) -1H-pyrazol-3-yl], [BC 428; 5-cyclopropyl-4-fluoro-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 429; 1- (2-butynyl) -5-cyclopropyl-4-fluoro-1H-pyrazol-3-yl], [BC 430; 5-cyclopropyl-1-cyclopropylmethyl-4-fluoro-1H-pyrazole 5-Cyclopropyl-4-fluoro-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC432; 5-cyclopropyl-4 -Fluoro-1-propyl-1H-pyrazol-3-yl], [BC 433; 1-butyl-5-cyclopropyl-4-fluoro-1H-pyrazo 5-cyclopropyl-4-fluoro-1-pentyl-1H-pyrazol-3-yl], [BC 435; 5-cyclopropyl-4-fluoro-1-isobutyl-1H- Pyrazol-3-yl], [BC 436; 5-cyclopropyl-4-fluoro-1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC 437; 5-cyclopropyl-4-fluoro- 1- (4-Methyl-pentyl) -1H-pyrazol-3-yl], [BC 438; 4-chloro-5-cyclopropyl-1-methyl-1H-pyrazol-3-yl], [BC 439; 4-chloro -5-cyclopropyl-1-ethyl-1H-pyrazol-3-yl], [BC 440; 4-chloro-5-cyclopropyl-1-isopropyl-1H-pyrazol-3-yl], [BC 441; 4-chloro -5-Cyclopropyl-1- (2,2-difluoroethyl) -1H-pyrazol-3-yl], [BC 442; 4-chloro-5-cyclopropyl-1- (2-propynyl) -1H-pyrazole- 3-yl], [BC 443; 1- (2-butynyl) -4-chloro-5-cyclopropyl-1H-pyrazol-3-yl], [BC 444; 4-chloro-1-cyclopropyl ester Ethyl 5-Cyclopropyl-1H-pyrazol-3-yl], [BC 445; 4-Chloro-5-cyclopropyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl] , [BC446; 4-chloro-5-cyclopropyl-1-propyl-1H-pyrazol-3-yl], [BC 447; 4-chloro-5-cyclopropyl-1-butyl-1H-pyrazol-3-yl] , [BC448; 4-chloro-5-cyclopropyl-1-pentyl-1H-pyrazol-3-yl], [BC449; 4-chloro-5-cyclopropyl-1-isobutyl-1H-pyrazol-3-yl] , [BC450; 4-bromo-5-cyclopropyl-1-methyl-1H-pyrazol-3-yl], [BC 451; 4-bromo-5-cyclopropyl-1-ethyl-1H-pyrazol-3-yl] [BC 452; 4-bromo-5-cyclopropyl-1-isopropyl-1H-pyrazol-3-yl], [BC 453; 4-bromo-5-cyclopropyl-1- (2,2-difluoroethyl) -1 H 4-Pyrazol-3-yl], [BC 454; 4-bromo-5-cyclopropyl-1- (2-propynyl) -1 H-pyrazol-3-yl], [BC 455; 4-bromo- 1- (2-butynyl) -5-cyclopropyl-1H-pyrazol-3-yl], [BC 456; 4-bromo-1-cyclopropylmethyl-5-cyclopropyl-1H-pyrazol-3-yl], BC 457; 4-bromo-5-cyclopropyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 458; 4-bromo-5-cyclopropyl-1-propyl- 1H-pyrazol-3-yl], [BC 459; 4-bromo-1-butyl-5-cyclopropyl-1H-pyrazol-3-yl], [BC 460; 4-bromo-5-cyclopropyl-1-pentyl- 1H-pyrazol-3-yl], [BC 461; 4-bromo-5-cyclopropyl-1-isobutyl-1H-pyrazol-3-yl], [BC 462; 5-isopropyl-1-methyl-1H-pyrazole-3 -Yl], [BC463; 1-ethyl-5-isopropyl-1H-pyrazol-3-yl], [BC464; 1,5-diisopropyl-1H-pyrazol-3-yl], [BC465; 1- (2, 2-Difluoroethyl) -5-isopropyl-1H-pyrazol-3-yl], [BC 466; 5-isopropyl-1- (2-propynyl) -1H-pyrazol-3-yl ], [BC 467; 1- (2-butynyl) -5-isopropyl-1 H-pyrazol-3-yl], [BC 468; 1-cyclopropylmethyl-5-isopropyl-1 H-pyrazol-3-yl], [BC 469] 5-isopropyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 470; 5-isopropyl-1-propyl-1H-pyrazol-3-yl], [BC 471; 1-butyl-5-isopropyl-1H-pyrazol-3-yl], [BC 472; 5-isopropyl-1-pentyl-1H-pyrazol-3-yl], [BC 473; 1-isobutyl-5-isopropyl-1 H; -Pyrazol-3-yl], [BC 474; 5-isopropyl-1- (3-methyl-butyl) -1 H-pyrazol-3-yl], [BC 475; 5-isopropyl-1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 476; 1,4-dimethyl-5-isopropyl-1H-pyrazol-3-yl], [BC 477; 1-ethyl-5-isopropyl-4-methyl-1H-pyrazole -3-yl], [BC 478; 1,5-diisopropyl-4-methyl-1H-pyrazol-3-yl], [BC 479; 1- (2,2-difluoroethyl) -5-iso] Ropyl-4-methyl-1H-pyrazol-3-yl], [BC 480; 5-isopropyl-4-methyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 481; 1- (2 -Butynyl) -5-isopropyl-4-methyl-1H-pyrazol-3-yl], [BC 482; 1-cyclopropylmethyl-5-isopropyl-4-methyl-1 H-pyrazol-3-yl], [BC 483; 5-isopropyl-4-methyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 484; 5-isopropyl-1-propyl-4-methyl-1H-pyrazole- 3-yl], [BC 485; 1-butyl-5-isopropyl-4-methyl-1H-pyrazol-3-yl], [BC 486; 5-isopropyl-4-methyl-1-pentyl-1H-pyrazole-3- [,,,, 5] 4-isopropyl-4-methyl-1-isobutyl-1H-pyrazol-3-yl], [BC 488; 5-isopropyl-1- (3-methyl-butyl) -4-methyl-1H- Pyrazol-3-yl], [BC 489; 5-isopropyl-4-methyl-1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC 490; 4-fluoro-5-iso Propyl-1-methyl-1H-pyrazol-3-yl], [BC 491; 4-fluoro-5-isopropyl-1-ethyl-1H-pyrazol-3-yl], [BC 492; 4-fluoro-1,5- Diisopropyl-1H-pyrazol-3-yl], [BC 493; 4-fluoro-5-isopropyl-1- (2,2-difluoroethyl) -1H-pyrazol-3-yl], [BC 494; 4-fluoro-5 -Isopropyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 495; 4-fluoro-5-isopropyl-1- (2-butynyl) -1H-pyrazol-3-yl], [BC 496 4-fluoro-5-isopropyl-1-cyclopropylmethyl-1H-pyrazol-3-yl], [BC 497; 4-fluoro-5-isopropyl-1- (2,2,2-trifluoroethyl) -1H 4-Pyrazol-3-yl], [BC 498; 4-fluoro-5-isopropyl-1-propyl-1H-pyrazol-3-yl], [BC 499; 4-fluoro-5-isopropyl-1-butyl-1H-pyrazole -4-yl], [BC 500; 4-fluoro-5-isopropyl-1-pentyl-1H-pyrazol-3-yl],

[BC501; 4-fluoro-5-isopropyl-1-isobutyl-1H-pyrazol-3-yl], [BC502; 4-fluoro-5-isopropyl-1- (3-methyl-butyl) -1H-pyrazole-3 -Yl], [BC 503; 4-fluoro-5-isopropyl-1- (4-methyl-pentyl) -1H-pyrazol-3-yl], [BC504; 4-chloro-5-isopropyl-1-methyl-1 H 4-Pyrazol-3-yl], [BC 505; 4-chloro-5-isopropyl-1-ethyl-1H-pyrazol-3-yl], [BC 506; 4-chloro-1,5-diisopropyl-1H-pyrazole-3 -Yl], [BC507; 4-chloro-1- (2,2-difluoroethyl) -5-isopropyl-1H-pyrazol-3-yl], [BC508; 4-chloro-5-isopropyl-1- (2) -Propynyl) -1H-pyrazol-3-yl], [BC 509; 1- (2-butynyl) -4-chloro-5-isopropyl-1H-pyrazol-3-yl], [BC510; 4-chloro-5- Isopropyl-1-cyclopropylmethyl-1H-pyrazol-3-yl], [BC511; 4-chloro-5-isopropyl-1- (2,2,2-trifluoroethyl) -1H-pyrazo 4-chloro-5-isopropyl-1-propyl-1H-pyrazol-3-yl], [BC513; 4-chloro-5-isopropyl-1-butyl-1H-pyrazole- 3-yl], [BC514; 4-chloro-5-isopropyl-1-pentyl-1H-pyrazol-3-yl], [BC515; 4-chloro-5-isopropyl-1-isobutyl-1H-pyrazole-3- 3 4-chloro-5-isopropyl-1- (3-methyl-butyl) -1H-pyrazol-3-yl], [BC 517; 4-chloro-5-isopropyl-1- (4-methyl) -Pentyl) -1H-pyrazol-3-yl], [BC518; 4-bromo-5-isopropyl-1-methyl-1H-pyrazol-3-yl], [BC519; 4-bromo-1-ethyl-5- Isopropyl-1H-pyrazol-3-yl], [BC520; 4-bromo-1,5-diisopropyl-1H-pyrazol-3-yl], [BC521; 4-bromo-1- (2,2-difluoroethyl) -5-isopropyl-1H-pyrazol-3-yl], [BC 522; 4-bromo-5-isopropyl-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 523; 4-bromo-1 -(2- Tynyl) -5-isopropyl-1H-pyrazol-3-yl], [BC 524; 4-bromo-1-cyclopropylmethyl-5-isopropyl-1H-pyrazol-3-yl], [BC 525; 4-bromo-5 -Isopropyl-1- (2,2,2-trifluoroethyl) -1H-pyrazol-3-yl], [BC 526; 4-bromo-5-isopropyl-1-propyl-1H-pyrazol-3-yl], [BC527; 4-bromo-1-butyl-5-isopropyl-1H-pyrazol-3-yl], [BC528; 4-bromo-5-isopropyl-1-pentyl-1H-pyrazol-3-yl], [BC529 4-bromo-5-isopropyl-1-isobutyl-1H-pyrazol-3-yl], [BC 530; 4-bromo-5-isopropyl-1- (3-methyl-butyl) -1H-pyrazol-3-yl ], [BC 531; 4-bromo-5-isopropyl-1- (4-methyl-pentyl) -1 H-pyrazol-3-yl], [BC 532; 5-methoxy-1-methyl-1 H-pyrazol-3-yl ], [BC 533; 1-ethyl-5-methoxy-1H-pyrazol-3-yl], [BC 534; 5-methoxy-1-isopropyl-1H-pyrazol-3-yl], [BC 535; 1- (2,2-difluoroethyl) -5-methoxy-1H-pyrazol-3-yl], [BC 536; 5-methoxy-1- (2-propynyl) -1H-pyrazol-3-yl], [BC 537; 1- (2-butynyl) -5-methoxy-1H-pyrazol-3-yl], [BC 538; 1-cyclopropylmethyl-5-methoxy-1H-pyrazol-3-yl], [BC 539; 1 , 4-Dimethyl-5-methoxy-1H-pyrazol-3-yl], [BC540; 1-ethyl-5-methoxy-4-methyl-1H-pyrazol-3-yl], [BC 541; 5-methoxy-1 -Isopropyl-4-methyl-1H-pyrazol-3-yl], [BC 542; 1- (2, 2-difluoroethyl) -5-methoxy-4-methyl-1 H-pyrazol-3-yl], [BC 543; 5-methoxy-1- (2-propynyl) -4-methyl-1H-pyrazol-3-yl], [BC 544; 1- (2-butynyl) -5-methoxy-4-methyl-1H-pyrazole-3- 1-Cyclopropylmethyl-5-methoxy-4-methyl-1H-pyrazol-3-yl], [BC546; 4-fluoro-5-methoxy-1-methyl-1H-pyrazole-3-yl], [BC 545; [, 4 5 Xyl-1-ethyl-1H-pyrazol-3-yl], [BC 548; 4-fluoro-5-methoxy-1-isopropyl-1H-pyrazol-3-yl], [BC 549; 1- (2,2-difluoro) Ethyl) -4-fluoro-5-methoxy-1H-pyrazol-3-yl], [BC550; 4-fluoro-5-methoxy-1- (2-propynyl) -1H-pyrazol-3-yl], [BC551 1- (2-butynyl) -4-fluoro-5-methoxy-1H-pyrazol-3-yl], [BC 552; 1-cyclopropylmethyl-4-fluoro-5-methoxy-1H-pyrazol-3-yl ], [BC553; 4-chloro-5-methoxy-1-methyl-1H-pyrazol-3-yl], [BC554; 4-chloro-5-methoxy-1-ethyl-1H-pyrazol-3-yl], [BC 555; 4,5-Dichloro-1-ethyl-1H-pyrazol-3-yl], [BC 556; 4-Chloro-1-ethyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC 557] 1-ethyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC 558; 1-ethyl-4-methyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC559; -Chloro- 1-ethyl-1H-pyrazol-3-yl], [BC 560; 5-chloro-1-ethyl-4-methyl-1H-pyrazol-3-yl], [BC 561; 4, 5-dichloro-1-methyl- 1H-pyrazol-3-yl], [BC 562; 4-chloro-1-methyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC 563; 1-methyl-5-trifluoromethyl-1H- Pyrazol-3-yl], [BC 564; 1,4-dimethyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC 565; 5-chloro-1-methyl-1H-pyrazol-3-yl] , [BC566; 5-chloro-1,4-dimethyl-1H-pyrazol-3-yl], [BC 567; 5,6-dihydro-4H-pyrrolo [1,2-b] pyrazol-2-yl], BC 568; 4,5,6,7-tetrahydro-pyrazolo [1,2-a] pyridin-2-yl], [BC569; 5,6-dihydro-3-methyl-4H-pyrrolo [1,2-b] Pyrazol-2-yl], [BC 570; 4,5,6,7-3-methyl-tetrahydro-pyrazolo [1,2-a] pyridin-2-yl], [BC571; 1-methyl-1H-pyrazole- 4-yl], [BC572; 1,5-dimethyl-1H-pyrazol-4-yl], [BC573; 1-ethyl-1H-pyra 1-ethyl-5-methyl-1H-pyrazol-4-yl], [BC575; 1,3-dimethyl-1H-pyrazol-4-yl], [BC 576; 1 , 3,5-trimethyl-1H-pyrazol-4-yl], [BC577; 1-ethyl-3-methyl-1H-pyrazol-4-yl], [BC578; 3,5-dimethyl-1-ethyl-1H -Pyrazol-4-yl], [BC 579; 1- (2-propynyl) -1H-pyrazol-4-yl], [BC 580; 5-methyl-1- (2-propynyl) -1H-pyrazol-4-yl ], [BC 581; 3-methyl-1- (2-propynyl) -1H-pyrazol-4-yl], [BC 582; 3,5-dimethyl-1- (2-propynyl) -1H-pyrazol-4-yl] ], [BC 583; 1-cyclopropylmethyl-1H-pyrazol-4-yl], [BC584; 1-cyclopropylmethyl-3-methyl-1H-pyrazol-4-yl], [BC585; 1-cyclopropylmethyl] -5-methyl-1H-pyrazol-4-yl], [BC 586; 1-cyclopropylmethyl-3,5-dimethyl-1H-pyrazol-4-yl], [BC 587; 1- (2, 2-difluoroethyl) ) -1H-Pyrazol-4-yl], [BC 588; 1- (2,2-difluo) Roethyl) -3-methyl-1H-pyrazol-4-yl], [BC 589; 1- (2,2-difluoroethyl) -5-methyl-1H-pyrazol-4-yl], [BC 590; 1- (2) , 2-Difluoroethyl) -3,5-dimethyl-1H-pyrazol-4-yl], [BC 591; 1-methyl-1H-pyrazol-5-yl], [BC 592; 1,4-dimethyl-1H-pyrazole 4-chloro-1-methyl-1H-pyrazol-5-yl], [BC594; 4-chloro-1-methyl-1H-pyrazol-5-yl], [BC595; -Bromo-1-methyl-1H-pyrazol-5-yl], [BC596; 1-ethyl-1H-pyrazol-5-yl], [BC 597; 1-ethyl-4-methyl-1H-pyrazol-5-yl ], [BC598; 1-ethyl-4-fluoro-1H-pyrazol-5-yl], [BC599; 4-chloro-1-ethyl-1H-pyrazol-5-yl], [BC600; 4-bromo-1 -Ethyl-1H-pyrazol-5-yl],

[BC601; 1-propyl-1H-pyrazol-5-yl], [BC602; 4-methyl-1-propyl-1H-pyrazol-5-yl], [BC603; 4-fluoro-1-propyl-1H-pyrazole 4-chloro-1-propyl-1H-pyrazol-5-yl], [BC605; 4-bromo-1-propyl-1H-pyrazol-5-yl], [BC 606; 1 -Butyl-1H-pyrazol-5-yl], [BC 607; 1-butyl-4-methyl-1H-pyrazol-5-yl], [BC 608; 1-butyl-4-fluoro-1H-pyrazol-5-yl ], [BC609; 1-butyl-4-chloro-1H-pyrazol-5-yl], [BC610; 1-butyl-4-bromo-1H-pyrazol-5-yl], [BC611; 1,3-dimethyl] -1H-pyrazol-5-yl], [BC612; 1,3,4-trimethyl-1H-pyrazol-5-yl], [BC 613; 1,3-dimethyl-4-fluoro-1H-pyrazol-5-yl ], [BC614; 4-chloro-1,3-dimethyl-1H-pyrazol-5-yl], [BC615; 4-bromo-1,3-dimethyl-1H-pyrazol-5-yl], [BC 616; 1] -Ethyl-3-methyl-1H-pyrazol-5-yl], [BC 617; 3,4-dimethyl-1-ethyl] -1H-pyrazol-5-yl], [BC 618; 1-ethyl-4-fluoro-3-methyl-1H-pyrazol-5-yl], [BC 619; 4-chloro-1-ethyl-3-methyl-1H 4-pyrazol-5-yl], [BC 620; 4-bromo-1-ethyl-3-methyl-1H-pyrazol-5-yl], [BC 621; 3-methyl-1-propyl-1H-pyrazol-5-yl [BC 622; 3,4-dimethyl-1-propyl-1H-pyrazol-5-yl], [BC 623; 3-methyl-4-fluoro-1-propyl-1H-pyrazol-5-yl], [BC 624] 4-chloro-3-methyl-1-propyl-1H-pyrazol-5-yl], [BC 625; 4-bromo-3-methyl-1-propyl-1H-pyrazol-5-yl], [BC 626; 1 -Butyl-3-methyl-1H-pyrazol-5-yl], [BC 627; 1-butyl-3,4-dimethyl-1H-pyrazol-5-yl], [BC 628; 1-butyl-4-fluoro-3 -Methyl-1H-pyrazol-5-yl], [BC629; 1-butyl-4-chloro-3-methyl-1H-pyrazol-5-yl], [BC630; 1-butyl-4-bromo-3-methyl] -1H-pyrazol-5-yl], [BC 631; 3-ethyl-1-methyl-1H-pylazo -4-yl], [BC 632; 1,4-dimethyl-3-ethyl-1H-pyrazol-5-yl], [BC 633; 3-ethyl-4-fluoro-1-methyl-1H-pyrazol-5-yl ], [BC634; 4-chloro-3-ethyl-1-methyl-1H-pyrazol-5-yl], [BC635; 4-bromo-3-ethyl-1-methyl-1H-pyrazol-5-yl], [BC 636; 1,3-diethyl-1H-pyrazol-5-yl], [BC 637; 1,3-diethyl-4-methyl-1H-pyrazol-5-yl], [BC 638; 1,3-diethyl-4 -Fluoro-1H-pyrazol-5-yl], [BC639; 4-chloro-1,3-diethyl-1H-pyrazol-5-yl], [BC640; 4-bromo-1,3-diethyl-1H-pyrazole -5-yl], [BC 641; 4-fluoro-1,3-diethyl-1H-pyrazol-5-yl], [BC 642; 3-ethyl-1-propyl-1H-pyrazol-5-yl], [BC643] 3-ethyl-4-methyl-1-propyl-1H-pyrazol-5-yl], [BC644; 4-fluoro-3-ethyl-1-propyl-1H-pyrazol-5-yl], [BC645; -Chloro-3-ethyl-1-propyl-1H-pyrazol-5-yl], [BC 646; 4-bromo-3-ethyl] -1-propyl-1H-pyrazol-5-yl], [BC 647; 1-butyl-3-ethyl-1H-pyrazol-5-yl], [BC 648; 1-butyl-3-ethyl-4-methyl-1H -Pyrazol-5-yl], [BC 649; 1-butyl-3-ethyl-4-fluoro-1H-pyrazol-5-yl], [BC 650; 1-butyl-4-chloro-3-ethyl-1H-pyrazole 4-bromo-1-butyl-3-ethyl-1H-pyrazol-5-yl], [BC652; 1- (2-propynyl) -1H-pyrazol-5-yl], [BC653; 4-methyl-1- (2-propynyl) -1H-pyrazol-5-yl], [BC654; 3-methyl-1- (2-propynyl) -1H-pyrazol-5-yl], [BC655 3,4-dimethyl-1- (2-propynyl) -1H-pyrazol-5-yl], [BC 656; 1-cyclopropylmethyl-1H-pyrazol-5-yl], [BC 657; 1-cyclopropylmethyl -4-Methyl-1H-pyrazol-5-yl], [BC 658; 1-cyclopropylmethyl-3-methyl-1H-pyrazol-5-yl], [BC 659; 1-cyclopropylmethyl-3,4-dimethyl] -1H-pyrazol-5-yl], [BC 660; 1- (2- Butynyl) -1H-pyrazol-5-yl], [BC 661; 1,5-dimethyl-4-iodo-1H-pyrazol-3-yl], [BC 662; 4-cyano-1,5-dimethyl-1H-pyrazole -3-yl], [BC663; 5-ethyl-1-methyl-4-iodo-1H-pyrazol-3-yl], [BC664; 4-cyano-5-ethyl-1-methyl-1H-pyrazole-3 -Yl], [BC665; 1,5-diethyl-4-iodo-1H-pyrazol-3-yl], [BC666; 4-cyano-1,5-diethyl-1H-pyrazol-3-yl], [BC667] 1,4-dimethyl-5-ethoxy-1H-pyrazol-3-yl], [BC 668; 4-ethyl-1-methyl-5-ethoxy-1H-pyrazol-3-yl], [BC 669; 1-ethyl -4-Methyl-5-ethoxy-1H-pyrazol-3-yl], [BC 670; 1,4-dimethyl-5-methylthio-1H-pyrazol-3-yl], [BC 671; 1,4-dimethyl-5 -Ethylthio-1H-pyrazol-3-yl], [BC 672; 1,4-diethyl-5-methylthio-1H-pyrazol-3-yl], [BC 673; 5-cyano-1,4-dimethyl-1H-pyrazole -3-yl], [BC 674; 5-cyano-1,4-diethyl-1H-pyrazole-3- , [BC 675; 5-cyano-4-ethyl-1-methyl-1H-pyrazol-3-yl], [BC 676; 5-cyano-1-ethyl-4-methyl-1H-pyrazol-3-yl] [BC 677; 5-Difluoromethoxy-1,4-dimethyl-1H-pyrazol-3-yl], [BC 678; 1,4-dimethyl-5-trifluoromethoxy-1H-pyrazol-3-yl], BC 679; 1,4-dimethyl-5- (2-propynyloxy) -1H-pyrazol-3-yl], [BC 680; 1,4-dimethyl-5- (2-butynyloxy) -1H-pyrazol-3-yl 5-chloro-1-methyl-1H-pyrazol-3-yl], [BC682; 5-bromo-1-methyl-1H-pyrazol-3-yl], [BC 683; 5-ethoxy-1] -Methyl-1H-pyrazol-3-yl], [BC684; 5-cyano-1-methyl-1H-pyrazol-3-yl], [BC685; 5-difluoromethyl-1-methyl-1H-pyrazole-3- 3 , [BC686; 4,5-difluoro-1-methyl-1H-pyrazol-3-yl], [BC 687; 5-chloro-4-fluoro-1-methyl-1H-pyrazol-3-yl], BC 688; 5-bromo-4-fluoro-1-methyl-1H-pi Zol-3-yl], [BC 689; 5-ethoxy-4-fluoro-1-methyl-1H-pyrazol-3-yl], [BC 690; 5-cyano-4-fluoro-1-methyl-1H-pyrazole- 3-yl], [BC691; 5-difluoromethyl-4-fluoro-1-methyl-1H-pyrazol-3-yl], [BC692; 5-trifluoromethyl-4-fluoro-1-methyl-1H-pyrazole 4-chloro-5-fluoro-1-methyl-1H-pyrazol-3-yl], [BC694; 5-bromo-4-chloro-1-methyl-1H-pyrazole-3. -Yl], [BC695; 4-chloro-5-ethyl-1-methyl-1H-pyrazol-3-yl], [BC696; 4-chloro-5-ethoxy-1-methyl-1H-pyrazol-3-yl ], [BC 697; 4-chloro-5-cyano-1-methyl-1H-pyrazol-3-yl], [BC 698; 4-chloro-5-difluoromethyl-1-methyl-1H-pyrazol-3-yl] , [BC699; 4-bromo-5-fluoro-1-methyl-1H-pyrazol-3-yl], [BC700; 4-bromo-5-chloro-1-methyl-1H-pyrazol-3-yl],

[BC 701; 4, 5-dibromo-1-methyl-1H-pyrazol-3-yl], [BC 702; 4-bromo-5-methoxy-1-methyl-1 H-pyrazol-3-yl], [BC 703; 4 4-bromo-5-ethoxy-1-methyl-1H-pyrazol-3-yl], [BC704; 4-bromo-5-cyano-1-methyl-1H-pyrazol-3-yl], [BC 705; 4-bromo -5-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC706; 4-bromo-5-trifluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 707; 5- Fluoro-1, 4-dimethyl-1H-pyrazol-3-yl], [BC 708; 5-bromo-1, 4-dimethyl-1 H-pyrazol-3-yl], [BC 709; 5-ethoxy-1, 4- Dimethyl-1H-pyrazol-3-yl], [BC710; 5-cyclopropyl-1,4-dimethyl-1H-pyrazol-3-yl], [BC711; 5-difluoromethyl-1,4-dimethyl-1H- Pyrazol-3-yl], [BC 712; 4-ethyl-5-fluoro-1-methyl-1H-pyrazol-3-yl], [BC 713; 4-ethyl-5-chloro-1-methylpyrazol-3-yl ], [BC 714; 5-bromo-4-ethyl-1- Thilpyrazol-3-yl], [BC 715; 4-ethyl-5-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 716; 5-cyclopropyl-4-ethyl-1-methyl-1H- Pyrazol-3-yl], [BC717; 4-ethyl-5-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 718; 4-ethyl-5-trifluoromethyl-1-methyl-1H 4-Pyrazol-3-yl], [BC 719; 4-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 720; 5-fluoro-4-methoxy-1-methyl-1H-pyrazol-3-yl ], [BC 721; 5-chloro-4-methoxy-1-methyl-1 H-pyrazol-3-yl], [BC 722; 5-bromo-4-methoxy-1-methyl-1 H-pyrazol-3-yl], [BC 723; 4-methoxy-1,5-dimethyl-1H-pyrazol-3-yl], [BC 724; 5-ethyl-4-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 725; 4 , 5-Dimethoxy-1-methyl-1H-pyrazol-3-yl], [BC 726; 5-ethoxy-4-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 727; 5-cyano-4 -Methoxy-1-methyl-1H- Razol-3-yl], [BC 728; 5-cyclopropyl-4-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 729; 5-difluoromethyl-4-methoxy-1-methyl-1 H- Pyrazol-3-yl], [BC 730; 5-trifluoromethyl-4-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 731; 4-ethoxy-1-methyl-1H-pyrazole-3- 5-fluoro-4-ethoxy-1-methyl-1H-pyrazol-3-yl], [BC733; 5-chloro-4-ethoxy-1-methyl-1H-pyrazol-3-yl] [BC734; 5-bromo-4-ethoxy-1-methyl-1H-pyrazol-3-yl], [BC 735; 4-ethoxy-1,5-dimethyl-1H-pyrazol-3-yl], [BC 736; 5-ethyl-4-ethoxy-1-methyl-1H-pyrazol-3-yl], [BC 737; 4-ethoxy-5-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 738; 5-diethoxy-1-methyl-1H-pyrazol-3-yl], [BC 739; 5-cyano-4-ethoxy-1-methyl-1H-pyrazol-3-yl], [BC 740; 5-cyclopropyl-4. -Ethoxy-1-me Ethyl-1H-pyrazol-3-yl], [BC 741; 5-difluoromethyl-4-ethoxy-1-methyl-1H-pyrazol-3-yl], [BC 742; 5-trifluoromethyl-4-ethoxy-1 -Methyl-1H-pyrazol-3-yl], [BC 743; 4-cyano-1-methyl-1H-pyrazol-3-yl], [BC 744; 4-cyano-5-fluoro-1-methyl-1H-pyrazole 4-Cyclo-5-chloro-1-methyl-1H-pyrazol-3-yl], [BC 746; 5-bromo-4-cyano-1-methyl-1H-pyrazole-3 -Yl], [BC 747; 4-cyano-5-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 748; 4-cyano-5-ethoxy-1-methyl-1 H-pyrazol-3-yl [BC 749; 4,5-dicyano-1-methyl-1H-pyrazol-3-yl], [BC750; 4-cyano-5-cyclopropyl-1-methyl-1H-pyrazol-3-yl], [BC750; BC 751; 4-cyano-5-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 752; 4-cyano-1-methyl-5-trifluoro-1H-methylpyrazol-3-yl], [BC 753; 4-difluoro Ethyl-1-methyl-1H-pyrazol-3-yl], [BC 754; 5-fluoro-4-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 755; 5-chloro-4-difluoro Methyl-1-methyl-1H-pyrazol-3-yl], [BC 756; 5-bromo-4-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 757; 4-difluoromethyl-1, 5-Dimethyl-1H-pyrazol-3-yl], [BC 758; 5-ethyl-4-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 759; 4-difluoromethyl-5-methoxy- 1-methyl-1H-pyrazol-3-yl], [BC 760; 5-ethoxy-4-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 761; 5-cyano-4-difluoromethyl- 1-methyl-1H-pyrazol-3-yl], [BC 762; 5-cyclopropyl-4-difluoromethyl-1-methyl-1H-pyrazol-3-yl], [BC 763; 4, 5-bis (difluoromethyl) ) -1-Methyl-1H-pyrazol-3-yl], [BC 764; 4-difluoromethyl-1-methyl-5-trifluorome 1-methyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC766; 5-fluoro-1-methyl-4-trifluoromethyl- 1H-pyrazol-3-yl], [BC 767; 5-chloro-1-methyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 768; 5-bromo-1-methyl-4-trifluoro] Methyl-1H-pyrazol-3-yl], [BC 769; 1,5-dimethyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 770; 5-ethyl-1-methyl-4-trifluoro] Methyl-1H-pyrazol-3-yl], [BC 771; 5-methoxy-1-methyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 772; 5-ethoxy-1-methyl-4- 4 Trifluoromethyl-1H-pyrazol-3-yl], [BC 773; 5-cyano-1-methyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 774; 5-cyclopropyl-1-methyl] -4-trifluoromethyl-1H-pyrazol-3-yl], [BC 775; 5-difluoromethyl-1-methyl-4-trifluro Methyl-1H-pyrazol-3-yl], [BC 776; 1-Methyl-4,5-bis (trifluoromethyl) -1H-pyrazol-3-yl], [BC 777; 1-ethyl-5-fluoro-1H -Pyrazol-3-yl], [BC 778; 5-bromo-1-ethyl-1H-pyrazol-3-yl], [BC 779; 5-cyano-1-ethyl-1H-pyrazol-3-yl], [BC 780] 1-ethyl-5-difluoromethyl-1H-pyrazol-3-yl], [BC 781; 1-ethyl-4, 5-difluoro-1 H-pyrazol-3-yl], [BC 782; 1-ethyl-4- Chloro-1H-pyrazol-3-yl], [BC 783; 1-ethyl-5-bromo-4-fluoro-1 H-pyrazol-3-yl], [BC 784; 1-ethyl-5-cyano-4-fluoro- 1H-Pyrazol-3-yl], [BC 785; 1-ethyl-5-difluoromethyl-4-fluoro-1H-pyrazol-3-yl], [BC 786; 1-ethyl-5-trifluoromethyl-4-fluoro -1H-pyrazol-3-yl], [BC 787; 4-chloro-1-ethyl-5-fluoro-1H-pyrazol-3-yl], [BC 788; 5-bromo-4-chloro-1-ethyl-1H -Pyrazol-3-yl], [BC 789; 4-chloro-1,5-diethyl-1H-pyrazol-3-yl], [BC 790; 1-ethyl-5-cyano-4-chloro-1H-pyrazol-3-yl], [BC 791; Ethyl 4-chloro-5-difluoromethyl-1H-pyrazol-3-yl], [BC 792; 4-bromo-1-ethyl-5-fluoro-1H-pyrazol-3-yl], [BC 793; 4-bromo 4-chloro-1-ethyl-1H-pyrazol-3-yl], [BC 794; 4-bromo-1-ethyl-5-methoxy-1H-pyrazol-3-yl], [BC795; 4-bromo-5 -Cyano-1-ethyl-1H-pyrazol-3-yl], [BC 796; 5-fluoro-1-ethyl-4-methyl-1H-pyrazol-3-yl], [BC 797; 5-bromo-1-ethyl -4-Methyl-1H-pyrazol-3-yl], [BC 798; 5-cyclopropyl-1-ethyl-4-methyl-1H-pyrazol-3-yl], [BC 799; 1-ethyl-5-difluoromethyl -4-Methyl-1H-pyrazol-3-yl], [BC 800; 1,4-diethyl-1H-pyrazol-3-yl],

[BC801; 1,4-diethyl-5-fluoro-1H-pyrazol-3-yl], [BC802; 1,4-diethyl-5-chloro-1H-pyrazol-3-yl], [BC 803; 1,4 -Diethyl-5-methoxy-1-methyl-1H-pyrazol-3-yl], [BC 804; 4-methoxy-1-ethyl-1H-pyrazol-3-yl], [BC 805; 5-fluoro-1-ethyl] -4-methoxy-1H-pyrazol-3-yl], [BC 806; 5-chloro-1-ethyl-4-methoxy-1H-pyrazol-3-yl], [BC 807; 5-bromo-1-ethyl-4 -Methoxy-1H-pyrazol-3-yl], [BC 808; 1-ethyl-5-methoxy-4-methyl-1H-pyrazol-3-yl], [BC 809; 1,5-diethyl-4-methoxy-1H -Pyrazol-3-yl], [BC 810; 1-ethyl-4,5-dimethoxy-1H-pyrazol-3-yl], [BC811; 1-ethyl-5-cyano-4-methoxy-1H-pyrazole-3 -Yl], [BC 812; 5-cyclopropyl-1-ethyl-4-methoxy-1H-pyrazol-3-yl], [BC 813; 1-ethyl-5-difluoromethyl-4-methoxy-1H-pyrazole-3 -Yl], [BC 814; 1-ethyl-4-methoxy -5-trifluoromethyl-1H-pyrazol-3-yl], [BC 815; 4-cyano-1-ethyl-1H-pyrazol-3-yl], [BC 816; 4-cyano-5-fluoro-1-ethyl -1H-pyrazol-3-yl], [BC 817; 4-cyano-5-chloro-1-ethyl-1H-pyrazol-3-yl], [BC 818; 5-bromo-4-cyano-1-ethyl-1H 4-Pyrazol-3-yl], [BC 819; 4-cyano-1-ethyl-5-methoxy-1H-pyrazol-3-yl], [BC 820; 4, 5-dicyano-1-ethyl-1 H-pyrazole-3 -Yl], [BC 821; 4-cyano-5-cyclopropyl-1-ethyl-1H-pyrazol-3-yl], [BC 822; 4-cyano-5-difluoromethyl-1-ethyl-1H-pyrazole-3 -Yl], [BC 823; 4-cyano-1-ethyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC 824; 4-difluoromethyl-1-ethyl-1H-pyrazol-3-yl] [BC 825; 5-fluoro-4-difluoromethyl-1-ethyl-1H-pyrazol-3-yl], [BC 826; 5-chloro-4-difluoromethyl-1-ethyl-1H-pyrazol-3-yl] , [BC 827; 4 -Difluoromethyl-1-ethyl-4-methyl-1H-pyrazol-3-yl], [BC 828; 4-difluoromethyl-1-ethyl-5-methoxyl-1H-pyrazol-3-yl], [BC 829; 5 -Cyano-4-difluoromethyl-1-ethyl-1H-pyrazol-3-yl], [BC 830; 1-ethyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 831; 5-fluoro- 1-ethyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 832; 5-chloro-1-ethyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 833; 1- Ethyl-4-trifluoromethyl-5-methyl-1H-pyrazol-3-yl], [BC 834; 1-ethyl-4-trifluoromethyl-5-methoxy-1 H-pyrazol-3-yl], [BC 835; 5-Cyano-1-ethyl-4-trifluoromethyl-1H-pyrazol-3-yl], [BC 836; 4-methoxy-5-methylpyrazol-1-yl], [BC 837; 4-ethoxy-5-methyl Pyrazol-1-yl], [BC 838; 4-cyclopropyl-5-methylpyrazol-1-yl], [BC 839; 4-triful Omethyl-5-methylpyrazol-1-yl], [BC 840; 4-bromo-3-methylpyrazol-1-yl], [BC 841; 4-ethyl-3-methylpyrazol-1-yl], [BC 842; 4 -Methoxy-3-methylpyrazol-1-yl], [BC843; 4-ethoxy-3-methylpyrazol-1-yl], [BC844; 4-cyclopropyl-3-methylpyrazol-1-yl], [BC845 5-fluoro-3-methylpyrazol-1-yl], [BC 846; 4,5-difluoro-3-methylpyrazol-1-yl], [BC 847; 4-chloro-5-fluoro-3-methylpyrazole- 1-yl], [BC 848; 4-bromo-5-fluoro-3-methylpyrazol-1-yl], [BC 849; 5-fluoro-3,4-dimethylpyrazol-1-yl], [BC 850; Ethyl-5-fluoro-3-methylpyrazol-1-yl], [BC 851; 5-fluoro-4-methoxy-3-methylpyrazol-1-yl], [BC 852; 4-ethoxy-5-fluoro-3- Methylpyrazol-1-yl], [BC 853; 4-cyano-5-fluoro-3-methylpyrazol-1-yl], [BC 854; 4-cyclopropyl 5-fluoro-3-methylpyrazol-1-yl], [BC 855; 4-difluoromethyl-5-fluoro-3-methylpyrazol-1-yl], [BC 856; 4-trifluoromethyl-5-fluoro- 3-Methylpyrazol-1-yl], [BC 857; 5-chloro-3-methylpyrazol-1-yl], [BC 858; 5-chloro-4-fluoro-3-methylpyrazol-1-yl], [BC 859 4,5-dichloro-3-methylpyrazol-1-yl], [BC 860; 4-bromo-5-chloro-3-methylpyrazol-1-yl], [BC 861; 5-chloro-3,4-dimethyl Pyrazol-1-yl], [BC 862; 5-chloro-4-ethyl-3-methylpyrazol-1-yl], [BC 863; 5-chloro-4-methoxy-3-methylpyrazol-1-yl], [BC BC864; 5-chloro-4-ethoxy-3-methylpyrazol-1-yl], [BC865; 5-chloro-4-cyano-3-methylpyrazol-1-yl], [BC866; 5-chloro-4- Cyclopropyl-3-methylpyrazol-1-yl], [BC 867; 5-chloro-4-difluoro-3-methylpyrazol-1-yl], [BC 868; 5-chloro-4- Fluoromethyl-3-methylpyrazol-1-yl], [BC 869; 5-bromo-3-methylpyrazol-1-yl], [BC 870; 5-bromo-4-fluoro-3-methylpyrazol-1-yl ], [BC 871; 5-bromo-4-chloro-3-methylpyrazol-1-yl], [BC 872; 4, 5-dibromo-3-methylpyrazol-1-yl], [BC 873; 5-bromo-3] , 4-Dimethylpyrazol-1-yl], [BC 874; 5-bromo-4-ethyl-3-methylpyrazol-1-yl], [BC 875; 5-bromo-4-methoxy-3-methylpyrazole-1-] 5-bromo-4-ethoxy-3-methylpyrazol-1-yl], [BC 877; 5-bromo-4-cyano-3-methylpyrazol-1-yl], [BC 878; 5- Bromo-4-cyclopropyl-3-methylpyrazol-1-yl], [BC 879; 5-bromo-4-difluoromethyl-3-methylpyrazol-1-yl], [BC 880; 5-bromo-4-trifluoro Methyl-3-methylpyrazol-1-yl], [BC 881; 3,5-dimethylpyrazol-1-yl], [BC 882; 5-ethyl-4-fluoro-3-methyl] Pyrazol-1-yl], [BC 883; 5-ethyl-4-methoxy-3-methylpyrazol-1-yl], [BC 884; 4-ethoxy-5-ethyl-3-methylpyrazol-1-yl], [BC BC885; 5-trifluoromethyl-4-methoxy-3-methylpyrazol-1-yl], [BC886; 5-methoxy-3-methylpyrazol-1-yl], [BC887; 4-fluoro-5-methoxy- 3-Methylpyrazol-1-yl], [BC 888; 4-chloro-5-methoxy-3-methylpyrazol-1-yl], [BC 889; 4-bromo-5-methoxy-3-methylpyrazol-1-yl ], [BC 890; 5-methoxy-3,4-dimethylpyrazol-1-yl], [BC891; 4-ethyl-5-methoxy-3-methylpyrazol-1-yl], [BC 892; -3-Methylpyrazol-1-yl], [BC 893; 4-ethoxy-5-methoxy-3-methylpyrazol-1-yl], [BC 894; 4-cyano-5-methoxy-3-methylpyrazole-1 4-cyclopropyl-5-methoxy-3-methylpyrazol-1-yl], [BC 896; 4-difluoro-5-methoxy- 3-Methylpyrazol-1-yl], [BC897; 5-methoxy-3-methyl-4-trifluoromethylpyrazol-1-yl], [BC898; 5-ethoxy-3-methylpyrazol-1-yl], [BC 899; 5-ethoxy-4-fluoro-3-methylpyrazol-1-yl], [BC 900; 5-ethoxy-4-chloro-3-methylpyrazol-1-yl],

[BC 901; 5-ethoxy-4-bromo-3-methylpyrazol-1-yl], [BC 902; 5-ethoxy-3,4-dimethylpyrazol-1-yl], [BC 903; 5-ethoxy-4-ethyl] -3-Methylpyrazol-1-yl], [BC 904; 5-ethoxy-4-methoxy-3-methylpyrazol-1-yl], [BC 905; 4,5-diethoxy-3-methylpyrazol-1-yl] , [BC906; 4-cyano-5-ethoxy-3-methylpyrazol-1-yl], [BC 907; 4-cyclopropyl-5-ethoxy-3-methylpyrazol-1-yl], [BC 908; 4-difluoro Methyl-5-ethoxy-3-methylpyrazol-1-yl], [BC 909; 5-ethoxy-4-trifluoromethyl-3-methylpyrazol-1-yl], [BC 910; 5-cyano-3-methylpyrazole -1-yl], [BC 911; 5-cyano-4-fluoro-3-methylpyrazol-1-yl], [BC 912; 5-cyano-4-chloro-3-methylpyrazol-1-yl], [BC 913 5-cyano-4-bromo-3-methylpyrazol-1-yl], [BC 914; 5-cyano-3,4-dimethylpyrazol-1-yl], [BC 915; 5-cyano-4-ethyl-3-methylpyrazol-1-yl], [BC 916; 5-cyano-4-methoxy-3-methylpyrazol-1-yl], [BC 917; 5-cyano-4- Ethoxy 3-methylpyrazol-1-yl], [BC 918; 4,5-dicyano-3-methylpyrazol-1-yl], [BC 919; 5-cyano-4-cyclopropyl-3-methylpyrazol-1-yl ], [BC920; 5-cyano-4-difluoro-3-methylpyrazol-1-yl], [BC 921; 5-cyano-4-trifluoromethyl-3-methylpyrazol-1-yl], [BC 922; 5] -Difluoromethyl-3-methylpyrazol-1-yl], [BC 923; 5-difluoromethyl-4-fluoro-3-methylpyrazol-1-yl], [BC 924; 4-chloro-5-difluoromethyl-3- Methylpyrazol-1-yl], [BC 925; 4-bromo-5-difluoromethyl-methylpyrazol-1-yl], [BC 926; 5-difluoromethyl-3,4-dimethylpyrazol-1-yl], [BC 927 4-ethyl-5-difluoromethyl-3-methylpyrazol-1-yl], [BC 928; 5-di Luomethyl-4-methoxy-3-methylpyrazol-1-yl], [BC 929; 4-ethoxy-5-difluoromethyl-3-methylpyrazol-1-yl], [BC 930; 4-cyano-5-difluoromethyl- 3-methylpyrazol-1-yl], [BC 931; 4-cyclopropyl-5-difluoromethyl-3-methylpyrazol-1-yl], [BC 932; 4,5-bis (difluoromethyl) -3-methylpyrazole -1-yl], [BC 933; 5-difluoromethyl-3-methyl-4-trifluoromethylpyrazol-1-yl], [BC 934; 3-methyl-5-trifluoromethylpyrazole-1-yl], [BC 935; 4-fluoro-3-methyl-5-trifluoromethylpyrazol-1-yl], [BC 936; 4-chloro-3-methyl-5-trifluoromethylpyrazol-1-yl], [BC 937 4-bromo-3-methyl-5-trifluoromethylpyrazol-1-yl], [BC 938; 3,4-dimethyl-5-trifluoromethylpyrazol-1-yl], [BC 939; 4-ethyl; -3-Methyl-5-trifluoromethyl pyra -1-yl], [BC 940; 4-methoxy-3-methyl-5-trifluoromethylpyrazol-1-yl], [BC 941; 4-ethoxy-3-methyl-5-trifluoromethylpyrazole -4-yl], [BC942; 4-cyano-3-methyl-5-trifluoromethylpyrazol-1-yl], [BC943; 4-cyclopropyl-3-methyl-5-trifluoromethylpyrazole- 1-yl], [BC 944; 4-difluoro-3-methyl-5-trifluoromethylpyrazol-1-yl], [BC 945; 4,5-bis (trifluoromethyl) -3-methylpyrazole-1-] [BC946; 3-ethyl-4-ethoxy-5-methylpyrazol-1-yl], [BC947; 3-ethyl-4-cyano-5-methylpyrazol-1-yl], [BC 948; 3- Ethyl-4-cyclopropyl-5-methylpyrazol-1-yl], [BC 949; 3-fluoro-5-methylpyrazol-1-yl], [BC950; 3,4-difluoro-5-methylpyrazole-1-] 4-chloro-3-fluoro-5-methylpyrazol-1-yl], [BC 952; 4-bromo-3-fluo] Ro-5-methylpyrazol-1-yl], [BC953; 3-fluoro-4,5-dimethylpyrazol-1-yl], [BC954; 4-ethyl-3-fluoro-5-methylpyrazole-1-yl ], [BC 955; 3-fluoro-4-methoxy-5-methylpyrazol-1-yl], [BC 956; 4-ethoxy-3-fluoro-5-methylpyrazol-1-yl], [BC 957; 4-cyano 4-fluoro-5-methylpyrazol-1-yl], [BC 958; 4-cyclopropyl-3-fluoro-5-methylpyrazol-1-yl], [BC 959; 4-difluoro-3-fluoro-5-l Methylpyrazol-1-yl], [BC960; 3-fluoro-5-methyl-4-trifluoromethylpyrazol-1-yl], [BC961; 3-chloro-5-methylpyrazol-1-yl], [BC962 3-chloro-4-fluoro-5-methylpyrazol-1-yl], [BC 963; 3,4-dichloro-5-methylpyrazol-1-yl], [BC 964; 4-bromo-3-chloro-5 -Methylpyrazol-1-yl], [BC 965; 3-chloro-4,5-dimethylpyrazol-1-yl], [BC 966; 3-chloro-4-ethyl-5-methyl Lupyrazol-1-yl], [BC967; 3-chloro-4-methoxy-5-methylpyrazol-1-yl], [BC968; 3-chloro-4-ethoxy-5-methylpyrazol-1-yl], [BC BC969; 3-chloro-4-cyano-5-methylpyrazol-1-yl], [BC 970; 3-chloro-4-cyclopropyl-5-methylpyrazol-1-yl], [BC 971; 3-chloro-4 -Difluoro-5-methylpyrazol-1-yl], [BC 972; 3-chloro-5-methyl-4-trifluoromethylpyrazol-1-yl], [BC 973; 3-methoxy-5-methylpyrazole-1-] 4-fluoro-3-methoxy-5-methylpyrazol-1-yl], [BC 975; 4-chloro-3-methoxy-5-methylpyrazol-1-yl], [BC 976; 4- Bromo-3-methoxy-5-methylpyrazol-1-yl], [BC 977; 3-methoxy-4,5-dimethylpyrazol-1-yl], [BC978; 4-ethyl-3-methoxy-5-methylpyrazole -1-yl], [BC979; 3,4-dimethoxy-5-methylpyrazol-1-yl], [BC 980; 4-ethoxy-3-methoxy-5-methyl] Pyrazol-1-yl], [BC 981; 4-cyano-3-methoxy-5-methylpyrazol-1-yl], [BC 982; 4-cyclopropyl-3-methoxy-5-methylpyrazol-1-yl], [BC983; 4-difluoro-3-methoxy-5-methylpyrazol-1-yl], [BC984; 5-methyl-3-methoxy-4-trifluoromethylpyrazol-1-yl], [BC985; 3-cyano -5-methylpyrazol-1-yl], [BC 986; 3-cyano-4-fluoro-5-methylpyrazol-1-yl], [BC 987; 4-chloro-3-cyano-5-methylpyrazole-1-l 4-bromo-3-cyano-5-methylpyrazol-1-yl], [BC 989; 3-cyano-4,5-dimethylpyrazol-1-yl], [BC 990; 3-cyano- 4-ethyl-5-methylpyrazol-1-yl], [BC991; 3-cyano-4-methoxy-5-methylpyrazol-1-yl], [BC992; 3-cyano-4-ethoxy-5-methylpyrazole -1-yl], [BC993; 3,4-dicyano-5-methylpyrazol-1-yl], [BC994; 3-cyano-4-cyclopropyl-5-methylpi Zol-1-yl], [BC995; 3-cyano-4-difluoro-5-methylpyrazol-1-yl], [BC996; 3-cyano-5-methyl-4-trifluoromethylpyrazol-1-yl] , [BC997; 3-cyclopropyl-4-methoxy-5-methylpyrazol-1-yl], [BC 998; 3-cyclopropyl-4-ethoxy-5-methylpyrazol-1-yl], [BC 999; 3 -Cyclopropyl-4-cyano-5-methylpyrazol-1-yl], [BC1000; 3-difluoromethyl-5-methylpyrazol-1-yl],

[BC1001; 4-fluoro-3-difluoromethyl-5-methylpyrazol-1-yl], [BC1002; 4-chloro-3-difluoromethyl-5-methylpyrazol-1-yl], [BC1003; 4-bromo -3-difluoromethyl-5-methylpyrazol-1-yl], [BC 1004; 3-difluoromethyl-4, 5-dimethylpyrazol-1-yl], [BC 1005; 3-difluoromethyl-4-ethyl-5- Methylpyrazol-1-yl], [BC 1006; 3-difluoromethyl-4-methoxy-5-methylpyrazol-1-yl], [BC 1007; 3-difluoromethyl-4-ethoxy-5-methylpyrazol-1-yl ], [BC1008; 3-difluoromethyl-4-cyano-5-methylpyrazol-1-yl], [BC1009; 3-difluoromethyl-4-cyclopropyl-5-methylpyrazol-1-yl], [BC1010; 4-Difluoromethyl-5-methylpyrazol-1-yl], [BC1011; 5-methyl-4-trifluoromethylpyrazol-1-yl], [BC1012; 5-methyl-3-trifluoromethylpyrazole-1 -Yl], [BC1013; 4-fluoro-5-methyl-3-trifluoromethylpyrazol-1-yl], [BC1014; 4-chloro-5-methyl-3-trifluoropyrazolyl-1-yl], [BC1015; 4- Bromo-5-methyl-3-trifluoromethylpyrazol-1-yl], [BC1016; 4,5-dimethyl-3-trifluoromethylpyrazol-1-yl], [BC1017; 4-ethyl-5- Methyl-3-trifluoromethylpyrazol-1-yl], [BC1018; 4-methoxy-5-methyl-3-trifluoromethylpyrazol-1-yl], [BC1019; 4-ethoxy-5-methyl- 3-Trifluoromethylpyrazol-1-yl], [BC1020; 4-cyano-5-methyl-3-trifluoromethylpyrazol-1-yl], [BC1021; 4-cyclopropyl-5-methyl-3 4-Trifluoromethylpyrazol-1-yl], [BC 1022; 4-difluoro-5-methyl-3-trifluoromethylpyrazol-1-yl], [BC 1023; 5-methyl-3,4-bis (triyl) Fluoromethyl (pyrazol-1-yl), [BC 1024; 3-fluoro-1,4-di 3-chloro-1,4-dimethyl-1H-pyrazol-5-yl], [BC1026; 3-bromo-1,4-dimethyl-1H-pyrazole- 5-yl], [BC1027; 3-cyano-1,4-dimethyl-1H-pyrazol-5-yl], [BC1028; 3-methoxy-1,4-dimethyl-1H-pyrazol-5-yl], BC 1029; 3-ethoxy-1, 4-dimethyl-1H-pyrazol-5-yl], [BC 1030; 3-fluoro-1-ethyl-4-methyl-1H-pyrazol-5-yl], [BC 1031; 3- Chloro-1-ethyl-4-methyl-1H-pyrazol-5-yl], [BC1032; 3-bromo-1-ethyl-4-methyl-1H-pyrazol-5-yl], [BC1033; 3-cyano- 1-ethyl-4-methyl-1H-pyrazol-5-yl], [BC1034; 3-methoxy-1-ethyl-4-methyl-1H-pyrazol-5-yl], [BC1035; Ethyl-4-methyl-1H-pyrazol-5-yl], [BC1036; 3,4-difluoro-1-methyl-1H-pyrazol-5-yl], [BC1037; 3-chloro-1-methyl-4- 4 Fluoro-1 H-pyrazol-5-yl], [BC 1038; 3-bromo-1-methyl-4- 4- Fluoro-1H-pyrazol-5-yl], [BC1039; 3-cyano-1-methyl-4-fluoro-1H-pyrazol-5-yl], [BC1040; 3-methoxy-1-methyl-4-fluoro- 1H-pyrazol-5-yl], [BC1041; 3-ethoxy-1-methyl-4-fluoro-1H-pyrazol-5-yl], [BC1042; 3,4-dichloro-1-methyl-1H-pyrazole- 5-yl], [BC1043; 3-bromo-1-methyl-4-chloro-1H-pyrazol-5-yl], [BC1044; 3-cyano-1-methyl-4-chloro-1H-pyrazole-5 , [BC 1045; 3-methoxy-1-methyl-4-chloro-1H-pyrazol-5-yl], [BC 1046; 3-ethoxy-1-methyl-4-chloro-1H-pyrazol-5-yl] , [BC1047; 3,4-dicyano-1-methyl-1H-pyrazol-5-yl], [BC1048; 3-fluoro-4-methoxy-1-methyl-1H-pyrazol-5yl], [BC1049; 3 -Chloro-4-methoxy-1-methyl-1H-pyrazol-5yl], [BC1050; 3-bromo-4-methoxy-1-methyl-1H-pyrazol-5yl], [BC1051; 3-cyano-4 -Methoxy-1-methyl-1H-pyrazole- 5-yl], [BC1052; 3,4- dimethoxy-1-methyl -1H- pyrazol -5-yl], [BC1053; C (= O) CH 3], [BC1054; C (= O) CH 2 CH 3] , [BC1055; C (= O ) CH 2 CH 2 CH 3], [BC1056; C (= O) CH 2 CH 2 CH 2 CH 3], [BC1057; C (= O) CH 2 CH 2 CH 2 CH ₂ CH ₃ ], [BC 1058; C (= O) CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ CH ₃ ], [BC 1059; C (= O) OCH (CH ₃ ) ₂ ], [BC 1060; C (= O) _{) C (CH 3) 3]} , [BC1061; C (= O) CH2CH (CH 3) 2], [BC1062; C (= O) CF 3], [BC1063; C (= O) CCl 3], [ BC1064; C (= O) CH 2 CHF 2], [BC1065; C (= O) -c-Pr], [BC1066; C (= O) -c-Bu], [BC1067; C (= O) - c-Hex], [BC1068; C (= O)-(2-fluorocyclopropyl)], [BC1069; C (= O)-(2-chlorocyclopropyl)], [BC1070; C (= O)- (2,2-difluorocyclopropyl), [BC1071; C ((O)-(2,2,3,3-tetrafluorocyclopropyl)], [BC1072; C (= O)-(1,2,5 2,3,3-Pentafluorocyclopropyl)], [BC1073; 1-cyclopropyl-1H-pyrazol-3-yl], [BC1074; 1-cyclopropyl-5-fluoro-1H-pyrazol-3-yl] , [BC1075; 5-chloro-1-cyclopropyl-1H-pyrazol-3-yl], [BC1076 5-bromo-1-cyclopropyl-1H-pyrazol-3-yl], [BC1077; 5-cyano-1-cyclopropyl-1H-pyrazol-3-yl], [BC1078; 1-cyclopropyl-5-yl; Methyl-1H-pyrazol-3-yl], [BC1079; 1-cyclopropyl-5-ethyl-1H-pyrazol-3-yl], [BC1080; 1-cyclopropyl-5-difluoromethyl-1H-pyrazole-3 -Yl], [BC1081; 1-cyclopropyl-5-trifluoromethyl-1H-pyrazol-3-yl], [BC1082; 1-cyclopropyl-5-methoxy-1H-pyrazol-3-yl], [BC1083 1-Cyclopropyl-5-ethoxy-1H-pyrazol-3-yl], [BC1084; 1-cyclopropyl-5-thiomethoxy-1H-pyrazol-3-yl], [BC1085; 1-cyclopropyl-5-yl; Thiodifluoromethoxy-1H-pyrazol-3-yl], [BC 1086; 1-cyclopropyl-5-thiotrifluoromethoxy-1H-pyrazol-3-yl].

  Below, a substituent number (MC2) BC1087-BC2879 is described.

Substituent No. (MC2) E ¹⁰³ represents one of the following E601 to E616: BC1087 to BC2879. Represents a binding site. ). For example, substituent number (MB2) BC1087 represents a group in which R ^{613 to} R ⁶¹⁵ and R ⁶¹⁶ are a hydrogen atom in the following E601.

[Substituent group number ^{(MC2); E 103],} [BC1087; E601, R613: H, R614: H, R615: H, R616: H], [BC1088; E601, R613: Me, R614: H, R615: H , R 616: H], [BC 1089; E 601, R 613: Me, R 614: H, R 616: H], [BC 10 90; E 601, R 613: H, R 614: H, R 615: Me, R 616: H], [BC1091; E601, R613: H, R614: H, R615: H, R616: Me], [BC1092; E601, R613: Me, R614: Me, R615: H, R616: H], [BC1093; E601, R613 : Me, R 614: H, R 615: Me, R 616: H], [BC 1094; E 601, R 613: Me, R 614: H, R 615: H, R 616: Me], [BC 10 95; E 601, R 613: H, R 614: Me , R615: Me, R616: H], [BC1096; E601, R613: H, R614: Me, R615: H, R616: Me], [BC1097; E601, R613: H, R614: H, R615: Me, R616 : Me], [BC 1098; E 601, R 613: H, R 614: Me, R 615: H, R 616: H], [BC 10 99; E 601, R 613: Me, R 614: Me, R 615: Me, R 616: H], [BC 1100] E601, R613: Me, R 614: Me, R 615: H, R 616: Me],

[BC1101; E601, R613: Me, R614: H, R615: Me, R616: Me], [BC1102; E601, R613: H, R614: Me, R615: Me, R616: Me], [BC1103; E601, R613 : Me, R614: Me, R615: Me, R616: Me], [BC1104; E601, R613: Me, R614: F, R615: H, R616: H], [BC1105; E601, R613: Me, R614: H , R615: F, R616: H], [BC1106; E601, R613: Me, R614: H, R615: H, R616: F], [BC1 107; E601, R613: Me, R614: F, R615: F, R616] : H], [BC1108; E601, R613: Me, R614: F, R615: H, R616: F], [BC1109; E601, R613: Me, R614: H, R615: F, R616: F], [BC1 110] E601, R613: Me, R614: F, R615: F, R616: F], [BC1111; E601, R613: F, R614: Me, R615: H, R616: H], [BC1112; E601, R613: H , R614: Me, R615: F, R616: H], [BC1113; E601, R613: H, R614: Me, R615: H, R616: F], [BC1114; E601, R613: F, R614: Me, R615] : F, R 616: H], [BC 1115; E 601, R 613: F, R 614: Me, R 615: H, R 616: F], [BC 1 116; E 601, R 613: H, R 614: Me, R 615: F, R 616: F ], [BC1117; E601, R613: F, R614: Me, R615: F, R616: F], [BC1118; E601, R613: F, R614: H, R615: Me, R616: H], [BC1119; E601] , R 613: H, R 614: F, R 615: Me, R 616: H], [BC1 120; E601, R 613: H, R 614: H, R 615: Me, R 616: F], [BC 1121; : F, R 615: Me, R 616: H], [BC 1122; E 601, R 613: F, R 614: H, R 615: Me, R 616: F], [BC 1 123; E 601, R 613: H, R 614: F, R 615: Me , R 616: F], [BC 1 124; E601, R613: F, R 614: F, R 615: Me, R 616: F], [BC 1 125; E 601, R 613: F, R 614: H, R 615: H, R 616: Me], [BC 1 126; E 601, R 613: H, R 614: F, R 615: H, R 616: Me], [BC1 127; E601, R 613: H, R 614: H, R 615: F, R 616: Me], [BC 1 128; E 601, R 613: F, R 614: F, R615: H, R616: Me], [BC1129; E601, R613: F, R614: H, R615: F, R616: Me], [BC1 130; E601, R613: H, R614: F, R615: F, R616: Me], [BC1131; E601, R613: F, R614: F, R615: F, R616: Me], [BC1132; E601, R613: Me, R614: Me, R615: F, R616: H], [BC1133; E601, R613: Me, R614: Me, R615: H, R616: F], [BC1134; E601, R613: Me, R614: F, R615: Me, R616: H], [BC1 135; E601, R613: Me, R614: H, R615: Me, R616: F], [BC1136; E601, R613: Me, R614: F, R615: H, R616: Me], [BC1137; E601, R613: Me, R614: H, R615: F, R616: Me], [BC1138; E601, R613: Me, R614: Me, R615: Cl, R616: H], [BC1139; E601, R613: Me, R614: Me, R615: H, R616: Cl] , [BC1140; E601, R613: Me, R614: Cl, R615: Me, R616: H], [BC1141; E601, R613: Me, R614: H, R615: Me, R616: Cl], [BC1142; R613: Me, R 614: Cl, R 615: H, R 616: Me], [BC 1143; E601, R 613: Me, R 614: H, R 615: Cl, R 616: Me], [BC 1 144; E 601, R 613: Me, R 614: Cl, R615: H, R616: H], [BC1145; E601, R613: Me, R614: H, R615: Cl, R616: H], [BC1146; E601, R613: Me, R614: H, R615: H, R61 6: Cl], [BC 1147; E601, R 613: Me, R 614: Cl, R 615: Cl, R 616: H], [BC 1148; E 601, R 613: Me, R 614: Cl, R 615: H, R 616: Cl], [ BC1149; E601, R613: Me, R614: H, R615: Cl, R616: Cl], [BC1150; E601, R613: Cl, R614: Me, R615: H, R616: H], [BC1151; E601, R613: H, R614: Me, R615: Cl, R616: H], [BC1152; E601, R613: H, R614: Me, R615: H, R616: Cl], [BC1153; E601, R613: Cl, R614: Me, R615: Cl, R 616: H], [BC 1154; E601, R 613: Cl, R 614: Me, R 615: H, R 616: Cl], [BC 1 155; E 601, R 613: H, R 614: Me, R 615: Cl, R 616: Cl], [BC1156; E601, R613: Cl, R614: H, R615: Me, R616: H], [BC1 157; E601, R613: H, R614: Cl, R615: Me, R616: H], [BC1158; E601, R613: H, R614: H, R615: Me, R616: Cl], [BC1159; E601, R613: Cl, R614: Cl, R615: Me, R616: H], [BC1 160; E601, R613: Cl, R614: H, R615: Me, R616: Cl], [BC1161; E601, R613: H, R614: Cl, R615: Me, R616: Cl], [BC1162; E601, R613: Cl, R614: H, R615: H, R616: Me], [BC1163; E601, R613: H, R614: Cl, R615: H, R616: Me], [BC1164; E601, R613: H, R614: H, R615: Cl, R616: Me] , [BC1165; E601, R613: Cl, R614: Cl, R615: H, R616: Me], [BC1166; E601, R613: Cl, R614: H, R615: Cl, R616: Me], [BC1167; E601, E601, E601, R613: H, R 614: Cl, R 615: Cl, R 616: Me], [BC1 168; E601, R 613: Me, R 614: Br, R 615: H, R 616: H], [BC 1 169; E 601, R 613: Me, R 614: H, R 615: Br, R 616: H], [BC1170; E601, R 613: Me, R 614: H, R 615: H, R 616: Br], [BC1171; E601, R613: Br, R 614: Me, R615: H, R616: H], [BC1172; E601, R613: H, R614: Me, R615: Br, R616: H], [BC1173; E601, R613: H, R614: Me, R615: H, R616: Br], [BC1174; E601, R613: Br, R614: H, R615: Me, R616: H], [BC1175; E601, R613: H, R614: Br, R615: Me, R616: H], [ BC1176; E601, R613: H, R614: H, R615: Me, R616: Br], [BC1177; E601, R613: Br, R614: H, R615: H, R616: Me], [BC1178; E601, R613: H, R614: Br, R615: H, R616: Me], [BC1179; E601, R613: H, R614: H, R615: Br, R616: Me], [BC1180; E601, R613: Me, R614: Me, R615: Br, R616: H], [BC1181; E601, R613: Me, R614: Me, R615: H, R616: Br], [BC1182; E601, R613: Me, R614: Br, R615: Me, R616: H], [BC1183; E601, R613: Me, R614: H, R615: Me, R616: Br], [BC1184; E601, R613: Me, R614: Br, R615: H, R616: Me], [BC1185; E601, R613: Me, R614: H, R615: Br, R616: Me], [BC1186; E601, R613: Me, R614: CN, R615: H, R616: H], [BC1187; E601, R613: Me, R614: H, R615: CN, R616: H], [BC1188; E601, R613: Me, R614: H, R615: H, R616: CN], [BC1189; E601, R613: CN, R614: Me, R615: H, R 616: H], [BC 1190; E 601, R 613: H, R 614: Me, R 615: CN, R 616: H], [BC 1191; E 601, R 613: H, R 614: Me, R 615: H, R 616: CN], [BC1192; E601, R613: CN, R614: H, R615: Me, R616: H], [BC1193; E601, R613: H, R614: CN, R615: Me, R616: H], [BC1194; E601, R613: H, R614: H, R615: Me, R616: CN], [BC1195; E601, R613: CN, R614: H, R615: H, R616: Me], [BC1196; E601, R613: H, R614: CN, R615: H, R616: Me], [BC1197; E601, R613: H, R614: H, R615: CN, R616: Me], [BC1198; E601, R613: Me, R614: Me, R615: CN, R616: H], [BC1 199; E601, R613: Me, R614: Me, R615: H, R616: CN], [BC1200; E601, R613: Me, R614: CN, R615: Me, R616: H] ,

[BC1201; E601, R613: Me, R614: H, R615: Me, R616: CN], [BC1202; E601, R613: Me, R614: CN, R615: H, R616: Me], [BC1203; E601, R613 : Me, R 614: H, R 615: CN, R 616: Me], [BC 1204; E 601, R 613: Me, R 614: OMe, R 615: H, R 616: H], [BC 1205; E 601, R 613: Me, R 614: H , R615: OMe, R616: H], [BC1206; E601, R613: Me, R614: H, R615: H, R616: OMe], [BC1207; E601, R613: OMe, R614: Me, R615: H, R616] : H], [BC1208; E601, R613: H, R614: Me, R615: OMe, R616: H], [BC1209; E601, R613: H, R614: Me, R615: H, R616: OMe], [BC1210] E601, R613: OMe, R614: H, R615: Me, R616: H], [BC1211; E601, R613: H, R614: OMe, R615: Me, R616: H], [BC1212; E601, R613: H , R614: H, R615: Me, R616: OMe], [BC1213; E601, R613: OMe, R614: H, R615: H, R616: Me], [BC1214; E601, R613: H, R614: OMe, R615 : H, R616: Me], [BC1215; E601, R613: H, R614: H, R615: OMe, R616: Me], [BC1216; E601, R613: Me, R614: Me, R615: OMe, R616: H ], [BC1217; E601, R613: Me, R614: Me, R615: H, R616: OMe], [BC1218; E601, R613: Me, R614: OMe, R615: Me, R616: H], [BC1219; , R 613: Me, R 614: H, R 615: Me, R 616: OMe], [BC 1220; E 601, R 613: Me, R 614: OMe, R 615: H, R 616: Me], [BC 122] E601, R 613: Me, R 614 : H, R 615: OMe, R 616: Me], [BC 1222; E601, R 613: Me, R 614: OEt, R 615: H, R 616: H], [BC 1 223; E601, R613: Me, R614: H, R615: OEt, R616: H], [BC1224; E601, R613: Me, R614: H, R615: H, R616: OEt], [BC1225; E601, R613: OEt, R614: Me, R615: H, R616: H], [BC1226; E601, R613: H, R614: Me, R615: OEt, R616: H], [BC1227; E601, R613: H, R614: Me, R615: H, R616: OEt], [BC1228; E601, R613: OEt, R614: H, R615: Me, R616: H], [BC1 229; E601, R613: H, R614: OEt, R615: Me, R616: H], [BC1230; E601, R613: H, R614: H, R615: Me, R616: OEt], [BC1231; E601, R613: OEt, R614: H, R615: H, R616: Me], [BC1232; E601, R613: H, R 614: OEt, R615: H, R616: Me], [BC1233; E601, R613: H, R614: H, R615: OEt, R616: Me], [BC1234; E601, R613: Me, R614: Me, R615: OEt, R616: H], [BC1235; E601, R613: Me, R614: Me, R615: H, R616: OEt], [BC1236; E601, R613: Me, R614: OEt, R615: Me, R616: H], [BC1237; E601, R613: Me, R614: H, R615: Me, R616: OEt], [BC1238; E601, R613: Me, R614: OEt, R615: H, R616: Me] , [BC1239; E601, R613: Me, R614: H, R615: OEt, R616: Me], [BC1240; E601, R613: Me, R614: Et, R615: H, R616: H], [BC 1241; E601, R613: Me, R 614: H, R 615: Et, R 616: H], [BC 1242; E601, R 613: Me, R 614: H, R 615: H, R 616: Et], [BC 1243; E601, R 613: Et, R 614: Me, R 615: H, R 616: H], [BC 1244; E 601, R 613: H, R 614: Me, R 615: Et, R 616: H], [BC 12 45; E 601, R613: H, R 614: Me, R 615: H, R 616: Et], [BC 1246; E601, R 613: Et, R 614: H, R 615: Me, R 616: H], [BC 1247; E 601, R 613: H, R 614: Et, R615: Me, R616: H], [BC1248; E601, R613: H, R614: H, R615: Me, R616: Et], [BC1249; E601, R613: Et, R614: H, R615: H, R616: Me], [BC1250; E601, R613: H, R614: Et, R615: H, R616: Me], [BC1251; E601, R613: H, R614: H, R615: Et, R616: Me], [ BC1252; E601, R613: Me, R614: Me, R615: Et, R616: H], [BC1253; E601, R613: Me, R614: Me, R615: H, R616: Et], [BC1254; E601, R613: Me, R 614: Et, R 615: Me, R 616: H], [BC1 255; E601, R 613: Me, R 614: H, R 615: Me, R 616: Et], [BC 1 256; E601, R 613: Me, R 614: Et, R615: H, R616: Me] , [BC1257; E601, R613: Me, R614: H, R615: Et, R616: Me], [BC1258; E601, R613: Me, R614: CF 3, R615: H, R616 : H], [BC1259; E601 , R613: Me, R614: H, R615: CF 3, R616: H], [BC1260; E601, R613: Me, R614: H, R615: H, R616: CF 3], [BC1261; E601, R613: CF 3, R614: Me, R615: H, R616: H], [BC1262; E601, R613: H, R614: Me, R615: CF 3, R616: H], [BC1263; E601 , R613: H, R614: Me , R615: H, R616: CF 3], [BC1264; E601, R613: CF 3, R614: H, R615: Me, R616: H], [BC1265; E601, R613: H _{, R614: CF 3, R615:} Me, R616: H], [BC1266; E601, R613: H, R614: H, R615: Me, R616: CF 3], [BC1267; E601 _{, R613: CF 3, R614:} H, R615: H, R616: Me], [BC1268; E601, R613: H, R614: CF 3, R615: H, R616: Me], [BC1269; E601, R613: H , R614: H, R615: CF 3, R616: Me], [BC1270; E601, R613: Me, R614: c-Pr, R615: H, R616: H], [BC1271; E601, R613: Me, R614: H, R615: c-Pr, R616: H], [BC1272; E601, R613: Me, R614: H, R615: H, R616: c-Pr], [BC1273; E601, R613: c-Pr, R614: Me, R615: H, R616: H], [BC1274; E601, R613: H, R614: Me, R615: c-Pr, R616: H], [BC1275; E601, R613: H, R614: Me, R615: H, R616: c-Pr], [BC1276; E601, R613: c-Pr, R614: H, R615: Me, R616: H], [BC1277; E601, R613: H, R614: c-Pr, R615: Me, R 616: H], [BC 1278; E 601, R 613: H, R 614: H, R 615: Me, R 616: c-Pr], [BC 1279; E 601, R 613: c-Pr, R 614: H, R 615: H, R616: Me], [BC 1280; E601, R 613: H, R 614: c-Pr, R 615: H, R 616: Me], [BC 1281; E 601, R 613: H, R 614: H, R 615: c-Pr, R 616: Me], [BC1282; E601, R613: Et, R614: H, R615: H, R616: H], [BC1283; E601, R613: H, R614: Et, R615: H, R616: H], [BC1284; E601, R 613: H, R 614: H, R 615: Et, R 616: H], [BC 1285; E 601, R 613: H, R 614: H, R 615: H, R 616: Et], [BC 1286; E 601, R 613: Et, R614: Et, R615: H, R616: H], [BC1287; E601, R613: Et, R614: H, R615: Et, R616: H], [BC1 288; E601, R613: Et, R614: H, R615: H, R 616: Et], [BC 1 289; E 601, R 6 13: H, R 614: Et, R 615: Et, R 616: H], [BC 1290; E 601, R 613: H, R 614: Et, R 615: H, R 616: Et], [BC 1291; E 601, R 613: H, R 614: H, R615: Et, R616: Et], [BC1292; E601, R613: Et, R614: Et, R615: Et, R615: H], [BC1293; E601, R613: Et, R614: Et, R615: H, R616: Et], [BC1294; E601, R613: Et, R614: F, R615: H, R616: H], [BC 1295; E601, R613: Et, R614: H, R615: F, R616: H], [ BC1296; E601, R613: Et, R614: H, R615: H, R616: F], [BC1297; E601, R613: Et, R614: F, R615: F, R616: H], [BC 1298; E601, R613: Et, R614: F, R615: H, R616: F], [BC1299; E601, R613: Et, R614: H, R615: F, R616: F], [BC1300; E601, R613: F, R614: Et, R 615: H, R 616: H],

[BC1301; E601, R613: H, R614: Et, R615: F, R616: H], [BC1302; E601, R613: H, R614: Et, R615: H, R616: F], [BC1303; E601, R613 : F, R 614: Et, R 615: F, R 616: H], [BC1 304; E601, R 613: F, R 614: Et, R 615: H, R 616: F], [BC 1 305; E 601, R 613: H, R 614: Et , R615: F, R616: F], [BC1306; E601, R613: F, R614: H, R615: Et, R616: H], [BC1307; E601, R613: H, R614: F, R615: Et, R616] : H], [BC1308; E601, R613: H, R614: H, R615: Et, R616: F], [BC1309; E601, R613: F, R614: F, R615: Et, R616: H], [BC1310 E601, R 613: F, R 614: H, R 615: Et, R 616: F], [BC 1311; E 601, R 613: H, R 614: F, R 615: Et, R 616: F], [BC 1312; E 601, R 613: F , R 614: H, R 615: H, R 616: Et], [BC 1313; E 601, R 613: H, R 614: F, R 615: H, R 616: Et], [BC 1314; E 601, R 613: H, R 614: H, R 615 : F, R 616: Et], [BC 1315; E 601, R 613: F, R 614: F, R 615: H, R 616: Et], [BC 1316; E 601, R 613: F, R 614: H, R 615: F, R 616: Et ], [BC1317; E601, R613: H, R614: F, R615: F, R616: Et], [BC1318; E601, R613: Et, R614: Et, R615: F, R616: H], [BC 1319; E601] , R613: Et, R614: Et, R615: H, R616: F], [BC1320; E601, R613: Et, R614: F, R615: Et, R616: H], [BC1321; E601, R613: Et, R614] : H, R615: Et, R616: F], [BC1322; E601, R613: Et, R614: F, R615: H, R616: Et], [BC1323; E601, R613: Et, R614: Et, R615: Cl , R 616: H], [BC 1 324; E601, R613: Et, R614: Et, R615: H, R616: Cl], [BC1325; E601, R613: Et, R614: Cl, R615: Et, R616: H], [BC1326; E601, R613: Et, R614: H, R615: Et, R616: Cl], [BC1327; E601, R613: Et, R614: Cl, R615: H, R616: Et], [BC1328; E601, R613: Et, R614: H, R615: Cl, R616: Et], [BC1329; E601, R613: Et, R614: Cl, R615: H, R616: H], [BC1330; E601, R613: Et, R614: H, R615: Cl, R616: H], [BC1331; E601, R613: Et, R614: H, R615: H, R616: Cl], [BC1332; E601, R613: Et, R614: Cl, R615: Cl, R616: H], [BC1333; E601, R613: Et, R614: Cl, R615: H, R616: Cl], [BC1334; E601, R613: Et, R614: H, R615: Cl, R616: Cl], [BC1335; E601, R613: Cl, R614: Et, R615: H, R616: H], [BC1336; E601, R613: H, R614: Et, R615: Cl, R616: H], [BC1337; E601, R613: H, R614: Et, R615: H, R616: Cl], [BC1338; E601, R613: Cl, R614: Et, R615: Cl, R616: H], [BC1339; E601, R613: Cl, R614: Et, R615: H, R616: Cl] , [BC1340; E601, R613: H, R614: Et, R615: Cl, R616: Cl], [BC1341; E601, R613: Cl, R614: H, R615: Et, R616: H], [BC1342; R613: H, R 614: Cl, R 615: Et, R 616: H], [BC 1343; E601, R 613: H, R 614: H, R 615: Et, R 616: Cl], [BC 1344; E 601, R 613: Cl, R 614: Cl, R615: Et, R616: H], [BC1345; E601, R613: Cl, R614: H, R615: Et, R616: Cl], [BC1346; E601, R613: H, R61 4: Cl, R615: Et, R616: Cl], [BC1347; E601, R613: Cl, R614: H, R615: H, R616: Et], [BC1348; E601, R613: H, R614: Cl, R615: H, R 616: Et], [BC 1 349; E 601, R 613: H, R 614: H, R 615: Cl, R 616: Et], [BC 1 350; E 601, R 613: Cl, R 614: Cl, R 615: H, R 616: Et] [BC1351; E601, R613: Cl, R614: H, R615: Cl, R616: Et], [BC1352; E601, R613: H, R614: Cl, R615: Cl, R616: Et], [BC1353; E601, E601, R613: Et, R614: CN, R615: H, R616: H], [BC1354; E601, R613: Et, R614: H, R615: CN, R616: H], [BC1 355; E601, R613: Et, R614: H, R615: H, R616: CN], [BC1356; E601, R613: CN, R614: Et, R615: H, R616: H], [BC1 357; E601, R613: H, R614: Et, R615: CN, R616: H], [BC1358; E601, R613: H, R614: Et, R615: H, R616: CN], [BC1359; E601, R613: CN, R614: H, R615: Et, R616: H], [ BC1360; E601, R613: H, R614: CN, R615: Et, R616: H], [BC1361; E601, R613: H, R614: H, R615: Et, R616: CN], [BC1362; E601, R613: CN, R 614: H, R 615: H, R 616: Et], [BC 1363; E601, R 613: H, R 614: CN, R 615: H, R 616: Et], [BC 1364; E 601, R 613: H, R 614: H, R615: CN, R616: Et] , [BC1365; E601, R613: Et, R614: CF 3, R615: H, R616: H], [BC1366; E601, R613: Et, R614: H, R615: CF 3, R 616: H], [BC 1367; E 601, R 613: Et, R 614: H, R 615: H, R 616: CF ₃ ], [BC 1 368; E 601, R 613: CF ₃ , R 614: Et, R 615: H, R 61 6: H], [BC1369; E601, R613: H, R614: Et, R615: CF 3, R616: H], [BC1370; E601, R613: H, R614: Et, R615: H, R616: CF 3] , [BC1371; E601, R613: CF 3, R614: H, R615: Et, R616: H], [BC1372; E601, R613: H, R614: CF 3, R615: Et, R616: H], [BC1373; E601, R613: H, R614: H, R615: Et, R616: CF 3], [BC1374; E601, R613: CF 3, R614: H, R615: H, R616: Et], [BC1375; E601, R613: _{H, R614: CF 3, R615} : H, R616: Et], [BC1376; E601, R613: H, R614: H, R615: CF 3, R616: Et], [BC1377; E601, R613: Et, R614: OMe, R615: H, R616: H], [BC1378; E601, R613: Et, R614: H, R615: OMe, R616: H], [BC1379; E601, R613: Et, R614: H, R615: H, R616: OMe], [BC1380; E601, R613: OMe, R614: Et, R615: H, R616: H], [BC1381; E601, R613: H, R614: Et, R615: OMe, R616: H], [ BC1382; E601, R613: H, R614: Et, R615: H, R616: OMe], [BC1383; E601, R613: OMe, R614: H, R615: Et, R616: H], [BC1384; E601, R613: H, R614: OMe, R615: Et, R616: H], [BC1385; E601, R613: H, R614: H, R615: Et, R616: OMe], [BC1386; E601, R613: OMe, R614: H, R615: H, R616: Et], [BC1387; E601, R613: H, R614: OMe, R615: H, R616: Et], [BC1388; E601, R613: H, R614: H, R615: OMe, R616: Et], [BC1389; E601, R613: F, R614: H, R615: H, R616: H], [BC1390; E601, R613: H, R614: F, R615: H, R61 6: H], [BC1391; E601, R613: H, R614: H, R615: F, R616: H], [BC1392; E601, R613: H, R614: H, R615: H, R616: F], [ BC1393; E601, R613: F, R614: F, R615: H, R616: H], [BC1394; E601, R613: F, R614: H, R615: F, R616: H], [BC 1395; E601, R613: F, R 614: H, R 615: H, R 616: F], [BC 1396; E 601, R 613: H, R 614: F, R 615: F, R 616: H], [BC 1397; E 601, R 613: H, R 614: F, R615: H, R 616: F], [BC 1398; E 601, R 613: H, R 614: F, R 615: F, R 616: F], [BC 1 399; H], [BC1400; E601, R613: F, R 614: H, R 615: F, R 616: F],

[BC1401; E601, R613: F, R614: F, R615: H, R616: F], [BC1402; E601, R613: Cl, R614: H, R615: H, R616: H], [BC1403; E601, R613 : H, R 614: Cl, R 615: H, R 616: H], [BC1404; E601, R 613: H, R 614: H, R 615: Cl, R 616: H], [BC 1 405; E 601, R 613: H, R 614: H , R615: H, R616: Cl], [BC1406; E601, R613: Cl, R614: Cl, R615: H, R616: H], [BC1407; E601, R613: Cl, R614: H, R615: Cl, R616 : H], [BC1408; E601, R613: Cl, R614: H, R615: H, R616: Cl], [BC1409; E601, R613: H, R614: Cl, R615: Cl, R616: H], [BC1410 E601, R 613: H, R 614: Cl, R 615: H, R 616: Cl], [BC 1411; E 601, R 613: H, R 614: H, R 615: Cl, R 616: Cl], [BC 1412; E 601, R 613: Cl , R614: H, R615: Cl, R616: Cl], [BC 1413; E601, R613: Cl, R614: Cl, R615: H, R616: Cl], [BC 1414; E601, R613: Cl, R614: Cl, R615 : Cl, R 616: H], [BC 1415; E 601, R 613: F, R 614: Cl, R 615: H, R 616: H], [BC 1416; E 601, R 613: F, R 614: H, R 615: Cl, R 616: H ], [BC1417; E601, R613: F, R614: H, R615: H, R616: Cl], [BC1418; E601, R613: Cl, R614: F, R615: H, R616: H], [BC 1419; E601] , R 613: H, R 614: F, R 615: Cl, R 616: H], [BC 1420; E 601, R 613: H, R 614: F, R 615: H, R 616: Cl], [BC 1421; : H, R 615: F, R 616: H], [BC 1422; E 601, R 613: H, R 614: Cl, R 615: F, R 616: H], [BC 1423; E 601, R 613: H, R 614: H, R 615: F , R 616: Cl], [BC1424; E601, R613: Cl, R614: H, R615: H, R616: F], [BC1425; E601, R613: H, R614: Cl, R615: H, R616: F], [BC1426; E601, R613 : H, R 614: H, R 615: Cl, R 616: F], [BC 1427; E601, R 613: Pr, R 614: H, R 615: H, R 616: H], [BC 1428; E 601, R 613: H, R 614: Pr , R 615: H, R 616: H], [BC 1429; H 601, R 613: H, R 614: H, R 615: Pr, R 616: H], [BC 1430; : Pr], [BC1431; E601, R613: isopropyl, R614: H, R615: H, R616: H], [BC1432; E601, R613: H, R614: isopropyl, R615: H, R616: H], [BC1433 E601, R 613: H, R 614: H, R 615: isopropyl, R 616: H], [BC 1434; E 601, R 613: H, R 614: H, R 615: H, R 616: isopropyl], [BC 1435; E 601, R 613: c -Pr, R 614: H, R 615: H, R 616: H], [BC 1436; E601, R 613: H, R 614: c-Pr, R 615: H, R 616: H], [BC 1 437; E 601, R 613: H, R 614 : H, R 615: c-Pr, R 616: H], [BC 1438; E 601, R 613: H, R 614: H, R 615: H, R 616: c-Pr], [BC 1439; E 601, R 613: c-Pr, R 614 : F, R 615: H, R 616: H], [BC 1440; E 601, R 613: c-Pr, R 614: H, R 615: F, R 616: H], [BC 1441; E 601, R 613: c-Pr, R 614: H , R615: H, R616: F], [BC1442; E601, R613: F, R614: c-Pr, R615: H, R616: H], [BC 1443; E601, R613: H, R614: c-Pr, R615 : F, R 616: H], [BC 1444; E 601, R 613: H, R 614: c-Pr, R 615: H, R 616: F], [BC 1445; E 601, R 613: F, R 614: H, R 615: c-Pr , R 616: H], [BC 1 446; E601, R613: H, R 614: F, R 615: c-Pr, R 616: H], [BC1447; E601, R 613: H, R 614: H, R 615: c-Pr, R 616: F], [BC 1448; E601, R 613: F, R 614: H, R 615: H, R 616: c-Pr], [BC1449; E601, R 613: H, R 614: F, R 615: H, R 616: c-Pr], [BC 1450; R613: H, R 614: H, R 615: F, R 616: c-Pr], [BC 1451; E601, R 613: c-Pr, R 614: Cl, R 615: H, R 616: H], [BC 1452; c-Pr, R614: H, R615: Cl, R616: H], [BC1453; E601, R613: c-Pr, R614: H, R615: H, R616: Cl], [BC1454; E601, R613: Cl, R614: c-Pr, R615: H, R616: H], [BC1455; E601, R613: H, R614: c-Pr, R615: Cl, R616: H], [BC1456; E601, R613: H, R614: c-Pr, R615: H, R616: Cl], [BC1457; E601, R613: Cl, R614: H, R615: c-Pr, R616: H], [BC1458; E601, R613: H, R614: Cl, R615: c-Pr, R616: H], [BC1459; E601, R613: H, R614: H, R615: c-Pr, R616: Cl], [BC 1460; E601, R613: Cl, R614: H, R615: H, R 616: c-Pr], [BC 1461; E 601, R 613: H, R 614: Cl, R 615: H, R 616: c-Pr], [BC 1462; E 601, R 613: H, R 614: H, R 615: Cl, R616: c-Pr], [BC1463; E601, R613: OMe, R614: H, R615: H, R616: H], [BC1464; E601, R613: H, R614: H, R615: H, R616: OMe] , [BC1465; E601, R613: OMe, R614: H, R615: H, R616: H], [BC1466; E601, R613: OMe, R614: H, R615: H, R616: H], [BC1467; R613: H, R 614: OMe, R 615: H, R 616: H], [BC 1468] E601, R613: H, R614: H, R615: OMe, R616: H], [BC1469; E601, R613: H, R614: H, R615: H, R616: OMe], [BC 1470; E601, R613: OMe] , R614: F, R615: H, R616: H], [BC1471; E601, R613: OMe, R614: H, R615: F, R616: H], [BC1472; E601, R613: OMe, R614: H, R615 : H, R 616: F], [BC 1 473; E 601, R 613: F, R 614: OMe, R 615: H, R 616: H], [BC 1 474; ], [BC1475; E601, R613: H, R614: OMe, R615: H, R616: F], [BC1476; E601, R613: F, R614: H, R615: OMe, R616: H], [BC1477; , R613: H, R 614: F, R 615: OMe, R 616: H], [BC1478; E601, R613: H, R 614: H, R 615: OMe, R 616: F], [BC1479; : H, R615: H, R616: OMe], [BC1480; E601, R613: H, R614: F, R615: H, R616: OMe], [BC1481; E601, R613: H, R614: H, R615: F , R616: OMe], [BC1482; E601, R613: Cl, R614: Cl, R615: H, R616: H], [BC1483; E601, R613: OMe, R614: H, R615: Cl, R616: H], [BC1484; E601, R613: OMe, R614: H, R615: H, R616: Cl], [BC1485; E601, R613: Cl, R614: OMe, R615: H, R616: H], [BC1486; E601, R613 : H, R614: OMe, R615: Cl, R616: H], [BC1487; E601, R613: H, R614: OMe, R615: H, R616: Cl], [BC1488; E601, R613: Cl, R614: H , R615: OMe, R616: H], [BC1489; E601, R613: H, R614: Cl, R615: OMe, R616: H], [BC1490; E601, R613: H, R614: H, R615] : OMe, R616: Cl], [BC1491; E601, R613: Cl, R614: H, R615: H, R616: OMe], [BC1492; E601, R613: H, R614: Cl, R615: H, R616: OMe ], [BC1493; E601, R613: H, R614: H, R615: Cl, R616: OMe], [BC1494; E601, R613: CN, R614: H, R615: H, R616: H], [BC1495; E601] , R 613: H, R 614: CN, R 615: H, R 616: H], [BC 1496; E 601, R 613: H, R 614: H, R 615: CN, R 616: H], [BC 1497; : H, R615: H, R616: CN], [BC1498; E601, R613: CN, R614: F, R615: H, R616: H], [BC1499; E601, R613: CN, R614: H, R615: F , R 616: H], [BC 1500; E 601, R 613: CN, R 614: H, R 615: H, R 616: F],

[BC1501; E601, R613: F, R614: CN, R615: H, R616: H], [BC1502; E601, R613: H, R614: CN, R615: F, R616: H], [BC1503; E601, R613 : H, R 614: CN, R 615: H, R 616: F], [BC 1504; E 601, R 613: F, R 614: H, R 615: CN, R 616: H], [BC 1505; E 601, R 613: H, R 614: F , R615: CN, R616: H], [BC1506; E601, R613: H, R614: H, R615: CN, R616: F], [BC1507; E601, R613: F, R614: H, R615: H, R616] : CN], [BC1508; E601, R613: H, R614: F, R615: H, R616: CN], [BC1509; E601, R613: H, R614: H, R615: F, R616: CN], [BC1510] E601, R613: CN, R614: Cl, R615: H, R616: H], [BC1511; E601, R613: CN, R614: H, R615: Cl, R616: H], [BC1512; E601, R613: CN , R 614: H, R 615: H, R 616: Cl], [BC 1513; E 601, R 613: Cl, R 614: CN, R 615: H, R 616: H], [BC 1514; E 601, R 613: H, R 614: CN, R 615 : Cl, R 616: H], [BC 1515; E 601, R 613: H, R 614: CN, R 615: H, R 616: Cl], [BC 1516; E 601, R 613: Cl, R 614: H, R 615: CN, R 616: H ], [BC1517; E601, R613: H, R614: Cl, R615: CN, R616: H], [BC1518; E601, R613: H, R614: H, R615: CN, R616: Cl], [BC1519; E601] , R 613: Cl, R 614: H, R 615: H, R 616: CN], [BC 1520; E 601, R 613: H, R 614: Cl, R 615: H, R 616: CN], [BC 1521; E 601, R 613: H, R 614 : H, R615: Cl, R616 : CN], [BC1522; E601, R613: NH 2, R614: H, R615: H, R616: H], [BC1523; E601, R613: H, R614: NH 2, R615 : H, R 616: H], [BC1524; E601, R613: H, R614: H, R615: NH 2, R616: H], [BC1525; E601, R613: H, R614: H, R615: H, R616: NH 2] , [BC1526; E601, R613: NH 2, R614: F, R615: H, R616: H], [BC1527; E601, R613: NH 2, R614: H, R615: F, R616: H], [BC1528; _{E601, R613: NH 2, R614} : H, R615: H, R616: F], [BC1529; E601, R613: F, R614: NH 2, R615: H, R616: H], [BC1530; E601, R613: _{H, R614: NH 2, R615} : F, R616: H], [BC1531; E601, R613: H, R614: NH 2, R615: H, R616: F], [BC1532; E601, R613: F, R614: _{H, R615: NH 2, R616} : H], [BC1533; E601, R613: H, R614: F, R615: NH 2, R616: H], [BC1534; E601, R613: H, R614: H, R615: _{NH 2, R616: F],} [BC1535; E601, R613: F, R614: H, R615: H, R616: NH 2], [BC1536; E601, R613: H, R614: F, R615: H, R616: _{NH 2], [BC1537; E601} , R613: H, R614: H, R615: F, R616: NH 2], [BC1538; E601, R613: NH 2, R614: Cl, R615: H, R616: H], [BC1539; E601, R613: NH 2, R614: H, R615: Cl, R616: H], [BC1540; E601, R613: NH 2, R614: H, R615: H, R616: Cl], [BC1541; E601 , R613: Cl, R614: NH 2, R615: H, R616: H], [BC1542; E601, R613: H, R614: NH 2, R615: Cl, R616: H], [BC1543; E601, R613: H _{, R614: NH 2, R615:} H, R616: Cl], [BC1544; E601, R613: Cl, R614: H, R615: NH 2, R616: H], [BC1545; E601, R613: H, _{R614: Cl, R615: NH 2} , R616: H], [BC1546; E601, R613: H, R614: H, R615: NH 2, R616: Cl], [BC1547; E601, R613: Cl, R614: H, _{R615: H, R616: NH 2} ], [BC1548; E601, R613: H, R614: Cl, R615: H, R616: NH 2], [BC1549; E601, R613: H, R614: H, R615: Cl, R616: NH ₂ ], [BC1550; E601, R613: NHMe, R614: H, R615: H, R616: H], [BC1551; E601, R613: H, R614: NHMe, R615: H, R616: H], [BC1552; E601, R613: H, R614: H, R615: NHMe, R616: H], [BC1553; E601, R613: H, R614: H, R615: H, R616: NHMe], [BC1554; E601, R613 : NHMe, R 614: F, R 615: H, R 616: H], [BC 1555; E601, R 613: NHMe, R 614: H, R 615: F, R 616: H], [BC 1 556; , R615: H, R616: F], [BC1557; E601, R613: F, R614: NHMe, R615: H, R616: H], [BC1 558; E601, R613: H, R614: NHMe, R615: F, R616] : H], [BC1559; E601, R613: H, R614: NHMe, R615: H, R616: F], [BC1560; E601, R613: F, R614: H, R615: NHMe, R616: H], [BC1561 E601, R613: H, R614: F, R615: NHMe, R616: H], [BC1562; E601, R613: H, R614: H, R615: NHMe, R616: F], [BC1563; E601, R613: F , R614: H, R615: H, R616: NHMe], [BC1564; E601, R613: H, R614: F, R615: H, R616: NHMe], [BC1565; E601, R613: H, R614: H, R615] : F, R 616: NHMe], [BC 1566; E601, R 613: NHMe, R 614: Cl, R 615: H, R 616: H], [BC 1 567; E 601, R 613: N HMe, R614: H, R615: Cl, R616: H], [BC1568; E601, R613: NHMe, R614: H, R615: H, R616: Cl], [BC1569; E601, R613: Cl, R614: NHMe, R615: H, R616: H], [BC1570; E601, R613: H, R614: NHMe, R615: Cl, R616: H], [BC1571; E601, R613: H, R614: NHMe, R615: H, R616: Cl], [BC1572; E601, R613: Cl, R614: H, R615: NHMe, R616: H], [BC1573; E601, R613: H, R614: Cl, R615: NHMe, R616: H], [BC1574; E601, R613: H, R614: H, R615: NHMe, R616: Cl], [BC1575; E601, R613: Cl, R614: H, R615: H, R616: NHMe], [BC1 576; E601, R613: H, R614: Cl, R615: H, R616: NHMe], [BC1577; E601, R613: H, R614: H, R615: Cl, R616: NHMe], [BC1578; E601, R613: NMe 2, R614: H, R615 : H, R616: H], [BC1579; E601, R613: H, R614: NMe 2, R615: H, R616: H], [BC1580; E601, R613: H, R614: H, R615: NMe 2, R616 : H], [BC1581; E601 , R613: H, R614: H, R615: H, R616: NMe 2], [BC1582; E601, R613: NMe 2, R614: F, R615: H, R616: H], [BC1583; E601, R613: NMe 2, R614: H, R615: F, R616: H], [BC1584; E601, R613: NMe 2, R614: H, R615: H, R616: F], [BC1585; E601 , R613: F, R614: NMe 2, R615: H, R616: H], [BC1586; E601, R613: H, R614: NMe 2, R615: F, R616: H], [BC1587; E601, R613: H _{, R614: NMe 2, R615:} H, R616: F], [BC1588; E601, R613: F, R614: H, R615: NMe 2, R616 : H], [BC1589; E601 , R613: H, R614: F, R615: NMe 2, R616: H], [BC1590; E601, R613: H, R614: H, R615: NMe 2, R616: F], [BC1591; E601, R613: F , R614: H, R615: H, R616: NMe 2], [BC1592; E601, R613: H, R614: F, R615: H, R616: NMe 2], [BC1593; E601 , R613: H, R614: H , R615: F, R616: NMe 2], [BC1594; E601, R613: NMe 2, R614: Cl, R615: H, R616: H], [BC1595; E601, R613: NMe _{2, R614: H, R615:} Cl, R616: H], [BC1596; E601, R613: NMe 2, R614: H, R615: H, R616: Cl], [BC1597; E601, R613: Cl, R614: NMe _{2, R615: H, R616:} H], [BC1598; E601, R613: H, R614: NMe 2, R615: Cl, R616: H], [BC1599; E601, R613: H, R614: NMe 2, R615: H, R 616: Cl], [BC1600; E601, R 613: Cl, R 614: H, R 615: NMe ₂ , R 616: H],

[BC1601; E601, R613: H , R614: Cl, R615: NMe 2, R616: H], [BC1602; E601, R613: H, R614: H, R615: NMe 2, R616: Cl], [BC1603; E601 , R613: Cl, R614: H , R615: H, R616: NMe 2], [BC1604; E601, R613: H, R614: Cl, R615: H, R616: NMe 2], [BC1605; E601, R613: H , R614: H, R615: Cl , R616: NMe 2], [BC1606; E601, R613: SMe, R614: H, R615: H, R616: H], [BC1607; E601, R613: H, R614: SMe, R615: H, R616: H], [BC1608; E601, R613: H, R614: H, R615: SMe, R616: H], [BC1 609; E601, R613: H, R614: H, R 615: H, R616: SMe], [BC1610; E601, R613: SMe, R614: F, R615: H, R616: H], [BC1611; E601, R613: SMe, R614: H, R615: F, R616: H], [BC1612; E601, R613: SMe, R 614: H, R 615: H, R 616: F], [BC 1613; E 601, R 613: F, R 614: S Me, R 615: H, R 616: H], [BC 1614; E 601, R 613: H, R614: SMe, R615: F, R616: H], [BC1615; E601, R613: H, R614: SMe, R615: H, R616: F], [BC1616; E601, R613: F, R614: H, R615: SMe, R616: H], [BC1617; E601, R613: H, R614: F, R615: SMe, R616: H], [BC1618; E601, R613: H, R614: H, R615: SMe, R616: F] , [BC1619; E601, R613: F, R614: H, R615: H, R616: SMe], [BC1620; E601, R613: H, R614: F, R615: H, R616: SMe], [BC1621; E601, R613: H, R 614: H, R 615: F, R 616: SMe], [BC1622; E601, R613: SMe, R 614: Cl, R 615: H, R 616: H], [BC1623; 1, R613: SMe, R614: H, R615: Cl, R616: H], [BC1624; E601, R613: SMe, R614: H, R615: H, R616: Cl], [BC1625; E601, R613: Cl, R614: SMe, R615: H, R616: H], [BC1626; E601, R613: H, R614: SMe, R615: Cl, R616: H], [BC1627; E601, R613: H, R614: SMe, R615: H, R616: Cl], [BC1628; E601, R613: Cl, R614: H, R615: SMe, R616: H], [BC1629; E601, R613: H, R614: Cl, R615: SMe, R616: H] [BC1630; E601, R613: H, R614: H, R615: SMe, R616: Cl], [BC1631; E601, R613: Cl, R614: H, R615: H, R616: SMe], [BC1632; E601, R613: H, R614: Cl, R615: H, R616: SMe], [BC1633; E601, R613: H, R614: H, R615: Cl, R616: SMe], [BC1634; E601, R613: NO 2, R614 : H, R615: H, R616 : H], [BC1635; E601, R613: H, R614: NO 2, R615: H, R616: H], [BC1636; E601, R613: H, R614: H, R615: _{NO 2, R616: H],} [BC1637; E601, R613: H, R614: H, R615: H, R616: NO 2], [BC1638; E601, R613: NO 2, R614: F, R615: H, R616 : H], [BC1639; E601 , R613: NO 2, R614: H, R615: F, R616: H], [BC1640; E601, R613: NO 2, R614: H, R615: H, R616: F], [BC1641; E601, R613: F , R614: NO 2, R615: H, R616: H], [BC1642; E601, R613: H, R614: NO 2, R615: F, R616: H], [BC1643; E601 , R 613: H, R 614: NO ₂ , R 615: H, R 616: F], [BC 1644; E601, R 613: F, R 614: H, R 615: NO ₂ , R 616: H], [BC 1645; E 6 01, R 613: H, R 614: F, R 615: NO ₂ , R 616: H], [BC 1646; E 601, R 613: H, R 614: H, R 615: NO ₂ , R 616: F], [BC 1647; F, R614: H, R615: H, R616: NO 2], [BC1648; E601, R613: H, R614: F, R615: H, R616: NO 2], [BC1649; E601, R613: H, R614: H, R615: F, R616: NO 2], [BC1650; E601, R613: NO 2, R614: Cl, R615: H, R616: H], [BC1651; E601, R613: NO 2, R614: H, R615 : Cl, R616: H], [BC1652; E601, R613: NO 2, R614: H, R615: H, R616: Cl], [BC1653; E601, R613: Cl, R614: NO 2, R615: H, R616 : H], [BC1654; E601 , R613: H, R614: NO 2, R615: Cl, R616: H], [BC1655; E601, R613: H, R614: NO 2, R615: H, R616: Cl], [BC1656; E601, R613: Cl , R614: H, R615: NO 2, R616: H], [BC1657; E601, R613: H, R614: Cl, R615: NO 2, R616: H], [BC1658; E601 , R 613: H, R 614: H, R 615: NO ₂ , R 616: Cl], [BC 1659; E 601, R 613: Cl, R 614: H, R 615: H, R 616: NO ₂ ], [BC 1660; , R614: Cl, R615: H , R616: NO 2], [BC1661; E601, R613: H, R614: H, R615: Cl, R616: NO 2], [BC1662; E602, R612: H, R614: H , R615: H, R616: H], [BC1663; E602, R612: Me, R614: H, R615: H, R616: H], [BC1664; E602, R612: H, R614: Me, R615: H, R616] : H], [BC1665; E602, R612: H, R614: Me, R616: H], [BC1 666; E602, R612: H, R614: H, R615: H, R616: Me], [B C1667; E602, R612: Me, R614: Me, R615: H, R616: H], [BC1668; E602, R612: Me, R614: H, R615: Me, R616: H], [BC1669; E602, R612: Me, R614: H, R615: H, R616: Me], [BC1670; E602, R612: H, R614: Me, R615: Me, R616: H], [BC1671; E602, R612: H, R614: Me, R615: H, R616: Me], [BC1672; E602, R612: H, R614: H, R615: Me, R616: Me], [BC1673; E602, R612: H, R614: Me, R615: H, R616: H], [BC1674; E602, R612: Me, R614: Me, R615: Me, R616: H], [BC1 675; E602, R612: Me, R614: Me, R615: H, R616: Me], [BC1 676; E602, R612: Me, R614: H, R615: Me, R616: Me], [BC1677; E602, R612: H, R614: Me, R615: Me, R616: Me], [BC1678; E602, R612: Me, R614: Me, R615: Me, R616: Me], [BC1679; E602, R612: Me, R614: F, R615: H, R616: H], [BC1680; E602, R612: Me, R614: H, R615: F, R616: H], [BC1681; E602, R612: Me, R614: H, R615: H, R616: F], [BC1682; E602, R612: Me, R614: F, R615: F, R616: H] , [BC 1683; E 602, R 612: Me, R 614: F, R 615: H, R 616: F], [BC 1 684; E 602, R 612: Me, R 614: H, R 615: F, R 616: F], [BC 1 685; R612: Me, R614: F, R615: F, R616: F], [BC1686; E602, R612: F, R614: Me, R615: H, R616: H], [BC1687; E602, R612: H, R614: Me, R615: F, R616: H], [BC1688; E602, R612: H, R614: Me, R615: H, R616: F], [BC1689; E602, R612: F, R614: Me, R615: F, R616 : H], [BC1690; F602, R612: Me, R614: H, R616: F], [BC1691; E602, R612: H, R614: Me, R615: F, R616: F], [BC1692 E602, R612: F, R614: Me, R615: F, R616: F], [BC1693; E602, R612: F, R614: H, R615: Me, R616: H], [BC1694; E602, R612: H , R 614: F, R 615: Me, R 616: H], [BC 1695; E 602, R 612: H, R 614: H, R 615: Me, R 616: F], [BC 1 696; : Me, R 616: H], [BC 1697; E 602, R 612: F, R 614: H, R 615: Me, R 616: F], [BC 1698; E 602, R 612: H, R 614: F, R 615: Me, R 616: F ], [BC1699; E602, R612: F, R614: F, R615: Me, R616: F], [BC1700; E602, R612: F, R614: H, R615: H, R616: Me],

[BC1701; E602, R612: H, R614: F, R615: H, R616: Me], [BC1702; E602, R612: H, R614: H, R615: F, R616: Me], [BC1703; E602, R612 : F, R 614: F, R 615: H, R 616: Me], [BC 1704; E 602, R 612: F, R 614: H, R 615: F, R 616: Me], [BC 1 705; E 602, R 612: H, R 614: F , R615: F, R616: Me], [BC1706; E602, R612: F, R614: F, R615: F, R616: Me], [BC1707; E602, R612: Me, R614: Me, R615: F, R616] : H], [BC1708; E602, R612: Me, R614: Me, R615: H, R616: F], [BC1709; E602, R612: Me, R614: F, R615: Me, R616: H], [BC1710 E602, R612: Me, R614: H, R615: Me, R616: F], [BC1711; E602, R612: Me, R614: F, R615: H, R616: Me], [BC1712; E602, R612: Me , R614: H, R615: F, R616: Me], [BC1713; E602, R612: Me, R614: Me, R615: Cl, R616: H], [BC1714; E602, R612: Me, R614: Me, R615] : H, R 616: Cl], [BC 1715; E 602, R 612: Me, R 614: Cl, R 615: Me, R 616: H], [BC 1716; E 602, R 612: Me, R 614: H, R 615: Me, R 616: Cl ], [BC1717; E602, R612: Me, R614: Cl, R615: H, R616: Me], [BC1718; E602, R612: Me, R614: H, R615: Cl, R616: Me], [BC1719; , R612: Me, R614: Cl, R615: H, R616: H], [BC1720; E602, R612: Me, R614: H, R615: Cl, R616: H], [BC1721; E602, R612: Me, R614] : H, R615: H, R616: Cl], [BC1722; E602, R612: Me, R614: Cl, R615: Cl, R616: H], [BC1723; E602, R612: Me, R614: Cl, R6 15: H, R616: Cl], [BC1724; E602, R612: Me, R614: H, R615: Cl, R616: Cl], [BC1725; E602, R612: Cl, R614: Me, R615: H, R616: H], [BC1726; E602, R612: H, R614: Me, R615: Cl, R616: H], [BC1727; E602, R612: H, R614: Me, R615: H, R616: Cl], [BC1728; E602, R612: Cl, R614: Me, R615: Cl, R616: H], [BC1729; E602, R612: Cl, R614: Me, R615: H, R616: Cl], [BC1730; E602, R612: H, R614: Me, R615: Cl, R616: Cl], [BC1731; E602, R612: Cl, R614: H, R615: Me, R616: H], [BC1732; E602, R612: H, R614: Cl, R615: Me, R616: H], [BC1733; E602, R612: H, R614: Me, R616: Cl], [BC1734; E602, R612: Cl, R614: Cl, R615: Me, R616: H] [BC1735; E602, R612: Cl, R614: H, R615: Me, R616: Cl], [BC1736; E602, R612: H, R614: Cl, R615: Me, R616: Cl], [BC1 737; R612: Cl, R614: H, R615: H, R616: Me], [BC1738; E602, R612: H, R614: Cl, R615: H, R616: Me], [BC1739; E602, R612: H, R614: H, R615: Cl, R616: Me], [BC1740; E602, R612: Cl, R614: Cl, R615: H, R616: Me], [BC1741; E602, R612: Cl, R614: H, R615: Cl, R616: Me], [BC1742; E602, R612: H, R614: Cl, R615: Cl, R616: Me], [BC1743; E602, R612: Me, R614: Br, R615: H, R616: H], [ BC1744; E602, R612: Me, R614: H, R615: Br, R616: H], [BC1745; E602, R612: Me, R614: H, R615: H, R616: Br], [BC1746; E602, R612: Br, R614: Me, R615: H, R616: H], [BC1747; E602, R612: H, R614: Me, R615: Br, R616: H], [BC1 748; E602, R612: H, R614: Me, R615: H, R616: Br], [BC1749; E602, R612: Br, R614: H, R615: Me, R616: H], [BC1 750; E602, R612: H, R614: Br, R615: Me, R616: H], [BC1751; E602, R612: H, R614: H, R615: Me, R616: Br], [BC1752; E602, R612: Br, R614: H, R615: H, R616: Me] , [BC1753; E602, R612: H, R614: Br, R615: H, R616: Me], [BC1754; E602, R612: H, R614: H, R615: Br, R616: Me], [BC1 755; R612: Me, R614: Me, R615: Br, R616: H], [BC1756; E602, R612: Me, R614: Me, R615: H, R616: Br], [BC1757; E602, R612: Me, R614: Br, R615: Me, R616: H], [BC1758; E602, R612: Me, R614: H, R615: Me, R616: Br], [BC1759; E602, R612: Me, R614: Br, R615: H, R616: Me], [BC1760; E602, R612: H, R614: Br, R616: Me], [BC1761; E602, R612: Me, R614: CN, R615: H, R616: H], [ BC1762; E602, R612: Me, R614: H, R615: CN, R616: H], [BC1763; E602, R612: Me, R614: H, R615: H, R616: CN], [BC1764; E602, R612: CN, R 614: Me, R 615: H, R 616: H], [BC 1 765; E 602, R 612: H, R 614: Me, R 615: CN, R 616: H], [BC 1 766; E 602, R 612: H, R 614: Me, R615: H, R616: CN], [BC1767; E602, R612: CN, R614: H, R615: Me, R616: H], [BC1768; E602, R612: H, R614: CN, R615: M e, R 616: H], [BC 1769; E 602, R 612: H, R 614: Me, R 616: CN], [BC 1 770; E 602, R 612: CN, R 614: H, R 615: H, R 616: Me] , [BC1771; E602, R612: H, R614: CN, R615: H, R616: Me], [BC1772; E602, R612: H, R614: H, R615: CN, R616: Me], [BC1773; R612: Me, R614: Me, R615: CN, R616: H], [BC1774; E602, R612: Me, R614: Me, R615: H, R616: CN], [BC1 775; E602, R612: Me, R614: CN, R615: Me, R616: H], [BC1776; E602, R612: Me, R614: H, R615: Me, R616: CN], [BC1 777; E602, R612: Me, R614: CN, R615: H, R616: Me], [BC1778; E602, R612: H, R614: CN, R616: Me], [BC1779; E602, R612: Me, R614: OMe, R615: H, R616: H], [ BC1780; E602, R612: Me, R614: H, R615: OMe, R616: H], [BC1781; E602, R612: Me, R614: H, R615: H, R616: OMe], [BC1782; E602, R612: OMe, R614: Me, R615: H, R616: H], [BC1783; E602, R612: H, R614: Me, R615: OMe, R616: H], [BC1784; E602, R612: H, R614: Me, R615: H, R616: OMe], [BC1785; E602, R612: H, R614: Me, R616: H], [BC1 786; E602, R612: H, R614: OMe, R615: Me, R616: H], [BC1787; E602, R612: H, R614: Me, R615: Me, R616: OMe], [BC1 788; E602, R612: OMe, R614: H, R615: H, R616: Me], [BC1 789; E602, R612: H, R614: OMe, R615: H, R616: Me], [BC1790; E602, R612: H, R614: H, R615: OMe, R616: Me], [BC1 791; E602, R612: Me, R614: Me, R615: OMe, R616: H], [BC1792; E602, R612: Me, R614: Me, R615: H, R616: OMe], [BC1 793; E602, R612: Me, R614: OMe, R615: Me, R616: H], [BC1794; E602, R612: Me, R614: H, R615: Me, R616: OMe], [BC1795; E602, R612: Me, R614: OMe, R615: H, R616: Me], [BC1796; E602, R612: Me, R614: H, R615: OMe, R616: Me], [BC1 797; E602, R612: Me, R614: OET, R615: H, R616: H], [BC1798; E602, R612: Me, R614: H, R615: OEt, R616: H], [BC1799; E602, R612: Me, R614: H, R615: H, R616: OEt], [BC1800; E602, R612: OEt, R614: Me, R615: H, R616: H],

[BC1801; E602, R612: H, R614: Me, R615: OEt, R616: H], [BC1802; E602, R612: H, R614: Me, R615: H, R616: OEt], [BC1803; E602, R612 : OEt, R614: H, R615: Me, R616: H], [BC1804; E602, R612: H, R614: OEt, R615: Me, R616: H], [BC1805; E602, R612: H, R614: H , R615: Me, R616: OEt], [BC1806; E602, R612: H, R615: H, R615: H, R616: Me], [BC1807; E602, R612: H, R614: OEt, R615: H, R616] : Me], [BC1808; E602, R612: H, R614: H, R615: OEt, R616: Me], [BC1809; E602, R612: Me, R614: Me, R615: OEt, R616: H], [BC1810 E602, R612: Me, R614: Me, R615: H, R616: OEt], [BC 1811; E602, R612: Me, R614: OEt, R615: Me, R616: H], [BC1812; E602, R612: Me , R614: H, R615: Me, R616: OEt], [BC1813; E602, R612: Me, R614: OEt, R615: H, R616: Me], [BC1814; E602, R612: Me, R614: H, R615] : OEt, R616: Me], [BC1815; E602, R612: Me, R614: Et, R615: H, R616: H], [BC1816; E602, R612: Me, R614: H, R615: Et, R616: H ], [BC1817; E602, R612: Me, R614: H, R615: H, R616: Et], [BC1818; E602, R612: Et, R614: Me, R615: H, R616: H], [BC1819; , R612: H, R614: Me, R615: Et, R616: H], [BC1820; E602, R612: H, R614: Me, R615: H, R616: Et], [BC1821; E602, R612: Et, R614] : H, R 615: Me, R 616: H], [BC 1 822; E 602, R 612: H, R 614: Et, R 615: Me, R 616: H], [BC 1823; , R612: H, R614: H, R615: Me, R616: Et], [BC1824; E602, R612: Et, R614: H, R615: H, R616: Me], [BC1825; E602, R612: H, R614] : Et, R 615: H, R 616: Me], [BC 1826; E 602, R 612: H, R 614: H, R 615: Et, R 616: Me], [BC 1827; E 602, R 612: Me, R 614: Me, R 615: Et , R616: H], [BC1828; E602, R612: Me, R614: Me, R615: H, R616: Et], [BC1829; E602, R612: Me, R614: Et, R615: Me, R616: H], [BC1830; E602, R612: Me, R614: H, R615: Me, R616: Et], [BC1831; E602, R612: Me, R614: Et, R615: H, R616: Me], [BC1832; E602, R612 : Me, R614: H, R615 : Et, R616: Me], [BC1833; E602, R612: Me, R614: CF 3, R615: H, R616: H], [BC1834; E602, R612: Me, R614: _{H, R615: CF 3, R616} : H], [BC1835; E602, R612: Me, R614: H, R615: H, R616: CF 3], [BC1836; E602, R612: CF 3, R614: Me, R615 : H, R 616: H], [BC 1837; E 602, R 612: H, R 614: Me, R 615: CF ₃ , R 616: H], [BC 1838; E 602, R 612: H, R 614: Me, R 615: H, R 616: _{CF 3], [BC1839; E602} , R612: CF 3, R614: H, R615: Me, R616: H], [BC1840; E602, R612: H, R614: CF 3, R615: Me, R616: H], [BC1841; E602, R612: H , R614: H, R615: Me, R616: CF 3], [BC1842; E602, R612: CF 3, R614: H, R615: H, R616: Me], [BC1843; E602 , R612: H, R614: CF 3, R615: H, R616: Me], [BC1844; E602, R612: H, R614: H, R615: CF 3, R616: Me], [B C1845; E602, R612: Me, R614: c-Pr, R615: H, R616: H], [BC1846; E602, R612: Me, R614: H, R615: c-Pr, R616: H], [BC1847; E602, R612: Me, R614: H, R615: H, R616: c-Pr], [BC1848; E602, R612: c-Pr, R614: Me, R615: H, R616: H], [BC1849; E602, E602, R612: H, R614: Me, R615: c-Pr, R616: H], [BC1850; E602, R612: H, R614: Me, R615: H, R616: c-Pr], [BC1851; E602, R612: c-Pr, R 614: H, R 615: Me, R 616: H], [BC 1852; E 602, R 612: H, R 614: c-Pr, R 615: Me, R 616: H], [BC 1853; E 602, R 612: H, R614: H, R615: Me, R616: c-Pr], [BC1854; E602, R612: c-Pr, R614: H, R615: H, R616: Me], [BC1855; E602, R612: H, R614: c-Pr, R615: H, R616: Me], [BC1856; E602, R612: H, R614: H, R615: c-Pr, R616: Me], [BC1 857; E602, R612: Et, R614: H, R615: H, R616: H], [BC1858; E602, R612: H, R614: Et, R615: H, R616: H], [BC1859; E602, R612: H, R614: H, R615: Et, R616: H], [BC1860; E602, R612: H, R614: H, R615: H, R616: Et], [BC1861; E602, R612: Et, R614: Et, R615: H, R616: H], [BC1862; E602, R612: Et, R614: H, R615: Et, R616: H], [BC1863; E602, R612: Et, R614: H, R615: H, R616: Et], [BC 1864; E602, R612: H, R614: Et, R615: Et, R616: H], [BC1865; E602, R612: H, R614: Et, R615: H, R616: Et], [BC 1866; E602, R612: H, R614: H, R615: Et, R 616: Et], [BC 1867; E 602, R 612: Et, R614: Et, R615: Et, R616: H], [BC1868; E602, R612: Et, R614: Et, R615: H, R616: Et], [BC1869; E602, R612: Et, R614: F, R 615: H, R 616: H], [BC 1 870; E 602, R 612: Et, R 614: H, R 615: F, R 616: H], [BC 187 1; E 602, R 612: Et, R 614: H, R 615: H, R616: F], [BC1872; E602, R612: Et, R614: F, R615: F, R616: H], [BC1 873; E602, R612: Et, R614: F, R615: H, R616: F], [ BC1874; E602, R612: Et, R614: H, R615: F, R616: F], [BC1875; E602, R612: F, R614: Et, R615: H, R616: H], [BC1876; E602, R612: H, R 614: Et, R 615: F, R 616: H], [BC 1877; E 602, R 612: H, R 614: Et, R 615: H, R 616: F], [BC 1878; E 602, R 612: F, R 614: Et, R615: F, R 616: H], [BC 1879; E 602, R 612: F, R 614: Et, R 615: H, R 616: F], [BC 1 880; E 602, R 612: H, R 614: Et, R 615: F, R 616: F], [BC1881; E602, R612: F, R614: H, R615: Et, R616: H], [BC1882; E602, R612: H, R614: F, R615: Et, R616: H], [BC 1883; E602, R612: H, R614: H, R615: Et, R616: F], [BC1884; E602, R612: F, R614: F, R615: Et, R616: H], [BC1885; E602, R612: F, R614: H, R 615: Et, R 616: F], [BC 1886; E 602, R 612: H, R 614: F, R 615: Et, R 616: F], [BC 1887; E 602, R 612: F, R 614: H, R 615: H, R616: Et], [BC1888; E602, R612: F, R614: F, R615: H, R616: Et], [BC1889; E602, R612: H, R614: H, R615: F, R616: Et] , [BC1890; E602, R612: F, R 614: F, R615: H, R616: Et], [BC1891; E602, R612: F, R614: H, R615: F, R616: Et], [BC1892; E602, R612: H, R614: F, R615: F, R616: Et], [BC1893; E602, R612: Et, R614: Et, R615: F, R616: H], [BC1894; E602, R612: Et, R614: Et, R615: H, R616: F] , [BC1895; E602, R612: Et, R614: F, R615: Et, R616: H], [BC1896; E602, R612: Et, R614: H, R615: Et, R616: F], [BC1897; R612: Et, R614: F, R615: H, R616: Et], [BC1898; E602, R612: Et, R614: Et, R615: Cl, R616: H], [BC1899; E602, R612: Et, R614: Et, R615: H, R616: Cl], [BC 1900; E602, R612: Et, R614: Cl, R615: Et, R616: H],

[BC1901; E602, R612: Et, R614: H, R615: Et, R616: Cl], [BC1902; E602, R612: Et, R614: Cl, R615: H, R616: Et], [BC1903; E602, R612 : Et, R 614: H, R 615: Cl, R 616: Et], [BC 1904; E 602, R 612: Et, R 614: Cl, R 615: H, R 616: H], [BC 1 905; E 602, R 612: Et, R 614: H , R615: Cl, R616: H], [BC1906; E602, R612: Et, R614: H, R615: H, R616: Cl], [BC1907; E602, R612: Et, R614: Cl, R615: Cl, R616] : H], [BC1908; E602, R612: Et, R614: Cl, R615: H, R616: Cl], [BC1909; E602, R612: Et, R614: H, R615: Cl, R616: Cl], [BC1910 E602, R612: Cl, R614: Et, R615: H, R616: H], [BC1911; E602, R612: H, R614: Et, R615: Cl, R616: H], [BC 1912; E602, R612: H , R614: Et, R615: H, R616: Cl], [BC1913; E602, R612: Cl, R614: Et, R615: Cl, R616: H], [BC1914; E602, R612: Cl, R614: Et, R615 : H, R 616: Cl], [BC 1915; E 602, R 612: H, R 614: Et, R 615: Cl, R 616: Cl], [BC 1916; E 602, R 612: Cl, R 614: H, R 615: Et, R 616: H ], [BC1917; E602, R612: H, R614: Cl, R615: Et, R616: H], [BC1918; E602, R612: H, R614: H, R615: Et, R616: Cl], [BC1919; , R612: Cl, R614: Cl, R615: Et, R616: H], [BC1920; E602, R612: Cl, R614: H, R615: Et, R616: Cl], [BC1921; E602, R612: H, R614] : Cl, R615: Et, R616: Cl], [BC1922; E602, R612: Cl, R614: H, R615: H, R616: Et], [BC1923; E602, R612: H, R614: Cl, R615: H, R616: Et], [BC1924; E602, R612: H, R614: H, R615: Cl, R616: Et], [BC1925; E602, R612: Cl, R614: Cl, R615: H, R 616: Et], [BC 1926; E 602, R 612: Cl, R 614: H, R 615: Cl, R 616: Et], [BC 1 927; E 602, R 612: H, R 614: Cl, R 615: Cl, R 616: Et] , [BC1928; E602, R612: Et, R614: CN, R615: H, R616: H], [BC1929; E602, R612: Et, R614: H, R615: CN, R616: H], [BC1930; R612: Et, R614: H, R615: H, R616: CN], [BC1931; E602, R612: CN, R614: Et, R615: H, R616: H], [BC1932; E602, R612: H, R614: Et, R615: CN, R616: H], [BC1933; E602, R612: H, R614: Et, R615: H, R616: CN], [BC1 934; E602, R612: CN, R614: H, R615: Et, R615: Et, R 616: H], [BC 1935; E 602, R 612: H, R 614: CN, R 615: Et, R 616: H], [BC 1 936; E 602, R 612: H, R 614: H, R 615: Et, R 616: CN], [ BC1937; E602, R612: CN, R614: H, R615: H, R616: Et], [BC1938; E602, R612: H, R614: CN, R615: H, R616: Et], [BC 1939; E602, R612: H, R614: H, R615: CN, R616: Et], [BC1940; E602, R612: Et, R614: CF 3, R615: H, R616: H], [BC1941; E602, R612: Et, R614: H _{, R615: CF 3, R616:} H], [BC1942; E602, R612: Et, R614: H, R615: H, R616: CF 3], [BC1943; E602, R612: CF 3, R614: Et, R615: H, R 616: H], [BC 1 944; E 602, R 612: H, R 614: Et, R 615: CF ₃ , R 616: H], [BC 1 945; E 602, R 612: H, R 614: Et, R 615: H _{, R616: CF 3], [} BC1946; E602, R612: CF 3, R614: H, R615: Et, R616: H], [BC1947; E602, R612: H, R614: CF 3, R615: Et, R616: H], [BC1948; E602, R612: H, R614: H, R615: Et, R616: CF 3], [BC1949; E602, R612: CF 3, R614: H, R615: H, R616: Et], [ BC1950; E602, R612: H, R614: CF 3, R615: H, R616: Et], [BC1951; E602, R612: H, R614: H, R615: CF 3, R616: Et], [BC1952; E602, R612: Et, R614: OMe, R615: H, R616: H], [BC1953; E602, R612: Et, R614: H, R615: OMe, R616: H], [BC1954; E602, R612: Et, R614: H, R 615: H, R 616: OMe], [BC 1 955; E 602, R 612: OMe, R 614: Et, R 615: H, R 616: H], [BC 1956; E 602, R 612: H, R 614: Et, R 615: OMe, R616: H], [BC1957; E602, R612: H, R614: Et, R615: H, R616: OMe], [BC1958; E602, R612: OMe, R614: H, R615: Et, R616: H], [ BC1959; E602, R612: H, R614: OMe, R615: Et, R616: H], [BC1960; E602, R612: H, R614: H, R615: Et, R616: OMe], [BC1961; E602, R612: OMe, R614: H, R615: H, R616: Et], [BC1962; E602, R612: H, R614: OMe, R615: H, R616: Et], [BC1963; E602, R612: H, R614: H, R615: OMe, R616: Et], [BC1964, E602, R612: H, R614: H, R616: H], [BC1965; E602, R612: H, R614: F, R615: H, R616: H], [BC 1966; E 602, R 612: H, R 614: H, R 615: F, R 616: H], [BC 1967; E 602, R 612: H, R 614: H, R 615: H, R 616: F], [BC1968; E602, R612: F, R614: F, R615: H, R616: H], [BC1969; E602, R612: F, R614: H, R615: F, R616: H], [BC1970; E602, R612: F, R614: H, R615: H, R616: F], [BC1971; E602, R612: H, R614: F, R615: F, R616: H], [BC 1972; E602, R612: H, R 614: F, R 615: H, R 616: F], [BC 1973; E 602, R 612: H, R 614: H, R 615: F, R 616: F], [BC 1974; E 602, R 612: F, R 614: F, R 615: F, R 616: H], [BC 1975; E 602, R 612: F, R 614: H, R 615: F, R 616: F], [BC 1976; E 602, R 612: F, R 614: F, R 615: H, R 616: F] [BC1977; E602, R612: Cl, R614: H, R615: H, R616: H], [BC1978; E602, R612: H, R614: Cl, R615: H, R616: H], [BC 1979; E602, R612: H, R614: H, R615: Cl, R616: H], [BC1980; E602, R612: H, R614: H, R615: H, R616: Cl], [BC1981; E602, R612: Cl, R614: Cl, R 615: H, R 616: H], [BC 1982; E 602, R 612: Cl, R 614: H, R 615: Cl, R 616: H], [BC 1983; E 602, R 612: Cl, R 614: H, R 615: H, R616: Cl], [BC 1984; E 602, R 612: H, R 614: Cl, R 615: Cl, R 616: H], [BC 1985; E 602, R 612: H, R 614: Cl, R 615: H, R 616: Cl], [ BC1986; E602, R612: H, R614: H, R615: Cl, R616: Cl], [BC1987; E602, R612: Cl, R614: H, R615: Cl, R616: Cl], [BC1988; E602, R612: Cl, R614: Cl, R615: H, R616: Cl], [BC1989; E602, R612: Cl, R614: Cl, R615: Cl, R616: H], [BC1990; E602, R612: F, R614: Cl, R 615: H, R 616: H], [BC 19 91; E602, R612: F, R614: H, R615: Cl, R616: H], [BC 1992; E602, R612: F, R614: H, R615: H, R616: Cl], [BC1993; E602, R612: Cl, R 614: F, R 615: H, R 616: H], [BC 1994; E 602, R 612: H, R 614: F, R 615: Cl, R 616: H], [BC 1995; E 602, R 612: H, R 614: F, R615: H, R616: Cl], [BC1996; E602, R612: H, R614: F, R615: F, R616: H], [BC1997; E602, R612: H, R614: Cl, R615: F, R616: H], [BC1998; E602, R612: H, R614: H, R615: F, R616: Cl], [BC1999; E602, R612: Cl, R614: H, R615: H, R616: F], [BC2000; E602, R612: H, R614: Cl, R615: H, R616: F],

[BC2001; E602, R612: H, R614: H, R615: Cl, R616: F], [BC2002; E602, R612: Pr, R614: H, R615: H, R616: H], [BC2003; E602, R612 : H, R 614: Pr, R 615: H, R 616: H], [BC 2004; E 602, R 612: H, R 614: H, R 615: Pr, R 616: H], [BC 2005; E 602, R 612: H, R 614: H , R 615: H, R 616: Pr], [BC 2006; E 602, R 612: isopropyl, R 614: H, R 615: H, R 616: H], [BC 2007; E 602, R 612: H, R 614: isopropyl, R 615: H, R 616 : H], [BC2008; E602, R612: H, R614: isopropyl, R616: H], [BC2009; E602, R612: H, R614: H, R615: H, R616: isopropyl], [BC2010] E602, R612: c-Pr, R614: H, R615: H, R616: H], [BC2011; E602, R612: H, R614: c-Pr, R615: H, R616: H], [BC2012; E602 , R 612: H, R 614: H, R 615: c-Pr, R 616: H], [BC 2013; E 602, R 612: H, R 614: H, R 615: H, R 616: c-Pr], [BC 2014; E 602, R 612 : c-Pr, R 614: F, R 615: H, R 616: H], [BC2015; E 602, R 612: c-Pr, R 614: H, R 615: F, R 616: H], [BC 2016; E 602, R 612: c -Pr, R 614: H, R 615: H, R 616: F], [BC 2017; E 602, R 612: F, R 614: c-Pr, R 615: H, R 616: H], [BC 2018; E 602, R 612: H, R 614 : c-Pr, R 615: F, R 616: H], [BC 2019; E 602, R 612: H, R 614: c-Pr, R 615: H, R 616: F], [BC 2020; E 602, R 612: F, R 614: H , R615: c-Pr, R616: H], [BC2021; E602, R612: H, R614: F, R615: c-Pr, R616: H], [BC2022; E602, R612: H, R614: H, R615 : c-Pr, R 616: F], [BC2023; E602, R612: F, R614: H, R615: H, R616: c-Pr], [BC2024; E602, R612: H, R614: F, R615: H, R616: c-Pr], [BC2025 E602, R612: H, R614: H, R615: F, R616: c-Pr], [BC2026; E602, R612: c-Pr, R614: Cl, R615: H, R616: H], [BC2027; , R612: c-Pr, R614: H, R615: Cl, R616: H], [BC2028; E602, R612: c-Pr, R614: H, R615: H, R616: Cl], [BC2029; E602, R612 : Cl, R614: c-Pr, R615: H, R616: H], [BC2030; E602, R612: H, R614: c-Pr, R615: Cl, R616: H], [BC2031; E602, R612: H , R 614: c-Pr, R 615: H, R 616: Cl], [BC 2032; E602, R 612: Cl, R 614: H, R 615: c-Pr, R 616: H], [BC 2033; E 602, R 612: H, R 614 : Cl, R615: c-Pr, R616: H], [BC2034; E602, R612: H, R614: H, R615: c-Pr, R616: Cl], [BC2035; E602, R612: Cl, R614: H , R615: H, R616: c-Pr], [BC2036; E602, R612: H, R614: Cl, R615: H, R616: c-Pr], [BC2037; E602, R612: H, R614: H, R615 : Cl, R 616: c-Pr], [BC2038; E602, R612: H, R615: H, R615: H], [BC2039; E602, R612: H, R614: H, R615: H, R616 : OMe], [BC2040; E602, R612: H, R614: H, R616: H], [BC2041; E602, R612: OMe, R614: H, R615: H, R616: H], [BC2042 E602, R612: H, R614: OMe, R615: H, R616: H], [BC2043; E602, R612: H, R614: H, R615: OMe, R616: H], [BC 2044; E602, R612: H , R 614: H, R 615: H, R 616: OMe], [BC 20 45; E602, R612: OMe, R614: F, R615: H, R616: H], [BC2046; E602, R612: OMe, R614: H, R615: F, R616: H], [BC2047; E602, R612: OMe, R614: H, R615: H, R616: F], [BC2048; E602, R612: F, R614: OMe, R615: H, R616: H], [BC2049; E602, R612: H, R614: OMe, R615: F, R616: H], [BC2050; E602, R612: H, R614: OMe, R615: H, R616: F], [BC2051; E602, R612: F, R614: H, R615: OMe, R616: H], [BC2052; E602, R612: H, R614: F, R615: OMe, R616: H], [BC2053; E602, R612: H, R614: H, R615: OMe, R616: F], [BC2054; E602, R612: F, R614: H, R615: H, R616: OMe], [BC2055; E602, R612: H, R614: F, R615: H, R616: OMe], [BC2056; E602, R612: H, R614: H, R615: F, R616: OMe], [BC2057; E602, R612: OMe, R614: Cl, R615: H, R616: H], [BC2058; E602, R612: OMe, R614: H, R615: Cl, R616: H], [BC2059; E602, R612: H, R615: H, R615: H, R616: Cl], [BC2060; E602, R612: Cl, R614: OMe, R615: H, R616: H] , [BC2061; E602, R612: H, R614: Cl, R615: H], [BC2062; E602, R612: H, R614: OMe, R615: H, R616: Cl], [BC2063; E602, R612: Cl, R 614: H, R 615: OMe, R 616: H], [BC 2064; E 602, R 612: H, R 614: Cl, R 615: OMe, R 616: H], [BC 2065; E 602, R 612: H, R 614: H, R615: OMe, R616: Cl], [BC2066; E602, R612: Cl, R614: H, R615: H, R616: OMe], [BC2067; E602, R612: H, R614: Cl , R615: H, R616: OMe], [BC2068; E602, R612: H, R614: H, R615: Cl, R616: OMe], [BC2069; E602, R612: CN, R614: H, R615: H, R616] : H], [BC2070; E602, R612: H, R614: CN, R615: H, R616: H], [BC2071; E602, R612: H, R614: H, R615: CN, R616: H], [BC2072 E602, R612: H, R614: H, R615: H, R616: CN], [BC2073; E602, R612: CN, R614: F, R615: H, R616: H], [BC2074; E602, R612: CN , R 614: H, R 615: F, R 616: H], [BC 2075; E 602, R 612: CN, R 614: H, R 615: H, R 616: F], [BC 2076; E 602, R 612: F, R 614: CN, R 615 : H, R 616: H], [BC 2077; E 602, R 612: H, R 614: CN, R 615: F, R 616: H], [BC 2078; E 602, R 612: H, R 614: CN, R 615: H, R 616: F ], [BC2079; E602, R612: F, R614: H, R615: CN, R616: H], [BC2080; E602, R612: H, R614: F, R615: CN, R616: H], [BC2081; E602] , R612: H, R614: H, R615: CN, R616: F], [BC2082; E602, R612: F, R614: H, R615: H, R616: CN], [BC 2083; E602, R612: H, R614] : F, R 615: H, R 616: CN], [BC 2084; E 602, R 612: H, R 614: H, R 615: F, R 616: CN], [BC 2085; E 602, R 612: CN, R 614: Cl, R 615: H , R616: H], [BC 2086; E 602, R 612: CN, R 614: H, R 615: Cl, R 616: H], [BC 2087; E 602, R 612: CN, R 614: H, R 615: H, R 616: Cl], [BC 2088; E 602, R 612: Cl, R 614: CN, R 615: H, R 616: H], [BC 2089; E 602, R 612: H, R 614: CN, R 615: Cl, R 616: H], [BC 2090; E 602, R 612 : H, R 614: CN, R 615: H, R616: Cl], [BC2091; E602, R612: H, R614: CN, R616: H], [BC2092; E602, R612: H, R614: Cl, R615: CN, R616: H], [BC 2093; E 602, R 612: H, R 614: CN, R 615: CN, R 616: Cl], [BC 2094; E 602, R 612: Cl, R 614: H, R 615: H, R 616: CN], [BC 20 95; E602, R612: H, R614: Cl, R615: H, R616: CN], [BC2096; E602, R612: H, R614: H, R615: Cl, R616: CN], [BC2097; E602, R612: NH 2 , R 614: H, R 615: H, R 616: H], [BC 2098; E 602, R 612: H, R 614: NH ₂ , R 615: H, R 616: H], [BC 20 99; E 602, R 612: H, R 614: H, _{R615: NH 2, R616: H} ], [BC2100; E602, R612: H, R614: H, R615: H, R616: NH 2],

[BC2101; E602, R612: NH 2, R614: F, R615: H, R616: H], [BC2102; E602, R612: NH 2, R614: H, R615: F, R616: H], [BC2103; E602 _{, R612: NH 2, R614:} H, R615: H, R616: F], [BC2104; E602, R612: F, R614: NH 2, R615: H, R616: H], [BC2105; E602, R612: H _{, R614: NH 2, R615:} F, R616: H], [BC2106; E602, R612: H, R614: NH 2, R615: H, R616: F], [BC2107; E602, R612: F, R614: H _{, R615: NH 2, R616:} H], [BC2108; E602, R612: H, R614: F, R615: NH 2, R616: H], [BC2109; E602, R612: H, R614: H, R615: NH ₂ , R 616: F], [BC ₂ 110; E 602, R 612: F, R 614: H, R 615: H, R 616: NH ₂ ], [BC ₂ 111; E 602, R 612: H, R 614: F, R 615: H, R 616: NH _{2], [BC2112; E602,} R612: H, R614: H, R615: F, R616: NH 2], [BC2113; E602, R612: NH 2, R614: Cl, R615: H, R616: H], [ _{BC2114; E602, R612: NH 2} , R614: H, R615: Cl, R616: H], [BC2115; E602, R612: NH 2, R614: H, R615: H, R616: Cl], [BC2116; E602, _{R612: Cl, R614: NH 2} , R615: H, R616: H], [BC2117; E602, R612: H, R614: NH 2, R615: Cl, R616: H], [BC2118; E602, R612: H, _{R614: NH 2, R615: H} , R616: Cl], [BC2119; E602, R612: Cl, R614: H, R615: NH 2, R616: H], [BC2120; E602, R612: H, R614: Cl, _{R615: NH 2, R616: H} ], [BC2121; E602, R612: H, R614: H, R615: NH 2, R616: Cl], [BC2122; E602, R612: Cl, R614 : H, R615: H, R616 : NH 2], [BC2123; E602, R612: H, R614: Cl, R615: H, R616: NH 2], [BC2124; E602, R612: H, R614: H, R615 : Cl, R 616: NH ₂ ], [BC ₂ 125; E 602, R 612: NH Me, R 614: H, R 615: H, R 616: H], [BC 2 126; E 602, R 612: H, R 614: NH Me, R 615: H, R 616: H], [BC2127; E602, R612: H, R614: H, R615: NHMe, R616: H], [BC2128; E602, R612: H, R614: H, R615: H, R616: NHMe], [BC2129; E602, R612: NHMe, R614: F, R615: H, R616: H], [BC2130; E602, R612: NHMe, R614: H, R615: F, R616: H], [BC2131; E602, R612: NHMe, R614: H, R615: H, R616: F], [BC2132; E602, R612: F, R614: NHMe, R615: H, R616: H], [BC2133; E602, R612: H, R614: NHMe, R615: F, R 616: H], [BC 2 134; E 602, R 612: H, R 614: NH Me, R 615: H, R 616: F], [BC 2 135; E 602, R 612: F, R 614: H, R 615: NH Me, R 616: H] , [BC2136; E602, R612: H, R614: F, R615: NHMe, R616: H], [BC2137; E602, R612: H, R614: H, R615: NHMe, R616: F], [BC2138; R612: F, R614: H, R615: H, R616: NHMe], [BC2139; E602, R612: H, R614: F, R 615: H, R616: NHMe], [BC2140; E602, R612: H, R614: H, R 615: F, R 616: NHMe], [BC 2141; E 602, R 612: NH Me, R 614: Cl, R 615: H, R 616: H], [BC 2142; E 602, R 612: NH Me, R 614: H, R 615: Cl, R616: H], [BC2143; E602, R612: NHMe, R614: H, R615: H, R616: Cl], [BC2144; E602, R612: Cl, R614: NHMe, R615: H, R616: H], [BC2145; E602, R612: H, R614: NHMe, R615: Cl, R616: H], [BC2146; E602, R612: H, R614: NHMe, R615: H, R616: Cl], [BC2147; E602, R612: H, R614: NHMe, R616: H], [BC2148; E602, R612: H, R614: Cl, R615: NHMe, R616: H], [ BC2149; E602, R612: H, R614: H, R615: NHMe, R616: Cl], [BC2150; E602, R612: Cl, R614: H, R615: H, R616: NHMe], [BC2151; E602, R612: H, R 614: Cl, R 615: H, R 616: NHMe], [BC 2 152; E 602, R 612: H, R 614: H, R 615: Cl, R 616: NH Me], [BC ₂ 153; E 602, R 612: N Me ₂ , R 614: H , R 615: H, R 616: H], [BC 2 154; E 602, R 612: H, R 614: N Me ₂ , R 615: H, R 616: H], [BC 2 155; E 602, R 612: H, R 614: H, R 615: N Me2, R 616: H], [BC 2156; E 602, R 612: H, R 614: H, R 615: H, R 616: N Me ₂ ], [BC ₂ 157; E 602, R 612: N Me ₂ , R 614: F, R 615: H, R 616: H] , [BC2158; E602, R612: NMe 2, R614: H, R615: F, R616: H], [BC2159; E602, R612: NMe 2, R614: H, R615: H, R616: F], [BC2160; E602, R612: F, R614: NMe 2, R615: H, R616: H], [BC2161; E602, R612: H, R614: NMe 2, R615: F, R616: H], [BC2162; E602, R612: _{H, R614: NMe 2, R615} : H, R616: F], [BC2163; E602, R612: F, R614: H, R615: NMe 2, R616: H], [BC2164; E602, R612: H, R614: _{F, R615: NMe 2, R616} : H], [BC2165; E602, R612: H, R614: H, R615: NMe 2, R616: F], [BC 2166; E602, R612: F, R614: H, R615: H, R616: NMe 2], [BC2167; E602, R612: H, R614: F, R615: H, R616: NMe 2], [BC2168; E602, R612: H, R614: H, R615: F, R616: NMe 2], [BC2169; E602, R612: NMe 2, R614: Cl, R615: H, R616: H], [BC2170; E602, R612: NMe 2 , R614: H, R615: Cl , R616: H], [BC2171; E602, R612: NMe 2, R614: H, R615: H, R616: Cl], [BC2172; E602, R612: Cl, R614: NMe 2 , R 615: H, R 616: H], [BC 2 173; E 602, R 612: H, R 614: N Me ₂ , R 615: Cl, R 616: H], [BC 2 174; E 602, R 612: H, R 614: N Me ₂ , R 615: H , R616: Cl], [BC2175 ; E602, R612: Cl, R614: H, R615: NMe 2, R616: H], [BC2176; E602, R612: H, R614: Cl, R615: NMe 2, R616: H ], [BC2177; E602, R612 : H, R614: H, R615: NMe 2, R616: Cl], [BC2178; E602, R612: Cl, R614: H, R615: H, R616: NMe 2], [BC2179 ; E602, R612: H, R614 : Cl, R615: H, R616: NMe 2], [BC2180; E602, R612: H, R614: H, R615: Cl, R616: NMe 2], [BC2181; E602, R612 : SMe, R 614: H, R 615: H, R 616: H], [BC 2182; E 602, R 612: H, R 614: S Me, R 615: H, R 616: H], [BC 2 183; E 602, R 612: H, R 614: H , R615: SMe, R616: H], [BC2184; E602, R612: H, R614: H, R615: H, R616: SMe], [BC2185; E602, R612: SMe, R614: F, R615: H, R616] : H], [BC2186; E602, R612: SMe, R614: H, R615: F, R 616: H], [BC2187; E602, R612: SMe, R614: H, R615: H, R616: F], [BC2188; E602, R612: F, R614: SMe, R615: H, R616: H], [BC2189; E602, R612: H, R614: SMe, R615: F, R 616: H], [BC 2 190; E 602, R 612: H, R 614: S Me, R 615: H, R 616: F], [BC 2 191; E 602, R 612: F, R 614: H, R 615: S Me, R 616: H] , [BC2192; E602, R612: H, R614: F, R615: SMe, R616: H], [BC2193; E602, R612: H, R614: H, R615: SMe, R616: F], [BC2194; E602, R612: F, R614: H, R615: H, R616: SMe], [BC2195; E602, R612: H, R614: F, R 615: H, R616: SMe], [BC2196; E602, R612: H, R614: H, R615: F, R616: SMe], [BC2197; E602, R612: SMe, R614: Cl, R615: H, R616: H], [BC2198; E602, R612: SMe, R614: H, R615: Cl, R616: H], [BC2199; E602, R612: SMe, R614: H, R615: H, R616: Cl], [BC2 200; E602, R612: Cl, R614: SMe, R615: H, R616: H],

[BC2201; E602, R612: H, R614: SMe, R615: Cl, R616: H], [BC2202; E602, R612: H, R614: SMe, R615: H, R616: Cl], [BC2203; E602, R612 : Cl, R 614: H, R 615: SMe, R 616: H], [BC 2 204; E 602, R 612: H, R 614: Cl, R 615: S Me, R 616: H], [BC 2 205; E 602, R 612: H, R 614: H , R615: SMe, R616: Cl], [BC2206; E602, R612: H, R614: H, R615: H, R616: SMe], [BC2207; E602, R612: H, R614: Cl, R615: H, R616 : SMe], [BC2208; E602 , R612: H, R614: H, R615: Cl, R616: SMe], [BC2209; E602, R612: NO 2, R614: H, R615: H, R616: H], [ BC2210; E602, R612: H, R614: NO 2, R615: H, R616: H], [BC2211; E602, R612: H, R614: H, R615: NO 2, R616: H], [BC2212; E602, R612: H, R614: H, R615: H, R616: NO 2], [BC2213; E602, R612: NO 2, R614: F, R615: H, R616: H], [BC2214; E602, R612: NO 2 , R614: H, R615: F , R616: H], [BC2215; E602, R612: NO 2, R614: H, R615: H, R616: F], [BC2216; E602, R612: F, R614: NO 2 , R615: H, R616: H ], [BC2217; E602, R612: H, R614: NO 2, R615: F, R616: H], [BC2218; E602, R612: H, R614: NO 2, R615: H , R616: F], [BC2219 ; E602, R612: F, R614: H, R615: NO 2, R616: H], [BC2220; E602, R612: H, R614: F, R615: NO 2, R616: H ], [BC2221; E602, R612 : H, R614: H, R615: NO 2, R616: F], [BC2222; E602, R612: F, R614: H, R615: H, R616: NO _{2], [BC2223; E602,} R612: H, R614: F, R615: H, R616: NO 2], [BC2224; E602, R612: H, R614: H, R615: F, R616: NO 2], [ _{BC2225; E602, R612: NO 2} , R614: Cl, R615: H, R616: H], [BC2226; E602, R612: NO 2, R614: H, R615: Cl, R616: H], [BC2227; E602, _{R612: NO 2, R614: H} , R615: H, R616: Cl], [BC2228; E602, R612: Cl, R614: NO 2, R615: H, R616: H], [BC2229; E602, R612: H, _{R614: NO 2, R615: Cl} , R616: H], [BC2230; E602, R612: H, R614: NO 2, R615: H, R616: Cl], [BC2231; E602, R612: Cl, R614: H, _{R615: NO 2, R616: H} ], [BC2232; E602, R612: H, R614: Cl, R615: NO 2, R616: H], [BC2233; E602, R612: H, R614: H, R615: NO 2 , R 616: Cl], [BC 2 234; E 602, R 612: H, R 614: H, R 615: H, R 616: NO ₂ ], [BC ₂ 235; E 602, R 612: H, R 614: Cl, R 615: H, R 616: NO ₂ ], [BC2236; E602, R612 : H, R614: H, R615: Cl, R616: NO 2], [BC2237; E604, R613: Me, R614: H, R615: H], [BC2238; E604, R613: H, R614: Me, R615: H], [BC2239; E604, R613: Me, R614: Me, R615: H], [BC2240; E604, R613: Me, R614: H, R615: Me], [BC2241; E604, R613: Me, R614: Me, R615: Me], [BC2242; E604, R613: Me, R614: F, R615: H], [BC2243; E604, R613: Me, R614: H, R615: F] [BC2244; E604, R613: F, R614: Me, R615: H], [BC2245; E604, R613: Me, R614: F, R615: F], [BC2246; , R613: F, R 614: Me, R 615: F], [BC 2247; E 604, R 613: Me, R 614: Me, R 615: F], [BC 2 248; E 604, R 613: Me, R 614: F, R 615: Me], [BC2249; E604, R613: Me, R614: Cl, R615: H], [BC2250; E604, R613: Me, R614: H, R615: Cl], [BC2251; E604, R613: Cl, R614: Me, R615 : H], [BC 2252; E 604, R 613: Me, R 614: Cl, R 615: Cl], [BC 2 253; E 604, R 613: Cl, R 614: Me, R 615: Cl], [BC 2 254; E 604, R 613: Me, R 614 : Me, R615: Cl], [BC2255; E604, R613: Me, R614: Cl, R615: Me], [BC2256; E604, R613: Me, R614: Br, R615: H], [BC2257; E604, R613 : Me, R 614: H, R 615: Br], [BC 2258; E 604, R 613: Br, R 614: Me, R 615: H], [BC 2 259; E 604, R 613: Me, R 614: Br, R 615: Br], [BC 2 260 E604, R 613: Br, R 614: Me, R 615: Br], [BC 2261; E 604, R 613: Me, R 614: Me, R 615: Br], [BC 2262; E 604, R 613: Me, R 614: Br, R 615: Me ], [BC 2263; E 604, R 613: F, R 614: H, R 615: H], [BC 2 264; E 604, R 613: H, R 614: F, R 615: H], [BC 2 265; E 604, R 613: F, R 614: F , R615: H], [BC2266; E604, R613: H, R614: F], [BC2267; E604, R613: F, R614: F, R615: F], [BC2268; E604, R613: F] , R 614: Cl, R 615: H], [BC 2269; E 604, R 613: F, R 614: H, R 615: Cl], [BC 2 270; E 604, R 613: Cl, R 614: F, R 615: H], [BC 227 1; , R 613: F, R 614: Cl, R 615: Cl], [BC 2272; E 604, R 613: Cl, R 614: F, R 615: Cl], [BC 2 273; E 604, R 613: F , R614: F, R615: Cl], [BC2274; E604, R613: F, R614: Cl, R615: F], [BC2275; E604, R613: Et, R614: H, R615: H], [BC2276; , R 613: H, R 614: Et, R 615: H], [BC 2277; E 604, R 613: Et, R 614: Et, R 615: H], [BC 2 278; E 604, R 613: Et, R 614: H, R 615: Et], [BC2279; E604, R613: Et, R614: Et, R615: Et], [BC2280; E604, R613: Et, R614: F, R615: H], [BC2281; E604, R613: Et, R614: H, R615 : F], [BC2282; E604, R613: F, R614: Et, R615: H], [BC2283; E604, R613: Et, R614: F, R615: F], [BC2284; E604, R613: F, R614] : Et, R 615: F], [BC 2285; E 604, R 613: Et, R 614: Et, R 615: F], [BC 2286; E 604, R 613: Et, R 614: F, R 615: Et], [BC 2287; : Et, R 614: Cl, R 615: H], [BC 2 288; E 604, R 613: Et, R 614: H, R 615: Cl], [BC 2 289; E 604, R 613: Cl, R 614: Et, R 615: H], [BC 2 290 E604, R613: Et, R614: Cl, R615: Cl], [BC2291; E604, R613: Cl, R614: Et, R615: Cl], [BC2292; E604, R613: Et, R614: Et, R615: Cl ], [BC2293; E604, R613: Et, R614: Cl, R615: Et], [BC2294; E604, R613: OMe, R614: H, R615: H], [BC2295; E604, R613: H, R614: OMe] , R615: H], [BC2296; E604, R613: OMe, R615: H], [BC2297; E604, R613: OMe, R614: H, R615: OMe], [BC2298; E604, R613: OMe] , R 614: F, R 615: H], [BC 2 299; E 604, R 613: OMe, R 614: H, R 615: F], [BC 2 300; E 604, R 613: F, R 614: OMe, R 615: H],

[BC2301; E604, R613: OMe, R614: F, R615: F], [BC2302; E604, R613: F, R614: OMe, R615: F], [BC2303; E604, R613: OMe, R614: OMe, R615 : F], [BC 2304; E 604, R 613: OMe, R 614: F, R 615: OMe], [BC 2 305; E 604, R 613: OMe, R 614: Cl, R 615: H], [BC 2 306; : H, R615: Cl], [BC2307; E604, R613: Cl, R614: OMe, R615: H], [BC2308; E604, R613: OMe, R614: Cl, R615: Cl], [BC2309; E604, R613 : Cl, R614: OMe, R615: Cl], [BC2310; E604, R613: OMe, R614: OMe, R615: Cl], [BC2311; E604, R613: OMe, R614: Cl, R615: OMe], [BC2312] E604, R613: Pr, R614: H, R615: H], [BC2313; E604, R613: H, R614: Pr, R615: H], [BC2314; E604, R613: Pr, R614: H, R615: F ], [BC2315; E604, R613: F, R614: Pr, R615: H], [BC2316; E604, R613: Pr, R614: F, R615: F], [BC2317; E604, R613: F, R614: Pr] , R615: F], [BC2318; E604, R613: Pr, R614: Cl, R615: H], [BC2319; E604, R613: Pr, R614: H, R615: Cl], [BC2320; E604, R613: Cl , R614: Pr, R615: H], [BC2321; E604, R613: Pr, R614: Cl, R615: Cl], [BC2322; E604, R613: Cl, R614: Pr, R615: Cl], [BC2323; , R613: SMe, R614: H, R615: H], [BC2324; E604, R613: H, R614: SMe, R615: H], [BC2325; E604, R613: SMe, R614: H, R615: F], [BC2326; E604, R613: F, R614: SMe, R615: H], [BC2327; E604, R613: SMe, R61 4: F, R 615: F], [BC 2 328; E 604, R 613: F, R 614: S Me, R 615: F], [BC 2 329; E 604, R 613: S Me, R 614: Cl, R 615: H], [BC 2 330; R613: SMe, R614: H, R615: Cl], [BC2331; E604, R613: Cl, R614: SMe, R615: H], [BC2332; E604, R613: SMe, R614: Cl, R615: Cl], [ BC2333; E604, R613: Cl, R614: SMe, R615: Cl], [BC2334; E604, R613: CF 3, R614: H, R615: H], [BC2335; E604, R613: H, R614: CF 3, R615: H], [BC2336; E604, R613: CF 3, R614: H, R615: F], [BC2337; E604, R613: F, R614: CF 3, R615: H], [BC2338; E604, R613: CF ₃ , R 614: F, R 615: F], [BC 2339; E 604, R 613: F, R 614: CF ₃ , R 615: F], [BC 2 340; E 604, R 613: CF ₃ , R 614: Cl, R 615: H], [BC2341; E604, R613: CF 3, R614: H, R615: Cl], [BC2342; E604, R613: Cl, R614: CF 3, R615: H], [BC2343; E604, R613: CF 3, R614: Cl, R615: Cl], [BC2344; E604, R613: H, R614: H, R615: H], [BC2 345; E601, R613: n-Bu, R614: H, R615: H, R616: H], [ BC2346; E601, R613: H, R614: cyclobutyl, R615: H, R616: H], [BC2347; E601, R613: H, R614: H, R615: Ph, R616: H], [BC 2348; E601, R613: H, R 614: H, R 615: H, R 616: OPh], [BC 2349; E 601, R 613: c-Proxy, R 614: H, R 615: H, R 616: H], [BC 2 350; E 601, R 613: H, R 614: CF 2 H, R 615: H, R 616: H], [BC 2351; E 601, R 613: H, R 614: H, R 615: SO Me, R 616: H], [BC 2352; E601, R613: SO2 Me, R 614: H, R 615: H, R 616: H], [BC 2 353; E 601, R 613: H, R 614: SO 2 Et, R 615: H, R 616: H], [BC 2 354; R614: H, R615: Bn, R616: Me], [BC2355; E601, R613: Bn, R614: Me, R615: H, R616: H], [BC2356; E602, R612: CHO, R614: H, R615: H, R 616: H], [BC 2 357; E 602, R 612: H, R 614: CHO, R 615: H, R 616: H], [BC 2 358; E 602, R 612: H, R 614: H, R 615: acetyl, R 616: H] , [BC2359; E602, R612: H, R614: H, R615: H, R616: SPh], [BC2 360; E602, R612: SH, R614: Me, R615: H, R616: H], [BC 2361; R612: H, R613: H, R615: H, R616: H], [BC2362; E603, R612: Me, R613: H, R615: H, R616: H], [BC2363; E603, R612: H, R613: Me, R615: H, R616: H], [BC2364; E603, R612: H, R613: H, R615: Me, R616: H], [BC2365; E603, R612: H, R613: H, R615: H, R616: Me], [BC2366; E603, R612: Me, R613: Me, R615: H, R616: H], [BC2367; E603, R612: Me, R613: H, R615: Me, R616: H], [ BC2368; E603, R612: Me, R613: H, R615: H, R616: Me], [BC2369; E603, R612: H, R613: Me, R615: Me, R616: H], [BC2370; E603, R612: H, R613: Me, R615: H, R616: Me], [BC2371; E603, R612: H, R613: H, R615: Me, R616: Me], [BC2372; E603, R612: H, R613: Me, R615: H, R616: H], [BC2373; E603, R612: Me, R613: Me, R615: Me, R616: H], [BC2 374; E603, R612: Me, R613: Me, R615: H, R61 6: Me], [BC2375; E603, R612: Me, R613: H, R615: Me, R616: Me], [BC2376; E603, R612: H, R613: Me, R615: Me, R616: Me], [ BC2377; E603, R612: Me, R613: Me, R615: Me, R616: Me], [BC2378; E603, R612: Me, R613: F, R615: H, R616: H], [BC2379; E603, R612: Me, R 613: H, R 615: F, R 616: H], [BC 2 380; E 603, R 612: Me, R 613: H, R 615: H, R 616: F], [BC 2 381; E 603, R 612: Me, R 613: F, R615: F, R616: H], [BC2382; E603, R612: Me, R613: F, R615: H, R616: F], [BC2383; E603, R612: Me, R613: H, R615: F, R616: F], [BC2384; E603, R612: Me, R613: F, R615: F, R616: F], [BC2385; E603, R612: F, R613: Me, R615: H, R616: H], [BC2386; E603, R612: H, R613: Me, R615: F, R616: H], [BC2387; E603, R612: H, R613: Me, R615: H, R616: F], [BC2388; E603, R612: F, R613: Me, R615: F, R616: H], [BC2389; E603, R612: F, R613: Me, R615: H, R616: F], [BC2390; E603, R612: H, R613: Me, R615: F, R616: F], [BC2391; E603, R612: Me, R613: F, R616: F], [BC2392; E603, R612: F, R613: H, R615: Me, R616: H] [BC2393; E603, R612: H, R613: F, R615: Me, R616: H], [BC2394; E603, R612: H, R613: H, R615: Me, R616: F], [BC2395; E603, E603, R612: F, R613: F, R615: Me, R616: H], [BC2396; E603, R612: F, R613: H, R615: Me, R616: F], [BC2397; E603, R612: H, R613: F, R 615: Me, R 616: F ], [BC2398; E603, R612: F, R613: F, R615: Me, R616: F], [BC2399; E603, R612: F, R613: H, R615: H, R616: Me], [BC2400; , R 612: H, R 613: F, R 615: H, R 616: Me],

[BC2401; E603, R612: H, R613: H, R615: F, R616: Me], [BC2402; E603, R612: F, R613: F, R615: H, R616: Me], [BC2403; E603, R612 : F, R 613: H, R 615: F, R 616: Me], [BC 2404; E 603, R 612: H, R 613: F, R 615: F, R 616: Me], [BC 2 405; E 603, R 612: F, R 613: F , R615: F, R616: Me], [BC2406; E603, R612: Me, R613: Me, R615: F, R616: H], [BC2407; E603, R612: Me, R613: Me, R615: H, R616 : F], [BC2408; E603, R612: Me, R613: F, R615: Me, R616: H], [BC2409; E603, R612: Me, R613: H, R615: Me, R616: F], [BC2410 E603, R612: Me, R613: F, R615: H, R616: Me], [BC2411; E603, R612: Me, R613: H, R615: F, R616: Me], [BC 2412; E603, R612: Me , R613: Me, R615: Cl, R616: H], [BC2413; E603, R612: Me, R613: Me, R615: H, R616: Cl], [BC2414; E603, R612: Me, R613: Cl, R615 : Me, R 616: H], [BC 2415; E 603, R 612: Me, R 613: H, R 615: Me, R 616: Cl], [BC 2416; E 603, R 612: Me, R 613: Cl, R 615: H, R 616: Me ], [BC2417; E603, R612: Me, R613: H, R615: Cl, R616: Me], [BC2418; E603, R612: Me, R613: Cl, R615: H, R616: H], [BC2419; , R612: Me, R613: H, R615: Cl, R616: H], [BC2420; E603, R612: Me, R613: H, R615: H, R616: Cl], [BC2421; E603, R612: Me, R613 : Cl, R615: Cl, R616: H], [BC2422; E603, R612: Me, R613: Cl, R615: H, R616: Cl], [BC2423; E603, R612: Me, R613: H, R 615: Cl, R 616: Cl], [BC 2424; E 603, R 612: Me, R 615: H, R 616: H], [BC 24 25; E 603, R 612: H, R 613: Me, R 615: Cl, R 616: H], [BC2426; E603, R612: H, R613: Me, R615: H, R616: Cl], [BC2427; E603, R612: Cl, R613: Me, R615: Cl, R616: H], [BC2428; E603, R612: Cl, R613: Me, R615: H, R616: Cl], [BC2429; E603, R612: H, R613: Me, R615: Cl, R616: Cl], [BC2430; E603, R612: Cl, R613: H, R 615: Me, R 616: H], [BC 2431; E 603, R 612: H, R 613: Cl, R 615: Me, R 616: H], [BC 2432; E 603, R 612: H, R 613: H, R 615: Me, R616: Cl], [BC2433; E603, R612: Cl, R613: Cl, R615: Me, R616: H], [BC2434; E603, R612: Cl, R613: H, R615: Me, R616: Cl] [BC2435; E603, R612: H, R613: Cl, R615: Me, R616: Cl], [BC2436; E603, R612: Bn, R613: H, R615: H, R616: H], [BC2437; R612: Bn, R613: Me, R615: H, R616: H], [BC2438; E603, R612: n-Bu, R613: H, R615: H, R616: H], [BC2439; E603, R612: H, R613: cyclobutyl, R615: H, R616: H], [BC2440; E603, R612: H, R613: H, R615: Ph, R616: H], [BC2441; E603, R612: H, R613: H, R615: H, R616: OPh], [BC2442; E603, R612: c-Proxy, R613: H, R615: H, R616: H], [BC2443; E603, R612: H, R613: CF2H, R615: H, R616: H], [BC2444; E603, R612: H, R613: H, R615: SOMe, R616: H], [BC2445; E603, R612: SO2Me, R613: H, R615: H, R616] : H], [BC2446; E603, R612: H, R613: SO2Et, R615: H, R616: H], [BC2447; E603, R612: H, R613: H, R615: Bn, R616: Me], [BC2448 E605, R613: H, R615: H, R616: H], [BC2449; E605, R613: Me, R615: H, R616: H], [BC2450; E605, R613: H, R615: Me, R616: H ], [BC2451; E605, R613: H, R615: H, R616: Me], [BC2452; E605, R613: Me, R615: Me, R616: H], [BC2453; E605, R613: Me, R615: H] , R616: Me], [BC2454; E605, R613: Me, R615: Me, R616: Me], [BC2455; E605, R613: Me, R615: F, R616: H], [BC2456; E605, R613: Me , R615: H, R616: F], [BC2457; E605, R613: F, R615: Me, R616: H], [BC2458; E605, R613: Me, R615: F, R616: F], [BC2459; , R613: F, R615: Me, R616: F], [BC2460; E605, R613: Me, R615: Me, R616: F], [BC2461; E605, R613: Me, R615: F, R616: Me], [BC2462; E605, R613: Me, R615: Cl, R616: H], [BC2463; E605, R613: Me, R615: H, R616: Cl], [BC2464; E605, R613: Cl, R615: Me, R616 : H], [BC2465; E605, R613: Me, R615: Cl, R616: Cl], [BC2466; E605, R613: Cl, R615: Me, R616: Cl], [BC2467; E605, R613: Me, R615] : Me, R616: Cl], [BC2468; E605, R613: Me, R615: Cl, R616: Me], [BC2469; E605, R613: Me, R615: Br, R616: H], [BC2470; E605, R613 : Me, R615: H, R616: Br], [BC2471; E605, R613: Br, R615: Me, R616: H], [BC2472; E605, R613: Me, R6 15: Br, R616: Br], [BC2473; E605, R613: Br, R615: Me, R616: Br], [BC2474; E605, R613: Me, R615: Me, R616: Br], [BC2475; R613: Me, R615: Br, R616: Me], [BC2476; E605, R613: Et, R615: H, R616: H], [BC2477; E605, R613: H, R615: Et, R616: H], [ BC2478; E605, R613: Et, R615: Et, R616: H], [BC2479; E605, R613: Et, R615: H, R616: Et], [BC2480; E605, R613: Et, R615: Et, R616: Et], [BC2481; E605, R613: Et, R615: F, R616: H], [BC2482; E605, R613: Et, R615: H, R616: F], [BC2483; E605, R613: F, R615: Et, R616: H], [BC2484; E605, R613: Et, R615: F, R616: F], [BC2485; E605, R613: F, R615: Et, R616: F], [BC2486; E605, R613: Et, R615: Et, R616: F], [BC2487; E605, R613: Et, R615: F, R616: Et], [BC2488; E605, R613: Et, R615: Cl, R616: H], [BC2489; E605, R613: Et, R615: H, R616: Cl], [BC2490; E605, R613: Cl, R615: Et, R616: H], [BC2491; E605, R613: Et, R615: Cl, R616: Cl] [BC2492; E605, R613: Cl, R615: Et, R616: Cl], [BC2493; E605, R613: Et, R615: Et, R616: Cl], [BC2494; E605, R613: Et, R615: Cl, R616: Et], [BC2495; E605, R613: H, R616: H], [BC2496; E605, R613: H, R615: OMe, R616: H], [BC2497; E605, R613: OMe, R615: OMe, R616: H], [BC2498; E605, R613: OMe, R615: H, R616: OMe], [BC2499; E605, R613: OMe, R615: F, R616: H], [BC2500; E605, R613: OMe, R615: H, R616: F],

[BC2501; E605, R613: F, R615: OMe, R616: H], [BC2502; E605, R613: OMe, R615: F, R616: F], [BC2503; E605, R613: F, R615: OMe, R616 : F], [BC2504; E605, R613: OMe, R615: OMe, R616: F], [BC2505; E605, R613: OMe, R615: F, R616: OMe], [BC2506; E605, R613: OMe, R615] : Cl, R 616: H], [BC 2507; E 605, R 613: OMe, R 615: H, R 616: Cl], [BC 2 508; E 605, R 613: Cl, R 615: OMe, R 616: H], [BC 2 509; : OMe, R615: Cl, R616: Cl], [BC 2510; E605, R613: Cl, R615: OMe, R616: Cl], [BC 2511; E605, R613: OMe, R615: OMe, R616: Cl], [BC 2512 E605, R613: OMe, R615: Cl, R616: OMe], [BC2513; E605, R613: Pr, R615: H, R616: H], [BC2514; E605, R613: H, R615: Pr, R616: H ], [BC2515; E605, R613: Pr, R615: H, R616: F], [BC2516; E605, R613: F, R615: Pr, R616: H], [BC2517; E605, R613: Pr, R615: F] , R616: F], [BC2518; E605, R613: Pr, R615: Pr], [BC2519; E605, R613: Pr, R615: Cl, R616: H], [BC2520; E605, R613: Pr] , R615: H, R616: Cl], [BC2521; E605, R613: Cl, R615: Pr, R616: H], [BC2522; E605, R613: Pr, R615: Cl, R616: Cl], [BC2523; , R613: Cl, R615: Pr, R616: Cl], [BC2524; E605, R613: SMe, R615: H, R616: H], [BC2525; E605, R613: H, R615: SMe, R616: H], [BC2526; E605, R613: SMe, R615: H, R616: F], [BC2527; E605, R613: F, R615: SMe, R616: H], [BC2528; E605, R613: SMe, R615: F, R616: F], [BC2529; E605, R613: F, R615: SMe, R616: F], [BC2530; E605, R613: SMe, R615: Cl, R616: H], [BC2531; E605, R613: SMe, R615: H, R616: Cl], [BC 2532; E605, R613: Cl, R615: SMe, R616: H], [BC2533; E605, R613: SMe, R615: Cl, R616: Cl], [BC2534; E605, R613: Cl, R615: SMe, R616: Cl], [BC2535; E606, R612: H, R614: H, R616: H] , [BC2536; E606, R612: Me, R614: H, R616: H], [BC2537; E606, R612: H, R614: Me, R616: H], [BC2538; E606, R612: Me, R614: Me, R616: H], [BC2539; E606, R612: Me, R614: Me, [BC2540; E606, R612: Me, R614: Me, R616: Me], [BC2541; E606, R612: Me, R614: F, R616: H], [BC2542; E606, R612: Me, R614: H, R616: F], [BC 2543; E606, R612: F, R614: Me, R616: H], [BC2544; R612: Me, R614: F, R616: F], [BC2545; E606, R612: F, R614: Me, R616: F], [BC2546; E606, R612: Me, R614: Me, R616: F], [ BC2547; E606, R612: Me, R614: F, R616: Me], [BC2548; E606, R612: Me, R614: Cl, R616: H], [BC2549; E606, R612: Me, R614: H, R616: Cl], [BC2550; E606, R612: Me, R614: H], [BC2551; E606, R612: Me, R614: Cl, R616: Cl], [BC2552; E606, R612: Cl, R614: Me, R616: Cl], [BC2553; E606, R612: Me, R614: Me, R616: Cl], [BC2554; E606, R612: Me, R61 4: Cl, R 616: Me], [BC2 555; E 606, R 612: Me, R 614: Br, R 616: H], [BC 2 556; E 606, R 612: Me, R 614: H, R 616: Br], [BC 2 557; R612: Br, R614: Me, R616: H], [BC2558; E606, R612: Me, R614: Br, R616: Br], [BC2559; E606, R612: Br, R614: Me, R616: Br], [ BC2560; E606, R612: Me, R614: Me, R616: Br], [BC2561; E606, R612: Me, R614: Br, R616: Me], [BC2562; E606, R612: F, R614: H, R616: H], [BC2563; E606, R612: H, R614: F, R616: H], [BC2564; E606, R612: F, R614: F, R616: H], [BC2565; E606, R612: F, R614: H, R616: F], [BC2566; E606, R612: F, R614: F], [BC2567; E606, R612: F, R614: Cl, R616: H], [BC2568; E606, R612: F, R 614: H, R 616: Cl], [BC 2569; E 606, R 612: Cl, R 614: F, R 616: H], [BC 2 570; E 606, R 612: F, R 614: Cl, R 616: Cl], [BC 2571; E606, R612: Cl, R614: F, R616: Cl], [BC2572; E606, R612: F, R614: F, R616: Cl], [BC2573; E606, R612: F, R614: Cl, R616: F] , [BC2574; E606, R612: Et, R614: H], [BC2575; E606, R612: H, R614: Et, R616: H], [BC2576; E606, R612: Et, R614: Et, R 616: H], [BC 2577; E 606, R 612: Et, R 614: H, R 616: Et], [BC 2578; E 606, R 612: Et, R 614: Et, R 616: Et], [BC 2579; E 606, R 612: Et, R614: F, R616: H], [BC2580; E606, R612: Et, R614: H, R616: F], [BC2581; E606, R612: F, R614: Et, R616: H], [B C2582; E606, R612: Et, R614: F, R616: F], [BC 2583; E606, R612: F, R614: Et, R616: F], [BC2584; E606, R612: Et, R614: Et, R616: F], [BC2585; E606, R612: Et, R614: F, R616: Et], [BC2586; E606, R612: Et, R614: Cl, R616: H], [BC2587; E606, R612: Et, R614: H, R616: Cl], [BC2588; E606, R612: Cl, R614: Et, R616: H], [BC2589; E606, R612: Et, R614: Cl, R616: Cl], [BC2590; E606, R612: Cl, R614: Et, R616: Cl], [BC2591; E606, R612: Et, R614: Et, R616: Cl], [BC2592; E606, R612: Et, R614: Cl, R616: Et], [BC2593; E606, R612: OMe, R614: H, R616: H], [BC2594; E606, R612: H, R614: OMe, R616: H], [BC2595; E606, R612: OMe, R614: OMe, R616: H] , [BC2596; E606, R612: OMe, R614: H, R616: OMe], [BC2597; E606, R612: OMe, R614: F, R616: H], [BC2598; E606, R612: OMe, R614: H, R616: F], [BC2599; E606, R612: F, R614: OMe, R616: H], [BC2600; E606, R612: OMe, R614: F, R616: F],

[BC2601; E606, R612: F, R614: OMe, R616: F], [BC2602; E606, R612: OMe, R614: OMe, R616: F], [BC2603; E606, R612: OMe, R614: F, R616 : OMe], [BC2604; E606, R612: Cl, R616: H], [BC2605; E606, R612: OMe, R614: H, R616: Cl], [BC2606; E606, R612: Cl, R614] : OMe, R616: H], [BC2607; E606, R612: Cl, R614: Cl], [BC2608; E606, R612: Cl, R614: OMe, R616: Cl], [BC2609; E606, R612 : OMe, R614: OMe, R616: Cl], [BC2610; E606, R612: OMe, R614: Cl, R616: OMe], [BC2611; E606, R612: Pr, R614: H, R616: H], [BC2612 E606, R612: H, R614: Pr, R616: H], [BC2613; E606, R612: Pr, R614: H, R616: F], [BC2614; E606, R612: F, R614: Pr, R616: H ], [BC2615; E606, R612: Pr, R614: F, R616: F], [BC2616; E606, R612: F, R614: Pr, R616: F], [BC2617; E606, R612: Pr, R614: Cl] , R616: H], [BC2618; E606, R612: Pr, R614: Cl], [BC2619; E606, R612: Cl, R614: Pr, R616: H], [BC 2620; E606, R612: Pr , R614: Cl, R616: Cl], [BC2621; E606, R612: Pr, R614: Pr, R616: Cl], [BC2622; E606, R612: SMe, R614: H, R616: H], [BC2623; , R612: SMe, R616: H], [BC2624; E606, R612: SMe, R614: H, R616: F], [BC2625; E606, R612: F, R614: SMe, R616: H], [BC2626; E606, R612: SMe, R614: F, R616: F], [BC2627; E606, R612: F, R614: SMe, R616: F], [BC2628; E606, R612: SMe, R614: Cl, R616: H], [BC2629; E606, R612: SMe, R614: H, R616: Cl], [BC 2630; E606, R612: Cl, R614: SMe, R616: H], [BC2631; E606, R612: SMe, R614: Cl, R616: Cl], [BC2632; E606, R612: Cl, R614: SMe, R616: Cl], [BC2633; E607, R614: H, R615: H, R616: H], [BC2634; E607, R614: Me, R615: H, R616: H], [BC2635; E607, R614: H, R615: Me, R616: H] [BC2636; E607, R614: Me, R615: Me, R616: H], [BC2637; E607, R614: Me, R615: H, R616: Me], [BC2638; E607, R614: Me, R615: Me, R616: Me], [BC2639; E607, R614: F, R615: H], [BC2640; E607, R614: Me, R615: H, R616: F], [BC2641; E607, R614: F, R615: Me, R616: H], [BC 2642; E 607, R 614: F, R 616: F], [BC 2643; E 607, R 614: F, R 615: Me, R 616: F], [BC 2 644; R614: Me, R615: Me, R616: F], [BC2645; E607, R614: Me, R615: F, R616: Me], [BC2646; E607, R614: Me, R615: Cl, R616: H], [ BC2647; E607, R614: Me, R615: H, R616: Cl], [BC 2648; E607, R614: Cl, R615: Me, R616: H], [BC2649; E607, R614: Me, R615: Cl, R616: Cl], [BC2650; E607, R614: Cl, R615: Me, R616: Cl], [BC2651; E607, R614: Me, R615: Me, R616: Cl], [BC2652; E607, R614: Me, R615: Cl, R616: Me], [BC2653; E607, R614: Me, R615: Br, R616: H], [BC2654; E607, R614: Me, R6 15: H, R 616: Br], [BC 2655; E 607, R 614: Br, R 615: Me, R 616: H], [BC 2 656; E 607, R 614: Me, R 615: Br, R 616: Br], [BC 2 657; R614: Br, R615: Me, R616: Br], [BC2658; E607, R614: Me, R615: Me, R616: Br], [BC2659; E607, R614: Me, R615: Br, R616: Me], [ BC2660; E607, R614: F, R615: H, R616: H], [BC2661; E607, R614: H, R615: F, R616: H], [BC2662; E607, R614: F, R615: F, R616: H], [BC2663; E607, R614: F, R615: H, R616: F], [BC2664; E607, R614: F, R615: F, R616: F], [BC2665; E607, R614: F, R615: Cl, R 616: H], [BC 2 666; E 607, R 614: H, R 616: Cl], [BC 2 667; E 607, R 614: Cl, R 615: F, R 616: H], [BC 2668; E 607, R 614: F, R615: Cl, R616: Cl], [BC2669; E607, R614: Cl, R615: F, R616: Cl], [BC2 670; E607, R614: F, R615: F, R616: Cl], [BC2671; E607, R 614: F, R 615: Cl, R 616: F], [BC 2 672; E 607, R 614: Et, R 615: H, R 616: H], [BC 263; E 607, R 614: H, R 615: Et, R 616: H] [BC2674; E607, R614: Et, R615: Et, R616: H], [BC2675; E607, R614: Et, R615: H, R616: Et], [BC2 676; E607, R614: Et, R615: Et, R616: Et], [BC2677; E607, R614: Et, R615: F, R616: H], [BC2678; E607, R614: Et, R615: H, R616: F], [BC 2679; E607, R614: F, R615: Et, R616: H], [BC2680; E607, R614: Et, R615: F, R616: F], [BC2681; E607, R614: F, R615: Et, R616: F], [BC2 682; E607, R614: Et, R615: Et, R616: F], [BC2683; E607, R614: Et, R615: F, R616: Et], [BC2684; E607, R614: Et, R615: Cl, R616: H], [BC2685; E607, R614: Et, R615: H, R616: Cl], [BC2686; E607, R614: Cl, R615: Et, R616: H], [BC2687; E607, R614: Et, R615: Cl, R616: Cl], [BC2688; E607, R614: Cl, R615: Et, R616: Cl], [BC2689; E607, R614: Et, R615: Et, R616: Cl], [BC2690; E607, R614: Et, R615: Cl, R616: Et], [BC2691; E607, R614: OMe, R615: H, R616: H], [BC2692; E607, R614: H, R615: OMe, R616: H], [BC2693; E607, R614: OMe, R615: OMe, R616: H], [BC2694; E607, R614: OMe, R615: H, R616: OMe], [BC2695; E607, R614: OMe, R615: F, R616: H] , [BC2696; E607, R614: OMe, R615: H, R616: F], [BC2697; E607, R614: F, R615: OMe, R616: H], [BC2698; E607, R614: OMe, R615: F, R 616: F], [BC 2699; E 607, R 614: F, R 615: OMe, R 616: F], [BC 2 700; E 607, R 614: OMe, R 615: OMe, R 616: F],

[BC 2701; E 607, R 614: OMe, R 615: F, R 616: OMe], [BC 2702; E 607, R 614: Cl, R 615: Cl, R 616: H], [BC 2703; E 607, R 614: OMe, R 615: H, R 616 : [Cl], [BC2704; E607, R614: Cl, R615: OMe, R616: H], [BC2705; E607, R614: OMe, R615: Cl, R616: Cl], [BC2706; E607, R614: Cl, R615] : OMe, R616: Cl], [BC2707; E607, R614: OMe, R615: OMe, R616: Cl], [BC2708; E607, R614: OMe, R615: Cl, R616: OMe], [BC2709; E607, R614] : Pr, R 615: H, R 616: H], [BC 2710; E 607, R 614: Pr, R 615: Pr, R 616: H], [BC 2711; E 607, R 614: Pr, R 615: H, R 616: F], [BC 27 12 E607, R614: F, R615: Pr, R616: H], [BC2713; E607, R614: Pr, R615: F, R616: F], [BC2714; E607, R614: F, R615: Pr, R616: F ], [BC2715; E607, R614: Pr, R615: Cl, R616: H], [BC2716; E607, R614: Pr, R615: H, R616: Cl], [BC2717; E607, R614: Cl, R615: Pr] , R616: H], [BC2718; E607, R614: Cl, R615: Cl], [BC2719; E607, R614: Cl, R615: Pr, R616: Cl], [BC2720; E607, R614: SMe , R615: H, R616: H], [BC2721; E607, R614: SMe, R616: H], [BC2722; E607, R614: SMe, R615: H, R616: F], [BC2723; , R614: SMe, R616: H], [BC2724; E607, R614: SMe, R615: F, R616: F], [BC2725; E607, R614: F, R615: SMe, R616: F], [BC2726; E607, R614: SMe, R615: Cl, R616: H], [BC2727; E607, R614: SMe, R615 : H, R 616: Cl], [BC2 728; E 607, R 614: SMe, R 616: H], [BC 2 729; E 607, R 614: S Me, R 615: Cl, R 616: Cl], [BC 2730; E 607, R 614 : Cl, R615: SMe, R616: Cl], [BC2731; E607, R614: OEt, R615: H, R616: H], [BC2732; E607, R614: propargyloxy, R615: H, R616: H], [BC2733 E608, R612: H, R615: H, R616: H], [BC2734; E608, R612: Me, R615: H, R616: H], [BC2 735; E608, R612: H, R615: Me, R616: H ], [BC 2736; E 608, R 612: H, R 615: H, R 616: Me], [BC 2 737; E 608, R 612: Cl, R 615: H, R 616: H], [BC 2 738: E 608, R 612: H, R 615: Cl , R 616: H], [BC 2739; E 608, R 612: H, R 615: H, R 616: Cl], [BC 2740; E 608, R 612: F, R 615: H, R 616: H], [BC 274 1; E 608, R 612: H , R 615: F, R 616: H], [BC 2742; E 608, R 612: H, R 615: H, R 616: F], [BC 2 743; E 608, R 612: OMe, R 615: H, R 616: H], [BC 2 744; , R612: H, R615: OMe, R616: H], [BC2745; E608, R612: H, R615: H, R616: OMe], [BC2746; E608, R612: Et, R615: H, R616: H], [BC 2 747; E 608, R 612: H, R 615: Et, R 616: H], [BC 2 748; E 608, R 612: H, R 615: H, R 616: Et], [BC 2 749: E 608, R 612: Ph, R 615: H, R 616] : H], [BC 2750; E 608, R 612: H, R 615: Ph, R 616: H], [BC 2751; E 608, R 612: H, R 615: H, R 616: Ph], [BC 2752; E 608, R 612: NHCOCH ₃ , R615: H, R 616: H], [BC 2753; E 608, R 612: H, R 615: NHCOCH ₃ , R 616: H], [BC 2 754; E 608, R 612: H, _{R615: H, R616: NHCOCH 3} ], [BC2755; E609, R612: H, R613: H, R616: H], [BC2756; E609, R612: Me, R613: H, R616: H], [BC2757; E609 , R612: H, R613: Me, R616: H], [BC2758; E609, R612: H, R613: H, R616: Me], [BC2759; E609, R612: Cl, R613: H, R616: H], [BC2760; E609, R612: H, R613: Cl, R616: H], [BC2761; E609, R612: H, R613: H, R616: Cl], [BC2762; E609, R612: F, R613: H, R616 : H], [BC2763; E609, R612: H, R613: F, R616: H], [BC2764; E609, R612: H, R613: H, R616: F], [BC2 765; E609, R612: OMe, R613 : H, R 616: H], [BC 2766; E 609, R 612: H, R 613: OMe, R 616: H], [BC 2 767; E 609, R 612: H, R 613: H, R 616: OMe], [BC 2 768; : Et, R 613: H, R 616: H], [BC 2769; E 609, R 612: H, R 613: Et, R 616: H], [BC 2 770; E 609, R 612: H, R 613: H, R 616: Et], [BC 277] E609, R612: Ph, R613: H, R616: H], [BC2772; E609, R612: H, R613: Ph, R616: H], [BC2773; E609, R612: H, R613: H, R616: Ph] [BC2774; E609, R612: SPh, R613: H, R616: H], [BC2775; E609, R612: H, R613: SPh, R616: H], [BC2776; E609, R612: H, R613: H] , R616: SPh], [BC2777; H610, R613: H, R614: H], [BC 2778; E610, R613: Me, R614: H, R616: H], [BC2779; E610, R613: H , R614: Me, R616: H], [BC2780; E610, R613: H, R614: H, R616: Me], [BC2781; E610, R613: Cl, R614: H, R616: H], [BC2 782; E610, R613: H, R614: Cl, R616: H], [BC2783; E610, R613: H, R614: H, R616: Cl], [BC2784; E610, R613: F, R614: H, R616: H], [BC2785; E610, R613: H, R614: F, R616: H], [BC2786; E610, R613: H, R614: H, R616: F], [BC2787; E610, R613: OMe, R614: H, R 616: H], [BC 2 788; E 610, R 613: H, R 614: R 616: H], [BC 2 789; E 610, R 613: H, R 614: H, R 616: OMe], [BC 2 790: E 610, R 613: Et, R614: H, R616: H], [BC2791; E610, R613: H, R614: Et, R616: H], [BC2792; E610, R613: H, R614: H, R616: Et], [BC2793; E610, R 613: Ph, R 614: H, R 616: H], [BC 2 794; E 610, R 613: H, R 614: Ph, R 616: H], [BC 2795; E 610, R 613: H, R 614: H, R 616: Ph] [BC 2796; E610, R 613: benzyl, R 614: H, R 616: H], [BC 2 797; E 610, R 613: H, R 614: benzyl, R 616: H], [BC 2798; E 610, R 613: H, R 614: H, R616: benzyl], [BC2799; E611, R613: H, R615: H], [BC2800; E611, R613: Me, R615: H],

[BC2801; E611, R613: H, R615: Me], [BC2802; E611, R613: Cl, R615: H], [BC 2803; E611, R613: H, R615: Cl], [BC 2804; E611, R613: F , R615: H], [BC2805; E611, R613: H, R615: F], [BC2806; E611, R613: OMe, R615: H], [BC2807; E611, R613: H, R615: OMe], [BC2808] E611, R613: Et, R615: H], [BC2809; E611, R613: H, R615: Et], [BC 2810; E611, R613: Ph, R615: H], [BC 2811; E611, R613: H, R615] : Ph], [BC2812; E6052, R612: H, R613: H], [BC2813; E6052, R612: Me, R613: H], [BC2814; E6052, R612: H, R613: Me], [BC2815; , R612: Cl, R613: H], [BC2816; E6052, R612: H, R613: Cl], [BC2817; E6052, R612: F, R613: H], [BC2818; E6052, R612: H, R613: F [BC2819; E6052, R612: OMe, R613: H], [BC2820; E6052, R612: H, R613: OMe], [BC2821; E6052, R612: Et, R613: H], [BC2822; E6052, R612] : H, R613: Et], [BC2823; E6052, R612: Ph, R613: H], [BC2824; E6052, R612: H, R613: Ph], [BC2825; E613, R612: H, R616: H], [BC2826; E613, R612: Me, R616: H], [BC2827; E613, R612: H, R616: Me], [BC2828; E613, R612: Cl, R616: H], [BC2829; E613, R612: H , R616: Cl], [BC2830; E613, R612: F, R616: H], [BC2831; E613, R612: H, R616: F], [BC2832; E613, R612: OMe, R616: H], [BC2833 E613, R612: H, R616: OMe], [BC2834; E613, R612: Et, R616: H], [BC E 613, R 612: H, R 616: Et], [BC 2 836; E 613, R 612: Ph, R 616: H], [BC 28 37; E 613, R 612: H, R 616: Ph], [BC 2 838; E 614, R 612: H, R614: H], [BC2839; E614, R612: Me, R614: H], [BC2840; E614, R612: H, R614: Me], [BC2841; E614, R612: Cl, R614: H], [BC2842; E614, R612: H, R614: Cl], [BC2843; E614, R612: F, R614: H], [BC 2844; E614, R612: H, R614: F], [BC2845; E614, R612: OMe, R614: H], [BC2846; E614, R612: H, R614: OMe], [BC2847; E614, R612: Et, R614: H], [BC2848; E614, R612: H, R614: Et], [BC2849; E614, R612: Ph, R614: H], [BC2850; E614, R612: Ph, [BC2851; E615, R613: H, R616: H], [BC2852; E615, R613: Me, R616: H] [BC2853; E615, R613: H, R616: Me], [BC2854; E615, R613: Cl, R616: H], [BC2855; E615, R613: H, R616: Cl], [BC2856; E615, R613: F, R 616: H], [BC 2 857; E 615, R 613: H, R 616: F], [BC 2 858; E 615, R 613: OMe, R 616: H], [BC 2859; E 615, R 613: H, R 616: OMe], [ BC2860; E615, R613: Et, R616: H], [BC2861; E615, R613: H, R616: Et], [BC2862; E615, R613: Ph, R616: H], [BC2863; E615, R613: H, R616: Ph], [BC2864; E616, R613: H, R614: H], [BC 2865; E616, R613: Me, R614: H], [BC2866; E616, R613: H, R614: Me], [BC2867; E 616, R 613: Cl, R 614: H], [BC 2 868; E 616, R 613: H, R 614: Cl], [BC 2869; E 616, R 613: F, R614: H], [BC2870; E616, R613: H, R614: F], [BC2871; E616, R613: OMe, R614: H], [BC2872; E616, R613: H, R614: OMe], [BC2873; E616, R613: Et, R614: H], [BC2874; E616, R613: H, R614: Et], [BC2875; E616, R613: Ph, R614: H], [BC 2876; E616, R613: H, R614: Ph], [BC 2877; E 607, R 614: H, R 615: H, R 616: H], [BC 2 878; E 607, R 614: H, R 615: Cl, R 616: H], [BC 2879; H, R 616: Cl].

[Substituent number (MC2); E ¹⁰³ ], [BC 2 880; 1- (ethoxyimino) propyl], [BC2881; 1- (propoxyimino) propyl], [BC2882; 1- (n-butoxyimino) propyl], [BC2883; 1- (Pentyloxyimino) propyl], [BC2884; 1- (Hexyloxyimino) propyl], [BC2885; 1- (Isopropoxyimino) propyl], [BC2288; 1- (tert-butoxyimino) 1- (sec-butoxyimino) propyl], [BC2888; 1- (cyclopropyloxyimino) propyl], [BC2889; 1- (cyclopentyloxyimino) propyl], [BC2890; 1- (Cyclohexyloxyimino) propyl], [BC2891; 1- (3-allyloxyimino) propyl], [BC2892; 1- (3-butenyloxyimino) propyl], [BC2893; 1- (2-propynyloxyimino] ) Propyl], [BC 2894; 1- (3-butynyloxyimino) propyl], [BC 2 895; 1- (1-cyclohexyloxyimino) propyl], [BC2896; 1- (2,2,2-trifluoroethoxyimino) propyl], [BC 2897; 1- (benzyloxyimino) propyl], [BC 2898; 1- (2-fluorobenzyloxyimino) propyl], [BC2899; 1- (3-fluorobenzyloxyimino) propyl], [BC2900; 1- (4-fluorobenzyloxyimino) propyl], [BC2901; 1- (2-chlorobenzyloxyimino) propyl], [BC2902; 1- (3-chlorobenzyloxyimino) propyl], [BC2903; 1- (4-chlorobenzyloxyimino) propyl], [BC2904; 1- (2) -Methylbenzyloxyimino) propyl], [BC2905; 1- (3-methylbenzyloxyimino) propyl], [BC2906; 1- (4-methylbenzyloxyimino) propyl], [BC2907; 1- (2-cyano) Benzyloxyimino) propyl], [BC 2908; 1- (3- 1- (4-cyanobenzyloxyimino) propyl], [BC2910; 1- (2-trifluoromethylbenzyloxyimino) propyl], [BC2911; Trifluoromethylbenzyloxyimino) propyl], [BC2912; 1- (4-trifluoromethylbenzyloxyimino) propyl], [BC2913; 1- (2-difluoromethylbenzyloxyimino) propyl], [BC2914; 1- (3-Difluoromethylbenzyloxyimino) propyl], [BC2915; 1- (4-difluoromethylbenzyloxyimino) propyl], [BC2916; 1- (2-methoxybenzyloxyimino) propyl], [BC2917; 1- (3-methoxybenzyloxyimino) propyl], [BC2918; 1- (4-methoxybenzyloxyimino) propyl], [BC2919; 1- (2-vinylbenzyloxyimino) propyl], [BC2920; 1- 3-vinylbenzyloxyimino) propyl], [BC2921; 1- (4-vinylbenzyloxyimino) propyl], [BC2922; 1- (2-phenylbenzyloxyimino) propyl], [BC2923; 1- (3-) Phenylbenzyloxyimino) propyl], [BC2924; 1- (4-phenylbenzyloxyimino) propyl], [BC2925; 1- (2,3-difluorobenzyloxyimino) propyl], [BC2926; 1- (2, 2, 4-difluorobenzyloxyimino) propyl], [BC2 927; 1- (2,5-difluorobenzyloxyimino) propyl], [BC2 928; 1- (2,6-difluorobenzyloxyimino) propyl], [BC2 929; 1 -(3,4-difluorobenzyloxyimino) propyl], [BC2930; 1- (3,5-difluorobenzyloxyimino) propyl], [BC2931; 1- (2,3,4,5,6-pentafluoro) Benzyloxyimino) propi 1- (3-ethylbenzyloxyimino) propyl], [BC 2933; 1- (4-ethylbenzyloxyimino) propyl], [BC 2934; 1- (2-trifluoromethoxybenzyloxyimino) propyl] ], [BC2935; 1- (3-trifluoromethoxybenzyloxyimino) propyl], [BC2936; 1- (4-trifluoromethoxybenzyloxyimino) propyl], [BC2937; 1- (methoxyimino) propyl], [BC 2938; 1- (ethoxyimino) butyl], [BC 2939; 1- (propoxyimino) butyl], [BC 2940; 1- (n-butoxyimino) butyl], [BC 2941; 1- (pentyloxyimino) butyl] , [BC2942; 1- (hexyloxyimino) butyl], [BC2943; 1- (isopropoxyimino) butyl], [BC2944; 1- (tert-butoxyimino) butyl], [BC2945; 1- (sec-butoxy) Imino) butyl], [BC 2946; 1- (cyclopropyloxyl) Mino) butyl], [BC2947; 1- (cyclopentyloxyimino) butyl], [BC2948; 1- (cyclohexyloxyimino) butyl], [BC2949; 1- (3-allyloxyimino) butyl], [BC2950; 1- (3-Butenyloxyimino) butyl], [BC 2951; 1- (2-propynyloxyimino) butyl], [BC 2952; 1- (3-butynyloxyimino) butyl], 1-Cyclohexyloxyimino) butyl], [BC 2 954; 1- (2,2,2-trifluoroethoxyimino) butyl], [BC 2 955; 1- (benzyloxyimino) butyl], [BC 2 956; Fluorobenzyloxyimino) butyl], [BC2957; 1- (3-fluorobenzyloxyimino) butyl], [BC2958; 1- (4-fluorobenzyloxyimino) butyl], [BC2959; 1- (2-chlorobenzyl) Oximino) butyl], [BC2960; 1- (3-chlorobenzyloxyimino) butyl], [BC2961; 1- (4-chlorobenzyloxyimino) butyl], [BC2962; 1- (2-methylbenzyloxyimino) butyl], [BC2963; 1- (3-methylbenzyloxyimino) butyl], [BC2964; 1- (4-Methylbenzyloxyimino) butyl], [BC2965; 1- (2-cyanobenzyloxyimino) butyl], [BC2966; 1- (3-cyanobenzyloxyimino) butyl], [BC2967; 1- (4) -Cyanobenzyloxyimino) butyl], [BC2968; 1- (2-trifluoromethylbenzyloxyimino) butyl], [BC2969; 1- (3-trifluoromethylbenzyloxyimino) butyl], [BC2970; 1- (4-Trifluoromethylbenzyloxyimino) butyl], [BC2971; 1- (2-difluoromethylbenzyloxyimino) butyl], [BC2972; 1- (3-difluoromethylbenzyloxyimino) butyl], [BC2973; 1- (4-difluoromethylbenzylo Siimino) butyl], [BC2974; 1- (2-methoxybenzyloxyimino) butyl], [BC2975; 1- (3-methoxybenzyloxyimino) butyl], [BC2976; 1- (4-methoxybenzyloxyimino) Butyl], [BC2977; 1- (2-vinylbenzyloxyimino) butyl], [BC2978; 1- (3-vinylbenzyloxyimino) butyl], [BC2979; 1- (4-vinylbenzyloxyimino) butyl] ,

[BC 2 980; 1- (2-phenylbenzyloxyimino) butyl], [BC2981; 1- (3-phenylbenzyloxyimino) butyl], [BC2982; 1- (4-phenylbenzyloxyimino) butyl], [BC2983 1- (2,3-difluorobenzyloxyimino) butyl], [BC2984; 1- (2,4-difluorobenzyloxyimino) butyl], [BC2985; 1- (2,5-difluorobenzyloxyimino) butyl 1- (2,6-difluorobenzyloxyimino) butyl], [BC 2987; 1- (3,4-difluorobenzyloxyimino) butyl], [BC2988; 1- (3,5-difluorobenzyl)] Oxyimino) butyl], [BC2989; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) butyl], [BC2990; 1- (3-ethylbenzyloxyimino) butyl], [BC2991; 1- (4-ethylbenzyloxyimino) butyl], [BC 299 2; 1- (2- Trifluoromethoxybenzyloxyimino) butyl], [BC2993; 1- (3-trifluoromethoxybenzyloxyimino) butyl], [BC2994; 1- (4-trifluoromethoxybenzyloxyimino) butyl], [BC2995; 1 -(Methoxyimino) butyl], [BC2996; 1- (ethoxyimino) pentyl], [BC2997; 1- (propoxyimino) pentyl], [BC2998; 1- (n-butoxyimino) pentyl], [BC2999; 1 -(Pentyloxyimino) pentyl], [BC 3000; 1-(hexyloxyimino) pentyl], [BC 3001; 1-(isopropoxy imino) pentyl], [BC 3002; 1-(tert- butoxyimino) pentyl], [ BC3003; 1- (sec-butoxyimino) pentyl], [BC3004; 1- (cyclopropyloxyimino) pentyl], [BC3005; 1- (cyclopentyloxyimino) pentyl], [BC3006; 1- (cyclohexyloxyimino) ) Pentyl], [B C 3007; 1- (3-allyloxyimino) pentyl], [BC 3008; 1- (3-butenyloxy imino) pentyl], [BC 3009; 1- (2-propynyloxy imino) pentyl], [BC 3010; 1- (3-butynyloxyimino) pentyl], [BC3011; 1- (1-cyclohexyloxyimino) pentyl], [BC3012; 1- (2,2,2-trifluoroethoxyimino) pentyl], [BC3013; 1 -(Benzyloxyimino) pentyl, [BC3014; 1- (2-fluorobenzyloxyimino) pentyl], [BC3015; 1- (3-fluorobenzyloxyimino) pentyl], [BC3016; 1- (4-fluoro) Benzyloxyimino) pentyl], [BC3017; 1- (2-chlorobenzyloxyimino) pentyl], [BC3018; 1- (3-chlorobenzyloxyimino) pentyl], [BC3019; 1- (4-chlorobenzyloxy) Imino) pentyl], [BC 3020; 1- (2-methylbenzyloxy) Imino) pentyl], [BC3021; 1- (3-methylbenzyloxyimino) pentyl], [BC3022; 1- (4-methylbenzyloxyimino) pentyl], [BC3023; 1- (2-cyanobenzyloxyimino) Pentyl], [BC3024; 1- (3-cyanobenzyloxyimino) pentyl], [BC3025; 1- (4-cyanobenzyloxyimino) pentyl], [BC3026; 1- (2-trifluoromethylbenzyloxyimino) Pentyl], [BC3027; 1- (3-trifluoromethylbenzyloxyimino) pentyl], [BC3028; 1- (4-trifluoromethylbenzyloxyimino) pentyl], [BC3029; 1- (2-difluoromethylbenzyl) Oximino) pentyl], [BC3030; 1- (3-difluoromethylbenzyloxyimino) pentyl], [BC3031; 1- (4-difluoromethylbenzyloxyimino) pentyl], [BC3032; 1- (2-methoxybenzyl) Oki Imino) pentyl], [BC 3033; 1- (3-methoxybenzyloxyimino) pentyl], [BC 3034; 1- (4-methoxybenzyloxyimino) pentyl], [BC 3035; 1- (2-vinylbenzyloxyimino) Pentyl], [BC3036; 1- (3-vinylbenzyloxyimino) pentyl], [BC3037; 1- (4-vinylbenzyloxyimino) pentyl], [BC3038; 1- (2-phenylbenzyloxyimino) pentyl] [BC 3039; 1- (3-phenylbenzyloxyimino) pentyl], [BC3040; 1- (4-phenylbenzyloxyimino) pentyl], [BC3041; 1- (2,3-difluorobenzyloxyimino) pentyl] , [BC3042; 1- (2,4-difluorobenzyloxyimino) pentyl], [BC3043; 1- (2,5-difluorobenzyloxyimino) pentyl], [BC3044; 1- (2,6-difluorobenzyloxy) Imino) pentyl], [BC 3045; -(3,4-difluorobenzyloxyimino) pentyl], [BC 3046; 1- (3,5-difluorobenzyloxyimino) pentyl], [BC 3047; 1- (2,3,4,5,6-pentafluoro) Benzyloxyimino) pentyl], [BC3048; 1- (3-ethylbenzyloxyimino) pentyl], [BC3049; 1- (4-ethylbenzyloxyimino) pentyl], [BC3050; 1- (2-trifluoromethoxy) Benzyloxyimino) pentyl], [BC3051; 1- (3-trifluoromethoxybenzyloxyimino) pentyl], [BC3052; 1- (4-trifluoromethoxybenzyloxyiminopentyl], [BC3053; 1- (methoxyimino) ) Pentyl], [BC3054; 1- (3-fluorobenzyloxyimino) (phenyl) methyl], [BC3055; 1- (ethoxyimino) -2-methylpropyl], [BC3056; 1- (propoxyimino) -2 -Methylpropyl], [BC305 7; 1- (n-butoxyimino) -2-methylpropyl], [BC3058; 1- (pentyloxyimino) -2-methylpropyl], [BC3059; 1- (hexyloxyimino) -2-methylpropyl] 1- (Isopropoxyimino) -2-methylpropyl], [BC3061; 1- (tert-butoxyimino) -2-methylpropyl], [BC3062; 1- (sec-butoxyimino) -2-] Methylpropyl], [BC 3063; 1- (cyclopropyloxyimino) -2-methylpropyl], [BC 3064; 1- (cyclopentyloxyimino) -2-methylpropyl], [BC 3065; 1- (cyclohexyloxyimino) -2-Methylpropyl], [BC 3066; 1- (3-allyloxyimino) -2-methylpropyl], [BC 3067; 1- (3-butenyloxyimino) -2-methylpropyl], [BC 3068; 1 -(2-propynyloxyimino) -2-methylpropyl], [BC3069; 1- (3-butynyloxyimino)- -Methylpropyl], [BC3070; 1- (1-cyclohexyloxyimino) -2-methylpropyl], [BC3071; 1- (2,2,2-trifluoroethoxyimino) -2-methylpropyl], [BC3072 1- (benzyloxyimino) -2-methylpropyl], [BC 3073; 1- (2-fluorobenzyloxyimino) -2-methylpropyl], [BC 3074; 1- (3-fluorobenzyloxyimino) -2 -Methylpropyl], [BC 3075; 1- (4-fluorobenzyloxyimino) -2-methylpropyl], [BC 3076; 1- (2-chlorobenzyloxyimino) -2-methylpropyl], [BC 3077; 1- (3-chlorobenzyloxyimino) -2-methylpropyl], [BC3078; 1- (4-chlorobenzyloxyimino) -2-methylpropyl], [BC3079; 1- (2-methylbenzyloxyimino) -2 -Methylpropyl],

[BC 3080; 1- (3-methylbenzyloxyimino) -2-methylpropyl], [BC3081; 1- (4-methylbenzyloxyimino) -2-methylpropyl], [BC3082; 1- (2-cyanobenzyl) Oximino) -2-methylpropyl], [BC3083; 1- (3-cyanobenzyloxyimino) -2-methylpropyl], [BC3084; 1- (4-cyanobenzyloxyimino) -2-methylpropyl], [BC 3085; 1- (2-trifluoromethylbenzyloxyimino) -2-methylpropyl], [BC 3086; 1- (3-trifluoromethylbenzyloxyimino) -2-methylpropyl], [BC 3087; 4-trifluoromethylbenzyloxyimino) -2-methylpropyl], [BC3088; 1- (2-difluoromethylbenzyloxyimino) -2-methylpropyl], [BC3089; 1- (3-difluoromethylbenzyloxyimino] ) -2-Methylpropyl], [BC 3090; 1- (4-Dif Omethylbenzyloxyimino) -2-methylpropyl], [BC3091; 1- (2-methoxybenzyloxyimino) -2-methylpropyl], [BC3092; 1- (3-methoxybenzyloxyimino) -2-methyl] Propyl], [BC 3093; 1- (4-methoxybenzyloxyimino) -2-methylpropyl], [BC 3094; 1- (2-vinylbenzyloxyimino) -2-methylpropyl], [BC 3095; 1- (3) -Vinylbenzyloxyimino) -2-methylpropyl], [BC3096; 1- (4-vinylbenzyloxyimino) -2-methylpropyl], [BC3097; 1- (2-phenylbenzyloxyimino) -2-methyl] Propyl], [BC 3098; 1- (3-phenylbenzyloxyimino) -2-methylpropyl], [BC3099; 1- (4-phenylbenzyloxyimino) -2-methylpropyl], [BC 3100; 1- (2) , 3-Difluorobenzyloxyimino) -2-methylpropyl] , [BC3101; 1- (2,4-difluorobenzyloxyimino) -2-methylpropyl], [BC3102; 1- (2,5-difluorobenzyloxyimino) -2-methylpropyl], BC 3103; 1- (2,6-Difluorobenzyloxyimino) -2-methylpropyl], [BC 3104; 1- (3,4-Difluorobenzyloxyimino) -2-methylpropyl], [BC 3105; 1- (3,5-Difluorobenzyloxyimino) -2-methylpropyl], [BC 3106; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) -2-methylpropyl], [BC 3107; 1- (3-ethylbenzyloxyimino) -2-methylpropyl], [BC 3108; 1- (4-ethylbenzyloxyimino) -2-methylpropyl], [BC 3109; 1- (2-trifluoro) Methoxybenzyloxyimino) -2-methylpropyl], [BC 3110; 1- (3-trifluoromethoxybenzyl) Siimino) -2-methylpropyl], [BC3111; 1- (4-trifluoromethoxybenzyloxyimino) -2-methylpropyl], [BC3112; 1- (methoxyimino) -2-methylpropyl], [BC3113; 1- (Ethoxyimino) -2,2-dimethylpropyl], [BC3114; 1- (propoxyimino) -2,2-dimethylpropyl], [BC3115; 1- (n-butoxyimino) -2,2-dimethyl Propyl], [BC3116; 1- (pentyloxyimino) -2,2-dimethylpropyl], [BC3117; 1- (hexyloxyimino) -2,2-dimethylpropyl], [BC3118; 1- (isopropoxyimino) ) -2,2-dimethylpropyl], [BC3119; 1- (tert-butoxyimino) -2,2-dimethylpropyl], [BC3120; 1- (sec-butoxyimino) -2,2-dimethylpropyl], [BC 3121; 1- (cyclopropyloxyimino) -2,2-dimethylpropyl], [BC 3122; Lopentyloxyimino) -2,2-dimethylpropyl], [BC3123; 1- (cyclohexyloxyimino) -2,2-dimethylpropyl], [BC3124; 1- (3-allyloxyimino) -2,2- Dimethylpropyl], [BC3125; 1- (3-butenyloxyimino) -2,2-dimethylpropyl], [BC3126; 1- (2-propynyloxyimino) -2,2-dimethylpropyl], [BC3127; 1- (3-butynyloxyimino) -2,2-dimethylpropyl], [BC3128; 1- (1-cyclohexyloxyimino) -2,2-dimethylpropyl], [BC3129; 1- (2,2,7) 2-trifluoroethoxyimino) -2,2-dimethylpropyl], [BC3130; 1- (benzyloxyimino) -2,2-dimethylpropyl], [BC3131; 1- (2-fluorobenzyloxyimino) -2 , 2-Dimethylpropyl], [BC 3132; 1- (3-fluorobenzyloxyimino) -2,2-dime 1- (4-fluorobenzyloxyimino) -2,2-dimethylpropyl], [BC 3134; 1- (2-chlorobenzyloxyimino) -2,2-dimethylpropyl], [BC 3135; 1- (3-chlorobenzyloxyimino) -2,2-dimethylpropyl], [BC3136; 1- (4-chlorobenzyloxyimino) -2,2-dimethylpropyl], [BC3137; 1- (2-methyl) Benzyloxyimino) -2,2-dimethylpropyl], [BC3138; 1- (3-methylbenzyloxyimino) -2,2-dimethylpropyl], [BC3139; 1- (4-methylbenzyloxyimino) -2 , 2-Dimethylpropyl], [BC3140; 1- (2-cyanobenzyloxyimino) -2,2-dimethylpropyl], [BC3141; 1- (3-cyanobenzyloxyimino) -2,2-dimethylpropyl] , [BC 3142; 1- (4-cyanobenzyloxyimino) -2,2-dimethylpropyl ], [BC 3143; 1- (2-trifluoromethylbenzyloxyimino) -2,2-dimethylpropyl], [BC3144; 1- (3-trifluoromethylbenzyloxyimino) -2,2-dimethylpropyl], [BC 3145; 1- (4-trifluoromethylbenzyloxyimino) -2,2-dimethylpropyl], [BC 3146; 1- (2-difluoromethylbenzyloxyimino) -2,2-dimethylpropyl], [BC 3147; 1- (3-Difluoromethylbenzyloxyimino) -2,2-dimethylpropyl], [BC3148; 1- (4-difluoromethylbenzyloxyimino) -2,2-dimethylpropyl], [BC3149; 1- (2 -Methoxybenzyloxyimino) -2,2-dimethylpropyl], [BC3150; 1- (3-methoxybenzyloxyimino) -2,2-dimethylpropyl], [BC3151; 1- (4-methoxybenzyloxyimino) -2,2-Dimethylpropyl], [BC3152; 1- (2-vinylbenzyloxyimino) -2,2-dimethylpropyl], [BC 3153; 1- (3-vinylbenzyloxyimino) -2,2-dimethylpropyl], [BC 3154; 1- (4-vinyl] Benzyloxyimino) -2,2-dimethylpropyl], [BC3155; 1- (2-phenylbenzyloxyimino) -2,2-dimethylpropyl], [BC3156; 1- (3-phenylbenzyloxyimino) -2 , 2-Dimethylpropyl], [BC3157; 1- (4-phenylbenzyloxyimino) -2,2-dimethylpropyl], [BC3158; 1- (2,3-difluorobenzyloxyimino) -2,2-dimethyl Propyl], [BC 3159; 1- (2,4-difluorobenzyloxyimino) -2,2-dimethylpropyl], [BC 3160; 1- (2,5-difluorobenzyloxyimino) -2,2-dimethylpropyl] [BC 3161; 1- (2, 6-difluorobenzyloxyimino) -2, -Dimethylpropyl], [BC3162; 1- (3,4-difluorobenzyloxyimino) -2,2-dimethylpropyl], [BC3163; 1- (3,5-difluorobenzyloxyimino) -2,2-dimethyl Propyl], [BC 3 164; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) -2,2-dimethylpropyl], [BC3165; 1- (3-ethylbenzyloxyimino) -2, 2-Dimethylpropyl], [BC3166; 1- (4-ethylbenzyloxyimino) -2,2-dimethylpropyl], [BC3167; 1- (2-trifluoromethoxybenzyloxyimino) -2,2-dimethylpropyl ], [BC 3168; 1- (3-trifluoromethoxybenzyloxyimino) -2,2-dimethylpropyl], [BC 3169; 1- (4-trifluoromethoxybenzyloxyimino) -2,2-dimethylpropyl], [BC 3170; 1- (methoxyimino) -2,2-dimethyl Ropyl], [BC 3171; 1- (ethoxyimino) (cyclopropyl) methyl], [BC 3172; 1- (propoxyimino) (cyclopropyl) methyl], [BC 3173; 1- (n-butoxyimino) (cyclopropyl) Methyl], [BC3174; 1- (pentyloxyimino) (cyclopropyl) methyl], [BC3175; 1- (hexyloxyimino) (cyclopropyl) methyl], [BC3176; 1- (isopropoxyimino) (cyclopropyl) 1) (meth) methyl], [BC3177; 1- (tert- butoxyimino) (cyclopropyl) methyl], [BC 3178; 1-(sec- butoxyimino) (cyclopropyl) methyl], [BC 3179; ) (Cyclopropyl) methyl],

[BC 3180; 1- (cyclopentyloxyimino) (cyclopropyl) methyl], [BC3181; 1- (cyclohexyloxyimino) (cyclopropyl) methyl], [BC3182; 1- (3-allyloxyimino) (cyclopropyl] 1) (methyl), [BC3183; 1- (3-butenyloxyimino) (cyclopropyl) methyl], [BC3184; 1- (2-propynyloxyimino) (cyclopropyl) methyl], [BC3185; 1- (3) -Butynyloxyimino) (cyclopropyl) methyl], [BC3186; 1- (1-cyclohexyloxyimino) (cyclopropyl) methyl], [BC3187; 1- (2,2,2-trifluoroethoxyimino) ( Cyclopropyl) methyl], [BC3188; 1- (benzyloxyimino) (cyclopropyl) methyl], [BC3189; 1- (2-fluorobenzyloxyimino) (cyclopropyl) methyl], [BC3190; 1- (3) -Fluorobenzyloxy Imino) (cyclopropyl) methyl], [BC 3191; 1- (4-fluorobenzyloxyimino) (cyclopropyl) methyl], [BC3192; 1- (2-chlorobenzyloxyimino) (cyclopropyl) methyl], [BC3192; BC 3193; 1- (3-chlorobenzyloxyimino) (cyclopropyl) methyl], [BC3194; 1- (4-chlorobenzyloxyimino) (cyclopropyl) methyl], [BC3195; 1- (2-methylbenzyloxy) Imino) (cyclopropyl) methyl], [BC3196; 1- (3-methylbenzyloxyimino) (cyclopropyl) methyl], [BC3197; 1- (4-methylbenzyloxyimino) (cyclopropyl) methyl], BC 3198; 1- (2-cyanobenzyloxyimino) (cyclopropyl) methyl], [BC3199; 1- (3-cyanobenzyloxyimino) (cyclopropyl) methyl], [BC3200; 1- (4-cyanobenzyloxy) Imi ) (Cyclopropyl) methyl], [BC3201; 1- (2-trifluoromethylbenzyloxyimino) (cyclopropyl) methyl], [BC3202; 1- (3-trifluoromethylbenzyloxyimino) (cyclopropyl) methyl 1- (4-Trifluoromethylbenzyloxyimino) (cyclopropyl) methyl], [BC3204; 1- (2-difluoromethylbenzyloxyimino) (cyclopropyl) methyl], [BC3205; 1- (3-Difluoromethylbenzyloxyimino) (cyclopropyl) methyl], [BC3206; 1- (4-difluoromethylbenzyloxyimino) (cyclopropyl) methyl], [BC3207; 1- (2-methoxybenzyloxyimino) (Cyclopropyl) methyl], [BC3208; 1- (3-methoxybenzyloxyimino) (cyclopropyl) methyl], [BC3209; 1- (4-methoxybenzyloxyimime] 1) (cyclopropyl) methyl], [BC 3210; 1-(2-vinylbenzyloxyimino) (cyclopropyl) methyl], [BC 3211; 1-(3- vinylbenzyloxyimino) (cyclopropyl) methyl], [BC 32 12 1- (4-vinylbenzyloxyimino) (cyclopropyl) methyl], [BC3213; 1- (2-phenylbenzyloxyimino) (cyclopropyl) methyl], [BC3214; 1- (3-phenylbenzyloxyimino] 1) (cyclopropyl) methyl], [BC 3215; 1- (4-phenylbenzyloxyimino) (cyclopropyl) methyl], [BC 3216; 1-(2,3-difluorobenzyloxyimino) (cyclopropyl) methyl], [BC 3217; 1- (2,4-difluorobenzyloxyimino) (cyclopropyl) methyl], [BC 3218; 1-(2, 5-difluorobenzyloxyimino) (cyclopropyl) methyl], [BC 32 19; 2, -Difluorobenzyloxyimino) (cyclopropyl) methyl], [BC3220; 1- (3,4-difluorobenzyloxyimino) (cyclopropyl) methyl], [BC3221; 1- (3,5-difluorobenzyloxyimino) (Cyclopropyl) methyl], [BC3222; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (cyclopropyl) methyl], [BC3223; 1- (3-ethylbenzyloxyimino) ( Cyclopropyl) methyl], [BC3224; 1- (4-ethylbenzyloxyimino) (cyclopropyl) methyl], [BC3225; 1- (2-trifluoromethoxybenzyloxyimino) (cyclopropyl) methyl], [BC3226 1- (3-trifluoromethoxybenzyloxyimino) (cyclopropyl) methyl], [BC3227; 1- (4-trifluoromethoxybenzyloxyimino) (cyclopropyl) methyl 1- (Methoxyimino) (cyclopropyl) methyl], [BC3229; 1- (ethoxyimino) (cyclobutyl) methyl], [BC3230; 1- (propoxyimino) (cyclobutyl) methyl], [BC3231] 1- (n-butoxyimino) (cyclobutyl) methyl], [BC3232; 1- (pentyloxyimino) (cyclobutyl) methyl], [BC3233; 1- (hexyloxyimino) (cyclobutyl) methyl], [BC3234; 1- (Isopropoxyimino) (cyclobutyl) methyl], [BC3235; 1- (tert-butoxyimino) (cyclobutyl) methyl], [BC3236; 1- (sec-butoxyimino) (cyclobutyl) methyl], [BC3237; 1- (cyclopropyloxyimino) (cyclobutyl) methyl], [BC3238; 1- (cyclopentyloxyimino) (cyclobutyl) methyl], [BC3239; 1- (cyclohexyloxyimino) (cyclobutyl) methyl], [BC 3240; 1- (3-allyloxyimino) (cyclobutyl) methyl], [BC3241; 1- (3-butenyloxyimino) (cyclobutyl) methyl], [BC3242; 1- (2-propynyloxyimino) ( Cyclobutyl) methyl], [BC3243; 1- (3-butynyloxyimino) (cyclobutyl) methyl], [BC3244; 1- (1-cyclohexyloxyimino) (cyclobutyl) methyl], [BC3245; 2,2-trifluoroethoxyimino) (cyclobutyl) methyl], [BC3246; 1- (benzyloxyimino) (cyclobutyl) methyl], [BC3247; 1- (2-fluorobenzyloxyimino) (cyclobutyl) methyl], [BC 3248; 1- (3-fluorobenzyloxyimino) (cyclobutyl) methyl], [BC3249; 1- (4-fluorobenzyloxyimino) (cyclobutyl) methyl], [BC3250; 1- (2-chlorobenzyloxyimino) ) Cyclobutyl) methyl], [BC3251; 1- (3-chlorobenzyloxyimino) (cyclobutyl) methyl], [BC3252; 1- (4-chlorobenzyloxyimino) (cyclobutyl) methyl], [BC3253; 1- (2) -Methylbenzyloxyimino) (cyclobutyl) methyl], [BC3254; 1- (3-methylbenzyloxyimino) (cyclobutyl) methyl], [BC3255; 1- (4-methylbenzyloxyimino) (cyclobutyl) methyl], [BC 3256; 1- (2-cyanobenzyloxyimino) (cyclobutyl) methyl], [BC3257; 1- (3-cyanobenzyloxyimino) (cyclobutyl) methyl], [BC3258; 1- (4-cyanobenzyloxyimino] ) (Cyclobutyl) methyl], [BC3259; 1- (2-trifluoromethylbenzyloxyimino) (cyclobutyl) methyl], [BC3260; 1- (3-trifluoromethylbenzyloxyimino) ( Chlorobutyl) methyl], [BC3261; 1- (4-trifluoromethylbenzyloxyimino) (cyclobutyl) methyl], [BC3262; 1- (2-difluoromethylbenzyloxyimino) (cyclobutyl) methyl], [BC3263; 1 -(3-Difluoromethylbenzyloxyimino) (cyclobutyl) methyl], [BC3264; 1- (4-difluoromethylbenzyloxyimino) (cyclobutyl) methyl], [BC3265; 1- (2-methoxybenzyloxyimino) ( Cyclobutyl) methyl], [BC3266; 1- (3-methoxybenzyloxyimino) (cyclobutyl) methyl], [BC3267; 1- (4-methoxybenzyloxyimino) (cyclobutyl) methyl], [BC3268; 1- (2) -Vinylbenzyloxyimino) (cyclobutyl) methyl], [BC3269; 1- (3-vinylbenzyloxyimino) (cyclobutyl) methyl], [BC3270; 1- (4-vinylbenzene) Diloxyimino) (cyclobutyl) methyl], [BC 3271; 1- (2-phenylbenzyloxyimino) (cyclobutyl) methyl], [BC3272; 1- (4-phenylbenzyloxyimino) (cyclobutyl) methyl], [BC3274; 1- (2,3-difluorobenzyloxyimino) (cyclobutyl) methyl], [BC3275; 1- (2,4-difluorobenzyl) Oxyimino) (cyclobutyl) methyl], [BC3276; 1- (2,5-difluorobenzyloxyimino) (cyclobutyl) methyl], [BC3277; 1- (2,6-difluorobenzyloxyimino) (cyclobutyl) methyl] [BC 3278; 1- (3,4-difluorobenzyloxyimino) (cyclobutyl) methyl], [BC3279; 1- (3,5-difluorobenzyloxyimino) (cyclobutyl) Le],

[BC 3280; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (cyclobutyl) methyl], [BC3281; 1- (3-ethylbenzyloxyimino) (cyclobutyl) methyl], [BC3282; 1- (4-ethylbenzyloxyimino) (cyclobutyl) methyl], [BC3283; 1- (2-trifluoromethoxybenzyloxyimino) (cyclobutyl) methyl], [BC3284; 1- (3-trifluoromethoxybenzylo] Roxyimino) (cyclobutyl) methyl], [BC3285; 1- (4-trifluoromethoxybenzyloxyimino) (cyclobutyl) methyl], [BC3286; 1- (methoxyimino) (cyclobutyl) methyl], [BC3287; 1- (Ethoxyimino) (cyclopentyl) methyl], [BC3288; 1- (propoxyimino) (cyclopentyl) methyl], [BC3289; 1- (n-butoxyimino) (cyclopentyl) methyl], [BC3290; -(Pentyloxyimino) (cyclopentyl) methyl], [BC3291; 1-(hexyloxyimino) (cyclopentyl) methyl], [BC3292; 1-(isopropoxyimino) (cyclopentyl) methyl], [BC 3293; tert-Butoxyimino) (cyclopentyl) methyl], [BC3294; 1- (sec-butoxyimino) (cyclopentyl) methyl], [BC3295; 1- (cyclopropyloxyimino) (cyclopentyl) methyl], [BC3296; 1- (Cyclopentyloxyimino) (cyclopentyl) methyl], [BC3297; 1- (cyclohexyloxyimino) (cyclopentyl) methyl], [BC3298; 1- (3-allyloxyimino) (cyclopentyl) methyl], [BC3299; 1 -(3-Butenyloxyimino) (cyclopentyl) methyl], [BC3300; 1- (2-propynyloxyimino) (cyclopentyl) methyl], [BC3301; 1- (3-) Tynyloxyimino) (cyclopentyl) methyl], [BC3302; 1- (1-cyclohexyloxyimino) (cyclopentyl) methyl], [BC3303; 1- (2,2,2-trifluoroethoxyimino) (cyclopentyl) methyl 1- (benzyloxyimino) (cyclopentyl) methyl], [BC3305; 1- (2-fluorobenzyloxyimino) (cyclopentyl) methyl], [BC3306; 1- (3-fluorobenzyloxyimino)] (Cyclopentyl) methyl], [BC3307; 1- (4-fluorobenzyloxyimino) (cyclopentyl) methyl], [BC3308; 1- (2-chlorobenzyloxyimino) (cyclopentyl) methyl], [BC3309; 3-chlorobenzyloxyimino) (cyclopentyl) methyl], [BC 3310; 1- (4-chlorobenzyloxyimino) (cyclopentyl) methyl], [BC 3311; 1- (2-methyl bene) 1- (3-methylbenzyloxyimino) (cyclopentyl) methyl], [BC3313; 1- (4-methylbenzyloxyimino) (cyclopentyl) methyl], BC3314; 1- (2-cyanobenzyloxyimino) (cyclopentyl) methyl], [BC3315; 1- (3-cyanobenzyloxyimino) (cyclopentyl) methyl], [BC3316; 1- (4-cyanobenzyloxyimino) (Cyclopentyl) methyl], [BC3317; 1- (2-trifluoromethylbenzyloxyimino) (cyclopentyl) methyl], [BC3318; 1- (3-trifluoromethylbenzyloxyimino) (cyclopentyl) methyl], [BC3319 1- (4-trifluoromethylbenzyloxyimino) (cyclopentyl) methyl], [BC3320; 1- (2-difluoromethylbenzyloxyimino) (sic) Pentyl) methyl], [BC3321; 1- (3-difluoromethylbenzyloxyimino) (cyclopentyl) methyl], [BC3322; 1- (4-difluoromethylbenzyloxyimino) (cyclopentyl) methyl], [BC3323; 1- (2-methoxybenzyloxyimino) (cyclopentyl) methyl], [BC3324; 1- (3-methoxybenzyloxyimino) (cyclopentyl) methyl], [BC3325; 1- (4-methoxybenzyloxyimino) (cyclopentyl) methyl ], [BC3326; 1- (2-vinylbenzyloxyimino) (cyclopentyl) methyl], [BC3327; 1- (3-vinylbenzyloxyimino) (cyclopentyl) methyl], [BC3328; 1- (4-vinylbenzyl) Oxyimino) (cyclopentyl) methyl], [BC3329; 1- (2-phenylbenzyloxyimino) (cyclopentyl) methyl], [BC3330; 1- (3-phenylbenzene) 1- (4-phenylbenzyloxyimino) (cyclopentyl) methyl], [BC3332; 1- (2,3-difluorobenzyloxyimino) (cyclopentyl) methyl], [BC3333] 1- (2,4-difluorobenzyloxyimino) (cyclopentyl) methyl], [BC3334; 1- (2,5-difluorobenzyloxyimino) (cyclopentyl) methyl], [BC3335; 1- (2,6-) Difluorobenzyloxyimino) (cyclopentyl) methyl], [BC3336; 1- (3,4-difluorobenzyloxyimino) (cyclopentyl) methyl], [BC3337; 1- (3,5-difluorobenzyloxyimino) (cyclopentyl) Methyl], [BC3338; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (cyclopentyl) methyl], [BC3339; 1- (3-ethylbenzene] Dihydroxyimino) (cyclopentyl) methyl], [BC3340; 1- (4-ethylbenzyloxyimino) (cyclopentyl) methyl], [BC3341; 1- (2-trifluoromethoxybenzyloxyimino) (cyclopentyl) methyl], [BC 3342; 1- (3-trifluoromethoxybenzyloxyimino) (cyclopentyl) methyl], [BC 3343; 1- (4-trifluoromethoxybenzyloxyimino) (cyclopentyl) methyl], [BC 3344; 1- (methoxyimino) 1) (Cyclopentyl) methyl], [BC3345; 1- (ethoxyimino) (cyclohexyl) methyl], [BC3346; 1-(propoxyimino) (cyclohexyl) methyl], [BC 3347; 1-(n-butoxyimino) (cyclohexyl) ) Methyl], [BC3348; 1- (pentyloxyimino) (cyclohexyl) methyl], [BC3349; 1- (hexyloxyimino) (cyclohexyl) Methyl], [BC3350; 1- (isopropoxyimino) (cyclohexyl) methyl], [BC3351; 1- (tert-butoxyimino) (cyclohexyl) methyl], [BC3352; 1- (sec-butoxyimino) (cyclohexyl) Methyl], [BC3353; 1- (cyclopropyloxyimino) (cyclohexyl) methyl], [BC3354; 1- (cyclopentyloxyimino) (cyclohexyl) methyl], [BC3355; 1- (cyclohexyloxyimino) (cyclohexyl) Methyl], [BC3356; 1- (3-allyloxyimino) (cyclohexyl) methyl], [BC3357; 1- (3-butenyloxyimino) (cyclohexyl) methyl], [BC3358; 1- (2-propynyloxy) Imino) (cyclohexyl) methyl], [BC3359; 1- (3-butynyloxyimino) (cyclohexyl) methyl], [BC3360; 1- (1-cyclohexyloxyimino) (cyclohexene) Methyl), [BC3361; 1- (2,2,2-trifluoroethoxyimino) (cyclohexyl) methyl], [BC3362; 1- (benzyloxyimino) (cyclohexyl) methyl], [BC3363; 1- ( 2-Fluorobenzyloxyimino) (cyclohexyl) methyl], [BC3364; 1- (3-fluorobenzyloxyimino) (cyclohexyl) methyl], [BC3365; 1- (4-fluorobenzyloxyimino) (cyclohexyl) methyl] , [BC3366; 1- (2-chlorobenzyloxyimino) (cyclohexyl) methyl], [BC3367; 1- (3-chlorobenzyloxyimino) (cyclohexyl) methyl], [BC3368; 1- (4-chlorobenzyloxy) Imino) (cyclohexyl) methyl], [BC3369; 1- (2-methylbenzyloxyimino) (cyclohexyl) methyl], [BC3370; 1- (3-methylbenzyloxyimino) (cyclohexy] ) Methyl], [BC3371; 1- (4-methylbenzyloxyimino) (cyclohexyl) methyl], [BC3372; 1- (2-cyanobenzyloxyimino) (cyclohexyl) methyl], [BC3373; 1- (3-) Cyanobenzyloxyimino) (cyclohexyl) methyl], [BC3374; 1- (4-cyanobenzyloxyimino) (cyclohexyl) methyl], [BC3375; 1- (2-trifluoromethylbenzyloxyimino) (cyclohexyl) methyl] , [BC3376; 1- (3-trifluoromethylbenzyloxyimino) (cyclohexyl) methyl], [BC3377; 1- (4-trifluoromethylbenzyloxyimino) (cyclohexyl) methyl], [BC3 378; 1- (2) -Difluoromethylbenzyloxyimino) (cyclohexyl) methyl], [BC 3379; 1- (3-difluoromethylbenzyloxyimino) (cyclohexyl) methyl],

[BC 3380; 1- (4-difluoromethylbenzyloxyimino) (cyclohexyl) methyl], [BC3381; 1- (2-methoxybenzyloxyimino) (cyclohexyl) methyl], [BC3382; 1- (3-methoxybenzyloxy) Imino) (cyclohexyl) methyl], [BC 3383; 1- (4-methoxybenzyloxyimino) (cyclohexyl) methyl], [BC 3384; 1- (2-vinylbenzyloxyimino) (cyclohexyl) methyl], [BC 3385; 1 -(3-vinylbenzyloxyimino) (cyclohexyl) methyl], [BC3386; 1- (4-vinylbenzyloxyimino) (cyclohexyl) methyl], [BC3387; 1- (2-phenylbenzyloxyimino) (cyclohexyl) Methyl], [BC3388; 1- (3-phenylbenzyloxyimino) (cyclohexyl) methyl], [BC3389; 1- (4-phenylbenzyloxyimino) (cyclohexene) Xyl) methyl], [BC3390; 1- (2,3-difluorobenzyloxyimino) (cyclohexyl) methyl], [BC3391; 1- (2,4-difluorobenzyloxyimino) (cyclohexyl) methyl], [BC3392; 1- (2,5-difluorobenzyloxyimino) (cyclohexyl) methyl], [BC3393; 1- (2,6-difluorobenzyloxyimino) (cyclohexyl) methyl], [BC3394; 1- (3,4-difluoro) Benzyloxyimino) (cyclohexyl) methyl], [BC3395; 1- (3,5-difluorobenzyloxyimino) (cyclohexyl) methyl], [BC3396; 1- (2,3,4,5,6-pentafluorobenzyl) Oxyimino) (cyclohexyl) methyl], [BC 3397; 1- (3-ethylbenzyloxyimino) (cyclohexyl) methyl], [BC3398; 1- (4-ethylbenzyloxyimino) (cyclohexyl) Sil) methyl], [BC3399; 1- (2-trifluoromethoxybenzyloxyimino) (cyclohexyl) methyl], [BC3400; 1- (3-trifluoromethoxybenzyloxyimino) (cyclohexyl) methyl], [BC3401; 1- (4-trifluoromethoxybenzyloxyimino) (cyclohexyl) methyl], [BC3402; 1- (methoxyimino) (cyclohexyl) methyl], [BC3403; 1- (ethoxyimino) (1-cyclohexenyl) methyl] , [BC3404; 1- (propoxyimino) (1-cyclohexenyl) methyl], [BC3405; 1- (n-butoxyimino) (1-cyclohexenyl) methyl], [BC3406; 1- (pentyloxyimino) ( 1-cyclohexenyl) methyl], [BC3407; 1- (hexyloxyimino) (1-cyclohexenyl) methyl], [BC3408; 1- (isopropoxyimino) (1-cyclohexenyl) methyl], [BC3 3409; 1- (tert-butoxyimino) (1-cyclohexenyl) methyl], [BC 3410; 1- (sec-butoxyimino) (1-cyclohexenyl) methyl], [BC3411; 1- (cyclopropyloxyimino) (1-cyclohexenyl) methyl], [BC 3412; 1- (cyclopentyloxyimino) (1-cyclohexenyl) methyl], [BC 3413; 1- (cyclohexyloxyimino) (1-cyclohexenyl) methyl], [BC3414] 1- (3-allyloxyimino) (1-cyclohexenyl) methyl], [BC3415; 1- (3-butenyloxyimino) (1-cyclohexenyl) methyl], [BC3416; 1- (2-propynyl) Oxyimino) (1-cyclohexenyl) methyl], [BC3417; 1- (3-butynyloxyimino) (1-cyclohexenyl) methyl], [BC3418; 1- (1-cyclohexyloxyimino) (1-cyclo Hexenyl) methyl], [BC 3419; 1- (2,2,2-trifluoroethoxyimino) (1-cyclohexenyl) methyl], [BC3420; 1- (benzyloxyimino) (1-cyclohexenyl) methyl], [BC3421; 1- (2-fluorobenzyl) Oxyimino) (1-cyclohexenyl) methyl], [BC 3422; 1- (3-fluorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3423; 1- (4-fluorobenzyloxyimino) (1-) Cyclohexenyl) methyl], [BC3424; 1- (2-chlorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC3425; 1- (3-chlorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3426; 1- (4-chlorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3427; 1- (2-methylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3428; 1- ( 3-methylbenzyloxy Mino) (1-cyclohexenyl) methyl], [BC3429; 1- (4-methylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3430; 1- (2-cyanobenzyloxyimino) (1-cyclo) Hexenyl) methyl], [BC 3431; 1- (3-cyanobenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3432; 1- (4-cyanobenzyloxyimino) (1-cyclohexenyl) methyl], [BC BC 3433; 1- (2-trifluoromethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3434; 1- (3-trifluoromethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3435; 1- (4-trifluoromethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3436; 1- (2-difluoromethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3437; 3- Giff Omethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3438; 1- (4-difluoromethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3439; 1- (2-methoxybenzyloxyimino) ) (1-Cyclohexenyl) methyl], [BC3440; 1- (3-methoxybenzyloxyimino) (1-cyclohexenyl) methyl], [BC3441; 1- (4-methoxybenzyloxyimino) (1-cyclohexenyl) 1) (2-vinylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3443; 1- (3-vinylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3444) 1- (4-vinylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3445; 1- (2-phenylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3446; 1- (3-) Phenyl Benzyloxyimino) (1-cyclohexenyl) methyl], [BC3447; 1- (4-phenylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3448; 1- (2,3-difluorobenzyloxyimino) (1-Cyclohexenyl) methyl], [BC3449; 1- (2,4-difluorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC3450; 1- (2,5-difluorobenzyloxyimino) (1) -Cyclohexenyl) methyl], [BC3451; 1- (2,6-difluorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC3452; 1- (3,4-difluorobenzyloxyimino) (1-cyclo Hexenyl) methyl], [BC 3453; 1- (3,5-difluorobenzyloxyimino) (1-cyclohexenyl) methyl], [BC3454; 1- (2,3,4,5,6-pentafluorobenzyloxyimino] ) (1- Chlorohexenyl) methyl], [BC3455; 1- (3-ethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3456; 1- (4-ethylbenzyloxyimino) (1-cyclohexenyl) methyl], [BC3457; 1- (2-trifluoromethoxybenzyloxyimino) (1-cyclohexenyl) methyl], [BC3458; 1- (3-trifluoromethoxybenzyloxyimino) (1-cyclohexenyl) methyl], [BC3459 1- (4-trifluoromethoxybenzyloxyimino) (1-cyclohexenyl) methyl], [BC 3460; 1- (methoxyimino) (1-cyclohexenyl) methyl], [BC3461; 1- (ethoxyimino) ( Phenyl) methyl], [BC3462; 1- (propoxyimino) (phenyl) methyl], [BC3463; 1- (n-butoxyimino) (phenyl) methyl], [BC3464; 1- (pentyloxyimino) (phenyl) Methyl ], [BC3465; 1- (hexyloxyimino) (phenyl) methyl], [BC3466; 1- (isopropoxyimino) (phenyl) methyl], [BC3467; 1- (tert-butoxyimino) (phenyl) methyl] , [BC 3468; 1- (sec-butoxyimino) (phenyl) methyl], [BC 3469; 1-(cyclopropyloxyimino) (phenyl) methyl], [BC 3 470; 1-(cyclopentyloxyimino) (phenyl) methyl 1- (Cyclohexyloxyimino) (phenyl) methyl], [BC3472; 1- (3-allyloxyimino) (phenyl) methyl], [BC3473; 1- (3-butenyloxyimino) ( Phenyl) methyl], [BC3474; 1- (2-propynyloxyimino) (phenyl) methyl], [BC3475; 1- (3-butynyloxyimino) (phenyl) methyl], [BC3476; 1- (1-) Cyclohexyloxyimino) (phenyl) methyl], [BC 3477; 1- 2,2,2-trifluoroethoxyimino) (phenyl) methyl], [BC3478; 1- (benzyloxyimino) (phenyl) methyl], [BC3479; 1- (2-fluorobenzyloxyimino) (phenyl) methyl ],

[BC 3480; 1- (4-fluorobenzyloxyimino) (phenyl) methyl], [BC3481; 1- (2-chlorobenzyloxyimino) (phenyl) methyl], [BC3482; 1- (3-chlorobenzyloxyimino] 1) (phenyl) methyl], [BC3483; 1- (4-chlorobenzyloxyimino) (phenyl) methyl], [BC3484; 1- (2-methylbenzyloxyimino) (phenyl) methyl], [BC3485; (3-Methylbenzyloxyimino) (phenyl) methyl], [BC3486; 1- (4-methylbenzyloxyimino) (phenyl) methyl], [BC3487; 1- (2-cyanobenzyloxyimino) (phenyl) methyl 1- (3-cyanobenzyloxyimino) (phenyl) methyl], [BC3489; 1- (4-cyanobenzyloxyimino) (phenyl) methyl], [BC3490; 1- (2-trifluoro) Methyl benzyl oxyimino) (phenyl) Methyl], [BC3491; 1- (3-trifluoromethylbenzyloxyimino) (phenyl) methyl], [BC3492; 1- (4-trifluoromethylbenzyloxyimino) (phenyl) methyl], [BC3493; 1- (2-Difluoromethylbenzyloxyimino) (phenyl) methyl], [BC3494; 1- (3-difluoromethylbenzyloxyimino) (phenyl) methyl], [BC3495; 1- (4-difluoromethylbenzyloxyimino) ( Phenyl) methyl], [BC3496; 1- (2-methoxybenzyloxyimino) (phenyl) methyl], [BC3497; 1- (3-methoxybenzyloxyimino) (phenyl) methyl], [BC3498; 1- (4) -Methoxybenzyloxyimino) (phenyl) methyl], [BC3499; 1- (2-vinylbenzyloxyimino) (phenyl) methyl], [BC3500; 1- (3-vinylbenzyloxyimino) (phenyl) methyl] , [BC3501; 1- (4-vinylbenzyloxyimino) (phenyl) methyl], [BC3502; 1- (2-phenylbenzyloxyimino) (phenyl) methyl], [BC3503; 1- (3-phenylbenzyloxy) Imino) (phenyl) methyl], [BC3504; 1- (4-phenylbenzyloxyimino) (phenyl) methyl], [BC3505; 1- (2,3-difluorobenzyloxyimino) (phenyl) methyl], [BC3506 1- (2,4-difluorobenzyloxyimino) (phenyl) methyl], [BC3507; 1- (2,5-difluorobenzyloxyimino) (phenyl) methyl], [BC3508; 1- (2, 6-) Difluorobenzyloxyimino) (phenyl) methyl], [BC3509; 1- (3,4-difluorobenzyloxyimino) (phenyl) methyl], [BC 3510; 1- (3,5-difluorobenzyloxyimino) (phenyl) Methyl], [BC 3511; 1- (2 1,3,4,5,6-pentafluorobenzyloxyimino) (phenyl) methyl], [BC 3512; 1- (3-ethylbenzyloxyimino) (phenyl) methyl], [BC 3513; 1- (4-ethyl benzyl] Oxyimino) (phenyl) methyl], [BC 3514; 1- (2-trifluoromethoxybenzyloxyimino) (phenyl) methyl], [BC 3515; 1- (3-trifluoromethoxybenzyloxyimino) (phenyl) methyl] , [BC3516; 1- (4-trifluoromethoxybenzyloxyimino) (phenyl) methyl], [BC3517; 1- (methoxyimino) (phenyl) methyl], [BC3518; 1- (ethoxyimino) (2-chlorophenyl) 1) (propoxyimino) (2-chlorophenyl) methyl], [BC 3520; 1-(n-butoxyimino) (2- chlorophenyl) methyl], [BC 3521; 1-(pentyloxyimino) (2- black Lophenyl) methyl], [BC3522; 1- (hexyloxyimino) (2-chlorophenyl) methyl], [BC3523; 1- (isopropoxyimino) (2-chlorophenyl) methyl], [BC3524; 1- (tert-butoxy) Imino) (2-chlorophenyl) methyl], [BC3525; 1- (sec-butoxyimino) (2-chlorophenyl) methyl], [BC3526; 1- (cyclopropyloxyimino) (2-chlorophenyl) methyl], [BC3527 1- (cyclopentyloxyimino) (2-chlorophenyl) methyl], [BC3528; 1- (cyclohexyloxyimino) (2-chlorophenyl) methyl], [BC3529; 1- (3-allyloxyimino) (2-) Chlorophenyl) methyl], [BC3530; 1- (3-butenyloxyimino) (2-chlorophenyl) methyl], [BC3531; 1- (2-propynyloxyimino) (2-chlorophenyl) methyl], [BC3532; 1 -(3- Roxyimino) (2-chlorophenyl) methyl], [BC 3533; 1- (1-cyclohexyloxyimino) (2-chlorophenyl) methyl], [BC 3534; 1- (2,2,2-trifluoroethoxyimino) (2-) Chlorophenyl) methyl], [BC3535; 1- (benzyloxyimino) (2-chlorophenyl) methyl], [BC3536; 1- (2-fluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3537; 3-Fluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3538; 1- (4-fluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3539; 1- (2-chlorobenzyloxyimino) ( 2-chlorophenyl) methyl], [BC3540; 1- (3-chlorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3541; 1- (4-chlorobenzyloxyimino) (2-chlorophenyl) methyl ], [BC3542; 1- (2-methylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3543; 1- (3-methylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3544; 4-Methylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3545; 1- (2-cyanobenzyloxyimino) (2-chlorophenyl) methyl], [BC3546; 1- (3-cyanobenzyloxyimino) ( 2-chlorophenyl) methyl], [BC3547; 1- (4-cyanobenzyloxyimino) (2-chlorophenyl) methyl], [BC3548; 1- (2-trifluoromethylbenzyloxyimino) (2-chlorophenyl) methyl] , [BC3549; 1- (3-trifluoromethylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3550; 1- (4-trifluoromethylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3551; 1- ( -Difluoromethylbenzyloxyimino) (2-chlorophenyl) methyl], [BC 3552; 1- (3-difluoromethylbenzyloxyimino) (2-chlorophenyl) methyl], [BC 3553; 1- (4-difluoromethylbenzyloxyimino] ) (2-chlorophenyl) methyl], [BC3554; 1- (2-methoxybenzyloxyimino) (2-chlorophenyl) methyl], [BC3555; 1- (3-methoxybenzyloxyimino) (2-chlorophenyl) methyl] , [BC3556; 1- (2,5-difluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3557; 1- (4-methoxybenzyloxyimino) (2-chlorophenyl) methyl], [BC3558; 1- (2,6-difluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC 3559; 1- (2-vinylbenzyloxyimino) (2-chlorophenyl) methyl], [BC 3560; 1- (3,4-Difluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3561; 1- (3-vinylbenzyloroxyimino) (2-chlorophenyl) methyl], [BC3562; 1- (3,5-) Difluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC 3563; 1- (4-vinylbenzyloxyimino) (2-chlorophenyl) methyl], [BC 3564; 1- (2,3,4,5,6-) Pentafluorobenzyloxyimino) (2-chlorophenyl) methyl], [BC3565; 1- (2-phenylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3566; 1- (3-ethylbenzyloxyimino) (2) -Chlorophenyl) methyl], [BC3567; 1- (3-phenylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3568; 1- (4-ethylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3569 1- ( -Phenylbenzyloxyimino) (2-chlorophenyl) methyl], [BC3570; 1- (2-trifluoromethoxybenzyloxyimino) (2-chlorophenyl) methyl], [BC3571; 1- (2,3-difluorobenzyloxy) Imino) (2-chlorophenyl) methyl], [BC3572; 1- (3-trifluoromethoxybenzyloxyimino) (2-chlorophenyl) methyl], [BC3573; 1- (2,4-difluorobenzyloxyimino) (2) -Chlorophenyl) methyl], [BC3574; 1- (4-trifluoromethoxybenzyloxyimino) (2-chlorophenyl) methyl], [BC3575; 1- (methoxyimino) (2-chlorophenyl) methyl], [BC3576; 1 -(Ethoxyimino) (3-chlorophenyl) methyl], [BC 3577; 1- (propoxyimino) (3-chlorophenyl) methyl], [BC 3578; 1- (n-butoxyimino) (3-chlorophenyl) Henyl) methyl], [BC 3579; 1- (pentyloxyimino) (3-chlorophenyl) methyl],

[BC 3 580; 1- (Hexyloxyimino) (3-chlorophenyl) methyl], [BC3581; 1- (Isopropoxyimino) (3-chlorophenyl) methyl], [BC3582; 1- (tert-butoxyimino) (3-) Chlorophenyl) methyl], [BC 3583; 1- (sec-butoxyimino) (3-chlorophenyl) methyl], [BC 3584; 1- (cyclopropyloxyimino) (3-chlorophenyl) methyl], [BC 3585; 1- (cyclo) Pentyloxyimino) (3-chlorophenyl) methyl], [BC3586; 1- (cyclohexyloxyimino) (3-chlorophenyl) methyl], [BC3587; 1- (3-allyloxyimino) (3-chlorophenyl) methyl], [BC 3588; 1- (3-butenyloxyimino) (3-chlorophenyl) methyl], [BC3589; 1- (2-propynyloxyimino) (3-chlorophenyl) methyl], [BC3590; 1- (3-butyl] Nyloxyimino) ( -Chlorophenyl) methyl], [BC 3591; 1- (1-cyclohexyloxyimino) (3-chlorophenyl) methyl], [BC 3592; 1- (2,2,2-trifluoroethoxyimino) (3-chlorophenyl) methyl] , [BC3593; 1- (benzyloxyimino) (3-chlorophenyl) methyl], [BC3594; 1- (2-fluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3595; 1- (3-fluorobenzyl) Oxyimino) (3-chlorophenyl) methyl], [BC 3596; 1- (4-fluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC 3597; 1- (2-chlorobenzyloxyimino) (3-chlorophenyl) Methyl], [BC3598; 1- (3-chlorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3599; 1- (4-chlorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3600; 1- (2-Methyl Benzyloxyimino) (3-chlorophenyl) methyl], [BC 3601; 1- (3-methylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3602; 1- (4-methylbenzyloxyimino) (3-chlorophenyl) 1) (2-cyanobenzyloxyimino) (3-chlorophenyl) methyl], [BC 3604; 1-(3-cyanobenzyloxyimino) (3-chlorophenyl) methyl], [BC 3605; 1) -(4-Cyanobenzyloxyimino) (3-chlorophenyl) methyl], [BC3606; 1- (2-trifluoromethylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3607; 1- (3-trifluoro) Methylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3608; 1- (4-trifluoromethylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3609; 1- (2-difluoromethyl bene] 1- (3-Difluoromethylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3611; 1- (4-difluoromethylbenzyloxyimino) (b-hydroxyimino) (3-chlorophenyl) methyl], [BC 3610; 3-chlorophenyl) methyl], [BC 3612; 1- (2-methoxybenzyloxyimino) (3-chlorophenyl) methyl], [BC 3613; 1- (3-methoxybenzyloxyimino) (3-chlorophenyl) methyl], [BC BC 3614; 1- (4-methoxybenzyloxyimino) (3-chlorophenyl) methyl], [BC3615; 1- (2-vinylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3616; 1- (3-vinyl] Benzyloxyimino) (3-chlorophenyl) methyl], [BC3617; 1- (4-vinylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3618; 1- (2-phenylbenzyloxyimino) 3-chlorophenyl) methyl], [BC3619; 1- (3-phenylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3620; 1- (4-phenylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3620; BC 3621; 1- (2,3-difluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3622; 1- (2,4-difluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3623; 1- (2,5-difluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3624; 1- (2,6-difluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3625; 1- (3,4 -Difluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3626; 1- (3,5-difluorobenzyloxyimino) (3-chlorophenyl) methyl], [BC3627; 1- (2,3,4,5] , 6- Pentafu Orobenzyloxyimino) (3-chlorophenyl) methyl], [BC3628; 1- (3-ethylbenzyloxyimino) (3-chlorophenyl) methyl], [BC3629; 1- (4-ethylbenzyloxyimino) (3-) Chlorophenyl) methyl], [BC3630; 1- (2-trifluoromethoxybenzyloxyimino) (3-chlorophenyl) methyl], [BC3631; 1- (3-trifluoromethoxybenzyloxyimino) (3-chlorophenyl) methyl] , [BC3632; 1- (4-trifluoromethoxybenzyloxyimino) (3-chlorophenyl) methyl], [BC3633; 1- (methoxyimino) (3-chlorophenyl) methyl], [BC3634; 1- (ethoxyimino) (4-chlorophenyl) methyl], [BC3635; 1- (propoxyimino) (4-chlorophenyl) methyl], [BC3636; 1- (n-butoxyimino) (4-chlorophenyl) methyl], [BC3637; -(Pentyloxyimino) (4-chlorophenyl) methyl], [BC3638; 1- (hexyloxyimino) (4-chlorophenyl) methyl], [BC3639; 1- (isopropoxyimino) (4-chlorophenyl) methyl], [BC 3640; 1- (tert-butoxyimino) (4-chlorophenyl) methyl], [BC3641; 1- (sec-butoxyimino) (4-chlorophenyl) methyl], [BC3642; 1- (cyclopropyloxyimino) ( 4-chlorophenyl) methyl], [BC3643; 1- (cyclopentyloxyimino) (4-chlorophenyl) methyl], [BC3644; 1- (cyclohexyloxyimino) (4-chlorophenyl) methyl], [BC3645; 3-Allyloxyimino) (4-chlorophenyl) methyl], [BC3646; 1- (3-butenyloxyimino) (4-chlorophenyl) methyl], [BC3647; 1- (2-propynyloxyimino) (4-) Chlorophyll 1- (3-butynyloxyimino) (4-chlorophenyl) methyl], [BC3649; 1- (1-cyclohexyloxyimino) (4-chlorophenyl) methyl], [BC3650;) (4-chlorophenyl) methyl], [BC3651; 1- (benzyloxyimino) (4-chlorophenyl) methyl], [BC3652; 1- (2-fluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC3653; 1- (3-Fluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC3654; 1- (4-fluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC3655; 1- (2-chlorobenzyloxy) Imino) (4-chlorophenyl) methyl], [BC3656; 1- (3-chlorobenzyloxyimino) (4-chlorophenyl) methyl], [BC3657; 1- (4-chlorobenzyloxyimino) (4-chlorophenyl) methyl ], [BC3658; 1- (2-methylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3659; 1- (3-methylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3660; 1- (4-methylbenzyloxy) Imino) (4-chlorophenyl) methyl], [BC3661; 1- (2-cyanobenzyloxyimino) (4-chlorophenyl) methyl], [BC3662; 1- (3-cyanobenzyloxyimino) (4-chlorophenyl) methyl 1- (4-cyanobenzyloxyimino) (4-chlorophenyl) methyl], [BC3664; 1- (2-trifluoromethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3665; 1] -(3-Trifluoromethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3666; 1- (4-trifluoromethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3667; 1- (2- Giff Omethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC 3668; 1- (3-difluoromethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC 3669; 1- (4-difluoromethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3670; 1- (2-methoxybenzyloxyimino) (4-chlorophenyl) methyl], [BC3671; 1- (3-methoxybenzyloxyimino) (4-chlorophenyl) methyl], [BC 3672; 1- (4-methoxybenzyloxyimino) (4-chlorophenyl) methyl], [BC 3673; 1-(2-vinylbenzyloxyimino) (4- chlorophenyl) methyl], [BC 3674; Vinylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3675; 1- (4-vinylbenzyloxyimino) (4-chlorophenyl) methyl], [BC3676; 1- (2-phenylbenzylo) Ximino) (4-chlorophenyl) methyl], [BC 3677; 1- (3-phenylbenzyloxyimino) (4-chlorophenyl) methyl], [BC 3678; 1- (4-phenylbenzyloxyimino) (4-chlorophenyl) methyl ], [BC 3679; 1- (2,3-difluorobenzyloxyimino) (4-chlorophenyl) methyl],

[BC 3680; 1- (2,4-difluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC 3681; 1-(2, 5-difluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC 3682; 1 -(2,6-difluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC3683; 1- (3,4-difluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC3684; 1- (3, 5-Difluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC 3685; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (4-chlorophenyl) methyl], [BC 3686; 1- (3-ethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC 3687; 1- (4-ethylbenzyloxyimino) (4-chlorophenyl) methyl], [BC 3688; 1- (2-trifluoromethoxybenzyloxy) Imino (4-chlorophenyl) methyl], [BC3689; 1- (3-trifluoromethoxybenzyloxyimino) (4-chlorophenyl) methyl], [BC3690; 1- (4-trifluoromethoxybenzyloxyimino) (4-chlorophenyl) 1) (methoxyimino) (4-chlorophenyl) methyl], [BC 369 2; 1- (ethoxyimino) (2-fluorophenyl) methyl], [BC 369 3; 1- (propoxyimino) (2) -Fluorophenyl) methyl], [BC3694; 1- (n-butoxyimino) (2-fluorophenyl) methyl], [BC3695; 1- (pentyloxyimino) (2-fluorophenyl) methyl], [BC3696; 1 -(Hexyloxyimino) (2-fluorophenyl) methyl], [BC3697; 1- (isopropoxyimino) (2-fluorophenyl) methyl], [BC3698; 1- (tert-butoxyimino) (2-fluorophenyl) ) Ethyl, [BC3699; 1- (sec-butoxyimino) (2-fluorophenyl) methyl], [BC3700; 1- (cyclopropyloxyimino) (2-fluorophenyl) methyl], [BC3701; 1- (cyclo) Pentyloxyimino) (2-fluorophenyl) methyl], [BC 3702; 1- (cyclohexyloxyimino) (2-fluorophenyl) methyl], [BC 3703; 1- (3-allyloxyimino) (2-fluorophenyl) Methyl], [BC3704; 1- (3-butenyloxyimino) (2-fluorophenyl) methyl], [BC3705; 1- (2-propynyloxyimino) (2-fluorophenyl) methyl], [BC3706; 1 -(3-butynyloxyimino) (2-fluorophenyl) methyl], [BC3707; 1- (1-cyclohexyloxyimino) (2-fluorophenyl) methyl], [BC3708; 1- (2,2,2 -Trifluoroethoxyimino) (2-fluorofe Nyl) methyl], [BC3709; 1- (benzyloxyimino) (2-fluorophenyl) methyl], [BC3710; 1- (2-fluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC3711; -(3-Fluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC 3712; 1- (4-fluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC 3713; 1- (2-chlorobenzyl) Oxyimino) (2-fluorophenyl) methyl], [BC3714; 1- (3-chlorobenzyloxyimino) (2-fluorophenyl) methyl], [BC3715; 1- (4-chlorobenzyloxyimino) (2-) Fluorophenyl) methyl], [BC3716; 1- (2-methylbenzyloxyimino) (2-fluorophenyl) methyl], [BC3717; 1- (3-methylbenzyloxyimino) (2-fluorophenyl) methyl], [BC 3718; 1- (4-methyl (2-fluorophenyl) methyl], [BC3719; 1- (2-cyanobenzyloxyimino) (2-fluorophenyl) methyl], [BC3720; 1- (3-cyanobenzyloxyimino) ( 2-Fluorophenyl) methyl], [BC3721; 1- (4-cyanobenzyloxyimino) (2-fluorophenyl) methyl], [BC3722; 1- (2-trifluoromethylbenzyloxyimino) (2-fluorophenyl) ) Methyl], [BC 3723; 1- (3-trifluoromethylbenzyloxyimino) (2-fluorophenyl) methyl], [BC 3724; 1-(4- trifluoromethylbenzyloxyimino) (2- fluorophenyl) methyl ], [BC 3725; 1- (2-difluoromethylbenzyloxyimino) (2-fluorophenyl) methyl], [BC3726; 1- (3-difluoromethylbenzyloxyimino) (2-fluorophenyl) me Ethyl, [BC3727; 1- (4-difluoromethylbenzyloxyimino) (2-fluorophenyl) methyl], [BC3728; 1- (2-methoxybenzyloxyimino) (2-fluorophenyl) methyl], [BC3729] 1- (3-methoxybenzyloxyimino) (2-fluorophenyl) methyl], [BC3730; 1- (4-methoxybenzyloxyimino) (2-fluorophenyl) methyl], [BC3731; 1- (2-) Vinylbenzyloxyimino) (2-fluorophenyl) methyl], [BC 3732; 1- (3-vinylbenzyloxyimino) (2-fluorophenyl) methyl], [BC 3 733; 1- (4-vinylbenzyloxyimino) ( 2-Fluorophenyl) methyl], [BC3734; 1- (2-phenylbenzyloxyimino) (2-fluorophenyl) methyl], [BC3735; 1- (3-phenylbenzyloxyimino) (2-fluorophenyl) methyl ], [BC3736; 1- (4-phenylbenzyloxyimino) (2-fluorophenyl) methyl], [BC3737; 1- (2,3-difluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC3738; 1- (2) , 4-Difluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC 3739; 1- (2,5-difluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC 3740; 1- (2, 6) -Difluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC 3741; 1- (3,4-difluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC 3742; 1- (3,5-difluoro) Benzyloxyimino) (2-fluorophenyl) methyl], [BC 3743; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (2-fluorophenyl) methyl], [BC3744; 3-ethyl benzyloxy Imino) (2-fluorophenyl) methyl], [BC3745; 1- (4-ethylbenzyloxyimino) (2-fluorophenyl) methyl], [BC3746; 1- (2-trifluoromethoxybenzyloxyimino) (2) -Fluorophenyl) methyl], [BC3747; 1- (3-trifluoromethoxybenzyloxyimino) (2-fluorophenyl) methyl], [BC3748; 1- (4-trifluoromethoxybenzyloxyimino) (2-fluoro) Phenyl) methyl], [BC3749; 1- (methoxyimino) (2-fluorophenyl) methyl], [BC3750; 1- (ethoxyimino) (3-fluorophenyl) methyl], [BC3751; 1- (propoxyimino) (3-fluorophenyl) methyl], [BC3752; 1- (n-butoxyimino) (3-fluorophenyl) methyl], [BC3753; 1- (pentyloxyimino) (3-fluorophenyl) methyl], [BC3754 1- (F Siloxyimino) (3-fluorophenyl) methyl], [BC3755; 1- (isopropoxyimino) (3-fluorophenyl) methyl], [BC3756; 1- (tert-butoxyimino) (3-fluorophenyl) methyl ], [BC 3757; 1- (sec-butoxyimino) (3-fluorophenyl) methyl], [BC 3758; 1-(cyclopropyloxyimino) (3- fluorophenyl) methyl], [BC 3759; 1-(cyclopenty) Roxyimino) (3-fluorophenyl) methyl], [BC3760; 1- (cyclohexyloxyimino) (3-fluorophenyl) methyl], [BC3761; 1- (3-allyloxyimino) (3-fluorophenyl) methyl 1- (3-Butenyloxyimino) (3-fluorophenyl) methyl], [BC3763; 1- (2-propynyloxyimino) (3-fluorophenyl) methyl], [BC3764; 1- (3-butynyloxyimi B) (3-fluorophenyl) methyl], [BC3765; 1- (1-cyclohexyloxyimino) (3-fluorophenyl) methyl], [BC3766; 1- (2,2,2-trifluoroethoxyimino) ( 3-Fluorophenyl) methyl], [BC3767; 1- (benzyloxyimino) (3-fluorophenyl) methyl], [BC3768; 1- (2-fluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3768; BC 3769; 1- (3-fluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3770; 1- (4-fluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3771; 1- (2) -Chlorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3772; 1- (3-chlorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3773; 1- (4-chlorobenzyloxyimino) (3-fluorophenyl Methyl], [BC3774; 1- (2-methylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3775; 1- (3-methylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3776; 1- (4-methylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3777; 1- (2-cyanobenzyloxyimino) (3-fluorophenyl) methyl], [BC3778; 1- (3-cyano) Benzyloxyimino) (3-fluorophenyl) methyl], [BC3779; 1- (4-cyanobenzyloxyimino) (3-fluorophenyl) methyl],

[BC 3780; 1- (2-trifluoromethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC 3781; 1- (3-trifluoromethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC 3782 1- (4-trifluoromethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC 3783; 1- (2-difluoromethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3784; 1- (3-Difluoromethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3785; 1- (4-difluoromethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3786; 1- (2-methoxy) Benzyloxyimino) (3-fluorophenyl) methyl], [BC 3787; 1- (3-methoxybenzyloxyimino) (3-fluorophenyl) methyl], [BC 3788; 1- (4-methoxybenzyl) Siimino) (3-fluorophenyl) methyl], [BC3789; 1- (2-vinylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3790; 1- (3-vinylbenzyloxyimino) (3-fluoro Phenyl) methyl], [BC 3791; 1- (4-vinylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3792; 1- (2-phenylbenzyloxyimino) (3-fluorophenyl) methyl], [BC792] BC 3793; 1- (3-phenylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3794; 1- (4-phenylbenzyloxyimino) (3-fluorophenyl) methyl], [BC3795; 1- (2) , 3-Difluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC 3796; 1- (2,4-difluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC 3797; 1- (2,5 -Difluorobenzylo Siimino) (3-fluorophenyl) methyl], [BC 3798; 1- (2,6-difluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC 3799; 1- (3,4-difluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3800; 1- (3,5-difluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC3801; 1- (2,3,4,5,6-penta) Fluorobenzyloxyimino) (3-fluorophenyl) methyl], [BC 3802; 1- (3-ethylbenzyloxyimino) (3-fluorophenyl) methyl], [BC 3803; 1- (4-ethylbenzyloxyimino) ( 3-Fluorophenyl) methyl], [BC3804; 1- (2-trifluoromethoxybenzyloxyimino) (3-fluorophenyl) methyl], [BC3805; 1- (3-trifluoromethoxybenzyloxyimino) (3-) Fluorof 1- (4-trifluoromethoxybenzyloxyimino) (3-fluorophenyl) methyl], [BC3807; 1- (methoxyimino) (3-fluorophenyl) methyl], [BC3808; 1- (Ethoxyimino) (4-fluorophenyl) methyl], [BC3809; 1- (propoxyimino) (4-fluorophenyl) methyl], [BC3810; 1- (n-butoxyimino) (4-fluorophenyl) Methyl], [BC3811; 1- (pentyloxyimino) (4-fluorophenyl) methyl], [BC3812; 1- (hexyloxyimino) (4-fluorophenyl) methyl], [BC3813; 1- (isopropoxyimino) ) (4-fluorophenyl) methyl], [BC3814; 1- (tert-butoxyimino) (4-fluorophenyl) methyl], [BC3815; 1- (sec-butoxyimino) (4-fluorophenyl) methyl], [BC 3816; 1- (cyclopropyl) Ximino) (4-fluorophenyl) methyl], [BC3817; 1- (cyclopentyloxyimino) (4-fluorophenyl) methyl], [BC3818; 1- (cyclohexyloxyimino) (4-fluorophenyl) methyl], [BC 3819; 1- (3-allyloxyimino) (4-fluorophenyl) methyl], [BC3820; 1- (3-butenyloxyimino) (4-fluorophenyl) methyl], [BC 3821; 1- (2) -Propynyloxyimino) (4-fluorophenyl) methyl], [BC3822; 1- (3-butynyloxyimino) (4-fluorophenyl) methyl], [BC3823; 1- (1-cyclohexyloxyimino) (4) -Fluorophenyl) methyl], [BC3824; 1- (2,2,2-trifluoroethoxyimino) (4-fluorophenyl) methyl], [BC3825; 1- (benzyloxyimino) (4-fluorophenyl) methyl ], [BC 3826; 1- (2-full Lobenzyloxyimino) (4-fluorophenyl) methyl], [BC3827; 1- (3-fluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3828; 1- (4-fluorobenzyloxyimino) ( 4-Fluorophenyl) methyl], [BC3829; 1- (2-chlorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3830; 1- (3-chlorobenzyloxyimino) (4-fluorophenyl) methyl 1- (4-chlorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3832; 1- (2-methylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3833; 1] -(3-Methylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3834; 1- (4-methylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3835; 1- (2-cyanobenzyl) Oximino) 4-Fluorophenyl) methyl], [BC3836; 1- (3-cyanobenzyloxyimino) (4-fluorophenyl) methyl], [BC3837; 1- (4-cyanobenzyloxyimino) (4-fluorophenyl) methyl 1- (2-trifluoromethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC 3839; 1- (3-trifluoromethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC 3840; 1- (4-trifluoromethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3841; 1- (2-difluoromethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3842; 1- (3-difluoromethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3843; 1- (4-difluoromethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3844; -(2-methoxybenzyloxyimino) (4-fluorophenyl) methyl], [BC3845; 1- (3-methoxybenzyloxyimino) (4-fluorophenyl) methyl], [BC3846; 1- (4-methoxybenzyl) Oxyimino) (4-fluorophenyl) methyl], [BC3847; 1- (2-vinylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3848; 1- (3-vinylbenzyloxyimino) (4-) Fluorophenyl) methyl], [BC 3849; 1- (4-vinylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3850; 1- (2-phenylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3851; 1- (3-phenylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3852; 1- (4-phenylbenzyloxyimino) (4-fluorophenyl) methyl], [BC3853; 2,3-difluo Benzyloxyimino) (4-fluorophenyl) methyl (4-fluorophenyl) methyl], [BC 3854; 1- (2,4-difluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC 3855; 2,5-Difluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3856; 1- (2,6-difluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3857; 1- (3, 4-difluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3858; 1- (3,5-difluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC3859; 1- (2,3,3 4,5,6-pentafluorobenzyloxyimino) (4-fluorophenyl) methyl], [BC 3860; 1- (3-ethylbenzyloxyimino) (4-fluorophenyl) methyl], [BC 386 1; 1- (4) -Ethyl benzyl Oximino) (4-fluorophenyl) methyl], [BC3862; 1- (2-trifluoromethoxybenzyloxyimino) (4-fluorophenyl) methyl], [BC3863; 1- (3-trifluoromethoxybenzyloxyimino) (4-fluorophenyl) methyl], [BC3864; 1- (4-trifluoromethoxybenzyloxyimino) (4-fluorophenyl) methyl], [BC3865; 1- (methoxyimino) (4-fluorophenyl) methyl] , [BC3866; 1- (ethoxyimino) (4-fluorophenyl) methyl], [BC 3867; 1- (propoxyimino) (2-bromophenyl) methyl], [BC3868; 1- (n-butoxyimino) (2 -Bromophenyl) methyl], [BC 3869; 1- (pentyloxyimino) (2-bromophenyl) methyl], [BC3870; 1- (hexyloxyimino) (2-bromophenyl) methyl], [BC 3871; 1- (Isopropoki Imino) (2-bromophenyl) methyl], [BC3872; 1- (tert-butoxyimino) (2-bromophenyl) methyl], [BC3873; 1- (sec-butoxyimino) (2-bromophenyl) methyl] , [BC3874; 1- (cyclopropyloxyimino) (2-bromophenyl) methyl], [BC3875; 1- (cyclopentyloxyimino) (2-bromophenyl) methyl], [BC3876; 1- (cyclohexyloxyimino) ) (2-bromophenyl) methyl], [BC3877; 1- (3-allyloxyimino) (2-bromophenyl) methyl], [BC3878; 1- (3-butenyloxyimino) (2-bromophenyl) Methyl], [BC 3879; 1- (2-propynyloxyimino) (2-bromophenyl) methyl],

[BC 3 880; 1- (3-butynyloxyimino) (2-bromophenyl) methyl], [BC 3881; 1- (1-cyclohexyloxyimino) (2-bromophenyl) methyl], [BC 3882; 1- (2) , 2,2-trifluoroethoxyimino) (2-bromophenyl) methyl], [BC 3883; 1- (benzyloxyimino) (2-bromophenyl) methyl], [BC 3884; 1- (2-fluorobenzyloxyimino) ) (2-bromophenyl) methyl], [BC3885; 1- (3-fluorobenzyloxyimino) (2-bromophenyl) methyl], [BC3886; 1- (4-fluorobenzyloxyimino) (2-bromophenyl) ) Methyl], [BC 3887; 1- (2-chlorobenzyloxyimino) (2-bromophenyl) methyl], [BC 3888; 1-(3-chlorobenzyloxyimino) (2-bromophenyl) methyl], [BC 3889] 1- (4-chlorobenzyloxyimino) (2-b Mophenyl) methyl], [BC3890; 1- (2-methylbenzyloxyimino) (2-bromophenyl) methyl], [BC3891; 1- (3-methylbenzyloxyimino) (2-bromophenyl) methyl], BC3892; 1- (4-methylbenzyloxyimino) (2-bromophenyl) methyl], [BC3893; 1- (2-cyanobenzyloxyimino) (2-bromophenyl) methyl], [BC3894; 1- (3) -Cyanobenzyloxyimino) (2-bromophenyl) methyl], [BC3895; 1- (4-cyanobenzyloxyimino) (2-bromophenyl) methyl], [BC3896; 1- (2-trifluoromethylbenzyloxy) Imino) (2-bromophenyl) methyl], [BC3897; 1- (3-trifluoromethylbenzyloxyimino) (2-bromophenyl) methyl], [BC3898; 1- (4-trifluoromethylbenzyloxyimino) (2-bromophenyl Methyl], [BC3899; 1- (2-difluoromethylbenzyloxyimino) (2-bromophenyl) methyl], [BC3900; 1- (3-difluoromethylbenzyloxyimino) (2-bromophenyl) methyl], [BC3900; BC3901; 1- (4-difluoromethylbenzyloxyimino) (2-bromophenyl) methyl], [BC3902; 1- (2-methoxybenzyloxyimino) (2-bromophenyl) methyl], [BC3903; 3-methoxybenzyloxyimino) (2-bromophenyl) methyl], [BC3904; 1- (4-methoxybenzyloxyimino) (2-bromophenyl) methyl], [BC3905; 1- (2-vinylbenzyloxyimino) ) (2-bromophenyl) methyl], [BC3906; 1- (3-vinylbenzyloxyimino) (2-bromophenyl) methyl], [BC3907; 1- (4-vinylbenzyloxyimino) (2-bromophenyl) ) Methyl], [BC3908 1- (2-phenylbenzyloxyimino) (2-bromophenyl) methyl], [BC3909; 1- (3-phenylbenzyloxyimino) (2-bromophenyl) methyl], [BC3910; Phenylbenzyloxyimino) (2-bromophenyl) methyl], [BC 3911; 1- (2,3-difluorobenzyloxyimino) (2-bromophenyl) methyl], [BC3912; 1- (2,4-difluorobenzyl) Oxyimino) (2-bromophenyl) methyl], [BC3913; 1- (2,5-difluorobenzyloxyimino) (2-bromophenyl) methyl], [BC3914; 1- (2,6-difluorobenzyloxyimino] ) (2-bromophenyl) methyl], [BC3915; 1- (3,4-difluorobenzyloxyimino) (2-bromophenyl) methyl], [BC3916; 1- (3,5-difluorobenzyloxyimino) ( 2-bromophenyl) methyl] , [BC 3917; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (2-bromophenyl) methyl], [BC3918; 1- (3-ethylbenzyloxyimino) (2-bromophenyl) 1) (meth) methyl], [BC3919; 1- (4-ethylbenzyloxyimino) (2-bromophenyl) methyl], [BC 3920; 1-(2-trifluoromethoxybenzyloxyimino) (2-bromophenyl) methyl], [BC 3921; 1- (3-trifluoromethoxybenzyloxyimino) (2-bromophenyl) methyl], [BC3922; 1- (4-trifluoromethoxybenzyloxyimino) (2-bromophenyl) methyl], [BC3923 1- (methoxyimino) (2-bromophenyl) methyl], [BC3924; 1- (ethoxyimino) (3-bromophenyl) methyl], [BC3925; 1- (propoxyimino) (3-bromophenyl) methyl ], [BC 3926; 1- (n-butoxyi B) (3-bromophenyl) methyl], [BC3 927; 1- (pentyloxyimino) (3-bromophenyl) methyl], [BC3928; 1- (hexyloxyimino) (3-bromophenyl) methyl], [BC3928; BC 3929; 1- (Isopropoxyimino) (3-bromophenyl) methyl], [BC 3930; 1- (tert-butoxyimino) (3-bromophenyl) methyl], [BC 3931; 1- (sec-butoxyimino) ( 3-bromophenyl) methyl], [BC3932; 1- (cyclopropyloxyimino) (3-bromophenyl) methyl], [BC3933; 1- (cyclopentyloxyimino) (3-bromophenyl) methyl], [BC3934 1- (cyclohexyloxyimino) (3-bromophenyl) methyl], [BC 3935; 1- (3-allyloxyimino) (3-bromophenyl) methyl], [BC3936; 1- (3-butenyloxyimino] ) (3-bromophenyl) methyl], [BC 3937; 1- (2) -Propynyloxyimino) (3-bromophenyl) methyl], [BC 3938; 1- (3-butynyloxyimino) (3-bromophenyl) methyl], [BC 3939; 1- (1-cyclohexyloxyimino) (3) -Bromophenyl) methyl], [BC3940; 1- (2,2,2-trifluoroethoxyimino) (3-bromophenyl) methyl], [BC3941; 1- (benzyloxyimino) (3-bromophenyl) methyl 1- (2-fluorobenzyloxyimino) (3-bromophenyl) methyl], [BC3943; 1- (3-fluorobenzyloxyimino) (3-bromophenyl) methyl], [BC3944; 1] -(4-Fluorobenzyloxyimino) (3-bromophenyl) methyl], [BC3945; 1- (2-chlorobenzyloxyimino) (3-bromophenyl) methyl], [BC3946; 1- (3-chlorobenzyl) Oximino) (3-bromophenyl) Ethyl, [BC 3947; 1- (4-chlorobenzyloxyimino) (3-bromophenyl) methyl], [BC 3948; 1- (2-methylbenzyloxyimino) (3-bromophenyl) methyl], [BC 3949; 1- (3-methylbenzyloxyimino) (3-bromophenyl) methyl], [BC3950; 1- (4-methylbenzyloxyimino) (3-bromophenyl) methyl], [BC3951; 1- (2-cyano) Benzyloxyimino) (3-bromophenyl) methyl], [BC3952; 1- (3-cyanobenzyloxyimino) (3-bromophenyl) methyl], [BC3953; 1- (4-cyanobenzyloxyimino) (3 -Bromophenyl) methyl], [BC 3954; 1- (2-trifluoromethylbenzyloxyimino) (3-bromophenyl) methyl], [BC 3955; 1- (3-trifluoromethylbenzyloxyimino) (3-bromo Phenyl) methyl], [BC 3956; 1- (4-trif Luomethylbenzyloxyimino) (3-bromophenyl) methyl], [BC3957; 1- (2-difluoromethylbenzyloxyimino) (3-bromophenyl) methyl], [BC3958; 1- (3-difluoromethylbenzyl] Oxyimino) (3-bromophenyl) methyl], [BC3959; 1- (4-difluoromethylbenzyloxyimino) (3-bromophenyl) methyl], [BC3960; 1- (2-methoxybenzyloxyimino) (3) -Bromophenyl) methyl], [BC3961; 1- (3-methoxybenzyloxyimino) (3-bromophenyl) methyl], [BC3962; 1- (4-methoxybenzyloxyimino) (3-bromophenyl) methyl] , [BC3963; 1- (2-vinylbenzyloxyimino) (3-bromophenyl) methyl], [BC3964; 1- (3-vinylbenzyloxyimino) (3-bromophenyl) methyl], [BC3965; 1- (4-vinyl [(3-bromophenyl) methyl], [BC3966; 1- (2-phenylbenzyloxyimino) (3-bromophenyl) methyl], [BC3967; 1- (3-phenylbenzyloxyimino) ( 3-bromophenyl) methyl], [BC 3968; 1- (4-phenylbenzyloxyimino) (3-bromophenyl) methyl], [BC3969; 1- (2,3-difluorobenzyloxyimino) (3-bromophenyl] ) Methyl], [BC 3 970; 1- (2,4-difluorobenzyloxyimino) (3-bromophenyl) methyl], [BC 3971; 1-(2, 5-difluorobenzyloxyimino) (3-bromophenyl) methyl 1- (2,6-difluorobenzyloxyimino) (3-bromophenyl) methyl], [BC3973; 1- (3,4-difluorobenzyloxyimino) (3-bromophenyl) methyl], [BC 3 974; 1- (3,5- dif Orobenzyloxyimino) (3-bromophenyl) methyl], [BC3975; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (3-bromophenyl) methyl], [BC3976; 1- (3-ethylbenzyloxyimino) (3-bromophenyl) methyl], [BC 3977; 1- (4-ethylbenzyloxyimino) (3-bromophenyl) methyl], [BC 3978; 1- (2-trifluoromethoxy) Benzyloxyimino) (3-bromophenyl) methyl], [BC 3979; 1- (3-trifluoromethoxybenzyloxyimino) (3-bromophenyl) methyl],

[BC 3 980; 1- (4-trifluoromethoxybenzyloxyimino) (3-bromophenyl) methyl], [BC 3981; 1- (methoxyimino) (3-bromophenyl) methyl], [BC 3982; 1- (ethoxyimino) ) (4-bromophenyl) methyl], [BC 3983; 1- (propoxyimino) (4-bromophenyl) methyl], [BC 3984; 1-(n-butoxyimino) (4-bromophenyl) methyl], [BC 3985 1- (pentyloxyimino) (4-bromophenyl) methyl], [BC 3986; 1- (hexyloxyimino) (4-bromophenyl) methyl], [BC3987; 1- (isopropoxyimino) (4-bromo; Phenyl) methyl], [BC 3988; 1- (tert-butoxyimino) (4-bromophenyl) methyl], [BC 3989; 1- (sec-butoxyimino) (4-bromophenyl) methyl], [BC 3990; 1- (Cyclopropyloxyimino) (4-bromophenyl) Ethyl, [BC3991; 1- (cyclopentyloxyimino) (4-bromophenyl) methyl], [BC3992; 1- (cyclohexyloxyimino) (4-bromophenyl) methyl], [BC3993; 1- (3- Allyloxyimino) (4-bromophenyl) methyl], [BC 3994; 1- (3-butenyloxyimino) (4-bromophenyl) methyl], [BC 3995; 1- (2-propynyloxyimino) (4-) Bromophenyl) methyl], [BC 3996; 1- (3-butynyloxyimino) (4-bromophenyl) methyl], [BC3997; 1- (1-cyclohexyloxyimino) (4-bromophenyl) methyl], [BC BC 3998; 1- (2,2,2-trifluoroethoxyimino) (4-bromophenyl) methyl], [BC3999; 1- (benzyloxyimino) (4-bromophenyl) methyl], [BC4000; 2-Fluorobenzyloxyimino) (4-bromophenyl) methyl], [BC 4001; 1- (3-fluorobenzyloxyimino) (4-bromophenyl) methyl], [BC4002; 1- (4-fluorobenzyloxyimino) (4-bromophenyl) methyl], [BC4003; 1- (2) -Chlorobenzyloxyimino) (4-bromophenyl) methyl], [BC4004; 1- (3-chlorobenzyloxyimino) (4-bromophenyl) methyl], [BC4005; 1- (4-chlorobenzyloxyimino) (4-bromophenyl) methyl], [BC4006; 1- (2-methylbenzyloxyimino) (4-bromophenyl) methyl], [BC4007; 1- (3-methylbenzyloxyimino) (4-bromophenyl) Methyl], [BC4008; 1- (4-methylbenzyloxyimino) (4-bromophenyl) methyl], [BC4009; 1- (2-cyanobenzyloxyimino) (4-bromophenyl) methyl], [BC4010; 1- (3-cyanobenzyloxyimino) (4- Lomophenyl) methyl], [BC4011; 1- (4-cyanobenzyloxyimino) (4-bromophenyl) methyl], [BC4012; 1- (2-trifluoromethylbenzyloxyimino) (4-bromophenyl) methyl] [BC 4013; 1- (3-trifluoromethylbenzyloxyimino) (4-bromophenyl) methyl], [BC4014; 1- (4-trifluoromethylbenzyloxyimino) (4-bromophenyl) methyl], [BC4014; BC4015; 1- (2-difluoromethylbenzyloxyimino) (4-bromophenyl) methyl], [BC4016; 1- (3-difluoromethylbenzyloxyimino) (4-bromophenyl) methyl], [BC4017; 1- (4-Difluoromethylbenzyloxyimino) (4-bromophenyl) methyl], [BC4018; 1- (2-methoxybenzyloxyimino) (4-bromophenyl) methyl], [BC4019; 1- (3-methoxybenzyl) Oxyimino) (4-bromophenyl) methyl], [BC4020; 1- (4-methoxybenzyloxyimino) (4-bromophenyl) methyl], [BC4021; 1- (2-vinylbenzyloxyimino) (4-bromo) Phenyl) methyl], [BC4022; 1- (3-vinylbenzyloxyimino) (4-bromophenyl) methyl], [BC4023; 1- (4-vinylbenzyloxyimino) (4-bromophenyl) methyl], [BC4023; BC4024; 1- (2-phenylbenzyloxyimino) (4-bromophenyl) methyl], [BC4025; 1- (3-phenylbenzyloxyimino) (4-bromophenyl) methyl], [BC4026; 1- (4) -Phenylbenzyloxyimino) (4-bromophenyl) methyl], [BC4027; 1- (2,3-difluorobenzyloxyimino) (4-bromophenyl) methyl], [BC4028; 1- (2,4-difluoro) Benzyloxyimino) (4-bro Phenyl) methyl], [BC4029; 1- (2,5-difluorobenzyloxyimino) (4-bromophenyl) methyl], [BC4030; 1- (2,6-difluorobenzyloxyimino) (4-bromophenyl) Methyl], [BC4031; 1- (3,4-difluorobenzyloxyimino) (4-bromophenyl) methyl], [BC4032; 1- (3,5-difluorobenzyloxyimino) (4-bromophenyl) methyl] , [BC4033; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (4-bromophenyl) methyl], [BC4034; 1- (3-ethylbenzyloxyimino) (4-bromophenyl) ) Methyl], [BC 4035; 1- (4-ethylbenzyloxyimino) (4-bromophenyl) methyl], [BC 4036; 1-(2-trifluoromethoxybenzyloxyimino) (4-bromophenyl) methyl], [BC 4037; 1- (3-trifluorometh) Xybenzyloxyimino) (4-bromophenyl) methyl], [BC4038; 1- (4-trifluoromethoxybenzyloxyimino) (4-bromophenyl) methyl], [BC4039; 1- (methoxyimino) (4-) Bromophenyl) methyl], [BC 4040; 1- (ethoxyimino) (2-methylphenyl) methyl], [BC4041; 1- (propoxyimino) (2-methylphenyl) methyl], [BC4042; 1- (n-) Butoxyimino) (2-methylphenyl) methyl], [BC4043; 1- (pentyloxyimino) (2-methylphenyl) methyl], [BC4044; 1- (hexyloxyimino) (2-methylphenyl) methyl], [BC 4045; 1- (Isopropoxyimino) (2-methylphenyl) methyl], [BC 4046; 1-(tert-butoxyimino) (2-methylphenyl) methyl], [BC 4047; 1-(sec-butoxyimino) (2-methylphenyl) methyl], [BC4048; -(Cyclopropyloxyimino) (2-methylphenyl) methyl], [BC4049; 1- (cyclopentyloxyimino) (2-methylphenyl) methyl], [BC4050; 1- (cyclohexyloxyimino) (2-methyl Phenyl) methyl], [BC4051; 1- (3-allyloxyimino) (2-methylphenyl) methyl], [BC4052; 1- (3-butenyloxyimino) (2-methylphenyl) methyl], [BC4053 1- (2-propynyloxyimino) (2-methylphenyl) methyl], [BC4054; 1- (3-butynyloxyimino) (2-methylphenyl) methyl], [BC4055; 1- (1-cyclohexyl] Oxyimino) (2-methylphenyl) methyl], [BC 4056; 1- (2,2,2-trifluoroethoxyimino) (2-methylphenyl) methyl], [BC4057; 1- (benzyloxyimino) (2 -Methylphenyl) methyl], [BC 4058; 1- (2-fluo) Lobenzyloxyimino) (2-methylphenyl) methyl], [BC 4059; 1- (3-fluorobenzyloxyimino) (2-methylphenyl) methyl], [BC 4060; 1- (4-fluorobenzyloxyimino) ( 2-Methylphenyl) methyl], [BC4061; 1- (2-chlorobenzyloxyimino) (2-methylphenyl) methyl], [BC4062; 1- (3-chlorobenzyloxyimino) (2-methylphenyl) methyl 1- (4-chlorobenzyloxyimino) (2-methylphenyl) methyl], [BC4064; 1- (2-methylbenzyloxyimino) (2-methylphenyl) methyl], [BC4065; -(3-Methylbenzyloxyimino) (2-methylphenyl) methyl], [BC 4066; 1- (4-methylbenzyloxyimino) (2-methylphenyl) methyl], [BC 4067; 1- (2-cyanobenzyl) Oximino) (2-methylphenyl) Methyl], [BC4068; 1- (3-cyanobenzyloxyimino) (2-methylphenyl) methyl], [BC4069; 1- (4-cyanobenzyloxyimino) (2-methylphenyl) methyl], [BC4070; 1- (2-trifluoromethylbenzyloxyimino) (2-methylphenyl) methyl], [BC4071; 1- (3-trifluoromethylbenzyloxyimino) (2-methylphenyl) methyl], [BC4072; 1- (4-Trifluoromethylbenzyloxyimino) (2-methylphenyl) methyl], [BC 4073; 1- (2-difluoromethylbenzyloxyimino) (2-methylphenyl) methyl], [BC 4074; 1- (3- Difluoromethylbenzyloxyimino) (2-methylphenyl) methyl], [BC4075; 1- (4-difluoromethylbenzyloxyimino) (2-methylphenyl) methyl], [BC4076; 1- (2-methoxybenzyloxyimino) ) 2-Methylphenyl) methyl], [BC4077; 1- (3-methoxybenzyloxyimino) (2-methylphenyl) methyl], [BC4078; 1- (4-methoxybenzyloxyimino) (2-methylphenyl) methyl ], [BC 4079; 1- (2-vinylbenzyloxyimino) (2-methylphenyl) methyl],

[BC 4080; 1- (3-vinylbenzyloxyimino) (2-methylphenyl) methyl], [BC4081; 1- (4-vinylbenzyloxyimino) (2-methylphenyl) methyl], [BC4082; 2-phenylbenzyloxyimino) (2-methylphenyl) methyl], [BC4083; 1- (3-phenylbenzyloxyimino) (2-methylphenyl) methyl], [BC4084; 1- (4-phenylbenzyloxyimino) 1) (2-methylphenyl) methyl], [BC 4085; 1-(2,3-difluorobenzyloxyimino) (2-methylphenyl) methyl], [BC 4086; 1-(2,4-difluorobenzyloxyimino) ( 2-Methylphenyl) methyl], [BC4087; 1- (2,5-difluorobenzyloxyimino) (2-methylphenyl) methyl], [BC4088; 1- (2,6-difluorobenzyloxyimino) (2-) Methylphenyl) methyl], [BC 4089; 1- ( , 4-Difluorobenzyloxyimino) (2-methylphenyl) methyl], [BC 4090; 1- (3,5-difluorobenzyloxyimino) (2-methylphenyl) methyl], [BC4091; 1- (2,3 1,4,5,6-pentafluorobenzyloxyimino) (2-methylphenyl) methyl], [BC4092; 1- (3-ethylbenzyloxyimino) (2-methylphenyl) methyl], [BC4093; 4-ethylbenzyloxyimino) (2-methylphenyl) methyl], [BC 4094; 1- (2-trifluoromethoxybenzyloxyimino) (2-methylphenyl) methyl], [BC4095; 1- (3-trifluoro) Methoxybenzyloxyimino) (2-methylphenyl) methyl], [BC4096; 1- (4-trifluoromethoxybenzyloxyimino) (2-methylphenyl) methyl], [BC4097; 1- (methoxyimino) (2-) Methyl phenyl Methyl], [BC4098; 1- (ethoxyimino) (3-methylphenyl) methyl], [BC4099; 1- (propoxyimino) (3-methylphenyl) methyl], [BC4100; 1- (n-butoxyimino) (3-Methylphenyl) methyl], [BC4101; 1- (pentyloxyimino) (3-methylphenyl) methyl], [BC4102; 1- (hexyloxyimino) (3-methylphenyl) methyl], [BC4103; 1- (Isopropoxyimino) (3-methylphenyl) methyl], [BC4104; 1- (tert-butoxyimino) (3-methylphenyl) methyl], [BC4105; 1- (sec-butoxyimino) (3-) Methylphenyl) methyl], [BC4106; 1- (cyclopropyloxyimino) (3-methylphenyl) methyl], [BC4107; 1- (cyclopentyloxyimino) (3-methylphenyl) methyl], [BC4108; 1 -(Cyclohexyloxyimino) (3-methylphenyl) Ethyl, [BC4109; 1- (3-allyloxyimino) (3-methylphenyl) methyl], [BC4110; 1- (3-butenyloxyimino) (3-methylphenyl) methyl], [BC4111; 1 -(2-propynyloxyimino) (3-methylphenyl) methyl], [BC4112; 1- (3-butynyloxyimino) (3-methylphenyl) methyl], [BC4113; 1- (1-cyclohexyloxyimino) ) (3-Methylphenyl) methyl], [BC4114; 1- (2,2,2-trifluoroethoxyimino) (3-methylphenyl) methyl], [BC4115; 1- (benzyloxyimino) (3-methyl] Phenyl) methyl], [BC4116; 1- (2-fluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4117; 1- (3-fluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4117; BC 4118; 1- (4-fluorobenzyloxyimino) (3-methylpheny ) Methyl], [BC 4119; 1- (2-chlorobenzyloxyimino) (3-methylphenyl) methyl], [BC 4120; 1-(3-chlorobenzyloxyimino) (3-methylphenyl) methyl], [BC 4121 1- (4-chlorobenzyloxyimino) (3-methylphenyl) methyl], [BC4122; 1- (2-methylbenzyloxyimino) (3-methylphenyl) methyl], [BC4123; 1- (3-) Methylbenzyloxyimino) (3-methylphenyl) methyl], [BC4124; 1- (4-methylbenzyloxyimino) (3-methylphenyl) methyl], [BC4125; 1- (2-cyanobenzyloxyimino) ( 3-Methylphenyl) methyl], [BC4126; 1- (3-cyanobenzyloxyimino) (3-methylphenyl) methyl], [BC4127; 1- (4-cyanobenzyloxyimino) (3-methylphenyl) methyl ], [BC 4128; 1- (2-trifluoromethylbenzyl) Oxyimino) (3-methylphenyl) methyl], [BC4129; 1- (3-trifluoromethylbenzyloxyimino) (3-methylphenyl) methyl], [BC4130; 1- (4-trifluoromethylbenzyloxyimino) (3-Methylphenyl) methyl], [BC4131; 1- (2-difluoromethylbenzyloxyimino) (3-methylphenyl) methyl], [BC4132; 1- (3-difluoromethylbenzyloxyimino) (3-methyl] Phenyl) methyl], [BC4133; 1- (4-difluoromethylbenzyloxyimino) (3-methylphenyl) methyl], [BC4134; 1- (2-methoxybenzyloxyimino) (3-methylphenyl) methyl], [BC 4135; 1- (3-methoxybenzyloxyimino) (3-methylphenyl) methyl], [BC4136; 1- (4-methoxybenzyloxyimino) (3-methylphenyl) methyl], [BC4137; 2-bi Nylbenzyloxyimino) (3-methylphenyl) methyl], [BC4138; 1- (3-vinylbenzyloxyimino) (3-methylphenyl) methyl], [BC4139; 1- (4-vinylbenzyloxyimino) ( 3-Methylphenyl) methyl], [BC4140; 1- (2-phenylbenzyloxyimino) (3-methylphenyl) methyl], [BC4141; 1- (3-phenylbenzyloxyimino) (3-methylphenyl) methyl 1- (4-phenylbenzyloxyimino) (3-methylphenyl) methyl], [BC4143; 1- (2,3-difluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4144] 1- (2,4-difluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4145; 1- (2,5-difluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4146; 1; -(2,6-difluorobenzyl Xyimino) (3-methylphenyl) methyl], [BC4147; 1- (3,4-difluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4148; 1- (3,5-difluorobenzyloxyimino) (3-Methylphenyl) methyl], [BC4149; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (3-methylphenyl) methyl], [BC4150; 1- (3-ethylbenzyl) Oxyimino) (3-methylphenyl) methyl], [BC4151; 1- (4-ethylbenzyloxyimino) (3-methylphenyl) methyl], [BC4152; 1- (2-trifluoromethoxybenzyloxyimino) ( 3-methylphenyl) methyl], [BC 4153; 1- (3-trifluoromethoxybenzyloxyimino) (3-methylphenyl) methyl], [BC4154; 1- (4-trifluoromethoxybenzyloxyimino) (3-) Methylphenyl) Ethyl, [BC4155; 1- (methoxyimino) (3-methylphenyl) methyl], [BC4156; 1- (ethoxyimino) (4-methylphenyl) methyl], [BC4157; 1- (propoxyimino) (4) -Methylphenyl) methyl], [BC4158; 1- (n-butoxyimino) (4-methylphenyl) methyl], [BC4159; 1- (pentyloxyimino) (4-methylphenyl) methyl], [BC4160; 1 -(Hexyloxyimino) (4-methylphenyl) methyl], [BC4161; 1- (isopropoxyimino) (4-methylphenyl) methyl], [BC4162; 1- (tert-butoxyimino) (4-methylphenyl) 1) (meth) methyl], [BC 4163; 1- (sec-butoxyimino) (4-methylphenyl) methyl], [BC 4164; 1- (cyclopropyloxyimino) (4-methylphenyl) methyl], [BC 4165; Cyclopentyloxyimino) (4-methylphenyl) methyl], [BC 4166; -(Cyclohexyloxyimino) (4-methylphenyl) methyl], [BC4167; 1- (3-allyloxyimino) (4-methylphenyl) methyl], [BC4168; 1- (3-butenyloxyimino) ( 4-Methylphenyl) methyl], [BC4169; 1- (2-propynyloxyimino) (4-methylphenyl) methyl], [BC4170; 1- (3-butynyloxyimino) (4-methylphenyl) methyl] , [BC 4171; 1- (1-cyclohexyloxyimino) (4-methylphenyl) methyl], [BC 4172; 1- (2,2,2-trifluoroethoxyimino) (4-methylphenyl) methyl], [BC 4173 1- (benzyloxyimino) (4-methylphenyl) methyl], [BC 4174; 1- (2-fluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4175; 1- (3-fluorobenzyloxy) Imino) (4-methylphenyl) methyl], [BC 4176; 1- (4-Fluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4177; 1- (2-chlorobenzyloxyimino) (4-methylphenyl) methyl], [BC4178; 1- (3-chlorobenzyloxy) Imino) (4-methylphenyl) methyl], [BC 4179; 1- (4-chlorobenzyloxyimino) (4-methylphenyl) methyl],

[BC 4180; 1- (2-methylbenzyloxyimino) (4-methylphenyl) methyl], [BC4181; 1- (3-methylbenzyloxyimino) (4-methylphenyl) methyl], [BC4182; 4-Methylbenzyloxyimino) (4-methylphenyl) methyl], [BC4183; 1- (2-cyanobenzyloxyimino) (4-methylphenyl) methyl], [BC4184; 1- (3-cyanobenzyloxyimino] ) (4-Methylphenyl) methyl], [BC4185; 1- (4-cyanobenzyloxyimino) (4-methylphenyl) methyl], [BC4186; 1- (2-trifluoromethylbenzyloxyimino) (4-) Methylphenyl) methyl], [BC4187; 1- (3-trifluoromethylbenzyloxyimino) (4-methylphenyl) methyl], [BC4188; 1- (4-trifluoromethylbenzyloxyimino) (4-methylphenyl) ) Methyl], [BC 4189; 1- (2- Difluoromethylbenzyloxyimino) (4-methylphenyl) methyl], [BC4190; 1- (3-difluoromethylbenzyloxyimino) (4-methylphenyl) methyl], [BC4191; 1- (4-difluoromethylbenzyloxy) Imino) (4-methylphenyl) methyl], [BC4192; 1- (2-methoxybenzyloxyimino) (4-methylphenyl) methyl], [BC4193; 1- (3-methoxybenzyloxyimino) (4-methyl] Phenyl) methyl], [BC 4194; 1- (4-methoxybenzyloxyimino) (4-methylphenyl) methyl], [BC4195; 1- (2-vinylbenzyloxyimino) (4-methylphenyl) methyl], [BC4195; BC 4196; 1- (3-vinylbenzyloxyimino) (4-methylphenyl) methyl], [BC4197; 1- (4-vinylbenzyloxyimino) (4-methylphenyl) methyl], [BC4198; 1- (2) -Phenylben Roxyimino) (4-methylphenyl) methyl], [BC4199; 1- (3-phenylbenzyloxyimino) (4-methylphenyl) methyl], [BC4200; 1- (4-phenylbenzyloxyimino) (4-methyl] Phenyl) methyl], [BC4201; 1- (2,3-difluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4202; 1- (2,4-difluorobenzyloxyimino) (4-methylphenyl) Methyl], [BC 4203; 1- (2,5-difluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4204; 1- (2,6-difluorobenzyloxyimino) (4-methylphenyl) methyl] [BC 4205; 1- (3,4-difluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4206; 1- (3,5-difluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4205; BC 4207; 1- (2, 3, 4) , 5,6-pentafluorobenzyloxyimino) (4-methylphenyl) methyl], [BC4208; 1- (3-ethylbenzyloxyimino) (4-methylphenyl) methyl], [BC4209; 1- (4-) Ethylbenzyloxyimino) (4-methylphenyl) methyl], [BC 4210; 1- (2-trifluoromethoxybenzyloxyimino) (4-methylphenyl) methyl], [BC4211; 1- (3-trifluoromethoxybenzyl] Oxyimino) (4-methylphenyl) methyl], [BC 4212; 1- (4-trifluoromethoxybenzyloxyimino) (4-methylphenyl) methyl], [BC4213; 1- (methoxyimino) (4-methylphenyl) 1- (Ethoxyimino) (2-ethylphenyl) methyl], [BC4215; 1- (propoxyimino) (2-ethylphenyl) methyl], [BC4216; 1- (n-butoxyimino) ) (2-ethyl fe Methyl), [BC4217; 1- (pentyloxyimino) (2-ethylphenyl) methyl], [BC4218; 1- (hexyloxyimino) (2-ethylphenyl) methyl], [BC4219; 1- (iso) Propoxyimino) (2-ethylphenyl) methyl], [BC4220; 1- (tert-butoxyimino) (2-ethylphenyl) methyl], [BC4221; 1- (sec-butoxyimino) (2-ethylphenyl) methyl 1- (cyclopropyloxyimino) (2-ethylphenyl) methyl], [BC4223; 1- (cyclopentyloxyimino) (2-ethylphenyl) methyl], [BC4224; 1- (cyclohexyloxy) oxy] Imino) (2-ethylphenyl) methyl], [BC4225; 1- (3-allyloxyimino) (2-ethylphenyl) methyl], [BC4226; 1- (3-butenyloxyimino) (2-ethylphenyl) ) Methyl], [BC 4227; 1- (2-propynyloxy) B) (2-ethylphenyl) methyl], [BC 4228; 1- (3-butynyloxyimino) (2-ethylphenyl) methyl], [BC 4229; 1- (1-cyclohexyloxyimino) (2-ethylphenyl) ) Methyl], [BC 4230; 1- (2,2,2-trifluoroethoxyimino) (2-ethylphenyl) methyl], [BC4231; 1- (benzyloxyimino) (2-ethylphenyl) methyl], BC4232; 1- (2-fluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4233; 1- (3-fluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4234; 1- (4) -Fluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4235; 1- (2-chlorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4236; 1- (3-chlorobenzyloxyimino) (2-ethylphenyl) methyl], [BC 4237; 1- (4-q) Rolobenzyloxyimino) (2-ethylphenyl) methyl], [BC4238; 1- (2-methylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4239; 1- (3-methylbenzyloxyimino) ( 2-ethylphenyl) methyl], [BC4240; 1- (4-methylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4241; 1- (2-cyanobenzyloxyimino) (2-ethylphenyl) methyl 1- (3-cyanobenzyloxyimino) (2-ethylphenyl) methyl], [BC4243; 1- (4-cyanobenzyloxyimino) (2-ethylphenyl) methyl], [BC4244; 1] -(2-trifluoromethylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4245; 1- (3-trifluoromethylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4246; 4-trifluoromethylbenzyl Xyimino) (2-ethylphenyl) methyl], [BC4247; 1- (2-difluoromethylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4248; 1- (3-difluoromethylbenzyloxyimino) (2 -Ethylphenyl) methyl], [BC4249; 1- (4-difluoromethylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4250; 1- (2-methoxybenzyloxyimino) (2-ethylphenyl) methyl 1- (3-methoxybenzyloxyimino) (2-ethylphenyl) methyl], [BC4252; 1- (4-methoxybenzyloxyimino) (2-ethylphenyl) methyl], [BC4253; 1] -(2-vinylbenzyloxyimino) (2-ethylphenyl) methyl], [BC 4254; 1- (3-vinylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4255; 1- (4-vinylbenzyl) Oximino (2-ethylphenyl) methyl], [BC4256; 1- (2-phenylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4257; 1- (3-phenylbenzyloxyimino) (2-ethylphenyl) Methyl], [BC4258; 1- (4-phenylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4259; 1- (2,3-difluorobenzyloxyimino) (2-ethylphenyl) methyl], BC 4260; 1- (2,4-difluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4261; 1- (2,5-difluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4262; 1- (2,6-difluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4263; 1- (3,4-difluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4264; 1- (3,5-difluorobenzyloxyl Mino) (2-ethylphenyl) methyl], [BC4265; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (2-ethylphenyl) methyl], [BC4266; 1- (3- Ethylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4267; 1- (4-ethylbenzyloxyimino) (2-ethylphenyl) methyl], [BC4268; 1- (2-trifluoromethoxybenzyloxyimino] ) (2-Ethylphenyl) methyl], [BC4269; 1- (3-trifluoromethoxybenzyloxyimino) (2-ethylphenyl) methyl], [BC4270; 1- (4-trifluoromethoxybenzyloxyimino) ( 2-ethylphenyl) methyl], [BC4271; 1- (methoxyimino) (2-ethylphenyl) methyl], [BC4272; 1- (ethoxyimino) (3-ethylphenyl) methyl], [BC4273; Propoxyimino) (3-ethylphenyl ) 1- (n-Butoxyimino) (3-ethylphenyl) methyl], [BC4275; 1- (pentyloxyimino) (3-ethylphenyl) methyl], [BC4276; 1- (hexyl) Oxyimino) (3-ethylphenyl) methyl], [BC4277; 1- (isopropoxyimino) (3-ethylphenyl) methyl], [BC4278; 1- (tert-butoxyimino) (3-ethylphenyl) methyl] [BC 4279; 1- (sec-butoxyimino) (3-ethylphenyl) methyl],

[BC 4280; 1- (cyclopropyloxyimino) (3-ethylphenyl) methyl], [BC4281; 1- (cyclopentyloxyimino) (3-ethylphenyl) methyl], [BC4282; 1- (cyclohexyloxyimino) (3-ethylphenyl) methyl], [BC4283; 1- (3-allyloxyimino) (3-ethylphenyl) methyl], [BC4284; 1- (3-butenyloxyimino) (3-ethylphenyl) methyl 1- (2-propynyloxyimino) (3-ethylphenyl) methyl], [BC4286; 1- (3-butynyloxyimino) (3-ethylphenyl) methyl], [BC4287; 1- (1-Cyclohexyloxyimino) (3-ethylphenyl) methyl], [BC4288; 1- (2,2,2-trifluoroethoxyimino) (3-ethylphenyl) methyl], [BC4289; 1- (benzyloxy) Imino) (3-ethylphenyl) methyl], [BC 4290; 1- (2- Fluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4291; 1- (3-fluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4292; 1- (4-fluorobenzyloxyimino) ( 3-ethylphenyl) methyl], [BC4293; 1- (2-chlorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4294; 1- (3-chlorobenzyloxyimino) (3-ethylphenyl) methyl 1- (4-chlorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4296; 1- (2-methylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4297; 1] -(3-Methylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4298; 1- (4-methylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4299; 1- (2-cyanobenzyl) Oximino ((3-ethyl fe) 1- (3-cyanobenzyloxyimino) (3-ethylphenyl) methyl], [BC4301; 1- (4-cyanobenzyloxyimino) (3-ethylphenyl) methyl], [BC BC4302; 1- (2-trifluoromethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4303; 1- (3-trifluoromethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4304; 1- (4-trifluoromethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4305; 1- (2-difluoromethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4306; 3-Difluoromethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4307; 1- (4-difluoromethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4308; 1- (2-methoxybenzyl) Oxy B) (3-ethylphenyl) methyl], [BC 4309; 1- (3-methoxybenzyloxyimino) (3-ethylphenyl) methyl], [BC 4310; 1-(4-methoxybenzyloxyimino) (3-ethyl) Phenyl) methyl], [BC4311; 1- (2-vinylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4312; 1- (3-vinylbenzyloxyimino) (3-ethylphenyl) methyl], BC 4313; 1- (4-vinylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4314; 1- (2-phenylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4315; 1- (3) -Phenylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4316; 1- (4-phenylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4317; 1- (2,3-difluorobenzyloxy) Imino) (3-ethylphenyl) methi 1- (2,4-difluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4319; 1- (2,5-difluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC 4320; 1- (2,6-difluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4321; 1- (3,4-difluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4322 1- (3,5-difluorobenzyloxyimino) (3-ethylphenyl) methyl], [BC4323; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (3-ethylphenyl); Methyl], [BC4324; 1- (3-ethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4325; 1- (4-ethylbenzyloxyimino) (3-ethylphenyl) methyl], [BC4326; 1- (2-Trifluoromethoxybenzyloxyimi ) (3-ethylphenyl) methyl], [BC4327; 1- (3-trifluoromethoxybenzyloxyimino) (3-ethylphenyl) methyl], [BC4328; 1- (4-trifluoromethoxybenzyloxyimino) ( 3-ethylphenyl) methyl], [BC4329; 1- (methoxyimino) (3-ethylphenyl) methyl], [BC4330; 1- (ethoxyimino) (4-ethylphenyl) methyl], [BC4331; Propoxyimino) (4-ethylphenyl) methyl], [BC4332; 1- (n-butoxyimino) (4-ethylphenyl) methyl], [BC4333; 1- (pentyloxyimino) (4-ethylphenyl) methyl] , [BC4334; 1- (hexyloxyimino) (4-ethylphenyl) methyl], [BC4335; 1- (isopropoxyimino) (4-ethylphenyl) methyl], [BC4336; 1- (tert-butoxyimino) (4-ethylphenyl) methyl], [BC4337; -(Sec-butoxyimino) (4-ethylphenyl) methyl], [BC4338; 1- (cyclopropyloxyimino) (4-ethylphenyl) methyl], [BC4339; 1- (cyclopentyloxyimino) (4-) Ethylphenyl) methyl], [BC4340; 1- (cyclohexyloxyimino) (4-ethylphenyl) methyl], [BC4341; 1- (3-allyloxyimino) (4-ethylphenyl) methyl], [BC4342; 1 -(3-Butenyloxyimino) (4-ethylphenyl) methyl], [BC4343; 1- (2-propynyloxyimino) (4-ethylphenyl) methyl], [BC4344; 1- (3-butynyloxy) Imino) (4-ethylphenyl) methyl], [BC4345; 1- (1-cyclohexyloxyimino) (4-ethylphenyl) methyl], [BC4346; 1- (2,2,2-trifluoroethoxyimino) ( 4-ethylphenyl) methyl], [BC 4347; 1- (benzyl) Xyimino) (4-ethylphenyl) methyl], [BC 4348; 1- (2-fluorobenzyloxyimino) (4-ethylphenyl) methyl], [BC 4349; 1- (3-fluorobenzyloxyimino) (4-ethyl) Phenyl) methyl], [BC 4350; 1- (4-fluorobenzyloxyimino) (4-ethylphenyl) methyl], [BC 4351; 1- (2-chlorobenzyloxyimino) (4-ethylphenyl) methyl], [BC BC4352; 1- (3-chlorobenzyloxyimino) (4-ethylphenyl) methyl], [BC4353; 1- (4-chlorobenzyloxyimino) (4-ethylphenyl) methyl], [BC4354; 1- (2) -Methylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4355; 1- (3-methylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4356; 1- (4-methylbenzyloxyimino) (4-ethylphenyl) methyl], [B C4357; 1- (2-cyanobenzyloxyimino) (4-ethylphenyl) methyl], [BC4358; 1- (3-cyanobenzyloxyimino) (4-ethylphenyl) methyl], [BC4359; 1- (4) -Cyanobenzyloxyimino) (4-ethylphenyl) methyl], [BC4360; 1- (2-trifluoromethylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4361; 1- (3-trifluoromethyl) Benzyloxyimino) (4-ethylphenyl) methyl], [BC4362; 1- (4-trifluoromethylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4363; 1- (2-difluoromethylbenzyloxyimino] ) (4-Ethylphenyl) methyl], [BC 4364; 1- (3-Difluoromethylbenzyloxyimino) (4-ethylphenyl) methyl], [BC 4365; 1- (4-Difluoromethylbenzyloxyimino) (4-) ethyl 1- (2-methoxybenzyloxyimino) (4-ethylphenyl) methyl], [BC4367; 1- (3-methoxybenzyloxyimino) (4-ethylphenyl) methyl], [BC4366; BC 4368; 1- (4-methoxybenzyloxyimino) (4-ethylphenyl) methyl], [BC4369; 1- (2-vinylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4370; 1- (3) -Vinylbenzyloxyimino) (4-ethylphenyl) methyl], [BC 4371; 1- (4-vinylbenzyloxyimino) (4-ethylphenyl) methyl], [BC 4372; 1- (2-phenylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4373; 1- (3-phenylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4374; 1- (4-phenylbenzyloxyimino) (4-ethylphenyl) Methyl], [BC 4375; 1- (2,3- dif Fluorobenzyloxyimino) (4-ethylphenyl) methyl], [BC4376; 1- (2,4-difluorobenzyloxyimino) (4-ethylphenyl) methyl], [BC4377; 1- (2,5-difluoro] Benzyloxyimino) (4-ethylphenyl) methyl], [BC 4378; 1- (2,6-difluorobenzyloxyimino) (4-ethylphenyl) methyl], [BC 4379; 1- (3,4-difluorobenzyloxy) Imino) (4-ethylphenyl) methyl],

[BC 4380; 1- (3,5-difluorobenzyloxyimino) (4-ethylphenyl) methyl], [BC4381; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (4-ethyl] Phenyl) methyl], [BC4382; 1- (3-ethylbenzyloxyimino) (4-ethylphenyl) methyl], [BC4383; 1- (4-ethylbenzyloxyimino) (4-ethylphenyl) methyl], [BC BC 4384; 1- (2-trifluoromethoxybenzyloxyimino) (4-ethylphenyl) methyl], [BC4385; 1- (3-trifluoromethoxybenzyloxyimino) (4-ethylphenyl) methyl], [BC4386; 1- (4-Trifluoromethoxybenzyloxyimino) (4-ethylphenyl) methyl], [BC4387; 1- (methoxyimino) (4-ethylphenyl) methyl], [BC4388; 1- (ethoxyimino) [( 2-trifluoromethyl) fe [L] methyl], [BC 4 389; 1-(propoxy imino) [(2- trifluoromethyl) phenyl] methyl], [BC 4 390; 1-(n- butoxy imino) [(2- trifluoromethyl) phenyl] methyl] , [BC4391; 1- (pentyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4392; 1- (hexyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4393; 1- (Isopropoxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC 4394; 1- (tert-butoxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC 4395; sec-Butoxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC 4396; 1- (cyclopropyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC 4397; 1- (cyclopenty) Roxyimino) [(2- to Trifluoromethyl) phenyl] methyl], [BC 4398; 1- (cyclohexyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4399; 1- (3-allyloxyimino) [(2-trifluoro) Methyl) phenyl] methyl], [BC4400; 1- (3-butenyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4401; 1- (2-propynyloxyimino) [(2-triphenyl) methyl] Fluoromethyl) phenyl] methyl], [BC4402; 1- (3-butynyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4403; 1- (1-cyclohexyloxyimino) [(2-) Trifluoromethyl) phenyl] methyl], [BC4404; 1- (2,2,2-trifluoroethoxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4405; 1- (benzyloxyimino) [ (2-trifluoromethyl) 1) (2-Fluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4407; 1- (3-fluorobenzyloxyimino) [(2-triphenyl) methyl], [BC4406; Fluoromethyl) phenyl] methyl], [BC 4408; 1- (4-Fluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4409; 1- (2-chlorobenzyloxyimino) [(2 -Trifluoromethyl) phenyl] methyl], [BC 4410; 1- (3-chlorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4411; 1- (4-chlorobenzyloxyimino) [ (2-trifluoromethyl) phenyl] methyl], [BC 4412; 1- (2-methylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4413; 1- (3-methylbenzyloxyimino] ) [(2- Trifluoromethyl) phenyl] methyl], [BC4414; 1- (4-methylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4415; 1- (2-cyanobenzyloxyimino) [( 2-Trifluoromethyl) phenyl] methyl], [BC 4416; 1- (3-cyanobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4417; 1- (4-cyanobenzyloxyimino) [(2-Trifluoromethyl) phenyl] methyl], [BC4418; 1- (2-trifluoromethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4419; Fluoromethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC 4420; 1- (4-trifluoromethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [ BC 4421; 1- (2-difluoromethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4422; 1- (3-difluoromethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] Methyl], [BC 4423; 1- (4-difluoromethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4424; 1- (2-methoxybenzyloxyimino) [(2-trifluoromethyl) 1) (phenyl) methyl], [BC4425; 1- (3-methoxybenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4426; 1- (4-methoxybenzyloxyimino) [(2-tri) Fluoromethyl) phenyl] methyl], [BC4427; 1- (2-vinylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4428; 1- (3-vinylbenzyloxyimino] ) [(2-trifluoromethyl) phenyl] methyl], [BC4429; 1- (4-vinylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4430; 1- (2-phenylbenzyl) Oxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4431; 1- (3-phenylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4432; 1- (4-) Phenylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4433; 1- (2,3-difluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4434; 1 -(2,4-difluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4435; 1- (2,5-difluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] meth 1- (2,6-difluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4437; 1- (3,4-difluorobenzyloxyimino) [(2-tri) Fluoromethyl) phenyl] methyl], [BC4438; 1- (3,5-difluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4439; 1- (2,3,4,5, 6-pentafluorobenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4440; 1- (3-ethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4441; 1- (4-ethylbenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4442; 1- (2-trifluoromethoxybenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl] , [BC4443; 1- ( 3-trifluoromethoxybenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4444; 1- (4-trifluoromethoxybenzyloxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC 4445; 1- (methoxyimino) [(2-trifluoromethyl) phenyl] methyl], [BC4446; 1- (ethoxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4447; Propoxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC 4448; 1- (n-butoxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC 4449; 1- (pentyloxyimino) [(3-Trifluoromethyl) phenyl] methyl], [BC 4450; 1- (hexyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4451; 1- (isopropoxyimino) [(3- bird Fluoromethyl) phenyl] methyl], [BC4452; 1- (tert-butoxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4453; 1- (sec-butoxyimino) [(3-trifluoromethyl) ) Phenyl] methyl], [BC 4454; 1- (Cyclopropyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC 4455; 1- (Cyclopentyloxyimino) [(3-trifluoromethyl) phenyl 1- (Cyclohexyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4457; 1- (3-allyloxyimino) [(3-trifluoromethyl) phenyl] methyl 1- (3-Butenyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4459; 1- (2-propynyloxyimino) [(3-trifluoromethyl) phenyl] Methi 1- (3-butynyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4461; 1- (1-cyclohexyloxyimino) [(3-trifluoromethyl) phenyl] Methyl], [BC4462; 1- (2,2,2-trifluoroethoxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4463; 1- (benzyloxyimino) [(3-trifluoromethyl) 1) (2-Fluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4465; 1- (3-fluorobenzyloxyimino) [(3-triphenyl) methyl], [BC 4464; Fluoromethyl) phenyl] methyl], [BC4466; 1- (4-Fluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4467; 1- (2-chlorobenzyloxyimino) [(3 -Trifluoromethyl) [N-yl] methyl], [BC4468; 1- (3-chlorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4469; 1- (4-chlorobenzyloxyimino) [(3-trifluoro) Methyl) phenyl] methyl], [BC4470; 1- (2-methylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4471; 1- (3-methylbenzyloxyimino) [(3- Trifluoromethyl) phenyl] methyl], [BC4472; 1- (4-methylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4473; 1- (2-cyanobenzyloxyimino) [( 3-Trifluoromethyl) phenyl] methyl], [BC4474; 1- (3-cyanobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4475; 1- (4-cyanobenzyloxyimino) [(3-trifluoro Ethyl) phenyl] methyl], [BC 4476; 1- (2- trifluoromethyl benzyloxy imino) [(3- trifluoromethyl) phenyl] methyl], [BC 4477; 1-(3- trifluoromethyl benzyloxy imino) [(3-Trifluoromethyl) phenyl] methyl], [BC4478; 1- (4-trifluoromethylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4479; 1- (2-difluoro) Methylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl],

[BC 4480; 1- (3-difluoromethylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4481; 1- (4-difluoromethylbenzyloxyimino) [(3-trifluoromethyl) phenyl ] [Methyl], [BC4482; 1- (2-methoxybenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4483; 1- (3-methoxybenzyloxyimino) [(3-trifluoromethyl) 1) (phenyl) methyl], [BC4484; 1- (4-methoxybenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4485; 1- (2-vinylbenzyloxyimino) [(3-trile) Fluoromethyl) phenyl] methyl], [BC4486; 1- (3-vinylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4487; 1- (4-vinylbenzyloxyimino) [(3 - 1- (2-phenylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4489; 1- (3-phenylbenzyloxyimino) [(trifluoromethyl) phenyl] methyl], [BC4488; 3-Trifluoromethyl) phenyl] methyl], [BC 4490; 1- (4-phenylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4491; 1- (2,3-difluorobenzyloxy) Imino) [(3-trifluoromethyl) phenyl] methyl], [BC4492; 1- (2,4-difluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4493; 1- (2,5-difluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4494; 1- (2,6-difluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl ], [BC 4495; 1- (3,4-difluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4496; 1- (3,5-difluorobenzyloxyimino) [(3-trile) Fluoromethyl) phenyl] methyl], [BC 4497; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4498; 1- (3) -Ethylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4499; 1- (4-ethylbenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4500; 1- (2-Trifluoromethoxybenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4501; 1- (3-trifluoromethoxybenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl] , [BC45 02; 1- (4-trifluoromethoxybenzyloxyimino) [(3-trifluoromethyl) phenyl] methyl], [BC4503; 1- (methoxyimino) [(3-trifluoromethyl) phenyl] methyl], BC4504; 1- (Ethoxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4505; 1- (propoxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4506; 1- (n) -Butoxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4507; 1- (pentyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4508; 1- (hexyloxyimino) [(4-Trifluoromethyl) phenyl] methyl], [BC4509; 1- (isopropoxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4510; 1- (tert-butoxyimino) [(4 -Trifluoromethyl ) Phenyl] methyl], [BC 4511; 1- (sec-butoxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4512; 1- (cyclopropyloxyimino) [(4-trifluoromethyl) phenyl] 1- (cyclopentyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4514; 1- (cyclohexyloxyimino) [(4-trifluoromethyl) phenyl] methyl] , [BC 4515; 1- (3-allyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4516; 1- (3-butenyloxyimino) [(4-trifluoromethyl) phenyl] methyl 1- (2-propynyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4518; 1- (3-butynyloxyimino) [(4-trifluoromethyl) phenyl] Methyl], [BC 4519; 1- 1-Cyclohexyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC 4520; 1- (2,2,2-trifluoroethoxyimino) [(4-trifluoromethyl) phenyl] methyl], [ BC 4521; 1- (benzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4522; 1- (2-fluorobenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4523 1- (3-fluorobenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4524; 1- (4-fluorobenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC 4525; 1- (2-chlorobenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4526; 1- (3-chlorobenzyloxyimino) [(4-trifluoromethyl) phenyl] Ethyl, [BC4527; 1- (4-chlorobenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4528; 1- (2-methylbenzyloxyimino) [(4-trifluoromethyl) Phenyl] methyl], [BC4529; 1- (3-methylbenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4530; 1- (4-methylbenzyloxyimino) [(4-trifluoro) Methyl) phenyl] methyl], [BC 4531; 1- (2-cyanobenzyloxyimino) [(4-trifluoromethyl) phenyl] methyl], [BC4532; 1- (3-cyanobenzyloxyimino) [(4-) Trifluoromethyl) phenyl] methyl], [BC4533; 1- (4-cyanobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4534; 1- (2-trifluoromethylbenzyloxyimino) [ (2-difluoro Methyl) phenyl] methyl], [BC4535; 1- (3-trifluoromethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4536; 1- (4-trifluoromethylbenzyloxyimino) [ (2-Difluoromethyl) phenyl] methyl], [BC4537; 1- (2-difluoromethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4538; 1- (3-difluoromethylbenzyloxyimino] ) [(2-Difluoromethyl) phenyl] methyl], [BC4539; 1- (4-difluoromethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4540; 1- (2-methoxybenzyloxy) Imino) [(2-difluoromethyl) phenyl] methyl], [BC4541; 1- (3-methoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4542 1- (4-methoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4543; 1- (2-vinylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4544 1- (3-vinylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4545; 1- (4-vinylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4546; 1- (2-phenylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4547; 1- (3-phenylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4548; 1- (4-phenylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4549; 1- (2,3-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] Ethyl, [BC 4550; 1- (2,4-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4551; 1- (2,5-difluorobenzyloxyimino) [(2-difluoro) Methyl) phenyl] methyl], [BC4552; 1- (2,6-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4553; 1- (3,4-difluorobenzyloxyimino) [ (2-Difluoromethyl) phenyl] methyl], [BC4554; 1- (3,5-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4555; 1- (2,3,4,6 5,6-Pentafluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4556; 1- (3-ethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4557; 1- (4-Echi Benzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4558; 1- (2-trifluoromethoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4559; 1- (3) -Trifluoromethoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4560; 1- (4-trifluoromethoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4561; 1- (methoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4562; 1- (ethoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4563; 1- (propoxyimino) [ 2-Difluoromethyl) phenyl] methyl], [BC4564; 1- (n-butoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4565; 1- (pentyloxyimino) [ 2-Difluoromethyl) phenyl] methyl], [BC4566; 1- (hexyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4567; 1- (isopropoxyimino) [(2-difluoromethyl) phenyl 1- (tert-Butoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4569; 1- (sec-butoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4570; 1- (cyclopropyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4571; 1- (cyclopentyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4572; 1 -(Cyclohexyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4573; 1- (3-allyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4574; 1- (3- Bute Nyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4575; 1- (2-propynyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4576; 1- (3-butynyloxyimino] ) [(2-Difluoromethyl) phenyl] methyl], [BC 4577; 1- (1-cyclohexyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4578; 1- (2,2,2-tri) Fluoroethoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4579; 1- (benzyloxyimino) [(2-difluoromethyl) phenyl] methyl],

[BC 4580; 1- (2-fluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 451; 1- (3-fluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4582; 1- (4-fluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4583; 1- (2-chlorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4584; 1- (3-chlorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4585; 1- (4-chlorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4586; 1- (2-methylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4587; 1- (3-methylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl] , [BC4588; 1- (4-methylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4589; 1- (2-cyanobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl] , [BC 4590; 1- (3-cyanobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4591; 1- (4-cyanobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl] , [BC4592; 1- (2-trifluoromethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4593; 1- (3-trifluoromethylbenzyloxyimino) [(2-difluoromethyl) Phenyl] methyl], [BC 4594; 1- (4-trifluoromethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4595; 1- (2-difluoromethylbenzyloxyimino) (2-Difluoromethyl) phenyl] methyl], [BC 4596; 1- (3-difluoromethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4597; 1- (4-difluoromethylbenzyloxyimino] ) [(2-Difluoromethyl) phenyl] methyl], [BC 4598; 1- (2-methoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4599; 1- (3-methoxybenzyloxyimino] ) [(2-Difluoromethyl) phenyl] methyl], [BC4600; 1- (4-methoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4601; 1- (2-vinylbenzyloxyimino) ) [(2-difluoromethyl) phenyl] methyl], [BC4602; 1- (3-vinylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4603; 1- (4-vinylbenzene)] [(2-difluoromethyl) phenyl] methyl], [BC 4604; 1- (2-phenylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4605; 1- (3-) Phenylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4606; 1- (4-phenylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4607; 1- (2, 3-Difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4608; 1- (2,4-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4609; 1 -(2,5-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC 4610; 1- (2,6-difluorobenzyloxyimino) [(2-difluoromethyl) fe [L]-(3,4-difluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4612; 1- (3,5-difluorobenzyloxyimino) [(2 -Difluoromethyl) phenyl] methyl], [BC 4613; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4614; 1- (3) -Ethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4615; 1- (4-ethylbenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4616; 1- (2) -Trifluoromethoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4617; 1- (3-trifluoromethoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4618; 1- (4-Trifluoromethoxybenzyloxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4619; 1- (methoxyimino) [(2-difluoromethyl) phenyl] methyl], [BC4620; 1- (ethoxy) Imino) [(3-difluoromethyl) phenyl] methyl], [BC4621; 1- (propoxyimino [(3-difluoromethyl) phenyl] methyl], [BC4622; 1- (n-butoxyimino) [(3-difluoro) Methyl) phenyl] methyl], [BC 4623; 1- (pentyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4624; 1- (hexyloxyimino) [(3-difluoromethyl) phenyl] methyl] , [BC4625; 1- (isopropoxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4626; 1- (tert-butoxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4627 1- (sec-butoxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4628; 1- (cyclopropyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4629; Cyclopentyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4630; 1- (cyclohexyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4631; 1- (3-allyloxyimino] ) [(3-Difluoromethyl) phenyl] methyl], [BC4632; 1- (3-butenyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4633; 1- (2-propynyloxyimino) [(3-Difluoromethyl) phenyl] methyl], [BC4634; 1- (3-butynyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4635; 1- (1-cyclohexyloxyimino) [ (3-di Luomethyl) phenyl] methyl], [BC4636; 1- (2,2,2-trifluoroethoxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4637; 1- (benzyloxyimino) [(3- Difluoromethyl) phenyl] methyl], [BC 4638; 1- (2-fluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4639; 1- (3-fluorobenzyloxyimino) [(3-) Difluoromethyl) phenyl] methyl], [BC 4640; 1- (4-fluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4641; 1- (2-chlorobenzyloxyimino) [(3- Difluoromethyl) phenyl] methyl], [BC4642; 1- (3-chlorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4643; 1- (4-chlorobenzyloxyimino) [(3-) The Luomethyl) phenyl] methyl], [BC 4644; 1- (2-methylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4645; 1- (3-methylbenzyloxyimino) [(3-difluoro) Methyl) phenyl] methyl], [BC 4646; 1- (4-methylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4647; 1- (2-cyanobenzyloxyimino) [(3-difluoro) Methyl) phenyl] methyl], [BC 4648; 1- (3-cyanobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4649; 1- (4-cyanobenzyloxyimino) [(3-difluoro) Methyl) phenyl] methyl [(3-difluoromethyl) phenyl] methyl], [BC 4650; 1- (2-trifluoromethylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4 651; 1- (3-trifluoromethylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4652; 1- (4-trifluoromethylbenzyloxyimino) [(3-difluoromethyl) phenyl] Methyl], [BC4653; 1- (2-difluoromethylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4654; 1- (3-difluoromethylbenzyloxyimino) [(3-difluoromethyl) Phenyl] methyl], [BC 4655; 1- (4-difluoromethylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4656; 1- (2-methoxybenzyloxyimino) [(3-difluoromethyl) 1) (phenyl) methyl], [BC4657; 1- (3-methoxybenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4658; 1- (4-methoxybenzyloxy) Siimino) [(3-difluoromethyl) phenyl] methyl], [BC4659; 1- (2-vinylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4660; 1- (3-vinylbenzyloxy) Imino) [(3-difluoromethyl) phenyl] methyl], [BC4661; 1- (4-vinylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4662; 1- (2-phenylbenzyloxy) Imino) [(3-difluoromethyl) phenyl] methyl], [BC4663; 1- (3-phenylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4664; 1- (4-phenylbenzyloxy) Imino) [(3-difluoromethyl) phenyl] methyl], [BC4665; 1- (2,3-difluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4666; 1- (2,4 -Giff Orobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4667; 1- (2,5-difluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4668; 2,6-Difluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4669; 1- (3,4-difluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4670 1- (3,5-difluorobenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4671; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) [(3) -Difluoromethyl) phenyl] methyl], [BC 4672; 1- (3-ethylbenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4673; 1- (4-ethylbenzyloxyimino) [( -Difluoromethyl) phenyl] methyl], [BC 4674; 1- (2-trifluoromethoxybenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC4675; 1- (3-trifluoromethoxybenzyloxyimino] ) [(3-Difluoromethyl) phenyl] methyl], [BC 4676; 1- (4-trifluoromethoxybenzyloxyimino) [(3-difluoromethyl) phenyl] methyl], [BC 4677; 1- (methoxyimino) [ (3-Difluoromethyl) phenyl] methyl], [BC4678; 1- (ethoxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4679; 1- (propoxyimino) [(4-difluoromethyl) phenyl] Methyl],

[BC 4680; 1- (n-butoxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4681; 1- (pentyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4682; 1- (Hexyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4683; 1- (isopropoxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4684; 1- (tert-butoxyimino) [(4-Difluoromethyl) phenyl] methyl], [BC 4685; 1- (sec-butoxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4686; 1- (cyclopropyloxyimino) [(4- Difluoromethyl) phenyl] methyl], [BC 4687; 1- (Cyclopentyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4688; 1- (Cyclohexyloxyimino) [(4-difluoromethyl) fe] Nyl] methyl], [BC 4689; 1- (3-allyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4690; 1- (3-butenyloxyimino) [(4-difluoromethyl) phenyl 1- (2-propynyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4692; 1- (3-butynyloxyimino) [(4-difluoromethyl) phenyl] Methyl], [BC4693; 1- (1-cyclohexyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4694; 1- (2,2,2-trifluoroethoxyimino) [(4-difluoromethyl) ) Phenyl] methyl], [BC 4695; 1- (benzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4696; 1- (2-fluorobenzyloxyimino) [(4-difluoromethyl) phenyl] Methyl], [BC 4697; 1- ( -Fluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4698; 1- (4-fluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4699; 1- (2) -Chlorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4700; 1- (3-chlorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4701; 1- (4) -Chlorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4702; 1- (2-methylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4703; 1- (3) -Methylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4704; 1- (4-methylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4705; 1- (2) -Cyanobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4706; 1- (3-cyanobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4707; 1- (4) -Cyanobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4708; 1- (2-trifluoromethylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4709; 1- (3-Trifluoromethylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4710; 1- (4-trifluoromethylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [ BC 4711; 1- (2-difluoromethylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4712; 1- (3-difluoromethylbenzyloxyimino) [ 4-Difluoromethyl) phenyl] methyl], [BC 4713; 1- (4-difluoromethylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4714; 1- (2-methoxybenzyloxyimino) [ (4-Difluoromethyl) phenyl] methyl], [BC 4715; 1- (3-methoxybenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4716; 1- (4-methoxybenzyloxyimino) [ (4-Difluoromethyl) phenyl] methyl], [BC 4717; 1- (2-vinylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4718; 1- (3-vinylbenzyloxyimino) [ (4-Difluoromethyl) phenyl] methyl], [BC 4719; 1- (4-vinylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4720; 1- (2-phenylbenzyl oxy) Imino) [(4-difluoromethyl) phenyl] methyl], [BC4721; 1- (3-phenylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4722; 1- (4-phenylbenzyloxy) Imino) [(4-difluoromethyl) phenyl] methyl], [BC 4723; 1- (2,3-difluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4724; 1- (2,4 -Difluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4725; 1- (2,5-difluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4726; 1- (2,6-difluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4727; 1- (3,4-difluorobenzyloxyimino) [(4-difluoromethyl) phenyl] Methyl], [BC 4728; 1- (3,5-difluorobenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4729; 1- (2,3,4,5,6-pentafluorobenzyloxy) Imino) [(4-difluoromethyl) phenyl] methyl], [BC 4730; 1- (3-ethylbenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4731; 1- (4-ethylbenzyloxy) Imino) [(4-difluoromethyl) phenyl] methyl], [BC 4732; 1- (2-trifluoromethoxybenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC 4 733; 1- (3- tri) Fluoromethoxybenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4734; 1- (4-trifluoromethoxybenzyloxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4735; -(Methoxyimino) [(4-difluoromethyl) phenyl] methyl], [BC4736; 1- (ethoxyimino) (2-methoxyphenyl) methyl], [BC4737; 1- (propoxyimino) (2-methoxyphenyl) Methyl], [BC 4738; 1- (n-butoxyimino) (2-methoxyphenyl) methyl], [BC 4739; 1-(pentyloxyimino) (2-methoxyphenyl) methyl], [BC 4740; 1-(hexyloxy) Imino) (2-methoxyphenyl) methyl], [BC4741; 1- (isopropoxyimino) (2-methoxyphenyl) methyl], [BC4742; 1- (tert-butoxyimino) (2-methoxyphenyl) methyl], [BC 4743; 1- (sec-butoxyimino) (2-methoxyphenyl) methyl], [BC 4744; 1-(cyclopropyloxyimino) (2-methoxyphenyl) methyl], [BC 4745; 1-(cyclopentyloxyimino) ) (2-Methoxyf 1- (cyclohexyloxyimino) (2-methoxyphenyl) methyl], [BC4747; 1- (3-allyloxyimino) (2-methoxyphenyl) methyl], [BC4748; 1- (3-Butenyloxyimino) (2-methoxyphenyl) methyl], [BC4749; 1- (2-propynyloxyimino) (2-methoxyphenyl) methyl], [BC4750; 1- (3-butynyloxyimino] ) (2-methoxyphenyl) methyl], [BC4751; 1- (1-cyclohexyloxyimino) (2-methoxyphenyl) methyl], [BC4752; 1- (2,2,2-trifluoroethoxyimino) (2) -Methoxyphenyl) methyl], [BC4753; 1- (benzyloxyimino) (2-methoxyphenyl) methyl], [BC4754; 1- (2-fluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4755 1- (3-fluorobenzyloxyimi ) (2-methoxyphenyl) methyl], [BC 4756; 1- (4-fluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4757; 1- (2-chlorobenzyloxyimino) (2-methoxyphenyl) ) Methyl], [BC 4758; 1- (3-chlorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4759; 1-(4-chlorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4760 1- (2-methylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4761; 1- (3-methylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4762; Methylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4763; 1- (2-cyanobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4764; 1- (3-cyanobenzyloxyimino) ( 2-Methoxyphenyl) [BC4 765; 1- (4-cyanobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4766; 1- (2-trifluoromethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4765; BC 4767; 1- (3-trifluoromethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4768; 1- (4-trifluoromethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4769; 1- (2-Difluoromethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4770; 1- (3-difluoromethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4771; 1- (4) -Difluoromethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4772; 1- (2-methoxybenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4773; 1- (3-methoxybenzyl) Oxyimino) (2-methoxyphenyl) methyl], [BC 4774; 1- (4-methoxybenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4775; 1- (2-vinylbenzyloxyimino) (2-methoxy) Phenyl) methyl], [BC4776; 1- (3-vinylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4777; 1- (4-vinylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4777; BC 4778; 1- (2-phenylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC4779; 1- (3-phenylbenzyloxyimino) (2-methoxyphenyl) methyl],

[BC 4 780; 1- (4-phenylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4781; 1-(2,3-difluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4782; 1 -(2,4-difluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4783; 1- (2,5-difluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4784; 2,6-Difluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4785; 1- (3,4-difluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4786; 1- (3, 5-Difluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4787; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (2-methoxyphenyl) methyl], [BC4788; 1- (3-ethyl benzyl Xyimino) (2-methoxyphenyl) methyl], [BC 4789; 1- (4-ethylbenzyloxyimino) (2-methoxyphenyl) methyl], [BC 4790; 1- (2-trifluoromethoxybenzyloxyimino) (2) -Methoxyphenyl) methyl], [BC4791; 1- (3-trifluoromethoxybenzyloxyimino) (2-methoxyphenyl) methyl], [BC4792; 1- (4-trifluoromethoxybenzyloxyimino) (2-methoxy) Phenyl) methyl], [BC4793; 1- (methoxyimino) (2-methoxyphenyl) methyl], [BC4794; 1- (ethoxyimino) (3-methoxyphenyl) methyl], [BC4795; 1- (propoxyimino) (3-methoxyphenyl) methyl], [BC4796; 1- (n-butoxyimino) (3-methoxyphenyl) methyl], [BC4797; 1- (pentyloxyimino) (3-methoxyphenyl) methyl], [BC4798 1- (Hexyloxyimino) (3-methoxyphenyl) methyl], [BC 4799; 1- (isopropoxyimino) (3-methoxyphenyl) methyl], [BC 4800; 1- (tert-butoxyimino) (3-methoxyphenyl) Methyl], [BC4801; 1- (sec-butoxyimino) (3-methoxyphenyl) methyl], [BC4802; 1- (cyclopropyloxyimino) (3-methoxyphenyl) methyl], [BC4803; 1- (cyclo) Pentyloxyimino) (3-methoxyphenyl) methyl], [BC 4804; 1- (cyclohexyloxyimino) (3-methoxyphenyl) methyl], [BC 4805; 1- (3-allyloxyimino) (3-methoxyphenyl) Methyl], [BC4806; 1- (3-butenyloxyimino) (3-methoxyphenyl) methyl], [BC4807; 1- (2-propynyloxyimino) (3-methoxyphenyl) methyl], [BC4808; 1 -(3-butynylok Imino) (3-methoxyphenyl) methyl], [BC4809; 1- (1-cyclohexyloxyimino) (3-methoxyphenyl) methyl], [BC4810; 1- (2,2,2-trifluoroethoxyimino) ( 3-methoxyphenyl) methyl], [BC4811; 1- (benzyloxyimino) (3-methoxyphenyl) methyl], [BC4812; 1- (2-fluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4812; BC 4813; 1- (3-fluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4814; 1- (4-fluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4815; 1- (2) -Chlorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4816; 1- (3-chlorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4817; 1- (4-chlorobenzyloxyimino) (3-Methoxyf Nyl) methyl], [BC4818; 1- (2-methylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4819; 1- (3-methylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC BC4820; 1- (4-methylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4821; 1- (2-cyanobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4822; 1- (3) -Cyanobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4823; 1- (4-cyanobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4824; 1- (2-trifluoromethylbenzyloxy) Imino) (3-methoxyphenyl) methyl], [BC4825; 1- (3-trifluoromethylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4826; 1- (4-trifluoromethylbenzyloxyimino) (3-Metoki Ciphenyl) methyl], [BC4827; 1- (2-difluoromethylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4828; 1- (3-difluoromethylbenzyloxyimino) (3-methoxyphenyl) methyl] , [BC4829; 1- (4-difluoromethylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4830; 1- (2-methoxybenzyloxyimino) (3-methoxyphenyl) methyl], [BC4831; 1 -(3-Methoxybenzyloxyimino) (3-methoxyphenyl) methyl], [BC 4832; 1- (4-methoxybenzyloxyimino) (3-methoxyphenyl) methyl], [BC 4833; 1- (2-vinylbenzyl) Oxyimino) (3-methoxyphenyl) methyl], [BC4834; 1- (3-vinylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4835; 1- (4-vinylbenzyloxyimino) (3-) 1- (2-phenylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4837; 1- (3-phenylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC 4838; 1- (4-phenylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC 4839; 1-(2,3-difluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC 4840; 1 -(2,4-difluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4841; 1- (2,5-difluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4842; 2,6-Difluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4843; 1- (3,4-difluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4844; 1- (3, 5-difluoroben Dihydroxyimino) (3-methoxyphenyl) methyl], [BC4845; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (3-methoxyphenyl) methyl], [BC4846; 3-ethylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4847; 1- (4-ethylbenzyloxyimino) (3-methoxyphenyl) methyl], [BC4848; 1- (2-trifluoromethoxybenzyl) Oxyimino) (3-methoxyphenyl) methyl], [BC4849; 1- (3-trifluoromethoxybenzyloxyimino) (3-methoxyphenyl) methyl], [BC4850; 1- (4-trifluoromethoxybenzyloxyimino] ) (3-methoxyphenyl) methyl], [BC4851; 1- (methoxyimino) (3-methoxyphenyl) methyl], [BC4852; 1- (ethoxyimino) (4-methoxyphenyl) methyl], [BC4853; -(Propo Siimino) (4-methoxyphenyl) methyl], [BC4854; 1- (n-butoxyimino) (4-methoxyphenyl) methyl], [BC4855; 1- (pentyloxyimino) (4-methoxyphenyl) methyl], [BC 4856; 1- (hexyloxyimino) (4-methoxyphenyl) methyl], [BC4857; 1- (isopropoxyimino) (4-methoxyphenyl) methyl], [BC4858; 1- (tert-butoxyimino) ( 4-methoxyphenyl) methyl], [BC 4859; 1- (sec-butoxyimino) (4-methoxyphenyl) methyl], [BC 4860; 1- (cyclopropyloxyimino) (4-methoxyphenyl) methyl], [BC 4861 1- (cyclopentyloxyimino) (4-methoxyphenyl) methyl], [BC4862; 1- (cyclohexyloxyimino) (4-methoxyphenyl) methyl], [BC4863; 1- (3-allyloxyimino) ( 4-methoxyphenyl ) Methyl], [BC 4864; 1- (3-butenyloxyimino) (4-methoxyphenyl) methyl], [BC 4865; 1-(2-propynyloxyimino) (4-methoxyphenyl) methyl], [BC 4866; 1- (3-butynyloxyimino) (4-methoxyphenyl) methyl], [BC 4867; 1- (1-cyclohexyloxyimino) (4-methoxyphenyl) methyl], [BC 4868; 1- (2,2, 2-trifluoroethoxyimino) (4-methoxyphenyl) methyl], [BC 4869; 1- (benzyloxyimino) (4-methoxyphenyl) methyl], [BC4870; 1- (2-fluorobenzyloxyimino) (4) -Methoxyphenyl) methyl], [BC 4871; 1- (3-fluorobenzyloxyimino) (4-methoxyphenyl) methyl], [BC 4872; 1-(4-fluorobenzyloxyimino) (4-methoxyphenyl) methyl] , [BC 4873; 1- (2-chlorobenzyl) 1- (3-chlorobenzyloxyimino) (4-methoxyphenyl) methyl], [BC4875; 1- (4-chlorobenzyloxyimino) (4-methoxy) ximino) (4-methoxyphenyl) methyl], [BC4874; Phenyl) methyl], [BC4876; 1- (2-methylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4877; 1- (3-methylbenzyloxyimino) (4-methoxyphenyl) methyl], BC 4 878; 1- (4-methylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4879; 1- (2-cyanobenzyloxyimino) (4-methoxyphenyl) methyl],

[BC 4880; 1- (3-cyanobenzyloxyimino) (4-methoxyphenyl) methyl], [BC4881; 1- (4-cyanobenzyloxyimino) (4-methoxyphenyl) methyl], [BC4882; 2-trifluoromethylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4883; 1- (3-trifluoromethylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4884; 1- (4-) Trifluoromethylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4885; 1- (2-difluoromethylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4886; 1- (3-difluoromethylbenzyl] Oxyimino) (4-methoxyphenyl) methyl], [BC4887; 1- (4-difluoromethylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4888; 1- (2-methoxybenzyloxy) Mino) (4-methoxyphenyl) methyl], [BC4889; 1- (3-methoxybenzyloxyimino) (4-methoxyphenyl) methyl], [BC4890; 1- (4-methoxybenzyloxyimino) (4-methoxy Phenyl) methyl], [BC4891; 1- (2-vinylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4892; 1- (3-vinylbenzyloxyimino) (4-methoxyphenyl) methyl], BC 4893; 1- (4-vinylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC 4894; 1- (2-phenylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC 4895; 1- (3) -Phenylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4896; 1- (4-phenylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4897; 1- (2,3-difluorobenzyloxy) Imino) (4- 1- (2,4-Difluorobenzyloxyimino) (4-methoxyphenyl) methyl], [BC4899; 1- (2,5-difluorobenzyloxyimino) (4-methoxyphenyl)] ) Methyl], [BC 4900; 1- (2, 6-difluorobenzyloxyimino) (4-methoxyphenyl) methyl], [BC 4901; 1-(3,4- difluorobenzyloxyimino) (4-methoxyphenyl) methyl 1- (3,5-difluorobenzyloxyimino) (4-methoxyphenyl) methyl], [BC4903; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (4) -Methoxyphenyl) methyl], [BC 4904; 1- (3-ethylbenzyloxyimino) (4-methoxyphenyl) methyl], [BC4905; 1- (4-ethylbenzyloxyimino) (4-methoxyphenyl) methyl] , [BC 4906; 1- (2- Trifluoromethoxybenzyloxyimino) (4-methoxyphenyl) methyl], [BC4907; 1- (3-trifluoromethoxybenzyloxyimino) (4-methoxyphenyl) methyl], [BC4908; 1- (4-trifluoro) Methoxybenzyloxyimino) (4-methoxyphenyl) methyl], [BC4909; 1- (methoxyimino) (4-methoxyphenyl) methyl], [BC4910; 1- (ethoxyimino) (2-cyclohexylphenyl) methyl], [BC4911; 1- (propoxyimino) (2-cyclohexylphenyl) methyl], [BC4912; 1- (n-butoxyimino) (2-cyclohexylphenyl) methyl], [BC4913; 1- (pentyloxyimino) (2 -Cyclohexylphenyl) methyl], [BC 4914; 1- (hexyloxyimino) -1- (2-cyclohexylphenyl) -methyl], [BC 4915; 1- (isopropoxyimino) (2-) Clohexylphenyl) methyl], [BC 4916; 1- (tert-butoxyimino) (2-cyclohexylphenyl) methyl], [BC4917; 1- (sec-butoxyimino) (2-cyclohexylphenyl) methyl], [BC4918; 1- (cyclopropyloxyimino) (2-cyclohexylphenyl) methyl], [BC4919; 1- (cyclopentyloxyimino) (2-cyclohexylphenyl) methyl], [BC4920; 1- (cyclohexyloxyimino) (2-) 1- (3-Allyloxyimino) (2-cyclohexylphenyl) methyl], [BC4922; 1- (3-butenyloxyimino) (2-cyclohexylphenyl) methyl], [cyclohexylphenyl) methyl], [BC 4921; BC 4923; 1- (2-propynyloxyimino) (2-cyclohexylphenyl) methyl], [BC4924; 1- (3-butynyloxyimino) (2-cyclohexylphenyl) Ethyl, [BC 4925; 1- (1-cyclohexyloxyimino) (2-cyclohexylphenyl) methyl], [BC4926; 1- (2,2,2-trifluoroethoxyimino) (2-cyclohexylphenyl) methyl], [BC 4 927; 1- (benzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4928; 1- (2-fluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4929; 1- (3-fluoro) Benzyloxyimino) (2-cyclohexylphenyl) methyl], [BC 4930; 1- (4-fluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4931; 1- (2-chlorobenzyloxyimino) (2) -Cyclohexylphenyl) methyl], [BC4932; 1- (3-chlorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4933; 1- (4-chlorobenzyloxyimino) 2-Cyclohexylphenyl) methyl], [BC4934; 1- (2-methylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4935; 1- (3-methylbenzyloxyimino) (2-cyclohexylphenyl) methyl 1- (4-methylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4937; 1- (2-cyanobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4938; 1] -(3-Cyanobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4939; 1- (4-cyanobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4940; 1- (2-trifluoro) Methylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC 4941; 1- (3-trifluoromethylbenzyloxyimino) (2-cyclohexylphenyl) Ethyl, [BC4942; 1- (4-trifluoromethylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4943; 1- (2-difluoromethylbenzyloxyimino)], [BC4944; 1- (3) -Difluoromethylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC 4945; 1- (4-difluoromethylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4946; 1- (2-methoxybenzyloxy) Imino) (2-cyclohexylphenyl) methyl], [BC4947; 1- (3-methoxybenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4948; 1- (4-methoxybenzyloxyimino) (2-cyclohexyl] Phenyl) methyl], [BC 4949; 1- (2-vinylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC 4950; 1- (3-vinylbenzyloxy Mino) (2-cyclohexylphenyl) methyl], [BC4951; 1- (4-vinylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4952; 1- (2-phenylbenzyloxyimino) (2-cyclohexyl] Phenyl) methyl], [BC 4953; 1- (3-phenylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4954; 1- (4-phenylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC BC 4 955; 1- (2,3-difluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4956; 1- (2,4-difluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4957; 1- (2,5-difluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC 4958; 1- (2,6-difluorobenzyloxyimino) (2-silyl) Lohexylphenyl) methyl], [BC4959; 1- (3,4-difluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4960; 1- (3,5-difluorobenzyloxyimino) (2-cyclohexyl] Phenyl) methyl], [BC4961; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4962; 1- (3-ethylbenzyloxyimino) ( 2-Cyclohexylphenyl) methyl], [BC 4963; 1- (4-ethylbenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC4964; 1- (2-trifluoromethoxybenzyloxyimino) (2-cyclohexylphenyl) ) Methyl], [BC 4965; 1- (3-trifluoromethoxybenzyloxyimino) (2-cyclohexylphenyl) methyl], [BC 4966; 1- (4-trifluoromethoxy) 1 '-(methoxyimino) (2-cyclohexylphenyl) methyl], [BC4968; 1- (ethoxyimino) (3-cyclohexylphenyl) methyl], [BC 4969; 1- (propoxyimino) (3-cyclohexylphenyl) methyl], [BC4970; 1- (n-butoxyimino) (3-cyclohexylphenyl) methyl], [BC4971; 1- (pentyloxyimino) (3 -Cyclohexylphenyl) methyl], [BC4972; 1- (hexyloxyimino) (3-cyclohexylphenyl) methyl], [BC4973; 1- (isopropoxyimino) (3-cyclohexylphenyl) methyl], [BC4974; 1- (Tert-Butoxyimino) (3-cyclohexylphenyl) methyl], [BC 4975; 1- (sec-butoxyimino) (3-cyclohexylphenyl) methyl], [BC 4976; Propyloxyimino) (3-cyclohexylphenyl) methyl], [BC 4977; 1- (cyclopentyloxyimino) (3-cyclohexylphenyl) methyl], [BC4978; 1- (cyclohexyloxyimino) (3-cyclohexylphenyl) methyl ], [BC 4979; 1- (3-allyloxyimino) (3-cyclohexylphenyl) methyl],

[BC 4980; 1- (3-butenyloxyimino) (3-cyclohexylphenyl) methyl], [BC 4981; 1- (2-propynyloxyimino) (3-cyclohexylphenyl) methyl], [BC4982; 1- (3) -Butynyloxyimino) (3-cyclohexylphenyl) methyl], [BC4983; 1- (1-cyclohexyloxyimino) (3-cyclohexylphenyl) methyl], [BC4984; 1- (2,2,2-trifluoro] Ethoxyimino) (3-cyclohexylphenyl) methyl], [BC4985; 1- (benzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4986; 1- (2-fluorobenzyloxyimino) (3-cyclohexylphenyl) Methyl], [BC 4987; 1- (3-fluorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4988; 1- (4-fluorobenzyloxyimino) (3-cyclohexyl] Phenyl) methyl], [BC 4989; 1- (2-chlorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4990; 1- (3-chlorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC BC4991; 1- (4-chlorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4992; 1- (2-methylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4993; 1- (3) -Methylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4994; 1- (4-methylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC4995; 1- (2-cyanobenzyloxyimino) (3-Cyclohexylphenyl) methyl], [BC 4996; 1- (3-cyanobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC 4997; 1- (4-cyanobenzyloxyimime] B) (3-cyclohexylphenyl) methyl], [BC 4998; 1- (2-trifluoromethylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC 4999; 1- (3-trifluoromethylbenzyloxyimino) (3-Cyclohexylphenyl) methyl], [BC5000; 1- (4-trifluoromethylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5001; 1- (2-difluoromethylbenzyloxyimino) (3-) Cyclohexylphenyl) methyl], [BC5002; 1- (3-difluoromethylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5003; 1- (4-difluoromethylbenzyloxyimino) (3-cyclohexylphenyl) methyl ], [BC 5004; 1- (2-methoxybenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC 5005; 1- (3-methoxy) 1- (4-methoxybenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5007; 1- (2-vinylbenzyloxyimino) ( 3-Cyclohexylphenyl) methyl], [BC5008; 1- (3-vinylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5009; 1- (4-vinylbenzyloxyimino) (3-cyclohexylphenyl) methyl 1- (2-phenylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5011; 1- (3-phenylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5012; 1] -(4-phenylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5013; 1- (2,3-difluorobenzyloxyimino) (3-cyclohexy] -Phenyl) methyl], [BC5014; 1- (2,4-difluorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5015; 1- (2,5-difluorobenzyloxyimino) (3-cyclohexylphenyl) Methyl], [BC5016; 1- (2,6-difluorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5017; 1- (3,4-difluorobenzyloxyimino) (3-cyclohexylphenyl) methyl] , [BC5018; 1- (3,5-difluorobenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5019; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (3-) Cyclohexylphenyl) methyl], [BC5020; 1- (3-ethylbenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5021; 1- (4-ethylbenzyloxyimino) (3-) Clohexylphenyl) methyl], [BC5022; 1- (2-trifluoromethoxybenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5023; 1- (3-trifluoromethoxybenzyloxyimino) (3-cyclohexyl] Phenyl) methyl], [BC5024; 1- (4-trifluoromethoxybenzyloxyimino) (3-cyclohexylphenyl) methyl], [BC5025; 1- (methoxyimino) (3-cyclohexylphenyl) methyl], [BC5026; 1- (Ethoxyimino) (4-cyclohexylphenyl) methyl], [BC5027; 1- (propoxyimino) (4-cyclohexylphenyl) methyl], [BC5028; 1- (n-butoxyimino) (4-cyclohexylphenyl) Methyl], [BC5029; 1- (pentyloxyimino) (4-cyclohexylphenyl) methyl], [BC5030; 1- (hexyloxyimino) (4-cyclo) Xylphenyl) methyl], [BC 5031; 1- (isopropoxyimino) (4-cyclohexylphenyl) methyl], [BC 5032; 1-(tert-butoxyimino) (4-cyclohexylphenyl) methyl], [BC 5033; (Sec-Butoxyimino) (4-cyclohexylphenyl) methyl], [BC 5034; 1- (cyclopropyloxyimino) (4-cyclohexylphenyl) methyl], [BC5035; 1- (cyclopentyloxyimino) (4-cyclohexyl] Phenyl) methyl], [BC5036; 1- (cyclohexyloxyimino) (4-cyclohexylphenyl) methyl], [BC5037; 1- (3-allyloxyimino) (4-cyclohexylphenyl) methyl], [BC5038; 1- (3-Butenyloxyimino) (4-cyclohexylphenyl) methyl], [BC5039; 1- (2-propynyloxyimino) (4-cyclohexylphenyl) methyl], [BC5 040; 1- (3-butynyloxyimino) (4-cyclohexylphenyl) methyl], [BC5041; 1- (1-cyclohexyloxyimino) (4-cyclohexylphenyl) methyl], [BC5042; 1- (2, 2, 2,2-trifluoroethoxyimino) (4-cyclohexylphenyl) methyl], [BC 5043; 1- (benzyloxyimino) (4-cyclohexylphenyl) methyl], [BC 5044; 1- (2-fluorobenzyloxyimino) (4-Cyclohexylphenyl) methyl], [BC5045; 1- (3-fluorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5046; 1- (4-fluorobenzyloxyimino) (4-cyclohexylphenyl) Methyl], [BC5047; 1- (2-chlorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5048; 1- (3-chlorobenzyloxyimino) (4-cyclohexene) Silphenyl) methyl], [BC5049; 1- (4-chlorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5050; 1- (2-methylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5050; BC5051; 1- (3-methylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5052; 1- (4-methylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5053; 1- (2) -Cyanobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC 5054; 1- (3-cyanobenzyloxyimino) -1- (4-cyclohexylphenyl) -methyl], [BC 5055; 1- (4) -Cyanobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5056; 1- (2-trifluoromethylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5057; 1- (3-to) Fluoromethylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5058; 1- (4-trifluoromethylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5059; 1- (2-difluoromethylbenzyl) Oxyimino) (4-cyclohexylphenyl) methyl], [BC5060; 1- (3-difluoromethylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5061; 1- (4-difluoromethylbenzyloxyimino) ( 4-Cyclohexylphenyl) methyl], [BC5062; 1- (2-methoxybenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5063; 1- (3-methoxybenzyloxyimino) (4-cyclohexylphenyl) methyl ], [BC 5064; 1- (4-methoxybenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC 50 65; 2-vinylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5066; 1- (3-vinylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5067; 1- (4-vinylbenzyloxyimino) ) (4-Cyclohexylphenyl) methyl], [BC5068; 1- (2-phenylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5069; 1- (3-phenylbenzyloxyimino) (4-cyclohexylphenyl) ) Methyl], [BC 5070; 1- (4-phenylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5071; 1-(2,3-difluorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5072; 1- (2,4-difluorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5073; 1- (2,5-difluorobenzyloxy) Imino) (4-cyclohexylphenyl) methyl], [BC5074; 1- (2,6-difluorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5075; 1- (3,4-difluorobenzyloxyimino) (4-Cyclohexylphenyl) methyl], [BC5076; 1- (3,5-difluorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5077; 1- (2,3,4,5,6-penta) Fluorobenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5078; 1- (3-ethylbenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5079; 1- (4-ethylbenzyloxyimino) ( 4-cyclohexylphenyl) methyl],

[BC 5080; 1- (2-trifluoromethoxybenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5081; 1- (3-trifluoromethoxybenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC5082 1- (4-trifluoromethoxybenzyloxyimino) (4-cyclohexylphenyl) methyl], [BC 5083; 1- (methoxyimino) (4-cyclohexylphenyl) methyl], [BC 5084; 1- (ethoxyimino) ( 2-cyanophenyl) methyl], [BC5085; 1- (propoxyimino) (2-cyanophenyl) methyl], [BC5086; 1- (n-butoxyimino) (2-cyanophenyl) methyl], [BC5087; 1 -(Pentyloxyimino) (2-cyanophenyl) methyl], [BC5088; 1- (hexyloxyimino) (2-cyanophenyl) methyl], [BC5089; 1- (isopropoxyimino) (2-cyanophenyl] Nyl) methyl], [BC5090; 1- (tert-butoxyimino) (2-cyanophenyl) methyl], [BC5091; 1- (sec-butoxyimino) (2-cyanophenyl) methyl], [BC5092; (Cyclopropyloxyimino) (2-cyanophenyl) methyl], [BC5093; 1- (cyclopentyloxyimino) (2-cyanophenyl) methyl], [BC5094; 1- (cyclohexyloxyimino) (2-cyanophenyl) ) Methyl], [BC5095; 1- (3-allyloxyimino) (2-cyanophenyl) methyl], [BC5096; 1- (3-butenyloxyimino) (2-cyanophenyl) methyl], [BC5097; 1- (2-propynyloxyimino) (2-cyanophenyl) methyl], [BC5098; 1- (3-butynyloxyimino) (2-cyanophenyl) methyl], [BC5099; 1- (1-cyclohexyloxy) Imino) (2-cyanophenyl) methyl], [BC 5100; 1- (2) , 2,2-trifluoroethoxyimino) (2-cyanophenyl) methyl], [BC5101; 1- (benzyloxyimino) (2-cyanophenyl) methyl], [BC5102; 1- (2-fluorobenzyloxyimino) ) (2-cyanophenyl) methyl], [BC5103; 1- (3-fluorobenzyloxyimino) (2-cyanophenyl) methyl], [BC5104; 1- (4-fluorobenzyloxyimino) (2-cyanophenyl) ) Methyl], [BC 5105; 1- (2-chlorobenzyloxyimino) (2-cyanophenyl) methyl], [BC 5106; 1-(3-chlorobenzyloxyimino) (2-cyanophenyl) methyl], [BC 5107 1- (4-chlorobenzyloxyimino) (2-cyanophenyl) methyl], [BC5108; 1- (2-methylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5109; 1- (3-) Methyl benzyl oxyimino) (2-cyanofe Nyl) methyl], [BC5110; 1- (4-methylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5111; 1- (2-cyanobenzyloxyimino) (2-cyanophenyl) methyl], BC 5112; 1- (3-cyanobenzyloxyimino) (2-cyanophenyl) methyl], [BC5113; 1- (4-cyanobenzyloxyimino) (2-cyanophenyl) methyl], [BC5114; 1- (2) -Trifluoromethylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5115; 1- (3-trifluoromethylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5116; 1- (4-tri) Fluoromethylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5117; 1- (2-difluoromethylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5118; 1- (3-difluoromethylbenzyloxy] Imino) (2- Nophenyl) methyl], [BC5119; 1- (4-difluoromethylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5120; 1- (2-methoxybenzyloxyimino) (2-cyanophenyl) methyl], [BC5121; 1- (3-methoxybenzyloxyimino) (2-cyanophenyl) methyl], [BC5122; 1- (4-methoxybenzyloxyimino) (2-cyanophenyl) methyl], [BC5123; 2-vinylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5124; 1- (3-vinylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5125; 1- (4-vinylbenzyloxyimino) ) (2-cyanophenyl) methyl], [BC5126; 1- (2-phenylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5127; 1- (3-phenylbenzyloxyimino) (2-cyanophenyl) ) Methyl], [BC 5128; 1- (4-phenylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5129; 1- (2,3-difluorobenzyloxyimino) (2-cyanophenyl) methyl], [BC5130; 1- (2,4 -Difluorobenzyloxyimino) (2-cyanophenyl) methyl], [BC 5131; 1- (2,5-difluorobenzyloxyimino) (2-cyanophenyl) methyl], [BC 5132; 1- (2,6-difluoro) Benzyloxyimino) (2-cyanophenyl) methyl], [BC5133; 1- (3,4-difluorobenzyloxyimino) (2-cyanophenyl) methyl], [BC5134; 1- (3,5-difluorobenzyloxy) Imino) (2-cyanophenyl) methyl], [BC5135; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (2-cyanophenyl) methyl], [BC5136; 1- (3- Ethyl benzyl oxyimino) (2-cyano Phenyl) methyl], [BC5137; 1- (4-ethylbenzyloxyimino) (2-cyanophenyl) methyl], [BC5138; 1- (2-trifluoromethoxybenzyloxyimino) (2-cyanophenyl) methyl] [BC5139; 1- (3-trifluoromethoxybenzyloxyimino) (2-cyanophenyl) methyl], [BC5140; 1- (4-trifluoromethoxybenzyloxyimino) (2-cyanophenyl) methyl], BC5141; 1- (methoxyimino) (2-cyanophenyl) methyl], [BC5142; 1- (ethoxyimino) (3-cyanophenyl) methyl], [BC5143; 1- (propoxyimino) (3-cyanophenyl) Methyl], [BC5144; 1- (n-butoxyimino) (3-cyanophenyl) methyl], [BC5145; 1- (pentyloxyimino) (3-cyanophenyl) methyl], [BC5146; 1- (hexyloxy) Imino) (3-cyanophenyl Methyl], [BC5147; 1- (isopropoxyimino) (3-cyanophenyl) methyl], [BC5148; 1- (tert-butoxyimino) (3-cyanophenyl) methyl], [BC5149; 1- (sec- 1- (Cyclopropyloxyimino) (3-cyanophenyl) methyl], [BC5151; 1- (cyclopentyloxyimino) (3-cyanophenyl) methyl] 1- (cyclohexyloxyimino) (3-cyanophenyl) methyl], [BC5153; 1- (3-allyloxyimino) (3-cyanophenyl) methyl], [BC5154; 1- (3-cyanophenyl) methyl], [BC5154; Butenyloxyimino) (3-cyanophenyl) methyl], [BC5155; 1- (2-propynyloxyimino) (3-cyanophenyl) methyl], [BC5156; 1- (3-butynyloxyimino) (3) -Cyanophenyl) methyl], [BC5157; 1- (1-cyclohexyl) Oxyimino) (3-cyanophenyl) methyl], [BC5158; 1- (2,2,2-trifluoroethoxyimino) (3-cyanophenyl) methyl], [BC5159; 1- (benzyloxyimino) (3-) Cyanophenyl) methyl], [BC 5160; 1- (2-fluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5161; 1- (3-fluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5162; 1- (4-fluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5163; 1- (2-chlorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5164; 3-chlorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5165; 1- (4-chlorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5166; 1- (2-methylbenzyloxyimino) ) (3-cyanophenyl) methyl], [B C5 167; 1- (3-methylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5168; 1- (4-methylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5169; 1- (2) -Cyanobenzyloxyimino) (3-cyanophenyl) methyl], [BC5170; 1- (3-cyanobenzyloxyimino) (3-cyanophenyl) methyl], [BC5171; 1- (4-cyanobenzyloxyimino) (3-cyanophenyl) methyl], [BC5172; 1- (2-trifluoromethylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5173; 1- (3-trifluoromethylbenzyloxyimino) (3 -Cyanophenyl) methyl], [BC 5174; 1- (4-trifluoromethylbenzyloxyimino) (3-cyanophenyl) methyl], [BC 5175; 1-(2-difluoromethylbenzyloxyimino) (3-cyanophenyl) ) Methyl], [BC 517 6; 1- (3-difluoromethylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5177; 1- (4-difluoromethylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5178; 1- (2-methoxybenzyloxyimino) (3-cyanophenyl) methyl], [BC5179; 1- (3-methoxybenzyloxyimino) (3-cyanophenyl) methyl],

[BC 5180; 1- (4-methoxybenzyloxyimino) (3-cyanophenyl) methyl], [BC5181; 1- (2-vinylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5182; 3-vinylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5183; 1- (4-vinylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5184; 1- (2-phenylbenzyloxyimino) ) (3-cyanophenyl) methyl], [BC5185; 1- (3-phenylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5186; 1- (4-phenylbenzyloxyimino) (3-cyanophenyl) ) Methyl], [BC5187; 1- (2,3-difluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5188; 1- (2,4-difluorobenzyloxyimino) (3-cyanophenyl) methyl ], [BC 5189; 1- (2,5-difluo Lobenzyloxyimino) (3-cyanophenyl) methyl], [BC 5190; 1- (2,6-difluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5191; 1- (3,4-difluorobenzyl) Oxyimino) (3-cyanophenyl) methyl], [BC5192; 1- (3,5-difluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5193; 1- (2,3,4,5, 1) 6-Pentafluorobenzyloxyimino) (3-cyanophenyl) methyl], [BC5194; 1- (3-ethylbenzyloxyimino) (3-cyanophenyl) methyl], [BC5195; 1- (4-ethylbenzyloxy) Imino) (3-cyanophenyl) methyl], [BC5196; 1- (2-trifluoromethoxybenzyloxyimino) (3-cyanophenyl) methyl], [BC5197; 1- (3-trifluoromethoxybenzyloxyimino) (3-cyanopheny 1) (4-trifluoromethoxybenzyloxyimino) (3-cyanophenyl) methyl], [BC 5199; 1- (methoxyimino) (3-cyanophenyl) methyl], [BC 5200; -(Ethoxyimino) (4-cyanophenyl) methyl], [BC5201; 1- (propoxyimino) (4-cyanophenyl) methyl], [BC5202; 1- (n-butoxyimino) (4-cyanophenyl) methyl ], [BC5203; 1- (pentyloxyimino) (4-cyanophenyl) methyl], [BC5204; 1- (hexyloxyimino) (4-cyanophenyl) methyl], [BC5205; 1- (isopropoxyimino)] (4-cyanophenyl) methyl], [BC5206; 1- (tert-butoxyimino) (4-cyanophenyl) methyl], [BC5207; 1- (sec-butoxyimino) (4-cyanophenyl) methyl], [BC BC 5208; 1- (cyclopropyloxyimino) (4-cyano 1- (Cyclopentyloxyimino) (4-cyanophenyl) methyl], [BC5210; 1- (cyclohexyloxyimino) (4-cyanophenyl) methyl], [BC5211; 3-Allyloxyimino) (4-cyanophenyl) methyl], [BC5212; 1- (3-butenyloxyimino) (4-cyanophenyl) methyl], [BC5213; 1- (2-propynyloxyimino) ( 4-cyanophenyl) methyl], [BC5214; 1- (3-butynyloxyimino) (4-cyanophenyl) methyl], [BC5215; 1- (1-cyclohexyloxyimino) (4-cyanophenyl) methyl] , [BC5216; 1- (2,2,2-trifluoroethoxyimino) (4-cyanophenyl) methyl], [BC5217; 1- (benzyloxyimino) (4-cyanophenyl) methyl], [BC5218; 1 -(2-Fluorobenzyloxyimino) (4-cyanophenyl) Methyl], [BC5219; 1- (3-fluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5220; 1- (4-fluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5221; 1- (2-chlorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5222; 1- (3-chlorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5223; 1- (4-chloro) Benzyloxyimino) (4-cyanophenyl) methyl], [BC5224; 1- (2-methylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5225; 1- (3-methylbenzyloxyimino) (4 -Cyanophenyl) methyl], [BC5226; 1- (4-methylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5227; 1- (2-cyanobenzyloxyimino) (4-cyanophenyl) methyl] [BC 5228; 1- (3-cyanobenzyloxyl 1) (4-cyanophenyl) methyl], [BC5 229; 1- (4-cyanobenzyloxyimino) (4-cyanophenyl) methyl], [BC 5230; 1- (2-trifluoromethylbenzyloxyimino) (4) -Cyanophenyl) methyl], [BC5231; 1- (3-trifluoromethylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5232; 1- (4-trifluoromethylbenzyloxyimino) (4-cyano Phenyl) methyl], [BC 5233; 1- (2-difluoromethylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5234; 1- (3-difluoromethylbenzyloxyimino) (4-cyanophenyl) methyl] , [BC5235; 1- (4-difluoromethylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5236; 1- (2-methoxybenzyloroxyimino) (4-cyanophenyl) methyl], [BC5237; 1- (3- Methoxybenzyloxyimino) (4-cyanophenyl) methyl], [BC5238; 1- (4-methoxybenzyloxyimino) (4-cyanophenyl) methyl], [BC5239; 1- (2-vinylbenzyloxyimino) ( 4-cyanophenyl) methyl], [BC5240; 1- (3-vinylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5241; 1- (4-vinylbenzyloxyimino) (4-cyanophenyl) methyl 1- (2-phenylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5243; 1- (3-phenylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5244; 1] -(4-phenylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5245; 1- (2,3-difluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5246; 1- (2, 4-difluorobenzyloxyi B) (4-cyanophenyl) methyl], [BC5247; 1- (2,5-difluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5248; 1- (2,6-difluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5249; 1- (3,4-difluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5250; 1- (3,5-difluorobenzyloxyimino) (4) -Cyanophenyl) methyl], [BC5251; 1- (2,3,4,5,6-pentafluorobenzyloxyimino) (4-cyanophenyl) methyl], [BC5252; 1- (3-ethylbenzyloxyimino] ) (4-cyanophenyl) methyl], [BC5253; 1- (4-ethylbenzyloxyimino) (4-cyanophenyl) methyl], [BC5254; 1- (2-trifluoromethoxybenzyloxyimino) (4-) Cyanophenyl) methyl], [BC 5255; 1- (3- Trifluoromethoxybenzyloxyimino) (4-cyanophenyl) methyl], [BC5256; 1- (4-trifluoromethoxybenzyloxyimino) (4-cyanophenyl) methyl], [BC5257; 1- (methoxyimino) ( 4-cyanophenyl) methyl].

  Further, the present compounds AD1-BD1 to AD2160-BD558 can also be obtained according to the above-mentioned method.

The present compounds AD1-BD1 to AD2160-BD558 are compounds represented by the following formula (ADBD).
[Wherein, X ^{40 to} X ⁴⁹ each represent a substituent corresponding to each of the substituent numbers (MD 1) AD 1 to AD 2 160 shown below, wherein E ¹⁰⁴ is a substituent number (MD 2) BD 1 shown below ~ Represents BD 558. ]
For example, the present compound AD1-BD1 is a compound represented by the formula (ADBD) in which X ^{40 to} X ⁴⁹ have a substituent number MD 1 (X ^{40 to} X ⁴³ is CH, X ⁴⁵ is a fluorine atom, X ^{46 to} X ⁴⁸ is A hydrogen atom, X ⁴⁴ and X ¹⁷ are oxygen atoms, E ¹⁰⁴ is a compound in which the substituent number (MD 2) is BD 1 (phenyl group), and is represented by the following formula.
[Substituent number (MD1): X ⁴⁰ , X ⁴¹ , X ⁴² , X ⁴³ , X ⁴⁴ , X ⁴⁵ , X ⁴⁶ , X ⁴⁷ , X ⁴⁸ , X ⁴⁹ ], [AD 1; CH, CH, CH, CH, O, H, H, H, H, H, O], [AD 2; CH, CH, CH, CH, O, F, H, H, O], [AD 3; CH, CH, CH, CH, O, Cl, H, H, H, O], [AD4; CH, CH, CH, CH, CH, O, Br, H, H, H, O], [AD5; CH, CH, CH, CH, O, I, H, H, H, O], [AD6; CH, CH, CH, CH, CH, O, Me, H, H, H, O], [AD7; CH, CH, CH, CH, O, Et, H, H H, H, O], [AD8; CH, CH, CH, CH, CH, O, Pr, H, H, H, O], [AD9; CH, CH, CH, CH, O, i-Pr, H, H, H, O], [ AD10; CH, CH, CH, CH, O, CH = CH 2, H, H, H, O], [AD11; CH, CH, CH, CH, O, C (CH _{3) = CH 2, H,} H, H, O], [AD12; CH, CH, CH, CH, O, C≡CH, H, H, H, O], [AD13; CH, CH, CH, CH, O, C≡CCH ₃ , H, H, H, O], [AD 14; CH, CH, CH, CH, O, c-Pr, H, H, H, O], [AD 15; CH, CH , CH, CH, O, OMe, H, H, H, O, [AD16; CH, CH, CH, CH, CH, O, OEt, H, H, H, O], [AD17; CH, CH, CH , CH, O, Oi-Pr, H, H, H, H, O], [AD 18; CH, CH, CH, CH, O, SMe, H, H, H, O], [AD 19; CH, CH, CH , CH, O, SEt, H, H, H, H, O], [AD 20; CH, CH, CH, CH, O, CH ₂ F, H, H, H, O], [AD 21; CH, CH, CH _{, CH, O, CHF 2,} H, H, H, O], [AD22; CH, CH, CH, CH, O, CF 3, H, H, H, O], [AD23; CH, CH, CH _{, CH, O, OCH 2 F} , H, H, H, O], [AD24; CH, CH, CH, CH, O, OCHF 2, H, H, H, O], [AD25; CH, CH, _{CH, CH, O, OCF 3} , H, H, H, O], [AD26; CH, CH, CH, CH, O, SCH 2 F, H, H, H, O], [AD27; CH, CH , CH, CH, O, SCHF ₂ , H, H, H, O], [AD 28; CH, CH, CH, CH, O, SCF ₃ , H, H, H, O], [AD 29; CH, CH, CH, CH, O, CN, H, H, H, O] , [AD30; CH, CH, CH, CH, O, NO 2, H, H, H, O], [AD31; N, CH, CH, CH, O, H, H , H, H, O], [AD 32; N, CH, CH, CH, O, F, H, H, H, O], [AD 33; N, CH, CH, CH, O, Cl, H, H , H, O], [AD 34; N, CH, CH, CH, O, Br, H, H, H, O], [AD 35; N, CH, CH, CH, O, I, H, H, H N, CH, CH, CH, CH, O, Me, H, H, H, O], [AD 37; N, CH, CH, CH, CH, O, Et, H, H, H, O] , [AD 38; N, CH, CH, CH, O, Pr, H, H, H, O], [AD 39; N, CH, CH, CH, O, i-Pr, H, H, H, O] N, CH, CH, CH, O, CH = CH ₂ , H, H, H, O], [AD 41; N, CH, CH, CH, O, C (CH 3) = CH ₂ , H, H, H, O], [AD 42; N, CH, CH, CH, O, C≡CH, H, H, H, O], [AD 43; N, CH, CH, CH, O, C≡ CCH ₃ , H, H, H, O], [AD 44; N, CH, CH, CH, O, c-Pr, H, H, H, O], [AD 45; N, CH, CH, CH, O , OMe, H, H, H, O], [AD 46; N, CH, CH, CH, O, OEt, H, H, H, O], [AD 47; N, CH, CH, CH, O, Oi -Pr, H, H, H, O], [AD 48; N, CH, CH, CH, O, SMe, H, H, H, O], [AD 49; N, CH, CH, CH, O, SEt , H, H, H, O], [AD 50; N, CH, CH, CH, O, CH ₂ F, H, H, H, O], [AD 51; N, CH, CH, CH, O, CHF _{2, H, H, H,} O], [AD52; N, CH, CH, CH, O, CF 3, H, H, H, O], [AD53; N, CH, CH, CH, O, OCH ₂ F, H, H, H, O], [AD 54; N, CH, CH, CH, O, OCHF ₂ , H, H, H, O], [AD 55; N, CH, CH, CH, O, OCF ₃ , H, H, H, O], [AD 56; N, CH, CH, CH, O, SCH ₂ F, H, H, H, O], [AD 57; N, CH, CH, CH, O, SCHF ₂ , H, H, H, O, [AD 58; N, CH, CH, CH, O, SCF ₃ , H, H, H, O], [AD 59; N, CH, CH, CH, O, CN, H, H, H, H, O], [AD 60; N, CH, CH, CH, O, NO ₂ , H, H, H, O], [AD 61; CH, N, CH, CH , O, H, H, H, H, O, [AD 62; CH, N, CH, CH, O, F, H, H, H, O], [AD 63; CH, N, CH, CH, O , Cl, H, H, H, O], [AD 64; CH, N, CH, CH, O, Br, H, H, H, O], [AD 65; CH, N, CH, CH, O, I , H, H, H, O], [AD 66; CH, N, CH, CH, O, Me, H, H, H, O], [AD 67; CH, N, CH, CH, O, Et, H , H, H, O], [AD 68; CH, N, CH, CH, O, Pr, H, H, H, O], [AD 69; CH, N, CH, CH, O, i-Pr, H , H, H, O], [AD 70; CH, N, CH, CH, O, CH = CH ₂ , H, H, H, O], [AD 71; CH, N, CH, CH, O, C ( CH ₃ ) = CH ₂ , H, H, H, O], [AD 72; CH, N, CH, CH, O, C≡CH, H, H, H, O], [AD 73; CH, N, CH , CH, O, C≡CCH ₃ , H, H, H, O], [AD 74; CH, N, CH, CH, O, c-Pr, H, H, O, [AD 75; CH, N, CH, CH, O, OMe, H, H, H, O], [AD 76; CH, N, CH, CH, O, OEt, H, H, H, O], [AD 77; CH, N, CH, CH, O, Oi-Pr, H, H, H, O], [AD 78; CH, N, CH, CH, O, SMe, H, H, O, [AD 79; CH, N, CH, CH, O, SEt, H, H, H, O], [AD 80; CH, N, CH, CH, O, CH ₂ F, H, H, H, O], [AD 81; CH, N, _{CH, CH, O, CHF 2} , H, H, H, O], [AD82; CH, N, CH, CH, O, CF 3, H, H, H, O], [AD83; CH, N, _{CH, CH, O, OCH 2} F, H, H, H, O], [AD84; CH, N, CH, CH, O, OCHF 2, H, H, H, O], [AD85; CH, N , CH, CH, O, OCF 3, H, H, H, O], [AD86; CH, N, CH, CH, O, SCH 2 F, H, H, H, O], [AD8 7; CH, N, CH, CH, O, SCHF ₂ , H, H, H, O], [AD 88; CH, N, CH, CH, O, SCF ₃ , H, H, H, O], [[ AD 89; CH, N, CH, CH, O, CN, H, H, H, O], [AD 90; CH, N, CH, CH, O, NO ₂ , H, H, H, O], [AD 91 CH, CH, N, CH, O, H, H, H, H, O], [AD 92; CH, CH, N, CH, O, F, H, H, O], [AD 93; CH , CH, N, CH, O, Cl, H, H, H, O], [AD 94; CH, CH, N, CH, O, Br, H, H, O], [AD 95; CH, CH , N, CH, O, I, H, H, H, O], [AD 96; CH, CH, N, CH, O, Me, H, H, H, O], [AD 97; CH, CH, N , CH, O, Et, H, H, H, O, [AD 98; CH, CH, N, CH, O, Pr, H, H, H, O], [AD 99; CH, CH, N, CH , O, i-Pr, H, H, H, O, [AD 100; CH, CH, N, CH, O, CH = CH ₂ , H, H, H, O],

[AD101; CH, CH, N , CH, O, C (CH 3) = CH 2, H, H, H, O], [AD102; CH, CH, N, CH, O, C≡CH, H, H, H, O], [AD 103; CH, CH, N, CH, O, C≡CCH ₃ , H, H, H, O], [AD 104; CH, CH, N, CH, O, c-Pr , H, H, H, O], [AD 105; CH, CH, N, CH, O, OMe, H, H, H, O], [AD 106; CH, CH, N, CH, O, OE t, H , H, H, O], [AD 107; CH, CH, N, CH, O, Oi-Pr, H, H, H, O], [AD 108; CH, CH, N, CH, O, SMe, H , H, H, O], [AD 109; CH, CH, N, CH, O, SE t, H, H, H, O], [AD 110; CH, CH, N, CH, O, CH ₂ F, H , H, H, O], [AD111; CH, CH, N, CH, O, CHF 2, H, H, H, O], [AD112; CH, CH, N, CH, O, CF 3, H , H, H, O], [AD 113; CH, CH, N, CH, O, OCH ₂ F, H, H, H, O], [AD 114; CH, CH, N, CH, O, OCHF ₂ , H, H, H, O] , [AD115; CH, CH, N, CH, O, OCF 3, H, H, H, O], [AD116; CH, CH, N, CH, O, SCH 2 F , H, H, H, O], [AD 117; CH, CH, N, CH, O, SCHF ₂ , H, H, H, O], [AD 118; CH, CH, N, CH, O, SCF ₃ , H, H, H, O], [AD119; CH, CH, N, CH, O, CN, H, H, H, O], [AD 120; CH, CH, N, CH, O, NO ₂ , H, H, H, O], [AD 121; CH, CH, CH, N, O, H, H, H, H, O], [AD 122; CH, CH, CH, N, O, F, H, H H, H, O], [AD 123; CH, CH, CH, N, O, Cl, H, H, O], [AD 124; CH, CH, CH, N, O, Br, H, H, H, H, O], [AD 125; CH, CH, CH, N, O, I, H, H, H, O], [AD 126; CH, CH, CH, N, O, Me, H, H, H, H, O], [AD 127; CH, CH, CH, CH, N, O, Et, H, H, H, O], [AD 128; CH, CH, CH, N, O, Pr, H, H, H, O] [AD 129; CH, CH, CH, N, O, i-Pr, H, H, H, O ], [AD130; CH, CH , CH, N, O, CH = CH 2, H, H, H, O], [AD131; CH, CH, CH, N, O, C (CH 3) = CH 2 , H, H, H, O], [AD 132; CH, CH, CH, N, O, C≡CH, H, H, H, O], [AD 133; CH, CH, CH, N, O, C ≡CCH ₃ , H, H, H, O], [AD 134; CH, CH, CH, N, O, c-Pr, H, H, H, O], [AD 135; CH, CH, CH, N, O, OMe, H, H, H, O], [AD 136; CH, CH, CH, N, O, OEt, H, H, H, O], [AD 137; CH, CH, CH, N, O, Oi-Pr, H, H, H, O], [AD 138; CH, CH, CH, N, O, SMe, H, H, H, O], [AD 139; CH, CH, CH, N, O, SEt, H, H, H, O], [AD 140; CH, CH, CH, N, O, CH ₂ F, H, H, H, O], [AD 141; CH, CH, CH, N, O, CHF ₂ , H, H, H, O, [AD 142; CH, CH, CH, N, O, CF ₃ , H, H, H, O], [AD 143; CH, CH, CH, N, O, _{OCH 2 F, H, H,} H, O], [AD144; CH, CH, CH, N, O, OCHF 2, H, H, H, O], [AD145; CH, CH, CH, N, O _{, OCF 3, H, H,} H, O], [AD146; CH, CH, CH, N, O, SCH 2 F, H, H, H, O], [AD147; CH, CH, CH, N, O, SCHF ₂ , H, H, H, O, [AD 148; CH, CH, CH, N, O, SCF ₃ , H, H, H, O], [AD 149; CH, CH, CH, N, O, CN, H, H, H, O, [AD 150; CH, CH, CH, CH, N, O, NO ₂ , H, H, H, O], [AD 151; N, N, CH, CH, O , H, H, H, H, O], [AD 152; N, N, CH, CH, O, F, H, H, H, O], [AD 153; N, N, CH, CH, O, Cl , H, H, H, O], [AD 154; N, N, CH, CH, O, Br, H, H, H, O], [AD 155; N, N, CH, CH, O, I, H , H, H, O], [AD 156; N, N, CH, CH, O, Me, H, H, H, O], [AD 157; N, N, CH, CH, O, Et, H, H , H, O], [AD 158; N, N, CH, CH, O, Pr, H, H, H, O], [AD159; N, N, CH , CH, O, i-Pr, H, H, H, O], [AD160; N, N, CH, CH, O, CH = CH 2, H, H, H, O], [AD161; N, N, CH, CH, O, C (CH 3) = CH 2, H, H, H, O], [AD162; N, N, CH, CH, O, C≡CH , H, H, H, O], [AD 163; N, N, CH, CH, O, C≡CCH ₃ , H, H, H, O], [AD 164; N, N, CH, CH, O, c-Pr, H, H, H, O], [AD 165; N, N, CH, CH, O, OMe, H, H, H, O], [AD 166; N, N, CH, CH, O, OEt, H, H, H, O], [AD 167; N, N, CH, CH, O, Oi-Pr, H, H, H, O], [AD 168; N, N, CH, CH, O, SMe, H, H, H, O], [AD 169; N, N, CH, CH, O, SEt, H, H, H, O], [AD 170; N, N, CH, CH, O, CH ₂ F, H, H, H, O], [AD171; N, N, CH, CH, O, CHF 2, H, H, H, O], [AD172; N, N, CH, CH, O, CF ₃ , H, H, H, O], [AD 173; N, N, CH, CH, O, OCH ₂ F, H, H, H, O], [AD 174; N, N, CH, CH, O, _{OCHF 2, H, H, H} , O], [AD175; N, N, CH, CH, O, OCF 3, H, H, H, O], [AD176; N, N, CH, CH, O, SCH ₂ F, H, H, H, O], [AD 177; N, N, CH, CH, O, SCHF ₂ , H, H, H, O], [AD 178; N, N, CH, CH, O , SCF ₃ , H, H, H, O, [AD 179; N, N, CH, CH, O, CN, H, H, H, O], [AD 180; N, N, CH, CH, O, _{NO 2, H, H, H} , O], [AD181; N, CH, N, CH, O, H, H, H, H, O], [AD182; N, CH, N, CH, O, F , H, H, H, O], [AD 183; N, CH, N, CH, O, Cl, H, H, H, O], [AD 184; N, CH, N, CH, O, Br, H , H, H, O], [AD 185; N, CH, N, CH, O, I, H, H, H, O], [AD 186; N, CH, N, CH, O, Me, H, H , H, O], [AD 187; N, CH, N, CH, O, Et, H, H, H, O], [AD 188; N, CH, N, CH, O, Pr , H, H, H, O], [AD 189; N, CH, N, CH, O, i-Pr, H, H, H, O], [AD 190; N, CH, N, CH, O, CH _{= CH 2, H, H,} H, O], [AD191; N, CH, N, CH, O, C (CH 3) = CH 2, H, H, H, O], [AD192; N, CH , N, CH, O, C≡CH, H, H, H, O], [AD 193; N, CH, N, CH, O, C≡ CCH ₃ , H, H, H, O], [AD 194; N, CH, N, CH, O, c-Pr, H, H, H, O], [AD 195; N, CH, N, CH, O, OMe, H, H, H, O], [AD 196; N, CH, N, CH, O, OEt, H, H, H, O], [AD 197; N, CH, N, CH, O, Oi-Pr, H, H, H, O], [AD 198; N, CH, N, CH, O, SMe, H, H, H, O], [AD 199; N, CH, N, CH, O, SE, H, H, H, O], [AD 200; N, CH, N, CH, O, CH 2 F, H, H, H, O],

[AD201; N, CH, N , CH, O, CHF 2, H, H, H, O], [AD202; N, CH, N, CH, O, CF 3, H, H, H, O], [AD 203; N, CH, N, CH, O, OCH ₂ F, H, H, H, O], [AD 204; N, CH, N, CH, O, OCHF ₂ , H, H, H, O] , [AD205; N, CH, N, CH, O, OCF 3, H, H, H, O], [AD206; N, CH, N, CH, O, SCH 2 F, H, H, H, O N, CH, N, CH, O, SCHF ₂ , H, H, H, O], [AD 208; N, CH, N, CH, O, SCF ₃ , H, H, H, O] ], [AD 209; N, CH, N, CH, O, CN, H, H, H, O], [AD 210; N, CH, N, CH, O, NO ₂ , H, H, H, O] [AD 211; N, CH, CH, N, O, H, H, H, O], [AD 212; N, CH, CH, N, O, F, H, H, H, O], [AD 211; AD 213; N, CH, CH, N, O, Cl, H, H, O], [AD 214; N, CH, CH, N, O, Br, H, H, H, O], [AD 215; N, CH, CH, N, O, I, H, H, H, O], [AD 216; N, CH, CH, N, O, Me, H, H, O], [AD 217; N, CH, CH, N, O, Et, H, H, H, O], [AD 218; N, CH, CH, N, O, Pr, H, H, H, O], [AD 219; N, CH, CH, N, O, i- Pr, H, H, H, O], [AD220; N, CH, CH, N, O, CH = CH 2, H, H, H, O], [AD221; N , CH, CH, N, O , C (CH 3) = CH 2, H, H, H, O], [AD222; N, CH, CH, N, O, C≡CH, H, H, H, O], [AD 223; N, CH, CH, N, O, C≡CCH ₃ , H, H, H, O], [AD 224; N, CH, CH, N, O, c-Pr, H, H , H, O], [AD 225; N, CH, CH, N, O, OMe, H, H, H, O], [AD 226; N, CH, CH, N, O, OE t, H, H, H , O], [AD 227; N, CH, CH, N, O, Oi-Pr, H, H, H, O], [AD 228; N, CH, CH, N, O, SMe, H, H, H , O], [AD 229; N, CH, CH, N, O, SE, H, H, H, O], [AD 230; N, CH, CH, N, O, CH ₂ F , H, H, H, O], [AD 231; N, CH, CH, N, O, CHF ₂ , H, H, H, O], [AD 232; N, CH, CH, N, O, CF ₃ , H, H, H, O], [AD 233; N, CH, CH, N, O, OCH ₂ F, H, H, H, O], [AD 234; N, CH, CH, N, O, OCHF _{2, H, H, H,} O], [AD235; N, CH, CH, N, O, OCF 3, H, H, H, O], [AD236; N, CH, CH, N, O, SCH ₂ F, H, H, H, O], [AD 237; N, CH, CH, N, O, SCHF ₂ , H, H, H, O], [AD 238; N, CH, CH, N, O, SCF ₃ , H, H, H, O], [AD 239; N, CH, CH, N, O, CN, H, H, H, O], [AD 240; N, CH, CH, N, O, NO ₂ H, H, H, O], [AD 241; CH, N, N, CH, O, H, H, H, H, O], [AD 242; CH, N, N, CH, O, F, H, H, H, O], [AD 243; CH, N, N, CH, O, Cl, H, H, H, O], [AD 244; CH, N, N, CH, O, Br, H, H, H, O], [AD 245; CH, N, N, CH, O, I, H, H, H, O], [AD 246; CH, N, N, CH, O, Me, H, H, H, H, O], [AD 247; CH, N, N, CH, O, Et, H, H, H, O], [AD 248; CH, N, N, CH, O, Pr, H, H, H, H O], [AD249; CH, N, N, CH, O, i-Pr, H, H, H, O], [AD250; CH, N, N, CH, O, CH = CH 2, H, H , H, O], [AD251 ; CH, N, N, CH, O, C (CH 3) = CH 2, H, H, H, O], [AD252; CH, N, N, CH, O, C≡CH, H, H, H, O], [AD 253; CH, N, N, CH, O, C≡ CCH ₃ , H, H, H, O], [AD 254; CH, N, N, CH , O, c-Pr, H, H, H, O, [AD 255; CH, N, N, CH, O, OMe, H, H, H, O], [AD 256; CH, N, N, CH , O, OEt, H, H, H, O, [AD 257; CH, N, N, CH, O, Oi-Pr, H, H, H, O], [AD 258; CH, N, N, CH , O, SMe, H, H, H, O, [AD 259; CH, N, N, CH, O, SE, H, H, H, O], [AD 260; CH, N, N, C _{H, O, CH 2 F,} H, H, H, O], [AD261; CH, N, N, CH, O, CHF 2, H, H, H, O], [AD262; CH, N, N _{, CH, O, CF 3,} H, H, H, O], [AD263; CH, N, N, CH, O, OCH 2 F, H, H, H, O], [AD264; CH, N, _{N, CH, O, OCHF 2} , H, H, H, O], [AD265; CH, N, N, CH, O, OCF 3, H, H, H, O], [AD266; CH, N, _{N, CH, O, SCH 2} F, H, H, H, O], [AD267; CH, N, N, CH, O, SCHF 2, H, H, H, O], [AD268; CH, N , N, CH, O, SCF 3, H, H, H, O], [AD269; CH, N, N, CH, O, CN, H, H, H, O], [AD270; CH, N, _{N, CH, O, NO 2} , H, H, H, O], [AD271; CH, N, CH, N, O, H, H, H, H, O], [AD272; CH, N, CH , N, O, F, H, H, H, O, [AD 273; CH, N, CH, N, O, Cl, H, H, H, O], [AD 274; CH, N, CH, N , O, Br, H, H, H, O, [AD 275; CH, N, CH, N, O, I, H, H, H, O], [AD 276; CH, N, CH, N, O , Me, H, H, H, O], [AD 277; CH, N, CH, N, O, Et, H, H, H, O], [AD 278; CH, N, CH, N, O, Pr , H, H, H, O], [AD 279; CH, N, CH, N, O, i-Pr, H, H, H, O], [AD 280; CH, N, CH, N, O, CH _{= CH 2, H, H,} H, O], [AD281; CH, N, CH, N, O, C (CH 3) = CH 2, H, H, H, O], [AD282; CH, N , CH, N, O, C≡CH, H, H, H, O], [AD 283; CH, N, CH, N, O, C≡ CCH ₃ , H, H, H, O], [AD 284; CH, N, CH, N, O, c, Pr, H, H, H, O], [AD 285; CH, N, CH, N, O, OMe, H, H, H, O], [AD 286; CH, N, CH, N, O, OE, OEt, H, H, H, O], [AD 287; CH, N, CH, N, O, Oi-Pr, H, H, H, O], [AD 288; CH, N, CH, N, O, SMe, H, H, H, O], [AD 289; CH, N, CH, N, O, SE, t, H, H, O], [AD 29 0; CH, N, CH, N, O, CH 2 F, H, H, H, O], [AD291; CH, N, CH, N, O, CHF 2, H, H, H, O], [AD292; CH, N, CH , N, O, CF 3, H, H, H, O], [AD293; CH, N, CH, N, O, OCH 2 F, H, H, H, O] , [AD294; CH, N, CH, N, O, OCHF 2, H, H, H, O], [AD295; CH, N, CH, N, O, OCF 3, H, H, H, O] [AD 296; CH, N, CH, N, O, SCH ₂ F, H, H, H, O], [AD 297: CH, N, CH, N, O, SCHF ₂ , H, H, H, O ], [AD 298; CH, N, CH, N, O, SCF ₃ , H, H, H, O], [AD 299: CH, N, CH, N, O, CN, H, H, H, O] [AD 300; CH, N, CH, N, O, NO ₂ , H, H, H, O],

[AD 301; CH, CH, N, N, O, H, H, H, O], [AD 302; CH, CH, N, N, N, O, F, H, H, O], [AD 303 CH, CH, N, N, N, O, Cl, H, H, H, O], [AD 304; CH, CH, N, N, N, O, Br, H, H, O], [AD 305; CH , CH, N, N, O, I, H, H, H, O], [AD 306; CH, CH, N, N, O, Me, H, H, O], [AD 307; CH, CH , N, N, O, Et, H, H, H, O], [AD 308; CH, CH, N, N, O, Pr, H, H, H, O], [AD 309; CH, CH, N , N, O, i-Pr , H, H, H, O], [AD310; CH, CH, N, N, O, CH = CH 2, H, H, H, O], [AD311; CH, CH, N, N, O, C (CH 3) = CH 2, H, H, H, O], [AD312; CH, CH, N, N, O, C≡CH, H, H, H, O ], [AD 313; CH, CH, N, N, O, C≡CCH ₃ , H, H, H, O], [AD 314; CH, CH, N, N, N, O, c-Pr, H, H, H, O], [AD 315; CH, CH, N, N, O, OMe, H, H, H, O], [AD 316; CH, CH, N, N, O, OEt, H, H, H, O], [AD 317] CH, CH, N, N, O, Oi-Pr, H, H, H, O], [AD 318; CH, CH, N, N, O, SMe, H, H, H, O], [AD 319; CH, CH, N, N, O, SE, H, H, O], [AD 320; CH, CH, N, N, N, O, CH ₂ F, H, H, H, H O], [AD 321; CH, CH, N, N, O, CHF ₂ , H, H, H, O], [AD 322; CH, CH, N, N, O, CF ₃ , H, H, H, H O], [AD 323; CH, CH, N, N, O, OCH ₂ F, H, H, H, O], [AD 324; CH, CH, N, N, O, OCHF ₂ , H, H, H , O], [AD325; CH , CH, N, N, O, OCF 3, H, H, H, O], [AD326; CH, CH, N, N, O, SCH 2 F, H, H, H, O], [AD327; CH, CH, N, N, O, SCHF 2, H, H, H, O], [AD328; CH, CH, N, N, O, SCF 3, H, H, H, O], [AD 329; CH, CH, N, N, O, CN, H, H, H, O], [AD 330; CH, CH, N, N, O, NO ₂ , H, H, H, O], [AD 331; N, CH, N, N, O, H, H, H, H, O], [AD 332; N, CH, N, N, O, F, H , H, H, O], [AD 333; N, CH, N, N, O, Cl, H, H, H, O], [AD 334; N, CH, N, N, N, O, Br, H, H , H, O], [AD 335; N, CH, N, N, O, I, H, H, H, O], [AD 336: N, CH, N, N, O, Me, H, H, H , O], [AD 337; N, CH, N, N, O, Et, H, H, H, O], [AD 338; N, CH, N, N, O, Pr, H, H, H, O N, CH, N, N, O, i, Pr, H, H, H, O], [AD 340; N, CH, N, N, O, CH, CH ₂ , H, H, H] H, O], [AD341; N, CH, N, N, O, C (CH 3) = CH 2, H, H, H, O], [AD342; N, CH, N, N, O, C ≡CH, H, H, H, O], [AD 343; N, CH, N, N, O, C≡CCH ₃ , H, H, H, O], [AD 344; N, CH, N, N, O, c-Pr, H, H, H, O, [AD 345; N, CH, N, N, O, OMe, H, H, H, O], [AD 346; N, CH, N, N, O, OEt, H, H, H, O, [AD 347; N, CH, N, N, O, Oi-Pr, H, H, H, O], [AD 348; N, CH, N, N, O, SMe, H, H, H, O], [AD 349; N, CH, N, N, O, SE, H, H, H, O], [AD 350; N, CH, N, N, O, _{CH 2 F, H, H,} H, O], [AD351; N, CH, N, N, O, CHF 2, H, H, H, O], [AD352; N, CH, N, N, O _{, CF 3, H, H,} H, O], [AD353; N, CH, N, N, O, OCH 2 F, H, H, H, O], [AD354; N, CH, N, N, _{O, OCHF 2, H, H} , H, O], [AD355; N, CH, N, N, O, OCF 3, H, H, H, O], [AD356; N, CH, N, N, O, SCH ₂ F, H, H, H, O, [AD 357; N, CH, N, N, O, SCHF ₂ , H, H, H, O], [AD 358; N, CH, N, N , O, SCF ₃ , H, H, H, O], [AD 359: N, CH, N, N, O, CN, H, H, H, O], [AD 360; N, CH, N, N, O, NO ₂ , H, H, H, O], [AD 361: CH, CH, CH, CH, S, H, H, H, H, H, O], [AD 362: CH, CH, CH, CH, S, F, H, H, H, O], [AD 363: CH, CH, CH CH, CH, S, Cl, H, H, H, O, [AD 364] CH, CH, CH, CH, CH, S, Br, H, H, H, O], [AD 365; CH, CH, CH, CH CH, S, I, H, H, H, O, [AD 366; CH, CH, CH, CH, S, Me, H, H, H, O], [AD 367; CH, CH, CH, CH, CH S, Et, H, H, H, O, [AD 368; CH, CH, CH, CH, S, Pr, H, H, H, O], [AD 369; CH, CH, CH, CH, S, i-Pr, H, H, H, O], [AD370; CH, CH, CH, CH, S, CH = CH 2, H, H, H, O], [AD371; CH, CH, CH, CH _{, S, C (CH 3)} = CH 2, H, H, H, O], [AD372; CH, CH, CH, CH, S, C≡CH, H, H, H, O], [AD373; CH, CH, CH, CH, S, C≡CCH 3, H, H, H, O], [AD374; CH, CH, CH, CH, S, c-Pr, H, H, H, O], [AD 375; CH, CH, CH, CH, S, OMe, H, H, H, O], [AD 376; CH, CH, CH, CH, S, OEt, H, H, H, O], [AD 377] CH, CH, CH, CH, S, Oi-Pr, H, H, H, O], [AD 378; CH, CH, CH, CH, S, SMe, H, H, H, O], [AD 379; CH, CH, CH, CH, S, SE, SEt, H, H, H, O], [AD 380; CH, CH, CH, CH, S, CH ₂ F, H, H, H, O], [AD 381; ; CH, CH, CH, CH , S, CHF 2, H, H, H, O], [AD382; CH, CH, CH, CH, S, CF 3, H, H, H, O], [AD383 ; CH, CH, CH, CH , S, OCH 2 F, H, H, H, O], [AD384; CH, CH, CH, CH, S, OCHF 2, H, H, H, O], [ AD385; CH, CH, CH, CH, S, OCF 3, H, H, H, O], [AD386; CH, CH, CH, CH, S, SCH 2 F, H, H, H, O], [AD 387; CH, CH, CH, CH, S, SCHF ₂ , H, H, H, O], [AD 388; CH, CH, CH, CH, S, SCF ₃ , H, H, H, O], [AD 389; CH , CH, CH, CH, S , CN, H, H, H, O], [AD390; CH, CH, CH, CH, S, NO 2, H, H, H, O], [AD391; N, CH, CH, CH, S, H, H, H, H, H, O], [AD 392; N, CH, CH, CH, S, F, H, H, H, O], [AD 393; N, CH, CH, CH, S, Cl, H, H, H, H, O], [AD 394; N, CH, CH, CH, S, Br, H, H, H, O], [AD 395: N, CH, CH, CH, S, I, H, H, H, O, [AD396; N, CH, CH, CH, S, Me, H, H, H, O], [AD 397; N, CH, CH, CH, S, Et, H, H, H, O, [AD 398; N, CH, CH, CH, S, Pr, H, H, H, O], [AD 399; N, CH, CH, CH, S, i-Pr, H, H, H, O], [AD 400; N, CH, CH, CH, S, CH = CH ₂ , H, H, H, O],

[AD401; N, CH, CH , CH, S, C (CH 3) = CH 2, H, H, H, O], [AD402; N, CH, CH, CH, S, C≡CH, H, H, H, O], [ AD403; N, CH, CH, CH, S, C≡CCH 3, H, H, H, O], [AD404; N, CH, CH, CH, S, c-Pr , H, H, H, O], [AD 405; N, CH, CH, CH, S, OMe, H, H, H, O], [AD 406; N, CH, CH, CH, S, OE t, H , H, H, O], [AD 407; N, CH, CH, CH, S, Oi-Pr, H, H, H, O], [AD 408; N, CH, CH, CH, S, SMe, H , H, H, O], [AD 409; N, CH, CH, CH, S, SE t, H, H, H, O], [AD 410; N, CH, CH, CH, S, CH ₂ F, H , H, H, O], [AD411; N, CH, CH, CH, S, CHF 2, H, H, H, O], [AD412; N, CH, CH, CH, S, CF 3, H , H, H, O], [AD413; N, CH, CH, CH, S, OCH 2 F, H, H, H, O], [AD414; N, CH, CH, CH, S, OCHF 2, H, H, H, O] , [AD415; N, CH, CH, CH, S, OCF 3, H, H, H, O], [AD416; N, CH, CH, CH, S, SCH 2 F , H, H, H, O], [AD 417; N, CH, CH, CH, S, SCHF ₂ , H, H, H, O], [AD 418; N, CH, CH, CH, S, SCF ₃ , H, H, H, O], [AD 419; N, CH, CH, CH, S, CN, H, H, H, O], [AD 420; N, CH, CH, CH, S, NO ₂ , H, H, H, O], [AD 421; CH, N, CH, CH, S, H, H, H, H, O], [AD 422; CH, N, CH, CH, S, F, H, H H, H, O], [AD 423: CH, N, CH, CH, S, Cl, H, H, H, O], [AD 424; CH, N, CH, CH, S, Br, H, H, H H, O], [AD 425; CH, N, CH, CH, S, I, H, H, H, O], [AD 426; CH, N, CH, CH, S, Me, H, H, H, H, H O], [AD 427; CH, N, CH, CH, S, Et, H, H, H, O], [AD 428; CH, N, CH, CH, S, Pr, H, H, H, O] , [AD 429; CH, N, CH, CH, S, i-Pr, H, H, H, O ], [AD430; CH, N , CH, CH, S, CH = CH 2, H, H, H, O], [AD431; CH, N, CH, CH, S, C (CH 3) = CH 2 , H, H, H, O], [AD 432; CH, N, CH, CH, S, C≡CH, H, H, H, O], [AD 433; CH, N, CH, CH, S, C ≡CCH ₃ , H, H, H, O], [AD 434; CH, N, CH, CH, S, c-Pr, H, H, H, O], [AD 435; CH, N, CH, CH, S, OMe, H, H, H, O], [AD 436; CH, N, CH, CH, S, OEt, H, H, H, O], [AD 437; CH, N, CH, CH, S, Oi-Pr, H, H, H, O], [AD 438; CH, N, CH, CH, S, SMe, H, H, H, O], [AD 439: CH, N, CH, CH, S, SEt, H, H, H, O], [AD440; CH, N, CH, CH, S, CH 2 F, H, H, H, O], [AD441; CH, N, CH, CH, S, _{CHF 2, H, H, H} , O], [AD442; CH, N, CH, CH, S, CF 3, H, H, H, O], [AD443; CH, N, CH, CH, S, OCH ₂ F, H, H, H, O], [AD 444; CH, N, CH, CH, S, OCHF ₂ , H, H, H, O], [AD 445; CH, N, CH, CH, S _{, OCF 3, H, H,} H, O], [AD446; CH, N, CH, CH, S, SCH 2 F, H, H, H, O], [AD447; CH, N, CH, CH, _{S, SCHF 2, H, H} , H, O], [AD448; CH, N, CH, CH, S, SCF 3, H, H, H, O], [AD449; CH, N, CH, CH, S, CN, H, H, H, O, [AD 450; CH, N, CH, CH, S, NO ₂ , H, H, H, O], [AD 451: CH, CH, N, CH, S , H, H, H, H, O], [AD 452; CH, CH, N, CH, S, F, H, H, H, O], [AD 453: CH, CH, N, CH, S, Cl , H, H, H, O], [AD 454; CH, CH, N, CH, S, Br, H, H, H, O], [AD 455; CH, CH, N, CH, S, I, H , H, H, O], [AD 456; CH, CH, N, CH, S, Me, H, H, H, O], [AD 457; CH, CH, N, CH, S, Et, H, H , H, O], [AD 458; CH, CH, N, CH, S, Pr, H , H, H, O], [AD 459; CH, CH, N, CH, S, i-Pr, H, H, H, O], [AD 460; CH, CH, N, CH, S, CH = CH _{2, H, H, H,} O], [AD461; CH, CH, N, CH, S, C (CH 3) = CH 2, H, H, H, O], [AD462; CH, CH, N , CH, S, C≡CH, H, H, H, O, [AD 463; CH, CH, N, CH, S, C≡ CCH ₃ , H, H, H, O], [AD 464; CH, CH, N, CH, S, c-Pr, H, H, H, O], [AD 465; CH, CH, N, CH, S, OMe, H, H, H, O], [AD 466; CH, N, CH, S, OEt, H, H, H, O], [AD 467; CH, CH, N, CH, S, Oi-Pr, H, H, H, O], [AD 468; CH, N, CH, S, SMe, H, H, H, O], [AD 469; CH, CH, N, CH, S, SE, H, H, H, O], [AD 470; CH, CH, _{N, CH, S, CH 2} F, H, H, H, O], [AD471; CH, CH, N, CH, S, CHF 2, H, H, H, O], [AD472; CH, CH , N, CH, S, CF 3, H, H, H, O], [AD473; CH, CH, N, CH, S, OCH 2 F, H, H, H, O], [AD474; CH, CH, N, CH, S, OCHF 2, H, H, H, O], [AD475; CH, CH, N, CH, S, OCF 3, H, H, H, O], [AD476; CH, CH, N, CH, S, SCH ₂ F, H, H, H, O], [AD 477; CH, CH, N, CH, S, SCHF ₂ , H, H, H, O], [AD 478; CH , CH, N, CH, S , SCF 3, H, H, H, O], [AD479; CH, CH, N, CH, S, CN, H, H, H, O], [AD480; CH, CH, N, CH, S, NO 2, H, H, H, O], [AD481; CH, CH, CH, N, S, H, H, H, H, O], [AD482; CH, CH , CH, N, S, F, H, H, H, O], [AD 483; CH, CH, CH, CH, N, S, Cl, H, H, H, O], [AD 484; CH, CH, CH , N, S, Br, H, H, H, O, [AD 485; CH, CH, CH, N, S, I, H, H, O], [AD 486; CH, CH, CH, N , S, Me, H, H, H, O], [AD 487; CH, CH, CH, N, S, Et, H, H, H, H, O], [AD 488; CH, CH, CH, N, S, Pr, H, H, H, O], [AD 489; CH, CH, CH, N, S, i-Pr, H, H, H, O], [AD490; CH, CH, CH, N, S, CH = CH 2, H, H, H, O], [AD491; CH, CH, CH , N, S, C (CH 3) = CH 2, H, H, H, O], [AD492; CH, CH, CH, N, S, C≡CH, H, H, H, O], [ AD 493; CH, CH, CH, N, S, C≡CCH ₃ , H, H, H, O], [AD 494; CH, CH, CH, N, S, c-Pr, H, H, H, O ], [AD495; CH, CH, CH, N, S, OMe, H, H, H, O], [AD 496; CH, CH, CH, N, S, OEt, H, H, H, O], [AD 497: CH, CH, CH, N, S, Oi-Pr, H, H, H, O], [AD 498: CH, CH, CH, N, S, SMe, H, H, H, O], [AD499; CH, CH, CH , N, S, SEt, H, H, H, O], [AD500; CH, CH, CH, N, S, CH 2 F, H, H, H, O],

[AD501; CH, CH, CH , N, S, CHF 2, H, H, H, O], [AD502; CH, CH, CH, N, S, CF 3, H, H, H, O], [AD 503; CH, CH, CH, N, S, OCH ₂ F, H, H, H, O], [AD 504; CH, CH, CH, N, S, OCHF ₂ , H, H, H, O] , [AD505; CH, CH, CH, N, S, OCF 3, H, H, H, O], [AD506; CH, CH, CH, N, S, SCH 2 F, H, H, H, O ], [AD 507; CH, CH, CH, N, S, SCHF ₂ , H, H, H, O], [AD 508; CH, CH, CH, N, S, SCF ₃ , H, H, H, O] ], [AD 509; CH, CH, CH, N, S, CN, H, H, H, O], [AD 510; CH, CH, CH, N, S, NO ₂ , H, H, H, O] , [AD 511; N, N, CH, CH, S, H, H, H, H, O], [AD 512; N, N, CH, CH, S, F, H, H, H, O], [AD 511; AD 513; N, N, CH, CH, S, Cl, H, H, H, O], [AD 514; N, N, CH, CH, S, Br, H, H, H, O], [AD 515; N, N, CH, CH, S, I, H, H, H, O], [AD 516; N, N, CH, CH, S, Me, H, H, O], [AD 517; N, N, CH, CH, S, Et, H, H, H, O], [AD 518; N, N, CH, CH, S, Pr, H, H, H, O], [AD 519: N, N, N, CH, CH, S, i- Pr, H, H, H, O], [AD520; N, N, CH, CH, S, CH = CH 2, H, H, H, O], [AD521; N , N, CH, CH, S , C (CH 3) = CH 2, H, H, H, O], [AD522; N, N, CH, CH, S, C≡CH, H, H, H, O], [AD 523; N, N, CH, CH, S, C≡CCH ₃ , H, H, H, O], [AD 524: N, N, CH, CH, S, c-Pr, H, H , H, O], [AD 525; N, N, CH, CH, S, OMe, H, H, H, O], [AD 526; N, N, CH, CH, S, OE t, H, H, H N, N, CH, CH, S, Oi-Pr, H, H, H, O], [AD 528; N, N, CH, CH, S, SMe, H, H, H , O], [AD 529; N, N, CH, CH, S, SE t, H, H, H, O], [AD 530; N, N, CH, C _{H, S, CH 2 F,} H, H, H, O], [AD531; N, N, CH, CH, S, CHF 2, H, H, H, O], [AD532; N, N, CH _{, CH, S, CF 3,} H, H, H, O], [AD533; N, N, CH, CH, S, OCH 2 F, H, H, H, O], [AD534; N, N, _{CH, CH, S, OCHF 2} , H, H, H, O], [AD535; N, N, CH, CH, S, OCF 3, H, H, H, O], [AD536; N, N, CH, CH, S, SCH ₂ F, H, H, H, O], [AD 537; N, N, CH, CH, S, SCHF ₂ , H, H, H, O], [AD 538; N, N , CH, CH, S, SCF 3, H, H, H, O], [AD539; N, N, CH, CH, S, CN, H, H, H, O], [AD540; N, N, _{CH, CH, S, NO 2} , H, H, H, O], [AD541; N, CH, N, CH, S, H, H, H, H, O], [AD542; N, CH, N , CH, S, F, H, H, H, O, [AD 543; N, CH, N, CH, S, Cl, H, H, H, O], [AD 544; N, CH, N, CH , S, Br, H, H, H, O], [AD 545; N, CH, N, CH, S, I, H, H, H, O], [AD 546; N, CH, N, CH, S , Me, H, H, H, O], [AD 547; N, CH, N, CH, S, Et, H, H, H, O], [AD 548; N, CH, N, CH, S, Pr , H, H, H, O], [AD 549; N, CH, N, CH, S, i-Pr, H, H, H, O], [AD 550; N, CH, N, CH, S, CH _{= CH 2, H, H,} H, O], [AD551; N, CH, N, CH, S, C (CH 3) = CH 2, H, H, H, O], [AD552; N, CH , N, CH, S, C≡CH, H, H, H, O], [AD 553; N, CH, N, CH, S, C≡ CCH ₃ , H, H, H, O], [AD 554; N, CH, N, CH, S, c-Pr, H, H, H, O], [AD 555; N, CH, N, CH, S, OMe, H, H, H, O], [AD 556; N, CH, N, CH, S, OEt, H, H, H, O], [AD 557; N, CH, N, CH, S, Oi-Pr, H, H, H, O], [AD 558; N, CH, N, CH, S, SMe, H, H, H, O], [AD559; N, CH, N, CH, S, SE, H, H, H, O], [AD56 0; N, CH, N, CH, S, CH 2 F, H, H, H, O], [AD561; N, CH, N, CH, S, CHF 2, H, H, H, O], [AD562; N, CH, N , CH, S, CF 3, H, H, H, O], [AD563; N, CH, N, CH, S, OCH 2 F, H, H, H, O] , [AD564; N, CH, N, CH, S, OCHF 2, H, H, H, O], [AD565; N, CH, N, CH, S, OCF 3, H, H, H, O] , [AD566; N, CH, N, CH, S, SCH ₂ F, H, H, H, O], [AD 567; N, CH, N, CH, S, SCHF ₂ , H, H, H, O ], [AD568; N, CH , N, CH, S, SCF 3, H, H, H, O], [AD569; N, CH, N, CH, S, CN, H, H, H, O] , [AD570; N, CH, N, CH, S, NO 2, H, H, H, O], [AD571; N, CH, CH, N, S, H, H, H, H, O], [AD 572; N, CH, CH, N, S, F, H, H, H, O], [AD 573; N, CH, CH, N, S, Cl, H, H, H, O], [AD 574] N, CH, CH, N, S, Br, H, H, O], [AD 575; N, CH, CH, N, S, I, H, H, O], [AD 576; , CH, CH, N, S, Me, H, H, H, O], [AD 577; N, CH, CH, N, S, Et, H, H, O], [AD 578; N, CH , CH, N, S, Pr, H, H, H, O], [AD579; N, CH, CH, N, S, i-Pr, H, H, H, O], [AD 580; N, CH , CH, N, S, CH = CH 2, H, H, H, O], [AD581; N, CH, CH, N, S, C (CH 3) = CH 2, H, H, H, O N, CH, CH, N, S, C≡CH, H, H, H, O], [AD 583; N, CH, CH, N, S, C≡ CCH ₃ , H, H, H] H, O], [AD 584; N, CH, CH, N, S, c, Pr, H, H, H, O], [AD 585; N, CH, CH, N, S, OMe, H, H, H H, O], [AD 586; N, CH, CH, N, S, OEt, H, H, H, O], [AD 587; N, CH, CH, N, S, Oi-Pr, H, H, H, O], [AD 588; N, CH, CH, N, S, SMe, H, H, H, O], [AD 589; N, CH, CH, N, S, SE t, H, H, H H, O], [AD590; N, CH, CH, N, S, CH 2 F, H, H, H, O], [AD591; N, CH, CH, N, S, CHF 2, H, H , H, O], [AD592 ; N, CH, CH, N, S, CF 3, H, H, H, O], [AD593; N, CH, CH, N, S, OCH 2 F, H, H, H, O], [ AD594; N, CH, CH, N, S, OCHF 2, H, H, H, O], [AD595; N, CH, CH, N, S, OCF 3, H, H, H, O], [AD 596; N, CH, CH, N, S, SCH ₂ F, H, H, H, O], [AD 597; N, CH, CH, N, S, SCHF ₂ , H , H, H, O], [AD598; N, CH, CH, N, S, SCF 3, H, H, H, O], [AD599; N, CH, CH, N, S, CN, H, H, H, O], [ AD600; N, CH, CH, N, S, NO 2, H, H, H, O],

[AD601; CH, N, N, CH, S, H, H, H, H, O], [AD 602; CH, N, N, CH, S, F, H, H, O], [AD 603 CH, N, N, CH, S, Cl, H, H, H, O], [AD 604; CH, N, N, CH, S, Br, H, H, O], [AD 605; CH , N, N, CH, S, I, H, H, H, O], [AD 606; CH, N, N, CH, S, Me, H, H, O], [AD 607; CH, N , N, CH, S, Et, H, H, H, O], [AD 608; CH, N, N, CH, S, Pr, H, H, H, O], [AD 609; CH, N, N , CH, S, i-Pr , H, H, H, O], [AD610; CH, N, N, CH, S, CH = CH 2, H, H, H, O], [AD611; CH, N, N, CH, S, C (CH 3) = CH 2, H, H, H, O], [AD612; CH, N, N, CH, S, C≡CH, H, H, H, O ], [AD613; CH, N , N, CH, S, C≡CCH 3, H, H, H, O], [AD614; CH, N, N, CH, S, c-Pr, H, H, H, O], [AD 615; CH, N, N, CH, S, OMe, H, H, H, O], [AD 616; CH, N, N, CH, S, OEt, H, H, H, O], [AD 617; CH, N, N, CH, S, Oi-Pr, H, H, H, O], [AD 618; CH, N, N, CH, S, SMe, H, H, H, O], [AD 619; CH, N, N, CH, S, SE t, H, H, H, O], [AD 620; CH, N, N, CH, S, CH ₂ F, H, H, H, H O], [AD621; CH, N, N, CH, S, CHF 2, H, H, H, O], [AD622; CH, N, N, CH, S, CF 3, H, H, H, O], [AD623; CH, N, N, CH, S, OCH 2 F, H, H, H, O], [AD624; CH, N, N, CH, S, OCHF 2, H, H, H , O], [AD625; CH , N, N, CH, S, OCF 3, H, H, H, O], [AD626; CH, N, N, CH, S, SCH 2 F, H, H, H, O], [AD627; CH, N, N, CH, S, SCHF 2, H, H, H, O], [AD628; CH, N, N, CH, S, SCF 3, H, H, H, O], [AD 629; CH, N, N, CH, S, CN, H, H, H, O], [AD 630; CH, N, N, CH, S, NO ₂ , H, H, H, O], [AD 631; CH, N, CH, N, S, H, H, H, H, O], [AD 632; CH, N, CH, N, S, F, H , H, H, O], [AD 633; CH, N, CH, N, S, Cl, H, H, H, O], [AD 634; CH, N, CH, N, S, Br, H, H , H, O], [AD 635; CH, N, CH, N, S, I, H, H, H, O], [AD 636; CH, N, CH, N, S, Me, H, H, H , O], [AD 637; CH, N, CH, N, S, Et, H, H, H, O], [AD 638; CH, N, CH, N, S, Pr, H, H, H, O ], [AD639; CH, N , CH, N, S, i-Pr, H, H, H, O], [AD640; CH, N, CH, N, S, CH = CH 2, H, H, H, O], [AD641; CH, N, CH, N, S, C (CH 3) = CH 2, H, H, H, O], [AD642; CH, N, CH, N, S, C ≡CH, H, H, H, O], [AD643; CH, N, CH, N, S, C≡CCH ₃ , H, H, H, O], [AD 644; CH, N, CH, N, S, c-Pr, H, H, H, O, [AD 645; CH, N, CH, N, S, OMe, H, H, H, O], [AD 646; CH, N, CH, N, S, OEt, H, H, H, O], [AD 647; CH, N, CH, N, S, Oi-Pr, H, H, H, O], [AD 648; CH, N, CH, N, S, SMe, H, H, H, O], [AD 649; CH, N, CH, N, S, SE t, H, H, H, O], [AD 650; CH, N, CH, N, S, _{CH 2 F, H, H,} H, O], [AD651; CH, N, CH, N, S, CHF 2, H, H, H, O], [AD652; CH, N, CH, N, S _{, CF 3, H, H,} H, O], [AD653; CH, N, CH, N, S, OCH 2 F, H, H, H, O], [AD654; CH, N, CH, N, _{S, OCHF 2, H, H} , H, O], [AD655; CH, N, CH, N, S, OCF 3, H, H, H, O], [AD656; CH, N, CH, N, S, SCH ₂ F, H, H, H, O], [AD 657; CH, N, CH, N, S, SCHF ₂ , H, H, H, O], [AD 658; CH, N, CH, N , S, SCF ₃ , H, H, H, O], [AD 659; CH, N, CH, N, S, CN, H, H, H, O], [AD 660; CH, N, CH _{, N, S, NO 2,} H, H, H, O], [AD661; CH, CH, N, N, S, H, H, H, H, O], [AD662; CH, CH, N, N, S, F, H, H, H, O, [AD 663; CH, CH, N, N, S, Cl, H, H, H, O], [AD 664; CH, CH, N, N, S, Br, H, H, H, O], [AD 665; CH, CH, N, N, S, I, H, H, H, O], [AD 666; CH, CH, N, N, S, Me, H, H, H, O], [AD 667; CH, CH, N, N, S, Et, H, H, H, O], [AD 668; CH, CH, N, N, S, Pr, H, H, H, O], [AD 669; CH, CH, N, N, S, i-Pr, H, H, H, O], [AD 670; CH, CH, N, N, S, CH = CH ₂ , H, H, H, O, [AD 671; CH, CH, N, N, S, C (CH ₃ ) = CH ₂ , H, H, H, O], [AD 672; CH, CH, CH N, N, S, C≡CH, H, H, H, O], [AD 673; CH, CH, N, N, S, C≡ CCH ₃ , H, H, H, O], [AD 674; CH , CH, N, N, S, c-Pr, H, H, H, O], [AD 675; CH, CH, N, N, S, OMe, H, H, H] O, [AD 676; CH , CH, N, N, S, OEt, H, H, H, O], [AD 677; CH, CH, N, N, N, S, Oi-Pr, H, H, H, O], [AD 678; CH , CH, N, N, S, SMe, H, H, H, O], [AD 679; CH, CH, N, N, S, SE, H, H, H, O], [AD 680; CH, CH , N, N, S, CH 2 F, H, H, H, O], [AD681; CH, CH, N, N, S, CHF 2, H, H, H, O], [AD682; CH, CH, N, N, S, CF 3, H, H, H, O], [AD683; CH, CH, N, N, S, OCH 2 F, H, H, H, O], [AD684; CH , CH, N, N, S , OCHF 2, H, H, H, O], [AD685; CH, CH, N, N, S, OCF 3, H, H, H, O], [AD686; CH , CH, N, N, S, SCH ₂ F, H, H, H, O], [AD 687; CH, CH, N, N, S, SCHF ₂ , H, H, H, O], [AD 688; CH, CH, N, N, S, SCF 3, H, H, H, O], [AD689; CH, CH, N, N, S, CN, H, H, H, O], [AD6 90; CH, CH, N, N, S, NO 2, H, H, H, O], [AD691; N, CH, N, N, S, H, H, H, H, O], [AD692 N, CH, N, N, N, S, F, H, H, H, O], [AD 693; N, CH, N, N, S, Cl, H, H, O], [AD 694; N , CH, N, N, S, Br, H, H, H, O], [AD695; N, CH, N, N, S, I, H, H, O], [AD 696; N, CH N, N, S, Me, H, H, H, O, [AD 697; N, CH, N, N, S, Et, H, H, H, O], [AD 698; N, CH, N , N, S, Pr, H, H, H, H, O], [AD 699; N, CH, N, N, S, i-Pr, H, H, H, O], [AD 700; N, CH, N , N, S, CH = CH 2, H, H, H, O],

[AD701; N, CH, N , N, S, C (CH 3) = CH 2, H, H, H, O], [AD702; N, CH, N, N, S, C≡CH, H, H, H, O], [AD 703; N, CH, N, N, S, C≡CCH ₃ , H, H, H, O], [AD 704; N, CH, N, N, S, c-Pr , H, H, H, O], [AD 705; N, CH, N, N, S, OMe, H, H, H, O], [AD 706; N, CH, N, N, S, OEt, H , H, H, O], [AD 707; N, CH, N, N, S, Oi-Pr, H, H, H, O], [AD 708; N, CH, N, N, S, S Me, H , H, H, O], [AD 709; N, CH, N, N, S, SE t, H, H, H, O], [AD 710; N, CH, N, N, S, CH ₂ F, H , H, H, O], [AD711; N, CH, N, N, S, CHF 2, H, H, H, O], [AD712; N, CH, N, N, S, CF 3, H , H, H, O], [AD713; N, CH, N, N, S, OCH 2 F, H, H, H, O], [AD714; N, CH, N, N, S, OCHF 2, H, H, H, O] , [AD715; N, CH, N, N, S, OCF 3, H, H, H, O], [AD716; N, CH, N, N, S, SCH 2 F , H, H, H, O], [AD717; N, CH, N, N, S, SCHF ₂ , H, H, H, O], [AD 718; N, CH, N, N, S, SCF ₃ , H, H, H, O], [AD 719; N, CH, N, N, S, CN, H, H, H, O], [AD 720; N, CH, N, N, S, NO ₂ , H, H, H, H, O], [AD 721; CH, CH, CH, CH, CH, O, H, H, H, H, S], [AD 722: CH, CH, CH, CH, O, F, H, H H, H, S], [AD 723; CH, CH, CH, CH, CH, O, Cl, H, H, H, S], [AD 724; CH, CH, CH, CH, O, Br, H, H, H H, S], [AD 725; CH, CH, CH, CH, CH, O, I, H, H, H, S], [AD 726; CH, CH, CH, CH, O, Me, H, H, H, H, S], [AD 727; CH, CH, CH, CH, CH, O, Et, H, H, H, S], [AD 728; CH, CH, CH, CH, O, Pr, H, H, H, S] , [AD729; CH, CH, CH, CH, O, i-Pr, H, H, H, S], [AD730; CH, CH, CH, CH, O, CH = CH 2 , H, H, H, S ], [AD731; CH, CH, CH, CH, O, C (CH 3) = CH 2, H, H, H, S], [AD732; CH, CH, CH, CH, O, C≡CH, H, H, H, S], [AD733; CH, CH, CH, CH, O, C≡CCH 3, H, H, H, S], [AD734; CH, CH , CH, CH, O, c-Pr, H, H, H, S], [AD 735; CH, CH, CH, CH, CH, O, OMe, H, H, H, S], [AD 736; CH, CH , CH, CH, O, OEt, H, H, H, S], [AD 737; CH, CH, CH, CH, CH, O, Oi-Pr, H, H, H, S], [AD 738; CH, CH , CH, CH, O, SMe, H, H, H, S], [AD 739; CH, CH, CH, CH, CH, O, SE t, H, H, H, S], [AD 740; CH, CH, CH _{, CH, O, CH 2 F} , H, H, H, S], [AD741; CH, CH, CH, CH, O, CHF 2, H, H, H, S], [AD742; CH, CH, _{CH, CH, O, CF 3} , H, H, H, S], [AD743; CH, CH, CH, CH, O, OCH 2 F, H, H, H, S], [AD744; CH, CH , CH, CH, O, OCHF 2, H, H, H, S], [AD745; CH, CH, CH, CH, O, OCF 3, H, H, H, S], [AD746; CH, CH , CH, CH, O, SCH ₂ F, H, H, H, S], [AD 747; CH, CH, CH, CH, CH, O, SCHF ₂ , H, H, H, S], [AD 748; CH, CH, CH, CH, CH, O, SCF 3, H, H, H, S], [AD749; CH, CH, CH, CH, O, CN, H, H, H, S], [AD750; CH, CH , CH, CH, O, NO 2, H, H, H, S], [AD751; N, CH, CH, CH, O, H, H, H, H, S], [AD752; N, CH, CH, CH, O, F, H, H, H, S], [AD 753; N, CH, CH, CH, O, Cl, H, H, H, S], [AD 754; N, CH, CH, CH, O, Br, H, H, H, S, [AD 755; N, CH, CH, CH, O, I, H, H, H, S], [AD 756; N, CH, CH, CH, O, Me, H, H, H, S], [AD757; N, CH, CH, CH, O, Et, H, H, H, S], [AD 758; N, CH, CH, CH, O, Pr, H, H, H, S], [A D759; N, CH, CH, CH, O, i-Pr, H, H, H, S], [AD760; N, CH, CH, CH, O, CH = CH 2, H, H, H, S ], [AD761; N, CH , CH, CH, O, C (CH 3) = CH 2, H, H, H, S], [AD762; N, CH, CH, CH, O, C≡CH, H, H, H, S], [AD 763; N, CH, CH, CH, O, C≡CCH ₃ , H, H, H, S], [AD 764; N, CH, CH, CH, O, c -Pr, H, H, H, S], [AD 765; N, CH, CH, CH, O, OMe, H, H, H, S], [AD 766; N, CH, CH, CH, O, OEt , H, H, H, S], [AD 767; N, CH, CH, CH, O, Oi-Pr, H, H, H, S], [AD 768; N, CH, CH, CH, O, SMe , H, H, H, S], [AD 769; N, CH, CH, CH, O, SE t, H, H, H, S], [AD 770; N, CH, CH, CH, O, CH ₂ F , H, H, H, S ], [AD771; N, CH, CH, CH, O, CHF 2, H, H, H, S], [AD772; N, CH, CH, CH, O, CF 3 , H, H, H, S], [AD 773; N, CH, CH, CH, O, OCH ₂ F, H, H, H, S], [AD 774; N, CH, CH, CH, O, OCHF _{2, H, H, H,} S], [AD775; N, CH, CH, CH, O, OCF 3, H, H, H, S], [AD776; N, CH, CH, CH, O, SCH ₂ F, H, H, H, S], [AD 777; N, CH, CH, CH, O, SCHF ₂ , H, H, H, S], [AD 778; N, CH, CH, CH, O, SCF ₃ , H, H, H, S], [AD 779; N, CH, CH, CH, O, CN, H, H, H, S], [AD 780; N, CH, CH, CH, O, NO ₂ , H, H, H, S], [AD 781; CH, N, CH, CH, O, H, H, H, H, S], [AD 782; CH, N, CH, CH, O, F, H, H, H, S], [AD 783; CH, N, CH, CH, O, Cl, H, H, H, S], [AD 784; CH, N, CH, CH, O, Br, H, H, H, S], [AD 785; CH, N, CH, CH, O, I, H, H, H, S], [AD 786; CH, N, CH, CH, O, Me, H, H, H H, S], [AD 787; CH, N, CH, CH, O, Et, H, H , H, S], [AD 788; CH, N, CH, CH, O, Pr, H, H, H, S], [AD 789; CH, N, CH, CH, O, i-Pr, H, H , H, S], [AD790 ; CH, N, CH, CH, O, CH = CH 2, H, H, H, S], [AD791; CH, N, CH, CH, O, C (CH 3 ) = CH ₂ , H, H, H, S], [AD 792; CH, N, CH, CH, O, C≡CH, H, H, H, S], [AD 793; CH, N, CH, CH , O, C≡CCH ₃ , H, H, H, S], [AD 794; CH, N, CH, CH, O, c-Pr, H, H, H, S], [AD795; CH, N, CH, CH, O, OMe, H, H, H, S], [AD796; CH, N, CH, CH, O, OEt, H, H, H, S], [AD 797; CH, N, CH, CH, O, Oi-Pr, H, H, H, S, [AD 798; CH, N, CH, CH, O, SMe, H, H, H, S], [AD 799; CH, N, CH, CH, O, SEt, H, H, H, S], [AD 800; CH, N, CH, CH, O, CH ₂ F, H, H, H, S],

[AD801; CH, N, CH , CH, O, CHF 2, H, H, H, S], [AD802; CH, N, CH, CH, O, CF 3, H, H, H, S], [AD 803; CH, N, CH, CH, O, OCH ₂ F, H, H, H, S], [AD 804; CH, N, CH, CH, O, OCHF ₂ , H, H, H, S] , [AD805; CH, N, CH, CH, O, OCF 3, H, H, H, S], [AD806; CH, N, CH, CH, O, SCH 2 F, H, H, H, S ], [AD 807; CH, N, CH, CH, O, SCHF ₂ , H, H, H, S], [AD 808; CH, N, CH, CH, O, SCF ₃ , H, H, H, S ], [AD809; CH, N , CH, CH, O, CN, H, H, H, S], [AD810; CH, N, CH, CH, O, NO 2, H, H, H, S] [AD 811; CH, CH, N, CH, O, H, H, H, S], [AD 812; CH, CH, N, CH, O, F, H, H, H, S], [AD 811; AD 813; CH, CH, N, CH, O, Cl, H, H, S], [AD 814; CH, CH, N, CH, O, Br, H, H, H, S], [AD 815; CH, CH, N, CH, O, I, H, H, H, S], [AD 816; CH, CH, N, CH, O, Me, H, H, S, [AD 817; CH, CH, CH, N, CH, O, Et, H, H, H, S], [AD 818; CH, CH, N, CH, O, Pr, H, H, H, S], [AD 819; CH, CH, CH N, CH, O, i- Pr, H, H, H, S], [AD820; CH, CH, N, CH, O, CH = CH 2, H, H, H, S], [AD821; CH , CH, N, CH, O , C (CH 3) = CH 2, H, H, H, S], [AD822; CH, CH, N, CH, O, C≡CH, H, H, H, S], [AD 823; CH, CH, N, CH, O, C≡CCH ₃ , H, H, H, S], [AD 824; CH, CH, N, CH, O, c-Pr, H, H , H, S], [AD 825; CH, CH, N, CH, O, OMe, H, H, H, S], [AD 826; CH, CH, N, CH, O, OE t, H, H, H S, [AD 827; CH, CH, N, CH, O, Oi-Pr, H, H, H, S], [AD 828; CH, CH, N, CH, O, SMe, H, H, H , S], [AD 829; CH, CH, N, CH, O, SEt, H, H, H , S], [AD830; CH , CH, N, CH, O, CH 2 F, H, H, H, S], [AD831; CH, CH, N, CH, O, CHF 2, H, H, H, S], [AD832; CH, CH, N, CH, O, CF 3, H, H, H, S], [AD833; CH, CH, N, CH, O, OCH 2 F, H, H , H, S], [AD834 ; CH, CH, N, CH, O, OCHF 2, H, H, H, S], [AD835; CH, CH, N, CH, O, OCF 3, H, H , H, S], [AD 836; CH, CH, N, CH, O, SCH ₂ F, H, H, H, S], [AD 837; CH, CH, N, CH, O, SCHF ₂ , H, H, H, S], [ AD838; CH, CH, N, CH, O, SCF 3, H, H, H, S], [AD839; CH, CH, N, CH, O, CN, H, H , H, S], [AD840 ; CH, CH, N, CH, O, NO 2, H, H, H, S], [AD841; CH, CH, CH, N, O, H, H, H, H, S], [AD 842; CH, CH, CH, N, O, F, H, H, S], [AD 843; CH, CH, CH, N, O, Cl, H, H, H, H, H S], [AD844; CH, CH, CH, CH, N, O, Br, H, H, S], [AD 845; CH, CH, CH, N, O, I, H, H, H, S] [AD 846; CH, CH, CH, N, O, Me, H, H, H, S], [AD 847; CH, CH, CH, CH, N, O, Et, H, H, H, S], [AD 846; AD 848; CH, CH, CH, N, O, Pr, H, H, H, S], [AD 849; CH, CH, CH, N, O, i-Pr, H, H, H, S], [AD 8 49 AD 850; CH, CH, CH, N, O, CH = CH ₂ , H, H, H, S], [AD 851; CH, CH, CH, N, O, C (CH ₃ ) = CH ₂ , H, H, H, H, S], [AD 852; CH, CH, CH, N, O, C≡CH, H, H, H, S], [AD 853; CH, CH, CH, N, O, C≡ CCH ₃ , H, H, H, S], [AD 854; CH, CH, CH, N, O, c-Pr, H, H, H, S], [AD 855; CH, CH, CH, N, O, OMe , H, H, H, S], [AD 856; CH, CH, CH, N, O, OEt, H, H, H, S], [AD 857; CH, CH, CH, N, O, Oi-Pr , H, H, H, S], [AD 858; CH, CH, CH, N, O, SM e, H, H, H, S], [AD 859; CH, CH, CH, N, O, SE, H, H, H, S], [AD 860; CH, CH, CH, N, O, CH ₂ F, H, H, H, S], [AD861; CH, CH, CH, N, O, CHF 2, H, H, H, S], [AD862; CH, CH, CH, N, O, CF ₃ , H, H, H, S], [AD 863; CH, CH, CH, N, O, OCH ₂ F, H, H, H, S], [AD 864; CH, CH, CH, N, O, _{OCHF 2, H, H, H} , S], [AD865; CH, CH, CH, N, O, OCF 3, H, H, H, S], [AD866; CH, CH, CH, N, O, SCH ₂ F, H, H, H, S], [AD 867; CH, CH, CH, N, O, SCHF ₂ , H, H, H, S], [AD 868; CH, CH, CH, N, O , SCF ₃ , H, H, H, S], [AD 869; CH, CH, CH, N, O, CN, H, H, H, S], [AD 870; CH, CH, CH, N, O, _{NO 2, H, H, H} , S], [AD871; N, N, CH, CH, O, H, H, H, H, S], [AD872; N, N, CH, CH, O, F , H, H, H, S], [AD 873; N, N, CH, CH, O, Cl, H, H, H, S], [AD 874; N, N, CH, CH, O, Br, H , H, H, S], [AD 875; N, N, CH, CH, O, I, H, H, H, S], [AD 876; N, N, CH, CH, O, Me, H, H , H, S], [AD 877; N, N, CH, CH, O, Et, H, H, H, S], [AD 878; N, N, CH, CH, O, Pr, H, H, H , S], [AD879; N , N, CH, CH, O, i-Pr, H, H, H, S], [AD880; N, N, CH, CH, O, CH = CH 2, H, H, H, S], [ AD881; N, N, CH, CH, O, C (CH 3) = CH 2, H, H, H, S], [AD882; N, N, CH, CH, O , C≡CH, H, H, H, S], [AD 883; N, N, CH, CH, O, C≡ CCH ₃ , H, H, H, S], [AD 884; N, N, CH, CH, O, c-Pr, H, H, H, H, S], [AD885; N, N, CH, CH, O, OMe, H, H, H, S], [AD 886; N, N, CH, CH, O, OEt, H, H, H, S], [AD 887; N, N, CH, CH, O, Oi-Pr, H, H, H, S] , [AD 888; N, N, CH, CH, O, SMe, H, H, H, S], [AD 889; N, N, CH, CH, O, SE t, H, H, H, S], [ AD890; N, N, CH, CH, O, CH 2 F, H, H, H, S], [AD891; N, N, CH, CH, O, CHF 2, H, H, H, S], [AD892; N, N, CH , CH, O, CF 3, H, H, H, S], [AD893; N, N, CH, CH, O, OCH 2 F, H, H, H, S] , [AD894; N, N, CH, CH, O, OCHF 2, H, H, H, S], [AD895; N, N, CH, CH, O, OCF 3, H, H, H, S] , [AD 896; N, N, CH, CH, O, SCH ₂ F, H, H, H, S], [AD 897; N, N, CH, CH, O, SCHF ₂ , H, H, H, S N, N, CH, CH, O, SCF ₃ , H, H, H, S], [AD 899; N, N, CH, CH, O, CN, H, H, H, S] , [AD 900; N, N, CH, CH, O, NO ₂ , H, H, H, S],

[AD 901; N, CH, N, CH, O, H, H, H, S], [AD 902; N, CH, N, CH, O, F, H, H, H, S], [AD 903 N, CH, N, CH, O, Cl, H, H, H, S], [AD 904; N, CH, N, CH, O, Br, H, H, S, [AD 905; N] , CH, N, CH, O, I, H, H, H, S], [AD 906; N, CH, N, CH, O, Me, H, H, S, [AD 907; N, CH , N, CH, O, Et, H, H, H, S], [AD 908; N, CH, N, CH, O, Pr, H, H, H, S], [AD 909; N, CH, N , CH, O, i-Pr , H, H, H, S], [AD910; N, CH, N, CH, O, CH = CH 2, H, H, H, S], [AD911; N, CH, N, CH, O, C (CH 3) = CH 2, H, H, H, S], [AD912; N, CH, N, CH, O, C≡CH, H, H, H, S N, CH, N, CH, O, C≡CCH ₃ , H, H, H, S], [AD 914; N, CH, N, CH, O, c-Pr, H, H, H, S], [AD 915; N, CH, N, CH, O, OMe, H, H, H, S], [AD 916; N, CH, N, CH, O, OE t, H, H, H, S], [AD 917; N, CH, N, CH, O, Oi-Pr, H, H, H, S], [AD 918; N, CH, N, CH, O, SMe, H, H, H, S], [AD 919; N, CH, N, CH, O, SEt, H, H, H, S], [AD 920; N, CH, N, CH, O, CH ₂ F, H, H, H, S S], [AD921; N, CH, N, CH, O, CHF 2, H, H, H, S], [AD922; N, CH, N, CH, O, CF 3, H, H, H, S], [AD923; N, CH, N, CH, O, OCH 2 F, H, H, H, S], [AD924; N, CH, N, CH, O, OCHF 2, H, H, H , S], [AD925; N , CH, N, CH, O, OCF 3, H, H, H, S], [AD926; N, CH, N, CH, O, SCH 2 F, H, H, H, S], [AD927; N, CH, N, CH, O, SCHF 2, H, H, H, S], [AD928; N, CH, N, CH, O, SCF 3, H, H, H, S], [AD 929; N, CH, N, CH, O, CN, H, H, H, S], [AD 930; N, CH, N, CH, O, NO ₂ , H, H, H, S], [AD 931; N, CH, CH, N, O, H, H, H, H, S], [AD 932: N, CH, CH, N, O, F, H , H, H, S], [AD 933; N, CH, CH, N, O, Cl, H, H, H, S], [AD 934; N, CH, CH, N, O, Br, H, H , H, S], [AD 935; N, CH, CH, N, O, I, H, H, H, S], [AD 936; N, CH, CH, N, O, Me, H, H, H , S], [AD 937; N, CH, CH, N, O, Et, H, H, H, S], [AD 938; N, CH, CH, N, O, Pr, H, H, H, S ], [AD939; N, CH , CH, N, O, i-Pr, H, H, H, S], [AD940; N, CH, CH, N, O, CH = CH 2, H, H, H, S], [AD941; N, CH, CH, N, O, C (CH 3) = CH 2, H, H, H, S], [AD942; N, CH, CH, N, O, C ≡CH, H, H, H, S], [AD 943; N, CH, CH, N, O, C≡CCH ₃ , H, H, H, S], [AD 944; N, CH, CH, N, O, c-Pr, H, H, H, S, [AD 945; N, CH, CH, N, O, OMe, H, H, H, S], [AD 946; N, CH, CH, N, O, OEt, H, H, H, S], [AD 947; N, CH, CH, N, O, Oi-Pr, H, H, H, S], [AD 948; N, CH, CH, N, O, SMe, H, H, H, S], [AD 949; N, CH, CH, N, O, SE, H, H, H, S], [AD 950; N, CH, CH, N, O, _{CH 2 F, H, H,} H, S], [AD951; N, CH, CH, N, O, CHF 2, H, H, H, S], [AD952; N, CH, CH, N, O _{, CF 3, H, H,} H, S], [AD953; N, CH, CH, N, O, OCH 2 F, H, H, H, S], [AD954; N, CH, CH, N, _{O, OCHF 2, H, H} , H, S], [AD955; N, CH, CH, N, O, OCF 3, H, H, H, S], [AD956; N, CH, CH, N, O, SCH ₂ F, H, H, H, S], [AD 957; N, CH, CH, N, O, SCHF ₂ , H, H, H, S], [AD 958; N, CH, CH, N , O, SCF ₃ , H, H, H, S], [AD 959; N, CH, CH, N, O, CN, H, H, H, S], [AD 960; N, CH, CH _{, N, O, NO 2,} H, H, H, S], [AD961; CH, N, N, CH, O, H, H, H, H, S], [AD962; CH, N, N, CH, O, F, H, H, H, S], [AD 963; CH, N, N, CH, O, Cl, H, H, H, S], [AD 964; CH, N, N, CH, O, Br, H, H, H, S], [AD 965; CH, N, N, CH, O, I, H, H, H, S], [AD 966; CH, N, N, CH, O, Me, H, H, H, S], [AD 967; CH, N, N, CH, O, Et, H, H, H, S], [AD 968; CH, N, N, CH, O, Pr, H, H, H, S], [AD 969; CH, N, N, CH, O, i-Pr, H, H, H, S], [AD 970; CH, N, N, CH, O, CH = _{CH 2, H, H, H} , S], [AD971; CH, N, N, CH, O, C (CH 3) = CH 2, H, H, H, S], [AD972; CH, N, N, CH, O, C≡CH, H, H, H, S], [AD 973; CH, N, N, CH, O, C≡ CCH ₃ , H, H, H, S], [AD 974; CH , N, N, CH, O, c-Pr, H, H, H, S], [AD 975; CH, N, N, CH, O, OMe, H, H, H, S], [AD 976; CH , N, N, CH, O, OEt, H, H, H, S], [AD 977; CH, N, N, CH, O, Oi-Pr, H, H, H, S], [AD 978; CH , N, N, CH, O, SMe, H, H, H, S], [AD979; CH, N, N, CH, O, SE, H, H, H, S], [AD 980; CH, N , N, CH, O, CH 2 F, H, H, H, S], [AD981; CH, N, N, CH, O, CHF 2, H, H, H, S], [AD982; CH, N, N, CH, O, CF 3, H, H, H, S], [AD983; CH, N, N, CH, O, OCH 2 F, H, H, H, S], [AD984; CH , N, N, CH, O , OCHF 2, H, H, H, S], [AD985; CH, N, N, CH, O, OCF 3, H, H, H, S], [AD986; CH , N, N, CH, O, SCH ₂ F, H, H, H, S], [AD 987; CH, N, N, CH, O, SCHF ₂ , H, H, H, S], [AD 988; CH, N, N, CH, O, SCF 3, H, H, H, S], [AD989; CH, N, N, CH, O, CN, H, H, H, S], [AD9 90; CH, N, N, CH, O, NO 2, H, H, H, S], [AD991; CH, N, CH, N, O, H, H, H, H, S], [AD992 CH, N, CH, N, O, F, H, H, S], [AD 993; CH, N, CH, N, O, Cl, H, H, H, S], [AD 994; CH , N, CH, N, O, Br, H, H, H, S], [AD995; CH, N, CH, N, O, I, H, H, S], [AD 996; CH, N , CH, N, O, Me, H, H, H, S, [AD 997; CH, N, CH, N, O, Et, H, H, H, S], [AD 998; CH, N, CH , N, O, Pr, H, H, H, S, [AD 999; CH, N, CH, N, O, i-Pr, H, H, H, S], [AD 1000; CH, N, CH , N, O, CH = CH ₂ , H, H, H, S],

[AD1001; CH, N, CH , N, O, C (CH 3) = CH 2, H, H, H, S], [AD1002; CH, N, CH, N, O, C≡CH, H, H, H, S], [AD 1003; CH, N, CH, N, O, C≡CCH ₃ , H, H, H, S], [AD 1004; CH, N, CH, N, O, c-Pr , H, H, H, S], [AD 1005; CH, N, CH, N, O, OMe, H, H, H, S], [AD 1006; CH, N, CH, N, O, OE t, H , H, H, S], [AD 1007; CH, N, CH, N, O, Oi-Pr, H, H, H, S], [AD 1008; CH, N, CH, N, O, SMe, H , H, H, S], [AD 1009; CH, N, CH, N, O, SE, H, H, H, S], [AD 1010; CH, N, CH, N, O, CH ₂ F, H , H, H, S], [AD1011; CH, N, CH, N, O, CHF 2, H, H, H, S], [AD1012; CH, N, CH, N, O, CF 3, H , H, H, S], [AD1013; CH, N, CH, N, O, OCH 2 F, H, H, H, S], [AD1014; CH, N, CH, N, O, OCHF 2, H, H, H, S] , [AD1015; CH, N, CH, N, O, OCF 3, H, H, H, S], [AD1016; CH, N, CH, N, O, SCH 2 F , H, H, H, S], [AD 1017; CH, N, CH, N, O, SCHF ₂ , H, H, H, S], [AD 1018; CH, N, CH, N, O, SCF ₃ , H, H, H, S], [AD 1019; CH, N, CH, N, O, CN, H, H, H, S], [AD 1020; CH, N, CH, N, O, NO ₂ , H, H, H, S], [AD 1021; CH, CH, N, N, O, H, H, H, H, S], [AD 1022; CH, CH, N, N, O, F, H, H, H, S], [AD 1023; CH, CH, N, N, O, Cl, H, H, H, S], [AD 1024; CH, CH, N, N, N, O, Br, H, H, H H, S], [AD1025; CH, CH, N, N, O, I, H, H, S], [AD 1026; CH, CH, N, N, N, O, Me, H, H, H, H S], [AD 1027; CH, CH, N, N, N, O, Et, H, H, H, S], [AD 1028; CH, CH, N, N, O, Pr, H, H, H, S] , [AD 1029; CH, CH, N, N, O, i-Pr, H, H, H, S ], [AD1030; CH, CH , N, N, O, CH = CH 2, H, H, H, S], [AD1031; CH, CH, N, N, O, C (CH 3) = CH 2 , H, H, H, S], [AD 1032; CH, CH, N, N, O, C≡CH, H, H, H, S], [AD 1033; CH, CH, N, N, O, C ≡CCH ₃ , H, H, H, S], [AD 1034; CH, CH, N, N, O, c-Pr, H, H, H, S], [AD 10 35; CH, CH, N, N, O, OMe, H, H, H, S], [AD 1036; CH, CH, N, N, O, OEt, H, H, H, S], [AD 1037; CH, CH, N, N, O, Oi-Pr, H, H, H, S], [AD 1038; CH, CH, N, N, O, SMe, H, H, H, S], [AD 1039; CH, CH, N, N, O, SEt, H, H, H, S], [AD 1040; CH, CH, N, N, O, CH ₂ F, H, H, H, S], [AD 1041; CH, CH, N, N, O, _{CHF 2, H, H, H} , S], [AD1042; CH, CH, N, N, O, CF 3, H, H, H, S], [AD1043; CH, CH, N, N, O, OCH ₂ F, H, H, H, S], [AD 1044; CH, CH, N, N, O, OCHF ₂ , H, H, H, S], [AD 1045; CH, CH, N, N, O _{, OCF 3, H, H,} H, S], [AD1046; CH, CH, N, N, O, SCH 2 F, H, H, H, S], [AD1047; CH, CH, N, N, _{O, SCHF 2, H, H} , H, S], [AD1048; CH, CH, N, N, O, SCF 3, H, H, H, S], [AD1049; CH, CH, N, N, O, CN, H, H, H, S], [AD 1050; CH, CH, N, N, O, NO, NO ₂ , H, H, H, S], [AD 1051; N, CH, N, N, O , H, H, H, H, S], [AD 1052; N, CH, N, N, O, F, H, H, S, [AD 1053; N, CH, N, N, O, Cl , H, H, H, S], [AD1054; N, CH, N, N, O, Br, H, H, H, S], [AD 1055; N, CH, N, N, O, I, H , H, H, S], [AD 1056; N, CH, N, N, O, Me, H, H, H, S], [AD 1057; N, CH, N, N, O, Et, H, H , H, S], [AD 1058; N, CH, N, N, O, Pr, H, H, H, S], [AD1059; N, CH, N , N, O, i-Pr, H, H, H, S], [AD1060; N, CH, N, N, O, CH = CH 2, H, H, H, S], [AD 1061; N, CH, N, N, O, C, (CH ₃ ) = CH ₂ , H, H, H, S], [AD 1062; N, CH, N, N, O, C≡CH , H, H, H, S], [AD 1063; N, CH, N, N, O, C≡CCH ₃ , H, H, H, S], [AD 1064; N, CH, N, N, O, c-Pr, H, H, H, S], [AD 1065; N, CH, N, N, O, OMe, H, H, H, S], [AD 1066; N, CH, N, N, O, OEt, H, H, H, S], [AD 1067; N, CH, N, N, O, Oi-Pr, H, H, H, S], [AD 1068; N, CH, N, N, O, SMe, H, H, H, S], [AD 1069; N, CH, N, N, O, SE, H, H, H, S], [AD 1070; N, CH, N, N, O, CH ₂ F, H, H, H, S], [AD1071; N, CH, N, N, O, CHF 2, H, H, H, S], [AD1072; N, CH, N, N, O, CF ₃ , H, H, H, S], [AD 1073; N, CH, N, N, O, OCH ₂ F, H, H, H, S], [AD 1074; N, CH, N, N, O, _{OCHF 2, H, H, H} , S], [AD1075; N, CH, N, N, O, OCF 3, H, H, H, S], [AD1076; N, CH, N, N, O, SCH ₂ F, H, H, H, S], [AD 1077; N, CH, N, N, O, SCHF ₂ , H, H, H, S], [AD 1078; N, CH, N, N, O , SCF ₃ , H, H, H, S], [AD 1079; N, CH, N, N, O, CN, H, H, H, S], [AD 1080; N, CH, N, N, O, _{NO 2, H, H, H} , S], [AD1081; CH, CH, CH, CH, O, H, F, H, H, O], [AD1082; CH, CH, CH, CH, O, F , F, H, H, O], [AD1083; CH, CH, CH, CH, CH, O, Cl, F, H, H, O], [AD1084; CH, CH, CH, CH, O, Br, F , H, H, O], [AD 1085; CH, CH, CH, CH, CH, O, I, F, H, H, O], [AD 1086; CH, CH, CH, CH, O, Me, F, H , H, O], [AD 1087; CH, CH, CH, CH, O, Et, F, H, H, O], [AD1088; CH, CH, CH, CH, CH, O, Pr, F, H, H, O], [AD 1089; CH, CH, CH, CH, O, i-Pr, F, H, H, O], [AD1090; CH, CH, CH , CH, O, CH = CH 2, F, H, H, O], [AD1091; CH, CH, CH, CH, O, C (CH 3) = CH 2, F , H, H, O], [AD1092; CH, CH, CH, CH, O, C≡CH, F, H, H, O], [AD1093; CH, CH, CH, CH, O, C≡ CCH ₃ , F, H, H, O], [AD 1094; CH, CH, CH, CH, O, c-Pr, F, H, H, O], [AD 1095; CH, CH, CH, CH, O, OMe, F, H, H, O], [AD 1096; CH, CH, CH, CH, O, OEt, F, H, H, O], [AD 1097; CH, CH, CH, CH, O, Oi- Pr, F, H, H, O], [AD 1098; CH, CH, CH, CH, O, SMe, F, H, H, O], [AD 1099; CH, CH, CH, CH, O, SEt, F, H, H, O], [AD 1100; CH, CH, CH, CH, O, CH ₂ F, F, H, H, O],

[AD1101; CH, CH, CH , CH, O, CHF 2, F, H, H, O], [AD1102; CH, CH, CH, CH, O, CF 3, F, H, H, O], [AD1103; CH, CH, CH , CH, O, OCH 2 F, F, H, H, O], [AD1104; CH, CH, CH, CH, O, OCHF 2, F, H, H, O] , [AD1105; CH, CH, CH, CH, O, OCF 3, F, H, H, O], [AD1106; CH, CH, CH, CH, O, SCH 2 F, F, H, H, O ], [AD 1107; CH, CH, CH, CH, CH, O, SCHF ₂ , F, H, H, O], [AD 1108; CH, CH, CH, CH, O, SCF ₃ , F, H, H, O] ], [AD 1109; CH, CH, CH, CH, O, CN, F, H, H, O], [AD 1110; CH, CH, CH, CH, O, NO ₂ , F, H, H, O] [AD 1111, N, CH, CH, CH, CH, O, H, F, H, H, O], [AD 1112; N, CH, CH, CH, O, F, F, H, H, O], [AD 1112; AD 1113; N, CH, CH, CH, CH, O, Cl, F, H, H, O], [AD 1114; N, CH, CH, CH, O, Br, F, H, H, O], [AD 1115; N, CH, CH, CH, O, I, F, H, H, O], [AD 1116; N, CH, CH, CH, O, Me, F, H, O, [AD 1 117; N, CH, CH, CH, O, Et, F, H, H, O], [AD 1118; N, CH, CH, CH, O, Pr, F, H, H, O], [AD 1 119; N, CH, CH, CH, O, i- Pr, F, H, H, O], [AD1120; N, CH, CH, CH, O, CH = CH 2, F, H, H, O], [AD1121; N , CH, CH, CH, O , C (CH 3) = CH 2, F, H, H, O], [AD1122; N, CH, CH, CH, O, C≡CH, F, H, H, O], [AD 1123; N, CH, CH, CH, O, C≡CCH ₃ , F, H, H, O], [AD 1 124; N, CH, CH, CH, O, c-Pr, F, H , H, O], [AD 1 125; N, CH, CH, CH, O, OMe, F, H, H, O], [AD 1 126; N, CH, CH, CH, O, OEt, F, H, H N, CH, CH, CH, O, Oi-Pr, F, H, H, O], [AD 1 128; N, CH, CH, CH, O, SMe, F, H, H, O], [AD 1 129; N, CH, CH, CH, O, SE t, F, H, H, O], [AD 1130; N, CH, CH, CH, O, CH ₂ F, F, H, H, O], [AD 1131; N, CH, CH, CH, O, CHF ₂ , F, H, H, O], [AD 1132; N, CH, CH, CH, O, CF ₃ , F, H, H, O], [AD 1 133; N, CH, CH, CH, O, OCH ₂ F, F, H, H, O], [AD 1 134; N, CH, CH, CH, O, OCHF ₂ , F, H, H, O ], [AD1135; N, CH, CH, CH, O, OCF 3, F, H, H, O], [AD1136; N, CH, CH, CH, O, SCH 2 F, F, H, H, O], [AD 1137; N, CH, CH, CH, O, SCHF ₂ , F, H, H, O], [AD 1138; N, CH, CH, CH, O, SCF ₃ , F, H, H, O], [AD 1139; N, CH, CH, CH, O, CN, F, H, H, O], [AD 1 140; N, CH, CH, CH, O, NO ₂ , F, H, H, O], [AD 1141; CH, N, CH, CH, O, H, F, H, H, O], [AD 1142; CH, N, CH, CH, O, F, F , H, H, O], [AD1143; CH, N, CH, CH, O, Cl, F, H, H, O], [AD 1144; CH, N, CH, CH, O, Br, F, H , H, O], [AD 1145; CH, N, CH, CH, O, I, F, H, H, O], [AD 1146; CH, N, CH, CH, O, Me, F, H, H CH, N, CH, CH, O, Et, F, H, H, O], [AD 1148; CH, N, CH, CH, O, Pr, F, H, H, O ], [AD1149; CH, N , CH, CH, O, i-Pr, F, H, H, O], [AD1150; CH, N, CH, CH, O, CH = CH 2, F, H, H, O], [AD1151; CH, N, CH, CH, O, C (CH 3) = CH 2, F, H, H, O], [AD1152; CH, N, CH, CH, O, C ≡CH, F, H, H, O], [AD 1153; CH, N, CH, CH, O, C≡CCH ₃ , F, H, H, O], [AD 1154; CH, N, CH, CH, O, c-Pr, F, H, H, O], [AD 1 155; CH, N, CH, CH, O, OMe, F, H, H, O], [AD 1156; CH, N, CH, CH, O, OEt, F, H, H, O], [AD 1 157; CH, N, CH, CH, O, Oi-Pr, F, H, H, O], [AD 1158; CH, N, CH, CH, O, SMe, F, H, H, O], [AD 1159; CH, N, CH, CH, O, SE t, F, H, H, O], [AD 1 160; CH, N, CH, CH, O, CH ₂ F, F, H, H, O] , [AD1161; CH, N, CH, CH, O, CHF 2, F, H, H, O], [AD1162; CH, N, CH, CH, O, CF 3, F, H, H, O] , [AD1163; CH, N, CH, CH, O, OCH 2 F, F, H, H, O], [AD1164; CH, N, CH, CH, O, OCHF 2 , F, H, H, O ], [AD1165; CH, N, CH, CH, O, OCF 3, F, H, H, O], [AD1166; CH, N, CH, CH, O, SCH 2 F, F, H, H, O], [AD 1167; CH, N, CH, CH, O, SCHF ₂ , F, H, H, O], [AD 1 168; CH, N, CH, CH, O, SCF ₃ , F, H, H, O], [AD 1169; CH, N, CH, CH, O, CN, F, H, H, O], [AD 1170; CH, N, CH, CH, O, NO ₂ , F, H, H, O], [AD1171; CH, CH, N, CH, O, H, F, H, H, O], [AD1172; CH, CH, N, CH, O, F, F , H, H, O], [AD1173; CH, CH, N, CH, O, Cl, F, H, H, O], [AD 1174; CH, CH, N, CH, O, Br, F, H , H, O], [AD 1175; CH, CH, N, CH, O, I, F, H, H, O], [AD 1176; CH, CH, N, CH, O, Me, F, H, H CH, CH, N, CH, O, Et, F, H, H, O], [AD 1178; CH, CH, N, CH, O, Pr, F, H, H, O ], [AD1179; CH, CH , N, CH, O, i-Pr, F, H, H, O], [AD1180; CH, CH, N, CH, O, CH = CH 2, F, H, H, O], [AD1181; CH, CH, N, CH, O, C (CH 3) = CH 2, F, H, H, O], [AD1182; CH, CH, N, CH, O, C ≡CH, F, H, H, O], [AD1183; CH, CH, N, CH, O, C≡CCH 3, F, H, H, O], [AD1184; CH, CH, N, CH, O, cP r, F, H, H, O], [AD 1185; CH, CH, N, CH, O, OMe, F, H, H, O], [AD 1186; CH, CH, N, CH, O, OE t, F, H, H, O], [AD 1187; CH, CH, N, CH, O, Oi-Pr, F, H, H, O], [AD 1188; CH, CH, N, CH, O, SMe, F, H, H, O], [AD 1189; CH, CH, N, CH, O, SE t, F, H, H, O], [AD 1190; CH, CH, N, CH, O, CH ₂ F, F, H, H, O] , [AD1191; CH, CH, N, CH, O, CHF 2, F, H, H, O], [AD1192; CH, CH, N, CH, O, CF 3, F, H, H, O] , [AD1193; CH, CH, N, CH, O, OCH 2 F, F, H, H, O], [AD1194; CH, CH, N, CH, O, OCHF 2 , F, H, H, O ], [AD1195; CH, CH, N, CH, O, OCF 3, F, H, H, O], [AD1196; CH, CH, N, CH, O, SCH 2 F, F, H, H, O], [AD 1197; CH, CH, N, CH, O, SCHF ₂ , F, H, H, O], [AD 1198; CH, CH, N, CH, O, SCF ₃ , F, H, H, O], [AD 1199; CH, CH, N, CH, O, CN, F, H, H, O], [AD 1200; CH, CH, N, CH, O, NO ₂ , F, H, H, O],

[AD 1201; CH, CH, CH, N, O, H, F, H, O], [AD 1202; CH, CH, CH, CH, N, O, F, F, H, H, O], [AD 1203 CH, CH, CH, CH, N, O, Cl, F, H, H, O], [AD 1204; CH, CH, CH, CH, N, O, Br, F, H, H, O], [AD 1205; CH , CH, CH, N, O, I, F, H, H, O], [AD 1206; CH, CH, CH, CH, N, O, Me, F, H, O], [AD 1207; CH, CH , CH, N, O, Et, F, H, H, O], [AD 1208; CH, CH, CH, CH, N, O, Pr, F, H, H, O], [AD 1 209; CH, CH, CH , N, O, i-Pr , F, H, H, O], [AD1210; CH, CH, CH, N, O, CH = CH 2, F, H, H, O], [AD1211; CH, CH, CH, N, O, C (CH 3) = CH 2, F, H, H, O], [AD1212; CH, CH, CH, N, O, C≡CH, F, H, H, O ], [AD 1213; CH, CH, CH, N, O, C≡CCH ₃ , F, H, H, O], [AD 1214; CH, CH, CH, N, O, c-Pr, F, H, H, O], [AD 1215; CH, CH, CH, N, O, OMe, F, H, H, O], [AD 1216; CH, CH, CH, N, O, OE t, F, H, H, O], [AD 1217; CH, CH, CH, N, O, Oi-Pr, F, H, H, O], [AD 1218; CH, CH, CH, N, O, SMe, F, H, H, O, [AD 1219; CH, CH, CH, N, O, SE, SEt, F, H, H, O], [AD 1220; CH, CH, CH, N, O, CH ₂ F, F, H, H, O], [AD1221; CH, CH, CH, N, O, CHF 2, F, H, H, O], [AD1222; CH, CH, CH, N, O, CF 3, F, H, H, O], [AD1223; CH, CH, CH, N, O, OCH 2 F, F, H, H, O], [AD1224; CH, CH, CH, N, O, OCHF 2, F, H, H , O], [AD1225; CH , CH, CH, N, O, OCF 3, F, H, H, O], [AD1226; CH, CH, CH, N, O, SCH 2 F, F, H, H, O], [AD 1227; CH, CH, CH, N, O, SCHF ₂ , F, H, H, O], [AD 1228; CH, CH, CH, N, O, SCF ₃ , F, H, H, O] [AD 1229; CH, CH, CH, N, O, CN, F, H, H, O], [AD 1230; CH, CH, CH, N, O, NO ₂ , F, H, H, O], [AD 1231; N, N, CH, CH, O, H, F, H, H, O], [AD 1232; N, N, CH, CH, O, F, F, H, H, O], [AD 1233 N, N, CH, CH, O, Cl, F, H, H, O], [AD 1234; N, N, CH, CH, O, Br, F, H, H, O], [AD 1235; N , N, CH, CH, O, I, F, H, H, O], [AD 1236; N, N, CH, CH, O, Me, F, H, O], [AD 1237; N, N , CH, CH, O, Et, F, H, H, O], [AD 1238; N, N, CH, CH, O, Pr, F, H, H, O], [AD 1239; N, N, CH , CH, O, i-Pr , F, H, H, O], [AD1240; N, N, CH, CH, O, CH = CH 2, F, H, H, O], [AD1241; N, N, CH, CH, O, C (CH 3) = CH 2, F, H, H, O], [AD1242; N, N, CH, CH, O, C≡CH, F, H, H, O N, N, CH, CH, O, C≡CCH ₃ , F, H, H, O], [AD 1244; N, N, CH, CH, O, c-Pr, F, H, H, O], [AD 1245; N, N, CH, CH, O, OMe, F, H, H, O], [AD 1246; N, N, CH, CH, O, OEt, F, H, H, O], [AD 1247; N, N, CH, CH, O, Oi-Pr, F, H, H, O], [AD 1248; N, N, CH, CH, O, SMe, F, H, H, O], [AD 1249; N, N, CH, CH, O, SEt, F, H, H, O], [AD 1 250; N, N, CH, CH, O, CH ₂ F, F, H, H, O], [AD1251; N, N, CH, CH, O, CHF 2, F, H, H, O], [AD1252; N, N, CH, CH, O, CF 3, F, H, H, O], [AD1253; N, N, CH, CH, O, OCH 2 F, F, H, H, O], [AD1254; N, N, CH, CH, O, OCHF 2, F, H, H , O], [AD1255; N , N, CH, CH, O, OCF 3, F, H, H, O], [AD1256; N, N, CH, CH, O, SCH 2 F, F, H, H, O], [AD 1257; N, N, CH, CH, O, SCHF ₂ , F, H, H, O], [AD 1258; N, N, CH, CH, O, SCF ₃ , F, H, H, O], [AD 1259; N, N, CH, CH, O, CN, F, H , H, O], [AD1260 ; N, N, CH, CH, O, NO 2, F, H, H, O], [AD1261; N, CH, N, CH, O, H, F, H, H, O], [AD 1262; N, CH, N, CH, O, F, F, H, H, O], [AD 1263; N, CH, N, CH, O, Cl, F, H, H, O], [AD 1264; N, CH, N, CH, O, Br, F, H, O], [AD 1 265; N, CH, N, CH, O, I, F, H, H, O] , [AD1266; N, CH, N, CH, O, Me, F, H, H, O], [AD 1267; N, CH, N, CH, O, Et, F, H, H, O], [ AD1268; N, CH, N, CH, O, Pr, F, H, H, O], [AD 1269; N, CH, N, CH, O, i-Pr, F, H, H, O], [AD 1269; AD1270; N, CH, N, CH, O, CH = CH 2, F, H, H, O], [AD1271; N, CH, N, CH, O, C (CH 3) = CH 2, F, H, H, O], [AD 1272; N, CH, N, CH, O, C≡CH, F, H, H, O], [AD 1273; N, CH, N, CH, O, C≡ CCH ₃ , F, H, H, O], [AD 1274; N, CH, N, CH, O, c-Pr, F, H, H, O], [AD 1275; N, CH, N, CH, O, OMe , F, H, H, O], [AD 1276; N, CH, N, CH, O, OEt, F, H, H, O], [AD 1277; N, CH, N, CH, O, Oi-Pr , F, H, H, O], [AD 1278; N, CH, N, CH, O, SMe, F, H, O], [AD 1279; N, CH, N, CH, O, SE t, F , H, H, O], [AD1280; N, CH, N, CH, O, CH 2 F, F, H, H, O], [AD1281; N, CH, N, CH, O, CHF 2, F, H, H, O] , [AD1282; N, CH, N, CH, O, CF 3, F, H, H, O], [AD1283; N, CH, N, CH, O, OCH 2 F , F, H, H, O ], [AD1284; N, CH, N, CH, O, OCHF 2, F, H, H, O], [AD1285; N, CH, N, CH, O, OCF 3 , F, H, H, O], [AD 1286; N, CH, N, CH, O, SCH ₂ F , F, H, H, O], [AD 1287; N, CH, N, CH, O, SCHF ₂ , F, H, H, O], [AD 1 288; N, CH, N, CH, O, SCF ₃ , F, H, H, O], [AD1289; N, CH, N, CH, O, CN, F, H, H, O], [AD 1290; N, CH, N, CH, O, NO ₂ , F, H, H, O], [AD 1291; N, CH, CH, N, O, H, F, H, H, O], [AD 1292; N, CH, CH, N, O, F, F, H, H, O], [AD 1293; N, CH, CH, N, O, Cl, F, H, H, O], [AD 1 294; N, CH, CH, N, O, Br, F, H, H, O], [AD 1295; N, CH, CH, N, O, I, F, H, H, O], [AD 1296; N, CH, CH, N, O, Me, F, H, H, O], [AD 1297; N, CH, CH, N, O, Et, F, H, H, O], [AD 1298; N, CH, CH, N, O, Pr, F, H, H, O] , [AD1299; N, CH, CH, N, O, i-Pr, F, H, H, O], [AD1300; N, CH, CH, N, O, CH = CH 2, F, H, H , O],

[AD1301; N, CH, CH , N, O, C (CH 3) = CH 2, F, H, H, O], [AD1302; N, CH, CH, N, O, C≡CH, F, H, H, O], [ AD1303; N, CH, CH, N, O, C≡CCH 3, F, H, H, O], [AD1304; N, CH, CH, N, O, c-Pr , F, H, H, O], [AD 1305; N, CH, CH, N, O, OMe, F, H, H, O], [AD 1306; N, CH, CH, N, O, OEt, F , H, H, O], [AD 1307; N, CH, CH, N, O, Oi-Pr, F, H, H, O], [AD 1308; N, CH, CH, N, O, SMe, F , H, H, O], [AD 1309; N, CH, CH, N, O, SE t, F, H, H, O], [AD 1310; N, CH, CH, N, O, CH ₂ F, F , H, H, O], [AD 1311; N, CH, CH, N, O, CHF ₂ , F, H, H, O], [AD 1312; N, CH, CH, N, O, CF ₃ , F , H, H, O], [AD 1313; N, CH, CH, N, O, OCH ₂ F, F, H, H, O], [AD 1314; N, CH, CH, N, O, OCHF ₂ , F, H, H, O] , [AD1315; N, CH, CH, N, O, OCF 3, F, H, H, O], [AD1316; N, CH, CH, N, O, SCH 2 F , F, H, H, O], [AD 1317; N, CH, CH, N, O, SCHF ₂ , F, H, H, O], [AD 1318; N, CH, CH, N, O, SCF ₃ , F, H, H, O], [AD 1319; N, CH, CH, N, O, CN, F, H, H, O], [AD 1320; N, CH, CH, N, O, NO ₂ , F, H, H, O], [AD 1321; CH, N, N, CH, O, H, F, H, H, O], [AD 1322; CH, N, N, CH, O, F, F, H, H, O], [AD 1323; CH, N, N, CH, O, Cl, F, H, H, O], [AD 1324; CH, N, N, CH, O, Br, F, H, H, O], [AD 1325; CH, N, N, CH, O, I, F, H, H, O], [AD 1326; CH, N, N, CH, O, Me, F, H, H, O], [AD 1327; CH, N, N, CH, O, Et, F, H, H, O], [AD 1328; CH, N, N, CH, O, Pr, F, H, H, O] [AD 1329; CH, N, N, CH, O, i-Pr, F, H, H, O ], [AD1330; CH, N , N, CH, O, CH = CH 2, F, H, H, O], [AD1331; CH, N, N, CH, O, C (CH 3) = CH 2 , F, H, H, O], [AD1332; CH, N, N, CH, O, C≡CH, F, H, H, O], [AD 1333; CH, N, N, CH, O, C ≡CCH ₃ , F, H, H, O], [AD 1334; CH, N, N, CH, O, c-Pr, F, H, H, O], [AD 1335; CH, N, N, CH, O, OMe, F, H, H, O], [AD 1336; CH, N, N, CH, O, OEt, F, H, H, O], [AD 1337; CH, N, N, CH, O, Oi-Pr, F, H, H, O], [AD 1338; CH, N, N, CH, O, SMe, F, H, H, O], [AD 1339; CH, N, N, CH, O, SEt, F, H, H, O], [AD 1340; CH, N, N, CH, O, CH ₂ F, F, H, H, O], [AD 1341; CH, N, N, CH, O, _{CHF 2, F, H, H} , O], [AD1342; CH, N, N, CH, O, CF 3, F, H, H, O], [AD1343; CH, N, N, CH, O, OCH ₂ F, F, H, H, O], [AD 1344; CH, N, N, CH, O, OCHF ₂ , F, H, H, O], [AD 1 345; CH, N, N, CH, O _{, OCF 3, F, H,} H, O], [AD1346; CH, N, N, CH, O, SCH 2 F, F, H, H, O], [AD1347; CH, N, N, CH, _{O, SCHF 2, F, H} , H, O], [AD1348; CH, N, N, CH, O, SCF 3, F, H, H, O], [AD1349; CH, N, N, CH, O, CN, F, H, H, O], [AD 1350; CH, N, N, CH, O, NO ₂ , F, H, H, O], [AD 1351; CH, N, CH, N, O , H, F, H, H, O], [AD 1352; CH, N, CH, N, O, F, F, H, H, O], [AD 1353; CH, N, CH, N, O, Cl , F, H, H, O], [AD 1 354; CH, N, CH, N, O, Br, F, H, H] O, [AD 1 355; CH, N, CH, N, O, I, F , H, H, O], [AD 1356; CH, N, CH, N, O, Me, F, H, H, O], [AD 1 357; CH, N, CH, N, O, Et, F, H , H, O], [AD 1358; CH, N, CH, N, O, Pr, F , H, H, O], [AD 1359; CH, N, CH, N, O, i-Pr, F, H, H, O], [AD 1 360; CH, N, CH, N, O, CH = CH _{2, F, H, H,} O], [AD1361; CH, N, CH, N, O, C (CH 3) = CH 2, F, H, H, O], [AD1362; CH, N, CH , N, O, C≡CH, F, H, H, O], [AD 1363; CH, N, CH, N, O, C≡ CCH ₃ , F, H, H, O], [AD 1364; CH, N, CH, N, O, c-Pr, F, H, H, O], [AD 1365; CH, N, CH, N, O, OMe, F, H, H, O], [AD 1 366; CH, N, CH, N, O, OEt, F, H, H, O], [AD 1367; CH, N, CH, N, O, Oi-Pr, F, H, H, O], [AD 1 368; CH, N, CH, N, O, SMe, F, H, H, O], [AD 1369; CH, N, CH, N, O, SE, F, H, H, O], [AD 1 370; CH, N, _{CH, N, O, CH 2} F, F, H, H, O], [AD1371; CH, N, CH, N, O, CHF 2, F, H, H, O], [AD1372; CH, N , CH, N, O, CF 3, F, H, H, O], [AD1373; CH, N, CH, N, O, OCH 2 F, F, H, H, O], [AD1374; CH, N, CH, N, O, OCHF 2, F, H, H, O], [AD1375; CH, N, CH, N, O, OCF 3, F, H, H, O], [AD1376; CH, N, CH, N, O, SCH ₂ F, F, H, H, O], [AD 1377; CH, N, CH, N, O, SCHF ₂ , F, H, H, O], [AD 1378; CH , N, CH, N, O , SCF 3, F, H, H, O], [AD1379; CH, N, CH, N, O, CN, F, H, H, O], [AD1380; CH, N, CH, N, O, NO 2, F, H, H, O], [AD1381; CH, CH, N, N, O, H, F, H, H, O], [AD1382; CH, CH , N, N, O, F, F, H, H, O], [AD 1383; CH, CH, N, N, N, O, Cl, F, H, H, O], [AD 1384; CH, CH, N , N, O, Br, F, H, H, O], [AD 1385; CH, CH, N, N, O, I, F, H, H, O], [AD 1 386; CH, CH, N, N , O, Me, F, H, H, O], [AD 1387; CH, CH, N, N, O, Et, F, H, H, O], [AD 1388; CH, CH, N, N, O, Pr, F, H, H, O], [AD 1 389; CH, CH, N, N, O, i-Pr, F, H, H, O], [AD1390; CH, CH, N, N, O, CH = CH 2, F, H, H, O], [AD1391; CH, CH, N , N, O, C (CH 3) = CH 2, F, H, H, O], [AD1392; CH, CH, N, N, O, C≡CH, F, H, H, O], [ AD1393; CH, CH, N, N, O, C≡CCH 3, F, H, H, O], [AD1394; CH, CH, N, N, O, c-Pr, F, H, H, O ], [AD 1395; CH, CH, N, N, O, O, OMe, F, H, H, O], [AD 1396; CH, CH, N, N, O, OEt, F, H, H, O], [AD 1397; CH, CH, N, N, N, O, Oi-Pr, F, H, H, O], [AD 1398; CH, CH, N, N, O, SMe, F, H, H, O], [AD 1399; CH, CH, N, N, N, O, SEt, F, H, H, O], [AD 1400; CH, CH, N, N, N, O, CH ₂ F, F, H, H, O],

[AD1401; CH, CH, N , N, O, CHF 2, F, H, H, O], [AD1402; CH, CH, N, N, O, CF 3, F, H, H, O], [AD1403; CH, CH, N , N, O, OCH 2 F, F, H, H, O], [AD1404; CH, CH, N, N, O, OCHF 2, F, H, H, O] , [AD1405; CH, CH, N, N, O, OCF 3, F, H, H, O], [AD1406; CH, CH, N, N, O, SCH 2 F, F, H, H, O ], [AD 1407; CH, CH, N, N, N, O, SCHF ₂ , F, H, H, O], [AD 1408; CH, CH, N, N, O, SCF ₃ , F, H, H, O ], [AD 1409; CH, CH, N, N, O, CN, F, H, H, O], [AD 1410; CH, CH, N, N, O, NO ₂ , F, H, H, O] , [AD 1411; N, CH, N, N, O, H, F, H, O], [AD 1412; N, CH, N, N, O, F, F, H, H, O], [AD 1412; AD 1413; N, CH, N, N, N, O, Cl, F, H, H, O], [AD 1414; N, CH, N, N, N, O, Br, F, H, H, O], [AD 1415; N, CH, N, N, N, O, I, F, H, H, O], [AD 1416; N, CH, N, N, O, Me, F, H, O], [AD 1417; N, CH, N, N, O, Et, F, H, H, O], [AD1418; N, CH, N, N, O, Pr, F, H, H, O], [AD 1419; N, CH, N, N, O, i- Pr, F, H, H, O], [AD1420; N, CH, N, N, O, CH = CH 2, F, H, H, O], [AD1421; N , CH, N, N, O , C (CH 3) = CH 2, F, H, H, O], [AD1422; N, CH, N, N, O, C≡CH, F, H, H, O, [AD 1423; N, CH, N, N, O, C≡CCH ₃ , F, H, H, O], [AD 1424; N, CH, N, N, O, c-Pr, F, H , H, O], [AD 1425; N, CH, N, N, O, OMe, F, H, H, O], [AD 1426; N, CH, N, N, O, OEt, F, H, H , O], [AD 1427; N, CH, N, N, O, Oi-Pr, F, H, H, O], [AD 1428; N, CH, N, N, O, SMe, F, H, H , O], [AD 1429; N, CH, N, N, O, SE, t, F, H, H, O], [AD 1430; N, CH, N, _{N, O, CH 2 F,} F, H, H, O], [AD1431; N, CH, N, N, O, CHF 2, F, H, H, O], [AD1432; N, CH, N _{, N, O, CF 3,} F, H, H, O], [AD1433; N, CH, N, N, O, OCH 2 F, F, H, H, O], [AD1434; N, CH, _{N, N, O, OCHF 2} , F, H, H, O], [AD1435; N, CH, N, N, O, OCF 3, F, H, H, O], [AD1436; N, CH, N, N, O, SCH ₂ F, F, H, H, O, [AD 1437; N, CH, N, N, N, O, SCHF ₂ , F, H, H, O], [AD 1438; N, CH , N, N, O, SCF 3, F, H, H, O], [AD1439; N, CH, N, N, O, CN, F, H, H, O], [AD1440; N, CH, _{N, N, O, NO 2} , F, H, H, O], [AD1441; CH, CH, CH, CH, O, H, H, F, H, O], [AD1442; CH, CH, CH , CH, O, F, H, F, H, O], [AD 1443; CH, CH, CH, CH, CH, O, Cl, H, F, H, O], [AD 1444; CH, CH, CH, CH , O, Br, H, F, H, O], [AD 1445; CH, CH, CH, CH, CH, O, I, H, F, H, O], [AD 1446; CH, CH, CH, CH, O , Me, H, F, H, O], [AD 1447; CH, CH, CH, CH, CH, O, Et, H, F, H, O], [AD 1448; CH, CH, CH, CH, O, Pr , H, F, H, O], [AD 1449; CH, CH, CH, CH, O, i-Pr, H, F, H, O], [AD 1450; CH, CH, CH, CH, O, CH = CH ₂ , H, F, H, O], [AD 1451; CH, CH, CH, CH, CH, O, C (CH ₃ ) = CH ₂ , H, F, H, O], [AD 1452; CH, CH , CH, CH, O, C≡CH, H, F, H, O], [AD 1453; CH, CH, CH, CH, CH, O, C≡ CCH ₃ , H, F, H, O], [AD 1454; CH, CH, CH, CH, CH, O, c-Pr, H, F, H, O], [AD 1455; CH, CH, CH, CH, O, OMe, H, F, H, O], [AD 1456; CH, CH, CH, CH, CH, O, OEt, H, F, H, O], [AD 1457; CH, CH, CH, CH, O, Oi-Pr, H, F, H, O], [AD 1458; CH, CH, CH, C H, O, SMe, H, F, H, O], [AD1459; CH, CH, CH, CH, O, SEt, H, F, H, O], [AD 1460; CH, CH, CH, CH, _{O, CH 2 F, H,} F, H, O], [AD1461; CH, CH, CH, CH, O, CHF 2, H, F, H, O], [AD1462; CH, CH, CH, CH _{, O, CF 3, H,} F, H, O], [AD1463; CH, CH, CH, CH, O, OCH 2 F, H, F, H, O], [AD1464; CH, CH, CH, _{CH, O, OCHF 2, H} , F, H, O], [AD1465; CH, CH, CH, CH, O, OCF 3, H, F, H, O], [AD1466; CH, CH, CH, CH, O, SCH ₂ F, H, F, H, O], [AD 1467; CH, CH, CH, CH, CH, O, SCHF ₂ , H, F, H, O], [AD 1468; CH, CH, CH _{, CH, O, SCF 3,} H, F, H, O], [AD1469; CH, CH, CH, CH, O, CN, H, F, H, O], [AD1470; CH, CH, CH, _{CH, O, NO 2, H} , F, H, O], [AD1471; N, CH, CH, CH, O, H, H, F, H, O], [AD1472; N, CH, CH, CH , O, F, H, F, H, O], [AD 1 473; N, CH, CH, CH, O, Cl, H, F, H, O], [AD 1474; N, CH, CH, CH, O Br, H, F, H, O], [AD 1475; N, CH, CH, CH, O, I, H, F, H, O], [AD 1476; N, CH, CH, CH, O, Me , H, F, H, O], [AD 1477; N, CH, CH, CH, O, Et, H, F, H, O], [AD 1478; N, CH, CH, CH, O, Pr, H , F, H, O], [AD 1479; N, CH, CH, CH, O, i-Pr, H, F, H, O], [AD 1480; N, CH, CH, CH, O, CH = CH _{2, H, F, H,} O], [AD1481; N, CH, CH, CH, O, C (CH 3) = CH 2, H, F, H, O], [AD1482; N, CH, CH , CH, O, C≡CH, H, F, H, O], [AD 1483; N, CH, CH, CH, O, C≡ CCH ₃ , H, F, H, O], [AD 1484; N, CH, CH, CH, O, c, Pr, H, F, H, O], [AD 1 485; N, CH, CH, CH, O, OMe, H, F, H, O], [AD 14 86; N, CH, CH, CH, CH, O, OEt, H, F, H, O], [AD 1487; N, CH, CH, CH, O, Oi-Pr, H, F, H, O], [[ AD 1488; N, CH, CH, CH, CH, O, SMe, H, F, H, O], [AD 1489; N, CH, CH, CH, O, SE t, H, F, H, O], [AD 1490; N, CH, CH, CH, O, CH 2 F, H, F, H, O], [AD1491; N, CH, CH, CH, O, CHF 2, H, F, H, O], [AD1492 ; N, CH, CH, CH , O, CF 3, H, F, H, O], [AD1493; N, CH, CH, CH, O, OCH 2 F, H, F, H, O], [ AD1494; N, CH, CH, CH, O, OCHF 2, H, F, H, O], [AD1495; N, CH, CH, CH, O, OCF 3, H, F, H, O], [ AD1496; N, CH, CH, CH, O, SCH ₂ F, H, F, H, O], [AD 1497; N, CH, CH, CH, O, SCHF ₂ , H, F, H, O], [AD 1498; N, CH, CH, CH, O, SCF ₃ , H, F, H, O], [AD 1499; N, CH, CH, CH, O, CN, H, F, H, O], AD 1500; N, CH, CH, CH, O, NO ₂ , H, F, H, O],

[AD 1501; CH, N, CH, CH, O, H, H, F, H, O], [AD 1502; CH, N, CH, CH, O, F, H, F, H, O], [AD 1503 CH, N, CH, CH, O, Cl, H, F, H, O], [AD 1504; CH, N, CH, CH, O, Br, H, F, H, O], [AD 1505; CH , N, CH, CH, O, I, H, F, H, O], [AD 1506; CH, N, CH, CH, O, Me, H, F, H, O], [AD 1507; CH, N , CH, CH, O, Et, H, F, H, O], [AD1508; CH, N, CH, CH, O, Pr, H, F, H, O], [AD 1509; CH, N, CH , CH, O, i-Pr , H, F, H, O], [AD1510; CH, N, CH, CH, O, CH = CH 2, H, F, H, O], [AD1511; CH, N, CH, CH, O, C (CH 3) = CH 2, H, F, H, O], [AD1512; CH, N, CH, CH, O, C≡CH, H, F, H, O ], [AD1513; CH, N , CH, CH, O, C≡CCH 3, H, F, H, O], [AD1514; CH, N, CH, CH, O, c-Pr, H, F, H, O], [AD 1515; CH, N, CH, CH, O, OMe, H, F, H, O], [AD 1516; CH, N, CH, CH, O, OE t, H, F, H, O, [AD 1517; CH, N, CH, CH, O, Oi-Pr, H, F, H, O], [AD 1518; CH, N, CH, CH, O, SMe, H, F, H, O, [AD 1519; CH, N, CH, CH, O, SEt, H, F, H, O], [AD 1520; CH, N, CH, CH, O, CH ₂ F, H, F, H, O], [AD1521; CH, N, CH, CH, O, CHF 2, H, F, H, O], [AD1522; CH, N, CH, CH, O, CF 3, H, F, H, O], [AD1523; CH, N, CH, CH, O, OCH 2 F, H, F, H, O], [AD1524; CH, N, CH, CH, O, OCHF 2, H, F, H , O], [AD1525; CH , N, CH, CH, O, OCF 3, H, F, H, O], [AD1526; CH, N, CH, CH, O, SCH 2 F, H, F, H, O], [AD1527; CH, N, CH, CH, O, SCHF 2, H, F, H, O], [AD1528; CH, N, CH, CH, O, SCF 3, H, F, H, O] [AD 1529; CH, N, CH, CH, O, CN, H, F, H, O], [AD 1530; CH, N, CH, CH, O, NO ₂ , H, F, H, O], [AD 1531; CH, CH, N, CH, O, H, H, F, H, O], [AD 1532; CH, CH, N, CH, O, F, H, F, H, O], [AD 1533 CH, CH, N, CH, O, Cl, H, F, H, O], [AD1534; CH, CH, N, CH, O, Br, H, F, H, O], [AD 1535; CH , CH, N, CH, O, I, H, F, H, O], [AD 1536; CH, CH, N, CH, O, Me, H, F, H, O], [AD 1537; CH, CH , N, CH, O, Et, H, F, H, O], [AD1538; CH, CH, N, CH, O, Pr, H, F, H, O], [AD1539; CH, CH, N , CH, O, i-Pr , H, F, H, O], [AD1540; CH, CH, N, CH, O, CH = CH 2, H, F, H, O], [AD1541; CH, CH, N, CH, O, C (CH 3) = CH 2, H, F, H, O], [AD1542; CH, CH, N, CH, O, C≡CH, H, F, H, O , [AD 1543; CH, CH, N, CH, O, C≡CCH ₃ , H, F, H, O], [AD 1544; CH, CH, N, CH, O, c-Pr, H, F, H, O], [AD1545; CH, CH, N, CH, O, OMe, H, F, H, O], [AD 1546; CH, CH, N, CH, O, OEt, H, F, H, O, [AD1547; CH, CH, N, CH, O, Oi-Pr, H, F, H, O], [AD 1548; CH, CH, N, CH, O, SMe, H, F, H, CH, CH, N, CH, O, SEt, H, F, H, O], [AD 1550; CH, CH, N, CH, O, CH ₂ F, H, F, H, O], [AD 1 549; O], [AD1551; CH, CH, N, CH, O, CHF 2, H, F, H, O], [AD1552; CH, CH, N, CH, O, CF 3, H, F, H, O], [AD1553; CH, CH, N, CH, O, OCH 2 F, H, F, H, O], [AD1554; CH, CH, N, CH, O, OCHF 2, H, F, H , O], [AD1555; CH , CH, N, CH, O, OCF 3, H, F, H, O], [AD1556; CH, CH, N, CH, O, SCH 2 F, H, F, H, O], [AD 1 557; CH, CH, N, CH, O, SCHF ₂ , H, F, H, O], [AD 1558; CH, CH, N, CH, O, SCF ₃ , H, F, H, O], [ AD 1559; CH, CH, N, CH, O, CN, H, F, H, O], [AD 1560; CH, CH, N, CH, O, NO ₂ , H, F, H, O], [AD 1561 CH, CH, CH, N, O, H, H, F, H, O], [AD1562; CH, CH, CH, N, O, F, H, F, H, O], [AD 1563; CH , CH, CH, N, O, Cl, H, F, H, O], [AD 1564; CH, CH, CH, CH, N, O, Br, H, F, H, O], [AD 1 565; CH, CH , CH, N, O, I, H, F, H, O], [AD 1 566; CH, CH, CH, CH, N, O, Me, H, F, H, O], [AD 1567; CH, CH, CH , N, O, Et, H, F, H, O], [AD1568; CH, CH, CH, N, O, Pr, H, F, H, O], [AD 1569; CH, CH, CH, N , O, i-Pr, H , F, H, O], [AD1570; CH, CH, CH, N, O, CH = CH 2, H, F, H, O], [AD1571; CH, CH, CH, N, O, C ( CH 3) = CH 2, H, F, H, O], [AD1572; CH, CH, CH, N, O, C≡CH, H, F, H, O], [AD 1573; CH, CH, CH, N, O, C≡CCH ₃ , H, F, H, O], [AD 1574; CH, CH, CH, N, O, c-Pr, H, F, H, O], [AD 1575; CH, CH, CH, N, O, O, OMe, H, F, H, O], [AD 1 576; CH, CH, CH, N, O, OEt, H, F, H, O] , [AD 1577; CH, CH, CH, N, O, Oi-Pr, H, F, H, O], [AD 1578; CH, CH, CH, N, O, SMe, H, F, H, O] , [AD1579; CH, CH, CH, N, O, SE, H, F, H, O], [AD 1580; CH, CH, CH, N, O, CH ₂ F, H, F, H, O] , [AD1581; CH, CH, CH, N, O, CHF 2, H, F, H, O], [AD1582; CH, CH, CH, N, O, CF 3, H, F, H, O] , [AD1583; CH, CH, CH, N, O, OCH 2 F, H, F, H, O], [AD1584; CH, CH, CH, N, O, OCHF 2, H, F, H, O ], [AD 1585; C H, CH, CH, N, O, OCF 3, H, F, H, O], [AD1586; CH, CH, CH, N, O, SCH 2 F, H, F, H, O], [AD1587 ; CH, CH, CH, N , O, SCHF 2, H, F, H, O], [AD1588; CH, CH, CH, N, O, SCF 3, H, F, H, O], [AD1589 CH, CH, CH, N, O, CN, H, F, H, O], [AD 1590; CH, CH, CH, N, O, NO ₂ , H, F, H, O], [AD 1591; N, N, CH, CH, O, H, H, F, H, O], [AD1592; N, N, CH, CH, O, F, H, F, H, O], [AD 1593; N, N, CH, CH, O, Cl, H, F, H, O], [AD1594; N, N, CH, CH, O, Br, H, F, H, O], [AD 1595; N, N, CH, CH, O, I, H, F, H, O], [AD 1596; N, N, CH, CH, O, Me, H, F, H, O], [AD 1597; N, N, CH, CH, O, Et, H, F, H, O], [AD 1598; N, N, CH, CH, O, Pr, H, F, H, O], [AD 1599; N, N, CH, CH, O, i-Pr, H, F, H, O], [AD1600; N, N, CH, CH, O, CH = CH 2, H, F, H, O],

[AD1601; N, N, CH , CH, O, C (CH 3) = CH 2, H, F, H, O], [AD1602; N, N, CH, CH, O, C≡CH, H, F, H, O], [AD 1603; N, N, CH, CH, O, C≡CCH ₃ , H, F, H, O], [AD 1604; N, N, CH, CH, O, c-Pr , H, F, H, O], [AD 1605; N, N, CH, CH, O, OMe, H, F, H, O], [AD 1606; N, N, CH, CH, O, OEt, H , F, H, O], [AD 1607; N, N, CH, CH, O, Oi-Pr, H, F, H, O], [AD 1608; N, N, CH, CH, O, SMe, H , F, H, O], [AD 1609; N, N, CH, CH, O, SE t, H, F, H, O], [AD 1610; N, N, CH, CH, O, CH ₂ F, H , F, H, O], [AD 1611; N, N, CH, CH, O, CHF ₂ , H, F, H, O], [AD 1612; N, N, CH, CH, O, CF ₃ , H , F, H, O], [AD 1613; N, N, CH, CH, O, OCH ₂ F, H, F, H, O], [AD 1614; N, N, CH, CH, O, OCHF ₂ , H, F, H, O] , [AD1615; N, N, CH, CH, O, OCF 3, H, F, H, O], [AD1616; N, N, CH, CH, O, SCH 2 F , H, F, H, O], [AD 1617; N, N, CH, CH, O, SCHF ₂ , H, F, H, O], [AD 1618; N, N, CH, CH, O, SCF ₃ , H, F, H, O], [AD 1619; N, N, CH, CH, O, CN, H, F, H, O], [AD 1620; N, N, CH, CH, O, NO ₂ , H, F, H, O], [AD1621; N, CH, N, CH, O, H, H, F, H, O], [AD1622; N, CH, N, CH, O, F, H, F, H, O], [AD1623; N, CH, N, CH, O, Cl, H, F, H, O], [AD1624; N, CH, N, CH, O, Br, H, F, H, O], [AD 1625; N, CH, N, CH, O, I, H, F, H, O], [AD 1626; N, CH, N, CH, O, Me, H, F, H, O], [AD 1627; N, CH, N, CH, O, Et, H, F, H, O], [AD 1628; N, CH, N, CH, O, Pr, H, F, H, O] , [AD 1629; N, CH, N, CH, O, i-Pr, H, F, H, O ], [AD1630; N, CH , N, CH, O, CH = CH 2, H, F, H, O], [AD1631; N, CH, N, CH, O, C (CH 3) = CH 2 , H, F, H, O], [AD 1632; N, CH, N, CH, O, C≡CH, H, F, H, O], [AD 1633; N, CH, N, CH, O, C ≡CCH ₃ , H, F, H, O], [AD 1634; N, CH, N, CH, O, c-Pr, H, F, H, O], [AD 1635; N, CH, N, CH, O, OMe, H, F, H, O], [AD1636; N, CH, N, CH, O, OEt, H, F, H, O], [AD 1637; N, CH, N, CH, O, Oi-Pr, H, F, H, O], [AD1638; N, CH, N, CH, O, SMe, H, F, H, O], [AD 1639; N, CH, N, CH, O, SEt, H, F, H, O], [AD 1640; N, CH, N, CH, O, CH ₂ F, H, F, H, O], [AD 1641; N, CH, N, CH, O, _{CHF 2, H, F, H} , O], [AD1642; N, CH, N, CH, O, CF 3, H, F, H, O], [AD1643; N, CH, N, CH, O, OCH ₂ F, H, F, H, O], [AD 1644; N, CH, N, CH, O, OCHF ₂ , H, F, H, O], [AD 1645; N, CH, N, CH, O _{, OCF 3, H, F,} H, O], [AD1646; N, CH, N, CH, O, SCH 2 F, H, F, H, O], [AD1647; N, CH, N, CH, _{O, SCHF 2, H, F} , H, O], [AD1648; N, CH, N, CH, O, SCF 3, H, F, H, O], [AD1649; N, CH, N, CH, O, CN, H, F, H, O], [AD 1650; N, CH, N, CH, O, NO ₂ , H, F, H, O], [AD 1651; N, CH, CH, N, O , H, H, F, H, O], [AD 1652; N, CH, CH, N, O, F, H, F, H, O], [AD 1653; N, CH, CH, N, O, Cl , H, F, H, O], [AD1654; N, CH, CH, N, O, Br, H, F, H, O], [AD 1 655; N, CH, CH, N, O, I, H , F, H, O], [AD 1 656; N, CH, CH, N, O, Me, H, F, H, O], [AD 1657; N, CH, CH, N, O, Et, H, F , H, O], [AD 1658; N, CH, CH, N, O, Pr, H , F, H, O], [AD 1659; N, CH, CH, N, O, i-Pr, H, F, H, O], [AD 1660; N, CH, CH, N, O, CH = CH _{2, H, F, H,} O], [AD1661; N, CH, CH, N, O, C (CH 3) = CH 2, H, F, H, O], [AD1662; N, CH, CH , N, O, C≡CH, H, F, H, O], [AD 1663; N, CH, CH, N, O, C≡ CCH ₃ , H, F, H, O], [AD 1664; N, CH, CH, N, O, c, Pr, H, F, H, O], [AD1665; N, CH, CH, N, O, OMe, H, F, H, O], [AD 1 666; CH, CH, N, O, OEt, H, F, H, O], [AD 1 667; N, CH, CH, N, O, Oi-Pr, H, F, H, O], [AD 1668; CH, CH, N, O, SMe, H, F, H, O], [AD1669; N, CH, CH, N, O, SE, H, F, H, O], [AD 1670; N, CH, _{CH, N, O, CH 2} F, H, F, H, O], [AD1671; N, CH, CH, N, O, CHF 2, H, F, H, O], [AD1672; N, CH , CH, N, O, CF 3, H, F, H, O], [AD1673; N, CH, CH, N, O, OCH 2 F, H, F, H, O], [AD1674; N, CH, CH, N, O, OCHF 2, H, F, H, O], [AD1675; N, CH, CH, N, O, OCF 3, H, F, H, O], [AD1676; N, CH, CH, N, O, SCH ₂ F, H, F, H, O], [AD 1677; N, CH, CH, N, O, SCHF ₂ , H, F, H, O], [AD 1678; N , CH, CH, N, O , SCF 3, H, F, H, O], [AD1679; N, CH, CH, N, O, CN, H, F, H, O], [AD1680; N, CH, CH, N, O, NO 2, H, F, H, O], [AD1681; CH, N, N, CH, O, H, H, F, H, O], [AD1682; CH, N , N, CH, O, F, H, F, H, O], [AD 1683; CH, N, N, CH, O, Cl, H, F, H, O], [AD 1 684; CH, N, N , CH, O, Br, H, F, H, O], [AD 1 685; CH, N, N, CH, O, I, H, F, H, O], [AD 1686; CH, N, N, CH , O, Me, H, F, H, O], [AD 1687; CH, N, N, C H, O, Et, H, F, H, O], [AD 1688; CH, N, N, CH, O, Pr, H, F, H, O], [AD 1689; CH, N, N, CH, O, i-Pr, H, F, H, O], [AD1690; CH, N, N, CH, O, CH = CH 2, H, F, H, O], [AD1691; CH, N, N , CH, O, C (CH 3) = CH 2, H, F, H, O], [AD1692; CH, N, N, CH, O, C≡CH, H, F, H, O], [ AD 1693; CH, N, N, CH, O, C≡CCH ₃ , H, F, H, O], [AD 1694; CH, N, N, CH, O, c-Pr, H, F, H, O ], [AD 1695; CH, N, N, CH, O, OMe, H, F, H, O], [AD 1696; CH, N, N, CH, O, OEt, H, F, H, O], [AD 1697; CH, N, N, CH, O, Oi-Pr, H, F, H, O], [AD 1698; CH, N, N, CH, O, SMe, H, F, H, O], [AD1699; CH, N, N , CH, O, SEt, H, F, H, O], [AD1700; CH, N, N, CH, O, CH 2 F, H, F, H, O],

[AD1701; CH, N, N , CH, O, CHF 2, H, F, H, O], [AD1702; CH, N, N, CH, O, CF 3, H, F, H, O], [AD1703; CH, N, N , CH, O, OCH 2 F, H, F, H, O], [AD1704; CH, N, N, CH, O, OCHF 2, H, F, H, O] , [AD1705; CH, N, N, CH, O, OCF 3, H, F, H, O], [AD1706; CH, N, N, CH, O, SCH 2 F, H, F, H, O ], [AD 1707; CH, N, N, CH, O, SCHF ₂ , H, F, H, O], [AD 1 708; CH, N, N, CH, O, SCF ₃ , H, F, H, O ], [AD 1709; CH, N, N, CH, O, CN, H, F, H, O], [AD 1710; CH, N, N, CH, O, NO ₂ , H, F, H, O] [AD 1711; CH, N, CH, N, O, H, H, F, H, O], [AD 1712; CH, N, CH, N, O, F, H, F, H, O], [AD 1712; AD 1713; CH, N, CH, N, O, Cl, H, F, O], [AD 1714; CH, N, CH, N, O, Br, H, F, H, O], [AD 1715; CH, N, CH, N, O, I, H, F, H, O], [AD1716; CH, N, CH, N, O, Me, H, F, H, O], [AD1717; CH, N, CH, N, O, Et, H, F, H, O], [AD1718; CH, N, CH, N, O, Pr, H, F, H, O], [AD1719; CH, N, CH, N, O, i- Pr, H, F, H, O], [AD1720; CH, N, CH, N, O, CH = CH 2, H, F, H, O], [AD1721; CH , N, CH, N, O , C (CH 3) = CH 2, H, F, H, O], [AD1722; CH, N, CH, N, O, C≡CH, H, F, H, O, [AD1723; CH, N, CH, N, O, C≡CCH ₃ , H, F, H, O], [AD 1724; CH, N, CH, N, O, c-Pr, H, F , H, O], [AD 1725; CH, N, CH, N, O, OMe, H, F, H, O], [AD 1726; CH, N, CH, N, O, OEt, H, F, H CH, N, CH, N, O, Oi-Pr, H, F, H, O], [AD 1728; CH, N, CH, N, O, SMe, H, F, H , O], [AD 1 729; CH, N, CH, N, O, SE t, H, F, H , O], [AD 1730; CH, N, CH, N, O, CH ₂ F, H, F, H, O], [AD 1731; CH, N, CH, N, O, CHF ₂ , H, F, H, O], [AD1732; CH, N, CH, N, O, CF 3, H, F, H, O], [AD1733; CH, N, CH, N, O, OCH 2 F, H, F , H, O], [AD 1734; CH, N, CH, N, O, OCHF ₂ , H, F, H, O], [AD 1735; CH, N, CH, N, O, OCF ₃ , H, F , H, O], [AD 1 736; CH, N, CH, N, O, SCH ₂ F, H, F, H, O], [AD 1 737; CH, N, CH, N, O, SCHF ₂ , H, F, H, O], [AD 1 738; CH, N, CH, N, O, SCF ₃ , H, F, H, O], [AD 1739; CH, N, CH, N, O, CN, H, F , H, O], [AD 1740; CH, N, CH, N, O, NO, NO ₂ , H, F, H, O], [AD 1741; CH, CH, N, N, O, H, H, F, H, O], [AD 1742; CH, CH, N, N, N, O, F, H, F, H, O], [AD 1743; CH, CH, N, N, N, O, Cl, H, F, H, O], [AD 1 744; CH, CH, N, N, O, Br, H, H, O], [AD 1 745; CH, CH, N, N, O, I, H, F, H, O] [AD 1746; CH, CH, N, N, N, O, Me, H, F, H, O], [AD 1 747; CH, CH, N, N, O, Et, H, F, H, O], [AD 1 747; AD 1748; CH, CH, N, N, N, O, Pr, H, F, H, O], [AD 1749; CH, CH, N, N, O, i-Pr, H, F, H, O], [AD 1 749; AD1750; CH, CH, N, N, O, CH = CH 2, H, F, H, O], [AD1751; CH, CH, N, N, O, C (CH 3) = CH 2, H, F, H, O], [AD1752; CH, CH, N, N, O, C≡CH, H, F, H, O], [AD1753; CH, CH, N, N, O, C≡ CCH ₃ , H, F, H, O], [AD 1754; CH, CH, N, N, O, c, Pr, H, F, H, O], [AD 1755; CH, CH, N, N, O, OMe , H, F, H, O], [AD 1756; CH, CH, N, N, O, OEt, H, F, H, O], [AD 1757; CH, CH, N, N, O, Oi-Pr , H, F, H, O], [AD 1758; CH, CH, N, N, O, SM e, H, F, H, O], [AD 1759; CH, CH, N, N, O, SE, H, F, H, O], [AD 1760; CH, CH, N, N, O, CH ₂ F, H, F, H, O], [AD1761; CH, CH, N, N, O, CHF 2, H, F, H, O], [AD1762; CH, CH, N, N, O, CF _{3, H, F, H,} O], [AD1763; CH, CH, N, N, O, OCH 2 F, H, F, H, O], [AD1764; CH, CH, N, N, O, _{OCHF 2, H, F, H} , O], [AD1765; CH, CH, N, N, O, OCF 3, H, F, H, O], [AD1766; CH, CH, N, N, O, SCH ₂ F, H, F, H, O], [AD 1 767; CH, CH, N, N, O, SCHF ₂ , H, F, H, O], [AD 1 768; CH, CH, N, N, O SCF ₃ , H, F, H, O], [AD 1769; CH, CH, N, N, O, CN, H, F, H, O], [AD 1770; CH, CH, N, N, O, NO ₂ , H, F, H, O], [AD 1771; N, CH, N, N, O, H, H, F, H, O], [AD 1772; N, CH, N, N, O, F , H, F, H, O], [AD1773; N, CH, N, N, O, Cl, H, F, H, O], [AD 1774; N, CH, N, N, O, Br, H , F, H, O], [AD 1 775; N, CH, N, N, O, I, H, F, H, O], [AD 1 776; N, CH, N, N, O, Me, H, F , H, O], [AD 1 777; N, CH, N, N, O, Et, H, F, H, O], [AD 1778; N, CH, N, N, N, O, Pr, H, F, H , O], [AD1779; N , CH, N, N, O, i-Pr, H, F, H, O], [AD1780; N, CH, N, N, O, CH = CH 2, H, F, H, O], [ AD1781; N, CH, N, N, O, C (CH 3) = CH 2, H, F, H, O], [AD1782; N, CH, N, N, O , CCHCH, H, F, H, O], [AD 1783; N, CH, N, N, O, C≡CCH ₃ , H, F, H, O], [AD 1784; N, CH, N, N, O, c-Pr, H, F, H, O], [AD 1 785; N, CH, N, N, O, OMe, H, F, H, O], [AD 1 786; N, CH, N, N, O, OEt, H, F, H, O], [AD 1787; N, CH, N, N, O, Oi-Pr, H, F, H, O] , [AD 1 788; N, CH, N, N, O, SMe, H, F, H, O], [AD 1 789; N, CH, N, N, O, SE t, H, F, H, O], [ AD1790; N, CH, N, N, O, CH 2 F, H, F, H, O], [AD1791; N, CH, N, N, O, CHF 2, H, F, H, O], [AD1792; N, CH, N , N, O, CF 3, H, F, H, O], [AD1793; N, CH, N, N, O, OCH 2 F, H, F, H, O] , [AD1794; N, CH, N, N, O, OCHF 2, H, F, H, O], [AD1795; N, CH, N, N, O, OCF 3, H, F, H, O] , [AD 1796; N, CH, N, N, O, SCH ₂ F, H, F, H, O], [AD 1 797; N, CH, N, N, O, SCHF ₂ , H, F, H, O ], [AD1798; N, CH , N, N, O, SCF 3, H, F, H, O], [AD1799; N, CH, N, N, O, CN, H, F, H, O] , [AD1800; N, CH, N, N, O, NO ₂ , H, F, H, O],

[AD 1801; CH, CH, CH, CH, CH, O, H, H, H, F, O], [AD 1802; CH, CH, CH, CH, O, F, H, H, F, O], [AD 1803 CH, CH, CH, CH, CH, O, Cl, H, H, F, O], [AD 1804; CH, CH, CH, CH, CH, O, Br, H, F, O], [AD 1805; CH , CH, CH, CH, O, I, H, H, F, O], [AD 1806; CH, CH, CH, CH, CH, O, Me, H, F, O], [AD 1807; CH, CH , CH, CH, O, Et, H, H, F, O], [AD 1808; CH, CH, CH, CH, CH, O, Pr, H, H, F, O], [AD 1809; CH, CH, CH , CH, O, i-Pr , H, H, F, O], [AD1810; CH, CH, CH, CH, O, CH = CH 2, H, H, F, O], [AD1811; CH, CH, CH, CH, O, C (CH 3) = CH 2, H, H, F, O], [AD1812; CH, CH, CH, CH, O, C≡CH, H, H, F, O ], [AD 1813; CH, CH, CH, CH, CH, O, C≡CCH ₃ , H, H, F, O], [AD 1814; CH, CH, CH, CH, O, c-Pr, H, H, F, O], [AD 1815; CH, CH, CH, CH, O, OMe, H, H, F, O], [AD 1816; CH, CH, CH, CH, O, OE t, H, H, F, O, [AD 1817; CH, CH, CH, CH, CH, O, Oi-Pr, H, H, F, O], [AD 1818; CH, CH, CH, CH, O, SMe, H, H, F, O, [AD 1819; CH, CH, CH, CH, O, SE t, H, H, F, O], [AD 1820; CH, CH, CH, CH, O, CH ₂ F, H, H, F, O], [AD1821; CH, CH, CH, CH, O, CHF 2, H, H, F, O], [AD1822; CH, CH, CH, CH, O, CF 3, H, H, F, O, [AD 1823; CH, CH, CH, CH, CH, O, OCH ₂ F, H, H, F, O], [AD 1824; CH, CH, CH, CH, O, OCHF ₂ , H, H, F , O], [AD1825; CH , CH, CH, CH, O, OCF 3, H, H, F, O], [AD1826; CH, CH, CH, CH, O, SCH 2 F, H, H, F, O], [AD 1827; CH, CH, CH, CH, O, SCHF ₂ , H, H, F, O], [AD 1 828; C H, CH, CH, CH, O, SCF 3, H, H, F, O], [AD1829; CH, CH, CH, CH, O, CN, H, H, F, O], [AD1830; CH , CH, CH, CH, O , NO 2, H, H, F, O], [AD1831; N, CH, CH, CH, O, H, H, H, F, O], [AD1832; N, CH, CH, CH, CH, O, F, H, H, F, O], [AD1833; N, CH, CH, CH, CH, O, Cl, H, F, O], [AD1834; N, CH, CH, CH, O, Br, H, H, F, O], [AD1835; N, CH, CH, CH, O, I, H, F, O], [AD1836; N, CH, CH, CH, O, Me, H, H, F, O], [AD 1837; N, CH, CH, CH, O, Et, H, H, F, O], [AD 1838; N, CH, CH, CH, O, Pr, H, H, F, O], [AD 1839; N, CH, CH, CH, O, i-Pr, H, H, F, O], [AD 1840; N, CH, CH, CH, _{O, CH = CH 2, H} , H, F, O], [AD1841; N, CH, CH, CH, O, C (CH 3) = CH 2, H, H, F, O], [AD1842; N, CH, CH, CH, O, C≡CH, H, H, F, O], [AD1843; N, CH, CH, CH, O, C≡CCH 3, H, H, F, O], [AD 1844; N, CH, CH, CH, CH, O, c-Pr, H, H, F, O], [AD 1845; N, CH, CH, CH, O, OMe, H, H, F, O], [AD 1846; N, CH, CH, CH, CH, O, OEt, H, H, F, O], [AD 1 847; N, CH, CH, CH, O, Oi-Pr, H, H, F, O], [AD1848; N, CH, CH, CH, CH, O, SMe, H, H, F, O], [AD 1849; N, CH, CH, CH, O, SE t, H, H, F, O], [AD1850 ; N, CH, CH, CH , O, CH 2 F, H, H, F, O], [AD1851; N, CH, CH, CH, O, CHF 2, H, H, F, O], [ AD1852; N, CH, CH, CH, O, CF 3, H, H, F, O], [AD1853; N, CH, CH, CH, O, OCH 2 F, H, H, F, O], [AD1854; N, CH, CH , CH, O, OCHF 2, H, H, F, O], [AD1855; N, CH, CH, CH, O, OCF 3, H, H, F, O], [AD 1856; N, CH , CH, CH, O, SCH ₂ F, H, H, F, O], [AD 1857; N, CH, CH, CH, O, SCHF ₂ , H, H, F, O], [AD 1858; N, CH, CH, CH, O, SCF 3, H, H, F, O], [AD1859; N, CH, CH, CH, O, CN, H, H, F, O], [AD1860; N, CH , CH, CH, O, NO 2, H, H, F, O], [AD1861; CH, N, CH, CH, O, H, H, H, F, O], [AD1862; CH, N, CH, CH, O, F, H, H, F, O], [AD 1863; CH, N, CH, CH, O, Cl, H, H, F, O], [AD 1864; CH, N, CH, CH, O, Br, H, H, F, O], [AD 1865; CH, N, CH, CH, O, I, H, F, O], [AD 1866; CH, N, CH, CH, O, Me, H, H, F, O], [AD 1867; CH, N, CH, CH, O, Et, H, F, O], [AD 1868; CH, N, CH, CH, O, Pr, H, H, F, O], [AD 1869; CH, N, CH, CH, O, i-Pr, H, H, F, O], [AD 1870; CH, N, CH, CH, O, CH = CH ₂ , H, H, F, O], [AD 187 1; CH, N, CH, CH, O, C (CH ₃ ) = CH ₂ , H, H, F, O], [AD 187 2; CH, N, CH, CH, O, C≡CH, H, H, F, O], [AD 1 873; CH, N, CH, CH, O, C≡ CCH ₃ , H, H, F, O], [AD 1 874 CH, N, CH, CH, O, c-Pr, H, H, F, O], [AD 1875; CH, N, CH, CH, O, OMe, H, H, F, O], [AD 1876; CH, N, CH, CH, O, OEt, H, H, F, O], [AD 1877; CH, N, CH, CH, O, Oi-Pr, H, H, F, O], [AD 1878 CH, N, CH, CH, O, SMe, H, H, F, O], [AD 1879; CH, N, CH, CH, O, SE t, H, H, F, O], [AD 1 880; CH , N, CH, CH, O , CH 2 F, H, H, F, O], [AD1881; CH, N, CH, CH, O, CHF 2, H, H, F, O], [AD1882; CH, N, CH, CH, O, CF 3, H, H, F, O], [AD1883; CH, N, CH, CH, O, OCH 2 F, H, H, F, O], [AD1884 CH, N, CH, C _{H, O, OCHF 2, H} , H, F, O], [AD1885; CH, N, CH, CH, O, OCF 3, H, H, F, O], [AD1886; CH, N, CH, CH, O, SCH ₂ F, H, H, F, O], [AD 1887; CH, N, CH, CH, O, SCHF ₂ , H, H, F, O], [AD 1888; CH, N, CH _{, CH, O, SCF 3,} H, H, F, O], [AD1889; CH, N, CH, CH, O, CN, H, H, F, O], [AD1890; CH, N, CH, _{CH, O, NO 2, H} , H, F, O], [AD1891; CH, CH, N, CH, O, H, H, H, F, O], [AD1892; CH, CH, N, CH , O, F, H, H, F, O], [AD 1893; CH, CH, N, CH, O, Cl, H, F, O], [AD 1894; CH, CH, N, CH, O , Br, H, H, F, O], [AD 1895; CH, CH, N, CH, O, I, H, F, O], [AD 1896; CH, CH, N, CH, O, Me , H, H, F, O], [AD 1897; CH, CH, N, CH, O, Et, H, H, F, O], [AD 1898; CH, CH, N, CH, O, Pr, H , H, F, O], [AD 1899; CH, CH, N, CH, O, i-Pr, H, H, F, O], [AD 1900; CH, CH, N, CH, O, CH = CH ₂ , H, H, F, O],

[AD1901; CH, CH, N , CH, O, C (CH 3) = CH 2, H, H, F, O], [AD1902; CH, CH, N, CH, O, C≡CH, H, H, F, O], [AD 1903; CH, CH, N, CH, O, C≡CCH ₃ , H, H, F, O], [AD 1904; CH, CH, N, CH, O, c-Pr , H, H, F, O], [AD 1905; CH, CH, N, CH, O, OMe, H, H, F, O], [AD 1906; CH, CH, N, CH, O, OE t, H , H, F, O], [AD 1 907; CH, CH, N, CH, O, Oi-Pr, H, H, F, O], [AD 1908; CH, CH, N, CH, O, SMe, H , H, F, O], [AD 1 909; CH, CH, N, CH, O, SE t, H, H, F, O], [AD 1910; CH, CH, N, CH, O, CH ₂ F, H , H, F, O], [AD1911; CH, CH, N, CH, O, CHF 2, H, H, F, O], [AD1912; CH, CH, N, CH, O, CF 3, H , H, F, O], [AD 1913; CH, CH, N, CH, O, OCH ₂ F, H, H, F, O], [AD 1914; CH, CH, N, CH, O, OCHF ₂ , H, H, F, O] , [AD1915; CH, CH, N, CH, O, OCF 3, H, H, F, O], [AD1916; CH, CH, N, CH, O, SCH 2 F , H, H, F, O], [AD 1917; CH, CH, N, CH, O, SCHF ₂ , H, H, F, O], [AD 1918; CH, CH, N, CH, O, SCF ₃ , H, H, F, O], [AD 1919; CH, CH, N, CH, O, CN, H, H, F, O], [AD 1920; CH, CH, N, CH, O, NO ₂ , H, H, F, O], [AD1921; CH, CH, CH, N, O, H, H, H, F, O], [AD1922; CH, CH, CH, N, O, F, H, H, F, O], [AD 1 923; CH, CH, CH, N, O, Cl, H, F, O], [AD 1 924; CH, CH, CH, N, O, Br, H, H, F, O], [AD 1925; CH, CH, CH, N, O, I, H, F, O], [AD 1926; CH, CH, CH, N, O, Me, H, H, F, O], [AD 1 927; CH, CH, CH, CH, N, O, Et, H, F, O], [AD 1 928; CH, CH, CH, N, O, Pr, H, H, F, O] , [AD1 929; CH, CH, CH, N, O, i-Pr, H, H, F, O], [AD1930; CH, CH, CH, N, O, CH = CH 2, H, H, F, O ], [AD1931; CH, CH , CH, N, O, C (CH 3) = CH 2, H, H, F, O], [AD1932; CH, CH, CH, N, O, C≡CH, H, H, F, O], [AD 1933; CH, CH, CH, N, O, C≡CCH ₃ , H, H, F, O], [AD 1934; CH, CH, CH, N, O, c -Pr, H, H, F, O], [AD 1935; CH, CH, CH, N, O, OMe, H, H, F, O], [AD 1936; CH, CH, CH, N, O, OEt , H, H, F, O], [AD 1937; CH, CH, CH, N, O, Oi-Pr, H, H, F, O], [AD 1938; CH, CH, CH, N, O, SMe , H, H, F, O], [AD 1939; CH, CH, CH, N, O, SE, H, H, F, O], [AD 1940; CH, CH, CH, N, O, CH ₂ F , H, H, F, O ], [AD1941; CH, CH, CH, N, O, CHF 2, H, H, F, O], [AD1942; CH, CH, CH, N, O, CF 3 , H, H, F, O ], [AD1943; CH, CH, CH, N, O, OCH 2 F, H, H, F, O], [AD1944; CH, CH, CH, N, O, OCHF _{2, H, H, F,} O], [AD1945; CH, CH, CH, N, O, OCF 3, H, H, F, O], [AD1946; CH, CH, CH, N, O, SCH ₂ F, H, H, F, O], [AD 1947; CH, CH, CH, N, O, SCHF ₂ , H, H, F, O], [AD 1948; CH, CH, CH, N, O, SCF ₃ , H, H, F, O], [AD 1949; CH, CH, CH, N, O, CN, H, H, F, O], [AD 1950; CH, CH, CH, N, O, NO ₂ , H, H, F, O], [AD1951; N, N, CH, CH, O, H, H, H, F, O], [AD 1952; N, N, CH, CH, O, F, H, H, F, O], [AD1953; N, N, CH, CH, O, Cl, H, H, F, O], [AD1954; N, N, CH, CH, O, Br, H, H, F, O], [AD 1 955; N, N, CH, CH, O, I, H, F, O], [AD 1956; N, N, CH, CH, O, Me, H, H, F, O], [AD 195 7; N, N, CH, CH, O, Et, H, H, F, O], [AD 1958; N, N, CH, CH, O, Pr, H, H, F, O], [AD 1959; N, N, CH, CH, O, i-Pr, H, H, F, O], [AD1960; N, N, CH, CH, O, CH = CH 2, H, H, F, O], [AD1961; N, N, CH , CH, O, C (CH 3) = CH 2, H, H, F, O], [AD1962; N, N, CH, CH, O, C≡CH, H, H, F, O], [AD 1963; N, N, CH, CH, O, C≡CCH ₃ , H, H, F, O], [AD 1964; N, N, CH, CH, O, c-Pr , H, H, F, O], [AD 1 965; N, N, CH, CH, O, OMe, H, H, F, O], [AD 1966; N, N, CH, CH, O, OE t, H , H, F, O], [AD 1967; N, N, CH, CH, O, Oi-Pr, H, H, F, O], [AD 1968; N, N, CH, CH, O, SMe, H , H, F, O], [AD1969; N, N, CH, CH, O, SEt, H, H, F, O], [AD1970; N, N, CH, CH, O, CH ₂ F, H H, F, O], [AD 1971; N, N, CH, CH, O, CHF ₂ , H, H, F, O], [AD 1972; N, N, CH, CH, O, CF ₃ , H , H, F, O], [AD 1973; N, N, CH, CH, O, OCH ₂ F, H, H, F, O], [AD 1974; N, N, CH, CH, O, OCHF ₂ , H, H, F, O] , [AD1975; N, N, CH, CH, O, OCF 3, H, H, F, O], [AD1976; N, N, CH, CH, O, SCH 2 F , H, H, F, O], [AD 1977; N, N, CH, CH, O, SCHF ₂ , H, H, F, O], [AD1978; N, N, CH, CH, O, SCF ₃ , H, H, F, O], [AD 1979; N, N, CH, CH, O, CN, H, H, F, O], [AD1980; N, N, CH, CH, O, NO ₂ , H, H, F, O], [AD1981; N, CH, N, CH, O, H, H, H, F, O], [AD 1982; N, CH, N, CH, O, F, H, H, F, O], [AD 1983; N, CH, N, CH, O, Cl, H, F, O], [AD 1984; N, CH, N, CH, O, Br, H, H, H F, O], [AD 1985; N, CH, N, CH, O, I, H, H, F, O ], [AD 1986; N, CH, N, CH, O, Me, H, H, F, O], [AD 1987; N, CH, N, CH, O, Et, H, H, F, O], [AD 1988; N, CH, N, CH, O, Pr, H, H, F, O], [AD 1989; N, CH, N, CH, O, i-Pr, H, H, F, O], [AD1990; N, CH, N , CH, O, CH = CH 2, H, H, F, O], [AD1991; N, CH, N, CH, O, C (CH 3) = CH 2, H , H, F, O], [AD 1992; N, CH, N, CH, O, C≡CH, H, H, F, O], [AD 1993; N, CH, N, CH, O, C≡ CCH ₃ , H, H, F, O], [AD 1994; N, CH, N, CH, O, c-Pr, H, H, F, O], [AD 1995; N, CH, N, CH, O, OMe, H, H, F, O], [AD 1996; N, CH, N, CH, O, OEt, H, H, F, O], [AD 1997; N, CH, N, CH, O, Oi- Pr, H, H, F, O], [AD1998; N, CH, N, CH, O, SMe, H, H, F, O], [AD 1999; N, CH, N, CH, O, SEt, H, H, F, O], [AD 2000; N, CH, N, CH, O, CH ₂ F, H, H, F, O],

[AD2001; N, CH, N , CH, O, CHF 2, H, H, F, O], [AD2002; N, CH, N, CH, O, CF 3, H, H, F, O], [AD2003; N, CH, N , CH, O, OCH 2 F, H, H, F, O], [AD2004; N, CH, N, CH, O, OCHF 2, H, H, F, O] , [AD2005; N, CH, N, CH, O, OCF 3, H, H, F, O], [AD2006; N, CH, N, CH, O, SCH 2 F, H, H, F, O ], [AD 2007; N, CH, N, CH, O, SCHF ₂ , H, H, F, O], [AD 2008; N, CH, N, CH, O, SCF ₃ , H, H, F, O] ], [AD2009; N, CH , N, CH, O, CN, H, H, F, O], [AD2010; N, CH, N, CH, O, NO 2, H, H, F, O] , [AD2011; N, CH, CH, N, O, H, H, H, F, O], [AD 2012; N, CH, CH, N, O, F, H, H, F, O], [AD2011; AD 2013; N, CH, CH, N, O, Cl, H, F, O], [AD 2014; N, CH, CH, N, O, Br, H, F, O], [AD 2015; N, CH, CH, N, O, I, H, H, F, O], [AD2016; N, CH, CH, N, O, Me, H, F, O], [AD 2017; N, CH, CH, N, O, Et, H, H, F, O], [AD 2018; N, CH, CH, N, O, Pr, H, F, O], [AD 2019; N, CH, CH, N, O, i- Pr, H, H, F, O], [AD2020; N, CH, CH, N, O, CH = CH 2, H, H, F, O], [AD2021; N , CH, CH, N, O , C (CH 3) = CH 2, H, H, F, O], [AD2022; N, CH, CH, N, O, C≡CH, H, H, F, O, [AD 2023; N, CH, CH, N, O, C≡CCH ₃ , H, H, F, O], [AD 2024; N, CH, CH, N, O, c-Pr, H, H , F, O], [AD 2025; N, CH, CH, N, O, OMe, H, H, F, O], [AD 2026; N, CH, CH, N, O, OE t, H, H, F , O], [AD 2027; N, CH, CH, N, O, Oi-Pr, H, H, F, O], [AD 2028; N, CH, CH, N, O, SMe, H, H, F , O], [AD 2029; N, CH, CH, N, O, SE t, H, H, F , O], [AD 2030; N, CH, CH, N, O, CH ₂ F, H, H, F, O], [AD 2031; N, CH, CH, N, O, CHF ₂ , H, H, H F, O], [AD2032; N, CH, CH, N, O, CF 3, H, H, F, O], [AD2033; N, CH, CH, N, O, OCH 2 F, H, H , F, O], [AD 2034; N, CH, CH, N, O, OCHF ₂ , H, H, F, O], [AD 2035; N, CH, CH, N, O, OCF ₃ , H, H , F, O], [AD 2036; N, CH, CH, N, O, SCH ₂ F, H, H, F, O], [AD 2037; N, CH, CH, N, O, SCHF ₂ , H, H, F, O], [AD 2038; N, CH, CH, N, O, SCF ₃ , H, H, F, O], [AD 2039; N, CH, CH, N, O, CN, H, H , F, O], [AD 2040; N, CH, CH, N, O, NO ₂ , H, H, F, O], [AD 2041; CH, N, N, CH, O, H, H, H, H, F, O], [AD 2042; CH, N, N, CH, O, F, H, H, F, O], [AD 2043; CH, N, N, CH, O, Cl, H, H, F, O], [AD 2044; CH, N, N, CH, O, Br, H, F, O], [AD 2045; CH, N, N, CH, O, I, H, H, F, O] , [AD 2046; CH, N, N, CH, O, Me, H, H, F, O], [AD 2047; CH, N, N, CH, O, Et, H, F, O], [AD 2047; AD2048; CH, N, N, CH, O, Pr, H, H, F, O], [AD 2049; CH, N, N, CH, O, i-Pr, H, H, F, O], [[ AD2050; CH, N, N, CH, O, CH = CH 2, H, H, F, O], [AD2051; CH, N, N, CH, O, C (CH 3) = CH 2, H, H, F, O], [AD 2052; CH, N, N, CH, O, C≡CH, H, H, F, O], [AD 2053; CH, N, N, CH, O, C≡ CCH ₃ , H, H, F, O], [AD 2054; CH, N, N, CH, O, c-Pr, H, H, F, O], [AD 2055; CH, N, N, CH, O, OMe , H, H, F, O], [AD 2056; CH, N, N, CH, O, OEt, H, H, F, O], [AD 2057; CH, N, N, CH, O, Oi-Pr , H, H, F, O], [AD 2058; CH, N, N, CH, O, SM e, H, H, F, O], [AD 2059; CH, N, N, CH, O, SE t, H, H, F, O], [AD 2060; CH, N, N, CH, O, CH ₂ F, H, H, F, O], [AD2061; CH, N, N, CH, O, CHF 2, H, H, F, O], [AD2062; CH, N, N, CH, O, CF ₃ , H, H, F, O], [AD 2063; CH, N, N, CH, O, OCH ₂ F, H, H, F, O], [AD 2064; CH, N, N, CH, O, _{OCHF 2, H, H, F} , O], [AD2065; CH, N, N, CH, O, OCF 3, H, H, F, O], [AD2066; CH, N, N, CH, O, SCH ₂ F, H, H, F, O], [AD 2067; CH, N, N, CH, O, SCHF ₂ , H, H, F, O], [AD 2068; CH, N, N, CH, O SCF ₃ , H, H, F, O], [AD 2069; CH, N, N, CH, O, CN, H, H, F, O], [AD 2070; CH, N, N, CH, O, _{NO 2, H, H, F} , O], [AD2071; CH, N, CH, N, O, H, H, H, F, O], [AD2072; CH, N, CH, N, O, F , H, H, F, O], [AD 2073; CH, N, CH, N, O, Cl, H, F, O], [AD 2074; CH, N, CH, N, O, Br, H , H, F, O], [AD 2075; CH, N, CH, N, O, I, H, H, F, O], [AD 2076; CH, N, CH, N, O, Me, H, H , F, O], [AD 2077; CH, N, CH, N, O, Et, H, F, O], [AD 2078; CH, N, CH, N, O, Pr, H, H, F , O], [AD2079; CH , N, CH, N, O, i-Pr, H, H, F, O], [AD2080; CH, N, CH, N, O, CH = CH 2, H, H, F, O], [ AD2081; CH, N, CH, N, O, C (CH 3) = CH 2, H, H, F, O], [AD2082; CH, N, CH, N, O , C≡CH, H, H, F, O], [AD 2083; CH, N, CH, N, O, C≡CCH ₃ , H, H, F, O], [AD 2084; CH, N, CH, N, O, c-Pr, H, H, F, O], [AD 2085; CH, N, CH, N, O, OMe, H, H, F, O], [AD 2086; CH, N, CH, N, O, OEt, H, H, F, O], [AD 2087; CH, N, CH, N , O, Oi-Pr, H, H, F, O], [AD 2088; CH, N, CH, N, O, SMe, H, F, O], [AD 2089; CH, N, CH, N , O, SEt, H, H, F, O], [AD 2090; CH, N, CH, N, O, CH ₂ F, H, H, F, O], [AD 2091; CH, N, CH, N _{, O, CHF 2, H,} H, F, O], [AD2092; CH, N, CH, N, O, CF 3, H, H, F, O], [AD2093; CH, N, CH, N _{, O, OCH 2 F, H} , H, F, O], [AD2094; CH, N, CH, N, O, OCHF 2, H, H, F, O], [AD2095; CH, N, CH, _{N, O, OCF 3, H} , H, F, O], [AD2096; CH, N, CH, N, O, SCH 2 F, H, H, F, O], [AD2097; CH, N, CH , N, O, SCHF ₂ , H, H, F, O], [AD 2098; CH, N, CH, N, O, SCF ₃ , H, H, F, O], [AD 2099; CH, N, CH , N, O, CN, H, H, F, O], [AD 2 100; CH, N, CH, N, O, NO ₂ , H, H, F, O],

[AD2101; CH, CH, N, N, N, O, H, H, F, O], [AD 2102; CH, CH, N, N, N, O, F, H, F, O], [AD 2 103 CH, CH, N, N, N, O, Cl, H, H, F, O], [AD 2104; CH, CH, N, N, O, Br, H, F, O], [AD 2 105; CH , CH, N, N, O, I, H, H, F, O], [AD 2106; CH, CH, N, N, N, O, Me, H, F, O], [AD 2107; CH, CH , N, N, O, Et, H, H, F, O], [AD 2108; CH, CH, N, N, N, O, Pr, H, F, O], [AD 2 109; CH, CH, N , N, O, i-Pr , H, H, F, O], [AD2110; CH, CH, N, N, O, CH = CH 2, H, H, F, O], [AD2111; CH, CH, N, N, O, C (CH 3) = CH 2, H, H, F, O], [AD2112; CH, CH, N, N, O, C≡CH, H, H, F, O ], [AD 2 113; CH, CH, N, N, O, C≡CCH ₃ , H, H, F, O], [AD 2114; CH, CH, N, N, N, O, c-Pr, H, H, F, O], [AD 2 115; CH, CH, N, N, O, OMe, H, H, F, O], [AD 2116; CH, CH, N, N, O, OEt, H, H, F, O, [AD 2 117; CH, CH, N, N, O, Oi-Pr, H, H, F, O], [AD 2 118; CH, CH, N, N, O, SMe, H, H, F, O, [AD 2119; CH, CH, N, N, O, SE, H, H, F, O], [AD 2 120; CH, CH, N, N, O, CH ₂ F, H, H, F, O], [AD2121; CH, CH, N, N, O, CHF 2, H, H, F, O], [AD2122; CH, CH, N, N, O, CF 3, H, H, F, O], [AD 2123; CH, CH, N, N, O, OCH ₂ F, H, H, F, O], [AD 2 124; CH, CH, N, N, O, OCHF ₂ , H, H, F , O], [AD2125; CH , CH, N, N, O, OCF 3, H, H, F, O], [AD2126; CH, CH, N, N, O, SCH 2 F, H, H, F, O], [AD 2 127; CH, CH, N, N, O, SCHF ₂ , H, H, F, O], [AD 2 128; CH, CH, N, N, O, SCF ₃ , H, H, F, O], [AD 2 129; CH, CH, N, N, O, CN, H, H, F, O], [AD 2130; CH, CH, N, N, O, NO, NO ₂ , H, H, F, O], [AD 2 131; N, CH, N, N, N, O, H, H, H, F N, CH, N, N, N, O, F, H, F, O], [AD 2 133; N, CH, N, N, O, Cl, H, H, F, O ], [AD 2 134; N, CH, N, N, O, Br, H, F, O], [AD 2 135; N, CH, N, N, O, I, H, H, F, O], [AD 2136; N, CH, N, N, N, O, Me, H, H, F, O], [AD 2 137; N, CH, N, N, N, O, Et, H, H, F, O], [AD 2 138 N, CH, N, N, N, O, Pr, H, H, F, O], [AD 2 139; N, CH, N, N, O, i-Pr, H, H, F, O], [AD 2 140 ; N, CH, N, N , O, CH = CH 2, H, H, F, O], [AD2141; N, CH, N, N, O, C (CH 3) = CH 2, H, H , F, O], [AD2142; N, CH, N, N, O, C≡CH, H, H, F, O], [AD 2143; N, CH, N, N, O, C≡ CCH ₃ , H, H, F, O], [AD 2144; N, CH, N, N, O, c, Pr, H, H, F, O], [AD 2 145; N, CH, N, N, O, OMe, H, H, F, O], [AD 2146; N, CH, N, N, O, OEt, H, H, F, O], [AD 2 147; N, CH, N, N, O, Oi-Pr, H, H, F, O], [AD 2 148; N, CH, N, N, O, SMe, H, H, F, O], [AD 2 149; N, CH, N, N, O, SE t, H, H, F, O], [AD 2150; N, CH, N, N, O, CH ₂ F, H, H, F, O], [AD 2151; N, CH, N, N, O, CHF ₂ , H , H, F, O], [AD2152; N, CH, N, N, O, CF 3, H, H, F, O], [AD2153; N, CH, N, N, O, OCH 2 F, H, H, F, O], [AD 2154; N, CH, N, N, O, OCHF ₂ , H, H, F, O], [AD 2 155; N, CH, N, N, O, OCF ₃ , H, H, F, O], [AD 2156; N, CH, N, N, O, SCH ₂ F, H, H, F, O], [AD 2 157; N, CH, N, N, O, SCHF ₂ , H, H, F, O], [AD 2158; N, CH, N, N, O, SCF ₃ , H, H, F, O], [AD 2 159; N, CH, N, N, O, CN, H, H, F, O], [AD 2 160; N, CH, N, N, O, NO ₂ , H, H, F, O].

[Substituent group number ^{(MD2); E 104],} [BD1; phenyl], [BD2; 2-fluorophenyl], [BD3; 3- fluorophenyl], [BD4; 4-fluorophenyl], [BD5; 2, 3-difluorophenyl], [BD 6; 2,4-difluorophenyl], [BD 7; 2, 5-difluorophenyl], [BD 8; 2, 6-difluorophenyl], [BD 9; 3,4-difluorophenyl], [BD10; 3,5-Difluorophenyl], [BD11; 2,3,4-Trifluorophenyl], [BD12; 2,3,5-Trifluorophenyl], [BD13; 2,3,6-Trifluoro Phenyl], [BD14; 2,4,5-trifluorophenyl], [BD15; 2,4,6-trifluorophenyl], [BD16; 3,4,5-trifluorophenyl], [BD17; 3,4,6-tetrafluorophenyl], [BD18; 2,3,5,6-tetrafluorophenyl], [BD19; 2,3,4,5,6-pentafluorophenyl], [BD20; Chlorophenyl], [BD 21; 3-chlorophenyl], [BD 22; 4-chlorophenyl], [BD 23; 2,3-dichlorophenyl], [BD 24; 2,4-dichlorophenyl], [BD 25; 2, 5-dichlorophenyl], [BD 25; BD 26; 2,6-dichlorophenyl], [BD 27; 3,4-dichlorophenyl], [BD 28; 3,5-dichlorophenyl], [BD 29; 2, 3, 4- trichlorophenyl], [BD 30; 2, 3, 5 -Trichlorophenyl], [BD31; 2,3,6-trichlorophenyl], [BD32; 2,4,5-trichlorophenyl], [BD33; 2,4,6-trichlorophenyl], [BD34; 3,4 , 5-trichlorophenyl], [BD 35; 2, 3, 4, 6-tetrachlorophenyl], [BD 36; 2, 3, 5, 6-tetrachlorophenyl], [BD 37; 2, 3, 4, 5, 6- Pentachlorophenyl], [BD 38; 2-bromophenyl], [BD 39; 3-bromophenyl], [BD 40; 4-bromophenyl], [BD 41; 2,4-dibromophenyl], [BD 42; 2, 5-dibromo Phenyl], [BD 43; 2, 6-dibromophenyl], [BD 44; 2, 4, 6-tribromophenyl], [BD 45; 2, 3, 4, 5, 6-pentabromophenyl], [BD 46; -Iodophenyl], [BD 47; 3-iodophenyl], [BD 48; 4-iodophenyl], [BD 49; 2,4-diiodophenyl], [BD 50; 2-chloro-3-fluorophenyl], [BD 51 2-chloro-4-fluorophenyl ], [BD 52; 2-chloro-5-fluorophenyl], [BD 53; 2-chloro-6-fluorophenyl], [BD 54; 2-chloro-3-bromophenyl], [BD 55; 2-chloro-4- Bromophenyl], [BD56; 2-chloro-5-bromophenyl], [BD57; 2-chloro-6-bromophenyl], [BD58; 2-bromo-3-chlorophenyl], [BD59; 2-bromo-4 2-Chlorophenyl], [BD60; 2-bromo-5-chlorophenyl], [BD 61; 2-bromo-3-fluorophenyl], [BD 62; 2-bromo-4-fluorophenyl], [BD 63; 2-bromo-5 -Fluorophenyl], [BD 64; 2-bromo-6-fluorophenyl], [BD 65; 2-fluoro-3-chlorophenyl], [BD 66; 2-fluoro-4-chlorophenyl], [BD 67; 2-chlorophenyl], [BD 68; 2-fluoro-4-bromophenyl], [BD 69; 3-chloro-4-fluorophenyl], [BD 70; 3-chloro-5-fluorophenyl], [BD 71; 3-chloro- 4-bromophenyl], [BD 72; 3-chloro-5-bromophenyl], [BD 73; 3-fluoro-4-chlorophenyl], [BD 74; Oro-4-bromophenyl], [BD 75; 3-bromo-4-chlorophenyl], [BD 76; 3-bromo-4-fluorophenyl], [BD 77; 2, 6-dichloro-4-bromophenyl], [BD 78 2,3-difluoro-4-chlorophenyl], [BD 79; 2, 6-difluoro-4-chlorophenyl], [BD 80; 2, 5-difluoro-4-chlorophenyl], [BD 81; 3,5-difluoro-4 -Chlorophenyl], [BD 82; 2, 3, 5-trifluoro-4-chlorophenyl], [BD 83; 2, 3, 6-trifluoro-4-chlorophenyl], [BD 84; 2, 3, 5, 6-tetra Fluoro-4-chlorophenyl], [BD 85; 2,3-difluoro-4-bromophenyl], [BD 86; 2, 6-difluoro-4-bromophenyl], [BD 87; 2, 5-difluoro-4-bromophenyl ], [BD 88; 3,5-difluoro-4-bromophenyl], [BD 89; 2, 3, 5-trifluoro-4-bromophenyl], [BD 90; 2, 3, 6-trifluoro-4-bromo] Phenyl], [BD 91; 2, 3, 5, 6 tetrafluoro-4-bromophenyl], [BD 92; 2-fluoro-4-iodophenyl], [BD 93; Phenyl], [BD 94; 2,3-difluoro-4-iodophenyl], [BD 95; 2, 6-difluoro-4-iodophenyl], [BD 96; 2, 5-difluoro-4-iodophenyl], [BD 97 3,5-Difluoro-4-iodophenyl], [BD 98; 2,3,5-trifluoro-4-iodophenyl], [BD 99; 2,3,6-trifluoro-4-iodophenyl], [BD BD 100; 2, 3, 5, 6-tetrafluoro-4-iodophenyl],

[BD101; 2-methylphenyl], [BD102; 3-methylphenyl], [BD103; 4-methylphenyl], [BD104; 2,3-dimethylphenyl], [BD105; 2,4-dimethylphenyl], [BD101; BD106; 2,5-dimethylphenyl], [BD107; 2,6-dimethylphenyl], [BD108; 3,4-dimethylphenyl], [BD109; 3,5-dimethylphenyl], [BD110; 5-trimethylphenyl], [BD111; 2,3,4-trimethylphenyl], [BD112; 2,3,6-trimethylphenyl], [BD113; 2,4,5-trimethylphenyl], [BD114; 4,6-trimethylphenyl], [BD115; 3,4,5-trimethylphenyl], [BD116; 2,3,4,6- tetramethylphenyl], [BD117; 2,3,5,6-tetramethyl Phenyl], [BD118; 2,3,4,5,6-pentamethylphenyl], [BD119; 2-ethylphenyl], [BD120; 3-ethylphenyl], [BD121; 4-ethylphenyl], [BD122 2,4-diethylphenyl], [BD 123; 2, 6-diethylphenyl], [BD 124; 3,5-diethylphenyl], [BD 125; 2, 4, 6-triethylphenyl], [BD 126; -Propylphenyl] , [BD127; 3-n-propylphenyl], [BD128; 4-n-propylphenyl], [BD129; 2-isopropylphenyl], [BD130; 3-isopropylphenyl], [BD131; 4-isopropylphenyl], [BD 132; 2,4-diisopropylphenyl], [BD 133; 2, 6-diisopropylphenyl], [BD 134; 3,5-diisopropylphenyl], [BD 135; 2-s-butylphenyl], [BD 136; 3-s -Butylphenyl], [BD 137; 4-s-butylphenyl], [BD 138; 2-t-butylphenyl], [BD 139; 3-t-butylphenyl], [BD 140; 4-t-butylphenyl], [BD BD 141; 4-butylphenyl], [BD 142; 4-nonylphenyl], [BD 143; 2-methyl-4-t-butylphenyl], [BD 144; 2-methyl-6-t-butylphenyl], [BD 145; 2-Methyl-4-isopropylphenyl], [BD 146; 2-methyl-5-isopropylphenyl], [BD 147; 3-methyl-4-isopropylphenyl], [BD 148; 2-cyclopropylphenyl], [BD 149; -Cyclopropylphenyl], [BD 150; 4-cyclopropylphenyl], [BD 151; 4- Cyclobutylphenyl], [BD 152; 4-cyclopentylphenyl], [BD 153; 4-hydroxyphenyl], [BD 154; 2-methoxyphenyl], [BD 155; 3-methoxyphenyl], [BD 156; 4-methoxyphenyl], [BD 157; 2-ethoxyphenyl], [BD 158; 3-ethoxyphenyl], [BD 159; 4-ethoxyphenyl], [BD 160; 2-propyloxyphenyl], [BD 161; 3-propyloxyphenyl], [BD 162; 4-propyloxyphenyl], [BD 163; 2-isopropyloxyphenyl], [BD 164; 3-isopropyloxyphenyl], [BD 165; 4-isopropyloxyphenyl], [BD 166; 2-hexyloxyphenyl], [BD 167; 3-Hexyloxyphenyl], [BD 168; 4-Hexyloxyphenyl], [BD 169; 2-benzyloxyphenyl], [BD 170; 3-benzyloxyphenyl], [BD 171; 4-benzyloxyphenyl], [BD 172; 2,3-Dimethoxyphenyl], [BD 173; 2,4-dimethoxyphenyl], [BD 174; 2, 5-dimethoxyphenyl], [BD 175; 2,6-Dimethoxyphenyl], [BD 176; 3,4-Dimethoxyphenyl], [BD 177; 3,5-Dimethoxyphenyl], [BD 178; 2-t-butoxyphenyl], [BD 179; 3-t-butoxyphenyl ], [BD 180; 4-t-butoxyphenyl], [BD 181; 2-trifluoromethoxyphenyl], [BD 182; 3-trifluoromethoxyphenyl], [BD 183; 4-trifluoromethoxyphenyl], [BD 184; -Pentafluoroethoxyphenyl], [BD 185; 3-pentafluoroethoxyphenyl], [BD 186; 4-pentafluoroethoxyphenyl], [BD 187; 2-phenoxyphenyl], [BD 188; 3-phenoxyphenyl], [BD 189; 4-phenoxyphenyl], [BD190; 4- (2-fluorophenoxy) phenyl], [BD191; 4- (3-chlorophenoxy) phenyl], [BD192; 4- (4-chlorophenoxy) phenyl], [BD193 2,3,6-trimethyl-4-fluorophenyl], [BD194; 2,3,6-trimethyl-4-chlorophenyl], [BD195; 2,3,6-trimethyl-4-bromophenyl], [BD196; 2,4-di Methyl-6-fluorophenyl], [BD 197; 2,4-dimethyl-6-chlorophenyl], [BD 198; 2,4-dimethyl-6-bromophenyl], [BD 199; 2-isopropyl-4-chloro-5- Methylphenyl], [BD 200; 2-methyl-5-isopropyl-4-chlorophenyl],

[BD 201; 3-fluoro-2-methoxyphenyl], [BD 202; 4-fluoro-2-methoxyphenyl], [BD 203; 5-fluoro-2-methoxyphenyl], [BD 204; 6-fluoro-2-methoxyphenyl ], [BD 205; 2-fluoro-3-methoxyphenyl], [BD 206; 4-fluoro-3-methoxyphenyl], [BD 207; 5-fluoro-3-methoxyphenyl], [BD 208; 6-fluoro-3- Methoxyphenyl], [BD 209; 2-fluoro-4-methoxyphenyl], [BD 210; 3-fluoro-4-methoxyphenyl], [BD 211; 3,4-difluoro-2-methoxyphenyl], [BD 212; 5-difluoro-2-methoxyphenyl], [BD 213; 3, 6-difluoro-2-methoxyphenyl], [BD 214; 4, 5-difluoro-2-methoxyphenyl], [BD 215; 4, 6-difluoro-2 -Methoxyphenyl], [BD216; 5,6-difluoro-2-methoxyphenyl], [BD217; 2,4-difluoro-3-methoxyphenyl], [BD218; 2,5-difluoro-3-methoxyphenyl], [BD219; 2,6-difluoro-3-methoxyphenyl], [BD22 0; 4,5-difluoro-3-methoxyphenyl], [BD 221; 4, 6-difluoro-3-methoxyphenyl], [BD 222; 5, 6-difluoro-3-methoxyphenyl], [BD 223; -Difluoro-4-methoxyphenyl], [BD224; 2,5-difluoro-4-methoxyphenyl], [BD 225; 2,6-difluoro-4-methoxyphenyl], [BD226; 3,5-difluoro-4- 4- Methoxyphenyl], [BD 227; 3, 6-difluoro-4-methoxyphenyl], [BD 228; 2, 3, 5-trifluoro-4-methoxyphenyl], [BD 229; 2, 3, 5, 6- tetrafluoro] -4-methoxyphenyl], [BD 230; 3-chloro-2-methoxyphenyl], [BD 231; 4-chloro-2-methoxyphenyl], [BD 232; 5-chloro-2-methoxyphenyl], [BD 233; 6 -Chloro-2-methoxyphenyl], [BD 234; 2-chloro-3-methoxyphenyl], [BD 235; 4-chloro-3-methoxyphenyl], [BD 236; 5-chloro-3-methoxyphenyl], [BD 237 6-chloro-3-methoxyphenyl], [BD 238; 2-chloro-4-methoxyphenyl], [BD 239; 3-chloro -4-Methoxyphenyl], [BD 240; 3,4-Dichloro-2-methoxyphenyl], [BD 241; 3,5-Dichloro-2-methoxyphenyl], [BD 242; 3, 6-Dichloro-2-methoxyphenyl ], [BD 243; 4, 5-dichloro-2-methoxyphenyl], [BD 244; 4, 6-dichloro-2-methoxyphenyl], [BD 245; 5, 6-dichloro-2- methoxyphenyl], [BD 246; 2,4-Dichloro-3-methoxyphenyl], [BD 247; 2, 5-dichloro-3-methoxyphenyl], [BD 248; 2, 6-dichloro-3-methoxyphenyl], [BD 249; 4, 5-dichloro -3-methoxyphenyl], [BD 250; 4, 6-dichloro-3-methoxyphenyl], [BD 251; 5, 6-dichloro-3-methoxyphenyl], [BD 252; 2,3-dichloro-4-methoxyphenyl ], [BD253; 2,5-dichloro-4-methoxyphenyl], [BD254; 2,6-dichloro-4-methoxyphenyl], [BD255; 3,5-dichloro-4-methoxyphenyl], [BD256; 3,6-dichloro-4-methoxyphenyl], [BD 257; 3-fluoro-2-trifluoromethoxyphenyl], [BD 258; 4-fluo -2- trifluoromethoxyphenyl], [BD 259; 5-fluoro-2-trifluoromethoxyphenyl], [BD 260; 6-fluoro-2-trifluoromethoxyphenyl], [BD 261; Fluoromethoxyphenyl], [BD 262; 4-fluoro-3-trifluoromethoxyphenyl], [BD 263; 5-fluoro-3-trifluoromethoxyphenyl], [BD 264; 6-fluoro-3-trifluoromethoxyphenyl], [BD 265; 2-fluoro-4-trifluoromethoxyphenyl], [BD 266; 3-fluoro-4-trifluoromethoxyphenyl], [BD 267; 3,4-difluoro-2-trifluoromethoxyphenyl], [BD 268; 3,5-Difluoro-2-trifluoromethoxyphenyl], [BD 269; 3,6-difluoro-2-trifluoromethoxyphenyl], [BD 270; 4, 5-difluoro-2-trifluoromethoxyphenyl], [BD 271 4,6-difluoro-2-trifluoromethoxyphenyl], [BD 272; 5,6-difluoro-2-trifluoro Oromethoxyphenyl], [BD 273; 2,4-difluoro-3-trifluoromethoxyphenyl], [BD 274; 2, 5-difluoro-3-trifluoromethoxyphenyl], [BD 275; 2, 6-difluoro-3- Trifluoromethoxyphenyl], [BD 276; 4, 5-difluoro-3-trifluoromethoxyphenyl], [BD 277; 4, 6-difluoro-3-trifluoromethoxyphenyl], [BD 278; 5, 6-difluoro-3 -Trifluoromethoxyphenyl], [BD 279; 2,3-difluoro-4-trifluoromethoxyphenyl], [BD 280; 2, 5-difluoro-4-trifluoromethoxyphenyl], [BD 281; 2, 6-difluoro- 4-trifluoromethoxyphenyl], [BD 282; 3,5-difluoro-4-trifluoromethoxyphenyl], [BD 283; 3, 6-difluoro-4-trifluoromethoxyphenyl], [BD 284; 2, 3, 5 -Trifluoro-4-trifluoromethoxyphenyl], [BD 285; 2,3,5,6-tetrafluoro-4-trifluoromethoxyphenyl], [BD2 86; 3-chloro-2-trifluoromethoxyphenyl], [BD 287; 4-chloro-2-trifluoromethoxyphenyl], [BD 288; 5-chloro-2-trifluoromethoxyphenyl], [BD 289; 6-chloro -2-trifluoromethoxyphenyl], [BD 290; 2-chloro-3-trifluoromethoxyphenyl], [BD 291; 4-chloro-3-trifluoromethoxyphenyl], [BD 292; 5-chloro-3-trifluoro] 6-Chloro-3-trifluoromethoxyphenyl], [BD 294; 2-chloro-4-trifluoromethoxyphenyl], [BD 295; 3-chloro-4-trifluoromethoxyphenyl], [methoxyphenyl], [BD 293; BD 296; 3,4-dichloro-2-trifluoromethoxyphenyl], [BD 297; 3,5-dichloro-2-trifluoromethoxyphenyl], [BD 298; 3, 6-dichloro-2-trifluoromethoxyphenyl], [BD 299; 4, 5-dichloro-2-trifluoromethoxyphenyl], [BD 300; 4, 6-dichloro-2-trifluoromethoxyphenyl],

[BD 301; 5,6-dichloro-2-trifluoromethoxyphenyl], [BD 302; 2,4-dichloro-3-trifluoromethoxyphenyl], [BD 303; 2, 5-dichloro-3-trifluoromethoxyphenyl] , [BD 304; 2,6-dichloro-3-trifluoromethoxyphenyl], [BD 305; 4,5-dichloro-3-trifluoromethoxyphenyl], [BD 306; 4,6-dichloro-3-trifluoromethoxyphenyl ], [BD 307; 5,6-dichloro-3-trifluoromethoxyphenyl], [BD 308; 2,3-dichloro-4-trifluoromethoxyphenyl], [BD 309; 2, 5-dichloro-4-trifluoromethoxy Phenyl], [BD 310; 2,6-dichloro-4-trifluoromethoxyphenyl], [BD 311; 3,5-dichloro-4-trifluoromethoxyphenyl], [BD 312; 3, 6-dichloro-4-trifluoro] Methoxyphenyl], [BD 313; 2-carbamoylphenyl], [BD 314; 3-carbamoylphenyl], [BD 315; 4-carbamoylphenyl], [BD 316; 2- (N-methylamino) Bonyl) phenyl], [BD 317; 3- (N-methylaminocarbonyl) phenyl], [BD 318; 4- (N-methylaminocarbonyl) phenyl], [BD 319; 2- (N, N-dimethylaminocarbonyl) phenyl ], [BD 320; 3- (N, N-dimethylaminocarbonyl) phenyl], [BD 321; 4- (N, N-dimethylaminocarbonyl) phenyl], [BD 322; 2-methoxycarbonylphenyl], [BD 323; 3] -Methoxycarbonylphenyl], [BD 324; 4-Methoxycarbonylphenyl], [BD 325; 4- acetoxyphenyl], [BD 326; 2-methoxymethylphenyl], [BD 327; 3-methoxymethylphenyl], [BD 328; 4- Methoxymethylphenyl], [BD 329; 2-formylphenyl], [BD 330; 3-formylphenyl], [BD 331; 4-formylphenyl], [BD 332; 2-methyl-5-bromophenyl], [BD 333; 2- Methyl-6-bromophenyl], [BD 334; 2-chloro-3-methylphenyl], [BD 335; 2-chloro-4-methylphenyl], [BD 336; 2-chloro-5-methylphenyl] [BD 337; 2-fluoro-3-methylphenyl], [BD 338; 2-fluoro-4-methylphenyl], [BD 339; 2-fluoro-5-methylphenyl], [BD 340; 2-bromo-3-methyl Phenyl], [BD 341; 2-bromo-4-methylphenyl], [BD 342; 2-bromo-5-methylphenyl], [BD 343; 3-methyl-4-chlorophenyl], [BD 344; 3-methyl-5- Chlorophenyl], [BD 345; 3-methyl-4-fluorophenyl], [BD 346; 3-methyl-5-fluorophenyl], [BD 347; 3-methyl-4-bromophenyl], [BD 348; 3-methyl-5 -Bromophenyl], [BD 349; 3-fluoro-4-methylphenyl], [BD 350; 3-chloro-4-methylphenyl], [BD 351; 3-bromo-4-methylphenyl], [BD 352; 2-chloro -4,5-dimethylphenyl], [BD 353; 2-bromo-4,5-dimethylphenyl], [BD 354; 2-chloro-3,5-dimethylphenyl], [BD 355; 2-bromo-3,5- Dimethylphenyl], [BD 356; 2,6-dibromo-4-methylphenyl], [BD 357; 2,4-dichloro-6-methylphenyl], [BD 358; 2,4-difluoro- 6-methylphenyl], [BD 359; 2,4-dibromo-6-methylphenyl], [BD 360; 2, 6-dimethyl-4-fluorophenyl], [BD 361; 2, 6-dimethyl-4-chlorophenyl], [BD362; 2,6-dimethyl-4-bromophenyl], [BD 363; 3,5-dimethyl-4-fluorophenyl], [BD 364; 3,5-dimethyl-4-chlorophenyl], [BD 365; -Dimethyl-4-bromophenyl], [BD 366; 2,3-difluoro-4-methylphenyl], [BD 367; 2, 5-difluoro-4-methylphenyl], [BD 368; 3,5-difluoro-4- Methylphenyl], [BD 369; 2, 3, 5-trifluoro-4-methylphenyl], [BD 370; 2, 3, 6-trifluoro-4-methylphenyl], [BD 371; -Tetrafluoro-4-methylphenyl], [BD 372; 2-fluoro-4-ethylphenyl], [BD 373; 3-fluoro-4-ethylphenyl], [BD 374; 2,3-difluoro-4-ethylphenyl] [BD 375; 2, 6-difluoro-4-ethylphenyl], [BD 376; 2, 5-difluoro-4-ethylphenyl], [BD 377; [BD378; 2,3,5-trifluoro-4-ethylphenyl], [BD379; 2,3,6-trifluoro-4-ethylphenyl], [BD380; 2,3,5,6- Tetrafluoro-4-ethylphenyl], [BD 381; 2-trifluoromethylphenyl], [BD 382; 3-trifluoromethylphenyl], [BD 383; 4-trifluoromethylphenyl], [BD 384; 4- (2, 2,2-Trifluoro-1-trifluoromethyl-ethyl) phenyl], [BD 385; 4- (2,2-difluoroethoxy) phenyl], [BD 386; 4- (2,2,2-trifluoroethoxy) Phenyl], [BD 387; 2-nitrophenyl], [BD 388; 3-nitrophenyl, [BD 389; 4-nitrophenyl], [BD 390; 2-cyanophenyl], [BD 391; 3-cyanophenyl], [BD 392; 4-Cyanophenyl], [BD 393; 2-methyl-3-chlorophenyl], [BD 394; 2-methyl-4-chlorophenyl], [BD 395; 2-methyl-5-chlorophenyl], [BD 396; 2-methyl-6 -Chlorophenyl], [BD 397; 2-methyl-3-fluorophenyl], [BD 398; 2-methyl-4-fluoropheny ], [BD399; 2- methyl-5-fluorophenyl], [BD400; 2- methyl-6-fluorophenyl,

[BD 401; 2-methyl-3-bromophenyl], [BD 402; 2-methyl-4-bromophenyl], [BD 403; 4-methylthiophenyl], [BD 404; 4-methylsulfonylphenyl], [BD 405; Methylsulfinylphenyl], [BD406; 4-trifluoromethylthiophenyl], [BD407; 4-ethynylphenyl], [BD408; 4- (1-propynyl) phenyl], [BD409; 4-vinylphenyl], [BD410; 4- (2,2-dichlorovinyl) phenyl], [BD411; 4- (2,2-difluorovinyl) phenyl], [BD 412; cyclohexyl], [BD 413; 2-chlorocyclohexyl], [BD 414; 3-chloro Cyclohexyl], [BD 415; 4-chlorocyclohexyl], [BD 416; 4, 4-dichlorocyclohexyl], [BD 417; 2-bromocyclohexyl], [BD 418; 3-bromocyclohexyl], [BD 419; 4-bromocyclohexyl], [BD 420; 4, 4-dibromocyclohexyl], [BD 421; 2-iodocyclohexyl], [BD 422; 3-iodocyclohexyl], [BD 423; 4-iodocyclohexyl], [BD 424; Rocyclohexyl], [BD 425; 3-fluorocyclohexyl], [BD 426; 4-fluorocyclohexyl], [BD 427; 4, 4-difluorocyclohexyl], [BD 428; 4-methylcyclohexyl], [BD 429; 4-ethylcyclohexyl] , [BD430; 4-methoxycyclohexyl], [BD 431; 4-ethoxycyclohexyl], [BD 432; 4-trifluoromethoxycyclohexyl], [BD 433; 1-cyclohexenyl], [BD 434; 2-cyclohexenyl], [BD 435 3-Cyclohexenyl], [BD 436; 4-fluoro-1-cyclohexenyl], [BD 437; 4-fluoro-2-cyclohexenyl], [BD 438; 4-fluoro-3-cyclohexenyl], [BD 439; -Chloro-1-cyclohexenyl, [BD440; 3-chloro-1-cyclohexenyl], [BD 441; 4-chloro-1-cyclohexenyl], [BD 442; 5-chloro-1-cyclohexenyl], [BD 443; 6-chloro-1-cyclohexenyl], [BD 444; 1-chloro-2-cyclohexenyl], [BD 445; 2-chloro-2-cyclohexenyl], [BD 446; 3-chloro-2 -Cyclohexenyl], [BD 447; 4-chloro-2-cyclohexenyl], [BD 448; 5-chloro-2-cyclohexenyl], [BD 449; 6-chloro-2-cyclohexenyl], [BD 450; 1-chloro -3-cyclohexenyl], [BD 451; 2-chloro-3-cyclohexenyl], [BD 452; 3-chloro-3-cyclohexenyl], [BD 453; 4-chloro-3-cyclohexenyl], [BD 454; -Chloro-3-cyclohexenyl], [BD 455; 6-chloro-3-cyclohexenyl], [BD 456; 4-bromo-1-cyclohexenyl], [BD 457; 4-bromo-2-cyclohexenyl], [BD 458 4-bromo-3-cyclohexenyl], [BD 459; 4-methyl-1-cyclohexenyl], [BD 460; 4-methyl-2-cyclohexenyl], [BD 461; 4-methyl-3-cyclohexenyl], [BD 462: 4-ethyl-1-cyclohexenyl], [BD 463; 4-ethyl-2-cyclohexenyl], [BD 464; 4-ethyl-3-cyclohexenyl], [BD 465: 4-methoxy-1-cyclohexenyl ], [BD 466; 4-methoxy-2-cyclohexenyl], [BD 467; 4-trifluoro Methoxy-1-cyclohexenyl], [BD 468; 4-trifluoromethoxy-2-cyclohexenyl], [BD 469; morpholino], [BD 470; thiomorpholino], [BD 471; piperidino], [BD 472; 4-methoxy piperidine No, [BD 473; piperazinyl], [BD 474; N-methylpiperazinyl], [BD 475; pyrrolyl], [BD 476; imidazolyl], [BD 477; pyrazolyl], [BD 478; ], [BD 479; 4, 5-dimethyl-pyrazol-1-yl], [BD 480; 3-methyl-pyrazol-1-yl], [BD 481; 3,4-dimethyl-pyrazol-1-yl], [BD 482 4-methoxy-3,5-dimethyl-pyrazol-1-yl], [BD 483; 1-methyl-1H-pyrazol-3-yl], [BD 484; 1,4,5-trimethyl-1H-pyrazole-3; -Yl], [BD 485; 1,4-dimethyl-5-methoxy-1H-pyrazol-3-yl], [BD 486; 2-pyridyl], [BD 487; 3-pyridyl], [BD 488; 4-pyridyl], [BD 489; 5-methoxy-2-pyridyl], [BD 490; 5-trifluoromethoxy-2-pyridyl], [BD 491; 5-fluoro-2-pyridyl], [BD 492; 5-chloro-2-pyridyl], [BD 493; 6-methoxy-3-pyridyl], [BD 494; 6-trifluoromethoxy-3-pyridyl], [BD 495; 6-fluoro-3-pyridyl], [BD 496; 6-chloro-3-pyridyl], [BD 497; 5-methoxy-2-pyrazinyl], [BD 498; 5-trifluoromethoxy-2-pyrazinyl], [BD 499; 5-fluoro-2-pyrazinyl], [BD 500; 5-chloro-2-pyrazinyl],

[BD501; 5-methoxy-2-pyrimidinyl], [BD 502; 5-trifluoromethoxy-2-pyrimidinyl], [BD 503; 5-fluoro-2-pyrimidinyl], [BD 504; 5-chloro-2-pyrimidinyl], [BD 505; 6-methoxy-3-pyridazinyl], [BD 506; 6-trifluoromethoxy-3-pyridazinyl], [BD 507; 6-fluoro-3-pyridazinyl], [BD 508; 6-chloro-3-pyridazinyl], [BD 509; 1-naphthyl], [BD 510; 2-naphthyl], [BD 511; 2-quinolyl], [BD 512; 3-quinolyl], [BD 513; 4-quinolyl], [BD 514; 5-quinolyl], [BD 515 6-quinolyl], [BD 516; 7-quinolyl], [BD 517; 8-quinolyl], [BD 518; 3-isoquinolyl], [BD 519; 6-isoquinolyl], [BD 520; , 4- (methylenedioxy) phenyl], [BD 522; 2-ethoxy-4-methoxyphenyl], [BD 523; 2-isopropyloxy-4-methoxyphenyl], [BD 524; 4-ethoxy-2-methoxyphenyl] , [BD 525; 4-isopropyloxy-2-methoxyphenyl], [BD 526; 4-oxy-2-isopropyloxyphenyl], [BD 528; 4-bromo-2-isopropyloxyphenyl], [BD 529; 4-fluoro-2-ethoxyphenyl], [BD 530; 4 -Chloro-2-ethoxyphenyl], [BD 531; 4-bromo-2-ethoxyphenyl], [BD 532; 4-cyano-2-methoxyphenyl], [BD 533; 4-cyano-2-ethoxyphenyl], [BD 534 4-cyano-2-isopropyloxyphenyl], [BD 535; 2-methoxy-3-pyridyl], [BD 536; 6-chloro-2-methoxy-3-pyridyl], [BD 537; 6-fluoro-2-methoxy 6-Bromo-2-methoxy-3-pyridyl], [BD 539; 6-ethoxy-2-methoxy-3-pyridyl], [BD 540; 2, 6-dimethoxy-3-pyridyl] ], [BD 541; 6-trifluoromethyl-2-methoxy-3-pyridyl], [BD 542; 6-cyano-2-methoxy-3-pyridyl], [BD 543; 2-ethoxy-3-pyridyl], [BD 544] 6-chloro-2-ethoxy-3-pyridyl], [BD 545; 6-fluoro-2-ethoxy-3-pyridyl], [B D 546; 6-bromo-2-ethoxy-3-pyridyl], [BD 547; 2-ethoxy-6-methoxy-3-pyridyl], [BD 548; 2, 6-diethoxy-3- pyridyl], [BD 549; Trifluoromethyl-2-ethoxy-3-pyridyl], [BD 550; 6-cyano-2-ethoxy-3-pyridyl], [BD 551; 2-isopropyloxy-3-pyridyl], [BD 552; 6-chloro-2 -Isopropyloxy-3-pyridyl], [BD 553; 6-fluoro-2-isopropyloxy-3-pyridyl], [BD 554; 6-bromo-2-isopropyloxy-3-pyridyl], [BD 555; 2-isopropyloxy -6-Methoxy-3-pyridyl], [BD 556; 2,6-diisopropyloxy-3-pyridyl], [BD 557; 6-trifluoromethyl-2-isopropyloxy-3-pyridyl], [BD 558; 6-cyano -2-isopropyloxy-3-pyridyl].
.

  Further, the present compounds AE1-BE1 to AE5220-BE5982 can also be obtained according to the method described above.

The present compounds AE1-BE1 to AE5220-BE5982 are compounds represented by the following formula (AEBE).
[Wherein, X ^{51 to} X ⁵⁸ each represent a substituent corresponding to each of the substituent numbers (ME 1) AE 1 to AE 2 220 shown below, wherein E ¹⁰⁵ is a substituent number (ME 2) BE 1 shown below ~ BE 5982 is represented. ]
For example, the present compounds AE1-BE1, in the compounds of formula (AEBE), X ⁵¹ ~X ⁵⁸ substituents ID ^{ME1 (X 51, X 52,} X 54 ~X 56 and X ⁵⁷ is a hydrogen atom, X ⁵³ And X ⁵⁸ is an oxygen atom), and E ¹⁰⁵ is a compound in which the substituent number (ME 2) is BE 1 (pyridin-2-yl group), and is represented by the following formula.
[Substituent number (ME1): X ⁵¹ , X ⁵² , X ⁵³ , X ⁵⁴ , X ⁵⁵ , X ⁵⁶ , X ⁵⁷ , X ⁵⁸ ], [AE 1; H, H, O, H, H, H, H, H, O], [AE2; H, H, O, F, H, H, O], [AE3; H, H, O, Cl, H, H, H, O], [AE 4; H, H, H, O, Br, H, H, H, O], [AE5; H, H, O, I, H, H, H, O], [AE 6; H, H, O, Me, H, H, H, H, H O], [AE7; H, H, O, Et, H, H, O], [AE 8; H, H, O, Pr, H, H, H, O], [AE 9; H, H, H, O, i-Pr, H, H, H, O], [AE 10; H, H, O, CH = CH ₂ , H, H, H, O], [AE 11; H, H, O, C (Me ) = CH ₂ , H, H, H, O], [AE 12; H, H, O, C≡CH, H, H, H, O], [AE 13; H, H, O, C≡ CMe, H , H, H, O], [AE 14; H, H, O, c-Pr, H, H, H, O], [AE 15; H, H, O, OMe, H, H, H, O], [AE16; H, H, O, OEt, H, H, H, O], [AE 17; H, H, O, Oi-Pr, H, H, H, O], [AE 18; H, H, O , SMe, H, H, H, O], [AE 19; H, H, O, SEt, H, H, H, O], [AE 20; H, H, O, CH ₂ F, H, H, H , O], [AE21; H , H, O, CHF 2, H, H, H, O], [AE22; H, H, O, CF 3, H, H, H, O], [AE23; H _{, H, O, OCH 2 F} , H, H, H, O], [AE24; H, H, O, OCHF 2, H, H, H, O], [AE25; H, H, O, OCF 3 H, H, H, O], [AE 26; H, H, O, SCH ₂ F, H, H, H, O], [AE 27; H, H, O, SCHF ₂ , H, H, H, H, O, [AE 28; H, H, O, SCF ₃ , H, H, H, O], [AE 29; H, H, O, CN, H, H, H, O], [AE 30; H, H , O, NO ₂ , H, H, H, O], [AE 31; Me, H, O, H, H, H, H, O], [AE 32; Me, H, O, F, H, H, H, H, O], [AE 33; Me, H, O, Cl, H, H, H, O], [AE 34; Me, H, O, Br, H, H, H, O], [AE 35; Me, H, O, I, H, H, H, O], [AE 36; Me, H, O, Me, H, H, H, O], [AE 37; Me, H, O, Et, H, H, H, O], [AE 38; Me, H, O, Pr, H, H, H, O], [AE 39; Me, H, O, i-Pr, H, H, H, O], [AE 40; Me, H, O, CH = CH ₂ , H, H, H, O], [AE 41; Me, H, O, C (Me ) = CH ₂ , H, H, H, O], [AE 42; Me, H, O, C≡CH, H, H, H, O], [AE 43; Me, H, O, C≡ CMe, H , H, H, O], [AE 44; Me, H, O, c-Pr, H, H, H, O], [AE 45; Me, H, O, OMe, H, H, H, O], [AE 46; Me, H, O, OEt, H, H, H, O], [AE 47; Me, H, O, Oi-Pr, H, H, H, O], [AE 48: Me, H, O , SMe, H, H, H, O], [AE 49; Me, H, O, SEt, H, H, H, O], [AE 50; Me, H, O, CH ₂ F, H, H, H , O], [AE 51; Me, H, O, CHF ₂ , H, H, H, O], [AE 52; Me, H, O, CF ₃ , H, H, H, O], [AE 53; Me _{, H, O, OCH 2 F} , H, H, H, O], [AE54; Me, H, O, OCHF 2, H, H, H, O], [AE55; Me, H, O, OCF 3 , H, H, H, O], [AE56; Me, H, O, SCH ₂ F, H, H, H, O], [AE 57; Me, H, O, SCHF ₂ , H, H, H, H, O], [AE 58; Me, H, O, SCF ₃ , H, H, H, O], [AE 59; Me, H, O, CN, H, H, H, O], [AE 60; Me, H , O, NO ₂ , H, H, H, O], [AE 61; Et, H, O, H, H, H, H, O], [AE 62; Et, H, O, F, H, H, H, H, O], [AE 63; Et, H, O, Cl, H, H, H, O], [AE 64; Et, H, O, Br, H, H, H, O], [AE 65; Et, Et, H, O, I, H, H, H, O, [AE 66; Et, H, O, Me, H, H, H, O], [AE 67; Et, H, O, Et, H, H, H, H, O], [AE 68; Et, H, O, Pr, H, H, H, O], [AE 69; Et, H, O, i-Pr, H, H, H, O], [AE 70; Et, H, O, CH = CH 2, H, H, H, O], [AE71; Et, H, O, C (Me) = CH 2, H, H, H, O], [AE72; Et , H, O, C≡CH, H, H, H, O], [A E73; Et, H, O, C≡CMe, H, H, H, O], [AE 74; Et, H, O, c-Pr, H, H, H, O], [AE 75; Et, H, O, OMe, H, H, H, O], [AE 76; Et, H, O, OEt, H, H, H, O], [AE 77; Et, H, O, Oi-Pr, H, H, H, O], [AE 78; Et, H, O, SMe, H, H, H, O], [AE 79; Et, H, O, SE, H, H, H, O], [AE 80; Et, _{H, O, CH 2 F,} H, H, H, O], [AE81; Et, H, O, CHF 2, H, H, H, O], [AE82; Et, H, O, CF 3, H, H, H, O], [AE 83; Et, H, O, OCH ₂ F, H, H, H, O], [AE 84; Et, H, O, OCHF ₂ , H, H, H, O ], [AE85; Et, H , O, OCF 3, H, H, H, O], [AE86; Et, H, O, SCH 2 F, H, H, H, O], [AE87; Et, _{H, O, SCHF 2, H} , H, H, O], [AE88; Et, H, O, SCF 3, H, H, H, O], [AE89; Et, H, O, CN, H, H, H, O], [AE 90; Et, H, O, NO ₂ , H, H, O], [AE 91; F, H, O, H, H, H, H, O], [AE 92 F, H, O, F, H, H, H, O], [AE93; F, H, O, Cl, H, H, H, O], [AE94; F, H, O, Br, H] , H, H, O], [AE 95; F, H, O, I, H, H, H, O], [AE 96; F, H, O, Me, H, H, H, O], [AE 97 F, H, O, Et, H, H, H, O], [AE 98; F, H, O, Pr, H, H, H, O], [AE 99; F, H, O, i-Pr , H, H, H, O], [AE 100; F, H, O, CH = CH ₂ , H, H, H, O],

[AE 101; F, H, O, C (Me) = CH ₂ , H, H, H, O], [AE 102; F, H, O, C≡CH, H, H, H, O], [AE 103 F, H, O, C≡CMe, H, H, H, O], [AE 104; F, H, O, c-Pr, H, H, H, O], [AE 105; F, H, O , OMe, H, H, H, O], [AE 106; F, H, O, OEt, H, H, H, O], [AE 107; F, H, O, Oi-Pr, H, H, H , O], [AE108; F, H, O, SMe, H, H, H, O], [AE109; F, H, O, SEt, H, H, H, O], [AE 110; F, H _{, O, CH 2 F, H} , H, H, O], [AE111; F, H, O, CHF 2, H, H, H, O], [AE112; F, H, O, CF 3, H , H, H, O], [AE 113; F, H, O, OCH ₂ F, H, H, H, O], [AE 114; F, H, O, OCHF ₂ , H, H, H, O] , [AE115; F, H, O, OCF 3, H, H, H, O], [AE116; F, H, O, SCH 2 F, H, H, H, O], [AE117; F, H , O, SCHF ₂ , H, H, H, O], [AE 118; F, H, O, SCF ₃ , H, H, H, O], [AE 119; F, H, O, CN, H, H , H, O], [AE 120; F, H, O, NO ₂ , H, H, O], [AE 121; Cl, H, O, H, H, H, H, O], [AE 122; Cl, H, O, F, H, H, H, O], [AE 123; Cl, H, O, Cl, H, H, H, O], [AE 124; Cl, H, O, Br, H, H, H, O], [AE 125; Cl, H, O, I, H, H, H, O], [AE 126; Cl, H, O, Me, H, H, H, O], [AE 127; Cl, H, O, Et, H, H, H, O], [AE 128; Cl, H, O, Pr, H, H, H, O], [AE 129; Cl, H, O, i-Pr, H, H, H, O] , [AE130; Cl, H, O, CH = CH 2, H, H, H, O], [AE131; Cl, H, O, C (Me) = CH 2, H , H, H, O], [AE 132; Cl, H, O, C≡CH, H, H, H, O], [AE 133; Cl, H, O, C≡ C Me, H, H, H, O ], [AE134; Cl, H, O, c-Pr, H, H, H, O], [AE 135; Cl, H, O, OMe, H, H, H, O], [AE 136; Cl, H , O, O Et, H, H, H, O], [AE 137; Cl, H, O, Oi-Pr, H, H, H, O], [AE 138; Cl, H, O, SMe, H, H, H, O], [AE139; Cl, H, O, SEt, H, H, H, O], [AE140; Cl, H, O, CH 2 F, H, H, H, O], [AE141; Cl, _{H, O, CHF 2, H} , H, H, O], [AE142; Cl, H, O, CF 3, H, H, H, O], [AE143; Cl, H, O, OCH 2 F, H, H, H, O] , [AE144; Cl, H, O, OCHF 2, H, H, H, O], [AE145; Cl, H, O, OCF 3, H, H, H, O] [AE 146; Cl, H, O, SCH ₂ F, H, H, H, O], [AE 147; Cl, H, O, SCHF ₂ , H, H, H, O], [AE 148; Cl, H , O, SCF ₃ , H, H, H, O], [AE 149; Cl, H, O, CN, H, H, H, O], [AE 150; Cl, H, O, NO ₂ , H, H , H, O], [AE 151; Br, H, O, H, H, H, H, O], [AE 152; Br, H, O, F, H, H, H, O], [AE 153; Br , H, O, Cl, H, H, H, O, [AE 154; Br, H, O, Br, H, H, H, O], [AE 155; Br, H, O, I, H, H] , H, O], [AE156; Br, H, O, Me, H, H, H, O], [AE 157; Br, H, O, Et, H, H, H, O], [AE 158; Br , H, O, Pr, H, H, H, O, [AE 159; Br, H, O, i-Pr, H, H, H, O], [AE 160; Br, H, O, CH = CH _{2, H, H, H,} O], [AE161; Br, H, O, C (Me) = CH 2, H, H, H, O], [AE162; Br, H, O, C≡CH, H, H, H, O], [AE163; Br, H, O, C≡CMe, H, H, H, O], [AE 164; Br, H, O, c-Pr, H, H, H, H, O], [AE 165; Br, H, O, OMe, H, H, H, O], [AE 166; Br, H, O, OEt, H, H, H, O], [AE 167; Br, H, O, Oi-Pr, H, H, H, O], [AE 168; Br, H, O, SMe, H, H, H, O], [AE 169; Br, H, O, SEt, H, H, H, O], [AE170; Br, H, O, CH 2 F, H, H, H, O], [AE171; Br, H, O, CHF 2, H, H, H, O] , [AE172; Br, H, O, CF 3, H, H, H, O], [AE173; Br, H, O, OCH 2 F, H, H, H, O ], [AE174; Br, H , O, OCHF 2, H, H, H, O], [AE175; Br, H, O, OCF 3, H, H, H, O], [AE176; Br, H , O, SCH ₂ F, H, H, H, O, [AE 177; Br, H, O, SCHF ₂ , H, H, H, O], [AE 178; Br, H, O, SCF ₃ , H , H, H, O], [AE 179; Br, H, O, CN, H, H, H, O], [AE 180; Br, H, O, NO ₂ , H, H, H, O], [[ AE 181; I, H, O, H, H, H, H, O], [AE 182; I, H, O, F, H, H, H, O], [AE 183; I, H, O, Cl, H, H, H, O], [AE 184; I, H, O, Br, H, H, O], [AE 185; I, H, O, I, H, H, H, O], [A AE 186; I, H, O, Me, H, H, H, O], [AE 187; I, H, O, Et, H, H, H, O], [AE 188; I, H, O, Pr, H, H, H, O] , [AE189; I, H, O, i-Pr, H, H, H, O], [AE190; I, H, O, CH = CH 2, H, H, H , O], [AE191; I , H, O, C (Me) = CH 2, H, H, H, O], [AE192; I, H, O, C≡CH, H, H, H, O ], [AE193; I, H, O, C≡CMe, H, H, H, O], [AE 194; I, H, O, c-Pr, H, H, H, O], [AE 195; , H, O, OMe, H, H, H, O], [AE 196; I, H, O, OEt, H, H, H, O], [AE 197; I, H, O, Oi-Pr, H , H, H, O], [AE 198; I, H, O, SMe, H, H, H, O], [AE 199; I, H, O, SE t, H, H, H, O], [AE 200 I, H, O, CH ₂ F, H, H, H, O],

[AE201; I, H, O , CHF 2, H, H, H, O], [AE202; I, H, O, CF 3, H, H, H, O], [AE203; I, H, O , OCH ₂ F, H, H, H, O], [AE 204; I, H, O, OCHF ₂ , H, H, H, O], [AE 205; I, H, O, OCF ₃ , H, H , H, O], [AE 206; I, H, O, SCH ₂ F, H, H, H, O], [AE 207; I, H, O, SCHF ₂ , H, H, H, O], [[ AE208; I, H, O, SCF 3, H, H, H, O], [AE209; I, H, O, CN, H, H, H, O], [AE210; I, H, O, NO _{2, H, H, H,} O], [AE211; CHF 2, H, O, H, H, H, H, O], [AE212; CHF 2, H, O, F, H, H, H, _{O], [AE213; CHF 2} , H, O, Cl, H, H, H, O], [AE214; CHF 2, H, O, Br, H, H, H, O], [AE215; CHF 2 , H, O, I, H , H, H, O], [AE216; CHF 2, H, O, Me, H, H, H, O], [AE217; CHF 2, H, O, Et, H , H, H, O], [AE218; CHF 2, H, O, Pr, H, H, H, O], [AE219; CHF 2, H, O, i-Pr, H, H, H, O ], [AE 220; CHF ₂ , H, O, CH = CH ₂ , H, H, H, O], [AE 221; CHF ₂ , H, O, C (Me) = CH ₂ , H, H, H, H _{O], [AE222; CHF 2} , H, O, C≡CH, H, H, H, O], [AE223; CHF 2, H, O, C≡CMe, H, H, H, O], [ _{AE224; CHF 2, H, O} , c-Pr, H, H, H, O], [AE225; CHF 2, H, O, OMe, H, H, H, O], [AE226; CHF 2, H , O, OEt, H, H , H, O], [AE227; CHF 2, H, O, Oi-Pr, H, H, H, O], [AE228; CHF 2, H, O, SMe, H , H, H, O], [AE 229; CHF ₂ , H, O, SE t, H, H, H, O], [AE 230; CHF ₂ , H, O, CH ₂ F, H, H, H, O _{], [AE231; CHF 2,} H, O, CHF 2, H, H, H, O], [AE232; CHF 2, H, O, CF 3, H, H, H, O], [AE233; CH F ₂ , H, O, OCH ₂ F, H, H, H, O], [AE234; CHF ₂ , H, O, OCHF ₂ , H, H, H, O], [AE 235; CHF ₂ , H, H, O, _{O, OCF 3, H, H} , H, O], [AE236; CHF 2, H, O, SCH 2 F, H, H, H, O], [AE237; CHF 2, H, O, SCHF 2, H, H, H, O] , [AE238; CHF 2, H, O, SCF 3, H, H, H, O], [AE239; CHF 2, H, O, CN, H, H, H, O _{], [AE240; CHF 2,} H, O, NO 2, H, H, H, O], [AE241; CF 3, H, O, H, H, H, H, O], [AE242; CF 3 , H, O, F, H , H, H, O], [AE243; CF 3, H, O, Cl, H, H, H, O], [AE244; CF 3, H, O, Br, H , H, H, O], [AE245; CF 3, H, O, I, H, H, H, O], [AE246; CF 3, H, O, Me, H, H, H, O], _{[AE247; CF 3, H,} O, Et, H, H, H, O], [AE248; CF 3, H, O, Pr, H, H, H, O], [AE249; CF 3, H, O, i-Pr, H, H, H, O, [AE 250; CF ₃ , H, O, CH = CH ₂ , H, H, H, O], [AE 251; CF ₃ , H, O, C _{(Me) = CH 2, H} , H, H, O], [AE252; CF 3, H, O, C≡CH, H, H, H, O], [AE253; CF 3, H, O, C ≡CMe, H, H, H, O], [AE254; CF ₃ , H, O, c-Pr, H, H, H, O], [AE 255; CF ₃ , H, O, OMe, H, H , H, O], [AE256 ; CF 3, H, O, OEt, H, H, H, O], [AE257; CF 3, H, O, Oi-Pr, H, H, H, O], _{[AE258; CF 3, H,} O, SMe, H, H, H, O], [AE259; CF 3, H, O, SEt, H, H, H, O], [AE260; CF 3, H, _{O, CH 2 F, H,} H, H, O], [AE261; CF 3, H, O, CHF 2, H, H, H, O], [AE262; CF 3, H, O, CF 3, H, H, H, O] , [AE263; CF 3, H, O, OCH 2 F, H, H, H, O], [AE264; CF 3, H, O, OCHF 2 , H, H, H, O], [AE 265; CF ₃ , H, O, OCF ₃ , H, H, H, O], [AE 266; CF ₃ , H, O, SCH ₂ F, H, H, H H, O], [AE267; CF 3, H, O, SCHF 2, H, H, H, O], [AE268; CF 3, H, O, SCF 3, H, H, H, O], [ _{AE269; CF 3, H, O} , CN, H, H, H, O], [AE270; CF 3, H, O, NO 2, H, H, H, O], [AE271; OMe, H, O , H, H, H, H, O], [AE 272; OMe, H, O, F, H, H, H, O], [AE 273; OMe, H, O, Cl, H, H, H, O ], [AE 274; OMe, H, O, Br, H, H, O], [AE 275; OMe, H, O, I, H, H, H, O], [AE 276: OMe, H, O] , Me, H, H, H, O], [AE 277; OMe, H, O, Et, H, H, H, O], [AE 278; OMe, H, O, Pr, H, H, H, O] ], [AE279; OMe, H , O, i-Pr, H, H, H, O], [AE280; OMe, H, O, CH = CH 2, H, H, H, O], [AE281; OMe, H, O, C ( Me) = CH 2, H, H, H, O], [AE282; OMe, H, O, C≡CH, H, H, H, O], [AE283; OMe, H, O, C≡CMe, H, H, H, O], [AE 284; OMe, H, O, c-Pr, H, H, H, O], [AE 285; OMe, H, O, OMe, H, H, H, O], [AE 286; OMe, H, O, OEt, H, H, H, O], [AE 287; OMe, H, O, Oi-Pr, H, H, H, O] [AE 288; OMe, H, O, SMe, H, H, H, O], [AE 289; OMe, H, O, SE t, H, H, H, O], [AE 290; OMe, H, O, _{CH 2 F, H, H,} H, O], [AE291; OMe, H, O, CHF 2, H, H, H, O], [AE292; OMe, H, O, CF 3, H, H, H, O], [AE 293; OMe, H, O, OCH ₂ F, H, H, H, O], [AE 294; OMe, H, O, OCHF ₂ , H, H, H, O], [AE 295 ; OMe, H, O, OCF 3, H, H, H, O], [AE296; OMe, H, O, SCH 2 F, H, H, H, O], [AE297; OMe, H, O, SCHF ₂ , H, H, H, O ], [AE 298; OMe, H, O, SCF ₃ , H, H, H, O], [AE 299; OMe, H, O, CN, H, H, H, O], [AE 300; OMe, H, O, NO ₂ , H, H, H, O],

[AE301; OEt, H, O, H, H, H, H, O], [AE 302; OEt, H, O, F, H, H, H, O], [AE 303; OEt, H, O, Cl] , H, H, H, O], [AE 304; OEt, H, O, Br, H, H, H, O], [AE 305; OEt, H, O, I, H, H, H, O], [AE306; OEt, H, O, Me, H, H, H, O], [AE 307; OEt, H, O, Et, H, H, H, O], [AE 308; OEt, H, O, Pr , H, H, H, O ], [AE309; OEt, H, O, i-Pr, H, H, H, O], [AE310; OEt, H, O, CH = CH 2, H, H, H, O], [AE311; OEt, H, O, C (Me) = CH 2, H, H, H, O], [AE312; OEt, H, O, C≡CH, H, H, H, O], [AE 313; OEt, H, O, C≡CMe, H, H, H, O], [AE 314; OEt, H, O, c-Pr, H, H, H, O], [AE 315; OEt, H, O, OMe, H, H, H, O], [AE 316; OEt, H, O, OEt, H, H, H, O], [AE 317; OEt, H, O, Oi-Pr, H, H, H, O], [AE 318; OEt, H, O, SMe, H, H, H, O], [AE 319; OEt, H, O, SE t, H, H, H, O], [ AE320; OEt, H, O, CH 2 F, H, H, H, O], [AE321; OEt, H, O, CHF 2, H, H, H, O], [AE322; OEt, H, O _{, CF 3, H, H,} H, O], [AE323; OEt, H, O, OCH 2 F, H, H, H, O], [AE324; OEt, H, O, OCHF 2, H, H , H, O], [AE325 ; OEt, H, O, OCF 3, H, H, H, O], [AE326; OEt, H, O, SCH 2 F, H, H, H, O], [ AE327; OEt, H, O, SCHF 2, H, H, H, O], [AE328; OEt, H, O, SCF 3, H, H, H, O], [AE329; OEt, H, O, CN, H, H, H, O], [AE330; OEt, H, O, NO 2, H, H, H, O], [AE331; CN, H, O, H, H, H, H, O ], [AE 332; CN, H, O, F, H, H, O], [AE 333; CN, H, O, Cl, H, H, H, O], [AE 334; CN, H, O] , Br, H, H, H, O], [AE 335; CN, H, O, I, H, H, H, O], [AE 336; CN, H, O, Me, H, H, H, O], [AE 337; CN, H, O, Et, H, H, H, O] , [AE 338; CN, H, O, Pr, H, H, H, O], [AE 339; CN, H, O, i-Pr, H, H, H, O], [AE 340; _{O, CH = CH 2, H} , H, H, O], [AE341; CN, H, O, C (Me) = CH 2, H, H, H, O], [AE342; CN, H, O , C≡CH, H, H, H, O, [AE 343; CN, H, O, C≡ CMe, H, H, H, O], [AE 344; CN, H, O, c-Pr, H , H, H, O], [AE 345; CN, H, O, OMe, H, H, H, O], [AE 346; CN, H, O, OE t, H, H, H, O], [AE 347 CN, H, O, Oi-Pr, H, H, H, O], [AE 348; CN, H, O, SMe, H, H, H, O], [AE 349; CN, H, O, SEt , H, H, H, O ], [AE350; CN, H, O, CH 2 F, H, H, H, O], [AE351; CN, H, O, CHF 2, H, H, H, O], [AE352; CN, H, O, CF 3, H, H, H, O], [AE353; CN, H, O, OCH 2 F, H, H, H, O], [AE354; CN _{, H, O, OCHF 2,} H, H, H, O], [AE355; CN, H, O, OCF 3, H, H, H, O], [AE356; CN, H, O, SCH 2 F , H, H, H, O], [AE 357; CN, H, O, SCHF ₂ , H, H, H, O], [AE 358; CN, H, O, SCF ₃ , H, H, H, O ], [AE 359; CN, H, O, CN, H, H, H, O], [AE 360; CN, H, O, NO ₂ , H, H, H, O], [AE 361; H, Me, O, H, H, H, H, O, [AE 362; H, Me, O, F, H, H, H, O], [AE 363; H, Me, O, Cl, H, H, H, H, H O, [AE 364; H, Me, O, Br, H, H, O], [AE 365; H, Me, O, I, H, H, H, O], [AE 366; H, Me, O, Me, H, H, H, O, [AE 367; H, Me, O, Et, H, H, H, O], [AE 368; H, Me, O, Pr, H, H, H, H, O], [AE369; H, Me, O, i-Pr, H, H, H, O], [AE370; H, Me, O, CH = CH 2, H, H, H, O], [AE371; H, Me, O, C (Me) = CH 2, H, H, H, O], [AE372; H, Me, O, C≡CH, H, H, H, O] , [AE 373; H, Me, O, C≡CMe, H, H, H, O], [AE 374; H, Me, O, c-Pr, H, H, H, O], [AE 375; H, Me, O, OMe, H, H, H, O], [AE 376; H, Me, O, OEt, H, H, H, O], [AE 377; H, Me, O, Oi-Pr, H, H, H, O], [AE 378; H, Me, O, SMe, H, H, H, O], [AE 379; H, Me, O, SE t, H, H, H, O], [AE 380; _{H, Me, O, CH 2} F, H, H, H, O], [AE381; H, Me, O, CHF 2, H, H, H, O], [AE382; H, Me, O, CF ₃ , H, H, H, O], [AE 383; H, Me, O, OCH ₂ F, H, H, H, O], [AE 384; H, Me, O, OCHF ₂ , H, H, H , O], [AE385; H , Me, O, OCF 3, H, H, H, O], [AE386; H, Me, O, SCH 2 F, H, H, H, O], [AE387; _{H, Me, O, SCHF 2} , H, H, H, O], [AE388; H, Me, O, SCF 3, H, H, H, O], [AE389; H, Me, O, CN, H, H, H, O] , [AE390; H, Me, O, NO 2, H, H, H, O], [AE391; H, Et, O, H, H, H, H, O], [AE 392; H, Et, O, F, H, H, H, O], [AE 393; H, Et, O, Cl, H, H, H, O], [AE 394; H, Et, O, Br , H, H, H, O], [AE 395; H, Et, O, I, H, H, H, O], [AE 396; H, Et, O, Me, H, H, H, O], [AE 397; H, Et, O, Et, H, H, H, O], [AE 398; H, Et, O, Pr, H, H, H, O], [AE 399; H, Et, O, i -Pr, H, H, H, O], [AE400; H, Et, O, CH = CH 2, H, H, H, O],

[AE 401; H, Et, O, C (Me) = CH ₂ , H, H, H, O], [AE 402; H, Et, O, C≡CH, H, H, H, O], [AE 403 H, Et, O, C≡CMe, H, H, H, O], [AE 404; H, Et, O, c-Pr, H, H, H, O], [AE 405; H, Et, O , OMe, H, H, H, O], [AE 406; H, Et, O, OEt, H, H, H, O], [AE 407; H, Et, O, Oi-Pr, H, H, H H, Et, O, SMe, H, H, H, O], [AE 409; H, Et, O, SEt, H, H, H, O], [AE 410; H, Et] _{, O, CH 2 F, H} , H, H, O], [AE411; H, Et, O, CHF 2, H, H, H, O], [AE412; H, Et, O, CF 3, H , H, H, O], [AE413; H, Et, O, OCH 2 F, H, H, H, O], [AE414; H, Et, O, OCHF 2, H, H, H, O] , [AE415; H, Et, O, OCF 3, H, H, H, O], [AE416; H, Et, O, SCH 2 F, H, H, H, O], [AE417; H, Et , O, SCHF ₂ , H, H, H, O], [AE 418; H, Et, O, SCF ₃ , H, H, H, O], [AE 419; H, Et, O, CN, H, H , H, O], [AE 420; H, Et, O, NO ₂ , H, H, O], [AE 421; H, F, O, H, H, H, H, O], [AE 422; H, F, O, F, H, H, H, O], [AE 423; H, F, O, Cl, H, H, H, O], [AE 424; H, F, O, Br, H, H, H, O], [AE 425; H, F, O, I, H, H, H, O], [AE 426; H, F, O, Me, H, H, H, O], [AE 427; H, F, O, Et, H, H, H, O], [AE 428; H, F, O, Pr, H, H, H, O], [AE 429; H, F, O, i-Pr, H, H, H, O] , [AE430; H, F, O, CH = CH 2, H, H, H, O], [AE431; H, F, O, C (Me) = CH 2, H , H, H, O], [AE 432; H, F, O, C≡CH, H, H, H, O], [AE 433; H, F, O, C≡ C Me, H, H, H, O H, F, O, c-Pr, H, H, H, O], [AE 435; H, F, O, OMe, H, H, H, O], [AE 436; H, F] , O, OEt, H, H, H, O], [AE 437; H, F, O, Oi-Pr, H, H, H, O], [AE 438; H, F, O, SMe, H, H , H, O], [AE 439; H, F, O, SE t, H, H, H, O], [AE 440; H, F, O, CH ₂ F, H, H, H, O], [AE 441 ; H, F, O, CHF 2, H, H, H, O], [AE442; H, F, O, CF 3, H, H, H, O], [AE443; H, F, O, OCH ₂ F, H, H, H, O], [AE 444; H, F, O, OCHF ₂ , H, H, H, O], [AE 445; H, F, O, OCF ₃ , H, H, H , O], [AE 446; H, F, O, SCH ₂ F, H, H, H, O], [AE 447; H, F, O, SCHF ₂ , H, H, H, O], [AE 448; H, F, O, SCF ₃ , H, H, H, O], [AE 449; H, F, O, CN, H, H, H, O], [AE 450; H, F, O, NO ₂ , H, H, H, O], [AE 451; H, Cl, O, H, H, H, H, O], [AE 452; H, Cl, O, F, H, H, H, O], [[ H, Cl, O, Cl, H, H, H, O], [AE 454; H, Cl, O, Br, H, H, H, O], [AE 455; H, Cl, O, I, H, H, H, O], [AE 456; H, Cl, O, Me, H, H, H, O], [AE 457; H, Cl, O, Et, H, H, H, O], [ AE 458; H, Cl, O, Pr, H, H, H, O], [AE 459; H, Cl, O, i-Pr, H, H, H, O], [AE 460; H, Cl, O, _{CH = CH 2, H, H} , H, O], [AE461; H, Cl, O, C (Me) = CH 2, H, H, H, O], [AE462; H, Cl, O, C ≡CH, H, H, H, O], [AE 463; H, Cl, O, C≡CMe, H, H, H, O], [AE 464; H, Cl, O, c-Pr, H, H , H, O], [AE 465; H, Cl, O, OMe, H, H, H, O], [AE 466; H, Cl, O, OEt, H, H, H, O], [AE 467; H , Cl, O, Oi-Pr, H, H, H, O, [AE 468; H, Cl, O, SMe, H, H, H, O], [AE 469; H, Cl, O, SEt, H , H, H, O], [AE470; H, Cl, O, CH 2 F, H, H, H, O], [AE471; H, Cl, O, CHF 2, H, H, H, O] , [ AE472; H, Cl, O, CF 3, H, H, H, O], [AE473; H, Cl, O, OCH 2 F, H, H, H, O], [AE474; H, Cl, O _{, OCHF 2, H, H,} H, O], [AE475; H, Cl, O, OCF 3, H, H, H, O], [AE476; H, Cl, O, SCH 2 F, H, H , H, O], [AE 477; H, Cl, O, SCHF ₂ , H, H, H, O], [AE 478; H, Cl, O, SCF ₃ , H, H, H, O], [AE 479 H, Cl, O, CN, H, H, H, H, O], [AE 480; H, Cl, O, NO ₂ , H, H, H, O], [AE 481; H, Br, O, H, O H, H, H, O], [AE 482; H, Br, O, F, H, H, H, O], [AE 483; H, Br, O, Cl, H, H, H, O], [[ AE 484; H, Br, O, Br, H, H, H, O], [AE 485; H, Br, O, I, H, H, H, O], [AE 486; H, Br, O, Me, H, H, H, O], [AE 487; H, Br, O, Et, H, H, H, O], [AE 488; H, Br, O, Pr, H, H, H, O], [A AE489; H, Br, O, i-Pr, H, H, H, O], [AE490; H, Br, O, CH = CH 2, H, H, H, O], [AE491; H, Br , O, C (Me) = CH ₂ , H, H, H, O], [AE 492; H, Br, O, C≡CH, H, H, H, O], [AE 493; H, Br, O , C≡CMe, H, H, H, O], [AE 494; H, Br, O, c-Pr, H, H, H, O], [AE 495; H, Br, O, OMe, H, H H, O], [AE 496; H, Br, O, OEt, H, H, H, O], [AE 497; H, Br, O, Oi-Pr, H, H, H, O], [AE 498] H, Br, O, SMe, H, H, H, O, [AE 499; H, Br, O, SEt, H, H, H, O], [AE 500; H, Br, O, CH ₂ F , H, H, H, O],

[AE501; H, Br, O , CHF 2, H, H, H, O], [AE502; H, Br, O, CF 3, H, H, H, O], [AE503; H, Br, O OCH ₂ F, H, H, H, H, O], [AE 504; H, Br, O, OCHF ₂ , H, H, H, O], [AE 505; H, Br, O, OCF ₃ , H, H , H, O], [AE 506; H, Br, O, SCH ₂ F, H, H, H, O], [AE 507; H, Br, O, SCHF ₂ , H, H, H, O], [[ AE508; H, Br, O, SCF 3, H, H, H, O], [AE509; H, Br, O, CN, H, H, H, O], [AE510; H, Br, O, NO ₂ , H, H, H, O], [AE 511; H, I, O, H, H, H, H, O], [AE 512; H, I, O, F, H, H, H, O] H, I, O, Cl, H, H, H, O], [AE 514; H, I, O, Br, H, H, H, O], [AE 515; H, I, O, I, H, H, H, O], [AE 516; H, I, O, Me, H, H, H, O], [AE 517; H, I, O, Et, H, H, H, O] [AE 518; H, I, O, Pr, H, H, H, O], [AE 519: H, I, O, i-Pr, H, H, H, O], [AE 520; H, I, I, _{O, CH = CH 2, H} , H, H, O], [AE521; H, I, O, C (Me) = CH 2, H, H, H, O], [AE522; H, I, O , CICH, H, H, H, O, [AE 523; H, I, O, C≡ CMe, H, H, H, O], [AE 524; H, I, O, c-Pr, H , H, H, O], [AE 525; H, I, O, OMe, H, H, H, O], [AE 526; H, I, O, OE t, H, H, H, O], [AE 527 H, I, O, Oi-Pr, H, H, H, O], [AE 528; H, I, O, SMe, H, H, H, O], [AE 529; H, I, O, SE t H, H, H, O], [AE 530; H, I, O, CH ₂ F, H, H, H, O], [AE 531; H, I, O, CHF ₂ , H, H, H, H, O, [AE 532; H, I, O, CF ₃ , H, H, H, O], [AE 533; H, I, O, OCH ₂ F, H, H, O], [AE 534; H _{, I, O, OCHF 2,} H, H, H, O], [AE535; H, I, O, OCF 3, H, H, H, O], [AE536; H, I, O, SCH 2 F , H, H, H, O], [AE 537; H, I, O, SCHF ₂ , H, H, H, O], [AE 538; H, I, O, SCF ₃ , H, H, H, O H, I, O, CN, H, H, H, O], [AE 540; H, I, O, NO ₂ , H, H, H, O], [AE 541; H, CHF _2] , O, H, H, H , H, O], [AE542; H, CHF 2, O, F, H, H, H, O], [AE543; H, CHF 2, O, Cl, H, H , H, O], [AE544 ; H, CHF 2, O, Br, H, H, H, O], [AE545; H, CHF 2, O, I, H, H, H, O], [AE546 _{; H, CHF 2, O,} Me, H, H, H, O], [AE547; H, CHF 2, O, Et, H, H, H, O], [AE548; H, CHF 2, O, Pr, H, H, H, O], [AE 549; H, CHF ₂ , O, i-Pr, H, H, H, O], [AE 550; H, CHF ₂ , O, CH 2CH ₂ , H , H, H, O], [AE 551; H, CHF ₂ , O, C (Me) = CH ₂ , H, H, H, O], [AE 552; H, CHF ₂ , O, CHCH, H , H, H, O], [AE553; H, CHF 2, O, C≡CMe, H, H, H, O], [AE554; H, CHF 2, O, c-Pr, H, H, H , O], [AE 555; H, CHF ₂ , O, OMe, H, H, H, O], [AE 556; H, CHF ₂ , O, OE t, H, H, H, O], [AE 557; H _{, CHF 2, O, Oi-} Pr, H, H, H, O], [AE558; H, CHF 2, O, SMe, H, H, H, O], [AE559; H, CHF 2, O, SEt, H, H, H, O], [AE560; H, CHF 2, O, CH 2 F, H, H, H, O], [AE561; H, CHF 2, O, CHF 2, H, H H, O], [AE 562; H, CHF ₂ , O, CF ₃ , H, H, O], [AE 563; H, CHF ₂ , O, OCH ₂ F, H, H, H, O] _{, [AE564; H, CHF 2} , O, OCHF 2, H, H, H, O], [AE565; H, CHF 2, O, OCF 3, H, H, H, O], [AE566; H, CHF ₂ , O, SCH ₂ F, H, H, H, O], [AE 567; H, CHF ₂ , O, SCHF ₂ , H, H, H, O], [[ _{AE568; H, CHF 2, O} , SCF 3, H, H, H, O], [AE569; H, CHF 2, O, CN, H, H, H, O], [AE570; H, CHF 2, _{O, NO 2, H, H} , H, O], [AE571; H, CF 3, O, H, H, H, H, O], [AE572; H, CF 3, O, F, H, H , H, O], [AE573 ; H, CF 3, O, Cl, H, H, H, O], [AE574; H, CF 3, O, Br, H, H, H, O], [AE575 _{; H, CF 3, O,} I, H, H, H, O], [AE576; H, CF 3, O, Me, H, H, H, O], [AE577; H, CF 3, O, Et, H, H, H, O], [AE 578; H, CF ₃ , O, Pr, H, H, H, O], [AE 579; H, CF ₃ , O, i-Pr, H, H, H, H, O], [AE580; H, CF 3, O, CH = CH 2, H, H, H, O], [AE581; H, CF 3, O, C (Me) = CH 2, H, H , H, O], [AE 582; H, CF ₃ , O, C≡CH, H, H, H, O], [AE 583; H, CF ₃ , O, C, C Me, H, H, H, O ], [AE584; H, CF 3, O, c-Pr, H, H, H, O], [AE585; H, CF 3, O, OMe, H, H, H, O], [AE586; H , CF ₃ , O, OEt, H, H, H, O, [AE 587; H, CF ₃ , O, Oi-Pr, H, H, H, O], [AE 588; H, CF ₃ , O, SMe, H, H, H, O], [AE 589; H, CF ₃ , O, SE t, H, H, H, O], [AE 590; H, CF ₃ , O, CH ₂ F, H, H, H, O], [AE591; H, CF 3, O, CHF 2, H, H, H, O], [AE592; H, CF 3, O, CF 3, H, H, H, O], [ _{AE593; H, CF 3, O} , OCH 2 F, H, H, H, O], [AE594; H, CF 3, O, OCHF 2, H, H, H, O], [AE595; H, CF _{3, O, OCF 3, H} , H, H, O], [AE596; H, CF 3, O, SCH 2 F, H, H, H, O], [AE597; H, CF 3, O, SCHF ₂ , H, H, H, O], [AE 598; H, CF ₃ , O, SCF ₃ , H, H, H, O], [AE 599; H, CF ₃ , O, CN, H , H, H, O], [AE 600; H, CF ₃ , O, NO ₂ , H, H, H, O],

[AE601; H, OMe, O, H, H, H, H, O], [AE 602; H, OMe, O, F, H, H, H, O], [AE 603; H, OMe, O, Cl , H, H, H, O], [AE 604; H, OMe, O, Br, H, H, H, O], [AE 605; H, OMe, O, I, H, H, H, O], [AE606; H, OMe, O, Me, H, H, H, O], [AE 607; H, OMe, O, Et, H, H, H, O], [AE 608; H, OMe, O, Pr , H, H, H, O ], [AE609; H, OMe, O, i-Pr, H, H, H, O], [AE610; H, OMe, O, CH = CH 2, H, H, H, O], [AE611; H, OMe, O, C (Me) = CH 2, H, H, H, O], [AE612; H, OMe, O, C≡CH, H, H, H, O], [AE 613; H, OMe, O, C≡CMe, H, H, H, O], [AE 614; H, OMe, O, c-Pr, H, H, H, O], [AE 615; H, OMe, O, OMe, H, H, H, O, [AE 616; H, OMe, O, OEt, H, H, H, O], [AE 617; H, OMe, O, Oi-Pr, H, H, H, O], [AE 618; H, OMe, O, SMe, H, H, H, O], [AE 619; H, OMe, O, SE t, H, H, H, O], [ AE620; H, OMe, O, CH 2 F, H, H, H, O], [AE621; H, OMe, O, CHF 2, H, H, H, O], [AE622; H, OMe, O , CF ₃ , H, H, H, O], [AE 623; H, OMe, O, OCH ₂ F, H, H, H, O], [AE 624; H, OMe, O, OCHF ₂ , H, H , H, O], [AE625 ; H, OMe, O, OCF 3, H, H, H, O], [AE626; H, OMe, O, SCH 2 F, H, H, H, O], [ AE 627; H, OMe, O, SCHF ₂ , H, H, H, O], [AE 628; H, OMe, O, SCF ₃ , H, H, H, O], [AE 629; H, OMe, O, CN, H, H, H, O], [AE 630; H, OMe, O, NO ₂ , H, H, H, O], [AE 631; H, OEt, O, H, H, H, H, O H, OEt, O, F, H, H, H, O], [AE 633; H, OEt, O, Cl, H, H, H, O], [AE 634; H, OEt, O] , Br, H, H, H, O], [AE 635; H, O Et, O, I, H, H, H, O], [AE 636; H, OEt, O, Me, H, H, H, O], [AE 637; H, OEt, O, Et, H, H, H, O], [AE 638; H, OEt, O, Pr, H, H, H, O], [AE 639; H, OE t, O, i-Pr, H, H, H, O], [AE 640; H, OEt, O, CH = CH 2, H, H, H, O], [AE641; H, OEt, O, C (Me) = CH 2, H, H, H, O], [AE642; H , OEt, O, C≡CH, H, H, H, O], [AE643; H, OEt, O, C≡ CMe, H, H, H, O], [AE 644; H, OEt, O, c -Pr, H, H, H, O], [AE645; H, OEt, O, OMe, H, H, H, O], [AE 646; H, OEt, O, OEt, H, H, H, O] H, OEt, O, Oi-Pr, H, H, H, O], [AE 648; H, OEt, O, SMe, H, H, H, O], [AE 649; H, OEt] , O, SEt, H, H , H, O], [AE650; H, OEt, O, CH 2 F, H, H, H, O], [AE651; H, OEt, O, CHF 2, H, H, H, O], [ AE652; H, OEt, O, CF 3, H, H, H, O], [AE653; H, OEt, O, OCH 2 F, H, H, H, O], [AE654; H, OEt, O , OCHF 2, H, H, H, O], [AE655; H, OEt, O, OCF 3, H, H, H, O], [AE656; H, OEt, O , SCH ₂ F, H, H, H, O], [AE 657; H, OEt, O, SCHF ₂ , H, H, H, O], [AE 658; H, OE t, O, SCF ₃ , H, H H, O], [AE 659; H, OEt, O, CN, H, H, H, O], [AE 660; H, OEt, O, NO ₂ , H, H, H, O], [AE 661; H, CN, O, H, H, H, H, H, O], [AE 662; H, CN, O, F, H, H, H, O], [AE 663; H, CN, O, Cl, H, H, H, O], [AE664; H, CN, O, Br, H, H, O], [AE665; H, CN, O, I, H, H, H, O], [AE 666; H, CN, O, Me, H, H, H, O, [AE 667; H, CN, O, Et, H, H, H, O], [AE 668; H, CN, O, Pr, H, H, H, O], [AE 669; H, CN, O, i-Pr, H, H, H, O] , [AE670; H, CN, O, CH = CH 2, H, H, H, O], [AE671; H, CN, O, C (Me) = CH 2, H, H, H, O], [AE 672; H, CN, O, C≡CH, H, H, H, O], [AE 673; H, CN, O, C≡ C Me, H, H, H, O], [AE 674; H, CN , O, c-Pr, H, H, H, O], [AE 675; H, CN, O, OMe, H, H, H, O], [AE 676; H, CN, O, OE t, H, H , H, O], [AE 677; H, CN, O, Oi-Pr, H, H, H, O], [AE 678; H, CN, O, SMe, H, H, H, O], [AE 679 H, CN, O, SEt, H, H, H, O], [AE 680; H, CN, O, CH ₂ F, H, H, H, O], [AE 681; H, CN, O, CHF _{2, H, H, H,} O], [AE682; H, CN, O, CF 3, H, H, H, O], [AE683; H, CN, O, OCH 2 F, H, H, H , O], [AE684; H , CN, O, OCHF 2, H, H, H, O], [AE685; H, CN, O, OCF 3, H, H, H, O], [AE686; H , CN, O, SCH ₂ F, H, H, H, O], [AE 687; H, CN, O, SCHF ₂ , H, H, H, O], [AE 688; H, CN, O, SCF ₃ H, H, H, O], [AE 689; H, CN, O, CN, H, H, H, O], [AE 690; H, CN, O, NO ₂ , H, H, H, O] , [AE 691; Me, Me, O, H, H, H, H, O], [AE 692; Me, Me, O, F, H, H, H, O], [AE 693; Me, Me, O, Cl, H, H, H, O], [AE 694; Me, Me, O, Br, H, H, H, O], [AE 695; Me, Me, O, I, H, H, H, O] [AE 696; Me, Me, O, Me, H, H, H, O], [AE 697; Me, Me, O, Et, H, H, H, O], [AE 698; Me, Me, O, Pr, H, H, H, O], [AE699; Me, Me, O, i-Pr, H, H, H, O], [AE700; Me, Me, O, CH = CH 2, H, H , H, O],

[AE 701; Me, Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 702; Me, Me, O, C≡CH, H, H, H, O], [AE 703 Me, Me, O, C≡CMe, H, H, H, O], [AE704; Me, Me, O, c-Pr, H, H, H, O], [AE 705; Me, Me, O , OMe, H, H, H, O], [AE 706; Me, Me, O, OEt, H, H, H, O], [AE 707; Me, Me, O, Oi-Pr, H, H, H , O], [AE 708; Me, Me, O, SMe, H, H, H, O], [AE 709; Me, Me, O, SE t, H, H, H, O], [AE 710; Me, Me _{, O, CH 2 F, H} , H, H, O], [AE711; Me, Me, O, CHF 2, H, H, H, O], [AE712; Me, Me, O, CF 3, H , H, H, O], [AE 713; Me, Me, O, OCH ₂ F, H, H, H, O], [AE 714; Me, Me, O, OCHF ₂ , H, H, H, O] , [AE715; Me, Me, O, OCF 3, H, H, H, O], [AE716; Me, Me, O, SCH 2 F, H, H, H, O], [AE717; Me, Me , O, SCHF ₂ , H, H, H, O], [AE 718; Me, Me, O, SCF ₃ , H, H, H, O], [AE 719; Me, Me, O, CN, H, H , H, O], [AE 720; Me, Me, O, NO ₂ , H, H, O], [AE 721; Et, Me, O, H, H, H, H, O], [AE 722; Et, Me, O, F, H, H, H, O, [AE 723; Et, Me, O, Cl, H, H, H, O], [AE 724; Et, Me, O, Br, H, H, H, O], [AE 725; Et, Me, O, I, H, H, H, O], [AE 726; Et, Me, O, Me, H, H, H, O], [AE 727; Et, Me, O, Et, H, H, H, H, O], [AE 728; Et, Me, O, Pr, H, H, H, O], [AE 729; Et, Me, O, i-Pr, H, H, H, O] , [AE730; Et, Me, O, CH = CH 2, H, H, H, O], [AE731; Et, Me, O, C (Me) = CH 2, H , H, H, O], [AE 732; Et, Me, O, C≡CH, H, H, H, O], [AE 733; Et, Me, O, C≡ C Me, H, H, H, O ], [AE 734; Et, Me, O, c- Pr, H, H, H, O], [AE 735; Et, Me, O, OMe, H, H, H, O], [AE 736; Et, Me, O, OEt, H, H, H, O] [AE 737; Et, Me, O, Oi-Pr, H, H, H, O], [AE 738; Et, Me, O, SMe, H, H, H, O], [AE 739; Et, Me, O, SEt, H, H, H, O], [AE740; Et, Me, O, CH 2 F, H, H, H, O], [AE741; Et, Me, O, CHF 2, H, H , H, O], [AE742 ; Et, Me, O, CF 3, H, H, H, O], [AE743; Et, Me, O, OCH 2 F, H, H, H, O], [ AE744; Et, Me, O, OCHF 2, H, H, H, O], [AE745; Et, Me, O, OCF 3, H, H, H, O], [AE746; Et, Me, O, SCH ₂ F, H, H, H, O], [AE 747; Et, Me, O, SCHF ₂ , H, H, H, O], [AE 748; Et, Me, O, SCF ₃ , H, H, H, O], [AE 749; Et, Me, O, CN, H, H, H, O], [AE 750; Et, Me, O, NO ₂ , H, H, H, O], [AE 751; F , Me, O, H, H, H, H, H, O], [AE 752; F, Me, O, F, H, H, H, O], [AE 753; F, Me, O, Cl, H, H] , H, O], [AE 754; F, Me, O, Br, H, H, O], [AE 755; F, Me, O, I, H, H, H, O], [AE 756; F , Me, O, Me, H, H, H, O, [AE757; F, Me, O, Et, H, H, H, O], [AE758; F, Me, O, Pr, H, H , H, O], [AE759 ; F, Me, O, i-Pr, H, H, H, O], [AE760; F, Me, O, CH = CH 2, H, H, H, O] , [AE 761; F, Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 762; F, Me, O, C≡CH, H, H, H, O], [[ AE 763; F, Me, O, C≡CMe, H, H, H, O], [AE764; F, Me, O, c-Pr, H, H, H, O], [AE 765; F, Me, O, OMe, H, H, H, O], [AE766; F, Me, O, OEt, H, H, H, O], [AE 767; F, Me, O, Oi-Pr, H, H, H, O], [AE 768; F, Me, O, SMe, H, H, H, O], [AE 769; F , Me, O, SEt, H , H, H, O], [AE770; F, Me, O, CH 2 F, H, H, H, O], [AE771; F, Me, O, CHF 2, H, H, H, O] , [AE772; F, Me, O, CF 3, H, H, H, O], [AE773; F, Me, O, OCH 2 F, H, H, H, O ], [AE774; F, Me , O, OCHF 2, H, H, H, O], [AE775; F, Me, O, OCF 3, H, H, H, O], [AE776; F, Me , O, SCH ₂ F, H, H, H, O], [AE 777; F, Me, O, SCHF ₂ , H, H, H, O], [AE 778; F, Me, O, SCF ₃ , H , H, H, O], [AE 779; F, Me, O, CN, H, H, H, O], [AE 780; F, Me, O, NO ₂ , H, H, H, O], [[ AE 781; Cl, Me, O, H, H, H, H, O], [AE 782; Cl, Me, O, F, H, H, H, O], [AE 783; Cl, Me, O, Cl, H, H, H, O], [AE 784; Cl, Me, O, Br, H, H, H, O], [AE 785; Cl, Me, O, I, H, H, H, O], [A AE 786; Cl, Me, O, Me, H, H, H, O], [AE 787; Cl, Me, O, Et, H, H, H, O], [AE 788; Cl, Me, O, Pr, H, H, H, O] , [AE789; Cl, Me, O, i-Pr, H, H, H, O], [AE790; Cl, Me, O, CH = CH 2, H, H, H , O], [AE 791; Cl, Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 792; Cl, Me, O, C≡CH, H, H, H, O ], [AE 793; Cl, Me, O, C≡CMe, H, H, H, O], [AE 794; Cl, Me, O, c-Pr, H, H, H, O], [AE 795; Cl , Me, O, OMe, H, H, H, O], [AE796; Cl, Me, O, OEt, H, H, H, O], [AE 797; Cl, Me, O, Oi-Pr, H , H, H, O], [AE 798; Cl, Me, O, SMe, H, H, H, O], [AE 799; Cl, Me, O, SE t, H, H, H, O], [AE 800] Cl, Me, O, CH ₂ F, H, H, H, O],

[AE801; Cl, Me, O , CHF 2, H, H, H, O], [AE802; Cl, Me, O, CF 3, H, H, H, O], [AE803; Cl, Me, O OCH ₂ F, H, H, H, O, [AE 804; Cl, Me, O, OCHF ₂ , H, H, H, O], [AE 805; Cl, Me, O, OCF ₃ , H, H , H, O], [AE 806; Cl, Me, O, SCH ₂ F, H, H, H, O], [AE 807; Cl, Me, O, SCHF ₂ , H, H, H, O], [[ AE808; Cl, Me, O, SCF 3, H, H, H, O], [AE809; Cl, Me, O, CN, H, H, H, O], [AE810; Cl, Me, O, NO ₂ , H, H, H, O], [AE 811; Br, Me, O, H, H, H, H, O], [AE 812; Br, Me, O, F, H, H, H, O] [AE813; Br, Me, O, Cl, H, H, H, O], [AE 814; Br, Me, O, Br, H, H, H, O], [AE 815; Br, Me, O, I, H, H, H, O], [AE 816; Br, Me, O, Me, H, H, H, O], [AE 817; Br, Me, O, Et, H, H, H, O] , [AE 818; Br, Me, O, Pr, H, H, H, O], [AE 819; Br, Me, O, i-Pr, H, H, H, O], [AE 820; Br, Me, _{O, CH = CH 2, H} , H, H, O], [AE821; Br, Me, O, C (Me) = CH 2, H, H, H, O], [AE822; Br, Me, O , CMeCH, H, H, H, O, [AE 823; Br, Me, O, C≡ CMe, H, H, H, O], [AE 824; Br, Me, O, c-Pr, H , H, H, O], [AE 825; Br, Me, O, OMe, H, H, H, O], [AE 826; Br, Me, O, OE t, H, H, H, O], [AE 827 Br, Me, O, Oi-Pr, H, H, H, O], [AE 828; Br, Me, O, SMe, H, H, H, O], [AE 829; Br, Me, O, SEt , H, H, H, O ], [AE830; Br, Me, O, CH 2 F, H, H, H, O], [AE831; Br, Me, O, CHF 2, H, H, H, O], [AE 832; Br, Me, O, CF ₃ , H, H, H, O], [AE 833; Br, Me, O, OCH ₂ F, H, H, H, O], [AE 834; Br , Me, O, OCHF ₂ , H, H, H, O] , [AE835; Br, Me, O, OCF 3, H, H, H, O], [AE836; Br, Me, O, SCH 2 F, H, H, H, O ], [AE837; Br, Me , O, SCHF 2, H, H, H, O], [AE838; Br, Me, O, SCF 3, H, H, H, O], [AE839; Br, Me , O, CN, H, H , H, O], [AE840; Br, Me, O, NO 2, H, H, H, O], [AE841; I, Me, O, H, H, H, H, O], [AE 842; I, Me, O, F, H, H, H, O], [AE 843; I, Me, O, Cl, H, H, H, O], [AE 844; Me, O, Br, H, H, H, O, [AE 845; I, Me, O, I, H, H, H, O], [AE 846; I, Me, O, Me, H, H, H, H, O], [AE 847; I, Me, O, Et, H, H, H, O], [AE 848; I, Me, O, Pr, H, H, H, O], [AE 849; Me, O, i-Pr, H, H, H, O], [AE850; I, Me, O, CH = CH 2, H, H, H, O], [AE851; I, Me, O, C _{(Me) = CH 2, H} , H, H, O], [AE852; I, Me, O, C≡CH, H, H, H, O], [AE853; I, Me, O, C≡CMe , H, H, H, O], [AE 854; I, Me, O, c-Pr, H, H, H, O], [AE 855; I, Me, O, OMe, H, H, H, O ], [AE 856; I, Me, O, OEt, H, H, H, O], [AE 857; I, Me, O, Oi-Pr, H, H, H, O], [AE 858; , O, SMe, H, H, H, O], [AE 859; I, Me, O, SEt, H, H, H, O], [AE 860; I, Me, O, CH ₂ F, H, H , H, O], [AE 861; I, Me, O, CHF ₂ , H, H, H, O], [AE 862; I, Me, O, CF ₃ , H, H, H, O], [AE 863 ; I, Me, O, OCH 2 F, H, H, H, O], [AE864; I, Me, O, OCHF 2, H, H, H, O], [AE865; I, Me, O, _{OCF 3, H, H, H} , O], [AE866; I, Me, O, SCH 2 F, H, H, H, O], [AE867; I, Me, O, SCHF 2, H, H, H, O], [AE 868; I, Me, O, SCF ₃ , H, H, H, O], [AE 869; I, Me, O, CN, H, H, H, O], [AE870; I, Me, O, NO 2, H, H, H, O], [AE871; CHF 2, Me, O, H, H, H, H, O], [ AE872; CHF 2, Me, O, F, H, H, H, O], [AE873; CHF 2, Me, O, Cl, H, H, H, O], [ _{AE874; CHF 2, Me, O} , Br, H, H, H, O], [AE875; CHF 2, Me, O, I, H, H, H, O], [AE876; CHF 2, Me, O , Me, H, H, H, O], [AE 877; CHF ₂ , Me, O, Et, H, H, H, O], [AE 878; CHF ₂ , Me, O, Pr, H, H, H , O], [AE879; CHF 2, Me, O, i-Pr, H, H, H, O], [AE880; CHF 2, Me, O, CH = CH 2, H, H, H, O] [AE 881; CHF ₂ , Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 882; CHF ₂ , Me, O, C≡CH, H, H, H, O] _{, [AE883; CHF 2, Me} , O, C≡CMe, H, H, H, O], [AE884; CHF 2, Me, O, c-Pr, H, H, H, O], [AE885; _{CHF 2, Me, O, OMe} , H, H, H, O], [AE886; CHF 2, Me, O, OEt, H, H, H, O], [AE887; CHF 2, Me, O, Oi -Pr, H, H, H, O], [AE888; CHF 2, Me, O, SMe, H, H, H, O], [AE889; CHF 2, Me, O, SEt, H, H, H , O], [AE890; CHF 2, Me, O, CH 2 F, H, H, H, O], [AE891; CHF 2, Me, O, CHF 2, H, H, H, O], [ AE 892; CHF ₂ , Me, O, CF ₃ , H, H, H, O], [AE 893; CHF ₂ , Me, O, OCH ₂ F, H, H, H, O], [AE 894; CHF ₂ , _{Me, O, OCHF 2, H} , H, H, O], [AE895; CHF 2, Me, O, OCF 3, H, H, H, O], [AE896; CHF 2, Me, O, SCH 2 F, H, H, H, O], [AE897; CHF 2, Me, O, SCHF 2, H, H, H, O], [AE898; CHF 2, Me, O, SCF 3, H, H, H, O], [AE 899; CHF ₂ , M e, O, CN, H, H, H, O], [AE900; CHF 2, Me, O, NO 2, H, H, H, O],

_{[AE901; CF 3, Me,} O, H, H, H, H, O], [AE902; CF 3, Me, O, F, H, H, H, O], [AE903; CF 3, Me, O, Cl, H, H, H, O, [AE 904; CF ₃ , Me, O, Br, H, H, H, O], [AE 905; CF ₃ , Me, O, I, H, H, H, H, O], [AE906; CF 3, Me, O, Me, H, H, H, O], [AE907; CF 3, Me, O, Et, H, H, H, O], [AE908; _{CF 3, Me, O, Pr} , H, H, H, O], [AE909; CF 3, Me, O, i-Pr, H, H, H, O], [AE910; CF 3, Me, O , CH = CH ₂ , H, H, H, O, [AE 911; CF ₃ , Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 912; CF ₃ , Me, O, C≡CH, H, H, H, H, O], [AE 913; CF ₃ , Me, O, C≡ CMe, H, H, H, O], [AE 914; CF ₃ , Me, O, c- Pr, H, H, H, O], [AE915; CF 3, Me, O, OMe, H, H, H, O], [AE916; CF 3, Me, O, OEt, H, H, H, _{O], [AE917; CF 3} , Me, O, Oi-Pr, H, H, H, O], [AE918; CF 3, Me, O, SMe, H, H, H, O], [AE919; _{CF 3, Me, O, SEt} , H, H, H, O], [AE920; CF 3, Me, O, CH 2 F, H, H, H, O], [AE921; CF 3, Me, O _{, CHF 2, H, H,} H, O], [AE922; CF 3, Me, O, CF 3, H, H, H, O], [AE923; CF 3, Me, O, OCH 2 F, H , H, H, O], [AE924; CF 3, Me, O, OCHF 2, H, H, H, O], [AE925; CF 3, Me, O, OCF 3, H, H, H, O _{], [AE926; CF 3,} Me, O, SCH 2 F, H, H, H, O], [AE927; CF 3, Me, O, SCHF 2, H, H, H, O], [AE928; _{CF 3, Me, O, SCF} 3, H, H, H, O], [AE929; CF 3, Me, O, CN, H, H, H, O], [AE930; CF 3, Me, O, NO ₂ , H, H, H, O], [AE 931; OMe, Me, O, H, H, H, H, O] [AE932; OMe, Me, O, F, H, H, H, O], [AE933; OMe, Me, O, Cl, H, H, H, O], [AE934; OMe, Me, O, Br, H, H, H, O], [AE 935; OMe, Me, O, I, H, H, H, O], [AE 936; OMe, Me, O, Me, H, H, H, O] [AE 937; OMe, Me, O, Et, H, H, H] O], [AE 938; OMe, Me, O, Pr, H, H, H, O], [AE 939; OMe, Me, O, i-Pr, H, H, H, O], [AE940; OMe, Me, O, CH = CH 2, H, H, H, O], [AE941; OMe, Me, O, C (Me) = CH ₂ , H, H, H, H, O], [AE942; OMe, Me, O, C≡CH, H, H, H, O], [AE943; OMe, Me, O, C≡ C Me, H, H , H, O], [AE 944; OMe, Me, O, c-Pr, H, H, H, O], [AE 945; OMe, Me, O, OMe, H, H, H, O], [AE 946 OMe, Me, O, OEt, H, H, H, O], [AE 947; OMe, Me, O, Oi-Pr, H, H, H, O], [AE 948; OMe, Me, O, SMe , H, H, H, O ], [AE949; OMe, Me, O, SEt, H, H, H, O], [AE950; OMe, Me, O, CH 2 F, H, H, H, O ], [AE 951; OMe, Me, O, CHF ₂ , H, H, H, O], [AE 952; OMe, Me, O, CF ₃ , H, H, H, O], [AE 953; OMe, Me , O, OCH ₂ F, H, H, H, O, [AE 954; OMe, Me, O, OCHF ₂ , H, H, H, O], [AE 955; OMe, Me, O, OCF ₃ , H , H, H, O], [AE 956; OMe, Me, O, SCH ₂ F, H, H, H, O], [AE 957; OMe, Me, O, SCHF ₂ , H, H, H, O] [AE 958; OMe, Me, O, SCF ₃ , H, H, H, O], [AE 959; OMe, Me, O, CN, H, H, H, O], [AE 960: OMe, Me, O , NO ₂ , H, H, H, O], [AE 961; OEt, Me, O, H, H, H, H, O], [AE 962; OEt, Me, O, F, H, H, H, H, O], [AE963; OEt, Me, O, Cl, H, H, H, O], [AE964; OEt, Me, O, Br, H, H, H, O], [A E965; OEt, Me, O, I, H, H, H, O], [AE 966; OEt, Me, O, Me, H, H, H, O], [AE 967; OEt, Me, O, Et, H, H, H, O], [AE968; OEt, Me, O, Pr, H, H, H, O], [AE 969; OEt, Me, O, i-Pr, H, H, H, O] , [AE970; OEt, Me, O, CH = CH 2, H, H, H, O], [AE971; OEt, Me, O, C (Me) = CH 2, H, H, H, O], [AE972; OEt, Me, O, C≡CH, H, H, H, O], [AE 973; OEt, Me, O, C≡CMe, H, H, H, O], [AE974; OEt, Me , O, c-Pr, H, H, H, O], [AE975; OEt, Me, O, OMe, H, H, H, O], [AE976; OEt, Me, O, OEt, H, H] , H, O], [AE977; OEt, Me, O, Oi-Pr, H, H, H, O], [AE978; OEt, Me, O, SMe, H, H, H, O], [AE979 ; OEt, Me, O, SEt , H, H, H, O], [AE980; OEt, Me, O, CH 2 F, H, H, H, O], [AE981; OEt, Me, O, CHF ₂ , H, H, H, O], [AE 982; OEt, Me, O, CF ₃ , H, H, H, O], [AE 983; OE t, Me, O, OCH ₂ F, H, H, H , O], [AE984; OEt , Me, O, OCHF 2, H, H, H, O], [AE985; OEt, Me, O, OCF 3, H, H, H, O], [AE986; OEt , Me, O, SCH ₂ F, H, H, H, O, [AE987; OEt, Me, O, SCHF ₂ , H, H, H, O], [AE 988; OEt, Me, O, SCF ₃ H, H, H, O], [AE 989; OEt, Me, O, CN, H, H, H, O], [AE 990; OEt, Me, O, NO ₂ , H, H, H, O] [AE 991; CN, Me, O, H, H, H, H, O], [AE 992; CN, Me, O, F, H, H, H, O], [AE 993; CN, Me, O, Cl, H, H, H, O], [AE 994; CN, Me, O, Br, H, H, H, O], [AE 995; CN, Me, O, I, H, H, H, O] [AE 996; CN, Me, O, Me, H, H, H, O], [AE 997; CN, Me, O, Et, H, H, H, O], [AE 998; CN, Me , O, Pr, H, H, H, O, [AE 999; CN, Me, O, i-Pr, H, H, H, O], [AE 1000; CN, Me, O, CH = CH ₂ , H, H, H, O],

[AE1001; CN, Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 1002; CN, Me, O, C≡CH, H, H, H, O], [AE 1003 CN, Me, O, C≡CMe, H, H, H, O], [AE 1004; CN, Me, O, c-Pr, H, H, H, O], [AE 1005; CN, Me, O , OMe, H, H, H, O], [AE 1006; CN, Me, O, OEt, H, H, H, O], [AE 1007; CN, Me, O, Oi-Pr, H, H, H , O], [AE 1008; CN, Me, O, SMe, H, H, H, O], [AE 1009; CN, Me, O, SE t, H, H, H, O], [AE 1010, CN, Me _{, O, CH 2 F, H} , H, H, O], [AE1011; CN, Me, O, CHF 2, H, H, H, O], [AE1012; CN, Me, O, CF 3, H , H, H, O], [AE1013; CN, Me, O, OCH 2 F, H, H, H, O], [AE1014; CN, Me, O, OCHF 2, H, H, H, O] , [AE1015; CN, Me, O, OCF 3, H, H, H, O], [AE1016; CN, Me, O, SCH 2 F, H, H, H, O], [AE1017; CN, Me , O, SCHF ₂ , H, H, H, O], [AE 1018; CN, Me, O, SCF ₃ , H, H, H, O], [AE 10 19; CN, Me, O, CN, H, H , H, O], [AE 1020; CN, Me, O, NO ₂ , H, H, O], [AE 1021; Me, Me, O, H, H, H, H, O], [AE 1022; Me, Me, O, F, H, H, H, O], [AE 1023; Me, Me, O, Cl, H, H, H, O], [AE 1024; Me, Me, O, Br, H, H, H, O], [AE 1025; Me, Me, O, I, H, H, H, O], [AE 1026; Me, Me, O, Me, H, H, H, O], [AE 1027; Me, Me, O, Et, H, H, H, O], [AE 1028; Me, Me, O, Pr, H, H, H, O], [AE 1029; Me, Me, O, i-Pr, H, H, H, O] , [AE1030; Me, Me, O, CH = CH 2, H, H, H, O], [AE1031; Me, Me, O, C (Me) = CH 2, H , H, H, O], [AE 1032; Me, Me, O, C≡CH, H, H, H, O], [AE 1033; Me, Me, O, C ≡CMe, H, H, H, O], [AE 1034; Me, Me, O, c-Pr, H, H, H, O], [AE 1035; Me, Me, O, OMe, H, H, H , O], [AE 1036; Me, Me, O, OEt, H, H, H, O], [AE 1037; Me, Me, O, Oi-Pr, H, H, H, O], [AE 1038; Me , Me, O, SMe, H, H, H, O, [AE 1039; Me, Me, O, SE t, H, H, H, O], [AE 1040; Me, Me, O, CH ₂ F, H , H, H, O], [AE1041; Me, Me, O, CHF 2, H, H, H, O], [AE1042; Me, Me, O, CF 3, H, H, H, O], [AE1043; Me, Me, O , OCH 2 F, H, H, H, O], [AE1044; Me, Me, O, OCHF 2, H, H, H, O], [AE1045; Me, Me, _{O, OCF 3, H, H} , H, O], [AE1046; Me, Me, O, SCH 2 F, H, H, H, O], [AE1047; Me, Me, O, SCHF 2, H, H, H, O], [ AE1048; Me, Me, O, SCF 3, H, H, H, O], [AE1049; Me, Me, O, CN, H, H, H, O], [AE1050 ; Me, Me, O, NO 2, H, H, H, O], [AE1051; Me, Et, O, H, H, H, H, O], [AE1052; Me, Et, O, F, H, H, H, O], [AE 1053; Me, Et, O, Cl, H, H, H, O], [AE 1054; Me, Et, O, Br, H, H, H, O], [ AE 1055; Me, Et, O, I, H, H, H, O], [AE 1056; Me, Et, O, Me, H, H, H, O], [AE 1057; Me, Et, O, Et, H, H, H, O], [AE 1058; Me, Et, O, Pr, H, H, H, O], [AE 1059; Me, Et, O, i-Pr, H, H, H, O] , [AE1060; Me, Et, O, CH = CH 2, H, H, H, O], [AE1061; Me, Et, O, C (Me) = CH 2, H, H, H, O], [AE1062; Me, Et, O, C≡CH, H, H, H, O], [AE1063; Me, Et, O, C≡CMe, H, H, H, O], [AE 1064; Me, Et , O, c-Pr, H, H, H, O], [AE 1065; Me, Et, O, OMe, H, H, H, O], [AE 1066; Me, Et, O, OEt, H, H, H, O, [AE 1067; Me, Et, O, Oi-Pr, H, H, H, O], [AE 1068; Me, Et, O, SMe, H, H, H, O], [AE 1069; Me, Et, O, SE t, H, H, H, O], [AE 1070; Me, Et, O, CH ₂ F, H, H, H, O], [ AE1071; Me, Et, O, CHF 2, H, H, H, O], [AE1072; Me, Et, O, CF 3, H, H, H, O], [AE1073; Me, Et, O, _{OCH 2 F, H, H,} H, O], [AE1074; Me, Et, O, OCHF 2, H, H, H, O], [AE1075; Me, Et, O, OCF 3, H, H, H, O], [AE 1076; Me, Et, O, SCH ₂ F, H, H, H, O], [AE 1077; Me, Et, O, SCHF ₂ , H, H, H, O], [AE 10 78 ; Me, Et, O, SCF 3, H, H, H, O], [AE1079; Me, Et, O, CN, H, H, H, O], [AE1080; Me, Et, O, NO 2 , H, H, H, O], [AE 1081; Me, F, O, H, H, H, H, O], [AE 1082; Me, F, O, F, H, H, H, O], [AE1083; Me, F, O, Cl, H, H, H, O], [AE1084; Me, F, O, Br, H, H, H, O], [AE1085; Me, F, O, I , H, H, H, O], [AE 1086; Me, F, O, Me, H, H, H, O], [AE 1087; Me, F, O, Et, H, H, H, O], [AE 10 88; Me, F, O, Pr, H, H, H, O], [AE 1089; Me, F, O, i-Pr, H, H, H, O], [AE 1090; Me, F, O _{, CH = CH 2, H,} H, H, O], [AE1091; Me, F, O, C (Me) = CH 2, H, H, H, O], [AE1092; Me, F, O, C≡CH, H, H, H, O], [AE1093; Me, F, O, C≡CMe, H, H, H, O], [AE1094; Me, F, O, c-Pr, H, H, H, O], [AE 1095; Me, F, O, OMe, H, H, H, O], [AE 1096; Me, F, O, OE t, H, H, H, O], [AE 1097; Me, F, O, Oi-Pr, H, H, H, O], [AE1098; Me, F, O, SMe, H, H, H, O], [AE 1099; Me, F, O, SEt, H, H, H, O ], [AE 1100; Me, F, O, CH ₂ F, H, H, H, O],

[AE1101; Me, F, O , CHF 2, H, H, H, O], [AE1102; Me, F, O, CF 3, H, H, H, O], [AE1103; Me, F, O OCH ₂ F, H, H, H, H, O], [AE 1 104; Me, F, O, OCHF ₂ , H, H, H, O], [AE 1 105; Me, F, O, OCF ₃ , H, H , H, O], [AE 1106; Me, F, O, SCH ₂ F, H, H, H, O], [AE 1 107; Me, F, O, SCHF ₂ , H, H, H, O], [[ AE 1108; Me, F, O, SCF ₃ , H, H, H, O], [AE 1 109; Me, F, O, CN, H, H, H, O], [AE 1110; Me, F, O, NO ₂ , H, H, H, O], [AE 1111; Me, Cl, O, H, H, H, H, O], [AE 1112; Me, Cl, O, F, H, H, H, O] , [AE1113; Me, Cl, O, Cl, H, H, H, O], [AE 1114; Me, Cl, O, Br, H, H, H, O], [AE 1115; Me, Cl, O, I, H, H, H, O], [AE 1 116; Me, Cl, O, Me, H, H, H, O], [AE 1 117; Me, Cl, O, Et, H, H, H, O] , [AE1118; Me, Cl, O, Pr, H, H, H, O], [AE 1119; Me, Cl, O, i-Pr, H, H, H, O], [AE 1120; _{O, CH = CH 2, H} , H, H, O], [AE1121; Me, Cl, O, C (Me) = CH 2, H, H, H, O], [AE1122; Me, Cl, O , C≡CH, H, H, H, O, [AE 1 123; Me, Cl, O, C≡CMe, H, H, H, O], [AE 1 124; Me, Cl, O, c-Pr, H , H, H, O], [AE 1 125; Me, Cl, O, OMe, H, H, H, O], [AE 1 126; Me, Cl, O, OE t, H, H, H, O], [AE 1 127 Me, Cl, O, Oi-Pr, H, H, H, O], [AE 1 128; Me, Cl, O, SMe, H, H, H, O], [AE 1 129; Me, Cl, O, SEt H, H, H, O], [AE 1130; Me, Cl, O, CH ₂ F, H, H, H, O], [AE 1131; Me, Cl, O, CHF ₂ , H, H, H, O], [AE 1132; Me, Cl, O, CF ₃ , H, H, H, O], [AE 1 133; Me, Cl, O, OCH ₂ F, H, H, H, O], [AE1134; Me, Cl, O , OCHF 2, H, H, H, O], [AE1135; Me, Cl, O, OCF 3, H, H, H, O], [AE1136; Me, Cl, O , SCH ₂ F, H, H, H, O], [AE 1137; Me, Cl, O, SCHF ₂ , H, H, H, O], [AE 1138; Me, Cl, O, SCF ₃ , H, H , H, O], [AE 1 139; Me, Cl, O, CN, H, H, H, O], [AE 1 140; Me, Cl, O, NO ₂ , H, H, H, O], [AE 1141; Me, Br, O, H, H, H, H, H, O], [AE1142; Me, Br, O, F, H, H, H, O], [AE1143; Me, Br, O, Cl, H, H, H, O], [AE 1 144; Me, Br, O, Br, H, H, H, O], [AE 1 145; Me, Br, O, I, H, H, H, O], [AE 1146; Me, Br, O, Me, H, H, H, H, O], [AE 1147; Me, Br, O, Et, H, H, H, O], [AE 1148; Me, Br, O, Pr, H, H, H, O], [ AE1149; Me, Br, O, i-Pr, H, H, H, O], [AE1150; Me, Br, O, CH = CH 2, H, H, H, O ], [AE1151; Me, Br , O, C (Me) = CH 2, H, H, H, O], [AE1152; Me, Br, O, C≡CH, H, H, H, O], [AE1153; Me, Br, O, C≡CMe, H, H, H, O], [AE 1154; Me, Br, O, c-Pr, H, H, H, O], [AE 1 155; Me, Br , O, OMe, H, H, H, O, [AE 1156; Me, Br, O, OEt, H, H, H, O], [AE 1 157; Me, Br, O, Oi-Pr, H, H , H, O], [AE 1158; Me, Br, O, SMe, H, H, H, O], [AE 1159; Me, Br, O, SE t, H, H, H, O], [AE 1 160; Me _{, Br, O, CH 2 F} , H, H, H, O], [AE1161; Me, Br, O, CHF 2, H, H, H, O], [AE1162; Me, Br, O, CF 3 , H, H, H, O ], [AE1163; Me, Br, O, OCH 2 F, H, H, H, O], [AE1164; Me, Br, O, OCHF 2, H, H, H, O], [AE 1165; Me, Br, O, OCF ₃ , H, H, H, O], [AE 1166; Me, Br, O, SCH ₂ F, H, H, H, O], [AE 1167; Me, Br, O, SCHF ₂ , H, H, H, O], [AE 1 168; Me, Br, O, SCF ₃ , H, H, H, O, [AE 1169; Me, Br, O, CN, H, H, H, O], [AE 1170; Me, Br, O, NO ₂ , H, H, H, O], [AE 1171; Me, I , O, H, H, H, H, O, [AE1172; Me, I, O, F, H, H, H, O], [AE1173; Me, I, O, Cl, H, H, H , O], [AE 1 174; Me, I, O, Br, H, H, H, O], [AE 1175; Me, I, O, I, H, H, H, O], [AE 1176; Me, I , O, Me, H, H, H, O, [AE 1177; Me, I, O, Et, H, H, H, O], [AE 1178; Me, I, O, Pr, H, H, H , O], [AE 1179; Me, I, O, i-Pr, H, H, H, O], [AE 1 180; Me, I, O, CH = CH ₂ , H, H, H, O], [, AE1181; Me, I, O, C (Me) = CH 2, H, H, H, O], [AE1182; Me, I, O, C≡CH, H, H, H, O], [AE1183; Me, I, O, C≡CMe, H, H, H, O], [AE 1184; Me, I, O, c-Pr, H, H, H, O], [AE 1 185; Me, I, O, OMe, H, H, H, O], [AE 1186; Me, I, O, OEt, H, H, H, O], [AE 1187; Me, I, O, Oi-Pr, H, H, H, O, [AE1188; Me, I, O, SMe, H, H, H, O], [AE 1189; Me, I, O, SEt, H, H, H, O], [AE 1190; Me, I, I _{O, CH 2 F, H,} H, H, O], [AE1191; Me, I, O, CHF 2, H, H, H, O], [AE1192; Me, I, O, CF 3, H, H, H, O], [ AE1193; Me, I, O, OCH 2 F, H, H, H, O], [AE1194; Me, I, O, OCHF 2, H, H, H, O], [AE 1195; Me, I, O, OCF ₃ , H, H, H, O], [AE 1196; Me, I, O, SCH ₂ F, H, H, H, O], [AE 1197; Me, I, _{O, SCHF 2, H, H} , H, O], [AE1198; Me, I, O, SCF 3, H, H, H, O], [AE1199; Me, I, O, CN, H, H, H, O], [AE 1200; Me , I, O, NO ₂ , H, H, H, O],

_{[AE1201; Me, CHF 2,} O, H, H, H, H, O], [AE1202; Me, CHF 2, O, F, H, H, H, O], [AE1203; Me, CHF 2, O, Cl, H, H, H, O], [AE1204; Me, CHF 2, O, Br, H, H, H, O], [AE1205; Me, CHF 2, O, I, H, H, H, O], [AE 1206; Me, CHF ₂ , O, Me, H, H, H, O], [AE 1207; Me, CHF ₂ , O, Et, H, H, H, O], [AE 1 208; _{Me, CHF 2, O, Pr} , H, H, H, O], [AE1209; Me, CHF 2, O, i-Pr, H, H, H, O], [AE1210; Me, CHF 2, O , CH = CH ₂ , H, H, H, O, [AE 1211; Me, CHF ₂ , O, C (Me) = CH ₂ , H, H, H, O], [AE 1212; Me, CHF ₂ , O, C≡CH, H, H, H, H, O], [AE 1213; Me, CHF ₂ , O, C≡ CMe, H, H, H, O], [AE 1214; Me, CHF ₂ , O, c − Pr, H, H, H, O], [AE1215; Me, CHF 2, O, OMe, H, H, H, O], [AE1216; Me, CHF 2, O, OEt, H, H, H, O], [AE1217; Me, CHF 2, O, Oi-Pr, H, H, H, O], [AE1218; Me, CHF 2, O, SMe, H, H, H, O], [AE1219; _{Me, CHF 2, O, SEt} , H, H, H, O], [AE1220; Me, CHF 2, O, CH 2 F, H, H, H, O], [AE1221; Me, CHF 2, O _{, CHF 2, H, H,} H, O], [AE1222; Me, CHF 2, O, CF 3, H, H, H, O], [AE1223; Me, CHF 2, O, OCH 2 F, H , H, H, O], [AE1224; Me, CHF 2, O, OCHF 2, H, H, H, O], [AE1225; Me, CHF 2, O, OCF 3, H, H, H, O ], [AE1226; Me, CHF 2, O, SCH 2 F, H, H, H, O], [AE1227; Me, CHF 2, O, SCHF 2, H, H, H, O], [AE1228; _{Me, CHF 2, O, SCF} 3, H, H, H, O], [AE1229; Me, CHF 2, O, CN, H, H, H, O], [ _{AE1230; Me, CHF 2, O} , NO 2, H, H, H, O], [AE1231; Me, CF 3, O, H, H, H, H, O], [AE1232; Me, CF 3, O, F, H, H, H, O], [AE1233; Me, CF 3, O, Cl, H, H, H, O], [AE1234; Me, CF 3, O, Br, H, H, H, O], [AE1235; Me, CF 3, O, I, H, H, H, O], [AE1236; Me, CF 3, O, Me, H, H, H, O], [AE1237; _{Me, CF 3, O, Et} , H, H, H, O], [AE1238; Me, CF 3, O, Pr, H, H, H, O], [AE1239; Me, CF 3, O, i -Pr, H, H, H, O], [AE 1240; Me, CF ₃ , O, CH = CH ₂ , H, H, H, O], [AE 1241; Me, CF ₃ , O, C (Me) = CH ₂ , H, H, H, O], [AE 1242; Me, CF ₃ , O, C≡CH, H, H, H, O], [AE 1243; Me, CF ₃ , O, C≡ CMe, H, H, H, O] , [AE1244; Me, CF 3, O, c-Pr, H, H, H, O], [AE1245; Me, CF 3, O, OMe, H, H, H, O], [AE1246; Me, CF 3, O, OEt, H, H, H, O], [AE1247; Me, CF 3, O, Oi-Pr, H, H, H, O], [AE1248; _{Me, CF 3, O, SMe} , H, H, H, O], [AE1249; Me, CF 3, O, SEt, H, H, H, O], [AE1250; Me, CF 3, O, CH ₂ F, H, H, H, O], [AE 1251; Me, CF ₃ , O, CHF ₂ , H, H, H, O], [AE 1252; Me, CF ₃ , O, CF ₃ , H, H , H, O], [AE1253 ; Me, CF 3, O, OCH 2 F, H, H, H, O], [AE1254; Me, CF 3, O, OCHF 2, H, H, H, O] _{, [AE1255; Me, CF 3} , O, OCF 3, H, H, H, O], [AE1256; Me, CF 3, O, SCH 2 F, H, H, H, O], [AE1257; Me , CF ₃ , O, SCHF ₂ , H, H, H, O, [AE 1258; Me, CF ₃ , O, SCF ₃ , H, H, H, O], [AE 1259; Me, CF ₃ , O, CN, H, H, H , O], [AE1260; Me , CF 3, O, NO 2, H, H, H, O], [AE1261; Me, OMe, O, H, H, H, H, O], [AE1262; Me , OMe, O, F, H, H, H, O], [AE 1263; Me, OMe, O, Cl, H, H, H, O], [AE 1264; Me, OMe, O, Br, H, H , H, O], [AE 1 265; Me, OMe, O, I, H, H, H, O], [AE 1266; Me, OMe, O, Me, H, H, H, O], [AE 1267; Me , OMe, O, Et, H, H, H, O, [AE 1268; Me, OMe, O, Pr, H, H, H, O], [AE 1269; Me, OMe, O, i-Pr, H , H, H, O], [AE 1 270; Me, OMe, O, CH = CH ₂ , H, H, H, O], [AE 1271; Me, OMe, O, C (Me) = CH ₂ , H, H, H, O], [AE 1272; Me, OMe, O, C≡CH, H, H, H, O], [AE 1273; Me, OMe, O, C≡ CMe, H, H, H, O] , [AE1274; Me, OMe, O, c-Pr, H, H, H, O], [AE 1275; Me, OMe, O, OMe, H, H, H, O], [AE 1276; Me, OMe, O, OEt, H, H, H, O, [AE 1277; Me, OMe, O, Oi-Pr, H, H, H, O], [AE 1278; Me, OMe, O, SMe, H, H, H, H, O], [AE 1279; Me, OMe, O, SEt, H, H, H, O], [AE 1280; Me, OMe, O, CH ₂ F, H, H, H, O], [AE 1281; _{Me, OMe, O, CHF 2} , H, H, H, O], [AE1282; Me, OMe, O, CF 3, H, H, H, O], [AE1283; Me, OMe, O, OCH 2 F, H, H, H, O], [AE1284; Me, OMe, O, OCHF 2, H, H, H, O], [AE1285; Me, OMe, O, OCF 3, H, H, H, O], [AE 1286; Me, OMe, O, SCH ₂ F, H, H, H, O], [AE 1287; Me, OMe, O, SCHF ₂ , H, H, H, O], [AE 1 288; Me , OMe, O, SCF ₃ , H, H, H, O], [AE 1 289; Me, OMe, O, CN, H, H, H, O], [AE 1290; Me, OMe, O, NO ₂ , H , H, H, O], [AE 1291; Me, OEt, O, H H, H, H, O], [AE1292; Me, OEt, O, F, H, H, H, O], [AE 1293; Me, OEt, O, Cl, H, H, H, O], [AE1294; Me, OEt, O, Br, H, H, H, O], [AE 1295; Me, OEt, O, I, H, H, H, O], [AE 1296; Me, OEt, O, Me, H, H, H, O], [AE 1297; Me, OEt, O, Et, H, H, H, O], [AE 1298; Me, OE t, O, Pr, H, H, H, O], [AE1299; Me, OEt, O , i-Pr, H, H, H, O], [AE1300; Me, OEt, O, CH = CH 2, H, H, H, O],

[AE1301; Me, OEt, O , C (Me) = CH 2, H, H, H, O], [AE1302; Me, OEt, O, C≡CH, H, H, H, O], [AE1303 Me, OEt, O, C≡CMe, H, H, H, O], [AE 1304; Me, OEt, O, c-Pr, H, H, H, O], [AE 1 305; Me, OEt, O , OMe, H, H, H, O], [AE 1306; Me, OEt, O, OEt, H, H, H, O], [AE 1307; Me, OEt, O, Oi-Pr, H, H, H , O], [AE1308; Me, OEt, O, SMe, H, H, H, O], [AE 1309; Me, OEt, O, SEt, H, H, H, O], [AE 1310; Me, OEt _{, O, CH 2 F, H} , H, H, O], [AE1311; Me, OEt, O, CHF 2, H, H, H, O], [AE1312; Me, OEt, O, CF 3, H , H, H, O], [AE 1313; Me, OEt, O, OCH ₂ F, H, H, H, O], [AE 1314; Me, OE t, O, OCHF ₂ , H, H, H, O] , [AE1315; Me, OEt, O, OCF 3, H, H, H, O], [AE1316; Me, OEt, O, SCH 2 F, H, H, H, O], [AE1317; Me, OEt , O, SCHF ₂ , H, H, H, O], [AE 1318; Me, OEt, O, SCF ₃ , H, H, H, O], [AE 1319; Me, OE t, O, CN, H, H , H, O], [AE 1320; Me, OEt, O, NO ₂ , H, H, O], [AE 1321; Me, CN, O, H, H, H, H, O], [AE 1322; Me, CN, O, F, H, H, H, O], [AE1323; Me, CN, O, Cl, H, H, H, O], [AE 1324; Me, CN, O, Br, H, H, H, O], [AE 1325; Me, CN, O, I, H, H, H, O], [AE 1326; Me, CN, O, Me, H, H, H, O], [AE 1327; Me, CN, O, Et, H, H, H, O], [AE1328; Me, CN, O, Pr, H, H, H, O], [AE 1329; Me, CN, O, i-Pr, H, H, H, O] , [AE1330; Me, CN, O, CH = CH 2, H, H, H, O], [AE1331; Me, CN, O, C (Me) = CH 2, H , H, H, O], [AE1332; Me, CN, O, C≡CH, H, H, H, O], [AE1333; Me, CN, O, C≡CMe, H, H, H, O], [AE 1334; Me, CN, O, c-Pr, H, H, H, O], [AE 1335; Me, CN, O, OMe, H, H, H, O], [AE 1336; Me, CN, O, OEt, H, H, H, O], [AE 1337; Me, CN, O, Oi-Pr, H, H, H, O], [AE 1 338; Me, CN, O, SMe, H, H, H, O], [AE 1339; Me, CN, O, SE t, H, H, H, O], [ AE1340; Me, CN, O, CH 2 F, H, H, H, O], [AE1341; Me, CN, O, CHF 2, H, H, H, O], [AE1342; Me, CN, O _{, CF 3, H, H,} H, O], [AE1343; Me, CN, O, OCH 2 F, H, H, H, O], [AE1344; Me, CN, O, OCHF 2, H, H , H, O], [AE 1345; Me, CN, O, OCF ₃ , H, H, O], [AE 1346; Me, CN, O, SCH ₂ F, H, H, H, O], [ AE 1347; Me, CN, O, SCHF ₂ , H, H, H, O], [AE 1348; Me, CN, O, SCF ₃ , H, H, H, O], [AE 1 349; Me, CN, O, CN, H, H, H, O], [AE 1350; Me, CN, O, NO ₂ , H, H, H, O], [AE 1351; Me, F, O, H, H, H, H, O ], [AE1352; Me, F, O, F, H, H, H, O], [AE1353; Me, F, O, Cl, H, H, H, O], [AE 1354; Me, F, O] , Br, H, H, H, O], [AE 1 355; Me, F, O, I, H, H, H, O], [AE 1356; Me, F, O, Me, H, H, H, O Me, F, O, Et, H, H, H, O], [AE 1358; Me, F, O, Pr, H, H, H, O], [AE 1359; Me, F, O] , i-Pr, H, H, H, O], [AE 1 360; Me, F, O, CH = CH ₂ , H, H, H, O], [AE 1361; Me, F, O, C (Me) = CH ₂ , H, H, H, O], [AE 1362; Me, F, O, C≡CH, H, H, H, O], [AE 1363; Me, F, O, C≡ C Me, H, H, H, O], [AE 1364; Me, F, O, c-Pr, H, H, H, O], [AE 1 365; Me, F, O, OMe, H, H, H, O], [ AE 136 6; Me, F, O, OEt, H, H, H, O], [AE 1367; Me, F, O, Oi-Pr, H, H, H, O], [AE 1 368; Me, F, O, SMe, H, H, H, O], [AE 1369; Me, F, O, SEt, H, H, H, O], [AE 1370; Me, F, O, CH ₂ F, H, H, H, O], [AE1371; Me, F, O, CHF 2, H, H, H, O], [AE1372; Me, F, O, CF 3, H, H, H, O], [AE1373; Me, _{F, O, OCH 2 F,} H, H, H, O], [AE1374; Me, F, O, OCHF 2, H, H, H, O], [AE1375; Me, F, O, OCF 3, H, H, H, O], [AE 1376; Me, F, O, SCH ₂ F, H, H, H, O], [AE 1377; Me, F, O, SCHF ₂ , H, H, H, O Me, F, O, SCF ₃ , H, H, H, O], [AE 1379; Me, F, O, CN, H, H, H, O], [AE 1 380; Me, F, _{O, NO 2, H, H} , H, O], [AE1381; Et, F, O, H, H, H, H, O], [AE1382; Et, F, O, F, H, H, H , O], [AE1383; Et, F, O, Cl, H, H, H, O], [AE 1384; Et, F, O, Br, H, H, H, O], [AE 1385; Et, F , O, I, H, H, H, O], [AE 1 386; Et, F, O, Me, H, H, H, O], [AE 1387; Et, F, O, Et, H, H, H , O], [AE1388; Et, F, O, Pr, H, H, H, O], [AE 1389; Et, F, O, i-Pr, H, H, H, O], [AE 1390; Et , F, O, CH = CH 2, H, H, H, O], [AE1391; Et, F, O, C (Me) = CH 2, H, H, H, O], [AE1392; Et, F, O, C≡CH, H, H, H, H, O], [AE1393; Et, F, O, C≡ CMe, H, H, H, O], [AE 1394; Et, F, O, c- Pr, H, H, H, O], [AE 1395; Et, F, O, OMe, H, H, H, O], [AE 1396; Et, F, O, OEt, H, H, H, O] [AE 1397; Et, F, O, Oi-Pr, H, H, H, O], [AE 1398; Et, F, O, SMe, H, H, H, O], [AE 1399; Et, F, O, SEt, H, H, H, O], [AE1400; _{Et, F, O, CH 2} F, H, H, H, O],

[AE1401; Et, F, O , CHF 2, H, H, H, O], [AE1402; Et, F, O, CF 3, H, H, H, O], [AE1403; Et, F, O , OCH ₂ F, H, H, H, O], [AE 1404; Et, F, O, OCHF ₂ , H, H, H, O], [AE 1 405; Et, F, O, OCF ₃ , H, H , H, O], [AE 1406; Et, F, O, SCH ₂ F, H, H, H, O], [AE 1407; Et, F, O, SCHF ₂ , H, H, H, O], [[ AE1408; Et, F, O, SCF 3, H, H, H, O], [AE1409; Et, F, O, CN, H, H, H, O], [AE1410; Et, F, O, NO ₂ , H, H, H, O], [AE 1411; F, F, O, H, H, H, H, O], [AE 1412; F, F, O, F, H, H, H, O] [AE 1413; F, F, O, Cl, H, H, H, O], [AE 1414; F, F, O, Br, H, H, O], [AE 1415; F, F, O, I, H, H, H, O], [AE 1416; F, F, O, Me, H, H, H, O], [AE 1417; F, F, O, Et, H, H, H, O] [AE 1418; F, F, O, Pr, H, H, H, O], [AE 1419; F, F, O, i-Pr, H, H, H, O], [AE 1420; F, F, _{O, CH = CH 2, H} , H, H, O], [AE1421; F, F, O, C (Me) = CH 2, H, H, H, O], [AE1422; F, F, O , C≡CH, H, H, H, O], [AE 1423; F, F, O, C≡ CMe, H, H, H, O], [AE 1424; F, F, O, c-Pr, H , H, H, O], [AE 1425; F, F, O, OMe, H, H, H, O], [AE 1426; F, F, O, OE t, H, H, H, O], [AE 1427 F, F, O, Oi-Pr, H, H, H, O], [AE1428; F, F, O, SMe, H, H, H, O], [AE 1429; F, F, O, SEt , H, H, H, O], [AE 1430; F, F, O, CH ₂ F, H, H, H, O], [AE 1431; F, F, O, CHF ₂ , H, H, H, O], [AE1432; F, F, O, CF 3, H, H, H, O], [AE1433; F, F, O, OCH 2 F, H, H, H, O], [AE1434; F , F, O, OCHF ₂ , H, H, H, O], [AE 1435; F, F, O, O _{CF 3, H, H, H} , O], [AE1436; F, F, O, SCH 2 F, H, H, H, O], [AE1437; F, F, O, SCHF 2, H, H, H, O], [AE1438; F, F, O, SCF 3, H, H, H, O], [AE1439; F, F, O, CN, H, H, H, O], [AE1440; F _{, F, O, NO 2,} H, H, H, O], [AE1441; Cl, F, O, H, H, H, H, O], [AE1442; Cl, F, O, F, H, H, H, O], [AE 1443; Cl, F, O, Cl, H, H, H, O], [AE 1444; Cl, F, O, Br, H, H, H, O], [AE 1445; Cl, F, O, I, H, H, H, O], [AE 1446; Cl, F, O, Me, H, H, H, O], [AE 1447; Cl, F, O, Et, H, H, H, O], [AE 1448; Cl, F, O, Pr, H, H, H, O], [AE 1449; Cl, F, O, i-Pr, H, H, H, O], [ AE 1450; Cl, F, O, CH = CH ₂ , H, H, H, O], [AE 1451; Cl, F, O, C (Me) = CH ₂ , H, H, H, O], [AE 1452 Cl, F, O, C≡CH, H, H, H, O], [AE 1453; Cl, F, O, C≡ CMe, H, H, H, O], [AE 1454; Cl, F, O , c-Pr, H, H, H, O], [AE 1455; Cl, F, O, OMe, H, H, H, O], [AE 1456; Cl, F, O, OEt, H, H, H , O], [AE 1457; Cl, F, O, Oi-Pr, H, H, H, O], [AE 1458; Cl, F, O, SMe, H, H, H, O], [AE 1459; Cl , F, O, SEt, H, H, H, O, [AE 1460; Cl, F, O, CH ₂ F, H, H, H, O], [AE 1461; Cl, F, O, CHF ₂ , H, H, H, O] , [AE1462; Cl, F, O, CF 3, H, H, H, O], [AE1463; Cl, F, O, OCH 2 F, H, H, H, O ], [AE 1464; Cl, F, O, OCHF ₂ , H, H, H, O], [AE 1465; Cl, F, O, OCF ₃ , H, H, H, O], [AE 1466; Cl, F , O, SCH ₂ F, H, H, H, O, [AE 1467; Cl, F, O, SCHF ₂ , H, H, H, O], [AE 1468; Cl, F, O, SCF ₃ , H , H, H, O], [AE 1469; Cl, F, O, CN, H, H, H, O, [AE 1470; Cl, F, O, NO ₂ , H, H, H, O], [AE 1471; Br, F, O, H, H, H , H, O], [AE1472; Br, F, O, F, H, H, H, O], [AE 1473; Br, F, O, Cl, H, H, H, O], [AE 1474; Br , F, O, Br, H, H, H, O, [AE 1475; Br, F, O, I, H, H, H, O], [AE 1476; Br, F, O, Me, H, H , H, O], [AE 1477; Br, F, O, Et, H, H, H, O], [AE 1478; Br, F, O, Pr, H, H, H, O], [AE 1479; Br , F, O, i-Pr , H, H, H, O], [AE1480; Br, F, O, CH = CH 2, H, H, H, O], [AE1481; Br, F, O, _{C (Me) = CH 2,} H, H, H, O], [AE1482; Br, F, O, C≡CH, H, H, H, O], [AE1483; Br, F, O, C≡ CMe, H, H, H, O], [AE 1484; Br, F, O, c-Pr, H, H, H, O], [AE 1485; Br, F, O, OMe, H, H, H, O], [AE 1486; Br, F, O, OEt, H, H, H, O], [AE 1487; Br, F, O, Oi-Pr, H, H, H, O], [AE 1 488; Br, F, O, SMe, H, H, H, O, [AE 1489; Br, F, O, SEt, H, H, H, O], [AE 1490; Br, F, O, CH ₂ F, H, H, H, O], [ AE1491; Br, F, O, CHF 2, H, H, H, O], [AE1492; Br, F, O, CF 3, H, H, H, O], [ AE1493; Br, F, O, OCH 2 F, H, H, H, O], [AE1494; Br, F, O, OCHF 2, H, H, H, O], [AE1495; Br, F, O Br, F, O, SCH ₂ F, H, H, H, O], [AE 1497; Br, F, O, SCHF ₂ , H, H], OCF ₃ , H, H, H, O], [AE 1496; , H, O], [AE 1498; Br, F, O, SCF ₃ , H, H, H, O], [AE 1499; Br, F, O, CN, H, H, H, O], [AE 1500; _{br, F, O, NO 2} , H, H, H, O],

[AE 1501; I, F, O, H, H, H, H, O], [AE 1502; I, F, O, F, H, H, H, O], [AE 1503; I, F, O, Cl , H, H, H, O], [AE 1504; I, F, O, Br, H, H, H, O], [AE 1505; I, F, O, I, H, H, H, O], [AE1506; I, F, O, Me, H, H, H, O], [AE 1507; I, F, O, Et, H, H, H, O], [AE 1508; I, F, O, Pr , H, H, H, O ], [AE1509; I, F, O, i-Pr, H, H, H, O], [AE1510; I, F, O, CH = CH 2, H, H, H, O], [AE1511; I, F, O, C (Me) = CH 2, H, H, H, O], [AE1512; I, F, O, C≡CH, H, H, H, O, [AE 1513; I, F, O, C≡CMe, H, H, H, O], [AE 1514; I, F, O, c-Pr, H, H, H, O], [AE 1515; I, F, O, OMe, H, H, H, O], [AE 1516; I, F, O, OEt, H, H, H, O], [AE 1517; I, F, O, Oi-Pr, H, H, H, O], [AE 1518; I, F, O, S Me, H, H, H, O], [AE 1519; I, F, O, SE t, H, H, H, O], [ AE1520; I, F, O, CH 2 F, H, H, H, O], [AE1521; I, F, O, CHF 2, H, H, H, O], [AE1522; I, F, O , CF ₃ , H, H, H, O], [AE 1523; I, F, O, OCH ₂ F, H, H, H, O], [AE 1524; I, F, O, OCHF ₂ , H, H , H, O], [AE1525 ; I, F, O, OCF 3, H, H, H, O], [AE1526; I, F, O, SCH 2 F, H, H, H, O], [ AE 1527; I, F, O, SCHF ₂ , H, H, H, O], [AE 1528; I, F, O, SCF ₃ , H, H, H, O], [AE 1529; I, F, O, CN, H, H, H, O], [AE 1530; I, F, O, NO ₂ , H, H, H, O], [AE 1531; CHF ₂ , F, O, H, H, H, H, H _{O], [AE1532; CHF 2} , F, O, F, H, H, H, O], [AE1533; CHF 2, F, O, Cl, H, H, H, O], [AE1534; CHF 2 , F, O, Br, H, H, H, O], [AE 1535; CHF ₂ , F, O, I, H, H , H, O], [AE1536 ; CHF 2, F, O, Me, H, H, H, O], [AE1537; CHF 2, F, O, Et, H, H, H, O], [AE1538 CHF ₂ , F, O, Pr, H, H, H, O, [AE 1539; CHF ₂ , F, O, i-Pr, H, H, H, O], [AE 1540; CHF ₂ , F, _{O, CH = CH 2, H} , H, H, O], [AE1541; CHF 2, F, O, C (Me) = CH 2, H, H, H, O], [AE1542; CHF 2, F , O, C≡CH, H, H, H, O, [AE 1543; CHF ₂ , F, O, C≡ CMe, H, H, H, O], [AE 1544; CHF ₂ , F, O, c -Pr, H, H, H, O], [AE1545; CHF 2, F, O, OMe, H, H, H, O], [AE1546; CHF 2, F, O, OEt, H, H, H , O], [AE1547; CHF 2, F, O, Oi-Pr, H, H, H, O], [AE1548; CHF 2, F, O, SMe, H, H, H, O], [AE1549 _{; CHF 2, F, O,} SEt, H, H, H, O], [AE1550; CHF 2, F, O, CH 2 F, H, H, H, O], [AE1551; CHF 2, F, _{O, CHF 2, H, H} , H, O], [AE1552; CHF 2, F, O, CF 3, H, H, H, O], [AE1553; CHF 2, F, O, OCH 2 F, H, H, H, O] , [AE1554; CHF 2, F, O, OCHF 2, H, H, H, O], [AE1555; CHF 2, F, O, OCF 3, H, H, H, _{O], [AE1556; CHF 2} , F, O, SCH 2 F, H, H, H, O], [AE1557; CHF 2, F, O, SCHF 2, H, H, H, O], [AE1558 CHF ₂ , F, O, SCF ₃ , H, H, H, O], [AE 1559; CHF ₂ , F, O, CN, H, H, H, O], [AE 1560; CHF ₂ , F, O _{, NO 2, H, H,} H, O], [AE1561; CF 3, F, O, H, H, H, H, O], [AE1562; CF 3, F, O, F, H, H, H, O], [AE 1563; CF ₃ , F, O, Cl, H, H, H, O], [AE 1564; CF ₃ , F, O, Br, H, H, H, O], [AE 1 565; _{CF 3, F, O, I} , H, H, H, O], [AE1566; CF 3, F, O, Me, H, H, H, O], [AE1567; CF 3, F, O, Et, H, H, H, O], [AE1568; _{CF 3, F, O, Pr} , H, H, H, O], [AE1569; CF 3, F, O, i-Pr, H, H, H, O], [AE1570; CF 3, F, O , CH = CH ₂ , H, H, H, O, [AE 1571; CF ₃ , F, O, C (Me) = CH ₂ , H, H, H, O], [AE 1572; CF ₃ , F, O, C≡CH, H, H, H, H, O], [AE 1573; CF ₃ , F, O, C≡ CMe, H, H, H, O], [AE 1574; CF ₃ , F, O, c − Pr, H, H, H, O], [AE 1575; CF ₃ , F, O, OMe, H, H, H, O], [AE 1576; CF ₃ , F, O, OE t, H, H, H, _{O], [AE1577; CF 3} , F, O, Oi-Pr, H, H, H, O], [AE1578; CF 3, F, O, SMe, H, H, H, O], [AE1579; _{CF 3, F, O, SEt} , H, H, H, O], [AE1580; CF 3, F, O, CH 2 F, H, H, H, O], [AE1581; CF 3, F, O _{, CHF 2, H, H,} H, O], [AE1582; CF 3, F, O, CF 3, H, H, H, O], [AE1583; CF 3, F, O, OCH 2 F, H , H, H, O], [AE 1584; CF ₃ , F, O, OCHF ₂ , H, H, H, O], [AE 1585; CF ₃ , F, O, OCF ₃ , H, H, H, O ], [AE 1586; CF ₃ , F, O, SCH ₂ F, H, H, H, O], [AE 1587; CF ₃ , F, O, SCHF ₂ , H, H, H, O], [AE 1588; _{CF 3, F, O, SCF} 3, H, H, H, O], [AE1589; CF 3, F, O, CN, H, H, H, O], [AE1590; CF 3, F, O, NO ₂ , H, H, H, O], [AE 1591; OMe, F, O, H, H, H, H, O], [AE 1592; OMe, F, O, F, H, H, H, O ], [AE 1593; OMe, F, O, Cl, H, H, H, O], [AE 1594; OMe, F, O, Br, H, H, H, O], [AE 1595; OMe, F, O] , I, H, H, H, O], [AE 1596; OMe, F, O, Me, H, H, H, O], [AE 1597; OMe, F, O, Et, H, H, H, O], [AE 1598; OMe, F, O, Pr, H, H, H, O], [AE 1599; OMe, F, O, i- Pr, H, H, H, O], [AE1600; OMe, F, O, CH = CH 2, H, H, H, O],

[AE 1601; OMe, F, O, C (Me) = CH ₂ , H, H, H, O], [AE 1602; OMe, F, O, C≡CH, H, H, H, O], [AE 1603 OMe, F, O, C≡CMe, H, H, H, O], [AE 1604, OMe, F, O, c-Pr, H, H, H, O], [AE 1605; OMe, F, O , OMe, H, H, H, O], [AE 1 606; OMe, F, O, OEt, H, H, H, O], [AE 1607; OMe, F, O, Oi-Pr, H, H, H , O], [AE 1 608; OMe, F, O, SMe, H, H, H, O], [AE 1609; OMe, F, O, SE t, H, H, H, O], [AE 1610; OMe, F _{, O, CH 2 F, H} , H, H, O], [AE1611; OMe, F, O, CHF 2, H, H, H, O], [AE1612; OMe, F, O, CF 3, H , H, H, O], [AE 1613; OMe, F, O, OCH ₂ F, H, H, H, O], [AE 1614; OMe, F, O, OCHF ₂ , H, H, H, O] , [AE1615; OMe, F, O, OCF 3, H, H, H, O], [AE1616; OMe, F, O, SCH 2 F, H, H, H, O], [AE1617; OMe, F , O, SCHF ₂ , H, H, H, O], [AE 1618; OMe, F, O, SCF ₃ , H, H, H, O], [AE 1619; OMe, F, O, CN, H, H , H, O], [AE 1620; OMe, F, O, NO ₂ , H, H, O], [AE1621; OEt, F, O, H, H, H, H, O], [AE 1622; OEt, F, O, F, H, H, H, O], [AE1623; OEt, F, O, Cl, H, H, H, O], [AE 1624; OEt, F, O, Br, H, H, H, O], [AE1625; OEt, F, O, I, H, H, H, O], [AE 1626; OEt, F, O, Me, H, H, H, O], [AE 1627; OEt, F, O, Et, H, H, H, O], [AE1628; OEt, F, O, Pr, H, H, H, O], [AE 1629; OEt, F, O, i-Pr, H, H, H, O] , [AE1630; OEt, F, O, CH = CH 2, H, H, H, O], [AE1631; OEt, F, O, C (Me) = CH 2, H , H, H, O], [AE 1632; OEt, F, O, C≡CH, H, H, H, O], [AE 1633; OE t, F, O, C ≡CMe, H, H, H, O], [AE1634; OEt, F, O, c-Pr, H, H, H, O], [AE 1635; OEt, F, O, OMe, H, H, H] , O], [AE1636; OEt, F, O, OEt, H, H, H, O], [AE 1637; OEt, F, O, Oi-Pr, H, H, H, O], [AE 1638; OEt , F, O, SMe, H, H, H, O, [AE 1639; OEt, F, O, SEt, H, H, H, O], [AE 1640; OEt, F, O, CH ₂ F, H , H, H, O], [AE1641; OEt, F, O, CHF 2, H, H, H, O], [AE1642; OEt, F, O, CF 3, H, H, H, O], [AE1643; OEt, F, O , OCH 2 F, H, H, H, O], [AE1644; OEt, F, O, OCHF 2, H, H, H, O], [AE1645; OEt, F, O, OCF ₃ , H, H, H, O], [AE 1 646; OEt, F, O, SCH ₂ F, H, H, H, O], [AE 1647; OEt, F, O, SCHF ₂ , H, H, H, O], [AE 1648; OEt, F, O, SCF ₃ , H, H, H, O], [AE 1 649; OE t, F, O, CN, H, H, H, O], [AE 16 50 ; OEt, F, O, NO 2, H, H, H, O], [AE1651; CN, F, O, H, H, H, H, O], [AE1652; CN, F, O, F, H, H, H, O], [AE 1653; CN, F, O, Cl, H, H, H, O], [AE 1654; CN, F, O, Br, H, H, H, O], [ AE 1655; CN, F, O, I, H, H, H, O], [AE 1656; CN, F, O, Me, H, H, H, O], [AE 1657; CN, F, O, Et, H, H, H, O], [AE 1658; CN, F, O, Pr, H, H, H, O], [AE 1659; CN, F, O, i-Pr, H, H, H, O] [AE 1660; CN, F, O, CH = CH ₂ , H, H, H, O], [AE 1661; CN, F, O, C (Me) = CH ₂ , H, H, H, O], [AE1662; CN, F, O, C≡CH, H, H, H, O], [AE1663; CN, F, O, C≡ CMe, H, H, H, O], [AE 1664; CN, F , O, c-Pr, H, H, H, O], [AE 1 665; CN, F, O, OMe, H, H, H, O], [AE 1 666; CN, F, O, OEt, H, H , H, O ], [AE1 667; CN, F, O, Oi-Pr, H, H, H, O], [AE 1668; CN, F, O, SMe, H, H, H, O], [AE 1 669; CN, F , O, SEt, H, H , H, O], [AE1670; CN, F, O, CH 2 F, H, H, H, O], [AE1671; CN, F, O, CHF 2, H, H, H, O], [ AE1672; CN, F, O, CF 3, H, H, H, O], [AE1673; CN, F, O, OCH 2 F, H, H, H, O], [AE1674; CN, F, O , OCHF 2, H, H, H, O], [AE1675; CN, F, O, OCF 3, H, H, H, O], [AE1676; CN, F, O , SCH ₂ F, H, H, H, O], [AE 1677; CN, F, O, SCHF ₂ , H, H, H, O], [AE 1678; CN, F, O, SCF ₃ , H, H , H, O], [AE 1679; CN, F, O, CN, H, H, H, O], [AE 1680; CN, F, O, NO ₂ , H, H, H, O], [AE 1681; F, Me, O, H, H, H, H, O, [AE1682; F, Me, O, F, H, H, H, O], [AE 1683; F, Me, O, Cl, H, H, H, O], [AE 1684; F, Me, O, Br, H, H, O], [AE 1 685; F, Me, O, I, H, H, H, O], [AE 1686; F, Me, O, Me, H, H, H, H, O], [AE 1687; F, Me, O, Et, H, H, H, O], [AE 1688; F, Me, O, Pr, H, H, H, O], [ AE1689; F, Me, O, i-Pr, H, H, H, O], [AE1690; F, Me, O, CH = CH 2, H, H, H, O F, Me, O, C (Me) = CH ₂ , H, H, H, O], [AE 1692; F, Me, O, C≡CH, H, H, H, O], [AE 1693; F, Me, O, C≡CMe, H, H, H, O], [AE 1694; F, Me, O, c-Pr, H, H, H, O], [AE 1695; F, Me , O, OMe, H, H, H, O], [AE 1696; F, Me, O, OEt, H, H, H, O], [AE 1697; F, Me, O, Oi-Pr, H, H , H, O], [AE 1698; F, Me, O, SMe, H, H, H, O], [AE 1699; F, Me, O, SE t, H, H, H, O], [AE 1700]; , Me, O, CH ₂ F, H, H, H, O],

[AE1701; F, Me, O , CHF 2, H, H, H, O], [AE1702; F, Me, O, CF 3, H, H, H, O], [AE1703; F, Me, O OCH ₂ F, H, H, H, H, O], [AE 1704; F, Me, O, OCHF ₂ , H, H, H, O], [AE 1705; F, Me, O, OCF ₃ , H, H , H, O], [AE 1706; F, Me, O, SCH ₂ F, H, H, H, O], [AE 1 707; F, Me, O, SCHF ₂ , H, H, H, O], [[ AE1708; F, Me, O, SCF 3, H, H, H, O], [AE1709; F, Me, O, CN, H, H, H, O], [AE1710; F, Me, O, NO ₂ , H, H, H, O], [AE 1711; F, Et, O, H, H, H, H, O], [AE 1712; F, Et, O, F, H, H, H, O] [AE 1713; F, Et, O, Cl, H, H, H, O], [AE 1714; F, Et, O, Br, H, H, H, O], [AE 1715; F, Et, O, I, H, H, H, O], [AE1716; F, Et, O, Me, H, H, H, O], [AE1717; F, Et, O, Et, H, H, H, O] [AE1718; F, Et, O, Pr, H, H, H, O], [AE1719; F, Et, O, i-Pr, H, H, H, O], [AE 1720; F, Et, _{O, CH = CH 2, H} , H, H, O], [AE1721; F, Et, O, C (Me) = CH 2, H, H, H, O], [AE1722; F, Et, O , C≡CH, H, H, H, O, [AE1723; F, Et, O, C≡CMe, H, H, H, O], [AE1724; F, Et, O, c-Pr, H , H, H, O], [AE1725; F, Et, O, OMe, H, H, H, O], [AE1726; F, Et, O, OEt, H, H, H, O], [AE 1727 F, Et, O, Oi-Pr, H, H, H, O], [AE1728; F, Et, O, SMe, H, H, H, O], [AE1729; F, Et, O, SEt , H, H, H, O ], [AE1730; F, Et, O, CH 2 F, H, H, H, O], [AE1731; F, Et, O, CHF 2, H, H, H, O], [AE 1732; F, Et, O, CF ₃ , H, H, H, O], [AE 1733; F, Et, O, OCH ₂ F, H, H, H, O], [AE 1734; F , Et, O, OCHF ₂ , H, H, H, O] , [AE1735; F, Et, O, OCF 3, H, H, H, O], [AE1736; F, Et, O, SCH 2 F, H, H, H, O F, Et, O, SCHF ₂ , H, H, H, O], [AE 1738; F, Et, O, SCF ₃ , H, H, H, O], [AE 1739; F, Et , O, CN, H, H, H, O, [AE 1740; F, Et, O, NO ₂ , H, H, H, O], [AE 1741; F, F, O, H, H, H, H, H, O], [AE 1742; F, F, O, F, H, H, H, O], [AE 1743; F, F, O, Cl, H, H, H, O], [AE 1 744; F, F, O, Br, H, H, H, O], [AE 1 745; F, F, O, I, H, H, H, O], [AE 1746; F, F, O, Me, H, H, H, O], [AE 1 747; F, F, O, Et, H, H, H, O], [AE 1 748; F, F, O, Pr, H, H, H, O], [AE 1 749; F, F, O, i-Pr, H, H, H, O], [AE1750; F, F, O, CH = CH 2, H, H, H, O], [AE1751; F, F, O, C _{(Me) = CH 2, H} , H, H, O], [AE1752; F, F, O, C≡CH, H, H, H, O], [AE1753; F, F, O, C≡CMe , H, H, H, O], [AE 1754; F, F, O, c-Pr, H, H, H, O], [AE 1 755; F, F, O, OMe, H, H, H, O F, F, O, OEt, H, H, H, O], [AE 1757; F, F, O, Oi-Pr, H, H, H, O], [AE 1758; F, F] , O, SMe, H, H, H, O], [AE1759; F, F, O, SEt, H, H, H, O], [AE 1760; F, F, O, CH ₂ F, H, H , H, O], [AE1761 ; F, F, O, CHF 2, H, H, H, O], [AE1762; F, F, O, CF 3, H, H, H, O], [AE1763 F, F, O, OCH ₂ F, H, H, H, O], [AE 1764; F, F, O, OCHF ₂ , H, H, H, O], [AE 1 765; F, F, O, OCF ₃ , H, H, H, O], [AE 1766; F, F, O, SCH ₂ F, H, H, H, O], [AE 1767; F, F, O, SCHF ₂ , H, H, H, O], [AE 1768; F, F, O, SCF ₃ , H, H, H, O], [AE 1769; F , F, O, CN, H, H, H, O, [AE 1 770; F, F, O, NO ₂ , H, H, H, O], [AE 1771; F, Cl, O, H, H, H, H, O], [AE1772; F, Cl, O, F, H, H, H, O], [AE1773; F, Cl, O, Cl, H, H, H, O], [AE 1774; F, Cl, O, Br, H, H, H, O, [AE 1775; F, Cl, O, I, H, H, H, O], [AE 1776; F, Cl, O, Me, H, H, H, O], [AE 1 777; F, Cl, O, Et, H, H, H, O], [AE 1778; F, Cl, O, Pr, H, H, H, O], [AE 1 779; F, Cl, O, i- Pr, H, H, H, O], [AE1780; F, Cl, O, CH = CH 2, H, H, H, O], [AE1781; F, Cl, O , C (Me) = CH ₂ , H, H, H, O], [AE 1782; F, Cl, O, C≡CH, H, H, H, O], [AE 1783; F, Cl, O, C ≡CMe, H, H, H, O], [AE 1784; F, Cl, O, c-Pr, H, H, H, O], [AE 1 785; F, Cl, O, OMe, H, H, H , O], [AE1786; F, Cl, O, OEt, H, H, H, O], [AE 1787; F, Cl, O, Oi-Pr, H, H, H, O], [AE 1788; F , Cl, O, SMe, H, H, H, O, [AE1 789; F, Cl, O, SEt, H, H, H, O], [AE 1 790; F, Cl, O, CH ₂ F, H , H, H, O], [AE1791; F, Cl, O, CHF 2, H, H, H, O], [AE1792; F, Cl, O, CF 3, H, H, H, O], [AE1793; F, Cl, O , OCH 2 F, H, H, H, O], [AE1794; F, Cl, O, OCHF 2, H, H, H, O], [AE1795; F, Cl, O, OCF ₃ , H, H, H, O], [AE 1796; F, Cl, O, SCH ₂ F, H, H, H, O], [AE 1797; F, Cl, O, SCHF ₂ , H, H, H, O], [ AE1798; F, Cl, O, SCF 3, H, H, H, O], [AE1799; F, Cl, O, CN, H, H, H, O], [AE1800 F, Cl, O, NO ₂ , H, H, H, O],

[AE 1801; F, Br, O, H, H, H, H, O], [AE 1802; F, Br, O, F, H, H, H, O], [AE 1803; F, Br, O, Cl , H, H, H, O], [AE1804; F, Br, O, Br, H, H, H, O], [AE 1805; F, Br, O, I, H, H, H, O], [AE1806; F, Br, O, Me, H, H, H, O], [AE 1807; F, Br, O, Et, H, H, H, O], [AE 1808; F, Br, O, Pr , H, H, H, O ], [AE1809; F, Br, O, i-Pr, H, H, H, O], [AE1810; F, Br, O, CH = CH 2, H, H, H, O], [AE1811; F, Br, O, C (Me) = CH 2, H, H, H, O], [AE1812; F, Br, O, C≡CH, H, H, H, O], [AE 1813; F, Br, O, C≡CMe, H, H, H, O], [AE 1814; F, Br, O, c-Pr, H, H, H, O], [AE 1815; F, Br, O, OMe, H, H, H, O], [AE 1816; F, Br, O, OEt, H, H, H, O], [AE 1817; F, Br, O, Oi-Pr, H, H, H, O], [AE1818; F, Br, O, SMe, H, H, H, O], [AE 1819; F, Br, O, SEt, H, H, H, O], [ AE 1820; F, Br, O, CH ₂ F, H, H, H, O], [AE 1821; F, Br, O, CHF ₂ , H, H, H, O], [AE 1822; F, Br, O , CF ₃ , H, H, H, O], [AE 1823; F, Br, O, OCH ₂ F, H, H, H, O], [AE 1824; F, Br, O, OCHF ₂ , H, H , H, O], [AE1825 ; F, Br, O, OCF 3, H, H, H, O], [AE1826; F, Br, O, SCH 2 F, H, H, H, O], [ AE1827; F, Br, O, SCHF 2, H, H, H, O], [AE1828; F, Br, O, SCF 3, H, H, H, O], [AE1829; F, Br, O, CN, H, H, H, O], [AE 1830; F, Br, O, NO ₂ , H, H, H, O], [AE 1831; F, I, O, H, H, H, H, O ], [AE 1832; F, I, O, F, H, H, H, O], [AE 1833; F, I, O, Cl, H, H, H, O], [AE 1834; F, I, O] , Br, H, H, H, O], [AE 1835; F, I, O, I, H, H, H, O], [AE 1836; F, I, O, Me, H, H, H, O], [AE 1837; F, I, O, Et, H, H, H, O] [AE 1839; F, I, O, Pr, H, H, H, O], [AE 1839; F, I, O, i-Pr, H, H, H, O], [AE 1840; F, I, _{O, CH = CH 2, H} , H, H, O], [AE1841; F, I, O, C (Me) = CH 2, H, H, H, O], [AE1842; F, I, O , C≡CH, H, H, H, O], [AE1843; F, I, O, C≡CMe, H, H, H, O], [AE 1844; F, I, O, c-Pr, H , H, H, O], [AE 1845; F, I, O, OMe, H, H, H, O], [AE 1846; F, I, O, OE t, H, H, H, O], [AE 1 847 F, I, O, Oi-Pr, H, H, H, O], [AE1848; F, I, O, SMe, H, H, H, O], [AE 1849; F, I, O, SEt , H, H, H, O], [AE 1850; F, I, O, CH ₂ F, H, H, H, O], [AE 1851; F, I, O, CHF ₂ , H, H, H, O], [AE1852; F, I, O, CF 3, H, H, H, O], [AE1853; F, I, O, OCH 2 F, H, H, H, O], [AE1854; F _{, I, O, OCHF 2,} H, H, H, O], [AE1855; F, I, O, OCF 3, H, H, H, O], [AE1856; F, I, O, SCH 2 F , H, H, H, O], [AE 1857; F, I, O, SCHF ₂ , H, H, H, O], [AE 1858; F, I, O, SCF ₃ , H, H, H, O ], [AE 1859; F, I, O, CN, H, H, H, O], [AE 1860; F, I, O, NO ₂ , H, H, H, O], [AE 1861; F, CHF ₂ , O, H, H, H , H, O], [AE1862; F, CHF 2, O, F, H, H, H, O], [AE1863; F, CHF 2, O, Cl, H, H , H, O], [AE1864 ; F, CHF 2, O, Br, H, H, H, O], [AE1865; F, CHF 2, O, I, H, H, H, O], [AE1866 F, CHF ₂ , O, Me, H, H, H, O, [AE 1867; F, CHF ₂ , O, Et, H, H, H, O], [AE 1868; F, CHF ₂ , O, Pr, H, H, H, O], [AE 1869; F, CHF ₂ , O, i-Pr, H, H, H, O], [AE1870; F, CHF 2, O, CH = CH 2, H, H, H, O], [AE1871; F, CHF 2, O, C _{(Me) = CH 2, H} , H, H, O], [AE1872; F, CHF 2, O, C≡CH, H, H, H, O], [AE1873; F, CHF 2, O, C ≡CMe, H, H, H, O], [AE 1874; F, CHF ₂ , O, c-Pr, H, H, H, O], [AE 1875; F, CHF ₂ , O, OMe, H, H , H, O], [AE1876 ; F, CHF 2, O, OEt, H, H, H, O], [AE1877; F, CHF 2, O, Oi-Pr, H, H, H, O], _{[AE1878; F, CHF 2,} O, SMe, H, H, H, O], [AE1879; F, CHF 2, O, SEt, H, H, H, O], [AE1880; F, CHF 2, _{O, CH 2 F, H,} H, H, O], [AE1881; F, CHF 2, O, CHF 2, H, H, H, O], [AE1882; F, CHF 2, O, CF 3, H, H, H, O] , [AE1883; F, CHF 2, O, OCH 2 F, H, H, H, O], [AE1884; F, CHF 2, O, OCHF 2, H, H, H , O], [AE1885; F , CHF 2, O, OCF 3, H, H, H, O], [AE1886; F, CHF 2, O, SCH 2 F, H, H, H, O], [ AE 1887; F, CHF ₂ , O, SCHF ₂ , H, H, H, O], [AE 1 888; F, CHF ₂ , O, SCF ₃ , H, H, H, O], [AE 1889; F, CHF ₂ , O, CN, H, H , H, O], [AE1890; F, CHF 2, O, NO 2, H, H, H, O], [AE1891; F, CF 3, O, H, H, H, H, O], [ AE1892; F, CF 3, O, F, H, H, H, O], [AE1893; F, CF 3, O, Cl, H, H, H, O], [ _{AE1894; F, CF 3, O} , Br, H, H, H, O], [AE1895; F, CF 3, O, I, H, H, H, O], [AE1896; F, CF 3, O , Me, H, H, H, O], [AE 1897; F, CF ₃ , O, Et, H, H, H, O], [AE 1898; F, CF ₃ , O, Pr, H, H, H , O], [AE 1899; F, CF ₃ , O, i-P r, H, H, H, O], [AE 1900; F, CF ₃ , O, CH = CH ₂ , H, H, H, O],

_{[AE1901; F, CF 3,} O, C (Me) = CH 2, H, H, H, O], [AE1902; F, CF 3, O, C≡CH, H, H, H, O], _{[AE1903; F, CF 3,} O, C≡CMe, H, H, H, O], [AE1904; F, CF 3, O, c-Pr, H, H, H, O], [AE1905; F , CF ₃ , O, OMe, H, H, H, O], [AE 1906; F, CF ₃ , O, OEt, H, H, H, O], [AE 1907; F, CF ₃ , O, Oi − Pr, H, H, H, O], [AE 1908; F, CF ₃ , O, SMe, H, H, H, O], [AE 1 909; F, CF ₃ , O, SE t, H, H, H, O, [AE 1910; F, CF ₃ , O, CH ₂ F, H, H, H, O], [AE 1911; F, CF ₃ , O, CHF ₂ , H, H, H, O], [AE 19 12 F, CF ₃ , O, CF ₃ , H, H, H, O], [AE1913; F, CF ₃ , O, OCH ₂ F, H, H, H, O], [AE 1914; F, CF ₃ , O, OCHF ₂ , H, H, H, O], [AE 1915; F, CF ₃ , O, OCF ₃ , H, H, H, O], [AE 1916; F, CF ₃ , O, SCH ₂ F , H, H, H, O ], [AE1917; F, CF 3, O, SCHF 2, H, H, H, O], [AE1918; F, CF 3, O, SCF 3, H, H, H , O], [AE1919; F , CF 3, O, CN, H, H, H, O], [AE1920; F, CF 3, O, NO 2, H, H, H, O], [AE1921; F, OMe, O, H, H, H, H, H, O], [AE1922; F, OMe, O, F, H, H, H, O], [AE 1923; F, OMe, O, Cl, H, H, H, O], [AE 1 924; F, OMe, O, Br, H, H, H, O], [AE 1 925; F, OMe, O, I, H, H, H, O], [AE 1 926; F, OMe, O, Me, H, H, H, H, O], [AE 1 927; F, OMe, O, Et, H, H, H, O], [AE 1 928; F, OMe, O, Pr, H, H, H, O], [ AE1929; F, OMe, O, i-Pr, H, H, H, O], [AE1930; F, OMe, O, CH = CH 2, H, H, H, O ], [AE1931; F, OMe , O, C (Me) = CH 2, H, H, H, O], [AE1932; F , OMe, O, C≡CH, H, H, H, O], [AE1933; F, OMe, O, C≡ CMe, H, H, H, O], [AE 1934; F, OMe, O, c -Pr, H, H, H, O], [AE 1935; F, OMe, O, OMe, H, H, H, O], [AE 1936; F, OMe, O, OEt, H, H, H, O F, OMe, O, Oi-Pr, H, H, H, O], [AE 1938; F, OMe, O, SMe, H, H, H, O], [AE 1939; F, OMe] , O, SEt, H, H, H, O], [AE 1940; F, OMe, O, CH ₂ F, H, H, H, O], [AE 1941; F, OMe, O, CHF ₂ , H, H, H, O], [ AE1942; F, OMe, O, CF 3, H, H, H, O], [AE1943; F, OMe, O, OCH 2 F, H, H, H, O], [AE1944; F, OMe, O , OCHF 2, H, H, H, O], [AE1945; F, OMe, O, OCF 3, H, H, H, O], [AE1946; F, OMe, O SCH ₂ F, H, H, H, H, O], [AE 1947; F, OMe, O, SCHF ₂ , H, H, H, O], [AE 1948; F, OMe, O, SCF ₃ , H, H , H, O], [AE 1949; F, OMe, O, CN, H, H, H, O], [AE 1950; F, OMe, O, NO ₂ , H, H, H, O], [AE 1951; F, OEt, O, H, H, H, H, H, O], [AE1952; F, OEt, O, F, H, H, H, O], [AE1953; F, OEt, O, Cl, H, H, H, O], [AE1954; F, OEt, O, Br, H, H, O], [AE 1 955; F, OEt, O, I, H, H, H, O], [AE 1956; F, OEt, O, Me, H, H, H, H, O], [AE 1957; F, OEt, O, Et, H, H, H, O], [AE 1958; F, OEt, O, Pr, H, H, H, O], [ AE1959; F, OEt, O, i-Pr, H, H, H, O], [AE1960; F, OEt, O, CH = CH 2, H, H, H, O ], [AE1961; F, OEt , O, C (Me) = CH 2, H, H, H, O], [AE1962; F, OEt, O, C≡CH, H, H, H, O], [AE1963; F, OEt, O, C≡CMe, H, H, H, O], [AE1964; F, OEt, O, c-Pr, H, H, H, O], [AE1 965; F, OEt, O, OMe, H, H, H, O], [AE1966; F, OEt, O, OEt, H, H, H, O], [AE 1967; F, OEt, O, Oi -Pr, H, H, H, O], [AE 1968; F, OEt, O, SMe, H, H, H, O], [AE 1969; F, OE t, O, SE t, H, H, H, O ], [AE1970; F, OEt , O, CH 2 F, H, H, H, O], [AE1971; F, OEt, O, CHF 2, H, H, H, O], [AE1972; F, _{OEt, O, CF 3, H} , H, H, O], [AE1973; F, OEt, O, OCH 2 F, H, H, H, O], [AE1974; F, OEt, O, OCHF 2, H, H, H, O] , [AE1975; F, OEt, O, OCF 3, H, H, H, O], [AE1976; F, OEt, O, SCH 2 F, H, H, H, O ], [AE1977; F, OEt , O, SCHF 2, H, H, H, O], [AE1978; F, OEt, O, SCF 3, H, H, H, O], [AE1979; F, OEt , O, CN, H, H, H, O, [AE1980; F, OEt, O, NO ₂ , H, H, H, O], [AE1981; F, CN, O, H, H, H, H, H H, O], [AE 1982; F, CN, O, F, H, H, H, O], [AE 1983; F, CN, O, Cl, H, H, H, O], [AE 1984; F, CN, O, Br, H, H, H, O], [AE1985; F, CN, O, I, H, H, H, O], [AE 1986; F, CN, O, Me, H, H, H H, O], [AE 1987; F, CN, O, Et, H, H, H, O], [AE 1988; F, CN, O, Pr, H, H, H, O], [AE 1989; F, CN, O, i-Pr, H, H, H, O], [AE1990; F, CN, O, CH = CH 2, H, H, H, O], [AE1991; F, CN, O, C (Me) = CH ₂ , H, H, H, O], [AE 1992; F, CN, O, C≡CH, H, H, H, O], [AE 1993; F, CN, O, C≡ CMe , H, H, H, O], [AE 1994; F, CN, O, c-Pr, H, H, H, O], [AE 1995; F, CN, O, OMe, H, H, H, O ], [AE 1996; F, CN, O, OEt, H, H, H, O], [AE 1997; F, CN, O, Oi-Pr, H, H, H, O], [AE 1998; F, CN] , O , SMe, H, H, H, O], [AE 1999; F, CN, O, SEt, H, H, H, O], [AE 2000; F, CN, O, CH ₂ F, H, H, H , O],

[AE2001; F, CN, O , CHF 2, H, H, H, O], [AE2002; F, CN, O, CF 3, H, H, H, O], [AE2003; F, CN, O OCH ₂ F, H, H, H, O], [AE 2004; F, CN, O, OCHF ₂ , H, H, H, O], [AE 2005; F, CN, O, OCF ₃ , H, H , H, O], [AE2006; F, CN, O, SCH ₂ F, H, H, H, O], [AE 2007; F, CN, O, SCHF ₂ , H, H, H, O], [[ AE2008; F, CN, O, SCF 3, H, H, H, O], [AE2009; F, CN, O, CN, H, H, H, O], [AE2010; F, CN, O, NO ₂ , H, H, H, O], [AE 2011; H, H, O, H, F, H, H, O], [AE 2012; H, H, O, F, F, H, H, O] , [AE2013; H, H, O, Cl, F, H, H, O], [AE 2014; H, H, O, Br, F, H, H, O], [AE 2015; H, H, O, I, F, H, H, O], [AE 2016; H, H, O, Me, F, H, H, O], [AE 2017; H, H, O, Et, F, H, H, O] H, H, O, Pr, F, H, H, O], [AE 2019; H, H, O, i-Pr, F, H, H, O], [AE 2020; H, H, _{O, CH = CH 2, F} , H, H, O], [AE2021; H, H, O, C (Me) = CH 2, F, H, H, O], [AE2022; H, H, O , C≡CH, F, H, H, O], [AE 2023; H, H, O, C≡ CMe, F, H, H, O], [AE 2024; H, H, O, c-Pr, F , H, H, O], [AE 2025; H, H, O, OMe, F, H, H, O], [AE 2026; H, H, O, OE t, F, H, H, O], [AE 20 27 H, H, O, Oi-Pr, F, H, H, O], [AE2028; H, H, O, SMe, F, H, H, O], [AE 2029; H, H, O, SEt , F, H, H, O], [AE 2030; H, H, O, CH ₂ F, F, H, H, O], [AE 2031; H, H, O, CHF ₂ , F, H, H, O, [AE 2032; H, H, O, CF ₃ , F, H, H, O], [AE 2033; H, H, O, OCH ₂ F, F, H, H, O], [AE 2034; H , H, O, OCHF ₂ , F, H, H, O], [AE 2035; H, H, O, O _{CF 3, F, H, H} , O], [AE2036; H, H, O, SCH 2 F, F, H, H, O], [AE2037; H, H, O, SCHF 2, F, H, H, O], [AE 2038; H, H, O, SCF ₃ , F, H, H, O], [AE 2039; H, H, O, CN, F, H, H, O], [AE 2040; H _{, H, O, NO 2,} F, H, H, O], [AE2041; Me, H, O, H, F, H, H, O], [AE2042; Me, H, O, F, F, H, H, O], [AE 2043; Me, H, O, Cl, F, H, H, O], [AE 2044; Me, H, O, Br, F, H, H, O], [AE 2045; Me, H, O, I, F, H, H, O], [AE 2046; Me, H, O, Me, F, H, H, O], [AE 2047; Me, H, O, Et, F, H, H, O], [AE 2048; Me, H, O, Pr, F, H, H, O], [AE 2049; Me, H, O, i-Pr, F, H, H, O], [[ AE2050; Me, H, O, CH = CH 2, F, H, H, O], [AE2051; Me, H, O, C (Me) = CH 2, F, H, H, O], [AE2052 Me, H, O, C≡CH, F, H, H, O], [AE 2053; Me, H, O, C≡ C Me, F, H, H, O], [AE 2054; Me, H, O , c-Pr, F, H, H, O], [AE2055; Me, H, O, OMe, F, H, H, O], [AE 2056; Me, H, O, OEt, F, H, H] , O], [AE2057; Me, H, O, Oi-Pr, F, H, H, O], [AE 2058; Me, H, O, SMe, F, H, H, O], [AE 2059; Me , H, O, SEt, F , H, H, O], [AE2060; Me, H, O, CH 2 F, F, H, H, O], [AE2061; Me, H, O, CHF 2, F, H, H, O] , [AE2062; Me, H, O, CF 3, F, H, H, O], [AE2063; Me, H, O, OCH 2 F, F, H, H, O ], [AE2064; Me, H , O, OCHF 2, F, H, H, O], [AE2065; Me, H, O, OCF 3, F, H, H, O], [AE2066; Me, H , O, SCH ₂ F, F, H, H, O], [AE 2067; Me, H, O, SCHF ₂ , F, H, H, O], [AE 2068; Me, H, O, SCF ₃ , F , H, H, O], [AE 2069; Me, H, O, CN, F, H, H, O], [AE2070; Me, H, O, NO 2, F, H, H, O], [AE2071; H, Me, O, H, F, H , H, O], [AE2072; H, Me, O, F, F, H, H, O], [AE 2073; H, Me, O, Cl, F, H, H, O], [AE 2074; H , Me, O, Br, F, H, H, O], [AE 2075; H, Me, O, I, F, H, H, O], [AE 2076; H, Me, O, Me, F, H , H, O], [AE 2077; H, Me, O, Et, F, H, H, O], [AE 2078; H, Me, O, Pr, F, H, H, O], [AE 2079; H , Me, O, i-Pr , F, H, H, O], [AE2080; H, Me, O, CH = CH 2, F, H, H, O], [AE2081; H, Me, O, _{C (Me) = CH 2,} F, H, H, O], [AE2082; H, Me, O, C≡CH, F, H, H, O], [AE2083; H, Me, O, C≡ CMe, F, H, H, O], [AE 2084; H, Me, O, c-Pr, F, H, H, O], [AE 2085; H, Me, O, OMe, F, H, H, O, [AE 2086; H, Me, O, OEt, F, H, H, O], [AE 2087; H, Me, O, Oi-Pr, F, H, H, O], [AE 2088; H, Me, O, SMe, F, H, H, O], [AE 2089; H, Me, O, SE t, F, H, H, O], [AE 2090; H, Me, O, CH ₂ F, F, H, H, O], [ AE2091; H, Me, O, CHF 2, F, H, H, O], [AE2092; H, Me, O, CF 3, F, H, H, O], [ AE2093; H, Me, O, OCH 2 F, F, H, H, O], [AE2094; H, Me, O, OCHF 2, F, H, H, O], [AE2095; H, Me, O _{, OCF 3, F, H,} H, O], [AE2096; H, Me, O, SCH 2 F, F, H, H, O], [AE2097; H, Me, O, SCHF 2, F, H H, O], [AE 2098; H, Me, O, SCF ₃ , F, H, H, O], [AE 2099; H, Me, O, CN, F, H, H, O], [AE 2 100; H, Me, O, NO ₂ , F, H, H, O],

[AE 2101; F, H, O, H, F, H, H, O], [AE 2102; F, H, O, F, F, H, H, O], [AE 2 103; F, H, O, Cl , F, H, H, O], [AE 2 104; F, H, O, Br, F, H, H, O], [AE 2 105; F, H, O, I, F, H, H, O], [AE 2 106; F, H, O, Me, F, H, H, O], [AE 2 107; F, H, O, Et, F, H, H, O], [AE 2 108; F, H, O, Pr , F, H, H, O ], [AE2109; F, H, O, i-Pr, F, H, H, O], [AE2110; F, H, O, CH = CH 2, F, H, H, O], [AE 2 111; F, H, O, C (Me) = CH ₂ , F, H, H, O], [AE 2 112; F, H, O, C≡CH, F, H, H, O, [AE 2 113; F, H, O, C≡CMe, F, H, H, O], [AE 2114; F, H, O, c-Pr, F, H, H, O], [AE 2 115; F, H, O, OMe, F, H, H, O], [AE 2116; F, H, O, OEt, F, H, H, O], [AE 2 117; F, H, O, Oi-Pr, F, H, H, O], [AE 2 118; F, H, O, S Me, F, H, H, O], [AE 2 119; F, H, O, SE t, F, H, H, O], [ AE ₂ 120; F, H, O, CH ₂ F, F, H, H, O], [AE 2121; F, H, O, CHF ₂ , F, H, H, O], [AE 2 122; F, H, O , CF ₃ , F, H, H, O], [AE ₂ 123; F, H, O, OCH ₂ F, F, H, H, O], [AE ₂ 124; F, H, O, OCHF ₂ , F, H , H, O], [AE 2 125; F, H, O, OCF ₃ , F, H, O], [AE ₂ 126; F, H, O, SCH ₂ F, F, H, H, O], [ AE 2127; F, H, O, SCHF ₂ , F, H, H, O], [AE 2 128; F, H, O, SCF ₃ , F, H, H, O], [AE 2 129; F, H, O, CN, F, H, H, O], [AE 2130; F, H, O, NO ₂ , F, H, H, O], [AE 2 131; H, F, O, H, F, H, H, O H, F, O, F, F, H, H, O], [AE 2133; H, F, O, Cl, F, H, H, O], [AE 2 134; H, F, O] , Br, F, H, H, O], [AE 2 135; H, F, O, I, F, H, H, O], [AE 2 136; H, F, O, Me, F, H, H, O], [AE 2137; H, F, O, Et, F, H, H, O], [AE 2138; H, F, O, Pr, F, H, H, O], [AE 2 139; H, F, O, i-Pr, F, H, H, O], [AE 2 140; H, F, O, CH = CH ₂ , F, H, H, O], [AE 2141; H, F, O _{, C (Me) = CH 2} , F, H, H, O], [AE2142; H, F, O, C≡CH, F, H, H, O], [AE2143; H, F, O, C ≡CMe, F, H, H, O], [AE 2144; H, F, O, c-Pr, F, H, H, O], [AE 2 145; H, F, O, OMe, F, H, H , O], [AE 2146; H, F, O, OEt, F, H, H, O], [AE 2147; H, F, O, Oi-Pr, F, H, H, O], [AE 2148; H , F, O, SMe, F, H, H, O], [AE 2 149; H, F, O, SE t, F, H, H, O], [AE ₂ 150; H, F, O, CH ₂ F, F , H, H, O], [AE2151; H, F, O, CHF 2, F, H, H, O], [AE2152; H, F, O, CF 3, F, H, H, O], [AE ₂ 153; H, F, O, OCH ₂ F, F, H, H, O], [AE ₂ 154; H, F, O, OCHF ₂ , F, H, H, O], [AE 2 155; H, F, _{O, OCF 3, F, H} , H, O], [AE2156; H, F, O, SCH 2 F, F, H, H, O], [AE2157; H, F, O, SCHF 2, F, H, H, O], [AE 2158; H, F, O, SCF ₃ , F, H, H, O], [AE 2 159; H, F, O, CN, F, H, H, O], [AE 2 160 H, F, O, NO ₂ , F, H, H, O], [AE2161; H, H, O, H, H, F, H, O], [AE 2162; H, H, O, F, H, F, H, O], [AE 2 163; H, H, O, Cl, H, F, H, O], [AE 2 164; H, H, O, Br, H, F, H, O], [[ H, H, O, I, H, F, H, O], [AE 2166; H, H, O, Me, H, F, H, O], [AE 2 167; H, H, O, Et, H, F, H, O], [AE 2 168; H, H, O, Pr, H, F, H, O], [AE 2 169; H, H, O, i-Pr, H, F, H, O] , [AE 2170; H, H, O, CH = CH ₂ , H, F, H, O], [AE 2171; H, H, O, C (Me) = CH ₂ , H , F, H, O], [AE2172 H, H, O, C≡CH, H, F, H, O], [AE 2173; H, H, O, CF C Me, H, F, H, O H, H, O, c-Pr, H, F, H, O], [AE 2175; H, H, O, OMe, H, F, H, O], [AE 2176; H, H] , O, OEt, H, F, H, O], [AE 2177; H, H, O, Oi-Pr, H, F, H, O], [AE 2 178; H, H, O, SMe, H, F , H, O], [AE 2 179; H, H, O, SE t, H, F, H, O], [AE ₂ 180; H, H, O, CH ₂ F, H, F, H, O], [AE 2181 ; H, H, O, CHF 2, H, F, H, O], [AE2182; H, H, O, CF 3, H, F, H, O], [AE2183; H, H, O, OCH ₂ F, H, F, H, O], [AE ₂ 184; H, H, O, OCHF ₂ , H, F, H, O], [AE 2 185; H, H, O, OCF ₃ , H, F, H H, H, O, SCH ₂ F, H, F, H, O], [AE 2187; H, H, O, SCHF ₂ , H, F, H, O], [AE 2 188; _{H, H, O, SCF 3} , H, F, H, O], [AE2189; H, H, O, CN, H, F, H, O], [AE2190; H, H, O, NO 2, H, F, H, O], [AE2191; Me, H, O, H, H, F, H, O], [AE 2 192; Me, H, O, F, H, F, H, O], [[ AE2193; Me, H, O, Cl, H, F, H, O], [AE 2 194; Me, H, O, Br, H, F, H, O], [AE 2195; Me, H, O, I, H, F, H, O], [AE 2196; Me, H, O, Me, H, F, H, O], [AE 2 197; Me, H, O, Et, H, F, H, O], [ AE 2198; Me, H, O, Pr, H, F, H, O], [AE 2199; Me, H, O, i-Pr, H, F, H, O], [AE 2 200; Me, H, O, CH = CH ₂ , H, F, H, O],

[AE2201; Me, H, O , C (Me) = CH 2, H, F, H, O], [AE2202; Me, H, O, C≡CH, H, F, H, O], [AE2203 Me, H, O, C≡CMe, H, F, H, O], [AE 2 204; Me, H, O, c-Pr, H, F, H, O], [AE 2 205; Me, H, O , OMe, H, F, H, O], [AE 2206; Me, H, O, OEt, H, F, H, O], [AE 2207; Me, H, O, Oi-Pr, H, F, H , O], [AE2208; Me, H, O, SMe, H, F, H, O], [AE 2209; Me, H, O, SEt, H, F, H, O], [AE 2210; Me, H _{, O, CH 2 F, H} , F, H, O], [AE2211; Me, H, O, CHF 2, H, F, H, O], [AE2212; Me, H, O, CF 3, H , F, H, O], [AE2213; Me, H, O, OCH 2 F, H, F, H, O], [AE2214; Me, H, O, OCHF 2, H, F, H, O] , [AE2215; Me, H, O, OCF 3, H, F, H, O], [AE2216; Me, H, O, SCH 2 F, H, F, H, O], [AE2217; Me, H , O, SCHF ₂ , H, F, H, O], [AE 2218; Me, H, O, SCF ₃ , H, F, H, O], [AE 2219; Me, H, O, CN, H, F , H, O], [AE 2220; Me, H, O, NO ₂ , H, F, H, O], [AE 2221; H, Me, O, H, H, F, H, O], [AE 2222; H, Me, O, F, H, F, H, O], [AE2223; H, Me, O, Cl, H, F, H, O], [AE 2224; H, Me, O, Br, H, F, H, O], [AE 2225; H, Me, O, I, H, F, H, O], [AE 2226; H, Me, O, Me, H, F, H, O], [AE 2 227; H, Me, O, Et, H, F, H, O], [AE 2 228; H, Me, O, Pr, H, F, H, O], [AE 2 229; H, Me, O, i-Pr, H, F, H, O], [AE 2 230; H, Me, O, CH = CH ₂ , H, F, H, O], [AE 2 231; H, Me, O, C (Me) = CH ₂ , H , F, H, O], [AE 2232; H, Me, O, C≡CH, H, F, H, O], [AE 2233; H, Me, O, C≡ C Me, H, F, H, O ], [AE2234; H, Me, O, c- Pr, H, F, H, O], [AE 2235; H, Me, O, OMe, H, F, H, O], [AE 2236; H, Me, O, OEt, H, F, H, O] H, Me, O, Oi-Pr, H, F, H, O], [AE 2238; H, Me, O, SMe, H, F, H, O], [AE 2239; H, Me, O, SEt, H, F, H, O], [AE ₂ 240; H, Me, O, CH ₂ F, H, F, H, O], [AE 2241; H, Me, O, CHF ₂ , H, F , H, O], [AE2242 ; H, Me, O, CF 3, H, F, H, O], [AE2243; H, Me, O, OCH 2 F, H, F, H, O], [ AE2244; H, Me, O, OCHF 2, H, F, H, O], [AE2245; H, Me, O, OCF 3, H, F, H, O], [AE2246; H, Me, O, SCH ₂ F, H, F, H, O], [AE 2247; H, Me, O, SCHF ₂ , H, F, H, O], [AE 2248; H, Me, O, SCF ₃ , H, F, H, O], [AE 2249; H, Me, O, CN, H, F, H, O], [AE ₂ 250; H, Me, O, NO ₂ , H, F, H, O], [AE 2251; F , H, O, H, H, F, H, O], [AE 2252; F, H, O, F, H, F, H, O], [AE 2 253; F, H, O, Cl, H, F , H, O], [AE 2 254; F, H, O, Br, H, H, O], [AE 2 255; F, H, O, I, H, F, H, O], [AE 2 256; F , H, O, Me, H, F, H, O], [AE 2 257; F, H, O, Et, H, F, H, O], [AE 2 258; F, H, O, Pr, H, F , H, O], [AE2259 ; F, H, O, i-Pr, H, F, H, O], [AE2260; F, H, O, CH = CH 2, H, F, H, O] [AE 2261; F, H, O, C (Me) = CH ₂ , H, F, H, O], [AE 2262; F, H, O, C≡CH, H, F, H, O], [[ AE 2263; F, H, O, C≡CMe, H, F, H, O], [AE 2 264; F, H, O, c-Pr, H, F, H, O], [AE 2 265; F, H, O, OMe, H, F, H, O], [AE 2 266; F, H, O, OEt, H, F, H, O], [AE 2 267; F, H, O, Oi-Pr, H, F, H, O], [AE 2268; F, H, O, SMe, H, F, H, O], [AE 2269; F, H, O, SEt, H, F, H, O], [AE ₂ 270; F, H, O, CH ₂ F, H, F, H, O], [AE 2271; F, H, O, CHF ₂ , H, F, H, O ], [AE2272; F, H, O, CF 3, H, F, H, O], [AE2273; F, H, O, OCH 2 F, H, F, H, O, [AE ₂ 274; F, H, O, OCHF ₂ , H, F, H, O], [AE 2275; F, H, O, OCF ₃ , H, F, H, O], [AE 2 276; F, H, O, SCH ₂ F, H, F, H, O], [AE 2277; F, H, O, SCHF ₂ , H, F, H, O], [AE 2 278; F, H, O, SCF ₃ , H, F, H, O], [AE 2279; F, H, O, CN, H, F, H, O], [AE ₂ 280; F, H, O, NO ₂ , H, F, H, O], [AE2281; H, F, O, H, H, F, H, O], [AE2282; H, F, O, F, H, F, H, O], [AE 2283; H, F, O, Cl , H, F, H, O], [AE 2284; H, F, O, Br, H, F, H, O], [AE 2285; H, F, O, I, H, F, H, O], [AE2286; H, F, O, Me, H, F, H, O], [AE 2287; H, F, O, Et, H, F, H, O], [AE 2288; H, F, O, Pr H, F, H, O], [AE 2 289; H, F, O, i-Pr, H, F, H, O], [AE 2 290; H, F, O, CHCHCH ₂ , H, F, H, O], [AE2291; H, F, O, C (Me) = CH 2, H, F, H, O], [AE2292; H, F, O, C≡CH, H, F, H, O, [AE2293; H, F, O, C≡CMe, H, F, H, O], [AE 2294; H, F, O, c-Pr, H, F, H, O], [AE 2295; H, F, O, OMe, H, F, H, O], [AE 2296; H, F, O, OEt, H, F, H, O], [AE 2 297; H, F, O, Oi-Pr, H, F, H, O], [AE2298; H, F, O, SMe, H, F, H, O], [AE 2299; H, F, O, SEt, H, F, H, O], [ AE 2300; H, F, O, CH ₂ F, H, F, H, O],

[AE2301; H, F, O , CHF 2, H, F, H, O], [AE2302; H, F, O, CF 3, H, F, H, O], [AE2303; H, F, O OCH ₂ F, H, F, H, O], [AE ₂ 304; H, F, O, OCHF ₂ , H, F, H, O], [AE 2 305; H, F, O, OCF ₃ , H, F , H, O], [AE 2306; H, F, O, SCH ₂ F, H, F, H, O], [AE ₂ 307; H, F, O, SCHF ₂ , H, F, H, O], [[ H, F, O, SCF ₃ , H, F, H, O], [AE 2 309; H, F, O, CN, H, F, H, O], [AE 2310; H, F, O, NO ₂ , H, F, H, O], [AE 2311; H, H, O, H, H, H, F, O], [AE 2312; H, H, O, F, H, H, F, O] H, H, O, Cl, H, F, O], [AE 2314; H, H, O, Br, H, F, O], [AE 2315; H, H, O, I, H, H, F, O], [AE2316; H, H, O, Me, H, H, F, O], [AE 2317; H, H, O, Et, H, H, F, O] H, H, O, Pr, H, F, O], [AE 2319; H, H, O, i-Pr, H, F, O], [AE 2 320; H, H, _{O, CH = CH 2, H} , H, F, O], [AE2321; H, H, O, C (Me) = CH 2, H, H, F, O], [AE2322; H, H, O , C≡CH, H, H, F, O], [AE2323; H, H, O, C≡CMe, H, H, F, O], [AE 2324; H, H, O, c-Pr, H , H, F, O], [AE2325; H, H, O, OMe, H, H, F, O], [AE 2326; H, H, O, OEt, H, H, F, O], [AE 2327 H, H, O, Oi-Pr, H, H, F, O], [AE2328; H, H, O, SMe, H, F, O], [AE 2329; H, H, O, SEt , H, H, F, O ], [AE2330; H, H, O, CH 2 F, H, H, F, O], [AE2331; H, H, O, CHF 2, H, H, F, O], [AE2332; H, H, O, CF 3, H, H, F, O], [AE2333; H, H, O, OCH 2 F, H, H, F, O], [AE2334; H _{, H, O, OCHF 2,} H, H, F, O], [AE2335; H, H, O, OCF 3, H, H, H, H, O, SCH ₂ F, H, F, O], [AE ₂ 337; H, H, O, SCHF ₂ , H, H, F, O], [AE 2 338] ; H, H, O, SCF 3, H, H, F, O], [AE2339; H, H, O, CN, H, H, F, O], [AE2340; H, H, O, NO 2 , H, H, F, O], [AE2341; Me, H, O, H, H, H, F, O], [AE 2342; Me, H, O, F, H, H, F, O], [AE 2343; Me, H, O, Cl, H, H, F, O], [AE 2344; Me, H, O, Br, H, F, O], [AE 2 345; Me, H, O, I , H, H, F, O], [AE 2346; Me, H, O, Me, H, H, F, O], [AE 2347; Me, H, O, Et, H, H, F, O], [AE2348; Me, H, O, Pr, H, H, F, O], [AE 2349; Me, H, O, i-Pr, H, H, F, O], [AE 2 350; Me, H, O _{, CH = CH 2, H,} H, F, O], [AE2351; Me, H, O, C (Me) = CH 2, H, H, F, O], [AE2352; Me, H, O, C≡CH, H, H, F, O], [AE2353; Me, H, O, C≡CMe, H, H, F, O], [AE 2354; Me, H, O, c-Pr, H, H, F, O], [AE 2 355; Me, H, O, OMe, H, H, F, O], [AE 2 356; Me, H, O, OE t, H, H, F, O], [AE 2 357; Me, H, O, Oi-Pr, H, H, F, O], [AE2358; Me, H, O, SMe, H, F, O], [AE 2359; Me, H, O, SEt, H, H, F, O], [AE ₂ 360; Me, H, O, CH ₂ F, H, H, F, O], [AE 2361; Me, H, O, CHF ₂ , H, H, F, O ], [AE2362; Me, H , O, CF 3, H, H, F, O], [AE2363; Me, H, O, OCH 2 F, H, H, F, O], [AE2364; Me, _{H, O, OCHF 2, H} , H, F, O], [AE2365; Me, H, O, OCF 3, H, H, F, O], [AE2366; Me, H, O, SCH 2 F, H, H, F, O] , [AE2367; Me, H, O, SCHF 2, H, H, F, O], [AE2368; Me, H, O, SCF 3, H, H, F, O] , [AE 2369; Me, H, O, CN, H, H , F, O], [AE 2370; Me, H, O, NO ₂ , H, F, O], [AE 2371; H, Me, O, H, H, H, F, O], [AE 2372; H, Me, O, F, H, F, O, [AE 2 373; H, Me, O, Cl, H, H, F, O], [AE 2 374; H, Me, O, Br, H, H, F, O], [AE 2 375; H, Me, O, I, H, H, F, O], [AE 2 376; H, Me, O, Me, H, H, F, O], [AE 2 377; H, Me, O, Et, H, F, O], [AE 2378; H, Me, O, Pr, H, H, F, O], [AE 2379; H, Me, O, i-Pr, H, H, F, O], [AE 2 380; H, Me, O, CH = CH ₂ , H, H, F, O], [AE 2 381; H, Me, O, C (Me) = CH ₂ , H H, F, O], [AE2382; H, Me, O, C≡CH, H, H, F, O], [AE 2383; H, Me, O, C≡CMe, H, H, F, O H, Me, O, c-Pr, H, H, F, O], [AE 2385; H, Me, O, OMe, H, H, F, O], [AE 2386; H, Me] , O, OEt, H, H, F, O], [AE2387; H, Me, O, Oi-Pr, H, H, F, O], [AE 2388; H, Me, O, SMe, H, H , F, O], [AE 2 389; H, Me, O, SE t, H, H, F, O], [AE ₂ 390; H, Me, O, CH ₂ F, H, H, F, O], [AE 239 1 ; H, Me, O, CHF 2, H, H, F, O], [AE2392; H, Me, O, CF 3, H, H, F, O], [AE2393; H, Me, O, OCH ₂ F, H, H, F, O], [AE 2394; H, Me, O, OCHF ₂ , H, H, F, O], [AE 2395; H, Me, O, OCF ₃ , H, H, F , O], [AE2396; H , Me, O, SCH 2 F, H, H, F, O], [AE2397; H, Me, O, SCHF 2, H, H, F, O], [AE2398; H, Me, O, SCF ₃ , H, H, F, O], [AE 2399; H, Me, O, CN, H, H, F, O], [AE 2400; H, Me, O, NO ₂ , H, H, F, O],

[AE 2401; F, H, O, H, H, H, F, O], [AE 2402; F, H, O, F, H, F, H, F, O], [AE 2403, F, H, O, Cl , H, H, F, O], [AE 2 404; F, H, O, Br, H, F, O], [AE 2 405; F, H, O, I, H, H, F, O], [AE2406; F, H, O, Me, H, H, F, O], [AE 2407; F, H, O, Et, H, F, O], [AE 2408; F, H, O, Pr , H, H, F, O ], [AE2409; F, H, O, i-Pr, H, H, F, O], [AE2410; F, H, O, CH = CH 2, H, H, F, O], [AE2411; F, H, O, C (Me) = CH 2, H, H, F, O], [AE2412; F, H, O, C≡CH, H, H, F, O], [AE 2413; F, H, O, C≡CMe, H, H, F, O], [AE 2414; F, H, O, c-Pr, H, H, F, O], [AE 2415; F, H, O, OMe, H, H, F, O], [AE 2416; F, H, O, OEt, H, H, F, O], [AE 24 17; F, H, O, Oi-Pr, H, H, F, O], [AE2418; F, H, O, SMe, H, H, F, O], [AE 2419; F, H, O, SEt, H, H, F, O], [ AE2420; F, H, O, CH 2 F, H, H, F, O], [AE2421; F, H, O, CHF 2, H, H, F, O], [AE2422; F, H, O , CF ₃ , H, H, F, O], [AE 2423; F, H, O, OCH ₂ F, H, H, F, O], [AE 2424; F, H, O, OCHF ₂ , H, H , F, O], [AE 2425; F, H, O, OCF ₃ , H, F, O], [AE 2426; F, H, O, SCH ₂ F, H, F, O], [ AE 2427; F, H, O, SCHF ₂ , H, H, F, O], [AE 2428; F, H, O, SCF ₃ , H, H, F, O], [AE 2429; F, H, O, CN, H, H, F, O], [AE 2430; F, H, O, NO ₂ , H, H, F, O], [AE 2431; H, F, O, H, H, H, F, O H, F, O, F, H, F, O], [AE 2433; H, F, O, Cl, H, F, O], [AE 2434; H, F, O] , Br, H, H, F, O], [AE 2435; H, F, O, I, H, H, F, O], [AE 2436; H, F, O, Me, H, H, F, O], [AE2437; H, F, O, Et, H, F, O], [AE 2438; H, F, O, Pr, H, H, F, O], [AE 2439; H, F, O, i- Pr, H, H, F, O], [AE2440; H, F, O, CH = CH 2, H, H, F, O], [AE2441; H, F, O , C (Me) = CH ₂ , H, H, F, O], [AE2442; H, F, O, C≡CH, H, H, F, O], [AE 2443; H, F, O, C ≡CMe, H, H, F, O], [AE 2444; H, F, O, c-Pr, H, H, F, O], [AE 2445; H, F, O, OMe, H, H, F H, F, O, OEt, H, H, F, O], [AE 2447; H, F, O, Oi-Pr, H, H, F, O], [AE 2448; H , F, O, SMe, H, H, F, O], [AE 2449; H, F, O, SE t, H, H, F, O], [AE 2450; H, F, O, CH ₂ F, H , H, F, O], [AE2451; H, F, O, CHF 2, H, H, F, O], [AE2452; H, F, O, CF 3, H, H, F, O], [AE2453; H, F, O , OCH 2 F, H, H, F, O], [AE2454; H, F, O, OCHF 2, H, H, F, O], [AE2455; H, F, _{O, OCF 3, H, H} , F, O], [AE2456; H, F, O, SCH 2 F, H, H, F, O], [AE2457; H, F, O, SCHF 2, H, H, F, O], [AE 2458; H, F, O, SCF ₃ , H, H, F, O], [AE 2459; H, F, O, CN, H, H, F, O], [AE 2460 H, F, O, NO ₂ , H, H, F, O], [AE2461; H, H, O, H, H, H, H, S], [AE 2462; H, H, O, F, H, H, H, S], [AE 2463; H, H, O, Cl, H, H, S], [AE 2464; H, H, O, Br, H, H, H, S], [ H, H, O, I, H, H, H, S], [AE 2466; H, H, O, Me, H, H, H, S], [AE 2467; H, H, O, Et, H, H, H, S], [AE 2468; H, H, O, Pr, H, H, H, S], [AE 2469; H, H, O, i-Pr, H, H, H, S] , [AE 2 470; H, H, O, CH = CH ₂ , H, H, H, S], [AE 2471; H, H, O, C (Me) = CH ₂ , H , H, H, S], [AE2472; H, H, O, C≡CH, H, H, H, S], [AE 2473; H, H, O, C≡ C Me, H, H, H, S H, H, O, c-Pr, H, H, H, S], [AE 2475; H, H, O, OMe, H, H, H, S], [AE 2476; H, H] , O, OEt, H, H, H, S], [AE2477; H, H, O, Oi-Pr, H, H, H, S], [AE 2478; H, H, O, SMe, H, H , H, S], [AE2479 ; H, H, O, SEt, H, H, H, S], [AE2480; H, H, O, CH 2 F, H, H, H, S], [AE2481 ; H, H, O, CHF 2, H, H, H, S], [AE2482; H, H, O, CF 3, H, H, H, S], [AE2483; H, H, O, OCH ₂ F, H, H, H, S], [AE 2484; H, H, O, OCHF ₂ , H, H, H, S], [AE 2 485; H, H, O, OCF ₃ , H, H, H H, H, O, SCH ₂ F, H, H, H, S], [AE 2487; H, H, O, SCHF ₂ , H, H, H, S], [AE 2 488; _{H, H, O, SCF 3} , H, H, H, S], [AE2489; H, H, O, CN, H, H, H, S], [AE2490; H, H, O, NO 2, H, H, H, S], [AE2491; Me, H, O, H, H, H, H, S], [AE2492; Me, H, O, F, H, H, H, S], [A AE 2493; Me, H, O, Cl, H, H, H, S], [AE2494; Me, H, O, Br, H, H, H, S], [AE 2495; Me, H, O, I, H, H, H, S], [AE 2496; Me, H, O, Me, H, H, H, S], [AE 2497; Me, H, O, Et, H, H, H, S], [ AE 2498; Me, H, O, Pr, H, H, H, S], [AE 2499; Me, H, O, i-Pr, H, H, H, S], [AE 2500] Me, H, O, CH = CH ₂ , H, H, H, S],

[AE2501; Me, H, O , C (Me) = CH 2, H, H, H, S], [AE2502; Me, H, O, C≡CH, H, H, H, S], [AE2503 Me, H, O, C≡CMe, H, H, H, S], [AE 2504; Me, H, O, c-Pr, H, H, H, S], [AE 2505; Me, H, O , OMe, H, H, H, S], [AE 2506; Me, H, O, OEt, H, H, H, S], [AE 2507; Me, H, O, Oi-Pr, H, H, H , S], [AE 2508; Me, H, O, SMe, H, H, H, S], [AE 2509; Me, H, O, SE t, H, H, H, S], [AE 2510; Me, H _{, O, CH 2 F, H} , H, H, S], [AE2511; Me, H, O, CHF 2, H, H, H, S], [AE2512; Me, H, O, CF 3, H , H, H, S], [AE 2513; Me, H, O, OCH ₂ F, H, H, H, S], [AE 2514; Me, H, O, OCHF ₂ , H, H, H, S] , [AE2515; Me, H, O, OCF 3, H, H, H, S], [AE2516; Me, H, O, SCH 2 F, H, H, H, S], [AE2517; Me, H , O, SCHF ₂ , H, H, H, S], [AE 2518; Me, H, O, SCF ₃ , H, H, H, S], [AE 2519; Me, H, O, CN, H, H , H, S], [AE 2520; Me, H, O, NO ₂ , H, H, S], [AE 2521; H, Me, O, H, H, H, H, S], [AE 2522; H, Me, O, F, H, H, H, S], [AE2523; H, Me, O, Cl, H, H, H, S], [AE 2524; H, Me, O, Br, H, H, H, S], [AE 2525; H, Me, O, I, H, H, H, S], [AE 2526; H, Me, O, Me, H, H, H, S], [AE 2 527; H, Me, O, Et, H, H, H, S], [AE 2528; H, Me, O, Pr, H, H, H, S], [AE 2529; H, Me, O, i-Pr, H, H, H, S] , [AE2530; H, Me, O, CH = CH 2, H, H, H, S], [AE2531; H, Me, O, C (Me) = CH 2, H H, H, S], [AE 2532; H, Me, O, C≡CH, H, H, H, S], [AE 2533; H, Me, O, C≡ C Me, H, H, H, S ], [AE2534; H, Me, O, c- Pr, H, H, H, S], [AE 2535; H, Me, O, OMe, H, H, H, S], [AE 2536; H, Me, O, OEt, H, H, H, S] H, Me, O, Oi-Pr, H, H, H, S], [AE 2538; H, Me, O, SMe, H, H, H, S], [AE 2539; H, Me, O, SEt, H, H, H, S], [AE 2540; H, Me, O, CH ₂ F, H, H, H, S], [AE 2541; H, Me, O, CHF ₂ , H, H , H, S], [AE2542 ; H, Me, O, CF 3, H, H, H, S], [AE2543; H, Me, O, OCH 2 F, H, H, H, S], [ AE2544; H, Me, O, OCHF 2, H, H, H, S], [AE2545; H, Me, O, OCF 3, H, H, H, S], [AE2546; H, Me, O, SCH ₂ F, H, H, H, S], [AE 2547; H, Me, O, SCHF ₂ , H, H, H, S], [AE 2548; H, Me, O, SCF ₃ , H, H, H, S], [AE 2 549; H, Me, O, CN, H, H, H, S], [AE 2550; H, Me, O, NO ₂ , H, H, H, S], [AE 2551; F , H, O, H, H, H, H, S], [AE2552; F, H, O, F, H, H, H, S], [AE 2553; F, H, O, Cl, H, H , H, S], [AE 2554; F, H, O, Br, H, H, S], [AE 2 555; F, H, O, I, H, H, H, S], [AE 2 556; F , H, O, Me, H, H, H, S], [AE 2 557; F, H, O, Et, H, H, H, S], [AE 2 558; F, H, O, Pr, H, H , H, S], [AE2559 ; F, H, O, i-Pr, H, H, H, S], [AE2560; F, H, O, CH = CH 2, H, H, H, S] , [AE 2561; F, H, O, C (Me) = CH ₂ , H, H, H, S], [AE 2562; F, H, O, C≡CH, H, H, H, S], [A AE 2563; F, H, O, C≡CMe, H, H, H, S], [AE 2564; F, H, O, c-Pr, H, H, H, S], [AE 2565; F, H, O, OMe, H, H, H, S], [AE 2566; F, H, O, OEt, H, H, H, S], [AE 2 567; F, H, O, Oi-Pr, H, H, H, S], [AE 2568; F, H, O, SMe, H, H, H, S], [AE 2569; F, H, O, SEt, H, H, H, S], [AE 2570; F, H, O, CH ₂ F, H, H, H, S], [AE 2571; F, H, O, CHF ₂ , H, H, H, S ], [AE2572; F, H, O, CF 3, H, H, H, S], [AE2573; F, H, O, OCH 2 F, H, H, H, S], [AE2574; F, H, O, OCHF 2, H, H, H, S], [AE2575; F, H, O, OCF 3, H, H, H, S], [AE2576; F, H, O, SCH ₂ F, H, H, H, S, [AE 2577; F, H, O, SCHF ₂ , H, H, H, S], [AE 2578; F, H, O, SCF ₃ , H, H, H, S], [AE 2579; F, H, O, CN, H, H, H, S], [AE 2580; F, H, O, NO ₂ , H, H, H, S], [AE 2581; H, F, O, H, H, H, H, S], [AE 2582; H, F, O, F, H, H, H, S], [AE 2583; H, F, O, Cl H, H, H, S], [AE 2584; H, F, O, Br, H, H, H, S], [AE 2585; H, F, O, I, H, H, H, S], [AE 2586; H, F, O, Me, H, H, H, S], [AE 2587; H, F, O, Et, H, H, H, S], [AE 2588; H, F, O, Pr , H, H, H, S ], [AE2589; H, F, O, i-Pr, H, H, H, S], [AE2590; H, F, O, CH = CH 2, H, H, H, S], [AE2591; H, F, O, C (Me) = CH 2, H, H, H, S], [AE2592; H, F, O, C≡CH, H, H, H, S, [AE 2593; H, F, O, C≡CMe, H, H, H, S], [AE 2594; H, F, O, c-Pr, H, H, H, S], [AE 2595; H, F, O, OMe, H, H, H, S], [AE 2596; H, F, O, OEt, H, H, H, S], [AE 2597; H, F, O, Oi-Pr, H, H, H, S], [AE 2598; H, F, O, S Me, H, H, H, S], [AE 2 599; H, F, O, SE t, H, H, H, S], [ AE 2600; H, F, O, CH ₂ F, H, H, H, S],

[AE2601; H, F, O , CHF 2, H, H, H, S], [AE2602; H, F, O, CF 3, H, H, H, S], [AE2603; H, F, O , OCH ₂ F, H, H, H, S], [AE 2604; H, F, O, OCHF ₂ , H, H, H, S], [AE 2605; H, F, O, OCF ₃ , H, H , H, S], [AE 2606; H, F, O, SCH ₂ F, H, H, H, S], [AE 2607; H, F, O, SCHF ₂ , H, H, H, S], [ H, F, O, SCF ₃ , H, H, H, S], [AE 2609; H, F, O, CN, H, H, H, S], [AE 2610; H, F, O, NO ₂ , H, H, H, S].

[Substituent number (ME2); E ¹⁰⁵ ], [BE 1; 2-Py], [BE 2; 3-F-2-Py], [BE 3; 4-Cl-3-F-2-Py], [BE 4 5-Cl-3-F-2-Py !, [BE5; 6-Cl-3-F-2-Py], [BE6; 4-Me-3-F-2-Py], [BE7; -Me-3-F-2- Py], [BE8; 6-Me-3-F-2-Py], [BE9; 4-CF 3 -3-F-2-Py], [BE10; 5- _{CF 3 -3-F-2-} Py], [BE11; 6-CF 3 -3-F-2-Py], [BE12; 4-CN-3-F-2-Py], [BE13; 5- CN-3-F-2-Py !, [BE14; 6-CN-3-F-2-Py], [BE15; 4-OMe-3-F-2-Py], [BE16; 5-OMe- 3-F-2-Py], [BE17; 6-OMe-3-F-2-Py], [BE18; 4-F-2-Py], [BE19; 3-Cl-4-F-2- Py], [BE20; 5-Cl-4-F-2-Py], [BE21; 6-Cl-4-F-2-Py], [BE22; 3-Me-4-F-2-Py] , [BE23; 5-Me- 4-F-2-Py], [BE24; 6-Me-4-F-2-Py], [BE25; 3-CF 3 -4-F-2-Py], _{[BE26; 5-CF 3 -4} -F-2-Py], [BE27; 6-CF 3 -4-F-2-Py], [BE28; 3-CN-4-F-2-Py], [BE29; 5-CN-4-F-2-Py], [BE30; 6-CN-4-F-2-Py], [BE31; 3-OMe-4-F-2-Py], [BE32 5-OMe-4-F-2-Py !, [BE 33; 6-OMe-4-F-2-Py], [BE 34; 5-F-2-Py], [BE 35; 3-Cl-5 -F-2-Py], [BE36; 4-Cl-5-F-2-Py], [BE 37; 6-Cl-5-F-2-Py], [BE 38; 3-Me-5-F -2-Py !, [BE 39; 4-Me-5-F-2-Py], [BE 40; 6-Me-5-F-2-Py], [BE 41; 3-CF ₃ -5-F- 2-Py], [BE42; 4-CF 3 -5-F-2-Py], [BE43; 6-CF 3 -5-F-2-Py], [BE44; 3-CN-5-F- 2-Py], [BE 45; 4-CN-5-F-2-Py], [BE 46; 6-CN-5-F-2-Py ], [BE 47; 3-OMe-5-F-2-Py], [BE 48; 4-OMe-5-F-2-Py], [BE 49; 6-OMe-5-F-2-Py], [BE50; 6-F-2-Py], [BE 51; 3-Cl-6-F-2-Py], [BE 52; 4-Cl-6-F-2-Py], [BE 53; 5-Cl -6-F-2-Py], [BE 54; 3-Me-6-F-2-Py], [BE 55; 4-Me-6-F-2-Py], [BE 56; 5-Me-6 -F-2-Py], [ BE57; 3-CF 3 -6-F-2-Py], [BE58; 4-CF 3 -6-F-2-Py], [BE59; 5-CF 3 - 6-F-2-Py], [BE60; 3-CN-6-F-2-Py], [BE61; 4-CN-6-F-2-Py], [BE62; 5-CN-6- F-2-Py !, [BE63; 3-OMe-6-F-2-Py], [BE64; 4-OMe-6-F-2-Py], [BE65; 5-OMe-6-F- 2-Py], [BE66; 3-Cl-2-Py], [BE 67; 4-Cl-3-Cl-2-Py], [BE 68; 5-Cl-3-Cl-2-Py], [BE 66] BE69; 6-Cl-3-Cl-2-Py], [BE70; 4-Me-3-Cl-2-Py], [BE71; 5-Me-3-Cl-2-Py], [BE 72; 6-Me-3-Cl-2-Py !, [BE 73; 4-CF ₃ -3-Cl-2-Py], [BE 74; 5-CF ₃ -3-Cl-2-Py], [BE 75; _{6-CF 3 -3-Cl-} 2-Py], [BE76; 4-CN-3-Cl-2-Py], [BE77; 5-CN-3-Cl-2-Py], [BE78; 6 -CN-3-Cl-2-Py], [BE 79; 4-OMe-3-Cl-2-Py], [BE 80; 5-OMe-3-Cl-2-Py], [BE 81; 6-OMe -3-Cl-2-Py !, [BE 82; 4-Cl-2-Py], [BE 83; 3-Cl-4-Cl-2-Py], [BE 84; 5-Cl-4-Cl-2 -Py], [BE 85; 6-Cl-4-Cl-2-Py], [BE 86; 3-Me-4-Cl-2-Py], [BE 87; 5-Me-4-Cl-2-Py ], [BE 88; 6-Me-4-Cl-2-Py], [BE 89; 3-CF ₃ -4-Cl-2-Py], [BE 90; 5-CF ₃ -4-Cl-2-Py] ], [BE 91; 6-CF ₃ -4-Cl-2-Py], [BE 92; 3-CN-4-Cl-2-Py], [BE93; 5-CN-4-Cl-2-Py], [BE94; 6-CN-4-Cl-2-Py], [BE95; OMe-4-Cl-2-Py], [BE96; 5-OMe-4-Cl-2-Py], [BE97; 6-OMe-4-Cl-2-Py], [BE98; 5-Cl- 2-Py], [BE 99; 4-Cl-5-Cl-2-Py], [BE 100; 5-Cl-5-Cl-2-Py], [BE 101; 6-Cl-5-Cl-2- Py],

[BE102; 4-Me-5-Cl-2-Py], [BE103; 5-Me-5-Cl-2-Py], [BE104; 6-Me-5-Cl-2-Py], [BE105] _{; 4-CF 3 -5-Cl} -2-Py], [BE106; 5-CF 3 -5-Cl-2-Py], [BE107; 6-CF 3 -5-Cl-2-Py], [ BE108; 4-CN-5-Cl-2-Py], [BE109; 3-CN-5-Cl-2-Py], [BE110; 6-CN-5-Cl-2-Py], [BE111; 4-OMe-5-Cl-2-Py], [BE112; 5-OMe-5-Cl-2-Py], [BE113; 6-OMe-5-Cl-2-Py], [BE114; 6- Cl-2-Py !, [BE115; 3-Cl-6-Cl-2-Py], [BE116; 4-Cl-6-Cl-2-Py], [BE117; 5-Cl-6-Cl- 2-Py], [BE118; 3-Me-6-Cl-2-Py], [BE119; 4-Me-6-Cl-2-Py], [BE120; 5-Me-6-Cl-2- Py], [BE121; 3- CF 3 -6-Cl-2-Py], [BE122; 4-CF 3 -6-Cl-2-Py], [BE123; 5-CF 3 -6-Cl-2 -Py], [BE124; 3-CN-6-Cl-2-Py], [BE 125; 4-CN-6-Cl-2-Py], [BE 126; 5-CN-6-Cl-2-Py ], [BE 127; 3-OMe-6-Cl-2-Py], [BE 128; 4-OMe-6-Cl-2-Py], [BE 129; 5-OMe-6-Cl-2-Py], [BE130; 3-Br-2-Py], [BE 131; 4-Cl-3-Br-2-Py], [BE 132; 5-Cl-3-Br-2-Py], [BE 133; 6-Cl -3-Br-2-Py !, [BE 134; 4-Me-3-Br-2-Py], [BE 135; 5-Me-3-Br-2-Py], [BE 136; 6-Me-3 -Br-2-Py], [ BE137; 4-CF 3 -3-Br-2-Py], [BE138; 5-CF 3 -3-Br-2-Py], [BE139; 6-CF 3 - 3-Br-2-Py], [BE140; 4-CN-3-Br-2-Py], [BE141; 5-CN-3-Br-2-Py], [BE142; 6-CN-3- Br-2-Py, [BE 143; 4-OMe-3-Br-2-Py], [BE 144; 5-O Me-3-Br-2-Py, [BE 145; 6-OMe-3-Br-2-Py], [BE 146; 4-Br-2-Py], [BE 147; 3-Cl-4-Br- 2-Py], [BE148; 5-Cl-4-Br-2-Py], [BE149; 6-Cl-4-Br-2-Py], [BE150; 3-Me-4-Br-2- Py], [BE151; 5- Me-4-Br-2-Py], [BE152; 6-Me-4-Br-2-Py], [BE153; 3-CF 3 -4-Br-2-Py ], [BE154; 5-CF 3 -4-Br-2-Py], [BE155; 6-CF 3 -4-Br-2-Py], [BE156; 3-CN-4-Br-2-Py ], [BE157; 5-CN-4-Br-2-Py], [BE158; 6-CN-4-Br-2-Py], [BE159; 3-OMe-4-Br-2-Py], [BE160; 5-OMe-4-Br-2-Py], [BE161; 6-OMe-4-Br-2-Py], [BE162; 5-Br-2-Py], [BE163; 3-Cl -5-Br-2-Py !, [BE 164; 4-Cl-5-Br-2-Py], [BE 165; 6-Cl-5-Br-2-Py], [BE 166; 3-Me-5 -Br-2-Py], [BE 167; 4-Me-5-Br-2-Py], [BE 168; 6-Me-5-Br-2-Py], [BE 169; 3-CF ₃ -5-] Br-2-Py], [ BE170; 4-CF 3 -5-Br-2-Py], [BE171; 6-CF 3 -5-Br-2-Py], [BE172; 3-CN-5- Br-2-Py, [BE 173; 4-CN-5-Br-2-Py], [BE 174; 6-CN-5-Br-2-Py], [BE 175; 3-OMe-5-Br- 2-Py], [BE 176; 4-OMe-5-Br-2-Py], [BE 177; 6-OMe-5-Br-2-Py], [BE 178; 6-Br-2-Py], BE 179; 3-Cl-6-Br-2-Py], [BE 180; 4-Cl-6-Br-2-Py], [BE 181; 5-Cl-6-Br-2-Py], [BE 182; 3-Me-6-Br-2-Py], [BE183; 4-Me-6-Br-2-Py], [BE184; 5-Me-6-Br-2-Py], [BE185; _{CF 3 -6-Br-2-} Py], [BE186; 4-CF 3 -6-Br-2-Py], [BE1 _{87; 5-CF 3 -6-} Br-2-Py], [BE188; 3-CN-6-Br-2-Py], [BE189; 4-CN-6-Br-2-Py], [BE190 5-CN-6-Br-2-Py !, [BE191; 3-OMe-6-Br-2-Py], [BE192; 4-OMe-6-Br-2-Py], [BE193; -OMe-6-Br-2-Py], [BE194; 3-I-2-Py], [BE195; 4-Cl-3-I-2-Py], [BE196; 5-Cl-3-I -2-Py !, [BE 197; 6-Cl-3-I-2-Py], [BE 198; 4-Me-3-I-2-Py], [BE 199; 5-Me-3-I-2 -Py], [BE200; 6- Me-3-I-2-Py], [BE201; 4-CF 3 -3-I-2-Py],

_{[BE202; 5-CF 3 -3} -I-2-Py], [BE203; 6-CF 3 -3-I-2-Py], [BE204; 4-CN-3-I-2-Py], [BE205; 5-CN-3-I-2-Py], [BE206; 6-CN-3-I-2-Py], [BE207; 4-OMe-3-I-2-Py], [BE208 5-OMe-3-I-2-Py !, [BE 209; 6-OMe-3-I-2-Py], [BE 210; 4-I-2-Py], [BE 211; 3-Cl-4 -I-2-Py, [BE 212; 5-Cl-4-I-2-Py], [BE 213; 6-Cl-4-I-2-Py], [BE 214; 3-Me-4-I -2-Py], [BE 215; 5-Me-4-I-2-Py], [BE 216; 6-Me-4-I-2-Py], [BE 217; 3-CF ₃ -4-I- 2-Py], [BE218; 5-CF 3 -4-I-2-Py], [BE219; 6-CF 3 -4-I-2-Py], [BE220; 3-CN-4-I- 2-Py], [BE221; 5-CN-4-I-2-Py], [BE222; 6-CN-4-I-2-Py], [BE223; 3-OMe-4-I-2-] Py], [BE224; 5-OMe-4-I-2-Py], [BE225; 6-OMe-4-I-2-Py], [BE226; 5-I-2-Py], [BE227; 3-Cl-5-I-2-Py], [BE 228; 4-Cl-5-I-2-Py], [BE 229; 6-Cl-5-I-2-Py], [BE 230; Me-5-I-2-Py], [BE 231; 4-Me-5-I-2-Py], [BE 232; 6-Me-5-I-2-Py], [BE 233; 3-CF ₃ -5-I-2-Py, [BE 234; 4-CF ₃ -5-I-2-Py], [BE 235; 6-CF ₃ -5-I-2-Py], [BE 236; 3-CN -5-I-2-Py], [BE 237; 4-CN-5-I-2-Py], [BE 238; 6-CN-5-I-2-Py], [BE 239; 3-OMe-5 -I-2-Py, [BE240; 4-OMe-5-I-2-Py], [BE241; 6-OMe-5-I-2-Py], [BE 242; 6-I-2-Py ], [BE 243; 3-Cl-6-I-2-Py], [BE 244; 4-Cl-6-I-2-Py], [BE 245; 5-Cl-6-I-2-Py], [BE 246; 3-Me-6- I-2-Py], [BE 247; 4-Me-6-I-2-Py], [BE 248; 5-Me-6-I-2-Py], [BE 249; 3-CF ₃ -6- I -2-Py !, [BE 250; 4-CF ₃ -6-I-2-Py], [BE 251; 5-CF ₃ -6-I-2-Py], [BE 252; 3-CN-6-I -2-Py], [BE253; 4-CN-6-I-2-Py], [BE254; 5-CN-6-I-2-Py], [BE255; 3-OMe-6-I-2 -Py], [BE256; 4-OMe-6-I-2-Py], [BE257; 5-OMe-6-I-2-Py], [BE258; 3-Me-2-Py], [BE259] 4-Cl-3-Me-2-Py !, [BE 260; 5-Cl-3-Me-2-Py], [BE 261; 6-Cl-3-Me-2-Py], [BE 262; -Me-3-Me-2-Py], [BE263; 5-Me-3-Me-2-Py], [BE264; 6-Me-3-Me-2-Py], [BE 265; 4-CF _{3 -3-Me-2-Py} ], [BE266; 5-CF 3 -3-Me-2-Py], [BE267; 6-CF 3 -3-Me-2-Py], [BE268; 4- CN-3-Me-2-Py !, [BE 269; 5-CN-3-Me-2-Py], [BE 270; 6-CN-3-Me-2-Py], [BE 271; 4-OMe- 3-Me-2-Py, [BE 272; 5-OMe-3-Me-2-Py], [BE 273; 6-OMe-3-Me-2-Py], [BE 274; 4-Me-2- Py], [BE 275; 3-Cl-4-Me-2-Py], [BE 276; 5-Cl-4-Me-2-Py], [BE 277; 6-Cl-4-Me-2-Py] , [BE 278; 3-Me-4-Me-2-Py], [BE 279; 5-Me-4-Me-2-Py], [BE 280; 6-Me-4-Me-2-Py], [BE BE 281; 3-CF ₃ -4-Me-2-Py !, [BE 282; 5-CF ₃ -4-Me-2-Py], [BE 283; 6-CF ₃ -4-Me-2-Py], [BE284; 3-CN-4-Me-2-Py], [BE 285; 5-CN-4-Me-2-Py], [BE 286; 6-CN-4-Me-2-Py], [BE 287] 3-OMe-4-Me-2-Py], [BE 288; 5-OMe-4-Me-2-Py], [BE 289; 6-OMe -4-Me-2-Py], [BE 290; 5-Me-2-Py], [BE 291; 3-Cl-5-Me-2-Py], [BE 292; 4-Cl-5-Me-2 -Py], [BE293; 6-Cl-5-Me-2-Py], [BE 294; 3-Me-5-Me-2-Py], [BE 295; 4-Me-5-Me-2-Py ], [BE296; 6-Me -5-Me-2-Py], [BE297; 3-CF 3 -5-Me-2-Py], [BE298; 4-CF 3 -5-Me-2-Py ], [BE299; 6-CF 3 -5-Me-2-Py], [BE300; 3-CN-5-Me-2-Py], [BE301; 4-CN-5-Me-2-Py] ,

[BE302; 6-CN-5-Me-2-Py], [BE303; 3-OMe-5-Me-2-Py], [BE304; 4-OMe-5-Me-2-Py], [BE305] 6-OMe-5-Me-2-Py], [BE306; 6-Me-2-Py], [BE 307; 3-Cl-6-Me-2-Py], [BE 308; 4-Cl-6 -Me-2-Py], [BE309; 5-Cl-6-Me-2-Py], [BE 310; 3-Me-6-Me-2-Py], [BE 311; 4-Me-6-Me -2-Py !, [BE 312; 5-Me-6-Me-2-Py], [BE 313; 3-CF ₃ -6-Me-2-Py], [BE 314; 4-CF ₃ -6-Me -2-Py !, [BE 315; 5-CF ₃ -6-Me-2-Py], [BE 316; 3-CN-6-Me-2-Py], [BE 317; 4-CN-6-Me- 2-Py], [BE 318; 5-CN-6-Me-2-Py], [BE 319; 3-OMe-6-Me-2-Py], [BE 320; 4-OMe-6-Me-2- 2 Py], [BE 321; 5-OMe-6-Me-2-Py], [BE 322; 3-OMe-2-Py], [BE 323; 4-Cl-3-OMe-2-Py], [BE 324; 5-Cl-3-OMe-2-Py, [BE 325; 6-Cl-3-OMe-2-Py], [BE 326; 4-Me-3-OMe-2-Py], [BE 327; Me-3-OMe-2-Py !, [BE 328; 6-Me-3-OMe-2-Py], [BE 329; 4-CF ₃ -3-OMe-2-Py], [BE 330; 5-CF ₃ -3-OMe-2-Py, [BE 331; 6-CF ₃ -3-OMe-2-Py], [BE 332; 4-CN-3-OMe-2-Py], [BE 333; 5-CN -3-OMe-2-Py !, [BE334; 6-CN-3-OMe-2-Py], [BE 335; 4-OMe-3-OMe-2-Py], [BE336; 5-OMe-3 -OMe-2-Py], [BE 337; 6-OMe-3-OMe-2-Py], [BE 338; 4-OMe-2-Py], [BE 339; 3-Cl-4-OMe-2-Py ], [BE340; 5-Cl-4-OMe-2-Py], [BE341; 6-Cl-4-OMe-2-Py], [BE342; 3-Me-4-OMe-2-Py], [BE 343; 5-Me-4-OMe-2-Py], [BE344; 6-Me-4 -OMe-2-Py], [BE345; 3-CF 3 -4-OMe-2-Py], [BE346; 5-CF 3 -4-OMe-2-Py], _{[BE347; 6-CF 3 -4} -OMe-2-Py], [BE348; 3-CN-4-OMe-2-Py], [BE349; 5-CN-4-OMe-2-Py], [ BE 350; 6-CN-4-OMe-2-Py], [BE 351; 3-OMe-4-OMe-2-Py], [BE 352; 5-OMe-4-OMe-2-Py], [BE 353; 6-OMe-4-OMe-2-Py], [BE 354; 5-OMe-2-Py], [BE 355; 3-Cl-5-OMe-2-Py], [BE 356; OMe-2-Py, [BE 357; 6-Cl-5-OMe-2-Py], [BE 358; 3-Me-5-OMe-2-Py], [BE 359; 4-Me-5-OMe- 2-Py], [BE360; 6-Me-5-OMe-2-Py], [BE361; 3-CF 3 -5-OMe-2-Py], [BE362; 4-CF 3 -5-OMe- 2-Py], [BE363; 6-CF 3 -5-OMe-2-Py], [BE364; 3-CN-5-OMe-2-Py], [BE365; 4-CN-5-OMe-2 -Py], [BE 366; 6-CN-5-OMe-2-Py], [BE 367; 3-OMe-5-OMe-2-Py], [BE 368; 4-OMe-5-OMe-2-Py ], [BE 369; 6-OMe-5-OMe-2-Py], [BE 370; 6-OMe-2-Py], [BE 371; 3-Cl-6-OMe-2-Py], [BE 372; 4] -Cl-6-OMe-2-Py], [BE 373; 5-Cl-6-OMe-2-Py], [BE 374; 3-Me-6-OMe-2-Py], [BE 375; -6-OMe-2-Py !, [BE 376; 5-Me-6-OMe-2-Py], [BE 377; 3-CF ₃ -6-OMe-2-Py], [BE 378; 4-CF ₃ -6-OMe-2-Py], [BE 379; 5-CF ₃ -6-OMe-2-Py], [BE 380; 3-CN-6-OMe-2-Py], [BE 381; 4-CN- 6-OMe-2-Py], [BE 382; 5-CN-6-OMe-2-Py], [BE 383; 3-OMe-6-OMe-2-Py], [BE 384; 4-OMe-6- O Me-2-Py], [ BE385; 5-OMe-6-OMe-2-Py], [BE386; 3-CF 3 -2-Py], [BE387; 4-Cl-3-CF 3 -2- Py], [BE388; 5- Cl-3-CF 3 -2-Py], [BE389; 6-Cl-3-CF 3 -2-Py], [BE390; 4-Me-3-CF 3 -2 5-Py], [BE 391; 5-Me-3-CF ₃ -2-Py], [BE 392; 6-Me-3-CF ₃ -2-Py], [BE 393; 4-CF ₃ -3-CF ₃ -2-Py], [BE 394; 5-CF ₃ -3-CF ₃ -2-Py], [BE 395; 6-CF ₃ -3-CF ₃ -2-Py], [BE 396; 4-CN-3 _{-CF 3 -2-Py], [} BE397; 5-CN-3-CF 3 -2-Py], [BE398; 6-CN-3-CF 3 -2-Py], [BE399; 4-OMe- _{3-CF 3 -2-Py]} , [BE400; 5-OMe-3-CF 3 -2-Py], [BE401; 6-OMe-3-CF 3 -2-Py],

_{[BE402; 4-CF 3 -2} -Py], [BE403; 3-Cl-4-CF 3 -2-Py], [BE404; 5-Cl-4-CF 3 -2-Py], [BE405; _{6-Cl-4-CF 3} -2-Py], [BE406; 3-Me-4-CF 3 -2-Py], [BE407; 5-Me-4-CF 3 -2-Py], [BE408 ; 6-Me-4-CF 3 -2-Py], [BE409; 3-CF 3 -4-CF 3 -2-Py], [BE410; 5-CF 3 -4-CF 3 -2-Py] _{, [BE411; 6-CF 3} -4-CF 3 -2-Py], [BE412; 3-CN-4-CF 3 -2-Py], [BE413; 5-CN-4-CF 3 -2- Py], [BE414; 6- CN-4-CF 3 -2-Py], [BE415; 3-OMe-4-CF 3 -2-Py], [BE416; 5-OMe-4-CF 3 -2 -Py], [BE417; 6- OMe-4-CF 3 -2-Py], [BE418; 5-CF 3 -2-Py], [BE419; 3-Cl-5-CF 3 -2-Py] , [BE420; 4-Cl- 5-CF 3 -2-Py], [BE421; 6-Cl-5-CF 3 -2-Py], [BE422; 3-Me-5-CF 3 -2-Py ], [BE423; 4-Me -5-CF 3 -2-Py], [BE424; 6-Me-5-CF 3 -2-Py], [BE425; 3-CF 3 -5-CF 3 -2 4-Py], [BE 426; 4-CF ₃ -5-CF ₃ -2-Py], [BE 427; 6-CF ₃ -5-CF ₃ -2-Py], [BE 428; ₃ -2-Py], [BE 429; 4-CN-5-CF ₃ -2-Py], [BE 430; 6-CN-5-CF ₃ -2-Py], [BE 431; 3-OMe -5-] CF ₃ -2-Py !, [BE 432; 4-OMe-5-CF ₃ -2-Py], [BE 433; 6-OMe -5-CF ₃ -2-Py], [BE 434; 6 CF _3- 2-Py], [BE435; 3-Cl-6-CF 3 -2-Py], [BE436; 4-Cl-6-CF 3 -2-Py], [BE437; 5-Cl-6-CF 3 -2-Py], [BE 438; 3-Me-6-CF ₃ -2-Py], [BE 439; 4-Me-6-CF ₃ -2-Py], [BE 440; 5-Me-6- CF 3 -2-Py], [BE441; 3-CF 3 -6-CF 3 -2-Py], [BE442; 4-CF 3 -6-CF 3 -2-Py ], [BE443; 5-CF 3 -6-CF 3 -2-Py], [BE444; 3-CN-6-CF 3 -2-Py], [BE445; 4-CN-6-CF 3 -2 -Py], [BE446; 5- CN-6-CF 3 -2-Py], [BE447; 3-OMe-6-CF 3 -2-Py], [BE448; 4-OMe-6-CF 3 - 2-Py], [BE449; 5-OMe-6-CF 3 -2-Py], [BE450; 3-OCF 3 -2-Py], [BE451; 4-Cl-3-OCF 3 -2-Py ], [BE452; 5-Cl -3-OCF 3 -2-Py], [BE453; 6-Cl-3-OCF 3 -2-Py], [BE454; 4-Me-3-OCF 3 -2- Py], [BE455; 5- Me-3-OCF 3 -2-Py], [BE456; 6-Me-3-OCF 3 -2-Py], [BE457; 4-CF 3 -3-OCF 3 - 2-Py], [BE 458; 5-CF ₃ -3-OCF ₃ -2-Py], [BE 459; 6-CF ₃ -3-OCF ₃ -2-Py], [BE 460; OCF ₃ -2-Py !, [BE 461; 5-CN-3-OCF ₃ -2-Py], [BE 462; 6-CN -3-OCF ₃ -2-Py], [BE 463; 4-OMe-3 _{-OCF 3 -2-Py], [} BE464; 5-OMe-3-OCF 3 -2-Py], [BE465; 6-OMe-3-OCF 3 -2-Py], [BE466; 4-OCF 3 -2-Py], [BE467; 3-Cl-4-OCF 3 -2-Py], [BE468; 5-Cl-4-OCF 3 -2-Py], [BE469; 6-Cl-4-OCF _{3 -2-Py], [BE470} ; 3-Me-4-OCF 3 -2-Py], [BE471; 5-Me-4-OCF 3 -2-Py], [BE472; 6-Me-4- OCF ₃ -2-Py !, [BE 473; 3-CF ₃ -4-OCF ₃ -2-Py], [BE 474; 5-CF ₃ -4-OCF ₃ -2-Py], [BE 475; 6-CF] ₃ -4-OCF ₃ -2-Py], [BE 476; 3-CN -4-OCF ₃ -2-Py !, [BE 477; 5-CN-4-OCF ₃ -2-Py], [BE 478; 6-CN-4-OCF ₃ -2-Py], [BE 479; 3-OMe -4- OCF ₃ -2-Py !, [BE 480; 5-OMe -4-OCF ₃ -2-Py], [BE 481; 6-OMe -4-OCF ₃ -2-Py], [BE 482; 5-OCF _3- 2-Py], [BE483; 3-Cl-5-OCF 3 -2-Py], [BE484; 4-Cl-5-OCF 3 -2-Py], [BE485; 6-Cl-5-OCF 3 -2-Py !, [BE 486; 3-Me-5-OCF ₃ -2-Py], [BE 487; 4-Me-5-OCF ₃ -2-Py], [BE 488; 6-Me-5-OCF ₃ -2-Py, [BE 489; 3-CF ₃ -5-OCF ₃ -2-Py], [BE 490; 4-CF ₃ -5-OCF ₃ -2-Py], [BE 491; 6-CF _{3 -5-OCF 3 -2-Py]} , [BE492; 3-CN-5-OCF 3 -2-Py], [BE493; 4-CN-5-OCF 3 -2-Py], [BE494; 6- _{CN-5-OCF 3 -2-} Py], [BE495; 3-OMe-5-OCF 3 -2-Py], [BE496; 4-OMe-5-OCF 3 -2-Py], [BE497; 6 _{-OMe-5-OCF 3 -2-} Py], [BE498; 6-OCF 3 -2-Py], [BE499; 3-Cl-6-OCF 3 -2-Py], [BE500; 4-Cl- _{6-OCF 3 -2-Py]} , [BE501; 5-Cl-6-OCF 3 -2-Py],

[BE502; 3-Me-6 -OCF 3 -2-Py], [BE503; 4-Me-6-OCF 3 -2-Py], [BE504; 5-Me-6-OCF 3 -2-Py] _{, [BE505; 3-CF 3} -6-OCF 3 -2-Py], [BE506; 4-CF 3 -6-OCF 3 -2-Py], [BE507; 5-CF 3 -6-OCF 3 - 2-Py], [BE508; 3-CN-6-OCF 3 -2-Py], [BE509; 4-CN-6-OCF 3 -2-Py], [BE510; 5-CN-6-OCF 3 -2-Py !, [BE 511; 3-OMe-6-OCF ₃ -2-Py], [BE 512; 4-OMe-6-OCF ₃ -2-Py], [BE 513; 5-OMe-6-OCF _{3 -2-Py], [BE514} ; 3-CHF 2 -2-Py], [BE515; 4-Cl-3-CHF 2 -2-Py], [BE516; 5-Cl-3-CHF 2 -2 -Py], [BE517; 6- Cl-3-CHF 2 -2-Py], [BE518; 4-Me-3-CHF 2 -2-Py], [BE519; 5-Me-3-CHF 2 - 2-Py], [BE520; 6-Me-3-CHF 2 -2-Py], [BE521; 4-CF 3 -3-CHF 2 -2-Py], [BE522; 5-CF 3 -3- _{CHF 2 -2-Py], [} BE523; 6-CF 3 -3-CHF 2 -2-Py], [BE524; 4-CN-3-CHF 2 -2-Py], [BE525; 5-CN- _{3-CHF 2 -2-Py]} , [BE526; 6-CN-3-CHF 2 -2-Py], [BE527; 4-OMe-3-CHF 2 -2-Py], [BE528; 5-OMe _{-3-CHF 2 -2-Py]} , [BE529; 6-OMe-3-CHF 2 -2-Py], [BE530; 4-CHF 2 -2-Py], [BE531; 3-Cl-4- _{CHF 2 -2-Py], [} BE532; 5-Cl-4-CHF 2 -2-Py], [BE533; 6-Cl-4-CHF 2 -2-Py], [BE534; 3-Me-4 _{-CHF 2 -2-Py], [} BE535; 5-Me-4-CHF 2 -2-Py], [BE536; 6-Me-4-CHF 2 -2-Py], [BE537; 3-CF 3 -4-CHF ₂ -2-Py], [BE 538; 5-CF ₃ -4-CHF ₂ -2-Py !, [BE 539; 6-CF ₃ -4-CHF ₂ -2-Py], [BE 540; 3-CN 4-CHF ₂ -2-Py], [BE 541; _{5-CN-4-CHF 2} -2-Py], [BE542; 6-CN-4-CHF 2 -2-Py], [BE543; 3-OMe-4-CHF 2 -2-Py], [BE544 ; 5-OMe-4-CHF 2 -2-Py], [BE545; 6-OMe-4-CHF 2 -2-Py], [BE546; 5-CHF 2 -2-Py], [BE547; 3- Cl-5-CHF ₂ -2-Py !, [BE 548; 4-Cl -5-CHF ₂ -2-Py], [BE 549; 6-Cl -5-CHF ₂ -2-Py], [BE 550; 3] -Me-5-CHF ₂ -2-Py, [BE 551; 4-Me-5-CHF ₂ -2-Py], [BE 552; 6-Me-5-CHF ₂ -2-Py], [BE 553; _{3-CF 3 -5-CHF 2} -2-Py], [BE554; 4-CF 3 -5-CHF 2 -2-Py], [BE555; 6-CF 3 -5-CHF 2 -2-Py] , [BE 556; 3-CN-5-CHF ₂ -2-Py], [BE 557; 4-CN -5-CHF ₂ -2-Py], [BE 558; 6-CN -5-CHF ₂ -2-Py ], [BE559; 3-OMe-5-CHF ₂ -2-Py], [BE 560; 4-OMe-5-CHF ₂ -2-Py], [BE 561; 6-OMe -5-CHF ₂ -2-] Py], [BE 562; 6-CHF ₂ -2-Py], [BE 563; 3-Cl-6-CHF ₂ -2-Py], [BE 564; 4-Cl 6-CHF ₂ -2-Py], [BE565; 5-Cl-6 -CHF 2 -2-Py], [BE566; 3-Me-6-CHF 2 -2-Py], [BE567; 4-Me-6-CHF 2 -2-Py] , [BE568; 5-Me- 6-CHF 2 -2-Py], [BE569; 3-CF 3 -6-CHF 2 -2-Py], [BE570; 4-CF 3 -6-CHF 2 -2 -Py], [BE571; 5- CF 3 -6-CHF 2 -2-Py], [BE572; 3-CN-6-CHF 2 -2-Py], [BE573; 4-CN-6-CHF 2 -2-Py], [BE 574; 5-CN-6-CHF ₂ -2-Py !, [BE 575; 3-OMe-6-CHF ₂ -2-Py], [BE 576; 4-OMe-6-CHF ₂ -2-Py], [BE 577; 5-OMe-6-CHF _{2 -2-Py], [BE578} ; 3-OCHF 2 -2-Py], [BE579; 4-Cl-3-OCHF 2 -2-Py], [BE580; 5-Cl-3-OCHF 2 -2 -Py], [BE581; 6- Cl-3-OCHF 2 -2-Py], [BE582; 4-Me-3-OCHF 2 -2-Py], [BE583; 5-Me-3-OCHF 2 - 2-Py], [BE 584; 6-Me-3-OCHF ₂ -2-Py], [BE 585; 4-CF ₃ -3-OCHF ₂ -2-Py], [BE 586; 5-CF ₃ -3- _{OCHF 2 -2-Py], [} BE587; 6-CF 3 -3-OCHF 2 -2-Py], [BE588; 4-CN-3-OCHF 2 -2-Py], [BE589; 5-CN- 3-OCHF ₂ 2-Py], [BE 590; 6-CN-3-OCHF ₂ 2-Py], [BE 591; 4-OMe 3-OCHF ₂ 2-Py], [BE 592; 5-OMe _{-3-OCHF 2 -2-Py]} , [BE593; 6-OMe-3-OCHF 2 -2-Py], [BE594; 4-OCHF 2 -2-Py], [BE595; 3-Cl-4- _{OCHF 2 -2-Py], [} BE596; 5-Cl-4-OCHF 2 -2-Py], [BE597; 6-Cl-4-OCHF 2 -2-Py], [BE598; 3-Me-4 _{-OCHF 2 -2-Py], [} BE599; 5-Me-4-OCHF 2 -2-Py], [BE600; 6-Me-4-OCHF 2 -2-Py], [BE601; 3-CF 3 -4-OCHF ₂ -2-Py],

_{[BE602; 5-CF 3 -4} -OCHF 2 -2-Py], [BE603; 6-CF 3 -4-OCHF 2 -2-Py], [BE604; 3-CN-4-OCHF 2 -2- Py], [BE605; 5- CN-4-OCHF 2 -2-Py], [BE606; 6-CN-4-OCHF 2 -2-Py], [BE607; 3-OMe-4-OCHF 2 -2 -Py], [BE608; 5- OMe-4-OCHF 2 -2-Py], [BE609; 6-OMe-4-OCHF 2 -2-Py], [BE610; 5-OCHF 2 -2-Py] , [BE 611; 3-Cl-5-OCHF ₂ -2-Py], [BE 612; 4-Cl -5-OCHF ₂ -2-Py], [BE 613; 6-Cl -5-OCHF ₂ -2-Py ], [BE 614; 3-Me-5-OCHF ₂ -2-Py], [BE 615; 4-Me-5-OCHF ₂ -2-Py], [BE 616; 6-Me-5-OCHF ₂ -2-] Py], [BE 617; 3-CF ₃ -5-OCHF ₂ -2-Py], [BE 618; 4-CF ₃ -5-OCHF ₂ -2-Py], [BE 619; 6-CF ₃ -5-OCHF _{2 -2-Py], [BE620} ; 3-CN-5-OCHF 2 -2-Py], [BE621; 4-CN-5-OCHF 2 -2-Py], [BE622; 6-CN-5- OCHF ₂ -2-Py !, [BE 623; 3-OMe-5-OCHF ₂ -2-Py], [BE 624; 4-OMe-5-OCHF ₂ -2-Py], [BE 625; 6-OMe-5] -OCHF ₂ -2-Py], [BE 626; 6-OCHF ₂ -2-Py], [BE 627; 3-Cl-6-OCHF ₂ -2-Py], [BE 628; 4-Cl -6-OCHF ₂ -2-Py !, [BE 629; 5-Cl-6-OCHF ₂ -2-Py], [BE 630; 3-Me-6-OCHF ₂ -2-Py], [BE 631; 4-Me-6-OCHF ₂ -2-Py !, [BE 632; 5-Me-6-OCHF ₂ -2-Py], [BE 633; 3-CF ₃ -6-OCHF ₂ -2-Py], [BE 634; 4-CF _3- 6-OCHF ₂ -2-Py], [BE 635; 5-CF ₃ -6-OCHF ₂ -2-Py], [BE 636; 3-CN 6-OCHF ₂ -2-Py], [BE637; 4-CN-6 -OCHF 2 -2-Py], [BE638; 5-CN-6-OCHF 2 -2-Py], [BE639; 3-OMe-6-OCHF 2 -2-Py] , [BE 640; 4-OMe-6-OCHF ₂ -2-Py], [BE 641; 5-OMe -6-OCHF ₂ -2-Py], [BE 642; 3-Et-2-Py], [BE 643; 4-Cl-3-Et-2-Py], [BE 644; 5-Cl-3-Et-2-Py], [BE 645; 6-Cl-3-Et-2-Py], [BE 646; Me-3-Et-2-Py], [BE 647; 5-Me-3-Et-2-Py], [BE 648; 6-Me-3-Et-2-Py], [BE 649; 4-CF ₃ -3-Et-2-Py], [BE 650; 5-CF ₃ -3-Et-2-Py], [BE 651; 6-CF ₃ -3-Et-2-Py], [BE 652; 4-CN -3-Et-2-Py !, [BE 653; 5-CN-3-Et-2-Py], [BE 654; 6-CN-3-Et-2-Py], [BE 655; 4-OMe-3 -Et-2-Py], [BE 656; 5-OMe-3-Et-2-Py], [BE 657; 6-OMe-3-Et-2-Py], [BE 658; 4-Et-2-Py ], [BE 659; 3-Cl-4-Et-2-Py], [BE 660; 5-Cl-4-Et-2-Py], [BE 661; 6-Cl-4-Et-2-Py], [BE662; 3-Me-4-Et-2-Py], [BE663; 5-Me-4-Et-2-Py], [BE664; 6-Me-4-Et-2-Py], [BE 665] 3-CF ₃ -4-Et-2-Py], [BE 666; 5-CF ₃ -4-Et-2-Py], [BE 667; 6-CF ₃ -4-Et-2-Py], [BE 667; BE668; 3-CN-4-Et-2-Py], [BE 669; 5-CN-4-Et-2-Py], [BE 670; 6-CN-4-Et-2-Py], [BE 671; 3-OMe-4-Et-2-Py], [BE 672; 5-OMe-4-Et-2-Py], [BE 673; 6-OMe-4-Et-2-Py], [BE 674; Et-2-Py, [BE 675; 3-Cl-5-Et-2-Py], [BE 676; 4-Cl-5-Et-2-Py], [BE 677; 6-Cl-5-Et- 2-Py], [BE 678; 3-Me-5-Et-2-P y], [BE 679; 4-Me-5-Et-2-Py], [BE 680; 6-Me-5-Et-2-Py], [BE 681; 3-CF ₃ -5-Et-2-Py ], [BE682; 4-CF 3 -5-Et-2-Py], [BE683; 6-CF 3 -5-Et-2-Py], [BE684; 3-CN-5-Et-2-Py ], [BE 685; 4-CN-5-Et-2-Py], [BE 686; 6-CN-5-Et-2-Py], [BE 687; 3-OMe-5-Et-2-Py], [BE 688; 4-OMe-5-Et-2-Py], [BE 689; 6-OMe-5-Et-2-Py], [BE 690; 6-Et-2-Py], [BE 691; 3-Cl -6-Et-2-Py], [BE692; 4-Cl-6-Et-2-Py], [BE693; 5-Cl-6-Et-2-Py], [BE 694; 3-Me-6 -Et-2-Py], [BE 695; 4-Me-6-Et-2-Py], [BE 696; 5-Me-6-Et-2-Py], [BE 697; 3-CF ₃ -6- Et-2-Py], [BE 698; 4-CF ₃ -6-Et-2-Py], [BE 699; 5-CF ₃ -6-Et-2-Py], [BE 700; Et-2-Py, [BE 701; 4-CN-6-Et-2-Py],

[BE702; 5-CN-6-Et-2-Py], [BE 703; 3-OMe-6-Et-2-Py], [BE704; 4-OMe-6-Et-2-Py], [BE 705] ; 5-OMe-6-Et -2-Py], [BE706; 3-CH 2 CF 3 -2-Py], [BE707; 4-Cl-3-CH 2 CF 3 -2-Py], [BE708 ; 5-Cl-3-CH 2 CF 3 -2-Py], [BE709; 6-Cl-3-CH 2 CF 3 -2-Py], [BE710; 4-Me-3-CH 2 CF 3 - 2-Py], [BE711; 5-Me-3-CH 2 CF 3 -2-Py], [BE712; 6-Me-3-CH 2 CF 3 -2-Py], [BE713; 4-CF 3 -3-CH ₂ CF ₃ -2-Py, [BE 714; 5-CF ₃ -3-CH ₂ CF ₃ -2-Py], [BE 715; 6-CF ₃ -3-CH ₂ CF ₃ -2- Py], [BE716; 4- CN-3-CH 2 CF 3 -2-Py], [BE717; 5-CN-3-CH 2 CF 3 -2-Py], [BE718; 6-CN-3- _{CH 2 CF 3 -2-Py]} , [BE719; 4-OMe-3-CH 2 CF 3 -2-Py], [BE720; 5-OMe-3-CH 2 CF 3 -2-Py], [BE721 ; 6-OMe-3-CH 2 CF 3 -2-Py], [BE722; 4-CH 2 CF 3 -2-Py], [BE723; 3-Cl-4-CH 2 CF 3 -2-Py] , [BE724; 5-Cl- 4-CH 2 CF 3 -2-Py], [BE725; 6-Cl-4-CH 2 CF 3 -2-Py], [BE726; 3-Me-4-CH 2 _{CF 3 -2-Py], [} BE727; 5-Me-4-CH 2 CF 3 -2-Py], [BE728; 6-Me-4-CH 2 CF 3 -2-Py], [BE729; 3 _{-CF 3 -4-CH 2 CF 3} -2-Py], [BE730; 5-CF 3 -4-CH 2 CF 3 -2-Py], [BE731; 6-CF 3 -4-CH 2 CF 3 -2-Py], [BE732; 3-CN-4-CH 2 CF 3 -2-Py], [BE733; 5-CN-4-CH 2 CF 3 -2-Py], [BE734; 6-CN -4-CH ₂ CF ₃ -2 -Py], [BE735; 3- OMe-4-CH 2 CF 3 -2-Py], [BE736; 5-OMe-4-CH 2 CF 3 -2-Py], [BE737; 6-OMe-4 _{-CH 2 CF 3 -2-Py]} , [BE738; 5-CH 2 CF 3 -2-Py], [BE739; 3-Cl-5-CH 2 CF 3 -2-Py], [BE740; 4- _{Cl-5-CH 2 CF 3} -2-Py], [BE741; 6-Cl-5-CH 2 CF 3 -2-Py], [BE742; 3-Me-5-CH 2 CF 3 -2-Py ], [BE 743; 4-Me-5-CH ₂ CF ₃ -2-Py], [BE 744; 6-Me-5-CH ₂ CF ₃ -2-Py], [BE 745; 3-CF ₃ -5-] _{CH 2 CF 3 -2-Py]} , [BE746; 4-CF 3 -5-CH 2 CF 3 -2-Py], [BE747; 6-CF 3 -5-CH 2 CF 3 -2-Py], [BE 748; 3-CN-5-CH ₂ CF ₃ -2-Py], [BE 749; 4-CN -5-CH ₂ CF ₃ -2-Py], [BE 750; 6-CN -5-CH ₂ CF _{3 -2-Py], [BE751} ; 3-OMe-5-CH 2 CF 3 -2-Py], [BE752; 4-OMe-5-CH 2 CF 3 -2-Py], [BE753; 6- _{OMe-5-CH 2 CF 3} -2-Py], [BE754; 6-CH 2 CF 3 -2-Py], [BE755; 3-Cl-6-CH 2 CF 3 -2-Py], [BE756 ; 4-Cl-6-CH 2 CF 3 -2-Py], [BE757; 5-Cl-6-CH 2 CF 3 -2-Py], [BE758; 3-Me-6-CH 2 CF 3 - 2-Py], [BE 759; 4-Me-6-CH ₂ CF ₃ -2-Py], [BE 760; 5-Me-6-CH ₂ CF ₃ -2-Py], [BE 761; 3-CF ₃ -6-CH ₂ CF ₃ -2-Py, [BE 762; 4-CF ₃ -6-CH ₂ CF ₃ -2-Py], [BE 763; 5-CF ₃ -6-CH ₂ CF ₃ -2- Py], [BE764; 3- CN-6-CH 2 CF 3 -2-Py], [BE765; 4-CN-6-CH 2 CF 3 -2-Py], [BE766; 5-CN-6- CH ₂ C _{F 3 -2-Py], [} BE767; 3-OMe-6-CH 2 CF 3 -2-Py], [BE768; 4-OMe-6-CH 2 CF 3 -2-Py], [BE769; 5 _{-OMe-6-CH 2 CF 3} -2-Py], [BE770; 3-OEt-2-Py], [BE771; 4-Cl-3-OEt-2-Py], [BE772; 5-Cl- 3-OEt-2-Py !, [BE 773; 6-Cl-3-OEt-2-Py], [BE 774; 4-Me-3-OEt-2-Py], [BE 775; 5-Me-3- OEt-2-Py], [ BE776; 6-Me-3-OEt-2-Py], [BE777; 4-CF 3 -3-OEt-2-Py], [BE778; 5-CF 3 -3- OEt-2-Py], [ BE779; 6-CF 3 -3-OEt-2-Py], [BE780; 4-CN-3-OEt-2-Py], [BE781; 5-CN-3-OEt -2-Py !, [BE 782; 6-CN-3-OEt-2-Py], [BE 783; 4-OMe-3-OEt-2-Py], [BE 784; 5-OMe-3-OEt-2 -Py], [BE 785; 6-OMe-3-OEt-2-Py], [BE 786; 4-OEt-2-Py], [BE 787; 3-Cl-4-OEt-2-Py], [BE 788] 5-Cl-4-OEt-2-Py !, [BE 789; 6-Cl-4-OEt-2-Py], [BE 790; 3-Me-4-OEt-2-Py], [BE 791; -Me-4-OEt-2- Py], [BE792; 6-Me-4-OEt-2-Py], [BE793; 3-CF 3 -4-OEt-2-Py], [BE794; 5- _{CF 3 -4-OEt-2-} Py], [BE795; 6-CF 3 -4-OEt-2-Py], [BE796; 3-CN-4-OEt-2-Py], [BE797; 5- CN-4-OEt-2-Py !, [BE 798; 6-CN-4-OEt-2-Py], [BE799; 3-OMe-4-OEt-2-Py], [BE 800; 5-OMe- 4-OEt-2-Py], [BE 801; 6-OMe-4-OEt-2-Py],

[BE802; 5-OEt-2-Py], [BE 803; 3-Cl-5-OEt-2-Py], [BE 804; 4-Cl-5-OEt-2-Py], [BE 805; 6-Cl -5-OEt-2-Py !, [BE 806; 3-Me-5-OEt-2-Py], [BE 807; 4-Me-5-OEt-2-Py], [BE 808; 6-Me-5 -OEt-2-Py], [ BE809; 3-CF 3 -5-OEt-2-Py], [BE810; 4-CF 3 -5-OEt-2-Py], [BE811; 6-CF 3 - 5-OEt-2-Py, [BE 812; 3-CN-5-OEt-2-Py], [BE 813; 4-CN-5-OEt-2-Py], [BE 814; 6-CN-5- OEt-2-Py, [BE 815; 3-OMe-5-OEt-2-Py], [BE 816; 4-OMe-5-OEt-2-Py], [BE 817; 6-OMe-5-OEt- 2-Py], [BE 818; 6-OEt-2-Py], [BE 819; 3-Cl-6-OEt-2-Py], [BE 820; 4-Cl-6-OEt-2-Py], BE 821; 5-Cl-6-OEt-2-Py], [BE 822; 3-Me-6-OEt-2-Py], [BE 823; 4-Me-6-OEt-2-Py], [BE 824; 5-Me-6-OEt- 2-Py], [BE825; 3-CF 3 -6-OEt-2-Py], [BE826; 4-CF 3 -6-OEt-2-Py], [BE827; _{5-CF 3 -6-OEt-} 2-Py], [BE828; 3-CN-6-OEt-2-Py], [BE829; 4-CN-6-OEt-2-Py], [BE830; 5 -CN-6-OEt-2-Py], [BE 831; 3-OMe-6-OEt-2-Py], [BE 832; 4-OMe-6-OEt-2-Py], [BE 833; 5-OMe -6-OEt-2-Py, [BE 834; 3-OCH ₂ CF ₃ -2-Py], [BE 835; 4-Cl-3-OCH ₂ CF ₃ -2-Py], [BE 836; 5-Cl _{-3-OCH 2 CF 3 -2-} Py], [BE837; 6-Cl-3-OCH 2 CF 3 -2-Py], [BE838; 4-Me-3-OCH 2 CF 3 -2-Py] , [BE839; 5-Me- 3-OCH 2 CF 3 -2-Py], [BE840; 6-Me-3-OCH 2 CF 3 -2-Py] _{, [BE841; 4-CF 3} -3-OCH 2 CF 3 -2-Py], [BE842; 5-CF 3 -3-OCH 2 CF 3 -2-Py], [BE843; 6-CF 3 -3 _{-OCH 2 CF 3 -2-Py]} , [BE844; 4-CN-3-OCH 2 CF 3 -2-Py], [BE845; 5-CN-3-OCH 2 CF 3 -2-Py], [ BE846; 6-CN-3- OCH 2 CF 3 -2-Py], [BE847; 4-OMe-3-OCH 2 CF 3 -2-Py], [BE848; 5-OMe-3-OCH 2 CF 3 -2-Py], [BE849; 6-OMe-3-OCH 2 CF 3 -2-Py], [BE850; 4-OCH 2 CF 3 -2-Py], [BE851; 3-Cl-4-OCH ₂ CF ₃ -2-Py !, [BE 852; 5-Cl-4-OCH ₂ CF ₃ -2-Py], [BE 853; 6-Cl 4-OCH ₂ CF ₃ -2-Py], [BE 854; _{3-Me-4-OCH 2} CF 3 -2-Py], [BE855; 5-Me-4-OCH 2 CF 3 -2-Py], [BE856; 6-Me-4-OCH 2 CF 3 -2 -Py], [BE857; 3- CF 3 -4-OCH 2 CF 3 -2-Py], [BE858; 5-CF 3 -4-OCH 2 CF 3 -2-Py], [BE859; 6-CF _{3 -4-OCH 2 CF 3 -2} -Py], [BE860; 3-CN-4-OCH 2 CF 3 -2-Py], [BE861; 5-CN-4-OCH 2 CF 3 -2-Py ], [BE862; 6-CN -4-OCH 2 CF 3 -2-Py], [BE863; 3-OMe-4-OCH 2 CF 3 -2-Py], [BE864; 5-OMe-4-OCH ₂ CF ₃ -2-Py !, [BE 865; 6-OMe -4-OCH ₂ CF ₃ -2-Py], [BE 866; 5-OCH ₂ CF ₃ -2-Py], [BE 867; 3-Cl- _{5-OCH 2 CF 3 -2-} Py], [BE868; 4-Cl-5-OCH 2 CF 3 -2-Py], [BE869; 6-Cl-5-OCH 2 CF 3 -2-Py], [BE 870; 3-Me-5-OCH ₂ CF ₃ -2-Py], [BE 871; 4-Me-5-OCH ₂ CF ₃ -2-Py], [BE 872; 6-Me-5-OCH ₂ CF ₃ -2-Py], [BE 873; 3-CF ₃ -5-OCH ₂ CF ₃ -2-Py], [BE 874; _{CF 3 -5-OCH 2 CF 3} -2-Py], [BE875; 6-CF 3 -5-OCH 2 CF 3 -2-Py], [BE876; 3-CN-5-OCH 2 CF 3 -2 4-Py], [BE 877; 4-CN-5-OCH ₂ CF ₃ -2-Py], [BE 878; 6-CN 5-OCH ₂ CF ₃ -2-Py], [BE 879; 3-OMe-5 _{-OCH 2 CF 3 -2-Py]} , [BE880; 4-OMe-5-OCH 2 CF 3 -2-Py], [BE881; 6-OMe-5-OCH 2 CF 3 -2-Py], [ BE 882; 6-OCH ₂ CF ₃ -2-Py], [BE 883; 3-Cl 6-OCH ₂ CF ₃ -2-Py], [BE 884; 4-Cl 6-OCH ₂ CF ₃ -2-Py ], [BE885; 5-Cl -6-OCH 2 CF 3 -2-Py], [BE886; 3-Me-6-OCH 2 CF 3 -2-Py], [BE887; 4-Me-6-OCH ₂ CF ₃ -2-Py], [BE 888; 5-Me-6-OCH ₂ CF ₃ -2-Py], [BE 889; 3-CF ₃ -6-OCH ₂ CF ₃ -2-Py], [BE 890] _{; 4-CF 3 -6-OCH} 2 CF 3 -2-Py], [BE891; 5-CF 3 -6-OCH 2 CF 3 -2-Py], [BE892; 3-CN-6-OCH 2 CF _{3 -2-Py], [BE893} ; 4-CN-6-OCH 2 CF 3 -2-Py], [BE894; 5-CN-6-OCH 2 CF 3 -2-Py], [BE895; 3- _{OMe-6-OCH 2 CF 3} -2-Py], [BE896; 4-OMe-6-OCH 2 CF 3 -2-Py], [BE897; 5-OMe-6-OCH 2 CF 3 -2-Py ], [BE 898; 4-Cl-3-Pr-2-Py], [BE 899; 5-Cl-3-Pr-2-Py], [BE 900; 6-Cl-3-Pr-2-Py], [BE 901; 4-Me-3-Pr-2-Py],

[BE902; 5-Me-3-Pr-2-Py], [BE 903; 6-Me-3-Pr-2-Py], [BE 904; 4-CF ₃ -3-Pr-2-Py], [BE 902; _{BE905; 5-CF 3 -3-} Pr-2-Py], [BE906; 6-CF 3 -3-Pr-2-Py], [BE907; 4-CN-3-Pr-2-Py], [ BE 908; 5-CN-3-Pr-2-Py !, [BE 909; 6-CN-3-Pr-2-Py], [BE 910; 4-OMe-3-Pr-2-Py], [BE 911; 5-OMe-3-Pr-2-Py !, [BE 912; 6-OMe-3-Pr-2-Py], [BE 913; 4-Pr-2-Py], [BE 914; 3-Cl-4- Pr-2-Py, [BE 915; 5-Cl-4-Pr-2-Py], [BE 916; 6-Cl-4-Pr-2-Py], [BE 917; 3-Me-4-Pr- 2-Py], [BE 918; 5-Me-4-Pr-2-Py], [BE 919; 6-Me-4-Pr-2-Py], [BE 920; 3-CF ₃ -4-Pr-2 -Py], [BE921; 5- CF 3 -4-Pr-2-Py], [BE922; 6-CF 3 -4-Pr-2-Py], [BE923; 3-CN-4-Pr-2 -Py], [BE 924; 5-CN-4-Pr-2-Py], [BE 925; 6-CN-4-Pr-2-Py], [BE 926; 3-OMe-4-Pr-2-Py ], [BE 927; 5-OMe-4-Pr-2-Py], [BE 928; 6-OMe-4-Pr-2-Py], [BE 929; 5-Pr-2-Py], [BE 930; 3] -Cl-5-Pr-2-Py], [BE 931; 4-Cl-5-Pr-2-Py], [BE 932; 6-Cl-5-Pr-2-Py], [BE 933; 3-Me -5-Pr-2-Py !, [BE 934; 4-Me-5-Pr-2-Py], [BE 935; 6-Me-5-Pr-2-Py], [BE 936; 3-CF _3- 5-Pr-2-Py, [BE 937; 4-CF ₃ -5-Pr-2-Py], [BE 938; 6-CF ₃ -5-Pr-2-Py], [BE 939; 3-CN- 5-Pr-2-Py, [BE 940; 4-CN-5-Pr-2-Py], [BE 941; 6-CN-5-Pr-2-Py], [BE 942; 3-OMe-5- Pr-2-Py, [BE943; 4-OMe-5-Pr-2-Py], [BE 944; 6- OMe-5-Pr-2-Py], [BE 945; 6-Pr-2-Py], [BE 946; 3-Cl-6-Pr-2-Py], [BE 947; 4-Cl-6-Pr- 2-Py], [BE948; 5-Cl-6-Pr-2-Py], [BE 949; 3-Me-6-Pr-2-Py], [BE 950; 4-Me-6-Pr-2- Py], [BE 951; 5-Me-6-Pr-2-Py], [BE 952; 3-CF ₃ -6-Pr-2-Py], [BE 953; 4-CF ₃ -6-Pr-2- Py], [BE954; 5- CF 3 -6-Pr-2-Py], [BE955; 3-CN-6-Pr-2-Py], [BE956; 4-CN-6-Pr-2-Py ], [BE957; 5-CN-6-Pr-2-Py], [BE958; 3-OMe-6-Pr-2-Py], [BE959; 4-OMe-6-Pr-2-Py], [BE 960; 5-OMe-6-Pr-2-Py], [BE 961; 3-OPr-2-Py], [BE 962; 4-Cl-3-OPr-2-Py], [BE 963; 5-Cl -3-OPr-2-Py, [BE964; 6-Cl-3-OPr-2-Py], [BE 965; 4-Me-3-OPr-2-Py], [BE 966; 5-Me-3 -OPr-2-Py], [ BE967; 6-Me-3-OPr-2-Py], [BE968; 4-CF 3 -3-OPr-2-Py], [BE969; 5-CF 3 -3 -OPr-2-Py], [ BE970; 6-CF 3 -3-OPr-2-Py], [BE971; 4-CN-3-OPr-2-Py], [BE972; 5-CN-3- OPr-2-Py], [BE 973; 6-CN-3-OPr-2-Py], [BE 974; 4-OMe-3-OPr-2-Py], [BE 975; 5-OMe-3-OPr- 2-Py], [BE976; 6-OMe-3-OPr-2-Py], [BE977; 4-OPr-2-Py], [BE978; 3-Cl-4-OPr-2-Py], [BE972; BE979; 5-Cl-4-OPr-2-Py], [BE 980; 6-Cl-4-OPr-2-Py], [BE 981; 3-Me-4-OPr-2-Py], [BE 982; 5-Me-4-OPr- 2-Py], [BE983; 6-Me-4-OPr-2-Py], [BE984; 3-CF 3 -4-OPr-2-Py], [BE985; 5 -CF ₃ -4-OPr-2-Py], [B _{E986; 6-CF 3 -4-} OPr-2-Py], [BE987; 3-CN-4-OPr-2-Py], [BE988; 5-CN-4-OPr-2-Py], [BE989 6-CN-4-OPr-2-Py !, [BE990; 3-OMe-4-OPr-2-Py], [BE991; 5-OMe-4-OPr-2-Py], [BE992; -OMe-4-OPr-2-Py], [BE993; 5-OPr-2-Py], [BE994; 3-Cl-5-OPr-2-Py], [BE995; 4-Cl-5-OPr -2-Py], [BE 996; 6-Cl-5-OPr-2-Py], [BE 997; 3-Me-5-OPr-2-Py], [BE 998; 4-Me-5-OPr-2 -Py], [BE999; 6- Me-5-OPr-2-Py], [BE1000; 3-CF 3 -5-OPr-2-Py], [BE1001; 4-CF 3 -5-OPr-2 -Py],

_{[BE1002; 6-CF 3 -5} -OPr-2-Py], [BE1003; 3-CN-5-OPr-2-Py], [BE1004; 4-CN-5-OPr-2-Py], [ BE 1005; 6-CN-5-OPr-2-Py], [BE 1006; 3-OMe-5-OPr-2-Py], [BE 1007; 4-OMe-5-OPr-2-Py], [BE 1008; 6-OMe-5-OPr-2-Py], [BE 1009; 6-OPr-2-Py], [BE 1010; 3-Cl-6-OPr-2-Py], [BE 1011; 4-Cl-6- OPr-2-Py], [BE1012; 5-Cl-6-OPr-2-Py], [BE1013; 3-Me-6-OPr-2-Py], [BE1014; 4-Me-6-OPr- 2-Py], [BE1015; 5-Me-6-OPr-2-Py], [BE1016; 3-CF 3 -6-OPr-2-Py], [BE1017; 4-CF 3 -6-OPr- 2-Py], [BE1018; 5-CF 3 -6-OPr-2-Py], [BE1019; 3-CN-6-OPr-2-Py], [BE1020; 4-CN-6-OPr-2 -Py], [BE 1021; 5-CN-6-OPr-2-Py], [BE 1022; 3-OMe-6-OPr-2-Py], [BE 1023; 4-OMe-6-OPr-2-Py ], [BE 1024; 5-OMe-6-OPr-2-Py], [BE 1025; 3-SMe-2-Py], [BE 1026; 4-Cl-3-SMe-2-Py], [BE 1027; -Cl-3-SMe-2-Py], [BE1028; 6-Cl-3-SMe-2-Py], [BE1029; 4-Me-3-SMe-2-Py], [BE1030; 5-Me -3-SMe-2-Py] , [BE1031; 6-Me-3-SMe-2-Py], [BE1032; 4-CF 3 -3-SMe-2-Py], [BE1033; 5-CF 3 -3-SMe-2-Py] , [BE1034; 6-CF 3 -3-SMe-2-Py], [BE1035; 4-CN-3-SMe-2-Py], [BE1036; 5-CN- 3-SMe-2-Py !, [BE1037; 6-CN-3-SMe-2-Py], [BE1038; 4-OMe-3-SMe-2-Py], [BE1039; 5-OMe-3- SMe-2-Py], [BE1040; 6-OMe-3-SMe-2-Py], [BE10] 41; 4-SMe-2-Py !, [BE1042; 3-Cl-4-SMe-2-Py], [BE1043; 5-Cl-4-SMe-2-Py], [BE1044; 6-Cl- 4-SMe-2-Py !, [BE1045; 3-Me-4-SMe-2-Py], [BE 1046; 5-Me-4-SMe-2-Py], [BE1047; 6-Me-4- 4 SMe-2-Py], [ BE1048; 3-CF 3 -4-SMe-2-Py], [BE1049; 5-CF 3 -4-SMe-2-Py], [BE1050; 6-CF 3 -4 -SMe-2-Py], [BE1051; 3-CN-4-SMe-2-Py], [BE1052; 5-CN-4-SMe-2-Py], [BE1053; 6-CN-4-SMe -2-Py], [BE1054; 3-OMe-4-SMe-2-Py], [BE1055; 5-OMe-4-SMe-2-Py], [BE1056; 6-OMe-4-SMe-2 -Py], [BE1057; 5-SMe-2-Py], [BE1058; 3-Cl-5-SMe-2-Py], [BE1059; 4-Cl-5-SMe-2-Py], [BE 1060] 6-Cl-5-SMe-2-Py !, [BE1061; 3-Me-5-SMe-2-Py], [BE1062; 4-Me-5-SMe-2-Py], [BE1063; -Me-5-SMe-2- Py], [BE1064; 3-CF 3 -5-SMe-2-Py], [BE1065; 4-CF 3 -5-SMe-2-Py], [BE1066; 6 _{-CF 3 -5-SMe-2-} Py], [BE1067; 3-CN-5-SMe-2-Py], [BE1068; 4-CN-5-SMe-2-Py], [BE1069; 6- CN-5-SMe-2-Py !, [BE 1070; 3-OMe-5-SMe-2-Py], [BE 1071; 4-OMe-5-SMe-2-Py], [BE 1072; 6-OMe- 5-SMe-2-Py !, [BE1073; 6-SMe-2-Py], [BE1074; 3-Cl-6-SMe-2-Py], [BE1075; 4-Cl-6-SMe-2-. Py], [BE1076; 5-Cl-6-SMe-2-Py], [BE1077; 3-Me-6-SMe-2-Py], [BE1078; 4-Me-6-SMe-2-Py] , [BE1079; 5-Me- 6-SMe-2-Py], [BE1080; 3-CF 3 -6-SMe -2-Py], [BE1081; 4-CF 3 -6-SMe-2-Py], [BE1082; 5-CF 3 -6-SMe-2-Py], [BE1083; 3-CN-6-SMe -2-Py !, [BE1084; 4-CN-6-SMe-2-Py], [BE1085; 5-CN-6-SMe-2-Py], [BE1086; 3-OMe-6-SMe-2 -Py], [BE1087; 4- OMe-6-SMe-2-Py], [BE1088; 5-OMe-6-SMe-2-Py], [BE1089; 3-SCF 3 -2-Py], [ BE1090; 4-Cl-3- SCF 3 -2-Py], [BE1091; 5-Cl-3-SCF 3 -2-Py], [BE1092; 6-Cl-3-SCF 3 -2-Py], [BE1093; 4-Me-3 -SCF 3 -2-Py], [BE1094; 5-Me-3-SCF 3 -2-Py], [BE1095; 6-Me-3-SCF 3 -2-Py] , [BE 1096; 4-CF ₃ -3-SCF ₃ -2-Py], [BE 1097; 5-CF ₃ -3-SCF ₃ -2-Py], [BE 1098; 6-CF ₃ -3-SCF _3- 2-Py], [BE1099; 4-CN-3-SCF 3 -2-Py], [BE1100; 5-CN-3-SCF 3 -2-Py], [BE1101; 6-CN-3-SCF 3 -2-Py],

[BE1102; 4-OMe-3 -SCF 3 -2-Py], [BE1103; 5-OMe-3-SCF 3 -2-Py], [BE1104; 6-OMe-3-SCF 3 -2-Py] _{, [BE1105; 4-SCF 3} -2-Py], [BE1106; 3-Cl-4-SCF 3 -2-Py], [BE1107; 5-Cl-4-SCF 3 -2-Py], [BE1108 ; 6-Cl-4-SCF 3 -2-Py], [BE1109; 3-Me-4-SCF 3 -2-Py], [BE1110; 5-Me-4-SCF 3 -2-Py], [ BE 1111; 6-Me-4-SCF ₃ -2-Py], [BE 11 12; 3-CF ₃ -4-SCF ₃ -2-Py], [BE 1113; 5-CF ₃ -4-SCF ₃ -2-Py] ], [BE1114; 6-CF 3 -4-SCF 3 -2-Py], [BE1115; 3-CN-4-SCF 3 -2-Py], [BE1116; 5-CN-4-SCF 3 -2 -Py], [BE1117; 6- CN-4-SCF 3 -2-Py], [BE1118; 3-OMe-4-SCF 3 -2-Py], [BE1119; 5-OMe-4-SCF 3 - 2-Py], [BE1120; 6-OMe-4-SCF 3 -2-Py], [BE1121; 5-SCF 3 -2-Py], [BE1122; 3-Cl-5-SCF 3 -2-Py ], [BE1123; 4-Cl -5-SCF 3 -2-Py], [BE1124; 6-Cl-5-SCF 3 -2-Py], [BE1125; 3-Me-5-SCF 3 -2- Py], [BE 1126; 4-Me-5-SCF ₃ -2-Py], [BE 1127; 6-Me-5-SCF ₃ -2-Py], [BE 1 128; 3-CF ₃ -5-SCF _3- 2-Py], [BE 1129; 4-CF ₃ -5-SCF ₃ -2-Py], [BE 1130; 6-CF ₃ -5-SCF ₃ -2-Py], [BE 1131; SCF ₃ -2-Py !, [BE 1132; 4-CN-5-SCF ₃ -2-Py], [BE 1133; 6-CN-5-SCF ₃ -2-Py], [BE 1 134; 3-OMe-5] -SCF ₃ -2-Py], [BE 1135; 4-OMe-5-SCF ₃ -2-Py], [BE 1136; 6-OMe-5-SCF ₃ -2-Py], [BE _{1137; 6-SCF 3 -2-} Py], [BE1138; 3-Cl-6-SCF 3 -2-Py], [BE1139; 4-Cl-6-SCF 3 -2-Py], [BE1140; 6 _{-Cl-6-SCF 3 -2-} Py], [BE1141; 3-Me-6-SCF 3 -2-Py], [BE1142; 4-Me-6-SCF 3 -2-Py], [BE1143; 6-Me-6-SCF ₃ -2-Py, [BE 1144; 3-CF ₃ -6-SCF ₃ -2-Py], [BE 1145; 4-CF ₃ -6-SCF ₃ -2-Py], _{[BE1146; 6-CF 3 -6} -SCF 3 -2-Py], [BE1147; 3-CN-6-SCF 3 -2-Py], [BE1148; 4-CN-6-SCF 3 -2-Py ], [BE 1149; 6-CN-6-SCF ₃ -2-Py], [BE 1150; 3-OMe-6-SCF ₃ -2-Py], [BE 1151; 4-OMe -6-SCF ₃ -2-] Py], [BE1152; 6- OMe-6-SCF 3 -2-Py], [BE1153; 3-S (O) Me-2-Py], [BE1154; 4-Cl-3-S (O) Me -2-Py !, [BE1 155; 5-Cl-3-S (O) Me-2-Py], [BE 1156; 6-Cl-3-S (O) Me-2-Py], [BE1 157; -Me-3-S (O) Me-2-Py], [BE1158; 5-Me-3-S (O) Me-2-Py], [BE1159; 6-Me-3-S (O) Me -2-Py !, [BE 1 160; 4-CF ₃ -3-S (O) Me-2-Py], [BE 1161; 5-CF ₃ -3-S (O) Me-2-Py], [BE 1162 _{; 6-CF 3 -3-S} (O) Me-2-Py], [BE1163; 4-CN-3-S (O) Me-2-Py], [BE1164; 5-CN-3-S ( O) Me-2-Py], [BE1165; 6-CN-3-S (O) Me-2-Py], [BE1166; 4-OMe-3-S (O) Me-2-Py], BE1167; 5-OMe-3-S (O) Me-2-Py], [BE1168; 6-OMe-3-S (O) Me-2-Py], [BE1169; 4-S (O) Me- 2-Py], [BE1170; 3-Cl-4-S (O) Me-2-Py], [BE1171; 5-Cl-4-S (O) Me-2-Py], [BE1172; 6- Cl-4 -S (O) Me-2-Py], [BE1173; 3-Me-4-S (O) Me-2-Py], [BE1174; 5-Me-4-S (O) Me-2-Py ], [BE1175; 6-Me -4-S (O) Me-2-Py], [BE1176; 3-CF 3 -4-S (O) Me-2-Py], [BE1177; 5-CF 3 -4-S (O) Me- 2-Py], [BE1178; 6-CF 3 -4-S (O) Me-2-Py], [BE1179; 3-CN-4-S (O) Me- 2-Py], [BE 1180; 5-CN-4-S (O) Me-2-Py], [BE1181; 6-CN-4-S (O) Me-2-Py], [BE1182; OMe-4-S (O) Me-2-Py], [BE1183; 5-OMe-4-S (O) Me-2-Py], [BE1184; 6-OMe-4-S (O) Me- 2-Py], [BE 1185; 5-S (O) Me-2-Py], [BE 1186; 3-Cl-5-S (O) Me-2-Py], [BE 1187; 4-Cl-5- S (O) Me-2-Py], [BE1188; 6-Cl-5-S (O) Me-2-Py], [BE1189; 3-Me-5-S (O) Me-2-Py] , [BE1190; 4-Me- 5-S (O) Me-2-Py], [BE1191; 6-Me-5-S (O) Me-2-Py], [BE1192; 3-CF 3 -5 -S (O) Me-2- Py], [BE1193; 4-CF 3 -5-S (O) Me-2-Py], [BE1194; 6-CF 3 -5-S (O) Me-2 -Py], [BE 1195; 3-CN-5-S (O) Me-2-Py], [BE 1196; 4-CN-5-S (O) Me-2-Py], [BE 1197; 6-CN -5-S (O) Me-2-Py], [BE 1198; 3-OMe-5-S (O) Me-2-Py], [BE 1199; 4-OMe-5-S (O) Me-2 -Py], [BE1200; 6-OMe-5-S (O) Me-2-Py], [BE1201; 6-S (O) Me-2-Py],

[BE1202; 3-Cl-6-S (O) Me-2-Py], [BE 1203; 4-Cl-6-S (O) Me-2-Py], [BE 1204; 5-Cl-6-S (O) Me-2-Py], [BE 1205; 3-Me-6-S (O) Me-2-Py], [BE 1206; 4-Me-6-S (O) Me-2-Py], [BE1207; 5-Me-6 -S (O) Me-2-Py], [BE1208; 3-CF 3 -6-S (O) Me-2-Py], [BE1209; 4-CF 3 -6 -S (O) Me-2- Py], [BE1210; 5-CF 3 -6-S (O) Me-2-Py], [BE1211; 3-CN-6-S (O) Me-2- Py], [BE 1212; 4-CN-6-S (O) Me-2-Py], [BE 1213; 5-CN-6-S (O) Me-2-Py], [BE 1214; 3-OMe- 6-S (O) Me-2-Py], [BE 1215; 4-OMe-6-S (O) Me-2-Py], [BE 1216; 5-OMe-6-S (O) Me-2- 2 Py], [BE1217; 3- S (O) CF 3 -2-Py], [BE1218; 4-Cl-3-S (O) CF 3 -2-Py], [BE1219; 5-Cl-3- _{S (O) CF 3 -2-} Py], [BE1220; 6-Cl-3-S (O) CF 3 -2-Py], [BE1221; 4-Me-3-S (O) CF 3 -2 -Py], [BE1222; 5- Me-3-S (O) CF 3 -2-Py], [BE1223; 6-Me-3-S (O) CF 3 -2-Py], [BE1224; 4 _{-CF 3 -3-S (O)} CF 3 -2-Py], [BE1225; 5-CF 3 -3-S (O) CF 3 -2-Py], [BE1226; 6-CF 3 -3- _{S (O) CF 3 -2-} Py], [BE1227; 4-CN-3-S (O) CF 3 -2-Py], [BE1228; 5-CN-3-S (O) CF 3 -2 -Py], [BE 1229; 6-CN-3-S (O) CF ₃ -2-Py], [BE 1230; 4-OMe-3-S (O) CF ₃ -2-Py], [BE 12 31; 5 -OMe-3-S (O) CF 3 -2-Py], [BE1232; 6-OMe-3-S (O) CF 3 -2-Py], [BE1233; 4-S (O) CF 3 - 2-Py], [BE 1234; 3-Cl-4-S (O) CF ₃ -2-Py], [BE 1235; 5-Cl-4-S ( O) CF 3 -2-Py], [BE1236; 6-Cl-4-S (O) CF 3 -2-Py], [BE1237; 3-Me-4-S ( _{O) CF 3 -2-Py]} , [BE1238; 5-Me-4-S (O) CF 3 -2-Py], [BE1239; 6-Me-4-S (O) CF 3 -2-Py ], [BE1240; 3-CF 3 -4-S (O) CF 3 -2-Py], [BE1241; 5-CF 3 -4-S (O) CF 3 -2-Py], [BE1242; 6 _{-CF 3 -4-S (O)} CF 3 -2-Py], [BE1243; 3-CN-4-S (O) CF 3 -2-Py], [BE1244; 5-CN-4-S ( _{O) CF 3 -2-Py]} , [BE1245; 6-CN-4-S (O) CF 3 -2-Py], [BE1246; 3-OMe-4-S (O) CF 3 -2-Py ], [BE1247; 5-OMe -4-S (O) CF 3 -2-Py], [BE1248; 6-OMe-4-S (O) CF 3 -2-Py], [BE1249; 5-S _{(O) CF 3 -2-Py} ], [BE1250; 3-Cl-5-S (O) CF 3 -2-Py], [BE1251; 4-Cl-5-S (O) CF 3 -2- Py], [BE1252; 6- Cl-5-S (O) CF 3 -2-Py], [BE1253; 3-Me-5-S (O) CF 3 -2-Py], [BE1254; 4- Me-5-S (O) CF 3 -2-Py], [BE1255; 6-Me-5-S (O) CF 3 -2-Py], [BE1256; 3-CF 3 -5-S (O ) CF ₃ -2-Py !, [BE 1257; 4-CF ₃ -5-S (O) CF ₃ -2-Py], [BE 1258; 6-CF ₃ -5-S (O) CF ₃ -2-] Py], [BE1259; 3- CN-5-S (O) CF 3 -2-Py], [BE1260; 4-CN-5-S (O) CF 3 -2-Py], [BE1261; 6- CN-5-S (O) CF 3 -2-Py], [BE1262; 3-OMe-5-S (O) CF 3 -2-Py], [BE1263; 4-OMe-5-S (O) _{CF 3 -2-Py], [} BE1264; 6-OMe-5-S (O) CF 3 -2-Py], [BE1265; 6-S (O) CF 3 -2-Py], [BE1266; 3 -Cl-6-S (O) CF ₃ -2-Py], [B E1267; 4-Cl-6- S (O) CF 3 -2-Py], [BE1268; 5-Cl-6-S (O) CF 3 -2-Py], [BE1269; 3-Me-6- _{S (O) CF 3 -2-} Py], [BE1270; 4-Me-6-S (O) CF 3 -2-Py], [BE1271; 5-Me-6-S (O) CF 3 -2 -Py], [BE1272; 3- CF 3 -6-S (O) CF 3 -2-Py], [BE1273; 4-CF 3 -6-S (O) CF 3 -2-Py], [BE1274 _{; 5-CF 3 -6-S} (O) CF 3 -2-Py], [BE1275; 3-CN-6-S (O) CF 3 -2-Py], [BE1276; 4-CN-6- _{S (O) CF 3 -2-} Py], [BE1277; 5-CN-6-S (O) CF 3 -2-Py], [BE1278; 3-OMe-6-S (O) CF 3 -2 -Py], [BE1279; 4- OMe-6-S (O) CF 3 -2-Py], [BE1280; 5-OMe-6-S (O) CF 3 -2-Py], [BE1281; 3 _{-S (O) 2 Me-2} -Py], [BE1282; 4-Cl-3-S (O) 2 Me-2-Py], [BE1283; 5-Cl-3-S (O) 2 Me- 2-Py], [BE1284; 6-Cl-3-S (O) 2 Me-2-Py], [BE1285; 4-Me-3-S (O) 2 Me-2-Py], [BE1286; 5-Me-3-S ( O) 2 Me-2-Py], [BE1287; 6-Me-3-S (O) 2 Me-2-Py], [BE1288; 4-CF 3 -3-S (O) ₂ Me-2-Py, [BE 1289; 5-CF ₃ -3-S (O) ₂ Me-2-Py], [BE 1290; 6-CF ₃ -3-S (O) ₂ Me- 2-Py], [BE1291; 4-CN-3-S (O) ₂ Me-2-Py], [BE1292; 5-CN-3-S (O) ₂ Me-2-Py], [BE1293; 6-CN-3-S ( O) 2 Me-2-Py], [BE1294; 4-OMe-3-S (O) 2 Me-2-Py], [BE1295; 5-OMe-3-S ( O) ₂ Me-2-Py], [BE 1296; 6-OMe-3-S (O) ₂ Me-2-Py], [BE 1297; 4-S (O) ₂ Me-2-Py], [BE 1298 3-Cl-4-S (O) ₂ Me-2- Py], [BE1299; 5-Cl-4-S (O) ₂ Me-2-Py], [BE1300; 6-Cl-4-S (O) ₂ Me-2-Py], [BE1301; Me-4-S (O) ₂ Me-2-Py],

[BE1302; 5-Me-4 -S (O) 2 Me-2-Py], [BE1303; 6-Me-4-S (O) 2 Me-2-Py], [BE1304; 3-CF 3 - _{4-S (O) 2 Me} -2-Py], [BE1305; 5-CF 3 -4-S (O) 2 Me-2-Py], [BE1306; 6-CF 3 -4-S (O) ₂ Me-2-Py !, [BE1307; 3-CN-4-S (O) ₂ Me-2-Py], [BE1308; 5-CN-4-S (O) ₂ Me-2-Py], [BE1309; 6-CN-4 -S (O) 2 Me-2-Py], [BE1310; 3-OMe-4-S (O) 2 Me-2-Py], [BE1311; 5-OMe-4 _{-S (O) 2 Me-2} -Py], [BE1312; 6-OMe-4-S (O) 2 Me-2-Py], [BE1313; 5-S (O) 2 Me-2-Py] , [BE 1314; 3-Cl-5-S (O) ₂ Me-2-Py], [BE 1315; 4-Cl-5-S (O) ₂ Me-2-Py], [BE 1316; 6-Cl- _{5-S (O) 2 Me} -2-Py], [BE1317; 3-Me-5-S (O) 2 Me-2-Py], [BE1318; 4-Me-5-S (O) 2 Me -2-Py], [BE 1319; 6-Me-5-S (O) ₂ Me-2-Py], [BE 1320; 3-CF ₃ -5-S (O) ₂ Me-2-Py], _{BE1321; 4-CF 3 -5-} S (O) 2 Me-2-Py], [BE1322; 6-CF 3 -5-S (O) 2 Me-2-Py], [BE1323; 3-CN- _{5-S (O) 2 Me} -2-Py], [BE1324; 4-CN-5-S (O) 2 Me-2-Py], [BE1325; 6-CN-5-S (O) 2 Me -2-Py !, [BE1326; 3-OMe-5-S (O) ₂ Me-2-Py], [BE1327; 4-OMe-5-S (O) ₂ Me-2-Py], [BE1328 ; 6-OMe-5-S (O) 2 Me-2-Py], [BE1329; 6-S (O) 2 Me-2-Py], [BE1330; 3-Cl-6-S (O) 2 Me-2-Py !, [BE1331; 4-Cl-6-S (O) ₂ Me-2-Py], [BE1332; 5-Cl-6-S (O) ₂ Me-2-Py], [BE1332; BE 1333; 3-Me-6-S (O) ₂ Me- 2-Py], [BE1334; 4-Me-6-S (O) ₂ Me-2-Py], [BE1335; 5-Me-6-S (O) ₂ Me-2-Py], [BE1336; _{3-CF 3 -6-S (} O) 2 Me-2-Py], [BE1337; 4-CF 3 -6-S (O) 2 Me-2-Py], [BE1338; 5-CF 3 -6 _{-S (O) 2 Me-2} -Py], [BE1339; 3-CN-6-S (O) 2 Me-2-Py], [BE1340; 4-CN-6-S (O) 2 Me- 2-Py], [BE1341; 5-CN-6-S (O) ₂ Me-2-Py], [BE1342; 3-OMe-6-S (O) ₂ Me-2-Py], [BE1343; 4-OMe-6-S ( O) 2 Me-2-Py], [BE1344; 5-OMe-6-S (O) 2 Me-2-Py], [BE1345; 3-S (O) 2 CF _{3 -2-Py], [BE1346} ; 4-Cl-3-S (O) 2 CF 3 -2-Py], [BE1347; 5-Cl-3-S (O) 2 CF 3 -2-Py] , [BE1348; 6-Cl- 3-S (O) 2 CF 3 -2-Py], [BE1349; 4-Me-3-S (O) 2 CF 3 -2-Py], [BE1350; 5- Me-3-S (O) 2 CF 3 -2-Py], [BE1351; 6-Me-3-S (O) 2 CF 3 -2-Py], [BE1352; 4-CF 3 -3-S _{(O) 2 CF 3 -2-} Py], [BE1353; 5-CF 3 -3-S (O) 2 CF 3 -2-Py], [BE1354; 6-CF 3 -3-S (O) 2 _{CF 3 -2-Py], [} BE1355; 4-CN-3-S (O) 2 CF 3 -2-Py], [BE1356; 5-CN-3-S (O) 2 CF 3 -2-Py ], [BE1357; 6-CN -3-S (O) 2 CF 3 -2-Py], [BE1358; 4-OMe-3-S (O) 2 CF 3 -2-Py], [BE1359; 5 -OMe-3-S (O) 2 CF 3 -2-Py], [BE1360; 6-OMe-3-S (O) 2 CF 3 -2-Py], [BE1361; 4-S (O) 2 _{CF 3 -2-Py], [} BE1362; 3-Cl-4-S (O) 2 CF 3 -2-Py], [BE1363; 5-Cl-4-S (O) 2 CF 3 -2-Py], [BE1364; 6-Cl-4-S (O) 2 CF 3 -2-Py], [BE1365; 3-Me-4-S (O) 2 CF 3 -2-Py], [BE1366; 5-Me-4 -S (O) 2 CF 3 -2-Py], [BE1367; 6-Me-4-S (O) 2 CF 3 -2-Py], [BE1368; 3-CF ₃ -4-S (O) ₂ CF ₃ -2-Py], [BE 1369; 5-CF ₃ -4-S (O) ₂ CF ₃ -2-Py], [BE 1370; 6-CF ₃ -4- _{S (O) 2 CF 3 -2} -Py], [BE1371; 3-CN-4-S (O) 2 CF 3 -2-Py], [BE1372; 5-CN-4-S (O) 2 CF _{3 -2-Py], [BE1373} ; 6-CN-4-S (O) 2 CF 3 -2-Py], [BE1374; 3-OMe-4-S (O) 2 CF 3 -2-Py] , [BE1375; 5-OMe- 4-S (O) 2 CF 3 -2-Py], [BE1376; 6-OMe-4-S (O) 2 CF 3 -2-Py], [BE1377; 5- _{S (O) 2 CF 3 -2} -Py], [BE1378; 3-Cl-5-S (O) 2 CF 3 -2-Py], [BE1379; 4-Cl-5-S (O) 2 CF _{3 -2-Py], [BE1380} ; 6-Cl-5-S (O) 2 CF 3 -2-Py], [BE1381; 3-Me-5-S (O) 2 CF 3 -2-Py] , [BE1382; 4-Me- 5-S (O) 2 CF 3 -2-Py], [BE1383; 6-Me-5-S (O) 2 CF 3 -2-Py], [BE1384; 3- _{CF 3 -5-S (O)} 2 CF 3 -2-Py], [BE1385; 4-CF 3 -5-S (O) 2 CF 3 -2-Py], [BE1386; 6-CF 3 -5 _{-S (O) 2 CF 3 -2} -Py], [BE1387; 3-CN-5-S (O) 2 CF 3 -2-Py], [BE1388; 4-CN-5-S (O) 2 _{CF 3 -2-Py], [} BE1389; 6-CN-5-S (O) 2 CF 3 -2-Py], [BE1390; 3-OMe-5-S (O) 2 CF 3 -2-Py ], [BE1391; 4-OMe -5-S (O) 2 CF 3 -2-Py], [BE1392; 6-OMe-5-S (O) 2 CF ₃ -2-Py, [BE 1393; 6-S (O) ₂ CF ₃ -2-Py], [BE 1394; 3-Cl-6-S (O) ₂ CF ₃ -2-Py], [BE 1395] ; 4-Cl-6-S (O) 2 CF 3 -2-Py], [BE1396; 5-Cl-6-S (O) 2 CF 3 -2-Py], [BE1397; 3-Me-6 _{-S (O) 2 CF 3 -2} -Py], [BE1398; 4-Me-6-S (O) 2 CF 3 -2-Py], [BE1399; 5-Me-6-S (O) 2 _{CF 3 -2-Py], [} BE1400; 3-CF 3 -6-S (O) 2 CF 3 -2-Py], [BE1401; 4-CF 3 -6-S (O) 2 CF 3 -2 -Py],

_{[BE1402; 5-CF 3 -6} -S (O) 2 CF 3 -2-Py], [BE1403; 3-CN-6-S (O) 2 CF 3 -2-Py], [BE1404; 4- CN-6-S (O) 2 CF 3 -2-Py], [BE1405; 5-CN-6-S (O) 2 CF 3 -2-Py], [BE1406; 3-OMe-6-S ( O) ₂ CF ₃ -2-Py, [BE 1407; 4-OMe-6-S (O) ₂ CF ₃ -2-Py], [BE 1408; 5-OMe-6-S (O) ₂ CF ₃ − 2-Py], [BE1409; 3-CN-2-Py], [BE 1410; 4-Cl-3-CN-2-Py], [BE 1411; 5-Cl-3-CN-2-Py], [BE 1410; BE 1412; 6-Cl-3-CN-2-Py], [BE 1413; 4-Me-3-CN-2-Py], [BE 1414; 5-Me-3-CN-2-Py], [BE 1415; 6-Me-3-CN-2-Py], [BE 1416; 4-CF ₃ -3-CN-2-Py], [BE 1417; 5-CF ₃ -3-CN-2-Py], [BE 14 18; _{6-CF 3 -3-CN-} 2-Py], [BE1419; 4-CN-3-CN-2-Py], [BE1420; 5-CN-3-CN-2-Py], [BE1421; 6 -CN-3-CN-2-Py], [BE1422; 4-OMe-3-CN-2-Py], [BE1423; 5-OMe-3-CN-2-Py], [BE1424; 6-OMe -3-CN-2-Py !, [BE1425; 4-CN-2-Py], [BE1426; 3-Cl-4-CN-2-Py], [BE1427; 5-Cl-4-CN-2 -Py], [BE1428; 6-Cl-4-CN-2-Py], [BE1429; 3-Me-4-CN-2-Py], [BE1430; 5-Me-4-CN-2-Py ], [BE1431; 6-Me -4-CN-2-Py], [BE1432; 3-CF 3 -4-CN-2-Py], [BE1433; 5-CF 3 -4-CN-2-Py ], [BE1434; 6-CF 3 -4-CN-2-Py], [BE1435; 3-CN-4-CN-2-Py], [BE1436; 5-CN-4-CN-2-Py] , [BE1437; 6-CN-4-CN-2-Py], [BE1438; 3-OMe-4-CN-2-Py], [BE1439; 5-OMe-4-CN-2-Py] , [BE1440; 6-OMe-4-CN-2-Py], [BE1441; 5-CN-2-Py], [BE1442; 3-Cl-5-CN-2-Py], [BE1443; Cl-5-CN-2-Py], [BE1444; 6-Cl-5-CN-2-Py], [BE1445; 3-Me-5-CN-2-Py], [BE1446; 4-Me- 5-CN-2-Py] , [BE1447; 6-Me-5-CN-2-Py], [BE1448; 3-CF 3 -5-CN-2-Py], [BE1449; 4-CF 3 - 5-CN-2-Py] , [BE1450; 6-CF 3 -5-CN-2-Py], [BE1451; 3-CN-5-CN-2-Py], [BE1452; 4-CN-5 -CN-2-Py], [BE1453; 6-CN-5-CN-2-Py], [BE1454; 3-OMe-5-CN-2-Py], [BE1455; 4-OMe-5-CN -2-Py], [BE1456; 6-OMe-5-CN-2-Py], [BE1457; 6-CN-2-Py], [BE1458; 3-Cl-6-CN-2-Py], [BE1459; 4-Cl-6-CN-2-Py], [BE 1460; 5-Cl-6-CN-2-Py], [BE1461; 3-Me-6-CN-2-Py], [BE1462 ; 4-Me-6-CN -2-Py], [BE1463; 5-Me-6-CN-2-Py], [BE1464; 3-CF 3 -6-CN-2-Py], [BE1465; _{4-CF 3 -6-CN-} 2-Py], [BE1466; 5-CF 3 -6-CN-2-Py], [BE1467; 3-CN-6-CN-2-Py], [BE1468; 4-CN-6-CN-2-Py], [BE1469; 5-CN-6-CN-2-Py], [BE1470; 3-OMe-6-CN-2-Py], [BE1471; OMe-6-CN-2-Py], [BE1472; 5-OMe-6-CN-2-Py], [BE1473; 3-COOMe-2-Py], [BE1474; 4-Cl-3-COOMe- 2-Py], [BE1475; 5-Cl-3-COOMe-2-Py], [BE1476; 6-Cl-3-COOMe-2-Py], [BE1477; 4-Me-3-COOMe-2-] Py], [BE1478; 5-Me-3-COOMe-2-Py], [BE1479; 6-Me-3-COOMe-2-Py], [BE1480; _{4-CF 3 -3-COOMe-} 2-Py], [BE1481; 5-CF 3 -3-COOMe-2-Py], [BE1482; 6-CF 3 -3-COOMe-2-Py], [BE1483 4-CN-3-COOMe-2-Py !, [BE1484; 5-CN-3-COOMe-2-Py], [BE1485; 6-CN-3-COOMe-2-Py], [BE1486; -OMe-3-COOMe-2-Py], [BE1487; 5-OMe-3-COOMe-2-Py], [BE1488; 6-OMe-3-COOMe-2-Py], [BE1489; 4-COOMe -2-Py !, [BE1490; 3-Cl-4-COOMe-2-Py], [BE1491; 5-Cl-4-COOMe-2-Py], [BE1492; 6-Cl-4-COOMe-2 -Py], [BE1493; 3-Me-4-COOMe-2-Py], [BE1494; 5-Me-4-COOMe-2-Py], [BE1495; 6-Me-4-COOMe-2-Py] ], [BE1496; 3-CF 3 -4-COOMe-2-Py], [BE1497; 5-CF 3 -4-COOMe-2-Py], [BE1498; 6-CF 3 -4-COOMe-2- Py], [BE1499; 3-CN-4-COOMe-2-Py], [BE1500; 5-CN-4-COOMe-2-Py], [BE1501; 6-CN-4-COOMe-2-Py] ,

[BE1502; 3-OMe-4-COOMe-2-Py], [BE1503; 5-OMe-4-COOMe-2-Py], [BE1504; 6-OMe-4-COOMe-2-Py], [BE1505] 5-COOMe-2-Py !, [BE1506; 3-Cl-5-COOMe-2-Py], [BE1507; 4-Cl-5-COOMe-2-Py], [BE1508; 6-Cl-5; -COOMe-2-Py], [BE1509; 3-Me-5-COOMe-2-Py], [BE1510; 4-Me-5-COOMe-2-Py], [BE1511; 6-Me-5-COOMe -2-Py], [BE 1512; 3-CF ₃ -5-COOMe 2-Py], [BE 1513; 4-CF ₃ -5-COOMe 2-Py], [BE 1514; 6-CF ₃ -5-] COOMe-2-Py !, [BE1515; 3-CN-5-COOMe-2-Py], [BE1516; 4-CN-5-COOMe-2-Py], [BE1517; 6-CN-5-COOMe- 2-Py], [BE 1518; 3-OMe-5-COOMe-2-Py], [BE 1519; 4-OMe-5-COOMe-2-Py], [BE 1520; 6-OMe-5-COOMe-2- Py], [BE1521; 6-COOMe-2-Py], [BE1522; 3-Cl-6-COOMe-2-Py], [BE1523; 4-Cl-6-COOMe-2-Py], [BE1524; 5-Cl-6-COOMe-2-Py], [BE1525; 3-Me-6-COOMe-2-Py], [BE1526; 4-Me-6-COOMe-2-Py], [BE1527; 5- Me-6-COOMe-2- Py], [BE1528; 3-CF 3 -6-COOMe-2-Py], [BE1529; 4-CF 3 -6-COOMe-2-Py], [BE1530; 5- _{CF 3 -6-COOMe-2-} Py], [BE1531; 3-CN-6-COOMe-2-Py], [BE1532; 4-CN-6-COOMe-2-Py], [BE1533; 5-CN -6-COOMe-2-Py], [BE1534; 3-OMe-6-COOMe-2-Py], [BE1535; 4-OMe-6-COOMe-2-Py], [BE1536; 5-OMe-6 -COOMe-2-Py], [ BE1537; 4-Cl-3-NO 2 -2-Py], [BE1538; 5-C _{l-3-NO 2 -2-} Py], [BE1539; 6-Cl-3-NO 2 -2-Py], [BE1540; 4-Me-3-NO 2 -2-Py], [BE1541; 5 _{-Me-3-NO 2 -2-} Py], [BE1542; 6-Me-3-NO 2 -2-Py], [BE1543; 4-CF 3 -3-NO 2 -2-Py], [BE1544 _{; 5-CF 3 -3-NO} 2 -2-Py], [BE1545; 6-CF 3 -3-NO 2 -2-Py], [BE1546; 4-CN-3-NO 2 -2-Py] , [BE1547; 5-CN- 3-NO 2 -2-Py], [BE1548; 6-CN-3-NO 2 -2-Py], [BE1549; 4-OMe-3-NO 2 -2-Py ], [BE1550; 5-OMe -3-NO 2 -2-Py], [BE1551; 6-OMe-3-NO 2 -2-Py], [BE1552; 4-NO 2 -2-Py], [ BE1553; 3-Cl-4- NO 2 -2-Py], [BE1554; 5-Cl-4-NO 2 -2-Py], [BE1555; 6-Cl-4-NO 2 -2-Py], [BE1556; 3-Me-4 -NO 2 -2-Py], [BE1557; 5-Me-4-NO 2 -2-Py], [BE1558; 6-Me-4-NO 2 -2-Py] _{, [BE1559; 3-CF 3} -4-NO 2 -2-Py], [BE1560; 5-CF 3 -4-NO 2 -2-Py], [BE1561; 6-CF 3 -4-NO 2 - 2-Py], [BE1562; 3-CN-4-NO 2 -2-Py], [BE1563; 5-CN-4-NO 2 -2-Py], [BE1564; 6-CN-4-NO 2 -2-Py], [BE1565; 3-OMe-4-NO 2 -2-Py], [BE1566; 5-OMe-4-NO 2 -2-Py], [BE1567; 6-OMe-4-NO _{2 -2-Py], [BE1568} ; 5-NO 2 -2-Py], [BE1569; 3-Cl-5-NO 2 -2-Py], [BE1570; 4-Cl-5-NO 2 -2 -Py], [BE1571; 6- Cl-5-NO 2 -2-Py], [BE1572; 3-Me-5-NO 2 -2-Py], [BE1573; 4-Me-5-NO 2 - 2-Py], [BE 1574; 6-Me-5-NO ₂ -2-Py ], [BE1575; 3-CF 3 -5-NO 2 -2-Py], [BE1576; 4-CF 3 -5-NO 2 -2-Py], [BE1577; 6-CF 3 -5-NO 2 -2-Py], [BE1578; 3-CN-5-NO 2 -2-Py], [BE1579; 4-CN-5-NO 2 -2-Py], [BE1580; 6-CN-5-NO ₂ -2-Py !, [BE 1581; 3-OMe-5-NO ₂ -2-Py], [BE 1582; 4-OMe-5-NO ₂ -2-Py], [BE 1583; 6-OMe -5- NO ₂ -2-Py !, [BE 1584; 6-NO ₂ -2-Py], [BE 1585; 3-Cl-6-NO ₂ -2-Py], [BE 1586; 4-Cl 6-NO ₂ − 2-Py], [BE1587; 5-Cl-6-NO 2 -2-Py], [BE1588; 3-Me-6-NO 2 -2-Py], [BE1589; 4-Me-6-NO 2 -2-Py], [BE1590; 5-Me-6-NO 2 -2-Py], [BE1591; 3-CF 3 -6-NO 2 -2-Py], [BE1592; 4-CF 3 -6 _{-NO 2 -2-Py], [} BE1593; 5-CF 3 -6-NO 2 -2-Py], [BE1594; 3-CN-6-NO 2 -2-Py], [BE1595; 4-CN _{-6-NO 2 -2-Py]} , [BE1596; 5-CN-6-NO 2 -2-Py], [BE1597; 3-OMe-6-NO 2 -2-Py], [BE1598; 4- _{OMe-6-NO 2 -2-} Py], [BE1599; 5-OMe-6-NO 2 -2-Py], [BE1600; 4-Cl-3-NH 2 -2-Py], [BE1601; 5 -Cl-3-NH ₂ -2-Py],

[BE1602; 6-Cl-3 -NH 2 -2-Py], [BE1603; 4-Me-3-NH 2 -2-Py], [BE1604; 5-Me-3-NH 2 -2-Py] , [BE1605; 6-Me- 3-NH 2 -2-Py], [BE1606; 4-CF 3 -3-NH 2 -2-Py], [BE1607; 5-CF 3 -3-NH 2 -2 -Py], [BE1608; 6- CF 3 -3-NH 2 -2-Py], [BE1609; 4-CN-3-NH 2 -2-Py], [BE1610; 5-CN-3-NH 2 -2-Py], [BE1611; 6-CN-3-NH 2 -2-Py], [BE1612; 4-OMe-3-NH 2 -2-Py], [BE1613; 5-OMe-3-NH _{2 -2-Py], [BE1614} ; 6-OMe-3-NH 2 -2-Py], [BE1615; 4-NH 2 -2-Py], [BE1616; 3-Cl-4-NH 2 -2 -Py], [BE1617; 5- Cl-4-NH 2 -2-Py], [BE1618; 6-Cl-4-NH 2 -2-Py], [BE1619; 3-Me-4-NH 2 - 2-Py], [BE1620; 5-Me-4-NH 2 -2-Py], [BE1621; 6-Me-4-NH 2 -2-Py], [BE1622; 3-CF 3 -4-NH _{2 -2-Py], [BE1623} ; 5-CF 3 -4-NH 2 -2-Py], [BE1624; 6-CF 3 -4-NH 2 -2-Py], [BE1625; 3-CN- _{4-NH 2 -2-Py]} , [BE1626; 5-CN-4-NH 2 -2-Py], [BE1627; 6-CN-4-NH 2 -2-Py], [BE1628; 3-OMe _{-4-NH 2 -2-Py]} , [BE1629; 5-OMe-4-NH 2 -2-Py], [BE1630; 6-OMe-4-NH 2 -2-Py], [BE1631; 5- _{NH 2 -2-Py], [} BE1632; 3-Cl-5-NH 2 -2-Py], [BE1633; 4-Cl-5-NH 2 -2-Py], [BE1634; 6-Cl-5 _{-NH 2 -2-Py], [} BE1635; 3-Me-5-NH 2 -2-Py], [BE1636; 4-Me-5-NH 2 -2-Py], [BE1637; 6-Me- 5-NH ₂ -2-Py, [BE 1638; 3-CF ₃ -5-NH ₂ -2-Py !, [BE 1639; 4-CF ₃ -5-NH ₂ -2-Py], [BE 1640; 6-CF ₃ -5-NH ₂ -2-Py], [BE 1641; _{3-CN-5-NH 2} -2-Py], [BE1642; 4-CN-5-NH 2 -2-Py], [BE1643; 6-CN-5-NH 2 -2-Py], [BE1644 3-OMe-5-NH ₂ 2-Py !, [BE1645; 4-OMe-5-NH ₂ 2-Py], [BE 1646; 6-OMe-5-NH ₂ 2-Py], _{BE1647; 6-NH 2 -2-} Py], [BE1648; 3-Cl-6-NH 2 -2-Py], [BE1649; 4-Cl-6-NH 2 -2-Py], [BE1650; 5 _{-Cl-6-NH 2 -2-} Py], [BE1651; 3-Me-6-NH 2 -2-Py], [BE1652; 4-Me-6-NH 2 -2-Py], [BE1653; _{5-Me-6-NH 2} -2-Py], [BE1654; 3-CF 3 -6-NH 2 -2-Py], [BE1655; 4-CF 3 -6-NH 2 -2-Py], _{[BE1656; 5-CF 3 -6} -NH 2 -2-Py], [BE1657; 3-CN-6-NH 2 -2-Py], [BE1658; 4-CN-6-NH 2 -2-Py ], [BE1659; 5-CN -6-NH 2 -2-Py], [BE1660; 3-OMe-6-NH 2 -2-Py], [BE1661; 4-OMe-6-NH 2 -2- Py], [BE1662; 5- OMe-6-NH 2 -2-Py], [BE1663; 3-NHMe-2-Py], [BE1664; 4-Cl-3-NHMe-2-Py], [BE1665 5-Cl-3-NHMe-2-Py, [BE1666; 6-Cl-3-NHMe-2-Py], [BE1667; 4-Me-3-NHMe-2-Py], [BE1668; -Me-3-NHMe-2- Py], [BE1669; 6-Me-3-NHMe-2-Py], [BE1670; 4-CF 3 -3-NHMe-2-Py], [BE1671; 5- _{CF 3 -3-NHMe-2-} Py], [BE1672; 6-CF 3 -3-NHMe-2-Py], [BE1673; 4-CN-3-NHMe-2-Py], [BE1674; 5- CN-3-NHMe-2-Py], [BE1 675; 6-CN-3-NHMe-2-Py, [BE1676; 4-OMe-3-NHMe-2-Py], [BE1677; 5-OMe-3-NHMe-2-Py], [BE1678; 6-OMe-3-NHMe-2-Py, [BE1679; 4-NHMe-2-Py], [BE1680; 3-Cl-4-NHMe-2-Py], [BE1681; 5-Cl-4- NHMe-2-Py, [BE1682; 6-Cl-4-NHMe-2-Py], [BE 1683; 3-Me-4-NHMe-2-Py], [BE 1684; 5-Me-4-NHMe- 2-Py], [BE1685; 6-Me-4-NHMe-2-Py], [BE1686; 3-CF 3 -4-NHMe-2-Py], [BE1687; 5-CF 3 -4-NHMe- 2-Py], [BE1688; 6-CF 3 -4-NHMe-2-Py], [BE1689; 3-CN-4-NHMe-2-Py], [BE1690; 5-CN-4-NHMe-2 -Py], [BE1691; 6-CN-4-NHMe-2-Py], [BE1692; 3-OMe-4-NHMe-2-Py], [BE1693; 5-OMe-4-NHMe-2-Py] ], [BE1694; 6-OMe-4-NHMe-2-Py], [BE1695; 5-NHMe-2-Py], [BE1696; 3-Cl-5-NHMe-2-Py], [BE1697; 4] -Cl-5-NHMe-2-Py], [BE1698; 6-Cl-5-NHMe-2-Py], [BE1699; 3-Me-5-NHMe-2-Py], [BE1700; 4-Me -5-NHMe-2-Py !, [BE 1701; 6-Me-5-NHMe-2-Py],

_{[BE1702; 3-CF 3 -5} -NHMe-2-Py], [BE1703; 4-CF 3 -5-NHMe-2-Py], [BE1704; 6-CF 3 -5-NHMe-2-Py] , [BE 1705; 3-CN-5-NHMe-2-Py], [BE 1706; 4-CN-5-NHMe-2-Py], [BE 1707; 6-CN-5-NHMe-2-Py], [BE 1705; BE1708; 3-OMe-5-NHMe-2-Py], [BE1709; 4-OMe-5-NHMe-2-Py], [BE1710; 6-OMe-5-NHMe-2-Py], [BE1711; 6-NHMe-2-Py, [BE 1712; 3-Cl-6-NHMe-2-Py], [BE 1713; 4-Cl-6-NHMe-2-Py], [BE 1714; 5-Cl-6- NHMe-2-Py, [BE1715; 3-Me-6-NHMe-2-Py], [BE1716; 4-Me-6-NHMe-2-Py], [BE1717; 5-Me-6-NHMe- 2-Py], [BE1718; 3-CF 3 -6-NHMe-2-Py], [BE1719; 4-CF 3 -6-NHMe-2-Py], [BE1720; 5-CF 3 -6-NHMe -2-Py !, [BE1721; 3-CN-6-NHMe-2-Py], [BE1722; 4-CN-6-NHMe-2-Py], [BE1723; 5-CN-6-NHMe-2 -Py], [BE1724; 3-OMe-6-NHMe-2-Py], [BE1725; 4-OMe-6-NHMe-2-Py], [BE1726; 5-OMe-6-NHMe-2-Py ], [BE1727; 3-NMe 2 -2-Py], [BE1728; 4-Cl-3-NMe 2 -2-Py], [BE1729; 5-Cl-3-NMe 2 -2-Py], [ BE1730; 6-Cl-3- NMe 2 -2-Py], [BE1731; 4-Me-3-NMe 2 -2-Py], [BE1732; 5-Me-3-NMe 2 -2-Py], [BE1733; 6-Me-3 -NMe 2 -2-Py], [BE1734; 4-CF 3 -3-NMe 2 -2-Py], [BE1735; 5-CF 3 -3-NMe 2 -2- Py], [BE1736; 6- CF 3 -3-NMe 2 -2-Py], [BE1737; 4-CN-3-NMe 2 -2-Py], [BE1738; 5-CN-3-NMe _{2 -2-Py], [BE1739} ; 6-CN-3-NMe 2 -2-Py], [BE1740; 4-OMe-3-NMe 2 -2-Py], [BE1741; 5-OMe-3- _{NMe 2 -2-Py], [} BE1742; 6-OMe-3-NMe 2 -2-Py], [BE1743; 4-NMe 2 -2-Py], [BE1744; 3-Cl-4-NMe 2 - 2-Py], [BE1745; 5-Cl-4-NMe 2 -2-Py], [BE1746; 6-Cl-4-NMe 2 -2-Py], [BE1747; 3-Me-4-NMe 2 -2-Py], [BE1748; 5-Me-4-NMe 2 -2-Py], [BE1749; 6-Me-4-NMe 2 -2-Py], [BE1750; 3-CF 3 -4- _{NMe 2 -2-Py], [} BE1751; 5-CF 3 -4-NMe 2 -2-Py], [BE1752; 6-CF 3 -4-NMe 2 -2-Py], [BE1753; 3-CN _{-4-NMe 2 -2-Py]} , [BE1754; 5-CN-4-NMe 2 -2-Py], [BE1755; 6-CN-4-NMe 2 -2-Py], [BE1756; 3- _{OMe-4-NMe 2 -2-} Py], [BE1757; 5-OMe-4-NMe 2 -2-Py], [BE1758; 6-OMe-4-NMe 2 -2-Py], [BE1759; 5 _{-NMe 2 -2-Py], [} BE1760; 3-Cl-5-NMe 2 -2-Py], [BE1761; 4-Cl-5-NMe 2 -2-Py], [BE1762; 6-Cl- _{5-NMe 2 -2-Py]} , [BE1763; 3-Me-5-NMe 2 -2-Py], [BE1764; 4-Me-5-NMe 2 -2-Py], [BE1765; 6-Me -5-NMe ₂ -2-Py !, [BE 1766; 3-CF ₃ -5-NMe ₂ -2-Py], [BE 1767; 4-CF ₃ -5-NMe ₂ -2-Py], [BE 1768; _{6-CF 3 -5-NMe 2} -2-Py], [BE1769; 3-CN-5-NMe 2 -2-Py], [BE1770; 4-CN-5-NMe 2 -2-Py], [ BE1771; 6-CN-5- NMe 2 -2-Py], [BE1772; 3-OMe-5-NMe 2 -2-Py], [BE1773; 4-OMe-5-NMe 2 -2 -Py], [BE1774; 6- OMe-5-NMe 2 -2-Py], [BE1775; 6-NMe 2 -2-Py], [BE1776; 3-Cl-6-NMe 2 -2-Py] , [BE1777; 4-Cl- 6-NMe 2 -2-Py], [BE1778; 5-Cl-6-NMe 2 -2-Py], [BE1779; 3-Me-6-NMe 2 -2-Py ], [BE1780; 4-Me -6-NMe 2 -2-Py], [BE1781; 5-Me-6-NMe 2 -2-Py], [BE1782; 3-CF 3 -6-NMe 2 -2 -Py], [BE1783; 4- CF 3 -6-NMe 2 -2-Py], [BE1784; 5-CF 3 -6-NMe 2 -2-Py], [BE1785; 3-CN-6-NMe ₂ -2-Py !, [BE 1 786; 4-CN-6-NMe ₂ -2-Py], [BE 1787; 5-CN-6-NMe ₂ -2-Py], [BE 1 788; 3-OMe -6- _{NMe 2 -2-Py], [} BE1789; 4-OMe-6-NMe 2 -2-Py], [BE1790; 5-OMe-6-NMe 2 -2-Py], [BE1791; 3-ACNH-2 4-Py], [BE1792; 4-Cl-3-ACNH-2-Py], [BE1793; 5-Cl-3-ACNH-2-Py], [BE1794; 6-Cl-3-ACNH-2-Py ], [BE1795; 4-Me-3-ACNH-2-Py], [BE1796; 5-Me-3-ACNH-2-Py], [BE1797; 6-Me-3-ACNH-2-Py], _{[BE1798; 4-CF 3 -3} -ACNH-2-Py], [BE1799; 5-CF 3 -3-ACNH-2-Py], [BE1800; 6-CF 3 -3-ACNH-2-Py] , [BE 1801; 4-CN-3-ACNH-2-Py],

[BE1802; 5-CN-3-ACNH-2-Py], [BE1803; 6-CN-3-ACNH-2-Py], [BE1804; 4-OMe-3-ACNH-2-Py], [BE1805 5-OMe-3-ACNH-2-Py !, [BE1806; 6-OMe-3-ACNH-2-Py], [BE1807; 4-ACNH-2-Py], [BE1808; 3-Cl-4; -ACNH-2-Py], [BE1809; 5-Cl-4-ACNH-2-Py], [BE1810; 6-Cl-4-ACNH-2-Py], [BE1811; 3-Me-4-ACNH -2-Py !, [BE 1812; 5-Me-4-ACNH-2-Py], [BE 1813; 6-Me-4-ACNH-2-Py], [BE 1814; 3-CF ₃ -4-ACNH- 2-Py], [BE1815; 5-CF 3 -4-ACNH-2-Py], [BE1816; 6-CF 3 -4-ACNH-2-Py], [BE1817; 3-CN-4-ACNH- 2-Py], [BE1818; 5-CN-4-ACNH-2-Py], [BE1819; 6-CN-4-ACNH-2-Py], [BE1820; 3-OMe-4-ACNH-2-] Py], [BE1821; 5-OMe-4-ACNH-2-Py], [BE1822; 6-OMe-4-ACNH-2-Py], [BE1823; 5-ACNH-2-Py], [BE1824; 3-Cl-5-ACNH-2-Py], [BE1825; 4-Cl-5-ACNH-2-Py], [BE1826; 6-Cl-5-ACNH-2-Py], [BE1827; Me-5-ACNH-2- Py], [BE1828; 4-Me-5-ACNH-2-Py], [BE1829; 6-Me-5-ACNH-2-Py], [BE1830; 3-CF 3 -5-ACNH-2-Py] , [BE1831; 4-CF 3 -5-ACNH-2-Py], [BE1832; 6-CF 3 -5-ACNH-2-Py], [BE1833; 3-CN -5-ACNH-2-Py, [BE1834; 4-CN-5-ACNH-2-Py], [BE1835; 6-CN-5-ACNH-2-Py], [BE1836; 3-OMe-5 -ACNH-2-Py], [BE 1837; 4-OMe-5-ACNH-2-Py], [BE 1838; 6-OMe-5-ACNH-2-Py], [BE 1839; 6-ACNH-2-Py ], [BE1840; 3-Cl-6-ACNH-2-Py], [BE1841; 4-Cl-6-ACNH-2-Py], [BE1842; 5-Cl-6-ACNH-2-Py], [BE1843 3-Me-6-ACNH-2-Py !, [BE1844; 4-Me-6-ACNH-2-Py], [BE1845; 5-Me-6-ACNH-2-Py], [BE1846; _{-CF 3 -6-ACNH-2-} Py], [BE1847; 4-CF 3 -6-ACNH-2-Py], [BE1848; 5-CF 3 -6-ACNH-2-Py], [BE1849; 3-CN-6-ACNH-2-Py], [BE1850; 4-CN-6-ACNH-2-Py], [BE1851; 5-CN-6-ACNH-2-Py], [BE1852; OMe-6-ACNH-2-Py !, [BE 1853; 4-OMe-6-ACNH-2-Py], [BE 1854; 5-OMe-6-ACNH-2-Py], [BE 1855; 3- (N (Ac) (Me))-2-Py] [BE1856; 4-Cl-3- (N (Ac) (Me))-2-Py], [BE1857; 5-Cl-3- (N (Ac)) (Me))-2-Py], [BE1858; 6-Cl-3- (N (Ac) (Me))-2-Py], [BE1859; 4-Me-3- (N (Ac) (Me) )) 2-Py], [BE1860; 5-Me-3- (N (Ac) (Me))-2-Py], [BE1861; 6-Me-3- (N (Ac) (Me)) -2-Py], [BE1862; 4-CF 3 -3- (N (Ac) (Me)) - 2-Py], [BE1863; 5-CF 3 -3- (N (Ac) (Me)) -2-Py !, [BE 1864; 6-CF ₃ -3- (N (Ac) (Me))-2-Py], [BE 1865; 4-CN-3- (N (Ac) (Me))- 2-Py], [BE1866; 5-CN-3- (N (Ac) (Me))-2-Py], [BE1867; 6-CN-3- (N (Ac) (Me))-2-] Py], [BE1868; 4-OMe-3- (N (Ac) (Me))-2-Py], [BE1869; 5-OMe-3- (N (Ac) (Me))-2-Py] , [BE1870; 6-OMe-3- (N (Ac) (Me))-2-Py], [BE1871; 4- (N (Ac) (Me))-2-Py], [BE1872; Cl-4- (N (Ac) (Me))-2-Py], [BE 1873; 5-Cl-4- (N (Ac) (Me))-2-Py], [BE1874; 6-Cl-4- (N (Ac) (Me))-2-Py], [BE1875; 3-Me-4- (N (Ac) (Me))-2-Py], [BE1876; 5-Me-4- (N (Ac) (Me))-2-Py], [BE1877; 6- Me-4- (N (Ac) (Me)) - 2-Py], [BE1878; 3-CF 3 -4- (N (Ac) (Me)) - 2-Py], [BE1879; 5-CF _{3 -4- (N (Ac) (} Me)) - 2-Py], [BE1880; 6-CF 3 -4- (N (Ac) (Me)) - 2-Py], [BE1881; 3-CN -4- (N (Ac) (Me))-2-Py], [BE1882; 5-CN-4- (N (Ac) (Me))-2-Py], [BE 1883; 6-CN-4 -(N (Ac) (Me))-2-Py], [BE1884; 3-OMe-4- (N (Ac) (Me))-2-Py], [BE1885; 5-OMe-4- (4) N (Ac) (Me))-2-Py], [BE 1886; 6-OMe-4- (N (Ac) (Me))-2-Py], [BE 1887; 5- (N (Ac) (Me) )) 2-Py], [BE 1888; 3-Cl-5- (N (Ac) (Me))-2-Py], [BE 1889; 4-Cl-5- (N (Ac) (Me)) -2-Py], [BE1890; 6-Cl-5- (N (Ac) (Me))-2-Py], [BE1891; 3-Me-5- (N (Ac) (Me))-2 -Py], [BE1892; 4-Me-5- (N (Ac) (Me))-2-Py], [BE1893; 6-Me-5- (N (Ac) (Me))-2-Py ], [BE1894; 3-CF 3 -5- (N (Ac) (Me)) - 2-Py], [BE1895; 4-CF 3 -5- (N (Ac) (Me)) - 2-Py ], [BE1896; 6-CF 3 -5- (N (Ac) (Me)) - 2-Py], [BE1897; 3-CN-5- (N (Ac) (Me)) - 2-Py] , [BE1898; 4-CN-5- (N (Ac) (Me))-2-Py], [BE1899; 6-CN-5- (N (Ac) (Me))-2-Py], [BE18 9; BE 1900; 3-OMe-5- (N (Ac) (Me))-2-Py], [BE1901; 4-OMe-5- (N (Ac) (Me))-2-Py],

[BE1902; 6-OMe-5- (N (Ac) (Me))-2-Py], [BE1903; 6- (N (Ac) (Me))-2-Py], [BE1904; 3-Cl -6- (N (Ac) (Me))-2-Py], [BE 1905; 4-Cl-6- (N (Ac) (Me))-2-Py], [BE 1906; 5-Cl-6 -(N (Ac) (Me))-2-Py], [BE1907; 3-Me-6- (N (Ac) (Me))-2-Py], [BE1908; 4-Me-6- ( N (Ac) (Me)) - 2-Py], [BE1909; 5-Me-6- (N (Ac) (Me)) - 2-Py], [BE1910; 3-CF 3 -6- (N (Ac) (Me)) - 2-Py], [BE1911; 4-CF 3 -6- (N (Ac) (Me)) - 2-Py], [BE1912; 5-CF 3 -6- (N (Ac) (Me))-2-Py], [BE1913; 3-CN-6- (N (Ac) (Me))-2-Py], [BE1914; 4-CN-6- (N (Ac) ) (Me))-2-Py], [BE1915; 5-CN-6- (N (Ac) (Me))-2-Py], [BE1916; 3-OMe-6- (N (Ac) ( Me))-2-Py], [BE1917; 4-OMe-6- (N (Ac) (Me))-2-Py], [BE1918; 5-OMe-6- (N (Ac) (Me)) )-[2-Py], [BE1919; 3-AC-2-Py], [BE1920; 4-Cl-3-AC-2-Py], [BE1921; 5-Cl-3-AC-2-Py] , [BE1922; 6-Cl-3-AC-2-Py], [BE1923; 4-Me-3-AC-2-Py], [BE1924; 5-Me-3-AC-2-Py], [BE2 922; BE 1925; 6-Me-3-AC-2-Py], [BE 1926; 4-CF ₃ -3-AC-2-Py], [BE 1 927; 5-CF ₃ -3-AC-2-Py], [BE 1 927; _{BE1928; 6-CF 3 -3-} AC-2-Py], [BE1929; 4-CN-3-AC-2-Py], [BE1930; 5-CN-3-AC-2-Py], [BE1931 6-CN-3-AC-2-Py !, [BE1932; 4-OMe-3-AC-2-Py], [BE1933; 5-OMe-3-AC-2-Py], [BE1934; -OMe-3-AC-2-Py], [BE 1935; 4-AC-2-Py], [BE 1936; 3-Cl-4-AC-2-P y], [BE1937; 5-Cl-4-AC-2-Py], [BE1938; 6-Cl-4-AC-2-Py], [BE1939; 3-Me-4-AC-2-Py] , [BE1940; 5-Me- 4-AC-2-Py], [BE1941; 6-Me-4-AC-2-Py], [BE1942; 3-CF 3 -4-AC-2-Py], _{[BE1943; 5-CF 3 -4} -AC-2-Py], [BE1944; 6-CF 3 -4-AC-2-Py], [BE1945; 3-CN-4-AC-2-Py], [BE1946; 5-CN-4-AC-2-Py], [BE1947; 6-CN-4-AC-2-Py], [BE1948; 3-OMe-4-AC-2-Py], [BE1949] 5-OMe-4-AC-2-Py !, [BE1950; 6-OMe-4-AC-2-Py], [BE1951; 5-AC-2-Py], [BE1952; 3-Cl-5; -AC-2-Py], [BE1953; 4-Cl-5-AC-2-Py], [BE1954; 6-Cl-5-AC-2-Py], [BE1955; 3-Me-5-AC -2-Py !, [BE1956; 4-Me-5-AC-2-Py], [BE1957; 6-Me-5-AC-2-Py], [BE1958; 3-CF ₃ -5-AC- 2-Py], [BE1959; 4-CF 3 -5-AC-2-Py], [BE1960; 6-CF 3 -5-AC-2-Py], [BE1961; 3-CN-5-AC- 2-Py], [BE1962; 4-CN-5-AC-2-Py], [BE1963; 6-CN-5-AC-2-Py], [BE1964] 3-OMe-5-AC-2- Py], [BE 1965; 4-OMe-5-AC-2-Py], [BE 1966; 6-OMe-5-AC-2-Py], [BE 1967; 6-AC-2-Py], [BE 1968; 3-Cl-6-AC-2-Py], [BE 1969; 4-Cl-6-AC-2-Py], [BE1970; 5-Cl-6-AC-2-Py], [BE 1971; 3- Me-6-AC-2-Py], [BE 1972; 4-Me-6-AC-2-Py], [BE 1973; 5-Me-6-AC-2-Py], [BE 1974; 3-CF ₃ -6-AC-2-Py] , [BE1975; 4-CF 3 -6-AC-2-Py], [BE1976; 5-CF 3 -6-AC-2-Py], [BE1977; 3-CN -6 -AC-2-Py], [BE1978; 4-CN-6-AC-2-Py], [BE 1979; 5-CN-6-AC-2-Py], [BE1980; 3-OMe-6-AC -2-Py], [BE1981; 4-OMe-6-AC-2-Py], [BE1982; 5-OMe-6-AC-2-Py], [BE1983; 2-F-3-Py], [BE1984; 4-Cl-2-F-3-Py], [BE1985; 5-Cl-2-F-3-Py], [BE1986; 6-Cl-2-F-3-Py], [BE 1987] 4-Me-2-F-3-Py !, [BE1988; 5-Me-2-F-3-Py], [BE1989; 6-Me-2-F-3-Py], [BE1990; _{-CF 3 -2-F-3-} Py], [BE1991; 5-CF 3 -2-F-3-Py], [BE1992; 6-CF 3 -2-F-3-Py], [BE1993; 4-CN-2-F-3-Py], [BE 1994; 5-CN-2-F-3-Py], [BE 1995; 6-CN-2-F-3-Py], [BE 1996; OMe-2-F-3-Py], [BE 1997; 5-OMe-2-F-3-Py], [BE1998; 6-OMe-2-F-3-Py], [BE 1999; 4-F- 3-Py], [BE2000; 2-Cl-4-F-3-Py], [BE2001; 5-Cl-4-F-3-Py],

[BE2002; 6-Cl-4-F-3-Py], [BE2003; 2-Me-4-F-3-Py], [BE2004; 5-Me-4-F-3-Py], [BE2005] ; 6-Me-4-F -3-Py], [BE2006; 2-CF 3 -4-F-3-Py], [BE2007; 5-CF 3 -4-F-3-Py], [BE2008 _{; 6-CF 3 -4-F} -3-Py], [BE2009; 2-CN-4-F-3-Py], [BE2010; 5-CN-4-F-3-Py], [BE2011; 6-CN-4-F-3-Py], [BE2012; 2-OMe-4-F-3-Py], [BE2013; 5-OMe-4-F-3-Py], [BE2014; 6- OMe-4-F-3-Py], [BE2015; 5-F-3-Py], [BE2016; 2-Cl-5-F-3-Py], [BE 2017; 4-Cl-5-F- 3-Py], [BE 2018; 6-Cl-5-F-3-Py], [BE 2019; 2-Me-5-F-3-Py], [BE 2020; 4-Me-5-F-3- Py], [BE2021; 6- Me-5-F-3-Py], [BE2022; 2-CF 3 -5-F-3-Py], [BE2023; 4-CF 3 -5-F-3- Py], [BE2024; 6- CF 3 -5-F-3-Py], [BE2025; 2-CN-5-F-3-Py], [BE2026; 4-CN-5-F-3-Py ], [BE2027; 6-CN-5-F-3-Py], [BE2028; 2-OMe-5-F-3-Py], [BE2029; 4-OMe-5-F-3-Py], [BE2030; 6-OMe-5-F-3-Py], [BE2031; 6-F-3-Py], [BE2032; 2-Cl-6-F-3-Py], [BE2033; 4-Cl -6-F-3-Py !, [BE2034; 5-Cl-6-F-3-Py], [BE2035; 2-Me-6-F-3-Py], [BE 2036; 4-Me-6 -F-3-Py], [ BE2037; 5-Me-6-F-3-Py], [BE2038; 2-CF 3 -6-F-3-Py], [BE2039; 4-CF 3 -6 -F-3-Py], [ BE2040; 5-CF 3 -6-F-3-Py], [BE2041; 2-CN-6-F-3-Py], [BE2042; 4-CN-6- F-3-Py], [BE2043; 5-CN-6-F-3-Py], [BE2044; 2-O Me-6-F-3-Py], [BE 2045; 4-OMe-6-F-3-Py], [BE 2046; 5-OMe-6-F-3-Py], [BE 2047; 2-Cl- 3-Py], [BE 2048; 4-Cl-2-Cl-3-Py], [BE 2049; 5-Cl-2-Cl-3-Py], [BE 2050; 6-Cl-2-Cl-3- Py], [BE2051; 4-Me-2-Cl-3-Py], [BE2052; 5-Me-2-Cl-3-Py], [BE2053; 6-Me-2-Cl-3-Py] , [BE 2054; 4-CF ₃ -2-Cl-3-Py], [BE 2055; 5-CF ₃ -2-Cl-3-Py], [BE 2056; 6-CF ₃ -2-Cl-3-Py] ], [BE 2057; 4-CN-2-Cl-3-Py], [BE 2058; 5-CN-2-Cl-3-Py], [BE 2059; 6-CN-2-Cl-3-Py], [BE2060; 4-OMe-2-Cl-3-Py], [BE2061; 5-OMe-2-Cl-3-Py], [BE2062; 6-OMe-2-Cl-3-Py], [BE2063 4-Cl-3-Py !, [BE 2064; 2-Cl-4-Cl-3-Py], [BE 2065; 5-Cl-4-Cl-3-Py], [BE 2066; 6-Cl-4 -Cl-3-Py], [BE 2067; 2-Me-4-Cl-3-Py], [BE 2068; 5-Me-4-Cl-3-Py], [BE 2069; 6-Me-4-Cl -3-Py], [BE2070; 2-CF 3 -4-Cl-3-Py], [BE2071; 5-CF 3 -4-Cl-3-Py], [BE2072; 6-CF 3 -4- Cl-3-Py], [BE 2073; 2-CN-4-Cl-3-Py], [BE 2074; 5-CN-4-Cl-3-Py], [BE 2075; 6-CN-4-Cl- 3-Py], [BE2076; 2-OMe-4-Cl-3-Py], [BE2077; 5-OMe-4-Cl-3-Py], [BE2078; 6-OMe-4-Cl-3- Py], [BE2079; 5-Cl-3-Py], [BE2080; 4-Cl-5-Cl-3-Py], [BE2081; 5-Cl-5-Cl-3-Py], [BE2082; 6-Cl-5-Cl-3-Py !, [BE 2083; 4-Me-5-Cl-3-Py], [BE 2084; 5-Me-5-Cl-3-Py], [BE 2085; 6- Me-5-Cl- 3-Py], [BE2086; 4-CF 3 -5-Cl-3-Py], [BE2087; 5-CF 3 -5-Cl-3-Py], [BE2088; 6-CF 3 -5-Cl -3-Py !, [BE 2089; 4-CN-5-Cl-3-Py], [BE 2090; 3-CN-5-Cl-3-Py], [BE 2091; 6-CN-5-Cl-3 -Py], [BE 2092; 4-OMe-5-Cl-3-Py], [BE 2093; 5-OMe-5-Cl-3-Py], [BE 2094; 6-OMe-5-Cl-3-Py ], [BE 2095; 6-Cl-3-Py], [BE 2096; 2-Cl-6-Cl-3-Py], [BE 2097; 4-Cl-6-Cl-3-Py], [BE 2098; 5] -Cl-6-Cl-3-Py], [BE 2099; 2-Me-6-Cl-3-Py], [BE 2100; 4-Me-6-Cl-3-Py], [BE 2101; 5-Me -6-Cl-3-Py],

_{[BE2102; 2-CF 3 -6} -Cl-3-Py], [BE2103; 4-CF 3 -6-Cl-3-Py], [BE2104; 5-CF 3 -6-Cl-3-Py] , [BE2105; 2-CN-6-Cl-3-Py], [BE2106; 4-CN-6-Cl-3-Py], [BE2107; 5-CN-6-Cl-3-Py], [BE2 10; BE2108; 2-OMe-6-Cl-3-Py], [BE2109; 4-OMe-6-Cl-3-Py], [BE2110; 5-OMe-6-Cl-3-Py], [BE2111; 2-Br-3-Py, [BE2112; 4-Cl-2-Br-3-Py], [BE2113; 5-Cl-2-Br-3-Py], [BE2114; 6-Cl-2- Br-3-Py, [BE2115; 4-Me-2-Br-3-Py], [BE2116; 5-Me-2-Br-3-Py], [BE2117; 6-Me-2-Br- 3-Py], [BE2118; 4-CF 3 -2-Br-3-Py], [BE2119; 5-CF 3 -2-Br-3-Py], [BE2120; 6-CF 3 -2-Br -3-Py], [BE2121; 4-CN-2-Br-3-Py], [BE2122; 5-CN-2-Br-3-Py], [BE2123; 6-CN-2-Br-3 4-Pe], [BE2124; 4-OMe-2-Br-3-Py], [BE2 125; 5-OMe-2-Br-3-Py], [BE 2126; 6-OMe-2-Br-3-Py ], [BE2127; 4-Br-3-Py], [BE2128; 2-Cl-4-Br-3-Py], [BE2129; 5-Cl-4-Br-3-Py], [BE2130; 6] -Cl-4-Br-3-Py], [BE2131; 2-Me-4-Br-3-Py], [BE2132; 5-Me-4-Br-3-Py], [BE2133; 6-Me -4-Br-3-Py] , [BE2134; 2-CF 3 -4-Br-3-Py], [BE2135; 5-CF 3 -4-Br-3-Py], [BE2136; 6-CF _3- 4-Br-3-Py], [BE 2137; 2-CN-4-Br-3-Py], [BE 2138; 5-CN-4-Br-3-Py], [BE 2139; 6-CN- 4-Br-3-Py !, [BE 2140; 2-OMe-4-Br-3-Py], [BE 2141; 5-OMe-4-Br-3-Py], [BE 2142; 6-OMe-4 -Br-3-Py], [BE2143; 5-Br-3-Py], [BE2144; 2-Cl-5-Br-3-Py], [BE2145; 4-Cl-5-Br-3-Py ], [BE2146; 6-Cl-5-Br-3-Py], [BE2147; 2-Me-5-Br-3-Py], [BE2148; 4-Me-5-Br-3-Py], [BE2149; 6-Me-5 -Br-3-Py], [BE2150; 2-CF 3 -5-Br-3-Py], [BE2151; 4-CF 3 -5-Br-3-Py], _{[BE2152; 6-CF 3 -5} -Br-3-Py], [BE2153; 2-CN-5-Br-3-Py], [BE2154; 4-CN-5-Br-3-Py], [ BE 2 155; 6-CN-5-Br-3-Py], [BE 2156; 2-OMe-5-Br-3-Py], [BE 2 157; 4-OMe-5-Br-3-Py], [BE 2158; 6-OMe-5-Br-3-Py], [BE2159; 6-Br-3-Py], [BE2160; 2-Cl-6-Br-3-Py], [BE2161; 4-Cl-6- Br-3-Py, [BE2162; 5-Cl-6-Br-3-Py], [BE2163; 2-Me-6-Br-3-Py], [BE2164; 4-Me-6-Br- 3-Py], [BE2165; 5-Me-6-Br-3-Py], [BE2166; 2-CF 3 -6-Br-3-Py], [BE2167; 4-CF 3 -6-Br- 3-Py], [BE2168; 5-CF 3 -6-Br-3-Py], [BE2169; 2-CN-6-Br-3-Py], [BE2170; 4-CN-6-Br-3 -Py], [BE 2171; 5-CN-6-Br-3-Py], [BE 2172; 2-OMe-6-Br-3-Py], [BE 2173; 4-OMe-6-Br-3-Py ], [BE2174; 5-OMe-6-Br-3-Py], [BE2175; 2-I-3-Py], [BE 2176; 4-Cl-2-I-3-Py], [BE 2177; 5] -Cl-2-I-3-Py, [BE2178; 6-Cl-2-I-3-Py], [BE2179; 4-Me-2-I-3-Py], [BE2180; 5-Me -2-I-3-Py !, [BE2181; 6-Me-2-I-3-Py], [BE2182; 4-CF ₃ -2-I-3-Py], [BE 2183; 5-CF ₃ -2-I-3-Py], _{[BE2184; 6-CF 3 -2} -I-3-Py], [BE2185; 4-CN-2-I-3-Py], [BE2186; 5-CN-2-I-3-Py], [ BE 2187; 6-CN-2-I-3-Py], [BE 2188; 4-OMe-2-I-3-Py], [BE 2189; 5-OMe-2-I-3-Py], [BE 2190; 6-OMe-2-I-3-Py, [BE2191; 4-I-3-Py], [BE2192; 2-Cl-4-I-3-Py], [BE2193; 5-Cl-4- I-3-Py, [BE2194; 6-Cl-4-I-3-Py], [BE2195; 2-Me-4-I-3-Py], [BE2196; 5-Me-4-I- 3-Py], [BE2197; 6-Me-4-I-3-Py], [BE2198; 2-CF 3 -4-I-3-Py], [BE2199; 5-CF 3 -4-I- 3-Py], [BE2200; 6-CF 3 -4-I-3-Py], [BE2201; 2-CN-4-I-3-Py],

[BE2202; 5-CN-4-I-3-Py], [BE 2203; 6-CN-4-I-3-Py], [BE 2204; 2-OMe-4-I-3-Py], [BE 2205] 5-OMe-4-I-3-Py !, [BE2206; 6-OMe-4-I-3-Py], [BE2207; 5-I-3-Py], [BE2208; 2-Cl-5; -I-3-Py, [BE2209; 4-Cl-5-I-3-Py], [BE2210; 6-Cl-5-I-3-Py], [BE2211; 2-Me-5-I -3-Py], [BE2212; 4-Me-5-I-3-Py], [BE2213; 6-Me-5-I-3-Py], [BE2214; 2-CF 3 -5-I- 3-Py], [BE2215; 4-CF 3 -5-I-3-Py], [BE2216; 6-CF 3 -5-I-3-Py], [BE2217; 2-CN-5-I- 3-Py], [BE2218; 4-CN-5-I-3-Py], [BE2219; 6-CN-5-I-3-Py], [BE2220; 2-OMe-5-I-3-3 Py], [BE2221; 4-OMe-5-I-3-Py], [BE2222; 6-OMe-5-I-3-Py], [BE2223; 6-I-3-Py], [BE2224; 2-Cl-6-I-3-Py, [BE2225; 4-Cl-6-I-3-Py], [BE2226; 5-Cl-6-I-3-Py], [BE2227; 2- Me-6-I-3- Py], [BE2228; 4-Me-6-I-3-Py], [BE2229; 5-Me-6-I-3-Py], [BE2230; 2-CF 3 -6-I-3-Py], [BE 2231; 4-CF ₃ -6-I-3-Py], [BE 2232; 5-CF ₃ -6-I-3-Py], [BE 2233; 2-CN -6-I-3-Py], [BE2234; 4-CN-6-I-3-Py], [BE2235; 5-CN-6-I-3-Py], [BE2236; 2-OMe-6 -I-3-Py, [BE2237; 4-OMe-6-I-3-Py], [BE2238; 5-OMe-6-I-3-Py], [BE2239; 2-Me-3-Py ], [BE2240; 4-Cl-2-Me-3-Py], [BE2241; 5-Cl-2-Me-3-Py], [BE2242; 6-Cl-2-Me-3-Py], [BE2243; 4-Me-2-Me-3-Py], [BE2244; 5-Me-2-Me -3-Py], [BE2245; 6-Me-2-Me-3-Py], [BE2246; 4-CF 3 -2-Me-3-Py], [BE2247; 5-CF 3 -2-Me -3-Py], [BE2248; 6-CF 3 -2-Me-3-Py], [BE2249; 4-CN-2-Me-3-Py], [BE2250; 5-CN-2-Me- 3-Py], [BE2251; 6-CN-2-Me-3-Py], [BE2252; 4-OMe-2-Me-3-Py], [BE2253; 5-OMe-2-Me-3- Py], [BE2254; 6-OMe-2-Me-3-Py], [BE2255; 4-Me-3-Py], [BE2256; 2-Cl-4-Me-3-Py], [BE2257; 5-Cl-4-Me-3-Py], [BE2258; 6-Cl-4-Me-3-Py], [BE2259; 2-Me-4-Me-3-Py], [BE2260; 5- Me-4-Me-3- Py], [BE2261; 6-Me-4-Me-3-Py], [BE2262; 2-CF 3 -4-Me-3-Py], [BE2263; 5-CF _{3 -4-Me-3-Py} ], [BE2264; 6-CF 3 -4-Me-3-Py], [BE2265; 2-CN-4-Me-3-Py], [BE2266; 5-CN -4-Me-3-Py], [BE2267; 6-CN-4-Me-3-Py], [BE2268; 2-OMe-4-Me-3-Py], [BE2269; 5-OMe-4 -Me-3-Py], [BE2270; 6-OMe-4-Me-3-Py], [BE2271; 5-Me-3-Py], [BE 2272; 2-Cl-5-Me-3-Py ], [BE2273; 4-Cl-5-Me-3-Py], [BE2274; 6-Cl-5-Me-3-Py], [BE2275; 2-Me-5-Me-3-Py], [BE2276; 4-Me-5 -Me-3-Py], [BE2277; 6-Me-5-Me-3-Py], [BE2278; 2-CF 3 -5-Me-3-Py], [ _{BE2279; 4-CF 3 -5-} Me-3-Py], [BE2280; 6-CF 3 -5-Me-3-Py], [BE2281; 2-CN-5-Me-3-Py], [ BE2282; 4-CN-5-Me-3-Py], [BE2283; 6-CN-5-Me-3-Py], [BE2284; 2-OMe-5-Me-3-Py], [BE2285; Four -OMe-5-Me-3-Py], [BE2286; 6-OMe-5-Me-3-Py], [BE2287; 6-Me-3-Py], [BE2288; 2-Cl-6-Me -3-Py], [BE2289; 4-Cl-6-Me-3-Py], [BE2290; 5-Cl-6-Me-3-Py], [BE 2291; 2-Me-6-Me-3 -Py], [BE2292; 4- Me-6-Me-3-Py], [BE2293; 5-Me-6-Me-3-Py], [BE2294; 2-CF 3 -6-Me-3- Py], [BE2295; 4- CF 3 -6-Me-3-Py], [BE2296; 5-CF 3 -6-Me-3-Py], [BE2297; 2-CN-6-Me-3- Py], [BE2298; 4-CN-6-Me-3-Py], [BE2299; 5-CN-6-Me-3-Py], [BE2300; 2-OMe-6-Me-3-Py] , [BE 2301; 4-OMe-6-Me-3-Py],

[BE 2302; 5-OMe-6-Me-3-Py], [BE 2303; 2-OMe-3-Py], [BE 2304; 4-Cl-2-OMe-3-Py], [BE 2 305; 5-Cl -2-OMe-3-Py !, [BE2306; 6-Cl-2-OMe-3-Py], [BE2307; 4-Me-2-OMe-3-Py], [BE2308; 5-Me-2 -OMe-3-Py], [ BE2309; 6-Me-2-OMe-3-Py], [BE2310; 4-CF 3 -2-OMe-3-Py], [BE2311; 5-CF 3 -2 -OMe-3-Py], [ BE2312; 6-CF 3 -2-OMe-3-Py], [BE2313; 4-CN-2-OMe-3-Py], [BE2314; 5-CN-2- OMe-3-Py !, [BE2315; 6-CN-2-OMe-3-Py], [BE2316; 4-OMe-2-OMe-3-Py], [BE2317; 5-OMe-2-OMe- 3-Py], [BE2318; 6-OMe-2-OMe-3-Py], [BE2319; 4-OMe-3-Py], [BE2320; 2-Cl-4-OMe-3-Py], [BE2 320; BE2321; 5-Cl-4-OMe-3-Py], [BE2322; 6-Cl-4-OMe-3-Py], [BE2323; 2-Me-4-OMe-3-Py], [BE2324; 5-Me-4-OMe- 3-Py], [BE2325; 6-Me-4-OMe-3-Py], [BE2326; 2-CF 3 -4-OMe-3-Py], [BE2327; 5 _{-CF 3 -4-OMe-3-} Py], [BE2328; 6-CF 3 -4-OMe-3-Py], [BE2329; 2-CN-4-OMe-3-Py], [BE2330; 5 -CN-4-OMe-3-Py], [BE2331; 6-CN-4-OMe-3-Py], [BE2332; 2-OMe-4-OMe-3-Py], [BE2333; 5-OMe -4-OMe-3-Py !, [BE2334; 6-OMe-4-OMe-3-Py], [BE2335; 5-OMe-3-Py], [BE2336; 2-Cl-5-OMe-3 -Py], [BE2337; 4-Cl-5-OMe-3-Py], [BE2338; 6-Cl-5-OMe-3-Py], [BE2339; 2-Me-5-OMe-3-Py ], [BE2340; 4-Me-5-OMe-3-Py], [BE2341; 6-Me-5-O Me-3-Py], [ BE2342; 2-CF 3 -5-OMe-3-Py], [BE2343; 4-CF 3 -5-OMe-3-Py], [BE2344; 6-CF 3 -5 -OMe-3-Py], [BE2345; 2-CN-5-OMe-3-Py], [BE2346; 4-CN-5-OMe-3-Py], [BE2347; 6-CN-5-OMe -3-Py], [BE2348; 2-OMe-5-OMe-3-Py], [BE2349; 4-OMe-5-OMe-3-Py], [BE2350; 6-OMe-5-OMe-3 -Py], [BE2351; 6-OMe-3-Py], [BE2352; 2-Cl-6-OMe-3-Py], [BE2353; 4-Cl-6-OMe-3-Py], [BE2354] 5-Cl-6-OMe-3-Py, [BE2355; 2-Me-6-OMe-3-Py], [BE2356; 4-Me-6-OMe-3-Py], [BE2357; -Me-6-OMe-3- Py], [BE2358; 2-CF 3 -6-OMe-3-Py], [BE2359; 4-CF 3 -6-OMe-3-Py], [BE2360; 5 _{-CF 3 -6-OMe-3-} Py], [BE2361; 2-CN-6-OMe-3-Py], [BE2362; 4-CN-6-OMe-3-Py], [BE2363; 5- CN-6-OMe-3-Py], [BE2364; 2-OMe-6-OMe-3-Py], [BE2365; 4-OMe-6-OMe-3-Py], [BE2366; 5-OMe- 6-OMe-3-Py] , [BE2367; 2-CF 3 -3-Py], [BE2368; 4-Cl-2-CF 3 -3-Py], [BE2369; 5-Cl-2-CF 3 -3-Py], [BE2370; 6-Cl-2-CF 3 -3-Py], [BE2371; 4-Me-2-CF 3 -3-Py], [BE2372; 5-Me-2-CF _{3 -3-Py], [BE2373} ; 6-Me-2-CF 3 -3-Py], [BE2374; 4-CF 3 -2-CF 3 -3-Py], [BE2375; 5-CF 3 - _{2-CF 3 -3-Py]} , [BE2376; 6-CF 3 -2-CF 3 -3-Py], [BE2377; 4-CN-2-CF 3 -3-Py], [BE2378; 5- _{CN-2-CF 3 -3-} Py], [BE2379; 6-CN-2-CF 3 -3-Py], [BE2380; 4-OMe-2-CF 3 -3-Py], [BE2381; 5-OMe-2-CF 3 -3-Py], [BE2382; 6-OMe-2-CF _{3 -3-Py], [BE2383} ; 4-CF 3 -3-Py], [BE2384; 2-Cl-4-CF 3 -3-Py], [BE2385; 5-Cl-4-CF 3 -3 -Py], [BE2386; 6- Cl-4-CF 3 -3-Py], [BE2387; 2-Me-4-CF 3 -3-Py], [BE2388; 5-Me-4-CF 3 - 3-Py], [BE2389; 6-Me-4-CF 3 -3-Py], [BE2390; 2-CF 3 -4-CF 3 -3-Py], [BE2391; 5-CF 3 -4- _{CF 3 -3-Py], [} BE2392; 6-CF 3 -4-CF 3 -3-Py], [BE2393; 2-CN-4-CF 3 -3-Py], [BE2394; 5-CN- _{4-CF 3 -3-Py]} , [BE2395; 6-CN-4-CF 3 -3-Py], [BE2396; 2-OMe-4-CF 3 -3-Py], [BE2397; 5-OMe _{-4-CF 3 -3-Py]} , [BE2398; 6-OMe-4-CF 3 -3-Py], [BE2399; 5-CF 3 -3-Py], [BE2400; 2-Cl-5- CF ₃ -3-Py], [BE 2401; 4-Cl-5-CF ₃ -3-Py],

[BE2402; 6-Cl-5 -CF 3 -3-Py], [BE2403; 2-Me-5-CF 3 -3-Py], [BE2404; 4-Me-5-CF 3 -3-Py] , [BE2405; 6-Me- 5-CF 3 -3-Py], [BE2406; 2-CF 3 -5-CF 3 -3-Py], [BE2407; 4-CF 3 -5-CF 3 -3 -Py], [BE2408; 6- CF 3 -5-CF 3 -3-Py], [BE2409; 2-CN-5-CF 3 -3-Py], [BE2410; 4-CN-5-CF 3 -3-Py], [BE 2411; 6-CN-5-CF ₃ -3-Py], [BE 2412; 2-OMe-5-CF ₃ -3-Py], [BE 2413; 4-OMe-5-CF _{3 -3-Py], [BE2414} ; 6-OMe-5-CF 3 -3-Py], [BE2415; 6-CF 3 -3-Py], [BE2416; 2-Cl-6-CF 3 -3 -Py], [BE2417; 4- Cl-6-CF 3 -3-Py], [BE2418; 5-Cl-6-CF 3 -3-Py], [BE2419; 2-Me-6-CF 3 - 3-Py], [BE2420; 4-Me-6-CF 3 -3-Py], [BE2421; 5-Me-6-CF 3 -3-Py], [BE2422; 2-CF 3 -6-CF _{3 -3-Py], [BE2423} ; 4-CF 3 -6-CF 3 -3-Py], [BE2424; 5-CF 3 -6-CF 3 -3-Py], [BE2425; 2-CN- _{6-CF 3 -3-Py]} , [BE2426; 4-CN-6-CF 3 -3-Py], [BE2427; 5-CN-6-CF 3 -3-Py], [BE2428; 2-OMe _{-6-CF 3 -3-Py]} , [BE2429; 4-OMe-6-CF 3 -3-Py], [BE2430; 5-OMe-6-CF 3 -3-Py], [BE2431; 2- _{OCF 3 -3-Py], [} BE2432; 4-Cl-2-OCF 3 -3-Py], [BE2433; 5-Cl-2-OCF 3 -3-Py], [BE2434; 6-Cl-2 _{-OCF 3 -3-Py], [} BE2435; 4-Me-2-OCF 3 -3-Py], [BE2436; 5-Me-2-OCF 3 -3-Py], [BE2437; 6-Me- 2-OCF ₃ -3-Py], [BE 2438 _{; 4-CF 3 -2-OCF} 3 -3-Py], [BE2439; 5-CF 3 -2-OCF 3 -3-Py], [BE2440; 6-CF 3 -2-OCF 3 -3-Py ], [BE2441; 4-CN -2-OCF 3 -3-Py], [BE2442; 5-CN-2-OCF 3 -3-Py], [BE2443; 6-CN-2-OCF 3 -3- Py], [BE2444; 4- OMe-2-OCF 3 -3-Py], [BE2445; 5-OMe-2-OCF 3 -3-Py], [BE2446; 6-OMe-2-OCF 3 -3 -Py], [BE2447; 4- OCF 3 -3-Py], [BE2448; 2-Cl-4-OCF 3 -3-Py], [BE2449; 5-Cl-4-OCF 3 -3-Py] , [BE2450; 6-Cl- 4-OCF 3 -3-Py], [BE2451; 2-Me-4-OCF 3 -3-Py], [BE2452; 5-Me-4-OCF 3 -3-Py ], [BE2453; 6-Me -4-OCF 3 -3-Py], [BE2454; 2-CF 3 -4-OCF 3 -3-Py], [BE2455; 5-CF 3 -4-OCF 3 - 3-Py], [BE2456; 6-CF 3 -4-OCF 3 -3-Py], [BE2457; 2-CN-4-OCF 3 -3-Py], [BE2458; 5-CN-4-OCF _{3 -3-Py], [BE2459} ; 6-CN-4-OCF 3 -3-Py], [BE2460; 2-OMe-4-OCF 3 -3-Py], [BE2461; 5-OMe-4- _{OCF 3 -3-Py], [} BE2462; 6-OMe-4-OCF 3 -3-Py], [BE2463; 5-OCF 3 -3-Py], [BE2464; 2-Cl-5-OCF 3 - 3-Py], [BE2465; 4-Cl-5-OCF 3 -3-Py], [BE2466; 6-Cl-5-OCF 3 -3-Py], [BE2467; 2-Me-5-OCF 3 -3-Py], [BE2468; 4-Me-5-OCF 3 -3-Py], [BE2469; 6-Me-5-OCF 3 -3-Py], [BE2470; 2-CF 3 -5- _{OCF 3 -3-Py], [} BE2471; 4-CF 3 -5-OCF 3 -3-Py], [BE2472; 6-CF 3 -5-OCF 3 -3-Py], [BE2 473; 2-CN-5- OCF 3 -3-Py], [BE2474; 4-CN-5-OCF 3 -3-Py], [BE2475; 6-CN-5-OCF 3 -3-Py], [BE2476; 2-OMe-5 -OCF 3 -3-Py], [BE2477; 4-OMe-5-OCF 3 -3-Py], [BE2478; 6-OMe-5-OCF 3 -3-Py] _{, [BE2479; 6-OCF 3} -3-Py], [BE2480; 2-Cl-6-OCF 3 -3-Py], [BE2481; 4-Cl-6-OCF 3 -3-Py], [BE2482 ; 5-Cl-6-OCF 3 -3-Py], [BE2483; 2-Me-6-OCF 3 -3-Py], [BE2484; 4-Me-6-OCF 3 -3-Py], [ BE2485; 5-Me-6- OCF 3 -3-Py], [BE2486; 2-CF 3 -6-OCF 3 -3-Py], [BE2487; 4-CF 3 -6-OCF 3 -3-Py ], [BE2488; 5-CF 3 -6-OCF 3 -3-Py], [BE2489; 2-CN-6-OCF 3 -3-Py], [BE2490; 4-CN-6-OCF 3 -3 -Py], [BE2491; 5- CN-6-OCF 3 -3-Py], [BE2492; 2-OMe-6-OCF 3 -3-Py], [BE2493; 4-OMe-6-OCF 3 - 3-Py], [BE2494; 5-OMe-6-OCF 3 -3-Py], [BE2495; 2-CHF 2 -3-Py], [BE2496; 4-Cl-2-CHF 2 -3-Py ], [BE2497; 5-Cl -2-CHF 2 -3-Py], [BE2498; 6-Cl-2-CHF 2 -3-Py], [BE2499; 4-Me-2-CHF 2 -3- Py], [BE2500; 5- Me-2-CHF 2 -3-Py], [BE2501; 6-Me-2-CHF 2 -3-Py],

_{[BE2502; 4-CF 3 -2} -CHF 2 -3-Py], [BE2503; 5-CF 3 -2-CHF 2 -3-Py], [BE2504; 6-CF 3 -2-CHF 2 -3 -Py], [BE2505; 4- CN-2-CHF 2 -3-Py], [BE2506; 5-CN-2-CHF 2 -3-Py], [BE2507; 6-CN-2-CHF 2 - 3-Py], [BE2508; 4-OMe-2-CHF 2 -3-Py], [BE2509; 5-OMe-2-CHF 2 -3-Py], [BE2510; 6-OMe-2-CHF 2 -3-Py, [BE 2511; 4-CHF ₂ -3-Py], [BE 2512; 2-Cl 4-CHF ₂ -3-Py], [BE 2513; 5-Cl 4-CHF ₂ -3- Py], [BE2514; 6- Cl-4-CHF 2 -3-Py], [BE2515; 2-Me-4-CHF 2 -3-Py], [BE2516; 5-Me-4-CHF 2 -3 -Py], [BE2517; 6- Me-4-CHF 2 -3-Py], [BE2518; 2-CF 3 -4-CHF 2 -3-Py], [BE2519; 5-CF 3 -4-CHF ₂ -3-Py, [BE 2520; 6-CF ₃ -4-CHF ₂ -3-Py], [BE 2521; 2-CN 4-CHF ₂ -3-Py], [BE 2522; 5-CN-4 _{-CHF 2 -3-Py], [} BE2523; 6-CN-4-CHF 2 -3-Py], [BE2524; 2-OMe-4-CHF 2 -3-Py], [BE2525; 5-OMe- _{4-CHF 2 -3-Py]} , [BE2526; 6-OMe-4-CHF 2 -3-Py], [BE2527; 5-CHF 2 -3-Py], [BE2528; 2-Cl-5-CHF _2-3 -Py, [BE 2529; 4-Cl-5-CHF ₂ -3-Py], [BE 2530; 6-Cl-5-CHF ₂ -3-Py], [BE 2531; 2-Me-5- CHF ₂ -3-Py !, [BE 2532; 4-Me-5-CHF ₂ -3-Py], [BE 2533; 6-Me-5-CHF ₂ -3-Py], [BE 2534; 2-CF _{3- 5-CHF 2 -3-Py]} , [BE2535; 4-CF 3 -5-CHF 2 -3-Py], [BE2536; 6-CF 3 -5-CHF 2 -3-P y], [BE2537; 2- CN-5-CHF 2 -3-Py], [BE2538; 4-CN-5-CHF 2 -3-Py], [BE2539; 6-CN-5-CHF 2 -3 -Py], [BE2540; 2- OMe-5-CHF 2 -3-Py], [BE2541; 4-OMe-5-CHF 2 -3-Py], [BE2542; 6-OMe-5-CHF 2 - 3-Py], [BE2543; 6-CHF 2 -3-Py], [BE2544; 2-Cl-6-CHF 2 -3-Py], [BE2545; 4-Cl-6-CHF 2 -3-Py ], [BE2546; 5-Cl -6-CHF 2 -3-Py], [BE2547; 2-Me-6-CHF 2 -3-Py], [BE2548; 4-Me-6-CHF 2 -3- Py], [BE2549; 5- Me-6-CHF 2 -3-Py], [BE2550; 2-CF 3 -6-CHF 2 -3-Py], [BE2551; 4-CF 3 -6-CHF 2 -3-Py], [BE2552; 5-CF 3 -6-CHF 2 -3-Py], [BE2553; 2-CN-6-CHF 2 -3-Py], [BE2554; 4-CN-6- _{CHF 2 -3-Py], [} BE2555; 5-CN-6-CHF 2 -3-Py], [BE2556; 2-OMe-6-CHF 2 -3-Py], [BE2557; 4-OMe-6 _{-CHF 2 -3-Py], [} BE2558; 5-OMe-6-CHF 2 -3-Py], [BE2559; 2-OCHF 2 -3-Py], [BE2560; 4-Cl-2-OCHF 2 -3-Py], [BE2561; 5-Cl-2-OCHF 2 -3-Py], [BE2562; 6-Cl-2-OCHF 2 -3-Py], [BE2563; 4-Me-2-OCHF _{2 -3-Py], [BE2564} ; 5-Me-2-OCHF 2 -3-Py], [BE2565; 6-Me-2-OCHF 2 -3-Py], [BE2566; 4-CF 3 -2 _{-OCHF 2 -3-Py], [} BE2567; 5-CF 3 -2-OCHF 2 -3-Py], [BE2568; 6-CF 3 -2-OCHF 2 -3-Py], [BE2569; 4- CN-2-OCHF ₂ -3-Py !, [BE 2570; 5-CN -2-OCHF ₂ -3-Py], [BE 2571; 6-CN -2-OCHF ₂ -3-Py !, [BE 2572; 4-OMe-2-OCHF ₂ -3-Py], [BE 2573; 5-OMe -2-OCHF ₂ -3-Py], [BE 2574; 6-OMe -2- OCHF _2-3 -Py], [BE 2575; 4-OCHF _2-3 -Py], [BE 2576; 2-Cl 4-OCHF _2-3 -Py], [BE 2577; 5-Cl 4-OCHF _2- 3-Py], [BE2578; 6-Cl-4-OCHF 2 -3-Py], [BE2579; 2-Me-4-OCHF 2 -3-Py], [BE2580; 5-Me-4-OCHF 2 -3-Py], [BE2581; 6-Me-4-OCHF 2 -3-Py], [BE2582; 2-CF 3 -4-OCHF 2 -3-Py], [BE2583; 5-CF 3 -4 _{-OCHF 2 -3-Py], [} BE2584; 6-CF 3 -4-OCHF 2 -3-Py], [BE2585; 2-CN-4-OCHF 2 -3-Py], [BE2586; 5-CN _{-4-OCHF 2 -3-Py]} , [BE2587; 6-CN-4-OCHF 2 -3-Py], [BE2588; 2-OMe-4-OCHF 2 -3-Py], [BE2589; 5- _{OMe-4-OCHF 2 -3-} Py], [BE2590; 6-OMe-4-OCHF 2 -3-Py], [BE2591; 5-OCHF 2 -3-Py], [BE2592; 2-Cl-5 _{-OCHF 2 -3-Py], [} BE2593; 4-Cl-5-OCHF 2 -3-Py], [BE2594; 6-Cl-5-OCHF 2 -3-Py], [BE2595; 2-Me- _{5-OCHF 2 -3-Py]} , [BE2596; 4-Me-5-OCHF 2 -3-Py], [BE2597; 6-Me-5-OCHF 2 -3-Py], [BE2598; 2-CF _{3 -5-OCHF 2 -3-Py} ], [BE2599; 4-CF 3 -5-OCHF 2 -3-Py], [BE2600; 6-CF 3 -5-OCHF 2 -3-Py], [BE2601 2-CN-5-OCHF ₂ -3-Py],

[BE2602; 4-CN-5 -OCHF 2 -3-Py], [BE2603; 6-CN-5-OCHF 2 -3-Py], [BE2604; 2-OMe-5-OCHF 2 -3-Py] , [BE2605; 4-OMe- 5-OCHF 2 -3-Py], [BE2606; 6-OMe-5-OCHF 2 -3-Py], [BE2607; 6-OCHF 2 -3-Py], [BE2608 ; 2-Cl-6-OCHF 2 -3-Py], [BE2609; 4-Cl-6-OCHF 2 -3-Py], [BE2610; 5-Cl-6-OCHF 2 -3-Py], [ BE2611; 2-Me-6- OCHF 2 -3-Py], [BE2612; 4-Me-6-OCHF 2 -3-Py], [BE2613; 5-Me-6-OCHF 2 -3-Py], _{[BE2614; 2-CF 3 -6} -OCHF 2 -3-Py], [BE2615; 4-CF 3 -6-OCHF 2 -3-Py], [BE2616; 5-CF 3 -6-OCHF 2 -3 -Py], [BE2617; 2- CN-6-OCHF 2 -3-Py], [BE2618; 4-CN-6-OCHF 2 -3-Py], [BE2619; 5-CN-6-OCHF 2 - 3-Py], [BE2620; 2-OMe-6-OCHF 2 -3-Py], [BE2621; 4-OMe-6-OCHF 2 -3-Py], [BE2622; 5-OMe-6-OCHF 2 -3-Py], [BE2623; 2-Et-3-Py], [BE2624; 4-Cl-2-Et-3-Py], [BE2625; 5-Cl-2-Et-3-Py], [BE2626; 6-Cl-2-Et-3-Py], [BE2627; 4-Me-2-Et-3-Py], [BE2628; 5-Me-2-Et-3-Py], [BE 2629] ; 6-Me-2-Et -3-Py], [BE2630; 4-CF 3 -2-Et-3-Py], [BE2631; 5-CF 3 -2-Et-3-Py], [BE2632 _{; 6-CF 3 -2-Et} -3-Py], [BE2633; 4-CN-2-Et-3-Py], [BE2634; 5-CN-2-Et-3-Py], [BE2635; 6-CN-2-Et-3-Py], [BE2636; 4-OMe-2-Et-3-Py], [BE2637; 5-OMe-2-Et-3-Py], [BE2638; 6- OMe-2 -Et-3-Py], [BE2639; 4-Et-3-Py], [BE2640; 2-Cl-4-Et-3-Py], [BE2641; 5-Cl-4-Et-3-Py ], [BE2642; 6-Cl-4-Et-3-Py], [BE2643; 2-Me-4-Et-3-Py], [BE2644; 5-Me-4-Et-3-Py], [BE2645; 6-Me-4 -Et-3-Py], [BE2646; 2-CF 3 -4-Et-3-Py], [BE2647; 5-CF 3 -4-Et-3-Py], [BE 2648; 6-CF ₃ -4-Et-3-Py], [BE 2649; 2-CN-4-Et-3-Py], [BE 2650; 5-CN-4-Et-3-Py], [BE 2 6 6 BE2651; 6-CN-4-Et-3-Py], [BE2652; 2-OMe-4-Et-3-Py], [BE2653; 5-OMe-4-Et-3-Py], [BE2654; 6-OMe-4-Et-3-Py], [BE 2655; 5-Et-3-Py], [BE 2656; 2-Cl-5-Et-3-Py], [BE 2657; Et-3-Py, [BE2658; 6-Cl-5-Et-3-Py], [BE2659; 2-Me-5-Et-3-Py], [BE2660; 4-Me-5-Et- 3-Py], [BE2661; 6-Me-5-Et-3-Py], [BE2662; 2-CF 3 -5-Et-3-Py], [BE2663; 4-CF 3 -5-Et- 3-Py], [BE2664; 6-CF 3 -5-Et-3-Py], [BE2665; 2-CN-5-Et-3-Py], [BE2666; 4-CN-5-Et-3 -Py], [BE2667; 6-CN-5-Et-3-Py], [BE2668; 2-OMe-5-Et-3-Py], [BE2669; 4-OMe-5-Et-3-Py ], [BE2670; 6-OMe-5-Et-3-Py], [BE2671; 6-Et-3-Py], [BE2672; 2-Cl-6-Et-3-Py], [BE 2673; 4] -Cl-6-Et-3-Py], [BE2674; 5-Cl-6-Et-3-Py], [BE2675; 2-Me-6-Et-3-Py], [BE2676; 4-Me -6-Et-3-Py] , [BE2677; 5-Me-6-Et-3-Py], [BE2678; 2-CF 3 -6-Et-3-Py], [BE2679; 4-CF 3 -6- Et-3-Py], [ BE2680; 5-CF 3 -6-Et-3-Py], [BE2681; 2-CN-6-Et-3-Py], [BE2682; 4-CN-6-Et -3-Py], [BE2683; 5-CN-6-Et-3-Py], [BE2684; 2-OMe-6-Et-3-Py], [BE2685; 4-OMe-6-Et-3 -Py], [BE2686; 5- OMe-6-Et-3-Py] 2691, [BE2687; 4-Cl-2-CH 2 CF 3 -3-Py], [BE2688; 5-Cl-2-CH _{2 CF 3 -3-Py],} [BE2689; 6-Cl-2-CH 2 CF 3 -3-Py], [BE2690; 4-Me-2-CH 2 CF 3 -3-Py], [BE2691; _{5-Me-2-CH 2} CF 3 -3-Py], [BE2692; 6-Me-2-CH 2 CF 3 -3-Py], [BE2693; 4-CF 3 -2-CH 2 CF 3 - 3-Py], [BE 2694; 5-CF ₃ -2-CH ₂ CF ₃ -3-Py], [BE 2 695; 6-CF ₃ -2-CH ₂ CF ₃ -3-Py], [BE ₂ 696; _{CN-2-CH 2 CF 3} -3-Py], [BE2697; 5-CN-2-CH 2 CF 3 -3-Py], [BE2698; 6-CN-2-CH 2 CF 3 -3-Py ], [BE2699; 4-OMe -2-CH 2 CF 3 -3-Py], [BE2700; 5-OMe-2-CH 2 CF 3 -3-Py], [BE2701; 6-OMe-2-CH ₂ CF ₃ -3-Py],

_{[BE2702; 4-CH 2 CF} 3 -3-Py], [BE2703; 2-Cl-4-CH 2 CF 3 -3-Py], [BE2704; 5-Cl-4-CH 2 CF 3 -3- Py], [BE2705; 6- Cl-4-CH 2 CF 3 -3-Py], [BE2706; 2-Me-4-CH 2 CF 3 -3-Py], [BE2707; 5-Me-4- _{CH 2 CF 3 -3-Py]} , [BE2708; 6-Me-4-CH 2 CF 3 -3-Py], [BE2709; 2-CF 3 -4-CH 2 CF 3 -3-Py], [ BE 2710; 5-CF ₃ -4-CH ₂ CF ₃ -3-Py], [BE 2711; 6-CF ₃ -4-CH ₂ CF ₃ -3-Py], [BE 2712; 2-CN -4-CH _{2 CF 3 -3-Py], [} BE2713; 5-CN-4-CH 2 CF 3 -3-Py], [BE2714; 6-CN-4-CH 2 CF 3 -3-Py], [BE2715; 2 _{-OMe-4-CH 2 CF 3} -3-Py], [BE2716; 5-OMe-4-CH 2 CF 3 -3-Py], [BE2717; 6-OMe-4-CH 2 CF 3 -3- Py], [BE2718; 5- CH 2 CF 3 -3-Py], [BE2719; 2-Cl-5-CH 2 CF 3 -3-Py], [BE2720; 4-Cl-5-CH 2 CF 3 -3-Py], [BE2721; 6-Cl-5-CH 2 CF 3 -3-Py], [BE2722; 2-Me-5-CH 2 CF 3 -3-Py], [BE2723; 4-Me _{-5-CH 2 CF 3 -3-} Py], [BE2724; 6-Me-5-CH 2 CF 3 -3-Py], [BE2725; 2-CF 3 -5-CH 2 CF 3 -3-Py ], [BE2726; 4-CF 3 -5-CH 2 CF 3 -3-Py], [BE2727; 6-CF 3 -5-CH 2 CF 3 -3-Py], [BE2728; 2-CN-5 _{-CH 2 CF 3 -3-Py]} , [BE2729; 4-CN-5-CH 2 CF 3 -3-Py], [BE2730; 6-CN-5-CH 2 CF 3 -3-Py], [ BE2731; 2-OMe-5- CH 2 CF 3 -3-Py], [BE2732; 4-OMe-5-CH 2 CF 3 -3 -Py], [BE2733; 6- OMe-5-CH 2 CF 3 -3-Py], [BE2734; 6-CH 2 CF 3 -3-Py], [BE2735; 2-Cl-6-CH 2 CF _{3 -3-Py], [BE2736} ; 4-Cl-6-CH 2 CF 3 -3-Py], [BE2737; 5-Cl-6-CH 2 CF 3 -3-Py], [BE2738; 2- _{Me-6-CH 2 CF 3} -3-Py], [BE2739; 4-Me-6-CH 2 CF 3 -3-Py], [BE2740; 5-Me-6-CH 2 CF 3 -3-Py ], [BE2741; 2-CF 3 -6-CH 2 CF 3 -3-Py], [BE2742; 4-CF 3 -6-CH 2 CF 3 -3-Py], [BE2743; 5-CF 3 - _{6-CH 2 CF 3 -3-} Py], [BE2744; 2-CN-6-CH 2 CF 3 -3-Py], [BE2745; 4-CN-6-CH 2 CF 3 -3-Py], [BE2746; 5-CN-6 -CH 2 CF 3 -3-Py], [BE2747; 2-OMe-6-CH 2 CF 3 -3-Py], [BE2748; 4-OMe-6-CH 2 CF _{3 -3-Py], [BE2749} ; 5-OMe-6-CH 2 CF 3 -3-Py], [BE2750; 4-Cl-2-OEt-3-Py], [BE2751; 5-Cl-2 -OEt-3-Py], [BE 2752; 6-Cl-2-OEt-3-Py], [BE 2753; 4-Me-2-OEt-3-Py], [BE 2754; 5-Me-2-OEt -3-Py], [BE2755; 6-Me-2-OEt-3-Py], [BE2756; 4-CF 3 -2-OEt-3-Py], [BE2757; 5-CF 3 -2-OEt -3-Py !, [BE 2758; 6-CF ₃ -2-OEt-3-Py], [BE 2759; 4-CN-2-OEt-3-Py], [BE 2760; 5-CN-2-OEt- 3-Py], [BE2761; 6-CN-2-OEt-3-Py], [BE2762; 4-OMe-2-OEt-3-Py], [BE2763; 5-OMe-2-OEt-3- 3 Py], [BE2764; 6-OMe-2-OEt-3-Py], [BE2765; 4-OEt-3-Py], [BE2766; 2-Cl-4-OEt-3-Py], [BE2767; 5-C l-4-OEt-3-Py], [BE2768; 6-Cl-4-OEt-3-Py], [BE2769; 2-Me-4-OEt-3-Py], [BE2770; 5-Me- 4-OEt-3-Py] , [BE2771; 6-Me-4-OEt-3-Py], [BE2772; 2-CF 3 -4-OEt-3-Py], [BE2773; 5-CF 3 - 4-OEt-3-Py] , [BE2774; 6-CF 3 -4-OEt-3-Py], [BE2775; 2-CN-4-OEt-3-Py], [BE2776; 5-CN-4 -OEt-3-Py], [BE2777; 6-CN-4-OEt-3-Py], [BE2778; 2-OMe-4-OEt-3-Py], [BE2779; 5-OMe-4-OEt -3-Py !, [BE2780; 6-OMe-4-OEt-3-Py], [BE2781; 5-OEt-3-Py], [BE2782; 2-Cl-5-OEt-3-Py], [BE 2783; 4-Cl-5-OEt-3-Py], [BE 2784; 6-Cl-5-OEt-3-Py], [BE 2 785; 2-Me-5-OEt-3-Py], [BE 2786] ; 4-Me-5-OEt -3-Py], [BE2787; 6-Me-5-OEt-3-Py], [BE2788; 2-CF 3 -5-OEt-3-Py], [BE2789; _{4-CF 3 -5-OEt-} 3-Py], [BE2790; 6-CF 3 -5-OEt-3-Py], [BE2791; 2-CN-5-OEt-3-Py], [BE2792; 4-CN-5-OEt-3-Py], [BE2793; 6-CN-5-OEt-3-Py], [BE2794; 2-OMe-5-OEt-3-Py], [BE2795; OMe-5-OEt-3-Py !, [BE2796; 6-OMe-5-OEt-3-Py], [BE2797; 6-OEt-3-Py], [BE2798; 2-Cl-6-OEt- 3-Py], [BE2799; 4-Cl-6-OEt-3-Py], [BE2800; 5-Cl-6-OEt-3-Py], [BE2801; 2-Me-6-OEt-3- Py],

[BE2802; 4-Me-6 -OEt-3-Py], [BE2803; 5-Me-6-OEt-3-Py], [BE2804; 2-CF 3 -6-OEt-3-Py], [ _{BE2805; 4-CF 3 -6-} OEt-3-Py], [BE2806; 5-CF 3 -6-OEt-3-Py], [BE2807; 2-CN-6-OEt-3-Py], [ BE2808; 4-CN-6-OEt-3-Py], [BE2809; 5-CN-6-OEt-3-Py], [BE2810; 2-OMe-6-OEt-3-Py], [BE2811; 4-OMe-6-OEt- 3-Py], [BE2812; 5-OMe-6-OEt-3-Py], [BE2813; 4-Cl-2-OCH 2 CF 3 -3-Py], [BE2814 ; 5-Cl-2-OCH 2 CF 3 -3-Py], [BE2815; 6-Cl-2-OCH 2 CF 3 -3-Py], [BE2816; 4-Me-2-OCH 2 CF 3 - 3-Py], [BE2817; 5-Me-2-OCH 2 CF 3 -3-Py], [BE2818; 6-Me-2-OCH 2 CF 3 -3-Py], [BE2819; 4-CF 3 -2-OCH ₂ CF ₃ -3-Py, [BE 2820; 5-CF ₃ -2-OCH ₂ CF ₃ -3-Py], [BE 2821; 6-CF ₃ -2-OCH ₂ CF ₃ -3- Py], [BE2822; 4- CN-2-OCH 2 CF 3 -3-Py], [BE2823; 5-CN-2-OCH 2 CF 3 -3-Py], [BE2824; 6-CN-2- _{OCH 2 CF 3 -3-Py]} , [BE2825; 4-OMe-2-OCH 2 CF 3 -3-Py], [BE2826; 5-OMe-2-OCH 2 CF 3 -3-Py], [BE2827 ; 6-OMe-2-OCH 2 CF 3 -3-Py], [BE2828; 4-OCH 2 CF 3 -3-Py], [BE2829; 2-Cl-4-OCH 2 CF 3 -3-Py] , [BE2830; 5-Cl- 4-OCH 2 CF 3 -3-Py], [BE2831; 6-Cl-4-OCH 2 CF 3 -3-Py], [BE2832; 2-Me-4-OCH 2 _{CF 3 -3-Py], [} BE2833; 5-Me-4-OCH 2 CF 3 -3-Py], [BE2834; 6-Me- _{4-OCH 2 CF 3 -3-} Py], [BE2835; 2-CF 3 -4-OCH 2 CF 3 -3-Py], [BE2836; 5-CF 3 -4-OCH 2 CF 3 -3-Py ], [BE 2837; 6-CF ₃ -4-OCH ₂ CF ₃ -3-Py], [BE 2 838; 2-CN 4-OCH ₂ CF ₃ -3-Py], [BE 2839; _{OCH 2 CF 3 -3-Py]} , [BE2840; 6-CN-4-OCH 2 CF 3 -3-Py], [BE2841; 2-OMe-4-OCH 2 CF 3 -3-Py], [BE2842 ; 5-OMe-4-OCH 2 CF 3 -3-Py], [BE2843; 6-OMe-4-OCH 2 CF 3 -3-Py], [BE2844; 5-OCH 2 CF 3 -3-Py] , [BE2845; 2-Cl- 5-OCH 2 CF 3 -3-Py], [BE2846; 4-Cl-5-OCH 2 CF 3 -3-Py], [BE2847; 6-Cl-5-OCH 2 CF ₃ -3-Py !, [BE 2848; 2-Me-5-OCH ₂ CF ₃ -3-Py], [BE 2849; 4-Me-5-OCH ₂ CF ₃ -3-Py], [BE 2850; 6 _{-Me-5-OCH 2 CF 3} -3-Py], [BE2851; 2-CF 3 -5-OCH 2 CF 3 -3-Py], [BE2852; 4-CF 3 -5-OCH 2 CF 3 - 3-Py], [BE2853; 6-CF 3 -5-OCH 2 CF 3 -3-Py], [BE2854; 2-CN-5-OCH 2 CF 3 -3-Py], [BE2855; 4-CN _{-5-OCH 2 CF 3 -3-} Py], [BE2856; 6-CN-5-OCH 2 CF 3 -3-Py], [BE2857; 2-OMe-5-OCH 2 CF 3 -3-Py] , [BE2858; 4-OMe- 5-OCH 2 CF 3 -3-Py], [BE2859; 6-OMe-5-OCH 2 CF 3 -3-Py], [BE2860; 6-OCH 2 CF 3 -3 -Py], [BE2861; 2- Cl-6-OCH 2 CF 3 -3-Py], [BE2862; 4-Cl-6-OCH 2 CF 3 -3-Py], [BE2863; 5-Cl-6 -OCH ₂ CF ₃ -3-Py], [BE 2864; 2 _{-Me-6-OCH 2 CF 3} -3-Py], [BE2865; 4-Me-6-OCH 2 CF 3 -3-Py], [BE2866; 5-Me-6-OCH 2 CF 3 -3- Py], [BE2867; 2- CF 3 -6-OCH 2 CF 3 -3-Py], [BE2868; 4-CF 3 -6-OCH 2 CF 3 -3-Py], [BE2869; 5-CF 3 _{-6-OCH 2 CF 3 -3-} Py], [BE2870; 2-CN-6-OCH 2 CF 3 -3-Py], [BE2871; 4-CN-6-OCH 2 CF 3 -3-Py] , [BE2872; 5-CN- 6-OCH 2 CF 3 -3-Py], [BE2873; 2-OMe-6-OCH 2 CF 3 -3-Py], [BE2874; 4-OMe-6-OCH 2 _{CF 3 -3-Py], [} BE2875; 5-OMe-6-OCH 2 CF 3 -3-Py], [BE2876; 2-Pr-3-Py], [BE2877; 4-Cl-2-Pr- 3-Py], [BE2878; 5-Cl-2-Pr-3-Py], [BE 2879; 6-Cl-2-Pr-3-Py], [BE 2880; 4-Me-2-Pr-3- Py], [BE2881; 5- Me-2-Pr-3-Py], [BE2882; 6-Me-2-Pr-3-Py], [BE2883; 4-CF 3 -2-Pr-3-Py ], [BE2884; 5-CF 3 -2-Pr-3-Py], [BE2885; 6-CF 3 -2-Pr-3-Py], [BE2886; 4-CN-2-Pr-3-Py ], [BE2887; 5-CN-2-Pr-3-Py], [BE2888; 6-CN-2-Pr-3-Py], [BE2889; 4-OMe-2-Pr-3-Py], [BE2890; 5-OMe-2-Pr-3-Py], [BE2891; 6-OMe-2-Pr-3-Py], [BE2892; 4-Pr-3-Py], [BE2893; 2-Cl -4-Pr-3-Py], [BE2894; 5-Cl-4-Pr-3-Py], [BE2895; 6-Cl-4-Pr-3-Py], [BE2896; 2-Me-4 -Pr-3-Py], [ BE2897; 5-Me-4-Pr-3-Py], [BE2898; 6-Me-4-Pr-3-Py], [BE2899; 2-CF 3 -4- Pr-3-Py], [BE 2 900; 5-CF ₃ -4-Pr -3-Py], [BE 2901; 6-CF ₃ -4-Pr-3-Py],

[BE2902; 2-CN-4-Pr-3-Py], [BE 2903; 5-CN-4-Pr-3-Py], [BE 2904; 6-CN-4-Pr-3-Py], [BE 2905] 2-OMe-4-Pr-3-Py !, [BE2906; 5-OMe-4-Pr-3-Py], [BE2907; 6-OMe-4-Pr-3-Py], [BE2908; -Pr-3-Py], [BE2909; 2-Cl-5-Pr-3-Py], [BE2910; 4-Cl-5-Pr-3-Py], [BE2911; 6-Cl-5-Pr -3-Py !, [BE2912; 2-Me-5-Pr-3-Py], [BE2913; 4-Me-5-Pr-3-Py], [BE2914; 6-Me-5-Pr-3 -Py], [BE2915; 2- CF 3 -5-Pr-3-Py], [BE2916; 4-CF 3 -5-Pr-3-Py], [BE2917; 6-CF 3 -5-Pr- 3-Py], [BE2918; 2-CN-5-Pr-3-Py], [BE2919; 4-CN-5-Pr-3-Py], [BE2920; 6-CN-5-Pr-3- Py], [BE2921; 2-OMe-5-Pr-3-Py], [BE2922; 4-OMe-5-Pr-3-Py], [BE2923; 6-OMe-5-Pr-3-Py] , [BE2924; 6-Pr-3-Py], [BE2925; 2-Cl-6-Pr-3-Py], [BE2926; 4-Cl-6-Pr-3-Py], [BE2927; 5- Cl-6-Pr-3-Py], [BE2928; 2-Me-6-Pr-3-Py], [BE2929; 4-Me-6-Pr-3-Py], [BE2930; 5-Me- 6-Pr-3-Py] , [BE2931; 2-CF 3 -6-Pr-3-Py], [BE2932; 4-CF 3 -6-Pr-3-Py], [BE2933; 5-CF 3 -6-Pr-3-Py], [BE2934; 2-CN-6-Pr-3-Py], [BE2935; 4-CN-6-Pr-3-Py], [BE2936; 5-CN-6 -Pr-3-Py], [BE2937; 2-OMe-6-Pr-3-Py], [BE2938; 4-OMe-6-Pr-3-Py], [BE2939; 5-OMe-6-Pr -3-Py !, [BE2940; 2-OPr-3-Py], [BE 2941; 4-Cl-2-OPr-3-Py], [BE2942; 5-Cl-2-OPr-3-Py], [ BE 2943; 6-Cl-2-OPr-3-Py], [BE 2944; 4-Me-2-OPr-3-Py], [BE 2 945; 5-Me-2-OPr-3-Py], [BE 2946; 6-Me-2-OPr- 3-Py], [BE2947; 4-CF 3 -2-OPr-3-Py], [BE2948; 5-CF 3 -2-OPr-3-Py], [BE2949; _{6-CF 3 -2-OPr-} 3-Py], [BE2950; 4-CN-2-OPr-3-Py], [BE2951; 5-CN-2-OPr-3-Py], [BE2952; 6 -CN-2-OPr-3-Py], [BE2953; 4-OMe-2-OPr-3-Py], [BE2954; 5-OMe-2-OPr-3-Py], [BE2955; 6-OMe -2-OPr-3-Py], [BE 2956; 4-OPr-3-Py], [BE 2957; 2-Cl-4-OPr-3-Py], [BE 2958; 5-Cl-4-OPr-3 -Py], [BE2959; 6-Cl-4-OPr-3-Py], [BE 2960; 2-Me-4-OPr-3-Py], [BE 296; 5-Me-4-OPr-3-Py ], [BE2962; 6-Me -4-OPr-3-Py], [BE2963; 2-CF 3 -4-OPr-3-Py], [BE2964; 5-CF 3 -4-OPr-3-Py ], [BE2965; 6-CF 3 -4-OPr-3-Py], [BE2966; 2-CN-4-OPr-3-Py], [BE2967; 5-CN-4-OPr-3-Py] , [BE2968; 6-CN-4-OPr-3-Py], [BE2969; 2-OMe-4-OPr-3-Py], [BE2970; 5-OMe-4-OPr-3-Py], [BE29 6; BE2971; 6-OMe-4-OPr-3-Py], [BE2972; 5-OPr-3-Py], [BE2 973; 2-Cl-5-OPr-3-Py], [BE 2974; 4-Cl- 5-OPr-3-Py, [BE2975; 6-Cl-5-OPr-3-Py], [BE2976; 2-Me-5-OPr-3-Py], [BE2977; 4-Me-5- OPr-3-Py], [ BE2978; 6-Me-5-OPr-3-Py], [BE2979; 2-CF 3 -5-OPr-3-Py], [BE2980; 4-CF 3 -5- OPr-3-Py], [BE 2981; 6-CF ₃ -5-OPr-3-Py], [BE 2982; 2-CN-5-OPr-3-Py], [BE2983; 4-CN-5-OPr-3-Py], [BE2984; 6-CN-5-OPr-3-Py], [BE2985; 2-OMe-5-OPr-3-Py], [BE2986; 4-OMe-5-OPr-3-Py], [BE2987; 6-OMe-5-OPr-3-Py], [BE2988; 6- OPr-3-Py], [BE2989; 2-Cl-6-OPr-3-Py], [BE2990; 4-Cl-6-OPr-3-Py], [BE 2991; 5-Cl-6-OPr- 3-Py], [BE2992; 2-Me-6-OPr-3-Py], [BE2993; 4-Me-6-OPr-3-Py], [BE2994; 5-Me-6-OPr-3- Py], [BE2995; 2- CF 3 -6-OPr-3-Py], [BE2996; 4-CF 3 -6-OPr-3-Py], [BE2997; 5-CF 3 -6-OPr-3 -Py], [BE2998; 2-CN-6-OPr-3-Py], [BE2999; 4-CN-6-OPr-3-Py], [BE 3000; 5-CN-6-OPr-3-Py ], [BE 3001; 2-OMe-6-OPr-3-Py],

[BE3002; 4-OMe-6-OPr-3-Py], [BE3003; 5-OMe-6-OPr-3-Py], [BE3004; 2-SMe-3-Py], [BE3005; -2-SMe-3-Py !, [BE 3006; 5-Cl-2-SMe-3-Py], [BE 3007; 6-Cl-2-SMe-3-Py], [BE 3008; 4-Me-2 5-SMe-3-Py !, [BE 3009; 5-Me-2-SMe-3-Py], [BE 3010; 6-Me-2-SMe-3-Py], [BE 3011; 4-CF ₃ -2- SMe-3-Py !, [BE 3012; 5-CF ₃ -2-SMe -3-Py], [BE 3013; 6-CF ₃ -2-SMe-3-Py], [BE 3014; SMe-3-Py !, [BE3015; 5-CN-2-SMe-3-Py], [BE3016; 6-CN-2-SMe-3-Py], [BE3017; 4-OMe-2-SMe- 3-Py], [BE3018; 5-OMe-2-SMe-3-Py], [BE3019; 6-OMe-2-SMe-3-Py], [BE3020; 4-SMe-3-Py], [BE30 20; BE3021; 2-Cl-4-SMe-3-Py], [BE3022; 5-Cl-4-SMe-3-Py], [BE3023; 6-Cl-4-SMe-3-Py], [BE3024; 2-Me-4-SMe-3-Py], [BE3025; 5-Me-4-SMe-3-Py], [BE3026; 6-Me-4-SMe-3-Py], [BE3027; _{CF 3 -4-SMe-3-} Py], [BE3028; 5-CF 3 -4-SMe-3-Py], [BE3029; 6-CF 3 -4-SMe-3-Py], [BE3030; 2 -CN-4-SMe-3-Py], [BE3031; 5-CN-4-SMe-3-Py], [BE3032; 6-CN-4-SMe-3-Py], [BE3033; 2-OMe -4-SMe-3-Py !, [BE 3034; 5-OMe-4-SMe-3-Py], [BE 3035; 6-OMe-4-SMe-3-Py], [BE 3036; 5-SMe-3 -Py], [BE3037; 2-Cl-5-SMe-3-Py], [BE3038; 4-Cl-5-SMe-3-Py], [BE3039; 6-Cl-5-SMe-3-Py ], [BE3040; 2-Me-5-SMe-3-Py], [BE3041; 4-Me-5 -SMe-3-Py], [ BE3042; 6-Me-5-SMe-3-Py], [BE3043; 2-CF 3 -5-SMe-3-Py], [BE3044; 4-CF 3 -5 -SMe-3-Py], [ BE3045; 6-CF 3 -5-SMe-3-Py], [BE3046; 2-CN-5-SMe-3-Py], [BE3047; 4-CN-5- SMe-3-Py !, [BE3048; 6-CN-5-SMe-3-Py], [BE3049; 2-OMe-5-SMe-3-Py], [BE3050; 4-OMe-5-SMe- 3-Py], [BE3051; 6-OMe-5-SMe-3-Py], [BE3052; 6-SMe-3-Py], [BE3053; 2-Cl-6-SMe-3-Py], [BE3053; BE 3054; 4-Cl-6-SMe-3-Py], [BE 3055; 5-Cl-6-SMe-3-Py], [BE 3056; 2-Me-6-SMe-3-Py], [BE 3057; 4-Me-6-SMe- 3-Py], [BE3058; 5-Me-6-SMe-3-Py], [BE3059; 2-CF 3 -6-SMe-3-Py], [BE3060; 4 _{-CF 3 -6-SMe-3-} Py], [BE3061; 5-CF 3 -6-SMe-3-Py], [BE3062; 2-CN-6-SMe-3-Py], [BE3063; 4 -CN-6-SMe-3-Py], [BE 3064; 5-CN-6-SMe-3-Py], [BE 3065; 2-OMe-6-SMe-3-Py], [BE 3066; 4-OMe -6-SMe-3-Py !, [BE3067; 5-OMe-6-SMe-3-Py], [BE3068; 2-SCF ₃ -3-Py], [BE 3069; 4-Cl-2-SCF ₃ -3-Py], [BE3070; 5-Cl-2-SCF 3 -3-Py], [BE3071; 6-Cl-2-SCF 3 -3-Py], [BE3072; 4-Me-2-SCF _{3 -3-Py], [BE3073} ; 5-Me-2-SCF 3 -3-Py], [BE3074; 6-Me-2-SCF 3 -3-Py], [BE3075; 4-CF 3 -2 _{-SCF 3 -3-Py], [} BE3076; 5-CF 3 -2-SCF 3 -3-Py], [BE3077; 6-CF 3 -2-SCF 3 -3-Py], [BE3078; 4- CN-2-SCF ₃ -3-Py], [BE 3079; 5-CN-2-SCF ₃ -3-Py, [BE 3080; 6-CN 2-SCF ₃ -3-Py], [BE 3081; 4-OMe 2-SCF ₃ -3-Py], [BE 308 2 ; 5-OMe-2-SCF 3 -3-Py], [BE3083; 6-OMe-2-SCF 3 -3-Py], [BE3084; 4-SCF 3 -3-Py], [BE3085; 2- _{Cl-4-SCF 3 -3-} Py], [BE3086; 5-Cl-4-SCF 3 -3-Py], [BE3087; 6-Cl-4-SCF 3 -3-Py], [BE3088; 2 _{-Me-4-SCF 3 -3-} Py], [BE3089; 5-Me-4-SCF 3 -3-Py], [BE3090; 6-Me-4-SCF 3 -3-Py], [BE3091; _{2-CF 3 -4-SCF 3} -3-Py], [BE3092; 5-CF 3 -4-SCF 3 -3-Py], [BE3093; 6-CF 3 -4-SCF 3 -3-Py] , [BE 3094; 2-CN-4-SCF ₃ -3-Py], [BE 3095; 5-CN 4-SCF ₃ -3-Py], [BE 3096; 6-CN 4-SCF ₃ -3-Py ], [BE3097; 2-OMe -4-SCF 3 -3-Py], [BE3098; 5-OMe-4-SCF 3 -3-Py], [BE3099; 6-OMe-4-SCF 3 -3- Py], [BE3100; 5- SCF 3 -3-Py], [BE3101; 2-Cl-5-SCF 3 -3-Py],

[BE3102; 4-Cl-5 -SCF 3 -3-Py], [BE3103; 6-Cl-5-SCF 3 -3-Py], [BE3104; 2-Me-5-SCF 3 -3-Py] , [BE3105; 4-Me- 5-SCF 3 -3-Py], [BE3106; 6-Me-5-SCF 3 -3-Py], [BE3107; 2-CF 3 -5-SCF 3 -3- Py], [BE3108; 4- CF 3 -5-SCF 3 -3-Py], [BE3109; 6-CF 3 -5-SCF 3 -3-Py], [BE3110; 2-CN-5-SCF 3 -3-Py], [BE3111; 4-CN-5-SCF 3 -3-Py], [BE3112; 6-CN-5-SCF 3 -3-Py], [BE3113; 2-OMe-5-SCF _{3 -3-Py], [BE3114} ; 4-OMe-5-SCF 3 -3-Py], [BE3115; 6-OMe-5-SCF 3 -3-Py], [BE3116; 6-SCF 3 -3 -Py], [BE3117; 2- Cl-6-SCF 3 -3-Py], [BE3118; 4-Cl-6-SCF 3 -3-Py], [BE3119; 6-Cl-6-SCF 3 - 3-Py], [BE3120; 2-Me-6-SCF 3 -3-Py], [BE3121; 4-Me-6-SCF 3 -3-Py], [BE3122; 6-Me-6-SCF 3 -3-Py], [BE 3123; 2-CF ₃ -6-SCF ₃ -3-Py], [BE 3124; 4-CF ₃ -6-SCF ₃ -3-Py], [BE ₃ 125; 6-CF _3- 6-SCF ₃ -3-Py !, [BE 3126; 2-CN-6-SCF ₃ -3-Py], [BE 3127; 4-CN-6-SCF ₃ -3-Py], [BE 3128; 6-CN _{-6-SCF 3 -3-Py]} , [BE3129; 2-OMe-6-SCF 3 -3-Py], [BE3130; 4-OMe-6-SCF 3 -3-Py], [BE3131; 6- _{OMe-6-SCF 3 -3-} Py], [BE3132; 2-S (O) Me-3-Py], [BE3133; 4-Cl-2-S (O) Me-3-Py], [BE3134 5-Cl-2-S (O) Me-3-Py], [BE3135; 6-Cl-2-S (O) Me-3-Py], [BE3136; 4-Me-2-S (O); ) Me-3-Py], [BE 313 7; 5-Me-2- S (O) Me-3-Py], [BE3138; 6-Me-2-S (O) Me-3-Py], [BE3139; 4-CF 3 -2-S (O) Me-3-Py ], [BE3140; 5-CF 3 -2-S (O) Me-3-Py], [BE3141; 6-CF 3 -2-S (O) Me-3-Py ], [BE3142; 4-CN-2-S (O) Me-3-Py], [BE3143; 5-CN-2-S (O) Me-3-Py], [BE3144; 6-CN-2 -S (O) Me-3-Py], [BE3145; 4-OMe-2-S (O) Me-3-Py], [BE3146; 5-OMe-2-S (O) Me-3-Py ], [BE3147; 6-OMe-2-S (O) Me-3-Py], [BE3148; 4-S (O) Me-3-Py], [BE3149; 2-Cl-4-S (O) ) Me-3-Py], [BE3150; 5-Cl-4-S (O) Me-3-Py], [BE3151; 6-Cl-4-S (O) Me-3-Py], [BE3152 2-Me-4-S (O) Me-3-Py], [BE3153; 5-Me-4-S (O) Me-3-Py], [BE3154; 6-Me-4-S (O ) Me-3-Py], [BE3155; 2-CF 3 -4-S (O) Me-3-Py], [BE3156; 5-CF 3 -4-S (O) Me-3-Py], _{[BE3157; 6-CF 3 -4} -S (O) Me-3-Py], [BE3158; 2-CN-4-S (O) Me-3-Py], [BE3159; 5-CN-4- S (O) Me-3-Py], [BE3160; 6-CN-4-S (O) Me-3-Py], [BE3161; 2-OMe-4-S (O) Me-3-Py] , [BE3162; 5-OMe-4-S (O) Me-3-Py], [BE3163; 6-OMe-4-S (O) Me-3-Py], [BE3164; 5-S (O) Me-3-Py !, [BE3165; 2-Cl-5-S (O) Me-3-Py], [BE3166; 4-Cl-5-S (O) Me-3-Py], [BE3167; 6-Cl-5-S (O) Me-3-Py], [BE3168; 2-Me-5-S (O) Me-3-Py], [BE3169; 4-Me-5-S (O) Me-3-Py], [ BE3170; 6-Me-5-S (O) Me-3-Py], [BE3171; 2-CF 3 -5-S (O) Me-3-Py], [BE3172 ;Four _{-CF 3 -5-S (O)} Me-3-Py], [BE3173; 6-CF 3 -5-S (O) Me-3-Py], [BE3174; 2-CN-5-S (O ) Me-3-Py], [BE3175; 4-CN-5-S (O) Me-3-Py], [BE3176; 6-CN-5-S (O) Me-3-Py], [BE3177] 2-OMe-5-S (O) Me-3-Py], [BE3178; 4-OMe-5-S (O) Me-3-Py], [BE3179; 6-OMe-5-S (O ) Me-3-Py], [BE3180; 6-S (O) Me-3-Py], [BE3181; 2-Cl-6-S (O) Me-3-Py], [BE3182; -6-S (O) Me-3-Py], [BE3183; 5-Cl-6-S (O) Me-3-Py], [BE3184; 2-Me-6-S (O) Me-3 -Py], [BE3185; 4-Me-6-S (O) Me-3-Py], [BE3186; 5-Me-6-S (O) Me-3-Py], [BE3187; 2-CF _{3 -6-S (O) Me} -3-Py], [BE3188; 4-CF 3 -6-S (O) Me-3-Py], [BE3189; 5-CF 3 -6-S (O) Me-3-Py !, [BE3190; 2-CN-6-S (O) Me-3-Py], [BE3191; 4-CN-6-S (O) Me-3-Py], [BE3192; 5-CN-6-S (O) Me-3-Py], [BE3193; 2-OMe-6-S (O) Me-3-Py], [BE3194; 4-OMe-6-S (O) Me-3-Py], [ BE3195; 5-OMe-6-S (O) Me-3-Py], [BE3196; 2-S (O) CF 3 -3-Py], [BE3197; 4-Cl _{-2-S (O) CF 3} -3-Py], [BE3198; 5-Cl-2-S (O) CF 3 -3-Py], [BE3199; 6-Cl-2-S (O) CF _{3 -3-Py], [BE3200} ; 4-Me-2-S (O) CF 3 -3-Py], [BE3201; 5-Me-2-S (O) CF 3 -3-Py],

[BE3202; 6-Me-2 -S (O) CF 3 -3-Py], [BE3203; 4-CF 3 -2-S (O) CF 3 -3-Py], [BE3204; 5-CF 3 _{-2-S (O) CF 3} -3-Py], [BE3205; 6-CF 3 -2-S (O) CF 3 -3-Py], [BE3206; 4-CN-2-S (O) _{CF 3 -3-Py], [} BE3207; 5-CN-2-S (O) CF 3 -3-Py], [BE3208; 6-CN-2-S (O) CF 3 -3-Py], [BE3209; 4-OMe-2 -S (O) CF 3 -3-Py], [BE3210; 5-OMe-2-S (O) CF 3 -3-Py], [BE3211; 6-OMe-2 _{-S (O) CF 3 -3-} Py], [BE3212; 4-S (O) CF 3 -3-Py], [BE3213; 2-Cl-4-S (O) CF 3 -3-Py] , [BE3214; 5-Cl- 4-S (O) CF 3 -3-Py], [BE3215; 6-Cl-4-S (O) CF 3 -3-Py], [BE3216; 2-Me- _{4-S (O) CF 3} -3-Py], [BE3217; 5-Me-4-S (O) CF 3 -3-Py], [BE3218; 6-Me-4-S (O) CF 3 -3-Py], [BE 3219; 2-CF ₃ -4-S (O) CF ₃ -3-Py], [BE 3220; 5-CF ₃ -4-S (O) CF ₃ -3-Py], _{[BE3221; 6-CF 3 -4} -S (O) CF 3 -3-Py], [BE3222; 2-CN-4-S (O) CF 3 -3-Py], [BE3223; 5-CN- _{4-S (O) CF 3} -3-Py], [BE3224; 6-CN-4-S (O) CF 3 -3-Py], [BE3225; 2-OMe-4-S (O) CF 3 -3-Py], [BE3226; 5-OMe-4-S (O) CF 3 -3-Py], [BE3227; 6-OMe-4-S (O) CF 3 -3-Py], [BE3228 ; 5-S (O) CF 3 -3-Py], [BE3229; 2-Cl-5-S (O) CF 3 -3-Py], [BE3230; 4-Cl-5-S (O) CF _{3 -3-Py], [BE3231} ; 6-Cl-5-S (O) CF 3 -3-Py], [BE3232; 2-Me-5-S (O) CF 3 -3-Py], [ BE 3233; 4-Me-5-S (O) CF _3- 3-Py], [BE3234; 6-Me-5-S (O) CF 3 -3-Py], [BE3235; 2-CF 3 -5-S (O) CF 3 -3-Py], [BE3236 _{; 4-CF 3 -5-S} (O) CF 3 -3-Py], [BE3237; 6-CF 3 -5-S (O) CF 3 -3-Py], [BE3238; 2-CN-5 _{-S (O) CF 3 -3-} Py], [BE3239; 4-CN-5-S (O) CF 3 -3-Py], [BE3240; 6-CN-5-S (O) CF 3 - 3-Py], [BE3241; 2-OMe-5-S (O) CF 3 -3-Py], [BE3242; 4-OMe-5-S (O) CF 3 -3-Py], [BE3243; 6-OMe-5-S ( O) CF 3 -3-Py], [BE3244; 6-S (O) CF 3 -3-Py], [BE3245; 2-Cl-6-S (O) CF 3 -3-Py], [BE3246; 4-Cl-6-S (O) CF 3 -3-Py], [BE3247; 5-Cl-6-S (O) CF 3 -3-Py], [BE3248 ; 2-Me-6-S (O) CF 3 -3-Py], [BE3249; 4-Me-6-S (O) CF 3 -3-Py], [BE3250; 5-Me-6-S _{(O) CF 3 -3-Py} ], [BE3251; 2-CF 3 -6-S (O) CF 3 -3-Py], [BE3252; 4-CF 3 -6-S (O) CF 3 - 3-Py], [BE3253; 5-CF 3 -6-S (O) CF 3 -3-Py], [BE3254; 2-CN-6-S (O) CF 3 -3-Py], [BE3255 ; 4-CN-6-S (O) CF 3 -3-Py], [BE3256; 5-CN-6-S (O) CF 3 -3-Py], [BE3257; 2-OMe-6-S _{(O) CF 3 -3-Py} ], [BE3258; 4-OMe-6-S (O) CF 3 -3-Py], [BE3259; 5-OMe-6-S (O) C

F ₃ -3-Py !, [BE 3260; 4-Cl-2-S (O) ₂ Me-3-Py], [BE 3261; 5-Cl-2-S (O) ₂ Me-3-Py], [BE3262; 6-Cl-2 -S (O) 2 Me-3-Py], [BE3263; 4-Me-2-S (O) 2 Me-3-Py], [BE3264; 5-Me-2 _{-S (O) 2 Me-3} -Py], [BE3265; 6-Me-2-S (O) 2 Me-3-Py], [BE3266; 4-CF 3 -2-S (O) 2 Me -3-Py], [BE3267; 5-CF 3 -2-S (O) 2 Me-3-Py], [BE3268; 6-CF 3 -2-S (O) 2 Me-3-Py], [BE3269; 4-CN-2 -S (O) 2 Me-3-Py], [BE3270; 5-CN-2-S (O) 2 Me-3-Py], [BE3271; 6-CN-2 _{-S (O) 2 Me-3} -Py], [BE3272; 4-OMe-2-S (O) 2 Me-3-Py], [BE3273; 5-OMe-2-S (O) 2 Me- 3-Py], [BE3274; 6-OMe-2-S (O) 2 Me-3-Py], [BE3275; 4-S (O) 2 Me-3-Py], [BE3276; 2-Cl- _{4-S (O) 2 Me} -3-Py], [BE3277; 5-Cl-4-S (O) 2 Me-3-Py], [BE3278; 6-Cl-4-S (O) 2 Me -3-Py !, [BE3279; 2-Me-4-S (O) ₂ Me-3-Py], [BE3280; 5-Me-4-S (O) ₂ Me-3-Py], [BE3281 ; 6-Me-4-S (O) 2 Me-3-Py], [BE3282; 2-CF 3 -4-S (O) 2 Me-3-Py], [BE3283; 5-CF 3 -4 _{-S (O) 2 Me-3} -Py], [BE3284; 6-CF 3 -4-S (O) 2 Me-3-Py], [BE3285; 2-CN-4-S (O) 2 Me -3-Py !, [BE3286; 5-CN-4-S (O) ₂ Me-3-Py], [BE3287; 6-CN-4-S (O) ₂ Me-3-Py], [BE3288] ; 2-OMe-4-S (O) 2 Me-3-Py], [BE3289; 5-OMe-4-S (O) 2 Me-3-Py], [BE3290; 6-OMe-4-S (O) ₂ Me-3-Py], [BE 3291; 5 _{-S (O) 2 Me-3} -Py], [BE3292; 2-Cl-5-S (O) 2 Me-3-Py], [BE3293; 4-Cl-5-S (O) 2 Me- 3-Py], [BE3294; 6-Cl-5-S (O) 2 Me-3-Py], [BE3295; 2-Me-5-S (O) 2 Me-3-Py], [BE3296; 4-Me-5-S ( O) 2 Me-3-Py], [BE3297; 6-Me-5-S (O) 2 Me-3-Py], [BE3298; 2-CF 3 -5-S (O) ₂ Me-3-Py, [BE 3299; 4-CF ₃ -5-S (O) ₂ Me-3-Py], [BE 3300; 6-CF ₃ -5-S (O) ₂ Me- 3-Py], [BE 3301; 2-CN-5-S (O) ₂ Me-3-Py],

[BE3302; 4-CN-5 -S (O) 2 Me-3-Py], [BE3303; 6-CN-5-S (O) 2 Me-3-Py], [BE3304; 2-OMe-5 _{-S (O) 2 Me-3} -Py], [BE3305; 4-OMe-5-S (O) 2 Me-3-Py], [BE3306; 6-OMe-5-S (O) 2 Me- 3-Py], [BE3307; 6-S (O) 2 Me-3-Py], [BE3308; 2-Cl-6-S (O) 2 Me-3-Py], [BE3309; 4-Cl- _{6-S (O) 2 Me} -3-Py], [BE3310; 5-Cl-6-S (O) 2 Me-3-Py], [BE3311; 2-Me-6-S (O) 2 Me -3-Py !, [BE 3312; 4-Me-6-S (O) ₂ Me-3-Py], [BE 3313; 5-Me-6-S (O) ₂ Me-3-Py], [BE 3314 _{; 2-CF 3 -6-S} (O) 2 Me-3-Py], [BE3315; 4-CF 3 -6-S (O) 2 Me-3-Py], [BE3316; 5-CF 3 - _{6-S (O) 2 Me} -3-Py], [BE3317; 2-CN-6-S (O) 2 Me-3-Py], [BE3318; 4-CN-6-S (O) 2 Me -3-Py !, [BE3319; 5-CN-6-S (O) ₂ Me-3-Py], [BE3320; 2-OMe-6-S (O) ₂ Me-3-Py], [BE3321 ; 4-OMe-6-S (O) 2 Me-3-Py], [BE3322; 5-OMe-6-S (O) 2 Me-3-Py], [BE3323; 2-S (O) 2 _{CF 3 -3-Py], [} BE3324; 4-Cl-2-S (O) 2 CF 3 -3-Py], [BE3325; 5-Cl-2-S (O) 2 CF 3 -3-Py ], [BE3326; 6-Cl -2-S (O) 2 CF 3 -3-Py], [BE3327; 4-Me-2-S (O) 2 CF 3 -3-Py], [BE3328; 5 -Me-2-S (O) 2 CF 3 -3-Py], [BE3329; 6-Me-2-S (O) 2 CF 3 -3-Py], [BE3330; 4-CF 3 -2- _{S (O) 2 CF 3 -3} -Py], [BE3331; 5-CF 3 -2-S (O) 2 CF 3 -3-Py], [BE3332; 6-CF 3 -2-S (O) ₂ CF ₃ -3 -Py], [BE3333; 4- CN-2-S (O) 2 CF 3 -3-Py], [BE3334; 5-CN-2-S (O) 2 CF 3 -3-Py], [BE3335 ; 6-CN-2-S (O) 2 CF 3 -3-Py], [BE3336; 4-OMe-2-S (O) 2 CF 3 -3-Py], [BE3337; 5-OMe-2 _{-S (O) 2 CF 3 -3} -Py], [BE3338; 6-OMe-2-S (O) 2 CF 3 -3-Py], [BE3339; 4-S (O) 2 CF 3 -3 -Py], [BE3340; 2- Cl-4-S (O) 2 CF 3 -3-Py], [BE3341; 5-Cl-4-S (O) 2 CF 3 -3-Py], [BE3342 ; 6-Cl-4-S (O) 2 CF 3 -3-Py], [BE3343; 2-Me-4-S (O) 2 CF 3 -3-Py], [BE3344; 5-Me-4 _{-S (O) 2 CF 3 -3} -Py], [BE3345; 6-Me-4-S (O) 2 CF 3 -3-Py], [BE3346; 2-CF 3 -4-S (O) ₂ CF ₃ -3-Py, [BE 3347; 5-CF ₃ -4-S (O) ₂ CF ₃ -3-Py], [BE 3348; 6-CF ₃ -4-S (O) ₂ CF _3- 3-Py], [BE3349; 2-CN-4-S (O) 2 CF 3 -3-Py], [BE3350; 5-CN-4-S (O) 2 CF 3 -3-Py], [ BE3351; 6-CN-4- S (O) 2 CF 3 -3-Py], [BE3352; 2-OMe-4-S (O) 2 CF 3 -3-Py], [BE3353; 5-OMe- _{4-S (O) 2 CF} 3 -3-Py], [BE3354; 6-OMe-4-S (O) 2 CF 3 -3-Py], [BE3355; 5-S (O) 2 CF 3 - 3-Py], [BE3356; 2-Cl-5-S (O) 2 CF 3 -3-Py], [BE3357; 4-Cl-5-S (O) 2 CF 3 -3-Py], [ BE3358; 6-Cl-5- S (O) 2 CF 3 -3-Py], [BE3359; 2-Me-5-S (O) 2 CF 3 -3-Py], [BE3360; 4-Me- _{5-S (O) 2 CF} 3 -3-Py], [BE3361; 6-Me-5-S (O) 2 CF 3 -3-Py], [BE3 _{362; 2-CF 3 -5-} S (O) 2 CF 3 -3-Py], [BE3363; 4-CF 3 -5-S (O) 2 CF 3 -3-Py], [BE3364; 6- _{CF 3 -5-S (O)} 2 CF 3 -3-Py], [BE3365; 2-CN-5-S (O) 2 CF 3 -3-Py], [BE3366; 4-CN-5-S _{(O) 2 CF 3 -3-} Py], [BE3367; 6-CN-5-S (O) 2 CF 3 -3-Py], [BE3368; 2-OMe-5-S (O) 2 CF 3 -3-Py], [BE3369; 4-OMe-5-S (O) 2 CF 3 -3-Py], [BE3370; 6-OMe-5-S (O) 2 CF 3 -3-Py], [BE3371; 6-S (O ) 2 CF 3 -3-Py], [BE3372; 2-Cl-6-S (O) 2 CF 3 -3-Py], [BE3373; 4-Cl-6-S _{(O) 2 CF 3 -3-} Py], [BE3374; 5-Cl-6-S (O) 2 CF 3 -3-Py], [BE3375; 2-Me-6-S (O) 2 CF 3 -3-Py], [BE3376; 4-Me-6-S (O) 2 CF 3 -3-Py], [BE3377; 5-Me-6-S (O) 2 CF 3 -3-Py], _{[BE3378; 2-CF 3 -6} -S (O) 2 CF 3 -3-Py], [BE3379; 4-CF 3 -6-S (O) 2 CF 3 -3-Py], [BE3380; 5 _{-CF 3 -6-S (O)} 2 CF 3 -3-Py], [BE3381; 2-CN-6-S (O) 2 CF 3 -3-Py], [BE3382; 4-CN-6- _{S (O) 2 CF 3 -3} -Py], [BE3383; 5-CN-6-S (O) 2 CF 3 -3-Py], [BE3384; 2-OMe-6-S (O) 2 CF _{3 -3-Py], [BE3385} ; 4-OMe-6-S (O) 2 CF 3 -3-Py], [BE3386; 5-OMe-6-S (O) 2 CF 3 -3-Py] , [BE3387; 2-CN-3-Py], [BE3388; 4-Cl-2-CN-3-Py], [BE3389; 5-Cl-2-CN-3-Py], [BE3390; 6- Cl-2-CN-3-Py, [BE3391; 4-Me-2-CN-3-Py], [BE3392; 5-Me-2-CN-3- Py], [BE3393; 6- Me-2-CN-3-Py], [BE3394; 4-CF 3 -2-CN-3-Py], [BE3395; 5-CF 3 -2-CN-3- Py], [BE3396; 6- CF 3 -2-CN-3-Py], [BE3397; 4-CN-2-CN-3-Py], [BE3398; 5-CN-2-CN-3-Py ], [BE3399; 6-CN-2-CN-3-Py], [BE3400; 4-OMe-2-CN-3-Py], [BE3401; 5-OMe-2-CN-3-Py],

[BE3402; 6-OMe-2-CN-3-Py], [BE3403; 4-CN-3-Py], [BE3404; 2-Cl-4-CN-3-Py], [BE3405; 5-Cl -4-CN-3-Py], [BE3406; 6-Cl-4-CN-3-Py], [BE3407; 2-Me-4-CN-3-Py], [BE3408; 5-Me-4 -CN-3-Py], [ BE3409; 6-Me-4-CN-3-Py], [BE3410; 2-CF 3 -4-CN-3-Py], [BE3411; 5-CF 3 -4 -CN-3-Py], [BE 3412; 6-CF ₃ -4-CN-3-Py], [BE 3413; 2-CN-4-CN-3-Py], [BE 3414; 5-CN-4- CN-3-Py !, [BE3415; 6-CN-4-CN-3-Py], [BE3416; 2-OMe-4-CN-3-Py], [BE3417; 5-OMe-4-CN- 3-Py], [BE3418; 6-OMe-4-CN-3-Py], [BE3419; 5-CN-3-Py], [BE3420; 2-Cl-5-CN-3-Py], [BE3 419; BE3421; 4-Cl-5-CN-3-Py], [BE3422; 6-Cl-5-CN-3-Py], [BE3423; 2-Me-5-CN-3-Py], [BE3424; 4-Me-5-CN- 3-Py], [BE3425; 6-Me-5-CN-3-Py], [BE3426; 2-CF 3 -5-CN-3-Py], [BE3427; 4 _{-CF 3 -5-CN-3-} Py], [BE3428; 6-CF 3 -5-CN-3-Py], [BE3429; 2-CN-5-CN-3-Py], [BE3430; 4 -CN-5-CN-3-Py], [BE3431; 6-CN-5-CN-3-Py], [BE3432; 2-OMe-5-CN-3-Py], [BE3433; 4-OMe -5-CN-3-Py !, [BE3434; 6-OMe-5-CN-3-Py], [BE3435; 6-CN-3-Py], [BE3436; 2-Cl-6-CN-3 -Py], [BE3437; 4-Cl-6-CN-3-Py], [BE3438; 5-Cl-6-CN-3-Py], [BE3439; 2-Me-6-CN-3-Py ], [BE3440; 4-Me -6-CN-3-Py], [BE3441; 5-Me-6-CN-3-Py], [BE3442; 2-CF 3 -6-CN-3-Py] , [BE _{3443; 4-CF 3 -6-} CN-3-Py], [BE3444; 5-CF 3 -6-CN-3-Py], [BE3445; 2-CN-6-CN-3-Py], [ BE3446; 4-CN-6-CN-3-Py], [BE3447; 5-CN-6-CN-3-Py], [BE 3448; 2-OMe-6-CN-3-Py], [BE3449; 4-OMe-6-CN-3-Py], [BE3450; 5-OMe-6-CN-3-Py], [BE3451; 2-COOMe-3-Py], [BE3452; 4-Cl-2- COOMe-3-Py !, [BE 3453; 5-Cl-2-COOMe-3-Py], [BE 3454; 6-Cl-2-COOMe-3-Py], [BE 3455; 4-Me-2-COOMe- 3-Py], [BE3456; 5-Me-2-COOMe-3-Py], [BE3457; 6-Me-2-COOMe-3-Py], [BE3458; 4-CF 3 -2-COOMe-3 -Py], [BE3459; 5- CF 3 -2-COOMe-3-Py], [BE3460; 6-CF 3 -2-COOMe-3-Py], [BE3461; 4-CN-2-COOMe-3 -Py], [BE3462; 5-CN-2-COOMe-3-Py], [BE3463; 6-CN-2-COOMe-3-Py], [BE 3464; 4-OMe-2-COOMe-3-Py ], [BE3465; 5-OMe-2-COOMe-3-Py], [BE3466; 6-OMe-2-COOMe-3-Py], [BE3467; 4-COOMe-3-Py], [BE3468; -Cl-4-COOMe-3-Py], [BE3469; 5-Cl-4-COOMe-3-Py], [BE3470; 6-Cl-4-COOMe-3-Py], [BE3471; 2-Me -4-COOMe-3-Py !, [BE3472; 5-Me-4-COOMe-3-Py], [BE3473; 6-Me-4-COOMe-3-Py], [BE3474; 2-CF _3- 4-COOMe-3-Py] , [BE3475; 5-CF 3 -4-COOMe-3-Py], [BE3476; 6-CF 3 -4-COOMe-3-Py], [BE3477; 2-CN- 4-COOMe-3-Py], [BE3478; 5-CN-4-COOMe-3-Py], [BE3479; 6-CN-4-COOMe-3-Py], [BE3480; 2-OMe-4-COOMe-3-Py], [BE3481; 5-OMe-4-COOMe-3-Py], [BE3482; 6-OMe-4-COOMe-3-Py], [BE3483; COOMe-3-Py], [BE3484; 2-Cl-5-COOMe-3-Py], [BE3485; 4-Cl-5-COOMe-3-Py], [BE3486; 6-Cl-5-COOMe- 3-Py], [BE3487; 2-Me-5-COOMe-3-Py], [BE3488; 4-Me-5-COOMe-3-Py], [BE3489; 6-Me-5-COOMe-3- Py], [BE3490; 2- CF 3 -5-COOMe-3-Py], [BE3491; 4-CF 3 -5-COOMe-3-Py], [BE3492; 6-CF 3 -5-COOMe-3 -Py], [BE3493; 2-CN-5-COOMe-3-Py], [BE3494; 4-CN-5-COOMe-3-Py], [BE3495; 6-CN-5-COOMe-3-Py ], [BE3496; 2-OMe-5-COOMe-3-Py], [BE3497; 4-OMe-5-COOMe-3-Py], [BE3498; 6-OMe-5-COOMe-3-Py], [BE3499; 6-COOMe-3-Py], [BE3500; 2-Cl-6-COOMe-3-Py], [BE3501; 4-Cl-6-COOMe-3-Py],

[BE3502; 5-Cl-6-COOMe-3-Py], [BE3503; 2-Me-6-COOMe-3-Py], [BE3504; 4-Me-6-COOMe-3-Py], [BE3505] ; 5-Me-6-COOMe -3-Py], [BE3506; 2-CF 3 -6-COOMe-3-Py], [BE3507; 4-CF 3 -6-COOMe-3-Py], [BE3508 _{; 5-CF 3 -6-COOMe} -3-Py], [BE3509; 2-CN-6-COOMe-3-Py], [BE3510; 4-CN-6-COOMe-3-Py], [BE3511; 5-CN-6-COOMe-3-Py], [BE 3512; 2-OMe-6-COOMe-3-Py], [BE 3513; 4-OMe-6-COOMe-3-Py], [BE 3514; OMe-6-COOMe-3- Py], [BE3515; 2-NO 2 -3-Py], [BE3516; 4-Cl-2-NO 2 -3-Py], [BE3517; 5-Cl-2- _{NO 2 -3-Py], [} BE3518; 6-Cl-2-NO 2 -3-Py], [BE3519; 4-Me-2-NO 2 -3-Py], [BE3520; 5-Me-2 _{-NO 2 -3-Py], [} BE3521; 6-Me-2-NO 2 -3-Py], [BE3522; 4-CF 3 -2-NO 2 -3-Py], [BE3523; 5-CF _{3 -2-NO 2 -3-Py} ], [BE3524; 6-CF 3 -2-NO 2 -3-Py], [BE3525; 4-CN-2-NO 2 -3-Py], [BE3526; _{5-CN-2-NO 2} -3-Py], [BE3527; 6-CN-2-NO 2 -3-Py], [BE3528; 4-OMe-2-NO 2 -3-Py], [BE3529 ; 5-OMe-2-NO 2 -3-Py], [BE3530; 6-OMe-2-NO 2 -3-Py], [BE3531; 4-NO 2 -3-Py], [BE3532; 2- _{Cl-4-NO 2 -3-} Py], [BE3533; 5-Cl-4-NO 2 -3-Py], [BE3534; 6-Cl-4-NO 2 -3-Py], [BE3535; 2 _{-Me-4-NO 2 -3-} Py], [BE3536; 5-Me-4-NO 2 -3-Py], [BE3537; 6-Me-4-NO 2 -3-Py], [BE3538; 2-CF _{3 -4-NO 2 -3-Py]} , [BE3539; 5-CF 3 -4-NO 2 -3-Py], [BE3540; 6-CF 3 -4-NO 2 -3-Py], [BE3541; _{2-CN-4-NO 2} -3-Py], [BE3542; 5-CN-4-NO 2 -3-Py], [BE3543; 6-CN-4-NO 2 -3-Py], [BE3544 ; 2-OMe-4-NO 2 -3-Py], [BE3545; 5-OMe-4-NO 2 -3-Py], [BE3546; 6-OMe-4-NO 2 -3-Py], [ BE 3547; 5-NO ₂ -3-Py], [BE 3548; 2-Cl -5-NO ₂ -3-Py], [BE 3 549; 4-Cl -5-NO ₂ -3-Py], [BE 3550; 6 _{-Cl-5-NO 2 -3-} Py], [BE3551; 2-Me-5-NO 2 -3-Py], [BE3552; 4-Me-5-NO 2 -3-Py], [BE3553; _{6-Me-5-NO 2} -3-Py], [BE3554; 2-CF 3 -5-NO 2 -3-Py], [BE3555; 4-CF 3 -5-NO 2 -3-Py], _{[BE3556; 6-CF 3 -5} -NO 2 -3-Py], [BE3557; 2-CN-5-NO 2 -3-Py], [BE3558; 4-CN-5-NO 2 -3-Py ], [BE3559; 6-CN -5-NO 2 -3-Py], [BE3560; 2-OMe-5-NO 2 -3-Py], [BE3561; 4-OMe-5-NO 2 -3- Py], [BE3562; 6- OMe-5-NO 2 -3-Py], [BE3563; 6-NO 2 -3-Py], [BE3564; 2-Cl-6-NO 2 -3-Py], [BE3565; 4-Cl-6 -NO 2 -3-Py], [BE3566; 5-Cl-6-NO 2 -3-Py], [BE3567; 2-Me-6-NO 2 -3-Py] , [BE3568; 4-Me- 6-NO 2 -3-Py], [BE3569; 5-Me-6-NO 2 -3-Py], [BE3570; 2-CF 3 -6-NO 2 -3- Py], [BE3571; 4- CF 3 -6-NO 2 -3-Py], [BE3572; 5-CF 3 -6-NO 2 -3-Py], [BE3573; 2-CN-6-NO 2 -3-Py], [BE 3574; 4-CN-6-NO ₂ -3-Py], [BE3575; 5-CN-6-NO 2 -3-Py], [BE3576; 2-OMe-6-NO 2 -3-Py], [BE3577; 4-OMe-6-NO _{2 -3-Py], [BE3578} ; 5-OMe-6-NO 2 -3-Py], [BE3579; 4-Cl-2-NH 2 -3-Py], [BE3580; 5-Cl-2- _{NH 2 -3-Py], [} BE3581; 6-Cl-2-NH 2 -3-Py], [BE3582; 4-Me-2-NH 2 -3-Py], [BE3583; 5-Me-2 _{-NH 2 -3-Py], [} BE3584; 6-Me-2-NH 2 -3-Py], [BE3585; 4-CF 3 -2-NH 2 -3-Py], [BE3586; 5-CF _{3 -2-NH 2 -3-Py} ], [BE3587; 6-CF 3 -2-NH 2 -3-Py], [BE3588; 4-CN-2-NH 2 -3-Py], [BE3589; _{5-CN-2-NH 2} -3-Py], [BE3590; 6-CN-2-NH 2 -3-Py], [BE3591; 4-OMe-2-NH 2 -3-Py], [BE3592 ; 5-OMe-2-NH 2 -3-Py], [BE3593; 6-OMe-2-NH 2 -3-Py], [BE3594; 4-NH 2 -3-Py], [BE3595; 2- _{Cl-4-NH 2 -3-} Py], [BE3596; 5-Cl-4-NH 2 -3-Py], [BE3597; 6-Cl-4-NH 2 -3-Py], [BE3598; 2 _{-Me-4-NH 2 -3-} Py], [BE3599; 5-Me-4-NH 2 -3-Py], [BE3600; 6-Me-4-NH 2 -3-Py], [BE3601; _{2-CF 3 -4-NH 2} -3-Py],

_{[BE3602; 5-CF 3 -4} -NH 2 -3-Py], [BE3603; 6-CF 3 -4-NH 2 -3-Py], [BE3604; 2-CN-4-NH 2 -3- Py], [BE3605; 5- CN-4-NH 2 -3-Py], [BE3606; 6-CN-4-NH 2 -3-Py], [BE3607; 2-OMe-4-NH 2 -3 -Py], [BE3608; 5- OMe-4-NH 2 -3-Py], [BE3609; 6-OMe-4-NH 2 -3-Py], [BE3610; 5-NH 2 -3-Py] , [BE3611; 2-Cl- 5-NH 2 -3-Py], [BE3612; 4-Cl-5-NH 2 -3-Py], [BE3613; 6-Cl-5-NH 2 -3-Py ], [BE3614; 2-Me -5-NH 2 -3-Py], [BE3615; 4-Me-5-NH 2 -3-Py], [BE3616; 6-Me-5-NH 2 -3- Py], [BE3617; 2- CF 3 -5-NH 2 -3-Py], [BE3618; 4-CF 3 -5-NH 2 -3-Py], [BE3619; 6-CF 3 -5-NH _{2 -3-Py], [BE3620} ; 2-CN-5-NH 2 -3-Py], [BE3621; 4-CN-5-NH 2 -3-Py], [BE3622; 6-CN-5- _{NH 2 -3-Py], [} BE3623; 2-OMe-5-NH 2 -3-Py], [BE3624; 4-OMe-5-NH 2 -3-Py], [BE3625; 6-OMe-5 _{-NH 2 -3-Py], [} BE3626; 6-NH 2 -3-Py], [BE3627; 2-Cl-6-NH 2 -3-Py], [BE3628; 4-Cl-6-NH 2 -3-Py], [BE3629; 5-Cl-6-NH 2 -3-Py], [BE3630; 2-Me-6-NH 2 -3-Py], [BE3631; 4-Me-6-NH _{2 -3-Py], [BE3632} ; 5-Me-6-NH 2 -3-Py], [BE3633; 2-CF 3 -6-NH 2 -3-Py], [BE3634; 4-CF 3 - _{6-NH 2 -3-Py]} , [BE3635; 5-CF 3 -6-NH 2 -3-Py], [BE3636; 2-CN-6-NH 2 -3-Py], [BE3637; 4- _{CN-6-NH 2 -3-} Py], [BE3638; _{5-CN-6-NH 2} -3-Py], [BE3639; 2-OMe-6-NH 2 -3-Py], [BE3640; 4-OMe-6-NH 2 -3-Py], [BE3641 ; 5-OMe-6-NH 2 -3-Py], [BE3642; 2-NHMe-3-Py], [BE3643; 4-Cl-2-NHMe-3-Py], [BE3644; 5-Cl- 2-NHMe-3-Py, [BE3645; 6-Cl-2-NHMe-3-Py], [BE3646; 4-Me-2-NHMe-3-Py], [BE3647; 5-Me-2- NHMe-3-Py !, [BE 3648; 6-Me-2-NHMe-3-Py], [BE 3649; 4-CF ₃ -2-NHMe-3-Py], [BE 3650; 5-CF ₃ -2-] NHMe-3-Py], [ BE3651; 6-CF 3 -2-NHMe-3-Py], [BE3652; 4-CN-2-NHMe-3-Py], [BE3653; 5-CN-2-NHMe -3-Py !, [BE3654; 6-CN-2-NHMe-3-Py], [BE 3655; 4-OMe-2-NHMe-3-Py], [BE 3656; 5-OMe-2-NHMe-3 -Py], [BE3657; 6-OMe-2-NHMe-3-Py], [BE3658; 4-NHMe-3-Py], [BE3659; 2-Cl-4-NHMe-3-Py], [BE3660] 5-Cl-4-NHMe-3-Py !, [BE3661; 6-Cl-4-NHMe-3-Py], [BE3662; 2-Me-4-NHMe-3-Py], [BE3663; -Me-4-NHMe-3- Py], [BE3664; 6-Me-4-NHMe-3-Py], [BE3665; 2-CF 3 -4-NHMe-3-Py], [BE3666; 5- _{CF 3 -4-NHMe-3-} Py], [BE3667; 6-CF 3 -4-NHMe-3-Py], [BE3668; 2-CN-4-NHMe-3-Py], [BE3669; 5- CN-4-NHMe-3-Py, [BE3670; 6-CN-4-NHMe-3-Py], [BE3671; 2-OMe-4-NHMe-3-Py], [BE3672; 5-OMe- 4-NHMe-3-Py, [BE3673; 6-OMe-4-NHMe-3-Py], [BE3674; 5-NHMe-3-Py], [BE3675; 2-Cl-5-NHMe-3- Py], [BE3 676; 4-Cl-5-NHMe-3-Py], [BE3677; 6-Cl-5-NHMe-3-Py], [BE3678; 2-Me-5-NHMe-3-Py], [BE3679; 4-Me-5-NHMe- 3-Py], [BE3680; 6-Me-5-NHMe-3-Py], [BE3681; 2-CF 3 -5-NHMe-3-Py], [BE3682; 4 _{-CF 3 -5-NHMe-3-} Py], [BE3683; 6-CF 3 -5-NHMe-3-Py], [BE3684; 2-CN-5-NHMe-3-Py], [BE3685; 4 -CN-5-NHMe-3-Py], [BE3686; 6-CN-5-NHMe-3-Py], [BE3687; 2-OMe-5-NHMe-3-Py], [BE3688; 4-OMe -5-NHMe-3-Py !, [BE3689; 6-OMe-5-NHMe-3-Py], [BE3690; 6-NHMe-3-Py], [BE3691; 2-Cl-6-NHMe-3 -Py], [BE3692; 4-Cl-6-NHMe-3-Py], [BE3693; 5-Cl-6-NHMe-3-Py], [BE3694; 2-Me-6-NHMe-3-Py ], [BE3695; 4-Me -6-NHMe-3-Py], [BE3696; 5-Me-6-NHMe-3-Py], [BE3697; 2-CF 3 -6-NHMe-3-Py] _{, [BE3698; 4-CF 3} -6-NHMe-3-Py], [BE3699; 5-CF 3 -6-NHMe-3-Py], [BE3700; 2-CN-6-NHMe-3-Py] , [BE3701; 4-CN-6-NHMe-3-Py],

[BE3702; 5-CN-6-NHMe-3-Py], [BE3703; 2-OMe-6-NHMe-3-Py], [BE3704; 4-OMe-6-NHMe-3-Py], [BE3705] ; 5-OMe-6-NHMe -3-Py], [BE3706; 2-NMe 2 -3-Py], [BE3707; 4-Cl-2-NMe 2 -3-Py], [BE3708; 5-Cl _{-2-NMe 2 -3-Py]} , [BE3709; 6-Cl-2-NMe 2 -3-Py], [BE3710; 4-Me-2-NMe 2 -3-Py], [BE3711; 5- _{Me-2-NMe 2 -3-} Py], [BE3712; 6-Me-2-NMe 2 -3-Py], [BE3713; 4-CF 3 -2-NMe 2 -3-Py], [BE3714; _{5-CF 3 -2-NMe 2} -3-Py], [BE3715; 6-CF 3 -2-NMe 2 -3-Py], [BE3716; 4-CN-2-NMe 2 -3-Py], [BE3717; 5-CN-2 -NMe 2 -3-Py], [BE3718; 6-CN-2-NMe 2 -3-Py], [BE3719; 4-OMe-2-NMe 2 -3-Py] , [BE3720; 5-OMe- 2-NMe 2 -3-Py], [BE3721; 6-OMe-2-NMe 2 -3-Py], [BE3722; 4-NMe 2 -3-Py], [BE3723 ; 2-Cl-4-NMe 2 -3-Py], [BE3724; 5-Cl-4-NMe 2 -3-Py], [BE3725; 6-Cl-4-NMe 2 -3-Py], [ BE3726; 2-Me-4- NMe 2 -3-Py], [BE3727; 5-Me-4-NMe 2 -3-Py], [BE3728; 6-Me-4-NMe 2 -3-Py], _{[BE3729; 2-CF 3 -4} -NMe 2 -3-Py], [BE3730; 5-CF 3 -4-NMe 2 -3-Py], [BE3731; 6-CF 3 -4-NMe 2 -3 -Py], [BE3732; 2- CN-4-NMe 2 -3-Py], [BE3733; 5-CN-4-NMe 2 -3-Py], [BE3734; 6-CN-4-NMe 2 - 3-Py], [BE3735; 2-OMe-4-NMe 2 -3-Py], [BE3736; 5-OMe-4-NMe 2 -3-Py], [BE3737; 6-OM _{e-4-NMe 2 -3-} Py], [BE3738; 5-NMe 2 -3-Py], [BE3739; 2-Cl-5-NMe 2 -3-Py], [BE3740; 4-Cl-5 _{-NMe 2 -3-Py], [} BE3741; 6-Cl-5-NMe 2 -3-Py], [BE3742; 2-Me-5-NMe 2 -3-Py], [BE3743; 4-Me- _{5-NMe 2 -3-Py]} , [BE3744; 6-Me-5-NMe 2 -3-Py], [BE3745; 2-CF 3 -5-NMe 2 -3-Py], [BE3746; 4- _{CF 3 -5-NMe 2 -3-} Py], [BE3747; 6-CF 3 -5-NMe 2 -3-Py], [BE3748; 2-CN-5-NMe 2 -3-Py], [BE3749 ; 4-CN-5-NMe 2 -3-Py], [BE3750; 6-CN-5-NMe 2 -3-Py], [BE3751; 2-OMe-5-NMe 2 -3-Py], [ BE3752; 4-OMe-5- NMe 2 -3-Py], [BE3753; 6-OMe-5-NMe 2 -3-Py], [BE3754; 6-NMe 2 -3-Py], [BE3755; 2 _{-Cl-6-NMe 2 -3-} Py], [BE3756; 4-Cl-6-NMe 2 -3-Py], [BE3757; 5-Cl-6-NMe 2 -3-Py], [BE3758; _{2-Me-6-NMe 2} -3-Py], [BE3759; 4-Me-6-NMe 2 -3-Py], [BE3760; 5-Me-6-NMe 2 -3-Py], [BE3761 _{; 2-CF 3 -6-NMe} 2 -3-Py], [BE3762; 4-CF 3 -6-NMe 2 -3-Py], [BE3763; 5-CF 3 -6-NMe 2 -3-Py ], [BE3764; 2-CN -6-NMe 2 -3-Py], [BE3765; 4-CN-6-NMe 2 -3-Py], [BE3766; 5-CN-6-NMe 2 -3- Py], [BE3767; 2- OMe-6-NMe 2 -3-Py], [BE3768; 4-OMe-6-NMe 2 -3-Py], [BE3769; 5-OMe-6-NMe 2 -3 -Py], [BE3770; 2-ACNH-3-Py], [BE3771; 4-Cl-2-ACNH-3-Py], [BE3772; 5-Cl-2-ACNH-3-Py], [BE3773; 6-Cl-2-ACNH-3-Py], [BE3774; 4-Me-2-ACNH-3-Py], [BE3775; 5-Me-2-ACNH-3-Py], [BE3776 ; 6-Me-2-ACNH -3-Py], [BE3777; 4-CF 3 -2-ACNH-3-Py], [BE3778; 5-CF 3 -2-ACNH-3-Py], [BE3779 _{; 6-CF 3 -2-ACNH} -3-Py], [BE3780; 4-CN-2-ACNH-3-Py], [BE3781; 5-CN-2-ACNH-3-Py], [BE3782; 6-CN-2-ACNH-3-Py, [BE 3783; 4-OMe-2-ACNH-3-Py], [BE 3784; 5-OMe-2-ACNH-3-Py], [BE 3 785; OMe-2-ACNH-3-Py !, [BE3786; 4-ACNH-3-Py], [BE3787; 2-Cl-4-ACNH-3-Py], [BE3788; 5-Cl-4-ACNH- 3-Py], [BE3789; 6-Cl-4-ACNH-3-Py], [BE3790; 2-Me-4-ACNH-3-Py], [BE3791; 5-Me-4-ACNH-3- Py], [BE3792; 6- Me-4-ACNH-3-Py], [BE3793; 2-CF 3 -4-ACNH-3-Py], [BE3794; 5-CF 3 -4-ACNH-3- Py], [BE3795; 6- CF 3 -4-ACNH-3-Py], [BE3796; 2-CN-4-ACNH-3-Py], [BE3797; 5-CN-4-ACNH-3-Py ], [BE 3798; 6-CN-4-ACNH-3-Py], [BE 3799; 2-OMe-4-ACNH-3-Py], [BE 3800; 5-OMe-4-ACNH-3-Py], [BE3801; 6-OMe-4-ACNH-3-Py],

[BE 3802; 5-ACNH-3-Py], [BE 3803; 2-Cl-5-ACNH-3-Py], [BE 3804; 4-Cl-5-ACNH-3-Py], [BE 3805; 6-Cl -5-ACNH-3-Py, [BE3806; 2-Me-5-ACNH-3-Py], [BE3807; 4-Me-5-ACNH-3-Py], [BE3808; 6-Me-5 -ACNH-3-Py], [ BE3809; 2-CF 3 -5-ACNH-3-Py], [BE3810; 4-CF 3 -5-ACNH-3-Py], [BE3811; 6-CF 3 - 5-ACNH-3-Py, [BE3812; 2-CN-5-ACNH-3-Py], [BE3813; 4-CN-5-ACNH-3-Py], [BE3814; 6-CN-5- ACNH-3-Py], [BE3815; 2-OMe-5-ACNH-3-Py], [BE3816; 4-OMe-5-ACNH-3-Py], [BE3817; 6-OMe-5-ACNH- 3-Py], [BE3818; 6-ACNH-3-Py], [BE3819; 2-Cl-6-ACNH-3-Py], [BE3820; 4-Cl-6-ACNH-3-Py], [BE3 20] BE 3821; 5-Cl-6-ACNH-3-Py], [BE3822; 2-Me-6-ACNH-3-Py], [BE3823; 4-Me-6-ACNH-3-Py], [BE3824; 5-Me-6-ACNH- 3-Py], [BE3825; 2-CF 3 -6-ACNH-3-Py], [BE3826; 4-CF 3 -6-ACNH-3-Py], [BE3827; _{5-CF 3 -6-ACNH-} 3-Py], [BE3828; 2-CN-6-ACNH-3-Py], [BE3829; 4-CN-6-ACNH-3-Py], [BE3830; 5 -CN-6-ACNH-3-Py], [BE3831; 2-OMe-6-ACNH-3-Py], [BE3832; 4-OMe-6-ACNH-3-Py], [BE3833; 5-OMe -6-ACNH-3-Py, [BE3834; 2- (N-AC-N-Me-N) -3-Py], [BE3835; 4-Cl-2- (N (Ac) (Me)) -3-Py !, [BE3836; 5-Cl-2- (N (Ac) (Me))-3-Py], [BE3837; 6-Cl-2- (N (Ac) (Me))-3 -Py], [BE 3838; 4-Me-2- (N (Ac)) (Me))-3-Py], [BE3839; 5-Me-2- (N (Ac) (Me))-3-Py], [BE3840; 6-Me-2- (N (Ac) (Me) )) 3-Py], [BE3841; 4-CF ₃ -2- (N (Ac) (Me))-3-Py], [BE3842; 5-CF ₃ -2- (N (Ac) (Me) )) 3-Py], [BE3843; 6-CF ₃ -2- (N (Ac) (Me))-3-Py], [BE3844; 4-CN-2- (N (Ac) (Me)) )-[3-Py], [BE3845; 5-CN-2- (N (Ac) (Me))-3-Py], [BE3846; 6-CN-2- (N (Ac) (Me))- 3-Py], [BE3847; 4-OMe-2- (N (Ac) (Me))-3-Py], [BE3848; 5-OMe-2- (N (Ac) (Me))-3- Py], [BE3849; 6-OMe-2- (N (Ac) (Me))-3-Py], [BE3850; 4- (N-AC-N-Me-N) -3-Py], BE3851; 2-Cl-4- (N (Ac) (Me))-3-Py], [BE3852; 5-Cl-4- (N (Ac) (Me))-3-Py], [BE3853; 6-Cl-4- (N (Ac) (Me))-3-Py], [BE3854; 2-Me-4- (N (Ac) (Me))-3-Py], [BE3855; 5- Me-4- (N (Ac) (Me)) - 3-Py], [BE3856; 6-Me-4- (N (Ac) (Me)) - 3-Py], [BE3857; 2-CF 3 -4- (N (Ac) (Me )) - 3-Py], [BE3858; 5-CF 3 -4- (N (Ac) (Me)) - 3-Py], [BE3859; 6-CF 3 -4- (N (Ac) (Me))-3-Py], [BE3860; 2-CN-4- (N (Ac) (Me))-3-Py], [BE3861; 5-CN-4 -(N (Ac) (Me))-3-Py], [BE3862; 6-CN-4- (N (Ac) (Me))-3-Py], [BE3863; 2-OMe-4- ( N (Ac) (Me))-3-Py], [BE3864; 5-OMe-4- (N (Ac) (Me))-3-Py], [BE3865; 6-OMe-4- (N ( Ac) (Me))-3-Py], [BE3866; 5- (N-AC-N-Me-N) -3-Py], [BE3867; 2-Cl-5- (N (Ac) (Me) ))-3-Py], [BE38] 68; 4-Cl-5- (N (Ac) (Me))-3-Py], [BE3869; 6-Cl-5- (N (Ac) (Me))-3-Py], [BE3870; 2-Me-5- (N (Ac) (Me))-3-Py], [BE 3871; 4-Me-5- (N (Ac) (Me))-3-Py], [BE 3872; 6- Me-5- (N (Ac) (Me)) - 3-Py], [BE3873; 2-CF 3 -5- (N (Ac) (Me)) - 3-Py], [BE3874; 4-CF _{3 -5- (N (Ac) (} Me)) - 3-Py], [BE3875; 6-CF 3 -5- (N (Ac) (Me)) - 3-Py], [BE3876; 2-CN -5- (N (Ac) (Me))-3-Py], [BE 3877; 4-CN-5- (N (Ac) (Me))-3-Py], [BE 3878; 6-CN-5 -(N (Ac) (Me))-3-Py], [BE 3879; 2-OMe-5- (N (Ac) (Me))-3-Py], [BE 3880; 4-OMe-5- ( N (Ac) (Me))-3-Py], [BE3881; 6-OMe-5- (N (Ac) (Me))-3-Py], [BE3882; 6- (N-AC-N-] Me-N) -3-Py], [BE 3883; 2-Cl-6- (N (Ac) (Me))-3-Py], [BE 3884; 4-Cl-6- (N (Ac) (Me) )) 3-Py], [BE3885; 5-Cl-6- (N (Ac) (Me))-3-Py], [BE3886; 2-Me-6- (N (Ac) (Me)) -3-Py !, [BE3887; 4-Me-6- (N (Ac) (Me))-3-Py], [BE3888; 5-Me-6- (N (Ac) (Me))-3] -Py], [BE3889; 2- CF 3 -6- (N (Ac) (Me)) - 3-Py], [BE3890; 4-CF 3 -6- (N (Ac) (Me)) - 3 -Py], [BE3891; 5- CF 3 -6- (N (Ac) (Me)) - 3-Py], [BE3892; 2-CN-6- (N (Ac) (Me)) - 3- Py], [BE3893; 4-CN-6- (N (Ac) (Me))-3-Py], [BE3894; 5-CN-6- (N (Ac) (Me))-3-Py] , [BE3895; 2-OMe-6- (N (Ac) (Me))-3-Py], [BE3896; 4-OMe-6- (N (Ac) (Me))-3-Py], [BE3896; BE3897; 5-OMe-6- (N (Ac) (M) e))-3-Py], [BE3898; 2-AC-3-Py], [BE3899; 4-Cl-2-AC-3-Py], [BE 3900; 5-Cl-2-AC-3- Py], [BE 3901; 6-Cl-2-AC-3-Py],

[BE 3902; 4-Me-2-AC-3-Py], [BE 3903; 5-Me-2-AC-3-Py], [BE 3904; 6-Me-2-AC-3-Py], [BE 3905] _{; 4-CF 3 -2-AC} -3-Py], [BE3906; 5-CF 3 -2-AC-3-Py], [BE3907; 6-CF 3 -2-AC-3-Py], [ BE3908; 4-CN-2-AC-3-Py], [BE3909; 5-CN-2-AC-3-Py], [BE3910; 6-CN-2-AC-3-Py], [BE3911; 4-OMe-2-AC-3-Py !, [BE3912; 5-OMe-2-AC-3-Py], [BE3913; 6-OMe-2-AC-3-Py], [BE3914; AC-3-Py !, [BE3915; 2-Cl-4-AC-3-Py], [BE3916; 5-Cl-4-AC-3-Py], [BE3917; 6-Cl-4-AC- 3-Py], [BE3918; 2-Me-4-AC-3-Py], [BE3919; 5-Me-4-AC-3-Py], [BE3920; 6-Me-4-AC-3- Py], [BE 3921; 2-CF ₃ -4-AC-3-Py], [BE 3922; 5-CF ₃ -4-AC-3-Py], [BE 3923; 6-CF ₃ -4-AC-3 -Py], [BE3924; 2-CN-4-AC-3-Py], [BE3925; 5-CN-4-AC-3-Py], [BE3926; 6-CN-4-AC-3-Py ], [BE3927; 2-OMe-4-AC-3-Py], [BE3928; 5-OMe-4-AC-3-Py], [BE3929; 6-OMe-4-AC-3-Py], [BE3930; 5-AC-3-Py], [BE 3931; 2-Cl-5-AC-3-Py], [BE 3932; 4-Cl-5-AC-3-Py], [BE 3933; 6-Cl -5-AC-3-Py, [BE3934; 2-Me-5-AC-3-Py], [BE 3935; 4-Me-5-AC-3-Py], [BE 3936; 6-Me-5 -AC-3-Py], [ BE3937; 2-CF 3 -5-AC-3-Py], [BE3938; 4-CF 3 -5-AC-3-Py], [BE3939; 6-CF 3 - 5-AC-3-Py, [BE3940; 2-CN-5-AC-3-Py], [BE3941; 4-CN-5-AC-3-Py], [BE3942; 6-CN-5- AC -3-Py], [BE3943; 2-OMe-5-AC-3-Py], [BE3944; 4-OMe-5-AC-3-Py], [BE3945; 6-OMe-5-AC-3 -Py], [BE3946; 6-AC-3-Py], [BE3947; 2-Cl-6-AC-3-Py], [BE3948; 4-Cl-6-AC-3-Py], [BE3949] 5-Cl-6-AC-3-Py !, [BE3950; 2-Me-6-AC-3-Py], [BE3951; 4-Me-6-AC-3-Py], [BE3952; -Me-6-AC-3- Py], [BE3953; 2-CF 3 -6-AC-3-Py], [BE3954; 4-CF 3 -6-AC-3-Py], [BE3955; 5 _{-CF 3 -6-AC-3-} Py], [BE3956; 2-CN-6-AC-3-Py], [BE3957; 4-CN-6-AC-3-Py], [BE3958; 5- CN-6-AC-3-Py, [BE3959; 2-OMe-6-AC-3-Py], [BE3960; 4-OMe-6-AC-3-Py], [BE3961; 5-OMe- 6-AC-3-Py], [BE3962; 4-Py], 0 [BE3963; 3-F-4-Py], [BE3964; 2-Cl-3-F-4-Py], [BE3965; -Cl-3-F-4-Py], [BE3966; 6-Cl-3-F-4-Py], [BE3967; 2-Me-3-F-4-Py], [BE 3968; 5-Me -3-F-4-Py !, [BE 3969; 6-Me-3-F-4-Py], [BE 3970; 2-CF ₃ -3-F-4-Py], [BE 3971; 5-CF ₃ -3-F-4-Py] , [BE3972; 6-CF 3 -3-F-4-Py], [BE3973; 2-CN-3-F-4-Py], [BE3974; 5-CN- 3-F-4-Py], [BE3975; 6-CN-3-F-4-Py], [BE3976; 2-OMe-3-F-4-Py], [BE3977; 5-OMe-3- F-4-Py !, [BE3978; 6-OMe-3-F-4-Py], [BE3979; 2-F-4-Py], [BE3980; 3-Cl-2-F-4-Py] [BE 3981; 5-Cl-2-F-4-Py], [BE 3982; 6-Cl-2-F-4-Py], [BE 3983; 3-Me-2-F-4-Py], [BE 3982; BE 3984; 5-Me-2-F-4-Py], [B E3985; 6-Me-2- F-4-Py], [BE3986; 3-CF 3 -2-F-4-Py], [BE3987; 5-CF 3 -2-F-4-Py], [ _{BE3988; 6-CF 3 -2-} F-4-Py], [BE3989; 3-CN-2-F-4-Py], [BE3990; 5-CN-2-F-4-Py], [BE3991 6-CN-2-F-4-Py !, [BE3992; 3-OMe-2-F-4-Py], [BE3993; 5-OMe-2-F-4-Py], [BE3994; -OMe-2-F-4-Py], [BE 3995; 5-F-4-Py], [BE 3996; 3-Cl-5-F-4-Py], [BE 3997; 2-Cl-5-F -4-Py], [BE 3998; 6-Cl-5-F-4-Py], [BE 3 999; 3-Me-5-F-4-Py], [BE 4000; 2-Me-5-F-4 -Py], [BE4001; 6-Me-5-F-4-Py],

_{[BE4002; 3-CF 3 -5} -F-4-Py], [BE4003; 2-CF 3 -5-F-4-Py], [BE4004; 6-CF 3 -5-F-4-Py] , [BE4005; 3-CN-5-F-4-Py], [BE4006; 2-CN-5-F-4-Py], [BE4007; 6-CN-5-F-4-Py], [BE4005; BE 4008; 3-OMe-5-F-4-Py], [BE 4009; 2-OMe-5-F-4-Py], [BE 4010; 6-OMe-5-F-4-Py], [BE 4011; 6-F-4-Py], [BE4012; 3-Cl-6-F-4-Py], [BE4013; 2-Cl-6-F-4-Py], [BE4014; 5-Cl-6- 6 F-4-Py !, [BE4015; 3-Me-6-F-4-Py], [BE4016; 2-Me-6-F-4-Py], [BE4017; 5-Me-6-F- 4-Py], [BE4018; 3-CF 3 -6-F-4-Py], [BE4019; 2-CF 3 -6-F-4-Py], [BE4020; 5-CF 3 -6-F -4-Py], [BE4021; 3-CN-6-F-4-Py], [BE4022; 2-CN-6-F-4-Py], [BE4023; 5-CN-6-F-4 -Py], [BE4024; 3-OMe-6-F-4-Py], [BE4025; 2-OMe-6-F-4-Py], [BE4026; 5-OMe-6-F-4-Py ], [BE 4027; 3-Cl-4-Py], [BE 4028; 2-Cl-3-Cl-4-Py], [BE 4029; 5-Cl-3-Cl-4-Py], [BE 4030; 6] -Cl-3-Cl-4-Py], [BE4031; 2-Me-3-Cl-4-Py], [BE4032; 5-Me-3-Cl-4-Py], [BE4033; 6-Me -3-Cl-4-Py !, [BE 4034; 2-CF ₃ -3-Cl-4-Py], [BE 4035; 5-CF ₃ -3-Cl-4-Py], [BE 4036; 6-CF _3- -3-Cl-4-Py], [BE4037; 2-CN-3-Cl-4-Py], [BE4038; 5-CN-3-Cl-4-Py], [BE4039; 6-CN- 3-Cl-4-Py], [BE 4040; 2-OMe-3-Cl-4-Py], [BE 4041; 5-OMe-3-Cl-4-Py], [BE 4042; 6-OMe-3- Cl-4-Py], [BE 4043; 2-Cl-4- Py], [BE4044; 3-Cl-2-Cl-4-Py], [BE 4045; 5-Cl-2-Cl-4-Py], [BE 4046; 6-Cl-2-Cl-4-Py] , [BE4047; 3-Me-2-Cl-4-Py], [BE4048; 5-Me-2-Cl-4-Py], [BE4049; 6-Me-2-Cl-4-Py], [BE40 49; _{BE4050; 3-CF 3 -2-} Cl-4-Py], [BE4051; 5-CF 3 -2-Cl-4-Py], [BE4052; 6-CF 3 -2-Cl-4-Py], [BE4053; 3-CN-2-Cl-4-Py], [BE4054; 5-CN-2-Cl-4-Py], [BE4055; 6-CN-2-Cl-4-Py], [BE 4056] 3-OMe-2-Cl-4-Py !, [BE4057; 5-OMe-2-Cl-4-Py], [BE4058; 6-OMe-2-Cl-4-Py], [BE4059; -Cl-4-Py], [BE 4060; 2-Cl-5-Cl-4-Py], [BE 4061; 5-Cl-5-Cl-4-Py], [BE 4062; 6-Cl-5-Cl -4-Py], [BE4063; 2-Me-5-Cl-4-Py], [BE 4064; 5-Me-5-Cl-4-Py], [BE 4065; 6-Me-5-Cl-4 -Py], [BE4066; 2- CF 3 -5-Cl-4-Py], [BE4067; 5-CF 3 -5-Cl-4-Py], [BE4068; 6-CF 3 -5-Cl- 4-Py], [BE4069; 2-CN-5-Cl-4-Py], [BE4070; 3-CN-5-Cl-4-Py], [BE4071; 6-CN-5-Cl-4- Py], [BE4072; 2-OMe-5-Cl-4-Py], [BE4073; 5-OMe-5-Cl-4-Py], [BE4074; 6-OMe-5-Cl-4-Py] [BE 4075; 6-Cl-4-Py], [BE 4076; 3-Cl-6-Cl-4-Py], [BE 4077; 2-Cl-6-Cl-4-Py], [BE 4078; Cl-6-Cl-4-Py], [BE4079; 3-Me-6-Cl-4-Py], [BE4080; 2-Me-6-Cl-4-Py], [BE4081; 5-Me- 6-Cl-4-Py] , [BE4082; 3-CF 3 -6-Cl-4-Py], [BE4083; 2-CF 3 -6-Cl-4-Py], [BE4084; 5-CF 3 - 6-Cl-4-Py, [BE 4085; 3-CN-6-Cl-4-Py], [BE 4086; 2-CN-6-Cl-4-Py], [BE 4087; 5-CN-6- Cl-4-Py], [BE4088; 3-OMe-6-Cl-4-Py], [BE4089; 2-OMe-6-Cl-4-Py], [BE4090; 5-OMe-6-Cl- 4-Py], [BE4091; 3-Br-4-Py], [BE4092; 2-Cl-3-Br-4-Py], [BE4093; 5-Cl-3-Br-4-Py], BE 4094; 6-Cl-3-Br-4-Py], [BE 4095; 2-Me-3-Br-4-Py], [BE 4096; 5-Me-3-Br-4-Py], [BE 4097; 6-Me-3-Br- 4-Py], [BE4098; 2-CF 3 -3-Br-4-Py], [BE4099; 5-CF 3 -3-Br-4-Py], [BE4100; _{6-CF 3 -3-Br-} 4-Py], [BE4101; 2-CN-3-Br-4-Py],

[BE4102; 5-CN-3-Br-4-Py], [BE4103; 6-CN-3-Br-4-Py], [BE4104; 2-OMe-3-Br-4-Py], [BE4105] 5-OMe-3-Br-4-Py !, [BE4106; 6-OMe-3-Br-4-Py], [BE4107; 2-Br-4-Py], [BE4108; 3-Cl-2 -Br-4-Py], [BE4109; 5-Cl-2-Br-4-Py], [BE4110; 6-Cl-2-Br-4-Py], [BE4111; 3-Me-2-Br -4-Py], [BE4112; 5-Me-2-Br-4-Py], [BE4113; 6-Me-2-Br-4-Py], [BE4114; 3-CF 3 -2-Br- 4-Py], [BE4115; 5-CF 3 -2-Br-4-Py], [BE4116; 6-CF 3 -2-Br-4-Py], [BE4117; 3-CN-2-Br- 4-Py], [BE4118; 5-CN-2-Br-4-Py], [BE4119; 6-CN-2-Br-4-Py], [BE4120; 3-OMe-2-Br-4- Py], [BE 4121; 5-OMe-2-Br-4-Py], [BE 4122; 6-OMe-2-Br-4-Py], [BE 4123; 5-Br-4-Py], [BE 4124; 3-Cl-5-Br-4-Py], [BE 4125; 2-Cl-5-Br-4-Py], [BE 4126; 6-Cl-5-Br-4-Py], [BE 4127; Me-5-Br-4- Py], [BE4128; 2-Me-5-Br-4-Py], [BE4129; 6-Me-5-Br-4-Py], [BE4130; 3-CF 3 -5-Br-4-Py], [BE 4131; 2-CF ₃ -5-Br-4-Py], [BE 4132; 6-CF ₃ -5-Br-4-Py], [BE 4133; 3-CN -5-Br-4-Py], [BE4134; 2-CN-5-Br-4-Py], [BE4135; 6-CN-5-Br-4-Py], [BE4136; 3-OMe-5 -Br-4-Py], [BE4137; 2-OMe-5-Br-4-Py], [BE4138; 6-OMe-5-Br-4-Py], [BE4139; 6-Br-4-Py ], [BE4140; 3-Cl-6-Br-4-Py], [BE4141; 2-Cl-6-Br-4-Py], [BE4142; 5-Cl-6-Br-4-Py], [BE4 143; 3-Me-6-Br-4-Py], [BE4144; 2-Me-6-Br-4-Py], [BE4145; 5-Me-6-Br-4-Py], [BE4146; _{3-CF 3 -6-Br-} 4-Py], [BE4147; 2-CF 3 -6-Br-4-Py], [BE4148; 5-CF 3 -6-Br-4-Py], [BE4149 3-CN-6-Br-4-Py !, [BE4150; 2-CN-6-Br-4-Py], [BE4151; 5-CN-6-Br-4-Py], [BE4152; -OMe-6-Br-4-Py], [BE 4153; 2-OMe-6-Br-4-Py], [BE 4154; 5-OMe-6-Br-4-Py], [BE 4155; 3-I -4-Py], [BE4156; 2-Cl-3-I-4-Py], [BE4157; 5-Cl-3-I-4-Py], [BE4158; 6-Cl-3-I-4 -Py], [BE 4159; 2-Me-3-I-4-Py], [BE 4160; 5-Me-3-I-4-Py], [BE 4161; 6-Me-3-I-4-Py ], [BE4162; 2-CF 3 -3-I-4-Py], [BE4163; 5-CF 3 -3-I-4-Py], [BE4164; 6-CF 3 -3-I-4- Py], [BE 4165; 2-CN-3-I-4-Py], [BE 4166; 5-CN-3-I-4-Py], [BE 4167; 6-CN-3-I-4-Py] , [BE4168; 2-OMe-3-I-4-Py], [BE4169; 5-OMe-3-I-4-Py], [BE4170; 6-OMe-3-I-4-Py], [BE4 168; BE 4171; 2-I-4-Py], [BE 4172; 3-Cl-2-I-4-Py], [BE 4173; 5-Cl-2-I-4-Py], [BE 4174; 6-Cl- 2-I-4-Py, [BE4175; 3-Me-2-I-4-Py], [BE4176; 5-Me-2-I-4-Py], [BE4177; 6-Me-2- I-4-Py], [ BE4178; 3-CF 3 -2-I-4-Py], [BE4179; 5-CF 3 -2-I-4-Py], [BE4180; 6-CF 3 -2 -I-4-Py], [BE4181; 3-CN-2-I-4-Py], [BE4182; 5-CN-2-I-4-Py], [BE4183; 6-CN-2-I -4-Py], [BE 4184; 3-OMe-2-I-4-Py], [B E4185; 5-OMe-2-I-4-Py, [BE4186; 6-OMe-2-I-4-Py], [BE4187; 5-I-4-Py], [BE4188; 3-Cl- 5-I-4-Py], [BE 4189; 2-Cl-5-I-4-Py], [BE 4190; 6-Cl-5-I-4-Py], [BE 4191; 3-Me-5-5 I-4-Py], [ BE4192; 2-Me-5-I-4-Py], [BE4193; 6-Me-5-I-4-Py], [BE4194; 3-CF 3 -5-I -4-Py], [BE4195; 2-CF 3 -5-I-4-Py], [BE4196; 6-CF 3 -5-I-4-Py], [BE4197; 3-CN-5-I -4-Py], [BE 4198; 2-CN-5-I-4-Py], [BE 4199; 6-CN-5-I-4-Py], [BE 4200; 3-OMe-5-I-4 -Py], [BE 4201; 2-OMe-5-I-4-Py],

[BE4202; 6-OMe-5-I-4-Py], [BE 4203; 6-I-4-Py], [BE 4204; 3-Cl-6-I-4-Py], [BE 4205; 2-Cl -6-I-4-Py], [BE4206; 5-Cl-6-I-4-Py], [BE4207; 3-Me-6-I-4-Py], [BE4208; 2-Me-6 -I-4-Py], [ BE4209; 5-Me-6-I-4-Py], [BE4210; 3-CF 3 -6-I-4-Py], [BE4211; 2-CF 3 -6 -I-4-Py], [ BE4212; 5-CF 3 -6-I-4-Py], [BE4213; 3-CN-6-I-4-Py], [BE4214; 2-CN-6- I-4-Py], [BE4215; 5-CN-6-I-4-Py], [BE4216; 3-OMe-6-I-4-Py], [BE4217; 2-OMe-6-I- 4-Py], [BE4218; 5-OMe-6-I-4-Py], [BE4219; 3-Me-4-Py], [BE4220; 2-Cl-3-Me-4-Py], BE4221; 5-Cl-3-Me-4-Py], [BE4222; 6-Cl-3-Me-4-Py], [BE4223; 2-Me-3-Me-4-Py], [BE4224; 5-Me-3-Me- 4-Py], [BE4225; 6-Me-3-Me-4-Py], [BE4226; 2-CF 3 -3-Me-4-Py], [BE4227; 5 _{-CF 3 -3-Me-4-} Py], [BE4228; 6-CF 3 -3-Me-4-Py], [BE4229; 2-CN-3-Me-4-Py], [BE4230; 5 -CN-3-Me-4-Py], [BE4231; 6-CN-3-Me-4-Py], [BE4232; 2-OMe-3-Me-4-Py], [BE4233; 5-OMe -3-Me-4-Py !, [BE4234; 6-OMe-3-Me-4-Py], [BE4235; 2-Me-4-Py], [BE4236; 3-Cl-2-Me-4 -Py], [BE4237; 5-Cl-2-Me-4-Py], [BE4238; 6-Cl-2-Me-4-Py], [BE4239; 3-Me-2-Me-4-Py ], [BE4240; 5-Me -2-Me-4-Py], [BE4241; 6-Me-2-Me-4-Py], [BE4242; 3-CF 3 -2-Me-4-Py] , [BE 4243; 5-CF ₃ -2-Me -4-Py], [BE4244; 6-CF 3 -2-Me-4-Py], [BE4245; 3-CN-2-Me-4-Py], [BE4246; 5-CN-2-Me- 4-Py], [BE4247; 6-CN-2-Me-4-Py], [BE4248; 3-OMe-2-Me-4-Py], [BE4249; 5-OMe-2-Me-4- 4 Py], [BE 4250; 6-OMe-2-Me-4-Py], [BE 4251; 5-Me-4-Py], [BE 4252; 3-Cl-5-Me-4-Py], [BE 4253; 2-Cl-5-Me-4-Py], [BE4254; 6-Cl-5-Me-4-Py], [BE4255; 3-Me-5-Me-4-Py], [BE4256; 2- Me-5-Me-4- Py], [BE4257; 6-Me-5-Me-4-Py], [BE4258; 3-CF 3 -5-Me-4-Py], [BE4259; 2-CF _{3 -5-Me-4-Py} ], [BE4260; 6-CF 3 -5-Me-4-Py], [BE4261; 3-CN-5-Me-4-Py], [BE4262; 2-CN -5-Me-4-Py !, [BE4263; 6-CN-5-Me-4-Py], [BE4264; 3-OMe-5-Me-4-Py], [BE4265; 2-OMe-5 -Me-4-Py], [BE4266; 6-OMe-5-Me-4-Py], [BE4267; 6-Me-4-Py], [BE4268; 3-Cl-6-Me-4-Py ], [BE 4269; 2-Cl-6-Me-4-Py], [BE 4270; 5-Cl-6-Me-4-Py], [BE 427 1; 3-Me-6-Me-4-Py], [BE4272; 2-Me-6 -Me-4-Py], [BE4273; 5-Me-6-Me-4-Py], [BE4274; 3-CF 3 -6-Me-4-Py], [ _{BE4275; 2-CF 3 -6-} Me-4-Py], [BE4276; 5-CF 3 -6-Me-4-Py], [BE4277; 3-CN-6-Me-4-Py], [ BE4278; 2-CN-6-Me-4-Py], [BE4279; 5-CN-6-Me-4-Py], [BE4280; 3-OMe-6-Me-4-Py], [BE4281; 2-OMe-6-Me-4-Py], [BE4282; 5-OMe-6-Me-4-Py], [BE4283; 3-OMe-4-Py], [BE4284; 2-Cl-3- OM e-4-Py], [BE4285; 5-Cl-3-OMe-4-Py], [BE4286; 6-Cl-3-OMe-4-Py], [BE4287; 2-Me-3-OMe- 4-Py], [BE4288; 5-Me-3-OMe-4-Py], [BE4289; 6-Me-3-OMe-4-Py], [BE4290; 2-CF 3 -3-OMe-4 -Py], [BE4291; 5- CF 3 -3-OMe-4-Py], [BE4292; 6-CF 3 -3-OMe-4-Py], [BE4293; 2-CN-3-OMe-4 -Py], [BE4294; 5-CN-3-OMe-4-Py], [BE4295; 6-CN-3-OMe-4-Py], [BE4296; 2-OMe-3-OMe-4-Py ], [BE4297; 5-OMe-3-OMe-4-Py], [BE4298; 6-OMe-3-OMe-4-Py], [BE4299; 2-OMe-4-Py], [BE4300; 3] -Cl-2-OMe-4-Py], [BE 4301; 5-Cl-2-OMe-4-Py],

[BE4302; 6-Cl-2-OMe-4-Py], [BE4303; 3-Me-2-OMe-4-Py], [BE 4304; 5-Me-2-OMe-4-Py], [BE 4305] ; 6-Me-2-OMe -4-Py], [BE4306; 3-CF 3 -2-OMe-4-Py], [BE4307; 5-CF 3 -2-OMe-4-Py], [BE4308 _{; 6-CF 3 -2-OMe} -4-Py], [BE4309; 3-CN-2-OMe-4-Py], [BE4310; 5-CN-2-OMe-4-Py], [BE4311; 6-CN-2-OMe-4-Py !, [BE4312; 3-OMe-2-OMe-4-Py], [BE4313; 5-OMe-2-OMe-4-Py], [BE4314; 6- OMe-2-OMe-4-Py], [BE4315; 5-OMe-4-Py], [BE4316; 3-Cl-5-OMe-4-Py], [BE4317; 2-Cl-5-OMe- 4-Py], [BE4318; 6-Cl-5-OMe-4-Py], [BE4319; 3-Me-5-OMe-4-Py], [BE4320; 2-Me-5-OMe-4- Py], [BE4321; 6- Me-5-OMe-4-Py], [BE4322; 3-CF 3 -5-OMe-4-Py], [BE4323; 2-CF 3 -5-OMe-4- Py], [BE4324; 6- CF 3 -5-OMe-4-Py], [BE4325; 3-CN-5-OMe-4-Py], [BE4326; 2-CN-5-OMe-4-Py ], [BE4327; 6-CN-5-OMe-4-Py], [BE4328; 3-OMe-5-OMe-4-Py], [BE4329; 2-OMe-5-OMe-4-Py], [BE4330; 6-OMe-5-OMe-4-Py], [BE4331; 6-OMe-4-Py], [BE4332; 3-Cl-6-OMe-4-Py], [BE4333; 2-Cl -6-OMe-4-Py], [BE4334; 5-Cl-6-OMe-4-Py], [BE4335; 3-Me-6-OMe-4-Py], [BE4336; 2-Me-6 -OMe-4-Py], [ BE4337; 5-Me-6-OMe-4-Py], [BE4338; 3-CF 3 -6-OMe-4-Py], [BE4339; 2-CF 3 -6 -OMe-4-Py], [BE 4340; 5-CF ₃ -6-OMe-4-Py], [B E4341; 3-CN-6-OMe-4-Py], [BE4342; 2-CN-6-OMe-4-Py], [BE4343; 5-CN-6-OMe-4-Py], [BE4344; 3-OMe-6-OMe-4-Py], [BE4345; 2-OMe-6-OMe-4-Py], [BE4346; 5-OMe-6-OMe-4-Py], [BE4347; _{CF 3 -4-Py], [} BE4348; 2-Cl-3-CF 3 -4-Py], [BE4349; 5-Cl-3-CF 3 -4-Py], [BE4350; 6-Cl-3 _{-CF 3 -4-Py], [} BE4351; 2-Me-3-CF 3 -4-Py], [BE4352; 5-Me-3-CF 3 -4-Py], [BE4353; 6-Me- _{3-CF 3 -4-Py]} , [BE4354; 2-CF 3 -3-CF 3 -4-Py], [BE4355; 5-CF 3 -3-CF 3 -4-Py], [BE4356; 6 _{-CF 3 -3-CF 3 -4-} Py], [BE4357; 2-CN-3-CF 3 -4-Py], [BE4358; 5-CN-3-CF 3 -4-Py], [BE4359 ; 6-CN-3-CF 3 -4-Py], [BE4360; 2-OMe-3-CF 3 -4-Py], [BE4361; 5-OMe-3-CF 3 -4-Py], [ BE4362; 6-OMe-3- CF 3 -4-Py], [BE4363; 2-CF 3 -4-Py], [BE4364; 3-Cl-2-CF 3 -4-Py], [BE4365; 5 _{-Cl-2-CF 3 -4-} Py], [BE4366; 6-Cl-2-CF 3 -4-Py], [BE4367; 3-Me-2-CF 3 -4-Py], [BE4368; _{5-Me-2-CF 3} -4-Py], [BE4369; 6-Me-2-CF 3 -4-Py], [BE4370; 3-CF 3 -2-CF 3 -4-Py], [ _{BE4371; 5-CF 3 -2-} CF 3 -4-Py], [BE4372; 6-CF 3 -2-CF 3 -4-Py], [BE4373; 3-CN-2-CF 3 -4-Py ], [BE4374; 5-CN -2-CF 3 -4-Py], [BE4375; 6-CN-2-CF 3 -4-Py], [BE4376; 3-OMe-2-CF 3 -4- Py], [BE 4377; 5-OMe-2-CF ₃ -4-Py] , [BE 4378; 6-OMe-2-CF ₃ -4-Py], [BE 4379; 5-CF ₃ -4-Py], [BE 4 380; 3-Cl -5-CF ₃ -4-Py], [BE 4 8 1 ; 2-Cl-5-CF 3 -4-Py], [BE4382; 6-Cl-5-CF 3 -4-Py], [BE4383; 3-Me-5-CF 3 -4-Py], [ BE 4384; 2-Me-5-CF ₃ -4-Py], [BE 4385; 6-Me-5-CF ₃ -4-Py], [BE 4386; 3-CF ₃ -5-CF ₃ -4-Py] _{, [BE4387; 2-CF 3} -5-CF 3 -4-Py], [BE4388; 6-CF 3 -5-CF 3 -4-Py], [BE4389; 3-CN-5-CF 3 -4 -Py], [BE4390; 2- CN-5-CF 3 -4-Py], [BE4391; 6-CN-5-CF 3 -4-Py], [BE4392; 3-OMe-5-CF 3 - 4-Py], [BE 4393; 2-OMe-5-CF ₃ -4-Py], [BE 4394; 6-OMe-5-CF ₃ -4-Py], [BE 4395; 6-CF ₃ -4-Py ], [BE4396; 3-Cl -6-CF 3 -4-Py], [BE4397; 2-Cl-6-CF 3 -4-Py], [BE4398; 5-Cl-6-CF 3 -4- Py], [BE4399; 3- Me-6-CF 3 -4-Py], [BE4400; 2-Me-6-CF 3 -4-Py], [BE4401; 5-Me-6-CF 3 -4 -Py],

_{[BE4402; 3-CF 3 -6} -CF 3 -4-Py], [BE4403; 2-CF 3 -6-CF 3 -4-Py], [BE4404; 5-CF 3 -6-CF 3 -4 -Py], [BE 4405; 3-CN-6-CF ₃ -4-Py], [BE 4406; 2-CN-6-CF ₃ -4-Py], [BE 4407; 5-CN-6-CF _3- 4-Py], [BE4408; 3-OMe-6-CF 3 -4-Py], [BE4409; 2-OMe-6-CF 3 -4-Py], [BE4410; 5-OMe-6-CF 3 -4-Py], [BE 4411; 3-OCF ₃ -4-Py], [BE 4412; 2-Cl-3-OCF ₃ -4-Py], [BE 4413; 5-Cl-3-OCF ₃ -4-] Py], [BE4414; 6- Cl-3-OCF 3 -4-Py], [BE4415; 2-Me-3-OCF 3 -4-Py], [BE4416; 5-Me-3-OCF 3 -4 -Py], [BE4417; 6- Me-3-OCF 3 -4-Py], [BE4418; 2-CF 3 -3-OCF 3 -4-Py], [BE4419; 5-CF 3 -3-OCF _{3 -4-Py], [BE4420} ; 6-CF 3 -3-OCF 3 -4-Py], [BE4421; 2-CN-3-OCF 3 -4-Py], [BE4422; 5-CN-3 _{-OCF 3 -4-Py], [} BE4423; 6-CN-3-OCF 3 -4-Py], [BE4424; 2-OMe-3-OCF 3 -4-Py], [BE4425; 5-OMe- _{3-OCF 3 -4-Py]} , [BE4426; 6-OMe-3-OCF 3 -4-Py], [BE4427; 2-OCF 3 -4-Py], [BE4428; 3-Cl-2-OCF ₃ -4-Py], [BE 4429; 5-Cl-2-OCF ₃ -4-Py], [BE 4430; 6-Cl 2-OCF ₃ -4-Py], [BE 4 43 1; _{OCF 3 -4-Py], [} BE4432; 5-Me-2-OCF 3 -4-Py], [BE4433; 6-Me-2-OCF 3 -4-Py], [BE4434; 3-CF 3 - _{2-OCF 3 -4-Py]} , [BE4435; 5-CF 3 -2-OCF 3 -4-Py], [BE4436; 6-CF 3 -2-OCF 3 -4-Py], [BE443 7; 3-CN-2- OCF 3 -4-Py], [BE4438; 5-CN-2-OCF 3 -4-Py], [BE4439; 6-CN-2-OCF 3 -4-Py], [BE4440; 3-OMe-2 -OCF 3 -4-Py], [BE4441; 5-OMe-2-OCF 3 -4-Py], [BE4442; 6-OMe-2-OCF 3 -4-Py] _{, [BE4443; 5-OCF 3} -4-Py], [BE4444; 3-Cl-5-OCF 3 -4-Py], [BE4445; 2-Cl-5-OCF 3 -4-Py], [BE4446 ; 6-Cl-5-OCF 3 -4-Py], [BE4447; 3-Me-5-OCF 3 -4-Py], [BE4448; 2-Me-5-OCF 3 -4-Py], [ BE4449; 6-Me-5- OCF 3 -4-Py], [BE4450; 3-CF 3 -5-OCF 3 -4-Py], [BE4451; 2-CF 3 -5-OCF 3 -4-Py ], [BE4452; 6-CF 3 -5-OCF 3 -4-Py], [BE4453; 3-CN-5-OCF 3 -4-Py], [BE4454; 2-CN-5-OCF 3 -4 -Py], [BE4455; 6- CN-5-OCF 3 -4-Py], [BE4456; 3-OMe-5-OCF 3 -4-Py], [BE4457; 2-OMe-5-OCF 3 - 4-Py], [BE 4458; 6-OMe-5-OCF ₃ -4-Py], [BE 4459; 6-OCF ₃ -4-Py], [BE 4460; 3-Cl -6-OCF ₃ -4-Py ], [BE4461; 2-Cl -6-OCF 3 -4-Py], [BE4462; 5-Cl-6-OCF 3 -4-Py], [BE4463; 3-Me-6-OCF 3 -4- Py], [BE 4464; 2-Me-6-OCF ₃ -4-Py], [BE 4465; 5-Me-6-OCF ₃ -4-Py], [BE 4466; 3-CF ₃ -6-OCF _3- 4-Py], [BE 4467; 2-CF ₃ -6-OCF ₃ -4-Py], [BE 4468; 5-CF ₃ -6-OCF ₃ -4-Py], [BE 4469; _{OCF 3 -4-Py], [} BE4470; 2-CN-6-OCF 3 -4-Py], [BE4471; 5-CN-6-OCF 3 -4-Py], [BE4472; 3-OM _{e-6-OCF 3 -4-} Py], [BE4473; 2-OMe-6-OCF 3 -4-Py], [BE4474; 5-OMe-6-OCF 3 -4-Py], [BE4475; 3 _{-CHF 2 -4-Py], [} BE4476; 2-Cl-3-CHF 2 -4-Py], [BE4477; 5-Cl-3-CHF 2 -4-Py], [BE4478; 6-Cl- _{3-CHF 2 -4-Py]} , [BE4479; 2-Me-3-CHF 2 -4-Py], [BE4480; 5-Me-3-CHF 2 -4-Py], [BE4481; 6-Me -3-CHF ₂ -4-Py !, [BE 4482; 2-CF ₃ -3-CHF ₂ -4-Py], [BE 4483; 5-CF ₃ -3-CHF ₂ -4-Py], [BE 4484; _{6-CF 3 -3-CHF 2} -4-Py], [BE4485; 2-CN-3-CHF 2 -4-Py], [BE4486; 5-CN-3-CHF 2 -4-Py], [ BE4487; 6-CN-3- CHF 2 -4-Py], [BE4488; 2-OMe-3-CHF 2 -4-Py], [BE4489; 5-OMe-3-CHF 2 -4-Py], [BE4490; 6-OMe-3 -CHF 2 -4-Py], [BE4491; 4-CHF 2 -4-Py], [BE4492; 3-Cl-4-CHF 2 -4-Py], [BE4493; _{5-Cl-4-CHF 2} -4-Py], [BE4494; 6-Cl-4-CHF 2 -4-Py], [BE4495; 3-Me-4-CHF 2 -4-Py], [BE4496 ; 5-Me-4-CHF 2 -4-Py], [BE4497; 6-Me-4-CHF 2 -4-Py], [BE4498; 3-CF 3 -4-CHF 2 -4-Py], _{[BE4499; 5-CF 3 -4} -CHF 2 -4-Py], [BE4500; 6-CF 3 -4-CHF 2 -4-Py], [BE4501; 3-CN-4-CHF 2 -4- Py],

[BE4502; 5-CN-4 -CHF 2 -4-Py], [BE4503; 6-CN-4-CHF 2 -4-Py], [BE4504; 3-OMe-4-CHF 2 -4-Py] , [BE4505; 5-OMe- 4-CHF 2 -4-Py], [BE4506; 6-OMe-4-CHF 2 -4-Py], [BE4507; 5-CHF 2 -4-Py], [BE4508 ; 3-Cl-5-CHF 2 -4-Py], [BE4509; 2-Cl-5-CHF 2 -4-Py], [BE4510; 6-Cl-5-CHF 2 -4-Py], [ BE 4511; 3-Me-5-CHF ₂ -4-Py], [BE 4512; 2-Me-5-CHF ₂ -4-Py], [BE 4513; 6-Me-5-CHF ₂ -4-Py], [BE 4514; 3-CF ₃ -5-CHF ₂ -4-Py], [BE 4515; 2-CF ₃ -5-CHF ₂ -4-Py], [BE 4516; 6-CF ₃ -5-CHF _2-4 -Py], [BE4517; 3- CN-5-CHF 2 -4-Py], [BE4518; 2-CN-5-CHF 2 -4-Py], [BE4519; 6-CN-5-CHF 2 - 4-Py], [BE 4520; 3-OMe-5-CHF ₂ -4-Py], [BE 4521; 2-OMe-5-CHF ₂ -4-Py], [BE 4522; 6-OMe -5-CHF ₂ -4-Py], [BE 4523; 6-CHF ₂ -4-Py], [BE 4524; 3-Cl-6-CHF ₂ -4-Py], [BE 4525; 2-Cl-6-CHF ₂ -4- Py], [BE4526; 5- Cl-6-CHF 2 -4-Py], [BE4527; 3-Me-6-CHF 2 -4-Py], [BE4528; 2-Me-6-CHF 2 -4 -Py], [BE 4529; 5-Me-6-CHF ₂ -4-Py], [BE 4530; 3-CF ₃ -6-CHF ₂ -4-Py], [BE 451; 2-CF ₃ -6-CHF ₂ -4-Py !, [BE 4532; 5-CF ₃ -6-CHF ₂ -4-Py], [BE 4533; 3-CN-6-CHF ₂ -4-Py], [BE 4534; 2-CN-6 _{-CHF 2 -4-Py], [} BE4535; 5-CN-6-CHF 2 -4-Py], [BE4536; 3-OMe-6-CHF 2 -4-Py], [BE45 37; 2-OMe-6- CHF 2 -4-Py], [BE4538; 5-OMe-6-CHF 2 -4-Py], [BE4539; 3-OCHF 2 -4-Py], [BE4540; 2 _{-Cl-3-OCHF 2 -4-} Py], [BE4541; 5-Cl-3-OCHF 2 -4-Py], [BE4542; 6-Cl-3-OCHF 2 -4-Py], [BE4543; _{2-Me-3-OCHF 2} -4-Py], [BE4544; 5-Me-3-OCHF 2 -4-Py], [BE4545; 6-Me-3-OCHF 2 -4-Py], [BE4546 _{; 2-CF 3 -3-OCHF} 2 -4-Py], [BE4547; 5-CF 3 -3-OCHF 2 -4-Py], [BE4548; 6-CF 3 -3-OCHF 2 -4-Py ], [BE 4549; 2-CN-3-OCHF ₂ -4-Py], [BE 4550; 5-CN-3-OCHF ₂ -4-Py], [BE 4551; 6-CN -3-OCHF ₂ -4-] Py], [BE4552; 2- OMe-3-OCHF 2 -4-Py], [BE4553; 5-OMe-3-OCHF 2 -4-Py], [BE4554; 6-OMe-3-OCHF 2 -4 -Py], [BE4555; 4- OCHF 2 -4-Py], [BE4556; 3-Cl-4-OCHF 2 -4-Py], [BE4557; 5-Cl-4-OCHF 2 -4-Py] , [BE4558; 6-Cl- 4-OCHF 2 -4-Py], [BE4559; 3-Me-4-OCHF 2 -4-Py], [BE4560; 5-Me-4-OCHF 2 -4-Py ], [BE4561; 6-Me -4-OCHF 2 -4-Py], [BE4562; 3-CF 3 -4-OCHF 2 -4-Py], [BE4563; 5-CF 3 -4-OCHF 2 - 4-Py], [BE 4564; 6-CF ₃ -4-OCHF ₂ -4-Py], [BE 4 565; 3-CN 4-OCHF ₂ -4-Py], [BE 4 566; ₂ -4-Py !, [BE 4567; 6-CN -4-OCHF ₂ -4-Py], [BE 4568; 3-OMe -4-OCHF ₂ -4-Py], [BE 4569; OCHF ₂ -4-Py], [BE 4570; 6-OMe -4-OCHF ₂ -4-Py], [BE 45] _{71; 5-OCHF 2 -4-} Py], [BE4572; 3-Cl-5-OCHF 2 -4-Py], [BE4573; 2-Cl-5-OCHF 2 -4-Py], [BE4574; 6 _{-Cl-5-OCHF 2 -4-} Py], [BE4575; 3-Me-5-OCHF 2 -4-Py], [BE4576; 2-Me-5-OCHF 2 -4-Py], [BE4577; 6-Me-5-OCHF ₂ -4-Py], [BE 4578; 3-CF ₃ -5-OCHF ₂ -4-Py], [BE 4579; 2-CF ₃ -5-OCHF ₂ -4-Py], _{[BE4580; 6-CF 3 -5} -OCHF 2 -4-Py], [BE4581; 3-CN-5-OCHF 2 -4-Py], [BE4582; 2-CN-5-OCHF 2 -4-Py ], [BE 4583; 6-CN-5-OCHF ₂ -4-Py], [BE 4584; 3-OMe-5-OCHF ₂ -4-Py], [BE 4585; 2-OMe -5-OCHF ₂ -4-] Py], [BE 4586; 6-OMe-5-OCHF ₂ -4-Py], [BE 4587; 6-OCHF ₂ -4-Py], [BE 4588; 3-Cl -6-OCHF ₂ -4-Py], [BE4589; 2-Cl-6 -OCHF 2 -4-Py], [BE4590; 5-Cl-6-OCHF 2 -4-Py], [BE4591; 3-Me-6-OCHF 2 -4-Py] , [BE4592; 2-Me-6-OCHF ₂ -4-Py], [BE 4593; 5-Me-6-OCHF ₂ -4-Py], [BE 4594; 3-CF ₃ -6-OCHF ₂ -4-] Py], [BE4595; 2- CF 3 -6-OCHF 2 -4-Py], [BE4596; 5-CF 3 -6-OCHF 2 -4-Py], [BE4597; 3-CN-6-OCHF 2 -4-Py], [BE 4598; 2-CN-6-OCHF ₂ -4-Py], [BE 4599; 5-CN-6-OCHF ₂ -4-Py], [BE 4600; 3-OMe -6-OCHF ₂ -4-Py], [BE 4601; 2-OMe-6-OCHF ₂ -4-Py],

[BE4602; 5-OMe-6 -OCHF 2 -4-Py], [BE4603; 3-Et-4-Py], [BE4604; 2-Cl-3-Et-4-Py], [BE4605; 5- Cl-3-Et-4-Py], [BE4606; 6-Cl-3-Et-4-Py], [BE4607; 2-Me-3-Et-4-Py], [BE4608; 5-Me- 3-Et-4-Py] , [BE4609; 6-Me-3-Et-4-Py], [BE4610; 2-CF 3 -3-Et-4-Py], [BE4611; 5-CF 3 - 3-Et-4-Py] , [BE4612; 6-CF 3 -3-Et-4-Py], [BE4613; 2-CN-3-Et-4-Py], [BE4614; 5-CN-3 -Et-4-Py], [BE4615; 6-CN-3-Et-4-Py], [BE4616; 2-OMe-3-Et-4-Py], [BE4617; 5-OMe-3-Et -4-Py], [BE4618; 6-OMe-3-Et-4-Py], [BE4619; 2-Et-4-Py], [BE4620; 3-Cl-2-Et-4-Py], [BE 4621; 5-Cl-2-Et-4-Py], [BE 4622; 6-Cl-2-Et-4-Py], [BE 4623; 3-Me-2-Et-4-Py], [BE 4624 ; 5-Me-2-Et -4-Py], [BE4625; 6-Me-2-Et-4-Py], [BE4626; 3-CF 3 -2-Et-4-Py], [BE4627; _{5-CF 3 -2-Et-} 4-Py], [BE4628; 6-CF 3 -2-Et-4-Py], [BE4629; 3-CN-2-Et-4-Py], [BE4630; 5-CN-2-Et-4-Py], [BE4631; 6-CN-2-Et-4-Py], [BE4632; 3-OMe-2-Et-4-Py], [BE4633; 5- OMe-2-Et-4-Py], [BE4634; 6-OMe-2-Et-4-Py], [BE4635; 5-Et-4-Py], [BE4636; 3-Cl-5-Et- 4-Py], [BE4637; 2-Cl-5-Et-4-Py], [BE4638; 6-Cl-5-Et-4-Py], [BE4639; 3-Me-5-Et-4- Py], [BE4640; 2- Me-5-Et-4-Py], [BE4641; 6-Me-5-Et-4-Py], [BE4642; 3-CF 3 -5-Et-4-Py ], [BE4643; 2-CF 3 -5-Et-4-Py], [BE4644; 6-CF 3 -5-Et-4-Py], [BE4645; 3-CN-5-Et-4-Py ], [BE 4646; 2-CN-5-Et-4-Py], [BE 4647; 6-CN-5-Et-4-Py], [BE 4648; 3-OMe-5-Et-4-Py], [BE 4649; 2-OMe-5-Et-4-Py], [BE 4650; 6-OMe-5-Et-4-Py], [BE 4651; 6-Et-4-Py], [BE 4652; 3-Cl -6-Et-4-Py], [BE 4653; 2-Cl-6-Et-4-Py], [BE 4564; 5-Cl-6-Et-4-Py], [BE 4655; 3-Me-6 -Et-4-Py], [BE 4656; 2-Me-6-Et-4-Py], [BE 4657; 5-Me-6-Et-4-Py], [BE 4658; 3-CF ₃ -6- Et-4-Py], [ BE4659; 2-CF 3 -6-Et-4-Py], [BE4660; 5-CF 3 -6-Et-4-Py], [BE4661; 3-CN-6- Et-4-Py !, [BE4662; 2-CN-6-Et-4-Py], [BE4663; 5-CN-6-Et-4-Py], [BE4664; 3-OMe-6-Et- 4-Py], [BE 4665; 2-OMe-6-Et-4-Py], [BE 4666; 5-OMe-6-Et-4-Py], [BE 4667; 3-CH ₂ CF ₃ -4-Py ], [BE 4668; 2-Cl-3-CH ₂ CF ₃ -4-Py], [BE 4 669; 5-Cl-3-CH ₂ CF ₃ -4-Py], [BE 4 670; 6-Cl-3-CH ₂ CF ₃ -4-Py], [BE 4671; 2-Me-3-CH ₂ CF ₃ -4-Py], [BE 4672; 5-Me-3-CH ₂ CF ₃ -4-Py], [BE 4 673; _{6-Me-3-CH 2} CF 3 -4-Py], [BE4674; 2-CF 3 -3-CH 2 CF 3 -4-Py], [BE4675; 5-CF 3 -3-CH 2 CF 3 -4-Py], [BE4676; 6-CF 3 -3-CH 2 CF 3 -4-Py], [BE4677; 2-CN-3-CH 2 CF 3 -4-Py], [BE4678; 5- _{CN-3-CH 2 CF 3} -4-Py], [BE4679; 6-CN-3-CH _{2 CF 3 -4-Py],} [BE4680; 2-OMe-3-CH 2 CF 3 -4-Py], [BE4681; 5-OMe-3-CH 2 CF 3 -4-Py], [BE4682; _{6-OMe-3-CH 2} CF 3 -4-Py], [BE4683; 2-CH 2 CF 3 -4-Py], [BE4684; 3-Cl-2-CH 2 CF 3 -4-Py], [BE4685; 5-Cl-2 -CH 2 CF 3 -4-Py], [BE4686; 6-Cl-2-CH 2 CF 3 -4-Py], [BE4687; 3-Me-2-CH 2 CF ₃ -4-Py !, [BE 4688; 5-Me-2-CH ₂ CF ₃ -4-Py], [BE 4689; 6-Me-2-CH ₂ CF ₃ -4-Py], [BE 4690; 3- CF ₃ -2-CH ₂ CF ₃ -4-Py], [BE 469 1; 5-CF ₃ -2-CH ₂ CF ₃ -4-Py], [BE 4 6 2; 6-CF ₃ -2-CH ₂ CF _3- 4-Py], [BE4693; 3-CN-2-CH 2 CF 3 -4-Py], [BE4694; 5-CN-2-CH 2 CF 3 -4-Py], [BE4695; 6-CN- _{2-CH 2 CF 3 -4-} Py], [BE4696; 3-OMe-2-CH 2 CF 3 -4-Py], [BE4697; 5-OMe-2-CH 2 CF 3 -4-Py], [BE 4698; 6-OMe-2-CH ₂ CF ₃ -4-Py], [BE 4699; 5-CH ₂ CF ₃ -4-Py], [BE 4700; 3-Cl-5-CH ₂ CF ₃ -4- Py], [BE 4701; 2-Cl-5-CH ₂ CF ₃ -4-Py],

[BE4702; 6-Cl-5 -CH 2 CF 3 -4-Py], [BE4703; 3-Me-5-CH 2 CF 3 -4-Py], [BE4704; 2-Me-5-CH 2 CF ₃ -4-Py], [BE 4705; 6-Me-5-CH ₂ CF ₃ -4-Py], [BE 4706; 3-CF ₃ -5-CH ₂ CF ₃ -4-Py], [BE 4 707; 2 _{-CF 3 -5-CH 2 CF 3} -4-Py], [BE4708; 6-CF 3 -5-CH 2 CF 3 -4-Py], [BE4709; 3-CN-5-CH 2 CF 3 - 4-Py], [BE4710; 2-CN-5-CH 2 CF 3 -4-Py], [BE4711; 6-CN-5-CH 2 CF 3 -4-Py], [BE4712; 3-OMe- _{5-CH 2 CF 3 -4-} Py], [BE4713; 2-OMe-5-CH 2 CF 3 -4-Py], [BE4714; 6-OMe-5-CH 2 CF 3 -4-Py], [BE 4715; 6-CH ₂ CF ₃ -4-Py], [BE 4716; 3-Cl-6-CH ₂ CF ₃ -4-Py], [BE 4 717; 2-Cl-6-CH ₂ CF ₃ -4- Py], [BE4718; 5- Cl-6-CH 2 CF 3 -4-Py], [BE4719; 3-Me-6-CH 2 CF 3 -4-Py], [BE4720; 2-Me-6- _{CH 2 CF 3 -4-Py]} , [BE4721; 5-Me-6-CH 2 CF 3 -4-Py], [BE4722; 3-CF 3 -6-CH 2 CF 3 -4-Py], [ BE 4723; 2-CF ₃ -6-CH ₂ CF ₃ -4-Py], [BE 4724; 5-CF ₃ -6-CH ₂ CF ₃ -4-Py], [BE 4 725; 3-CN -6-CH ₂ CF ₃ -4-Py !, [BE 4726; 2-CN-6-CH ₂ CF ₃ -4-Py], [BE 4727; 5-CN-6-CH ₂ CF ₃ -4-Py], [BE 4728; 3] _{-OMe-6-CH 2 CF 3} -4-Py], [BE4729; 2-OMe-6-CH 2 CF 3 -4-Py], [BE4730; 5-OMe-6-CH 2 CF 3 -4- Py], [BE 4731; 3-OEt-4-Py], [BE 4732; 2-Cl-3-OEt-4-Py], [BE 4 733; 5-Cl-3-OEt-4-Py !, [BE4734; 6-Cl-3-OEt-4-Py], [BE4735; 2-Me-3-OEt-4-Py], [BE4736; 5- Me-3-OEt-4- Py], [BE4737; 6-Me-3-OEt-4-Py], [BE4738; 2-CF 3 -3-OEt-4-Py], [BE4739; 5-CF ₃ -3-OEt-4-Py], [BE 4740; 6-CF ₃ -3-OEt-4-Py], [BE 474 1; 2-CN-3-OEt-4-Py], [BE 474 2; -3-OEt-4-Py !, [BE4743; 6-CN-3-OEt-4-Py], [BE4744; 2-OMe-3-OEt-4-Py], [BE4745; 5-OMe-3 -OEt-4-Py], [BE4746; 6-OMe-3-OEt-4-Py], [BE4747; 2-OEt-4-Py], [BE4748; 3-Cl-2-OEt-4-Py ], [BE 4749; 5-Cl-2-OEt-4-Py], [BE 4750; 6-Cl-2-OEt-4-Py], [BE 4751; 3-Me-2-OEt-4-Py], [BE4752; 5-Me-2 -OEt-4-Py], [BE4753; 6-Me-2-OEt-4-Py], [BE4754; 3-CF 3 -2-OEt-4-Py], [ _{BE4755; 5-CF 3 -2-} OEt-4-Py], [BE4756; 6-CF 3 -2-OEt-4-Py], [BE4757; 3-CN-2-OEt-4-Py], [ BE 4758; 5-CN-2-OEt-4-Py], [BE 4759; 6-CN-2-OEt-4-Py], [BE 4760; 3-OMe-2-OEt-4-Py], [BE 4761; 5-OMe-2-OEt-4-Py], [BE4762; 6-OMe-2-OEt-4-Py], [BE4763; 5-OEt-4-Py], [BE4764; 3-Cl-5-4 OEt-4-Py], [BE4765; 2-Cl-5-OEt-4-Py], [BE4766; 6-Cl-5-OEt-4-Py], [BE4767; 3-Me-5-OEt- 4-Py], [BE4768; 2-Me-5-OEt-4-Py], [BE4769; 6-Me-5-OEt-4-Py], [BE4770; 3-CF 3 -5-OEt-4 -Py], [BE4771; 2- CF 3 -5-OEt-4-Py], [BE4772; 6-CF _{3 -5-OEt-4-Py} ], [BE4773; 3-CN-5-OEt-4-Py], [BE4774; 2-CN-5-OEt-4-Py], [BE4775; 6-CN- 5-OEt-4-Py], [BE4776; 3-OMe-5-OEt-4-Py], [BE4777; 2-OMe-5-OEt-4-Py], [BE4778; 6-OMe-5- OEt-4-Py], [BE4779; 6-OEt-4-Py], [BE4780; 3-Cl-6-OEt-4-Py], [BE4781; 2-Cl-6-OEt-4-Py] , [BE 4782; 5-Cl-6-OEt-4-Py], [BE4783; 3-Me-6-OEt-4-Py], [BE4784; 2-Me-6-OEt-4-Py], [BE4782; BE4785; 5-Me-6- OEt-4-Py], [BE4786; 3-CF 3 -6-OEt-4-Py], [BE4787; 2-CF 3 -6-OEt-4-Py], [ _{BE4788; 5-CF 3 -6-} OEt-4-Py], [BE4789; 3-CN-6-OEt-4-Py], [BE4790; 2-CN-6-OEt-4-Py], [BE4791 5-CN-6-OEt-4-Py !, [BE4792; 3-OMe-6-OEt-4-Py], [BE4793; 2-OMe-6-OEt-4-Py], [BE4794; -OMe-6-OEt-4- Py], [BE4795; 3-OCH 2 CF 3 -4-Py], [BE4796; 2-Cl-3-OCH 2 CF 3 -4-Py], [BE4797; 5 _{-Cl-3-OCH 2 CF 3} -4-Py], [BE4798; 6-Cl-3-OCH 2 CF 3 -4-Py], [BE4799; 2-Me-3-OCH 2 CF 3 -4- Py], [BE4800; 5- Me-3-OCH 2 CF 3 -4-Py], [BE4801; 6-Me-3-OCH 2 CF 3 -4-Py],

_{[BE4802; 2-CF 3 -3} -OCH 2 CF 3 -4-Py], [BE4803; 5-CF 3 -3-OCH 2 CF 3 -4-Py], [BE4804; 6-CF 3 -3- _{OCH 2 CF 3 -4-Py]} , [BE4805; 2-CN-3-OCH 2 CF 3 -4-Py], [BE4806; 5-CN-3-OCH 2 CF 3 -4-Py], [BE4807 ; 6-CN-3-OCH 2 CF 3 -4-Py], [BE4808; 2-OMe-3-OCH 2 CF 3 -4-Py], [BE4809; 5-OMe-3-OCH 2 CF 3 - 4-Py], [BE4810; 6-OMe-3-OCH 2 CF 3 -4-Py], [BE4811; 2-OCH 2 CF 3 -4-Py], [BE4812; 3-Cl-2-OCH 2 CF ₃ -4-Py !, [BE 4813; 5-Cl-2-OCH ₂ CF ₃ -4-Py], [BE 4814; 6-Cl 2-OCH ₂ CF ₃ -4-Py], [BE 4815; 3 _{-Me-2-OCH 2 CF 3} -4-Py], [BE4816; 5-Me-2-OCH 2 CF 3 -4-Py], [BE4817; 6-Me-2-OCH 2 CF 3 -4- Py], [BE 4818; 3-CF ₃ -2-OCH ₂ CF ₃ -4-Py], [BE 4819; 5-CF ₃ -2-OCH ₂ CF ₃ -4-Py], [BE 4820; 6-CF _{3 -2-OCH 2 CF 3 -4-} Py], [BE4821; 3-CN-2-OCH 2 CF 3 -4-Py], [BE4822; 5-CN-2-OCH 2 CF 3 -4-Py] , [BE4823; 6-CN- 2-OCH 2 CF 3 -4-Py], [BE4824; 3-OMe-2-OCH 2 CF 3 -4-Py], [BE4825; 5-OMe-2-OCH 2 CF ₃ -4-Py !, [BE 48 26; 6-OMe -2-OCH ₂ CF ₃ -4-Py], [BE 4827; 5-OCH ₂ CF ₃ -4-Py], [BE 4 828; 3-Cl-5 _{-OCH 2 CF 3 -4-Py]} , [BE4829; 2-Cl-5-OCH 2 CF 3 -4-Py], [BE4830; 6-Cl-5-OCH 2 CF 3 -4-Py], [ BE 4831; 3-Me-5-OCH ₂ CF ₃ -4- Py], [BE4832; 2- Me-5-OCH 2 CF 3 -4-Py], [BE4833; 6-Me-5-OCH 2 CF 3 -4-Py], [BE4834; 3-CF 3 -5 -OCH ₂ CF ₃ -4-Py], [BE 4835; 2-CF ₃ -5-OCH ₂ CF ₃ -4-Py], [BE 4836; 6-CF ₃ -5-OCH ₂ CF ₃ -4-Py] , [BE4837; 3-CN- 5-OCH 2 CF 3 -4-Py], [BE4838; 2-CN-5-OCH 2 CF 3 -4-Py], [BE4839; 6-CN-5-OCH 2 _{CF 3 -4-Py], [} BE4840; 3-OMe-5-OCH 2 CF 3 -4-Py], [BE4841; 2-OMe-5-OCH 2 CF 3 -4-Py], [BE4842; 6 _{-OMe-5-OCH 2 CF 3} -4-Py], [BE4843; 6-OCH 2 CF 3 -4-Py], [BE4844; 3-Cl-6-OCH 2 CF 3 -4-Py], [ BE4845; 2-Cl-6- OCH 2 CF 3 -4-Py], [BE4846; 5-Cl-6-OCH 2 CF 3 -4-Py], [BE4847; 3-Me-6-OCH 2 CF 3 -4-Py], [BE4848; 2-Me-6-OCH 2 CF 3 -4-Py], [BE4849; 5-Me-6-OCH 2 CF 3 -4-Py], [BE4850; 3-CF _{3 -6-OCH 2 CF 3 -4} -Py], [BE4851; 2-CF 3 -6-OCH 2 CF 3 -4-Py], [BE4852; 5-CF 3 -6-OCH 2 CF 3 -4 -Py], [BE4853; 3- CN-6-OCH 2 CF 3 -4-Py], [BE4854; 2-CN-6-OCH 2 CF 3 -4-Py], [BE4855; 5-CN-6 _{-OCH 2 CF 3 -4-Py]} , [BE4856; 3-OMe-6-OCH 2 CF 3 -4-Py], [BE4857; 2-OMe-6-OCH 2 CF 3 -4-Py], [ BE 4858; 5-OMe-6-OCH ₂ CF ₃ -4-Py], [BE 4859; 3-Pr-4-Py], [BE 4860; 2-Cl-3-Pr-4-Py], [BE 4861; -Cl-3-Pr-4-Py], [BE 482; 6-Cl-3-Pr-4 -Py], [BE 4863; 2-Me-3-Pr-4-Py], [BE 4864; 5-Me-3-Pr-4-Py], [BE 4865; 6-Me-3-Pr-4-Py ], [BE4866; 2-CF 3 -3-Pr-4-Py], [BE4867; 5-CF 3 -3-Pr-4-Py], [BE4868; 6-CF 3 -3-Pr-4- Py], [BE 4869; 2-CN-3-Pr-4-Py], [BE 4870; 5-CN-3-Pr-4-Py], [BE 4871; 6-CN-3-Pr-4-Py] , [BE 4 872; 2-OMe-3-Pr-4-Py], [BE 4873; 5-OMe-3-Pr-4-Py], [BE 4874; 6-OMe-3-Pr-4-Py], [BE 4 872; BE 4875; 2-Pr-4-Py], [BE 4876; 3-Cl-2-Pr-4-Py], [BE 4877; 5-Cl-2-Pr-4-Py], [BE 4878; 6-Cl- 2-Pr-4-Py], [BE4879; 3-Me-2-Pr-4-Py], [BE4880; 5-Me-2-Pr-4-Py], [BE4881; 6-Me-2-] Pr-4-Py], [ BE4882; 3-CF 3 -2-Pr-4-Py], [BE4883; 5-CF 3 -2-Pr-4-Py], [BE4884; 6-CF 3 -2 -Pr-4-Py], [BE4885; 3-CN-2-Pr-4-Py], [BE4886; 5-CN-2-Pr-4-Py], [BE4887; 6-CN-2-Pr -4-Py], [BE4888; 3-OMe-2-Pr-4-Py], [BE4889; 5-OMe-2-Pr-4-Py], [BE4890; 6-OMe-2-Pr-4 -Py], [BE4891; 5-Pr-4-Py], [BE 4892; 3-Cl-5-Pr-4-Py], [BE4893; 2-Cl-5-Pr-4-Py], [BE 4894] 6-Cl-5-Pr-4-Py !, [BE4895; 3-Me-5-Pr-4-Py], [BE4896; 2-Me-5-Pr-4-Py], [BE4897; -Me-5-Pr-4- Py], [BE4898; 3-CF 3 -5-Pr-4-Py], [BE4899; 2-CF 3 -5-Pr-4-Py], [BE4900; 6 _{-CF 3 -5-Pr-4-} Py], [BE4901; 3-CN-5-Pr-4-Py],

[BE4902; 2-CN-5-Pr-4-Py], [BE4903; 6-CN-5-Pr-4-Py], [BE 4904; 3-OMe-5-Pr-4-Py], [BE 4905] 2-OMe-5-Pr-4-Py !, [BE4906; 6-OMe-5-Pr-4-Py], [BE4907; 6-Pr-4-Py], [BE4908; 3-Cl-6 -Pr-4-Py], [BE4909; 2-Cl-6-Pr-4-Py], [BE4910; 5-Cl-6-Pr-4-Py], [BE4911; 3-Me-6-Pr -4-Py !, [BE4912; 2-Me-6-Pr-4-Py], [BE4913; 5-Me-6-Pr-4-Py], [BE4914; 3-CF ₃ -6-Pr- 4-Py], [BE4915; 2-CF 3 -6-Pr-4-Py], [BE4916; 5-CF 3 -6-Pr-4-Py], [BE4917; 3-CN-6-Pr- 4-Py], [BE4918; 2-CN-6-Pr-4-Py], [BE4919; 5-CN-6-Pr-4-Py], [BE4920; 3-OMe-6-Pr-4- 4 Py], [BE4921; 2-OMe-6-Pr-4-Py], [BE4922; 5-OMe-6-Pr-4-Py], [BE4923; 3-OPr-4-Py], [BE4924; 2-Cl-3-OPr-4-Py], [BE4925; 5-Cl-3-OPr-4-Py], [BE4926; 6-Cl-3-OPr-4-Py], [BE4927; Me-3-OPr-4-Py], [BE 4928; 5-Me-3-OPr-4-Py], [BE 4929; 6-Me-3-OPr-4-Py], [BE 4930; 2-CF ₃ -3-OPr-4-Py] , [BE4931; 5-CF 3 -3-OPr-4-Py], [BE4932; 6-CF 3 -3-OPr-4-Py], [BE4933; 2-CN -3-OPr-4-Py !, [BE4934; 5-CN-3-OPr-4-Py], [BE4935; 6-CN-3-OPr-4-Py], [BE4936; 2-OMe-3 -OPr-4-Py], [BE4937; 5-OMe-3-OPr-4-Py], [BE4938; 6-OMe-3-OPr-4-Py], [BE4939; 2-OPr-4-Py ], [BE 4940; 3-Cl-2-OPr-4-Py], [BE 4941; 5-Cl-2-OPr-4-Py], [BE 49 42; 6] -Cl-2-OPr-4-Py], [BE 4943; 3-Me-2-OPr-4-Py], [BE 4944; 5-Me-2-OPr-4-Py], [BE 4945; 6-Me -2-OPr-4-Py] , [BE4946; 3-CF 3 -2-OPr-4-Py], [BE4947; 5-CF 3 -2-OPr-4-Py], [BE4948; 6-CF _{3 -2-OPr-4-Py} ], [BE4949; 3-CN-2-OPr-4-Py], [BE4950; 5-CN-2-OPr-4-Py], [BE4951; 6-CN- 2-OPr-4-Py], [BE4952; 3-OMe-2-OPr-4-Py], [BE4953; 5-OMe-2-OPr-4-Py], [BE4954; 6-OMe-2- OPr-4-Py], [BE4955; 5-OPr-4-Py], [BE4956; 3-Cl-5-OPr-4-Py], [BE4957; 2-Cl-5-OPr-4-Py] , [BE4958; 6-Cl-5-OPr-4-Py], [BE4959; 3-Me-5-OPr-4-Py], [BE4960; 2-Me-5-OPr-4-Py], [BE4959; BE4961; 6-Me-5- OPr-4-Py], [BE4962; 3-CF 3 -5-OPr-4-Py], [BE4963; 2-CF 3 -5-OPr-4-Py], [ _{BE4964; 6-CF 3 -5-} OPr-4-Py], [BE4965; 3-CN-5-OPr-4-Py], [BE4966; 2-CN-5-OPr-4-Py], [BE4967 6-CN-5-OPr-4-Py !, [BE4968; 3-OMe-5-OPr-4-Py], [BE4969; 2-OMe-5-OPr-4-Py], [BE4970; -OMe-5-OPr-4-Py], [BE4971; 6-OPr-4-Py], [BE4972; 3-Cl-6-OPr-4-Py], [BE4973; 2-Cl-6-OPr -4-Py], [BE 4974; 5-Cl-6-OPr-4-Py], [BE 4975; 3-Me-6-OPr-4-Py], [BE 4976; 2-Me-6-OPr-4 -Py], [BE 4977; 5-Me-6-OPr-4-Py], [BE 4978; 3-CF ₃ -6-OPr-4-Py], [BE 4979; 2-CF ₃ -6-OPr-4 -Py], [BE 4980; 5-CF ₃ -6-OPr-4-Py], [BE 4981; 3-C N-6-OPr-4-Py], [BE4982; 2-CN-6-OPr-4-Py], [BE4983; 5-CN-6-OPr-4-Py], [BE4984; 3-OMe- 6-OPr-4-Py], [BE4985; 2-OMe-6-OPr-4-Py], [BE4986; 5-OMe-6-OPr-4-Py], [BE4987; 3-SMe-4- Py], [BE4988; 2-Cl-3-SMe-4-Py], [BE4989; 5-Cl-3-SMe-4-Py], [BE4990; 6-Cl-3-SMe-4-Py] , [BE4991; 2-Me-3-SMe-4-Py], [BE4992; 5-Me-3-SMe-4-Py], [BE4993; 6-Me-3-SMe-4-Py], [BE4992; _{BE4994; 2-CF 3 -3-} SMe-4-Py], [BE4995; 5-CF 3 -3-SMe-4-Py], [BE4996; 6-CF 3 -3-SMe-4-Py], [BE4997; 2-CN-3-SMe-4-Py], [BE4998; 5-CN-3-SMe-4-Py], [BE4999; 6-CN-3-SMe-4-Py], [BE5000] 2-OMe-3-SMe-4-Py !, [BE 5001; 5-OMe-3-SMe-4-Py],

[BE5002; 6-OMe-3-SMe-4-Py], [BE5003; 2-SMe-4-Py], [BE5004; 3-Cl-2-SMe-4-Py], [BE5005; -2-SMe-4-Py !, [BE5006; 6-Cl-2-SMe-4-Py], [BE5007; 3-Me-2-SMe-4-Py], [BE5008; 5-Me-2 -SMe-4-Py], [ BE5009; 6-Me-2-SMe-4-Py], [BE5010; 3-CF 3 -2-SMe-4-Py], [BE5011; 5-CF 3 -2 -SMe-4-Py], [ BE5012; 6-CF 3 -2-SMe-4-Py], [BE5013; 3-CN-2-SMe-4-Py], [BE5014; 5-CN-2- SMe-4-Py !, [BE5015; 6-CN-2-SMe-4-Py], [BE5016; 3-OMe-2-SMe-4-Py], [BE5017; 5-OMe-2-SMe- 4-Py], [BE5018; 6-OMe-2-SMe-4-Py], [BE5019; 5-SMe-4-Py], [BE5020; 3-Cl-5-SMe-4-Py], [BE50 20; BE 5021; 2-Cl-5-SMe-4-Py], [BE5022; 6-Cl-5-SMe-4-Py], [BE5023; 3-Me-5-SMe-4-Py], [BE5024; 2-Me-5-SMe- 4-Py], [BE5025; 6-Me-5-SMe-4-Py], [BE5026; 3-CF 3 -5-SMe-4-Py], [BE5027; 2 _{-CF 3 -5-SMe-4-} Py], [BE5028; 6-CF 3 -5-SMe-4-Py], [BE5029; 3-CN-5-SMe-4-Py], [BE5030; 2 -CN-5-SMe-4-Py], [BE 5031; 6-CN-5-SMe-4-Py], [BE 5032; 3-OMe-5-SMe-4-Py], [BE 5033; 2-OMe -5-SMe-4-Py !, [BE5034; 6-OMe-5-SMe-4-Py], [BE5035; 6-SMe-4-Py], [BE5036; 3-Cl-6-SMe-4 -Py], [BE5037; 2-Cl-6-SMe-4-Py], [BE5038; 5-Cl-6-SMe-4-Py], [BE5039; 3-Me-6-SMe-4-Py ], [BE 5040; 2-Me-6-SMe-4-Py], [BE 5041; 5-Me-6- SMe-4-Py], [ BE5042; 3-CF 3 -6-SMe-4-Py], [BE5043; 2-CF 3 -6-SMe-4-Py], [BE5044; 5-CF 3 -6 -SMe-4-Py], [BE5045; 3-CN-6-SMe-4-Py], [BE5046; 2-CN-6-SMe-4-Py], [BE5047; 5-CN-6-SMe -4-Py], [BE5048; 3-OMe-6-SMe-4-Py], [BE5049; 2-OMe-6-SMe-4-Py], [BE5050; 5-OMe-6-SMe-4 -Py], [BE5051; 3- SCF 3 -4-Py], [BE5052; 2-Cl-3-SCF 3 -4-Py], [BE5053; 5-Cl-3-SCF 3 -4-Py] , [BE 5054; 6-Cl-3-SCF ₃ -4-Py], [BE 5055; 2-Me-3-SCF ₃ -4-Py], [BE 5056; 5-Me-3-SCF ₃ -4-Py ], [BE 5057; 6-Me-3-SCF ₃ -4-Py], [BE 5058; 2-CF ₃ -3-SCF ₃ -4-Py], [BE 5059; 5-CF ₃ -3-SCF _3- 4-Py], [BE5060; 6-CF 3 -3-SCF 3 -4-Py], [BE5061; 2-CN-3-SCF 3 -4-Py], [BE5062; 5-CN-3-SCF ₆ -4-Py !, [BE 5063; 6-CN-3-SCF ₃ -4-Py], [BE 5064; 2-OMe-3-SCF ₃ -4-Py], [BE 5065; 5-OMe -3-] SCF ₃ -4-Py !, [BE 5066; 6-OMe -3-SCF ₃ -4-Py], [BE 5067; 2-SCF ₃ -4-Py], [BE 5068; 3-Cl-2-SCF _3- 4-Py], [BE5069; 5-Cl-2-SCF ₃ -4-Py], [BE 5070; 6-Cl-2-SCF ₃ -4-Py], [BE 5071; 3-Me-2-SCF ₃ -4-Py], [BE5072; 5-Me-2-SCF 3 -4-Py], [BE5073; 6-Me-2-SCF 3 -4-Py], [BE5074; 3-CF 3 -2- SCF ₃ -4-Py !, [BE 5075; 5-CF ₃ -2-SCF ₃ -4-Py], [BE 5076; 6-CF ₃ -2-SCF ₃ -4-Py], [BE 5077; 3-CN] -2 -SCF ₃ -4-Py], [BE 5078; 5-CN-2-SCF ₃ -4-Py], [BE 5079; 6-CN 2-SCF ₃ -4-Py], [BE 5080; 3-OMe- _{2-SCF 3 -4-Py]} , [BE5081; 5-OMe-2-SCF 3 -4-Py], [BE5082; 6-OMe-2-SCF 3 -4-Py], [BE5083; 5-SCF ₃ -4-Py !, [BE 5084; 3-Cl-5-SCF ₃ -4-Py], [BE 5085; 2-Cl-5-SCF ₃ -4-Py], [BE 5086; 6-Cl-5- SCF ₃ -4-Py !, [BE 5087; 3-Me-5-SCF ₃ -4-Py], [BE 5088; 2-Me-5-SCF ₃ -4-Py], [BE 5089; 6-Me-5 -SCF ₃ -4-Py], [BE 5090; 3-CF ₃ -5-SCF ₃ -4-Py], [BE 50 1; 2-CF ₃ -5-SCF ₃ -4-Py], [BE 50 9 2; 6- _{CF 3 -5-SCF 3 -4-} Py], [BE5093; 3-CN-5-SCF 3 -4-Py], [BE5094; 2-CN-5-SCF 3 -4-Py], [BE5095; _{6-CN-5-SCF 3} -4-Py], [BE5096; 3-OMe-5-SCF 3 -4-Py], [BE5097; 2-OMe-5-SCF 3 -4-Py], [BE5098 ; 6-OMe-5-SCF 3 -4-Py], [BE5099; 6-SCF 3 -4-Py], [BE5100; 3-Cl-6-SCF 3 -4-Py], [BE5101; 2- Cl-6-SCF ₃ -4-Py],

[BE5102; 6-Cl-6-SCF ₃ -4-Py], [BE 5103; 3-Me-6-SCF ₃ -4-Py], [BE 5104; 2-Me-6-SCF ₃ -4-Py] , [BE5105; 6-Me- 6-SCF 3 -4-Py], [BE5106; 3-CF 3 -6-SCF 3 -4-Py], [BE5107; 2-CF 3 -6-SCF 3 -4 -Py], [BE5108; 6- CF 3 -6-SCF 3 -4-Py], [BE5109; 3-CN-6-SCF 3 -4-Py], [BE5110; 2-CN-6-SCF 3 -4-Py], [BE5111; 6-CN-6-SCF 3 -4-Py], [BE5112; 3-OMe-6-SCF 3 -4-Py], [BE5113; 2-OMe-6-SCF ₃ -4-Py !, [BE 5114; 6-OMe-6-SCF ₃ -4-Py], [BE 5115; 3-S (O) Me-4-Py], [BE 5116; 2-Cl-3-S (O) Me-4-Py], [BE5117; 5-Cl-3-S (O) Me-4-Py], [BE5118; 6-Cl-3-S (O) Me-4-Py], [BE5119; 2-Me-3-S (O) Me-4-Py], [BE5120; 5-Me-3-S (O) Me-4-Py], [BE5121; 6-Me-3-S (O) Me-4-Py ], [BE5122; 2-CF 3 -3-S (O) Me-4-Py], [BE5123; 5-CF 3 -3-S (O) Me-4-Py ], [BE5124; 6-CF 3 -3-S (O) Me-4-Py], [BE5125; 2-CN-3-S (O) Me-4-Py], [BE5126; 5-CN- 3-S (O) Me-4-Py], [BE5127; 6-CN-3-S (O) Me-4-Py], [BE5128; 2-OMe-3-S (O) Me-4- 4 Py], [BE5129; 5-OMe-3-S (O) Me-4-Py], [BE5130; 6-OMe-3-S (O) Me-4-Py], [BE5131; O) Me-4-Py], [BE 5132; 3-Cl-2-S (O) Me-4-Py], [BE 5133; 5-Cl-2-S (O) Me-4-Py], [BE BE5134; 6-Cl-2-S (O) Me-4-Py], [BE5135; 3-Me-2-S (O) Me-4-Py], [BE5136; 5-Me-2-S ( O) Me-4-Py], [BE 513 7; 6-Me-2- S (O) Me-4-Py], [BE5138; 3-CF 3 -2-S (O) Me-4-Py], [BE5139; 5-CF 3 -2- S (O) Me-4- Py], [BE5140; 6-CF 3 -2-S (O) Me-4-Py], [BE5141; 3-CN-2-S (O) Me-4-Py ], [BE5142; 5-CN-2-S (O) Me-4-Py], [BE5143; 6-CN-2-S (O) Me-4-Py], [BE5144; 3-OMe-2 -S (O) Me-4-Py], [BE5145; 5-OMe-2-S (O) Me-4-Py], [BE5146; 6-OMe-2-S (O) Me-4-Py ], [BE 5147; 5-S (O) Me-4-Py], [BE 5148; 3-Cl-5-S (O) Me-4-Py], [BE 5149; 2-Cl-5-S (O ) Me-4-Py], [BE5150; 6-Cl-5-S (O) Me-4-Py], [BE5151; 3-Me-5-S (O) Me-4-Py], [BE5152 ; 2-Me-5-S (O) Me-4-Py], [BE5153; 6-Me-5-S (O) Me-4-Py], [BE5154; 3-CF 3 -5-S ( O) Me-4-Py] , [BE5155; 2-CF 3 -5-S (O) Me-4-Py], [BE5156; 6-CF 3 -5-S (O) Me-4-Py] , [BE5157; 3-CN-5-S (O) Me-4-Py], [BE5158; 2-CN-5-S (O) Me-4-Py], [BE5159; 6-CN-5- S (O) Me-4-Py], [BE5160; 3-OMe-5-S (O) Me-4-Py], [BE5161; 2-OMe-5-S (O) Me-4-Py] , [BE5162; 6-OMe-5-S (O) Me-4-Py], [BE5163; 6-S (O) Me-4-Py], [BE5164; 3-Cl-6-S (O) Me-4-Py !, [BE5165; 2-Cl-6-S (O) Me-4-Py], [BE5166; 5-Cl-6-S (O) Me-4-Py], [BE5167; 3-Me-6-S (O) Me-4-Py], [BE5168; 2-Me-6-S (O) Me-4-Py], [BE5169; 5-Me-6-S (O) Me-4-Py], [ BE5170; 3-CF 3 -6-S (O) Me-4-Py], [BE5171; 2-CF 3 -6-S (O) Me-4-Py], [ BE 517 _{2; 5-CF 3 -6-} S (O) Me-4-Py], [BE5173; 3-CN-6-S (O) Me-4-Py], [BE5174; 2-CN-6-S (O) Me-4-Py], [BE5175; 5-CN-6-S (O) Me-4-Py], [BE5176; 3-OMe-6-S (O) Me-4-Py], [BE5177; 2-OMe-6-S (O) Me-4-Py], [BE5178; 5-OMe-6-S (O) Me-4-Py], [BE5179; 3-S (O) CF _{3 -4-Py], [BE5180} ; 2-Cl-3-S (O) CF 3 -4-Py], [BE5181; 5-Cl-3-S (O) CF 3 -4-Py], [ BE5182; 6-Cl-3- S (O) CF 3 -4-Py], [BE5183; 2-Me-3-S (O) CF 3 -4-Py], [BE5184; 5-Me-3- _{S (O) CF 3 -4-} Py], [BE5185; 6-Me-3-S (O) CF 3 -4-Py], [BE5186; 2-CF 3 -3-S (O) CF 3 - 4-Py], [BE 5187; 5-CF ₃ -3-S (O) CF ₃ -4-Py], [BE 5188; 6-CF ₃ -3-S (O) CF ₃ -4-Py], [4] BE5189; 2-CN-3- S (O) CF 3 -4-Py], [BE5190; 5-CN-3-S (O) CF 3 -4-Py], [BE5191; 6-CN-3- _{S (O) CF 3 -4-} Py], [BE5192; 2-OMe-3-S (O) CF 3 -4-Py], [BE5193; 5-OMe-3-S (O) CF 3 -4 -Py], [BE5194; 6- OMe-3-S (O) CF 3 -4-Py], [BE5195; 2-S (O) CF 3 -4-Py], [BE5196; 3-Cl-2 _{-S (O) CF 3 -4-} Py], [BE5197; 5-Cl-2-S (O) CF 3 -4-Py], [BE5198; 6-Cl-2-S (O) CF 3 - 4-Py], [BE5199; 3-Me-2-S (O) CF 3 -4-Py], [BE5200; 5-Me-2-S (O) CF 3 -4-Py], [BE5201; 6-Me-2-S ( O) CF 3 -4-Py],

_{[BE5202; 3-CF 3 -2} -S (O) CF 3 -4-Py], [BE5203; 5-CF 3 -2-S (O) CF 3 -4-Py], [BE5204; 6-CF _{3 -2-S (O) CF} 3 -4-Py], [BE5205; 3-CN-2-S (O) CF 3 -4-Py], [BE5206; 5-CN-2-S (O) _{CF 3 -4-Py], [} BE5207; 6-CN-2-S (O) CF 3 -4-Py], [BE5208; 3-OMe-2-S (O) CF 3 -4-Py], [BE5209; 5-OMe-2 -S (O) CF 3 -4-Py], [BE5210; 6-OMe-2-S (O) CF 3 -4-Py], [BE5211; 5-S (O ) CF ₃ -4-Py !, [BE 5212; 3-Cl-5-S (O) CF ₃ -4-Py], [BE 5213; 2-Cl-5-S (O) CF ₃ -4-Py] , [BE5214; 6-Cl- 5-S (O) CF 3 -4-Py], [BE5215; 3-Me-5-S (O) CF 3 -4-Py], [BE5216; 2-Me- _{5-S (O) CF 3} -4-Py], [BE5217; 6-Me-5-S (O) CF 3 -4-Py], [BE5218; 3-CF 3 -5-S (O) CF ₃ -4-Py], [BE 5219; 2-CF ₃ -5-S (O) CF ₃ -4-Py], [BE 5220; 6-CF ₃ -5-S (O) CF ₃ -4-Py] , [BE5221; 3-CN- 5-S (O) CF 3 -4-Py], [BE5222; 2-CN-5-S (O) CF 3 -4-Py], [BE5223; 6-CN- _{5-S (O) CF 3} -4-Py], [BE5224; 3-OMe-5-S (O) CF 3 -4-Py], [BE5225; 2-OMe-5-S (O) CF 3 -4-Py], [BE5226; 6-OMe-5-S (O) CF 3 -4-Py], [BE5227; 6-S (O) CF 3 -4-Py], [BE5228; 3-Cl _{-6-S (O) CF 3} -4-Py], [BE5229; 2-Cl-6-S (O) CF 3 -4-Py], [BE5230; 5-Cl-6-S (O) CF ₃ -4-Py !, [BE5231; 3-Me-6-S (O) CF ₃ -4-Py], [BE5232; 2-Me-6-S (O) CF ₃ -4-Py], BE 5233; 5-Me-6-S (O) CF _3- 4-Py], [BE5234; 3-CF 3 -6-S (O) CF 3 -4-Py], [BE5235; 2-CF 3 -6-S (O) CF 3 -4-Py], [ _{BE5236; 5-CF 3 -6-} S (O) CF 3 -4-Py], [BE5237; 3-CN-6-S (O) CF 3 -4-Py], [BE5238; 2-CN-6 _{-S (O) CF 3 -4-} Py], [BE5239; 5-CN-6-S (O) CF 3 -4-Py], [BE5240; 3-OMe-6-S (O) CF 3 - 4-Py], [BE5241; 2-OMe-6-S (O) CF 3 -4-Py], [BE5242; 5-OMe-6-S (O) CF 3 -4-Py], [BE5243; _{3-S (O) 2 Me} -4-Py], [BE5244; 2-Cl-3-S (O) 2 Me-4-Py], [BE5245; 5-Cl-3-S (O) 2 Me -4-Py], [BE5246; 6-Cl-3-S (O) 2 Me-4-Py], [BE5247; 2-Me-3-S (O) 2 Me-4-Py], [BE5248 ; 5-Me-3-S (O) 2 Me-4-Py], [BE5249; 6-Me-3-S (O) 2 Me-4-Py], [BE5250; 2-CF 3 -3- _{S (O) 2 Me-4} -Py], [BE5251; 5-CF 3 -3-S (O) 2 Me-4-Py], [BE5252; 6-CF 3 -3-S (O) 2 Me -4-Py], [BE5253; 2-CN-3-S (O) 2 Me-4-Py], [BE5254; 5-CN-3-S (O) 2 Me-4-Py], [BE5255 ; 6-CN-3-S (O) 2 Me-4-Py], [BE5256; 2-OMe-3-S (O) 2 Me-4-Py], [BE5257; 5-OMe-3-S (O) ₂ Me-4-Py], [BE5258; 6-OMe-3-S (O) ₂ Me-4-Py], [BE5259; 2-S (O) ₂ Me-4-Py], BE5260; 3-Cl-2- S (O) 2 Me-4-Py], [BE5261; 5-Cl-2-S (O) 2 Me-4-Py], [BE5262; 6-Cl-2- _{S (O) 2 Me-4} -Py], [BE5263; 3-Me-2-S (O) 2 Me-4-Py], [BE5264; 5-Me-2-S (O) 2 Me-4 -Py], [BE5265; 6-Me-2-S (O) _{2 Me-4-Py],} [BE5266; 3-CF 3 -2-S (O) 2 Me-4-Py], [BE5267; 5-CF 3 -2-S (O) 2 Me-4-Py ], [BE5268; 6-CF 3 -2-S (O) 2 Me-4-Py], [BE5269; 3-CN-2-S (O) 2 Me-4-Py], [BE5270; 5- CN-2-S (O) 2 Me-4-Py], [BE5271; 6-CN-2-S (O) 2 Me-4-Py], [BE5272; 3-OMe-2-S (O) ₂ Me-4-Py], [BE 5273; 5-OMe-2-S (O) ₂ Me-4-Py], [BE 5274; 6-OMe-2-S (O) ₂ Me-4-Py], [BE 5275; 5-S (O) ₂ Me-4-Py], [BE 5276; 3-Cl-5-S (O) ₂ Me-4-Py], [BE 5277; 2-Cl-5-S (O ) ₂ Me-4-Py], [BE5278; 6-Cl-5-S (O) ₂ Me-4-Py], [BE5279; 3-Me-5-S (O) ₂ Me-4-Py] , [BE5280; 2-Me- 5-S (O) 2 Me-4-Py], [BE5281; 6-Me-5-S (O) 2 Me-4-Py], [BE5282; 3-CF 3 _{-5-S (O) 2 Me} -4-Py], [BE5283; 2-CF 3 -5-S (O) 2 Me-4-Py], [BE5284; 6-CF 3 -5-S (O ) ₂ Me-4-Py], [BE 5285; 3-CN-5-S (O) ₂ Me-4-Py], [BE 5286; 2-CN-5-S (O) ₂ Me-4-Py] , [BE5287; 6-CN- 5-S (O) 2 Me-4-Py], [BE5288; 3-OMe-5-S (O) 2 Me-4-Py], [BE5289; 2-OMe- _{5-S (O) 2 Me} -4-Py], [BE5290; 6-OMe-5-S (O) 2 Me-4-Py], [BE5291; 6-S (O) 2 Me-4-Py ], [BE 5292; 3-Cl-6-S (O) ₂ Me-4-Py], [BE 5293; 2-Cl-6-S (O) ₂ Me-4-Py], [BE 5294; 5-Cl] _{-6-S (O) 2 Me} -4-Py], [BE5295; 3-Me-6-S (O) 2 Me-4-Py], [BE5296; 2-Me-6-S (O) 2 Me-4-Py], [BE5297; 5-Me- _{6-S (O) 2 Me} -4-Py], [BE5298; 3-CF 3 -6-S (O) 2 Me-4-Py], [BE5299; 2-CF 3 -6-S (O) _{2 Me-4-Py],} [BE5300; 5-CF 3 -6-S (O) 2 Me-4-Py], [BE5301; 3-CN-6-S (O) 2 Me-4-Py] ,

[BE5302; 2-CN-6 -S (O) 2 Me-4-Py], [BE5303; 5-CN-6-S (O) 2 Me-4-Py], [BE5304; 3-OMe-6 _{-S (O) 2 Me-4} -Py], [BE5305; 2-OMe-6-S (O) 2 Me-4-Py], [BE5306; 5-OMe-6-S (O) 2 Me- 4-Py], [BE5307; 3-S (O) 2 CF 3 -4-Py], [BE5308; 2-Cl-3-S (O) 2 CF 3 -4-Py], [BE5309; 5- Cl-3-S (O) 2 CF 3 -4-Py], [BE5310; 6-Cl-3-S (O) 2 CF 3 -4-Py], [BE5311; 2-Me-3-S ( O) ₂ CF ₃ -4-Py], [BE 53 12; 5-Me-3-S (O) ₂ CF ₃ -4-Py], [BE 53 13; 6-Me-3-S (O) ₂ CF _3- 4-Py], [BE5314; 2-CF 3 -3-S (O) 2 CF 3 -4-Py], [BE5315; 5-CF 3 -3-S (O) 2 CF 3 -4-Py] _{, [BE5316; 6-CF 3} -3-S (O) 2 CF 3 -4-Py], [BE5317; 2-CN-3-S (O) 2 CF 3 -4-Py], [BE5318; 5 -CN-3-S (O) 2 CF 3 -4-Py], [BE5319; 6-CN-3-S (O) 2 CF 3 -4-Py], [BE5320; 2-OMe-3-S _{(O) 2 CF 3 -4-} Py], [BE5321; 5-OMe-3-S (O) 2 CF 3 -4-Py], [BE5322; 6-OMe-3-S (O) 2 CF 3 -4-Py], [BE 5323; 2-S (O) ₂ CF ₃ -4-Py], [BE 5324; 3-Cl-2-S (O) ₂ CF ₃ -4-Py], [BE 5325; 5 -Cl-2-S (O) 2 CF 3 -4-Py], [BE5326; 6-Cl-2-S (O) 2 CF 3 -4-Py], [BE5327; 3-Me-2-S _{(O) 2 CF 3 -4-} Py], [BE5328; 5-Me-2-S (O) 2 CF 3 -4-Py], [BE5329; 6-Me-2-S (O) 2 CF 3 -4-Py], [BE 5330; 3-CF ₃ -2-S (O) ₂ CF ₃ -4-Py], [BE 5331; 5-CF ₃ -2-S (O ) ₂ CF ₃ -4-Py], [BE 5332; 6-CF ₃ -2-S (O) ₂ CF ₃ -4-Py], [BE 5333; 3-CN-2-S (O) ₂ CF _3- 4-Py], [BE5334; 5-CN-2-S (O) 2 CF 3 -4-Py], [BE5335; 6-CN-2-S (O) 2 CF 3 -4-Py], [ BE5336; 3-OMe-2- S (O) 2 CF 3 -4-Py], [BE5337; 5-OMe-2-S (O) 2 CF 3 -4-Py], [BE5338; 6-OMe- _{2-S (O) 2 CF} 3 -4-Py], [BE5339; 5-S (O) 2 CF 3 -4-Py], [BE5340; 3-Cl-5-S (O) 2 CF 3 - 4-Py], [BE5341; 2-Cl-5-S (O) 2 CF 3 -4-Py], [BE5342; 6-Cl-5-S (O) 2 CF 3 -4-Py], [ BE5343; 3-Me-5- S (O) 2 CF 3 -4-Py], [BE5344; 2-Me-5-S (O) 2 CF 3 -4-Py], [BE5345; 6-Me- _{5-S (O) 2 CF} 3 -4-Py], [BE5346; 3-CF 3 -5-S (O) 2 CF 3 -4-Py], [BE5347; 2-CF 3 -5-S ( O) ₂ CF ₃ -4-Py], [BE 5348; 6-CF ₃ -5-S (O) ₂ CF ₃ -4-Py], [BE 5 349; 3-CN-5-S (O) ₂ CF ₃ -4-Py], [BE 5350; 2-CN-5-S (O) ₂ CF ₃ -4-Py], [BE 5351; 6-CN-5-S (O) ₂ CF ₃ -4-Py], [BE5352; 3-OMe-5 -S (O) 2 CF 3 -4-Py], [BE5353; 2-OMe-5-S (O) 2 CF 3 -4-Py], [BE5354; 6-OMe _{-5-S (O) 2 CF} 3 -4-Py], [BE5355; 6-S (O) 2 CF 3 -4-Py], [BE5356; 3-Cl-6-S (O) 2 CF 3 -4-Py], [BE5357; 2-Cl-6-S (O) 2 CF 3 -4-Py], [BE5358; 5-Cl-6-S (O) 2 CF 3 -4-Py], [BE5359; 3-Me-6 -S (O) 2 CF 3 -4-Py], [BE5360; 2-Me-6-S (O) 2 CF _{3 -4-Py], [BE5361} ; 5-Me-6-S (O) 2 CF 3 -4-Py], [BE5362; 3-CF 3 -6-S (O) 2 CF 3 -4-Py ], [BE5363; 2-CF 3 -6-S (O) 2 CF 3 -4-Py], [BE5364; 5-CF 3 -6-S (O) 2 CF 3 -4-Py], [BE5365 ; 3-CN-6-S (O) 2 CF 3 -4-Py], [BE5366; 2-CN-6-S (O) 2 CF 3 -4-Py], [BE5367; 5-CN-6 _{-S (O) 2 CF 3 -4} -Py], [BE5368; 3-OMe-6-S (O) 2 CF 3 -4-Py], [BE5369; 2-OMe-6-S (O) 2 _{CF 3 -4-Py], [} BE5370; 5-OMe-6-S (O) 2 CF 3 -4-Py], [BE5371; 3-CN-4-Py], [BE5372; 2-Cl-3 -CN-4-Py], [BE5373; 5-Cl-3-CN-4-Py], [BE5374; 6-Cl-3-CN-4-Py], [BE5375; 2-Me-3-CN -4-Py], [BE5376; 5-Me-3-CN-4-Py], [BE5377; 6-Me-3-CN-4-Py], [BE5378; 2-CF 3 -3-CN- 4-Py], [BE5379; 5-CF 3 -3-CN-4-Py], [BE5380; 6-CF 3 -3-CN-4-Py], [BE5381; 2-CN-3-CN- 4-Py], [BE5382; 5-CN-3-CN-4-Py], [BE5383; 6-CN-3-CN-4-Py], [BE5384; 2-OMe-3-CN-4-] Py], [BE5385; 5-OMe-3-CN-4-Py], [BE5386; 6-OMe-3-CN-4-Py], [BE5387; 2-CN-4-Py], [BE5388; 3-Cl-2-CN-4-Py !, [BE5389; 5-Cl-2-CN-4-Py], [BE5390; 6-Cl-2-CN-4-Py], [BE5391; 3- Me-2-CN-4- Py], [BE5392; 5-Me-2-CN-4-Py], [BE5393; 6-Me-2-CN-4-Py], [BE5394; 3-CF 3 -2-CN-4-Py] , [BE5395; 5-CF 3 -2-CN-4-Py], [BE5396; 6-CF 3 -2-CN-4-Py], [BE 5397; 3-CN-2-CN-4-Py], [BE5398; 5-CN-2-CN-4-Py], [BE5399; 6-CN-2-CN-4-Py], [BE5400; 3-OMe-2-CN-4-Py], [BE5401; 5-OMe-2-CN-4-Py],

[BE5402; 6-OMe-2-CN-4-Py], [BE5403; 5-CN-4-Py], [BE5404; 3-Cl-5-CN-4-Py], [BE5405; -5-CN-4-Py !, [BE5406; 6-Cl-5-CN-4-Py], [BE5407; 3-Me-5-CN-4-Py], [BE5408; 2-Me-5 -CN-4-Py], [ BE5409; 6-Me-5-CN-4-Py], [BE5410; 3-CF 3 -5-CN-4-Py], [BE5411; 2-CF 3 -5 -CN-4-Py], [ BE5412; 6-CF 3 -5-CN-4-Py], [BE5413; 3-CN-5-CN-4-Py], [BE5414; 2-CN-5- CN-4-Py], [BE5415; 6-CN-5-CN-4-Py], [BE5416; 3-OMe-5-CN-4-Py], [BE5417; 2-OMe-5-CN- 4-Py], [BE5418; 6-OMe-5-CN-4-Py], [BE5419; 6-CN-4-Py], [BE5420; 3-Cl-6-CN-4-Py], [BE5 419; BE 5421; 2-Cl-6-CN-4-Py], [BE 5422; 5-Cl-6-CN-4-Py], [BE 5423; 3-Me-6-CN-4-Py], [BE 5424; 2-Me-6-CN- 4-Py], [BE5425; 5-Me-6-CN-4-Py], [BE5426; 3-CF 3 -6-CN-4-Py], [BE5427; 2 _{-CF 3 -6-CN-4-} Py], [BE5428; 5-CF 3 -6-CN-4-Py], [BE5429; 3-CN-6-CN-4-Py], [BE5430; 2 -CN-6-CN-4-Py], [BE5431; 5-CN-6-CN-4-Py], [BE5432; 3-OMe-6-CN-4-Py], [BE5433; 2-OMe -6-CN-4-Py !, [BE 5434; 5-OMe-6-CN-4-Py], [BE 5435; 3-COOMe-4-Py], [BE 5436; 2-Cl-3-COOMe-4 -Py], [BE5437; 5-Cl-3-COOMe-4-Py], [BE5438; 6-Cl-3-COOMe-4-Py], [BE5439; 2-Me-3-COOMe-4-Py ], [BE 5440; 5-Me-3-COOMe-4-Py], [BE5441; 6-Me-3-COOMe-4-Py], [BE5442; 2] _{-CF 3 -3-COOMe-4-} Py], [BE5443; 5-CF 3 -3-COOMe-4-Py], [BE5444; 6-CF 3 -3-COOMe-4-Py], [BE5445; 2-CN-3-COOMe-4-Py], [BE5446; 5-CN-3-COOMe-4-Py], [BE5447; 6-CN-3-COOMe-4-Py], [BE5448; OMe-3-COOMe-4-Py], [BE5449; 5-OMe-3-COOMe-4-Py], [BE5450; 6-OMe-3-COOMe-4-Py], [BE5451; 2-COOMe- 4-Py], [BE5452; 3-Cl-2-COOMe-4-Py], [BE5453; 5-Cl-2-COOMe-4-Py], [BE5454; 6-Cl-2-COOMe-4-] Py], [BE5455; 3-Me-2-COOMe-4-Py], [BE5456; 5-Me-2-COOMe-4-Py], [BE5457; 6-Me-2-COOMe-4-Py] _{, [BE5458; 3-CF 3} -2-COOMe-4-Py], [BE5459; 5-CF 3 -2-COOMe-4-Py], [BE5460; 6-CF 3 -2-COOMe-4-Py ], [BE5461; 3-CN-2-COOMe-4-Py], [BE5462; 5-CN-2-COOMe-4-Py], [BE5463; 6-CN-2-COOMe-4-Py], [BE5464; 3-OMe-2-COOMe-4-Py], [BE5465; 5-OMe-2-COOMe-4-Py], [BE5466; 6-OMe-2-COOMe-4-Py], [BE5467] 5-COOMe-4-Py !, [BE5468; 3-Cl-5-COOMe-4-Py], [BE5469; 2-Cl-5-COOMe-4-Py], [BE5470; 6-Cl-5; -COOMe-4-Py], [BE5471; 3-Me-5-COOMe-4-Py], [BE5472; 2-Me-5-COOMe-4-Py], [BE5473; 6-Me-5-COOMe -4-Py], [BE5474; 3-CF 3 -5-COOMe-4-Py], [BE5475; 2-CF 3 -5-COOMe-4-Py], [BE5476; 6-CF 3 -5- COOMe-4-Py], [BE5477; 3-CN-5-COOMe-4-Py], [BE5478; 2-CN-5 -COOMe-4-Py], [BE5479; 6-CN-5-COOMe-4-Py], [BE5480; 3-OMe-5-COOMe-4-Py], [BE5481; 2-OMe-5-COOMe -4-Py], [BE5482; 6-OMe-5-COOMe-4-Py], [BE5483; 6-COOMe-4-Py], [BE5484; 3-Cl-6-COOMe-4-Py], [BE5485; 2-Cl-6-COOMe-4-Py], [BE5486; 5-Cl-6-COOMe-4-Py], [BE5487; 3-Me-6-COOMe-4-Py], [BE5488] ; 2-Me-6-COOMe -4-Py], [BE5489; 5-Me-6-COOMe-4-Py], [BE5490; 3-CF 3 -6-COOMe-4-Py], [BE5491; _{2-CF 3 -6-COOMe-} 4-Py], [BE5492; 5-CF 3 -6-COOMe-4-Py], [BE5493; 3-CN-6-COOMe-4-Py], [BE5494; 2-CN-6-COOMe-4-Py], [BE5495; 5-CN-6-COOMe-4-Py], [BE5496; 3-OMe-6-COOMe-4-Py], [BE5497; OMe-6-COOMe-4- Py], [BE5498; 5-OMe-6-COOMe-4-Py], [BE5499; 3-NO 2 -4-Py], [BE5500; 2-Cl-3-NO ₂ -4-Py], [BE 5501; 5-Cl-3-NO ₂ -4-Py],

[BE5502; 6-Cl-3 -NO 2 -4-Py], [BE5503; 2-Me-3-NO 2 -4-Py], [BE5504; 5-Me-3-NO 2 -4-Py] , [BE5505; 6-Me- 3-NO 2 -4-Py], [BE5506; 2-CF 3 -3-NO 2 -4-Py], [BE5507; 5-CF 3 -3-NO 2 -4 -Py], [BE5508; 6- CF 3 -3-NO 2 -4-Py], [BE5509; 2-CN-3-NO 2 -4-Py], [BE5510; 5-CN-3-NO 2 -4-Py], [BE5511; 6-CN-3-NO 2 -4-Py], [BE5512; 2-OMe-3-NO 2 -4-Py], [BE5513; 5-OMe-3-NO _{2 -4-Py], [BE5514} ; 6-OMe-3-NO 2 -4-Py], [BE5515; 2-NO 2 -4-Py], [BE5516; 3-Cl-2-NO 2 -4 -Py], [BE5517; 5- Cl-2-NO 2 -4-Py], [BE5518; 6-Cl-2-NO 2 -4-Py], [BE5519; 3-Me-2-NO 2 - 4-Py], [BE5520; 5-Me-2-NO 2 -4-Py], [BE5521; 6-Me-2-NO 2 -4-Py], [BE5522; 3-CF 3 -2-NO ₂ -4-Py], [BE 5523; 5-CF ₃ -2-NO ₂ -4-Py], [BE 5524; 6-CF ₃ -2-NO ₂ -4-Py], [BE 5525; 3-CN- _{2-NO 2 -4-Py]} , [BE5526; 5-CN-2-NO 2 -4-Py], [BE5527; 6-CN-2-NO 2 -4-Py], [BE5528; 3-OMe _{-2-NO 2 -4-Py]} , [BE5529; 5-OMe-2-NO 2 -4-Py], [BE5530; 6-OMe-2-NO 2 -4-Py], [BE5531; 5- _{NO 2 -4-Py], [} BE5532; 3-Cl-5-NO 2 -4-Py], [BE5533; 2-Cl-5-NO 2 -4-Py], [BE5534; 6-Cl-5 _{-NO 2 -4-Py], [} BE5535; 3-Me-5-NO 2 -4-Py], [BE5536; 2-Me-5-NO 2 -4-Py], [BE5537; 6-Me- 5-NO ₂ -4-Py], [BE 5538; 3-CF ₃ -5-NO ₂ -4-Py], [BE 5539; 2-CF ₃ -5-NO ₂ -4-Py], [BE 5540; 6-CF ₃ -5-NO ₂ -4-Py], [BE 554 1; _{3-CN-5-NO 2} -4-Py], [BE5542; 2-CN-5-NO 2 -4-Py], [BE5543; 6-CN-5-NO 2 -4-Py], [BE5544 ; 3-OMe-5-NO 2 -4-Py], [BE5545; 2-OMe-5-NO 2 -4-Py], [BE5546; 6-OMe-5-NO 2 -4-Py], [ _{BE5547; 6-NO 2 -4-} Py], [BE5548; 3-Cl-6-NO 2 -4-Py], [BE5549; 2-Cl-6-NO 2 -4-Py], [BE5550; 5 _{-Cl-6-NO 2 -4-} Py], [BE5551; 3-Me-6-NO 2 -4-Py], [BE5552; 2-Me-6-NO 2 -4-Py], [BE5553; _{5-Me-6-NO 2} -4-Py], [BE5554; 3-CF 3 -6-NO 2 -4-Py], [BE5555; 2-CF 3 -6-NO 2 -4-Py], _{[BE5556; 5-CF 3 -6} -NO 2 -4-Py], [BE5557; 3-CN-6-NO 2 -4-Py], [BE5558; 2-CN-6-NO 2 -4-Py ], [BE5559; 5-CN -6-NO 2 -4-Py], [BE5560; 3-OMe-6-NO 2 -4-Py], [BE5561; 2-OMe-6-NO 2 -4- Py], [BE5562; 5- OMe-6-NO 2 -4-Py], [BE5563; 3-NH 2 -4-Py], [BE5564; 2-Cl-3-NH 2 -4-Py], [BE5565; 5-Cl-3 -NH 2 -4-Py], [BE5566; 6-Cl-3-NH 2 -4-Py], [BE5567; 2-Me-3-NH 2 -4-Py] , [BE5568; 5-Me- 3-NH 2 -4-Py], [BE5569; 6-Me-3-NH 2 -4-Py], [BE5570; 2-CF 3 -3-NH 2 -4- Py], [BE5571; 5- CF 3 -3-NH 2 -4-Py], [BE5572; 6-CF 3 -3-NH 2 -4-Py], [BE5573; 2-CN-3-NH 2 -4-Py], [BE 5574; 5-CN-3-NH ₂ -4-Py], [BE5575; 6-CN-3-NH 2 -4-Py], [BE5576; 2-OMe-3-NH 2 -4-Py], [BE5577; 5-OMe-3-NH ₂ -4-Py], [BE 5578; 6-OMe-3-NH ₂ -4-Py], [BE 5579; 2-NH ₂ -4-Py], [BE 5580; 3-Cl-2-NH _2-4 -Py], [BE5581; 5- Cl-2-NH 2 -4-Py], [BE5582; 6-Cl-2-NH 2 -4-Py], [BE5583; 3-Me-2-NH 2 - 4-Py], [BE5584; 5-Me-2-NH 2 -4-Py], [BE5585; 6-Me-2-NH 2 -4-Py], [BE5586; 3-CF 3 -2-NH ₂ -4-Py], [BE 5587; 5-CF ₃ -2-NH ₂ -4-Py], [BE 5588; 6-CF ₃ -2-NH ₂ -4-Py], [BE 5589; 3-CN- _{2-NH 2 -4-Py]} , [BE5590; 5-CN-2-NH 2 -4-Py], [BE5591; 6-CN-2-NH 2 -4-Py], [BE5592; 3-OMe _{-2-NH 2 -4-Py]} , [BE5593; 5-OMe-2-NH 2 -4-Py], [BE5594; 6-OMe-2-NH 2 -4-Py], [BE5595; 5- _{NH 2 -4-Py], [} BE5596; 3-Cl-5-NH 2 -4-Py], [BE5597; 2-Cl-5-NH 2 -4-Py], [BE5598; 6-Cl-5 _{-NH 2 -4-Py], [} BE5599; 3-Me-5-NH 2 -4-Py], [BE5600; 2-Me-5-NH 2 -4-Py], [BE5601; 6-Me- 5-NH ₂ -4-Py],

_{[BE5602; 3-CF 3 -5} -NH 2 -4-Py], [BE5603; 2-CF 3 -5-NH 2 -4-Py], [BE5604; 6-CF 3 -5-NH 2 -4 -Py], [BE5605; 3- CN-5-NH 2 -4-Py], [BE5606; 2-CN-5-NH 2 -4-Py], [BE5607; 6-CN-5-NH 2 - 4-Py], [BE5608; 3-OMe-5-NH 2 -4-Py], [BE5609; 2-OMe-5-NH 2 -4-Py], [BE5610; 6-OMe-5-NH 2 -4-Py], [BE 5611; 6-NH ₂ -4-Py], [BE 5612; 3-Cl-6-NH ₂ -4-Py], [BE 5613; 2-Cl-6-NH ₂ -4- Py], [BE5614; 5- Cl-6-NH 2 -4-Py], [BE5615; 3-Me-6-NH 2 -4-Py], [BE5616; 2-Me-6-NH 2 -4 -Py], [BE 5617; 5-Me-6-NH ₂ -4-Py], [BE 5618; 3-CF ₃ -6-NH ₂ -4-Py], [BE 5619; 2-CF ₃ -6-NH] _{2 -4-Py], [BE5620} ; 5-CF 3 -6-NH 2 -4-Py], [BE5621; 3-CN-6-NH 2 -4-Py], [BE5622; 2-CN-6 _{-NH 2 -4-Py], [} BE5623; 5-CN-6-NH 2 -4-Py], [BE5624; 3-OMe-6-NH 2 -4-Py], [BE5625; 2-OMe- _{6-NH 2 -4-Py]} , [BE5626; 5-OMe-6-NH 2 -4-Py], [BE5627; 3-NHMe-4-Py], [BE5628; 2-Cl-3-NHMe- 4-Py], [BE5629; 5-Cl-3-NHMe-4-Py], [BE5630; 6-Cl-3-NHMe-4-Py], [BE5631; 2-Me-3-NHMe-4- Py], [BE5632; 5- Me-3-NHMe-4-Py], [BE5633; 6-Me-3-NHMe-4-Py], [BE5634; 2-CF 3 -3-NHMe-4-Py ], [BE5635; 5-CF 3 -3-NHMe-4-Py], [BE5636; 6-CF 3 -3-NHMe-4-Py], [BE5637; 2-CN-3-NHMe-4-Py ], [BE 5638; 5-CN-3-N HMe-4-Py], [BE5639; 6-CN-3-NHMe-4-Py], [BE5640; 2-OMe-3-NHMe-4-Py], [BE5641; 5-OMe-3-NHMe- 4-Py], [BE5642; 6-OMe-3-NHMe-4-Py], [BE5643; 2-NHMe-4-Py], [BE5644; 3-Cl-2-NHMe-4-Py], [BE 564] BE 5645; 5-Cl-2-NHMe-4-Py], [BE 5646; 6-Cl-2-NHMe-4-Py], [BE 5647; 3-Me-2-NHMe-4-Py], [BE 5648; 5-Me-2-NHMe- 4-Py], [BE5649; 6-Me-2-NHMe-4-Py], [BE5650; 3-CF 3 -2-NHMe-4-Py], [BE5651; 5 _{-CF 3 -2-NHMe-4-} Py], [BE5652; 6-CF 3 -2-NHMe-4-Py], [BE5653; 3-CN-2-NHMe-4-Py], [BE5654; 5 -CN-2-NHMe-4-Py], [BE5655; 6-CN-2-NHMe-4-Py], [BE5656; 3-OMe-2-NHMe-4-Py], [BE5657; 5-OMe -2-NHMe-4-Py, [BE5658; 6-OMe-2-NHMe-4-Py], [BE 5659; 5-NHMe-4-Py], [BE 5660; 3-Cl-5-NHMe-4 -Py], [BE5661; 2-Cl-5-NHMe-4-Py], [BE5662; 6-Cl-5-NHMe-4-Py], [BE5663; 3-Me-5-NHMe-4-Py ], [BE5664; 2-Me -5-NHMe-4-Py], [BE5665; 6-Me-5-NHMe-4-Py], [BE5666; 3-CF 3 -5-NHMe-4-Py] _{, [BE5667; 2-CF 3} -5-NHMe-4-Py], [BE5668; 6-CF 3 -5-NHMe-4-Py], [BE5669; 3-CN-5-NHMe-4-Py] , [BE5670; 2-CN-5-NHMe-4-Py], [BE5671; 6-CN-5-NHMe-4-Py], [BE5672; 3-OMe-5-NHMe-4-Py], [BE5672; BE 5673; 2-OMe-5-NHMe-4-Py], [BE 5674; 6-OMe-5-NHMe-4-Py], [BE 5675; 6-NHMe-4-Py], [BE 5676; 3-Cl- 6-N HMe-4-Py], [BE5677; 2-Cl-6-NHMe-4-Py], [BE5678; 5-Cl-6-NHMe-4-Py], [BE5679; 3-Me-6-NHMe- 4-Py], [BE5680; 2-Me-6-NHMe-4-Py], [BE5681; 5-Me-6-NHMe-4-Py], [BE5682; 3-CF 3 -6-NHMe-4 -Py], [BE5683; 2- CF 3 -6-NHMe-4-Py], [BE5684; 5-CF 3 -6-NHMe-4-Py], [BE5685; 3-CN-6-NHMe-4 -Py], [BE5686; 2-CN-6-NHMe-4-Py], [BE5687; 5-CN-6-NHMe-4-Py], [BE5688; 3-OMe-6-NHMe-4-Py ], [BE5689; 2-OMe -6-NHMe-4-Py], [BE5690; 5-OMe-6-NHMe-4-Py], [BE5691; 3-NMe 2 -4-Py], [BE5692; _{2-Cl-3-NMe 2} -4-Py], [BE5693; 5-Cl-3-NMe 2 -4-Py], [BE5694; 6-Cl-3-NMe 2 -4-Py], [BE5695 ; 2-Me-3-NMe 2 -4-Py], [BE5696; 5-Me-3-NMe 2 -4-Py], [BE5697; 6-Me-3-NMe 2 -4-Py], [ _{BE5698; 2-CF 3 -3-} NMe 2 -4-Py], [BE5699; 5-CF 3 -3-NMe 2 -4-Py], [BE5700; 6-CF 3 -3-NMe 2 -4- Py], [BE5701; 2- CN-3-NMe 2 -4-Py],

[BE5702; 5-CN-3 -NMe 2 -4-Py], [BE5703; 6-CN-3-NMe 2 -4-Py], [BE5704; 2-OMe-3-NMe 2 -4-Py] , [BE5705; 5-OMe- 3-NMe 2 -4-Py], [BE5706; 6-OMe-3-NMe 2 -4-Py], [BE5707; 4-NMe 2 -4-Py], [BE5708 ; 3-Cl-4-NMe 2 -4-Py], [BE5709; 5-Cl-4-NMe 2 -4-Py], [BE5710; 6-Cl-4-NMe 2 -4-Py], [ BE5711; 3-Me-4- NMe 2 -4-Py], [BE5712; 5-Me-4-NMe 2 -4-Py], [BE5713; 6-Me-4-NMe 2 -4-Py], _{[BE5714; 3-CF 3 -4} -NMe 2 -4-Py], [BE5715; 5-CF 3 -4-NMe 2 -4-Py], [BE5716; 6-CF 3 -4-NMe 2 -4 -Py], [BE5717; 3- CN-4-NMe 2 -4-Py], [BE5718; 5-CN-4-NMe 2 -4-Py], [BE5719; 6-CN-4-NMe 2 - 4-Py], [BE5720; 3-OMe-4-NMe 2 -4-Py], [BE5721; 5-OMe-4-NMe 2 -4-Py], [BE5722; 6-OMe-4-NMe 2 -4-Py], [BE5723; 5-NMe 2 -4-Py], [BE5724; 3-Cl-5-NMe 2 -4-Py], [BE5725; 2-Cl-5-NMe 2 -4- Py], [BE5726; 6- Cl-5-NMe 2 -4-Py], [BE5727; 3-Me-5-NMe 2 -4-Py], [BE5728; 2-Me-5-NMe 2 -4 -Py], [BE5729; 6- Me-5-NMe 2 -4-Py], [BE5730; 3-CF 3 -5-NMe 2 -4-Py], [BE5731; 2-CF 3 -5-NMe ₂ -4-Py], [BE 5732; 6-CF ₃ -5-NMe ₂ -4-Py], [BE 5733; 3-CN-5-NMe ₂ -4-Py], [BE 5 734; 2-CN-5 _{-NMe 2 -4-Py], [} BE5735; 6-CN-5-NMe 2 -4-Py], [BE5736; 3-OMe-5-NMe 2 -4-Py], [BE57 37; 2-OMe-5- NMe 2 -4-Py], [BE5738; 6-OMe-5-NMe 2 -4-Py], [BE5739; 6-NMe 2 -4-Py], [BE5740; 3 _{-Cl-6-NMe 2 -4-} Py], [BE5741; 2-Cl-6-NMe 2 -4-Py], [BE5742; 5-Cl-6-NMe 2 -4-Py], [BE5743; _{3-Me-6-NMe 2} -4-Py], [BE5744; 2-Me-6-NMe 2 -4-Py], [BE5745; 5-Me-6-NMe 2 -4-Py], [BE5746 _{; 3-CF 3 -6-NMe} 2 -4-Py], [BE5747; 2-CF 3 -6-NMe 2 -4-Py], [BE5748; 5-CF 3 -6-NMe 2 -4-Py ], [BE5749; 3-CN -6-NMe 2 -4-Py], [BE5750; 2-CN-6-NMe 2 -4-Py], [BE5751; 5-CN-6-NMe 2 -4- Py], [BE5752; 3- OMe-6-NMe 2 -4-Py], [BE5753; 2-OMe-6-NMe 2 -4-Py], [BE5754; 5-OMe-6-NMe 2 -4 -Py], [BE5755; 3-ACNH-4-Py], [BE5756; 2-Cl-3-ACNH-4-Py], [BE5757; 5-Cl-3-ACNH-4-Py], [BE5758] 6-Cl-3-ACNH-4-Py !, [BE5759; 2-Me-3-ACNH-4-Py], [BE5760; 5-Me-3-ACNH-4-Py], [BE5761; -Me-3-ACNH-4- Py], [BE5762; 2-CF 3 -3-ACNH-4-Py], [BE5763; 5-CF 3 -3-ACNH-4-Py], [BE5764; 6 _{-CF 3 -3-ACNH-4-} Py], [BE5765; 2-CN-3-ACNH-4-Py], [BE5766; 5-CN-3-ACNH-4-Py], [BE5767; 6- CN-3-ACNH-4-Py, [BE5768; 2-OMe-3-ACNH-4-Py], [BE5769; 5-OMe-3-ACNH-4-Py], [BE5770; 6-OMe- 3-ACNH-4-Py, [BE5771; 2-ACNH-4-Py], [BE5772; 3-Cl-2-ACNH-4-Py], [BE5773; 5-Cl-2-ACNH-4- Py], [BE5774; 6-Cl-2-ACNH-4-Py], [BE5775; 3-Me-2-ACNH-4-Py], [BE5776; 5-Me-2-ACNH-4-Py] , [BE5777; 6-Me- 2-ACNH-4-Py], [BE5778; 3-CF 3 -2-ACNH-4-Py], [BE5779; 5-CF 3 -2-ACNH-4-Py] , [BE 5780; 6-CF ₃ 2-ACNH-4-Py], [BE 5781; 3-CN-2-ACNH-4-Py], [BE 578 2; 5-CN-2-ACNH-4-Py], [BE5783; 6-CN-2-ACNH-4-Py], [BE5784; 3-OMe-2-ACNH-4-Py], [BE 5785; 5-OMe-2-ACNH-4-Py], [BE5786] 6-OMe-2-ACNH-4-Py !, [BE5787; 5-ACNH-4-Py], [BE5788; 3-Cl-5-ACNH-4-Py], [BE5789; 2-Cl-5; -ACNH-4-Py], [BE5790; 6-Cl-5-ACNH-4-Py], [BE5791; 3-Me-5-ACNH-4-Py], [BE5792; 2-Me-5-ACNH -4-Py], [BE5793; 6-Me-5-ACNH-4-Py], [BE5794; 3-CF 3 -5-ACNH-4-Py], [BE5795; 2-CF 3 -5-ACNH -4-Py], [BE5796; 6-CF 3 -5-ACNH-4-Py], [BE5797; 3-CN-5-ACNH-4-Py], [BE5798; 2-CN-5-ACNH- 4-Py], [BE5799; 6-CN-5-ACNH-4-Py], [BE5800; 3-OMe-5-ACNH-4-Py], [BE5801; 2-OMe-5-ACNH-4- Py],

[BE 5802; 6-OMe-5-ACNH-4-Py], [BE 5803; 6-ACNH-4-Py], [BE 5804; 3-Cl-6-ACNH-4-Py], [BE 5805; 2-Cl -6-ACNH-4-Py], [BE5806; 5-Cl-6-ACNH-4-Py], [BE5807; 3-Me-6-ACNH-4-Py], [BE5808; 2-Me-6 -ACNH-4-Py], [ BE5809; 5-Me-6-ACNH-4-Py], [BE5810; 3-CF 3 -6-ACNH-4-Py], [BE5811; 2-CF 3 -6 -ACNH-4-Py], [ BE5812; 5-CF 3 -6-ACNH-4-Py], [BE5813; 3-CN-6-ACNH-4-Py], [BE5814; 2-CN-6- ACNH-4-Py !, [BE5815; 5-CN-6-ACNH-4-Py], [BE5816; 3-OMe-6-ACNH-4-Py], [BE5817; 2-OMe-6-ACNH- 4-Py], [BE5818; 5-OMe-6-ACNH-4-Py], [BE5819; 3- (N (Ac) (Me))-4-Py], [BE5820; 2-Cl-3- (N (Ac) (Me))-4-Py], [BE 5821; 5-Cl-3- (N (Ac) (Me))-4-Py], [BE 5822; 6-Cl-3- (N) (Ac) (Me))-4-Py], [BE 5823; 2-Me-3- (N (Ac) (Me))-4-Py], [BE 5824; 5-Me-3- (N (Ac) ) (Me))-4-Py], [BE 5825; 6-Me-3- (N (Ac) (Me))-4-Py], [BE 5826; 2-CF ₃ -3- (N (Ac)) (Me)) - 4-Py ], [BE5827; 5-CF 3 -3- (N (Ac) (Me)) - 4-Py], [BE5828; 6-CF 3 -3- (N (Ac) (Me))-4-Py], [BE5829; 2-CN-3- (N (Ac) (Me))-4-Py], [BE5830; 5-CN-3- (N (Ac) (Me) )) 4-Py], [BE5831; 6-CN-3- (N (Ac) (Me))-4-Py], [BE5832; 2-OMe-3- (N (Ac) (Me)) -4-Py], [BE5833; 5-OMe-3- (N (Ac) (Me))-4-Py], [BE5834; 6-OMe-3- (N (Ac) (Me))-4 -Py], [BE 5835; 2- (N (Ac ) (Me))-4-Py], [BE5836; 3-Cl-2- (N (Ac) (Me))-4-Py], [BE5837; 5-Cl-2- (N (Ac) ( Me))-4-Py], [BE5838; 6-Cl-2- (N (Ac) (Me))-4-Py], [BE5839; 3-Me-2- (N (Ac) (Me)) )-[4-Py], [BE 5840; 5-Me-2- (N (Ac) (Me))-4-Py], [BE5841; 6-Me-2- (N (Ac) (Me))- 4-Py], [BE5842; 3-CF 3 -2- (N (Ac) (Me)) - 4-Py], [BE5843; 5-CF 3 -2- (N (Ac) (Me)) - 4-Py], [BE5844; 6-CF 3 -2- (N (Ac) (Me)) - 4-Py], [BE5845; 3-CN-2- (N (Ac) (Me)) - 4 -Py], [BE5846; 5-CN-2- (N (Ac) (Me))-4-Py], [BE5847; 6-CN-2- (N (Ac) (Me))-4-Py ], [BE 5848; 3-OMe-2- (N (Ac) (Me))-4-Py], [BE 5849; 5-OMe-2- (N (Ac) (Me))-4-Py], [BE5850; 6-OMe-2- (N (Ac) (Me))-4-Py], [BE5851; 5- (N (Ac) (Me))-4-Py], [BE5852; 3-Cl -5- (N (Ac) (Me))-4-Py], [BE5853; 2-Cl-5- (N (Ac) (Me))-4-Py], [BE5854; 6-Cl-5 -(N (Ac) (Me))-4-Py], [BE5855; 3-Me-5- (N (Ac) (Me))-4-Py], [BE5856; 2-Me-5- ( N (Ac) (Me)) - 4-Py], [BE5857; 6-Me-5- (N (Ac) (Me)) - 4-Py], [BE5858; 3-CF 3 -5- (N (Ac) (Me)) - 4-Py], [BE5859; 2-CF 3 -5- (N (Ac) (Me)) - 4-Py], [BE5860; 6-CF 3 -5- (N (Ac) (Me))-4-Py], [BE5861; 3-CN-5- (N (Ac) (Me))-4-Py], [BE5862; 2-CN-5- (N (Ac) ) (Me))-4-Py], [BE5863; 6-CN-5- (N (Ac) (Me))-4-Py], [BE5864; 3-OMe-5- (N (Ac) ( Me))-4-Py], [BE 5865; 2-OMe -5- (N (Ac) (Me))-4-Py], [BE5866; 6-OMe-5- (N (Ac) (Me))-4-Py], [BE5867; 6- (N ( Ac) (Me))-4-Py], [BE5868; 3-Cl-6- (N (Ac) (Me))-4-Py], [BE5869; 2-Cl-6- (N (Ac)) (Me))-4-Py], [BE5870; 5-Cl-6- (N (Ac) (Me))-4-Py], [BE5871; 3-Me-6- (N (Ac) (Me) )) 4-Py], [BE 5872; 2-Me-6- (N (Ac) (Me))-4-Py], [BE 5873; 5-Me-6- (N (Ac) (Me)) -4-Py], [BE 5874; 3-CF ₃ -6- (N (Ac) (Me))-4-Py], [BE 5875; 2-CF ₃ -6- (N (Ac) (Me)) -4-Py], [BE5876; 5-CF 3 -6- (N (Ac) (Me)) - 4-Py], [BE5877; 3-CN-6- (N (Ac) (Me)) - 4-Py], [BE5878; 2-CN-6- (N (Ac) (Me))-4-Py], [BE5879; 5-CN-6- (N (Ac) (Me))-4- Py], [BE 5880; 3-OMe-6- (N (Ac) (Me))-4-Py], [BE 5881; 2-OMe-6- (N (Ac) (Me))-4-Py] , [BE 5882; 5-OMe-6- (N (Ac) (Me))-4-Py], [BE 5883; 3-AC-4-Py], [BE 5884; 2-Cl-3-AC-4- Py], [BE 5885; 5-Cl-3-AC-4-Py], [BE 5886; 6-Cl-3-AC-4-Py], [BE 5887; 2-Me-3-AC-4-Py] , [BE5888; 5-Me-3-AC-4-Py], [BE 5889; 6-Me-3-AC-4-Py], [BE 5890; 2-CF ₃ -3-AC-4-Py], _{[BE5891; 5-CF 3 -3} -AC-4-Py], [BE5892; 6-CF 3 -3-AC-4-Py], [BE5893; 2-CN-3-AC-4-Py], [BE5894; 5-CN-3-AC-4-Py], [BE5895; 6-CN-3-AC-4-Py], [BE5896; 2-OMe-3-AC-4-Py], [BE5897 5-OMe-3-AC-4-Py !, [BE 5898; 6-OMe-3-AC-4-Py], [BE5899; 2-AC-4-Py], [BE5900; 3-Cl-2-AC-4-Py], [BE5901; 5-Cl-2-AC-4-Py],

[BE5902; 6-Cl-2-AC-4-Py], [BE5903; 3-Me-2-AC-4-Py], [BE5904; 5-Me-2-AC-4-Py], [BE5905] ; 6-Me-2-AC -4-Py], [BE5906; 3-CF 3 -2-AC-4-Py], [BE5907; 5-CF 3 -2-AC-4-Py], [BE5908 _{; 6-CF 3 -2-AC} -4-Py], [BE5909; 3-CN-2-AC-4-Py], [BE5910; 5-CN-2-AC-4-Py], [BE5911; 6-CN-2-AC-4-Py, [BE5912; 3-OMe-2-AC-4-Py], [BE5913; 5-OMe-2-AC-4-Py], [BE5914; 6- OMe-2-AC-4-Py], [BE5915; 5-AC-4-Py], [BE5916; 3-Cl-5-AC-4-Py], [BE5917; 2-Cl-5-AC- 4-Py], [BE5918; 6-Cl-5-AC-4-Py], [BE5919; 3-Me-5-AC-4-Py], [BE5920; 2-Me-5-AC-4- 4 Py], [BE5921; 6- Me-5-AC-4-Py], [BE5922; 3-CF 3 -5-AC-4-Py], [BE5923; 2-CF 3 -5-AC-4- Py], [BE5924; 6- CF 3 -5-AC-4-Py], [BE5925; 3-CN-5-AC-4-Py], [BE5926; 2-CN-5-AC-4-Py ], [BE5927; 6-CN-5-AC-4-Py], [BE5928; 3-OMe-5-AC-4-Py], [BE5929; 2-OMe-5-AC-4-Py], [BE 5930; 6-OMe-5-AC-4-Py], [BE 5931; 6-AC-4-Py], [BE 5932; 3-Cl-6-AC-4-Py], [BE 5933; 2-Cl -6-AC-4-Py], [BE5934; 5-Cl-6-AC-4-Py], [BE5935; 3-Me-6-AC-4-Py], [BE5936; 2-Me-6 -AC-4-Py], [ BE5937; 5-Me-6-AC-4-Py], [BE5938; 3-CF 3 -6-AC-4-Py], [BE5939; 2-CF 3 -6 -AC-4-Py], [ BE5940; 5-CF 3 -6-AC-4-Py], [BE5941; 3-CN-6-AC-4-Py], [BE5942; 2-CN-6- AC -4-Py], [BE5943; 5-CN-6-AC-4-Py], [BE 5944; 3-OMe-6-AC-4-Py], [BE5945; 2-OMe-6-AC-4 -Py], [BE5946; 5-OMe-6-AC-4-Py], [BE5947; 1,2- (methylenedioxy) phenyl-4-yl], [BE5948; 2,3-dihydrobenzofuran-5] -Yl], [BE 5949; 2,3-dihydrobenzofuran-6-yl], [BE 5950; 1,3-dihydroisobenzofuran-5-yl], [BE 5951; benzofuran-5-yl], [BE 5952; benzofuran- 6-yl], [BE 595 3; 2,3-dihydrobenzothiophen-5-yl], [BE 595 4; 2,3-dihydrobenzothiophen-6-yl], [BE 5 955; 1,3-dihydroisobenzothiophene 5 -Yl], [BE 5956; benzothiophen-5-yl], [BE 5957; benzothiophen-6-yl], [BE 5958; benzodioxan-4-yl], [BE 5959; chroman-6-yl], [BE 5960; Chroman-7-yl], [BE 5961; isochroman-6-yl], [BE 5962; isochroman-7-yl], [BE 5963; 2-quinolyl], [BE 5964; 3-quinolyl], [BE 5 965; Methylenedioxyphenyl], [BE 5966; 2-indolyl], [ BE5967; 3-indolyl], [BE 5968; 2-benzoimidazolyl], [BE 5969; 2-thienyl], [BE 5970; 3-thienyl], [BE 5971; 2,3-dihydrobenzofuran-7-yl], [BE 5972; 2 -Pyrimidyl], [BE 5973; 5-Pyrimidyl], [BE 5 974; 2-thiazolyl], [BE 5 975; 4-thiazolyl], [BE 5976; 5-thiazolyl], [BE 5977; [BE5979; 2-benzoxazolyl], [BE5980; 2-benzothiazolyl], [BE5981; 2-quinazolyl], [BE5982; 2-quinoxalyl], [BE5983; phenyl], [BE5984; 2-fluorophenyl], [BE5983; BE5985; 3-fluoroPh], [BE5986; 4-fluoroPh], [BE5987; 2,4-difluorophenyl], [BE5988; 2,4,6-trifluorophenyl], [BE5989; 2,3,4,5,6- 2-fluorophenyl], [BE5992; 2-chlorophenyl], [BE5992; 3-chlorophenyl], [BE5993; 3-chlorophenyl], [BE5994; 2-3-dichlorophenyl], [BE5995; 2,4-dichlorophenyl], [BE5996; 2,5-dichlorophenyl], [BE5997; 2,6-dichlorophenyl], [BE5998; 3,4-dichlorophenyl], [BE5999; 3,5-dichlorophenyl], [BE6000; 2,3,4-trichlorophenol], [BE6001; 2,3,5-trichlorophenyl], [BE6002; 3,6-trichlorophenyl], [BE6003; 2,4,5-trichlorophenyl], [BE6004; 2,4,6-trichlorophenyl], [BE6005; 3,4,5-trichlorophenyl], [BE6006; 4,6-tetrachlorophenyl], [BE6007; 2,3,5,6-tetrachlorophenyl], [BE6008; 2,3,4,5,6-pentachlorophenyl], [BE6009; 2-bromophenyl], [BE6010; 3- bromophenyl], [BE6011; 4-bromophenyl], [BE6012; 2,4-dibromophenyl], [BE6013; 2,5-dibromophenyl], [BE6014; 2,6-dibromophenyl], [BE6015; 2,4,6- tribromophenyl], [BE6016; 2,3,4,5,6-pentabromophenyl], [BE6017; 2-iodophenyl], [BE6018; 3-iodophenyl], [BE6019; 4-iodophenyl], [BE6020; 2-chloro-3-fluorophenyl], [BE 60 22; 2-chloro-4-fluorophenyl], [BE 60 23; 2-chloro-5-fluorophenyl], [BE 60 24; 2-chloro-6-fluorophenyl] [BE 6025; 2-chloro-3-bromophenyl], [BE 6026; 2-chloro-4-bromophenyl], [BE 6027; 2-chloro-5-bromophenyl], [BE 6028; 2-chloro-6-bromophenyl], [BE 60 25 BE6029; 2-bromo-3-chlorophenyl], [BE6030; 2-bromo-4-chlorophenyl], [BE6031; 2-bromo-5-chlorophenyl], [BE6032; 2-bromo-3-fluorophenyl], [BE6033; 2-bromo-4-fluorophenyl, [BE6034; 2-bromo-5-fluorophenyl], [BE6035; 2-bromo-6-f luorophenyl], [BE6036; 2-fluoro-3-chlorophenyl], [BE6037; 2-fluoro-4-chlorophenyl], [BE6038; 2-fluoro-5-chlorophenyl], [BE6039; 2-fluoro-4-bromophenyl] [BE 6040; 3-chloro 4-fluorophenyl], [BE 6041; 3-chloro-5-fluorophenyl], [BE 6042; 3-chloro-4-bromophenyl], [BE 6043; 3-chloro-5-bromophenyl], [BE 6044; 3-fluoro-4-chlorophenyl], [BE 6045; 3-fluoro-4-bromophenyl], [BE 6046; 3-bromo-4-chlorophenyl], [BE 6047; 3-bromo-4-fluorophenyl], [BE 6048; 6-dichloro-4-bromophenyl], [BE6049; 2-3-difluoro-4-chlorophenyl], [BE6050; 2,6-difluoro-4-chlorophenyl], [BE6051; 2,5-difluoro-4-chlorophenyl] , [BE 6052; 3,5-difluoro-4-chlorophenyl], [BE 6053; 2, 3, 5-trifluoro-4-chlorophenyl], [BE 6054; 2, 3, 6-trifluoro-4-chlorophenyl], [BE 6055; 2,3,5,6-tetrafluoro-4-chlorophenyl], [BE 6056; 2-fluoro-4-bromophenyl], [BE 6057; 2-3-difluoro-4-bromophenyl], [BE 6058; 2, 6-difluoro- 4-bromophenyl], [BE6059; 2,5-difluoro-4-bromophenyl], [BE6060; 3,5-difluoro-4-bromophenyl], [BE6061; 2,3,5-trifluoro-4-bromophenyl], [BE6061] BE6062; 2,3,6-trifluoro-4-bromophenyl], [BE6063; 2,3,5,6-tetrafluoro-4-bromop 2-fluoro-4-iodophenyl], [BE 6065; 3-fluoro-4-iodophenyl], [BE 6066; 2-3-difluoro-4-iodophenyl], [BE 6067; 2, 6-difluoro- 4-iodophenyl], [BE 6068; 2,5-difluoro-4-iodophenyl], [BE 6069; 3,5-difluoro-4-iodophenyl], [BE 6070; 2, 3, 5-trifluoro-4-iodophenyl], [BE 60 70 BE6071; 2,3,6-trifluoro-4-iodophenyl], [BE6072; 2,3,5,6-tetrafluoro-4-iodophenyl], [BE6073; 2-methylphenyl], [BE6074; 3-methylphenyl], BE 6075; 4-methylphenyl, [BE 6076, 2-3-dimethylphenyl], [BE 6077; 2,4-dimethylphenyl], [BE 6078; 2, 5-dimethylphenyl], [BE 6079; 2, 6-dimethylphenyl], [BE 6080; 3,4-dimethylphenyl], [BE6081; 3,5-dimethylphenyl], [BE6082; 2,3,5-trimethylphenyl], [BE6083; 2,3,4-trimethylphenyl],

[BE 6084; 2,3,6-trimethylphenyl], [BE 6085; 2,4,5-trimethylphenyl], [BE 6086; 2,4,6-trimethylphenyl], [BE 6087; 3,4,5-trimethylphenyl], [BE 6088 2,3,4,6- tetramethylphenyl], [BE6089; 2,3,5,6- tetramethylphenyl], [BE6090; 2,3,4,5,6-pentamethylphenyl], [BE6091; 2-ethylphenyl], [BE6092; 3-ethylphenyl], [BE 6093; 4-ethylphenyl], [BE 6094; 2,4-diethylphenyl], [BE 6095; 2, 6-diethylphenyl], [BE 6096; 3,5-diethylphenyl], [BE 6097; 2 , 4,6-triethylphenyl], [BE 6098; 2-n-propylphenyl], [BE 6099; 3-n-propylphenyl], [BE 6100; 4-n-propylphenyl], [BE 6101; 2-isopropylphenyl], [BE 6102; 3 -isopropylphenyl], [BE 6103; 4-isopropylphenyl], [BE 6104; 2,4-diisopropylphenyl], [BE 6105; 2, 6-diisopropylphenyl], [BE 6106; 3,5-diisopropylphenyl], [BE 6107; 2-s-butylphenyl] ], [BE 6108; 3-s-butylphenyl], [BE 6109; 4-s-butylphenyl], [BE 6110; 2-t-butylphenyl], [BE 6111; 3-t-butylphenyl], [BE 6112; 4-t-butylphenyl] ], [BE6113; 4-n-butylphenyl], [BE6114; 4-n-nonylphenyl], [BE6115; 2-methyl-4-t-butylphenyl], [BE6116; 2-methyl-6-t-butylphenyl], [BE6117; 2-methyl-4-isopropylphenyl], [BE6118; 2-methyl-5-isopropylphenyl [BE 6119; 3-methyl-4-isopropylphenyl], [BE 6120; 2-cyclohexylphenyl], [BE 6121; 3-cyclohexylphenyl], [BE 6122; 4-cyclohexylphenyl], [BE 6123; 4-cyclopropylphenyl], [BE 6124; 4-cyclobutylphenyl], [BE6125; 4-cyclopentylphenyl], [BE6126; 2-chloro-4-phenylphenyl], [BE6127; 2-bromo-4-phenylphenyl], [BE6128; 4-hydroxyphenyl], [BE6129; methoxyphenyl], [BE6130; 3-methoxyphenyl], [BE6131; 4-methoxyphenyl], [BE6132; 2-ethoxyphenyl], [BE6133; 3-ethoxyphenyl], [BE6134; 4-ethoxyphenyl], [BE 6135; 2-n- [BE6 136; 3-n-propyloxyphenyl], [BE 6137; 4-n-propyloxyphenyl], [BE 6138; 2-isopropyloxyphenyl], [BE 6139; 3-isopropyloxyphenyl], [BE 6140; 4-isopropyloxyphenyl], [BE 6141; 2-n-hexyloxyphenyl], [BE6142; 3-n-hexyloxyphenyl], [BE6143; 4-n-hexyloxyphenyl], [BE6144; 2-benzyloxyphenyl], [BE6145; 3-benzyloxyphenyl], [BE6146; 4-benzyloxyphenyl] [BE 6147; 2-3-dimethoxyphenyl], [BE 6148; 2,4-dimethoxyphenyl], [BE 6149; 2, 5-dimethoxyphenyl], [BE 6150; 2, 6-dimethoxyphenyl], [BE 6151; 3,4-dimethoxyphenyl] [BE 6152; 3,5-dimethoxyphenyl], [BE 6153; 2-t-butoxyphenyl], [BE 6154; 3-t -butoxyphenyl], [BE 6155; 4-t-butylphenyl], [BE 6156; 3- (3-chlorophenyl) phenyl], [BE 6157; 4- (4-chlorophenyl) phenyl], [BE 6158; 2-phenoxyphenyl], [BE 6159 3-phenoxyphenyl], [BE 6160; 4-phenoxyphenyl], [BE 6161; 2- (2-fluorophenoxy) phenyl], [BE 6 16 2; 3- (3-chlorophenoxy) phenyl], [BE 6 16 3; 4- (4-chlorophenoxy) phenyl, [BE6164; 2,3,6-trimethyl-4-fluorophenyl], [BE6165; 2,3,6-trimethyl-4-chlorophenyl], [BE6166; 2,3,6-trimethyl-4-bromophenyl] [BE6167; 2,4-dimethyl-6-fluorophenyl], [BE6168; 2,4-dimethyl-6-chlorophenyl], [BE6169; 2,4-dimethyl-6-bromophenyl], [BE6170; 2-isopropyl- 4-chloro-5-methylphenyl], [BE6171; 2-chloro-4-nitrophenyl], [BE6172; 2-nitro-4-chlorophenyl], [BE6173; 2-methoxy-5-nitrophenyl], [BE6174; 4-dichloro-5-nitrophenyl], [BE 6175; 2,4-dichloro-6-nitrophenyl], [BE 6176; 2, 6-dichloro-4-nitrophenyl], [BE 6177; 2, 6-dibromo-4-nitrophenyl] , [BE6178; 2,6-diiodo-4-nitrophenyl], [BE6179; 2-methyl-5-isopropyl-4-chlorophenyl], [BE6180; 2-methoxycarbonylphenyl], [BE6181; 3-methoxycarbonylphenyl], [BE6182; 4-methoxycarbonylphenyl], [BE 6183; 4-acetoxyph enyl],

[BE 6184; 2-methoxymethylphenyl], [BE 6185; 3-methoxymethylphenyl], [BE 6186; 4-methoxymethylphenyl], [BE 6187; 2-phenylphenyl], [BE 6188; 3-phenylphenyl], [BE 6189; 4-phenylphenyl], [BE 6189] 2- (2-fluorophenyl) phenyl], [BE6191; 2-methyl-5-bromophenyl], [BE6192; 2-methyl-6-bromophenyl], [BE6193; 2-chloro-3-methylphenyl], [BE6194; 2-chloro-4-methylphenyl], [BE6195; 2-chloro-5-methylphenyl], [BE6196; 2-fluoro-3-methylphenyl], [BE6197; 2-fluoro-4-methylphenyl], [BE6198; 2- fluoro-5-methylphenyl, [BE 6199; 2-bromo-3-methylphenyl], [BE 6200; 2-bromo-4-methylphenyl], [BE 6201; 2-bromo-5-methylphenyl], [BE 6202; 3-methyl- 4-chlorophenyl], [BE 6203; 3-methyl-5-chlorophenyl], [BE 6204; 3-methyl-4-fluorophenyl], [BE 6205; 3-methyl-5-fluorophenyl], [BE 6206; 3-methyl-4- bromophenyl], [BE 6207; 3-methyl-5-bromophenyl], [BE 6208; 3-fluoro-4-methylphenyl], [BE 6209; 3-chloro-4-methylphenyl], [BE 6210; 3-bromo-4-methylphenyl] , [BE6211; 2-chloro-4,5-dimethylphenyl], [BE6212; 2-bromo-4,5-dimethylphenyl], [BE6213; 2-chloro-3,5-dimethylphenyl], [BE6214; 2-bromo- 3,5-dimethylphenyl], [BE 6215;], [BE6216;], [BE6217; Y, [BE6218; 2,6-dibromo-4-methylphenyl], [BE6219; 2,4-dichloro-6-methylphenyl], [BE6220; difluoro-6-methylphenyl, [BE 622; 2,4-dibromo-6-methylphenyl], [BE 622; 2, 6-dimethyl-4-fluorophenyl], [BE 6 22 3; 2, 6-dimethyl-4-chlorophenyl], [ BE6224; 2,6-dimethyl-4-bromophenyl], [BE6225; 3,5-dimethyl-4-fluorophenyl], [BE6226; 3,5-dimethyl-4-chlorophenyl], [BE6227; 3,5-dimethyl- 4-bromophenyl], [BE6228; 2-3-difluoro-4-methylphenyl], [BE6229; 2,5-difluoro-4-methylphenyl], [BE6230; 3,5-difluoro-4-methylphenyl], [BE6231; 2,3,5-trifluoro-4-methylphenyl], [BE6232; 2,3,6-trifluoro-4-methylphenyl], [BE6233; 2,3,5,6-tetrafluoro-4-methylphenyl], [BE6234; 2-fluoro-4-ethylphenyl], [BE6235; 3-fluoro-4-ethylphenyl], [BE6236; 2-3-difluoro-4-ethylphenyl], [BE6237; 2,6-difluoro-4-ethylphenyl], [BE6-237] BE6238; 2,5-difluoro-4-ethylphenyl], [BE6239; 3,5-difluoro-4-ethylphenyl], [BE6240; 2,3,5- trifluoro-4-ethylphenyl], [BE6241; 2,3, 6-trifluoro-4-ethylphenyl], [BE6242; 2,3,5,6-tetrafluoro-4-ethylphenyl], [BE6243; 2-trifluoromethylphenyl], [BE6244; 3 4-trifluoromethylphenyl], [BE6245; 4-trifluoromethylphenyl], [BE6246; 4- (2,2,2-trifluoro-1-trifluoromethylethyl) phenyl], [BE6247; 2-trifluoromethoxyphenyl], [BE6248; 3-trifluoromethoxyphenyl], [BE6248; BE6249; 4-trifluoromethoxyphenyl], [BE6250; 4- (2,2-difluoroethoxy) phenyl], [BE6251; 4- (2,2,2-trifluoroethoxy) phenyl], [BE6252; 2-nitrophenyl], [BE6253; 3-nitrophenyl, [BE6254; 4-nitrophenyl], [BE6255; 2-cyanophenyl], [BE6256; 3-cyanophenyl], [BE6257; 4-cyanophenyl], [BE6258; 2-methyl-3-chlorophenyl], [BE BE6259; 2-methyl-4-chlorophenyl], [BE6260; 2-methyl-5-chlorophenyl], [BE6261; 2-methyl-6-chlorophenyl], [BE6262; 2-methyl-3-fluorophenyl], [BE6263; 2-methyl-4-fluorophenyl], [BE6264; 2-methyl-5-fluorophenyl], [BE6265; 2-methyl-6-fluorophenyl], [BE6266; 2-methyl-3-bromophenyl], [BE6267; methyl-4-bromophenyl], [BE6268; 4-methylthiophenyl], [BE6269; 4-methylsulfonylphenyl], [BE 6270; 4-methylsulfinylphenyl], [BE 6271; 4-trifluoromethylthiophenyl], [BE 627 2; 4-ethynylphenyl], [BE 6 2 3 4- (1-propynyl) phenyl], [BE 6274; 4-vinylphenyl], [BE 6275; 4- (2, 2-dichlorovinyl) ph 4- (2,2-difluorovinyl) phenyl, [BE6277; cyclohexyl], [BE6278; 2-chlorocyclohexyl], [BE6279; 3-chlorocyclohexyl], [BE6280; 4-chlorocyclohexyl], [BE6281 4,4-dichlorocyclohexyl], [BE6282; 2-bromocyclohexyl], [BE6283; 3-bromocyclohexyl],

[BE6284; 4-bromocyclohexyl], [BE6285; 4, 4-difluorocyclohexyl], [BE 6286; 2-iodocyclohexyl], [BE 6287; 3-iodocyclohexyl], [BE 6288; [BE6290; 3-fluorocyclohexyl], [BE6291; 4-fluorocyclohexyl], [BE6292; 4, 4-difluorocyclohexyl], [BE6293; 4-methylcyclohexyl], [BE6294; 4-ethylcyclohexyl], [BE6295; 1-cyclohexyl], [BE6 296; 2-cyclohexenyl], [BE 6297; 3-cyclohexenyl], [BE 6298; 2-chloro-1-cyclohexenyl], [BE 6299; 3-chloro-1-cyclohexenyl], [BE 6300; 4-chloro-1-cyclohexenyl ], [BE6301; 5-chloro-1-cyclohexenyl], [BE6302; 6-chloro-1-cyclohexenyl], [BE6303; 1-chloro-2-cyclohexenyl], [BE6304; 2-chloro-2-cyclohexenyl], [BE6305; 3-chloro-2-cyclohexenyl], [BE6306; 4-chloro-2-cyclohexenyl], [BE6307; 5-chloro-2-cyclohexenyl], [BE6308; 6-chloro-2-cyclohexenyl], [BE6309 1-chloro-3-cyclohexenyl], [BE6310; 2-chloro-3-cyclohexenyl], [BE6311; 3-chloro-3-cyclohexenyl], [BE6312; 4-chloro-3-cyclohexenyl], [BE6313; -chloro-3-cyclohexenyl], [BE6314; 6-chloro-3-cyclohexenyl], [BE6315; 4-bromo-1-cyclohexyl], [BE6316; 4-bromo-2-cyclohexen [BE 6317; 4-bromo-3-cyclohexenyl], [BE 6318; 4-methyl-1-cyclohexyl], [BE 6319; 4-methyl-2-cyclohexyl], [BE 6320; 4-methyl-3-cyclohexenyl] , [BE6321; 4-ethyl-1-cyclohexenyl], [BE6322; 4-ethyl-2-cyclohexenyl], [BE6323; 4-ethyl-3-cyclohexenyl], [BE6324; trifluoromethyl], [BE6325; tert-butyl] [BE6326; 3-fluoro-2-methoxyphenyl], [BE6327; 4-fluoro-2-methoxyphenyl], [BE6328; 5-fluoro-2-methoxyphenyl], [BE6329; 6-fluoro-2-methoxyphenyl], [BE6326; BE6330; 3-chloro-2-methoxyphenyl], [BE6331; 4-chloro-2-methoxyphenyl], [BE6332; 5-chloro-2-methoxyphenyl], [BE6333; 6-chloro-2-methoxyphenyl], [BE6334; 3-bromo-2-methoxyphenyl], [BE6335; 4-bromo-2-methoxyphenyl], [BE6336; 5-bromo-2-methoxyphenyl], [BE6337; 6-bromo-2-methoxyphenyl], [BE6338; iodo-2-methoxyphenyl], [BE6339; 4-iodo-2-methoxyphenyl], [BE 6340; 5-iodo-2-methoxyphenyl], [BE6341; 6-iodo-2-methoxyphenyl], [BE6342; Dimethoxyphenyl], [BE 6343; 2,4-dimethoxyphenyl], [BE 6344; 2, 5-dimethoxyphenyl], [BE 6345; 2, 6-dimethoxyphenyl], [BE 6346; 3-methyl-2-methoxyphenyl], [BE 6347; methyl-2-methoxyphenyl], [BE6348; 5-methyl-2-methoxyphenyl], [BE6349; 6-methyl-2-methoxyphenyl], [BE6350; 3-ethyl-2-methoxyphenyl], [BE6351; 4-ethyl-2-methoxyphenyl], [BE6352; 5- Ethyl-2-methoxyphenyl], [BE6353; 6-ethyl-2-methoxyphenyl], [BE 6354; 3-trifluoromethoxy-2-methoxyphenyl], [BE 6355; 4-trifluoromethoxy-2-methoxyphenyl], [BE 6356; 5-trifluoromethoxy- 2-methoxyphenyl], [BE6357; 6-trifluoromethoxy-2-methoxyphenyl], [BE6358; 3-trifluoromethyl-2-methoxyphenyl], [BE6359; 4-trifluoromethyl-2-methoxyphenyl], [BE6360; 5-trifluoromethyl-2-] methoxyphenyl], [BE6361; 6-trifluoromethyl-2-methoxyphenyl], [BE6362; 3-methylthio-2-methoxyphenyl], [BE6363; 4-methylthio-2-methoxyphenyl], [BE6364; 5-methylthio-2-methoxyphenyl] [BE 6365; 6-methylthio-2-methoxyphenyl], [BE 6366; 3-trifluoromethylthio 2-methoxyphenyl], [BE 6367; 4-trifluoromethylthio 2-methoxyphenyl], [BE 6368; 5-trifluoromethyl 2-methoxyphenyl], [BE 6368; BE6369; 6-trifluoromethylthio-2-methoxyphenyl], [BE 6370; 3-ethynyl-2-methoxyphenyl], [BE 6371; 4-ethynyl-2-methoxyphenyl], [BE6372; 5-ethynyl-2-methoxyphenyl], [BE 6373; 6-ethyn yl-2-methoxyphenyl], [BE6374; 3-cyclopropyl-2-methoxyphenyl], [BE6375; 4-cyclopropyl-2-methoxyphenyl], [BE6376; 5-cyclopropyl-2-methoxyphenyl], [BE6377; 6-cyclopropyl- 2-methoxyphenyl], [BE6378; 3-cyclopropyloxy-2-methoxyphenyl], [BE6379; 4-cyclopropyloxy-2-methoxyphenyl], [BE 6380; 5-cyclopropyloxy-2-methoxyphenyl], [BE6381; 6-cyclopropyloxy-2-] methoxyphenyl], [BE6382; 2-ethoxy-3-fluorophenyl], [BE6383; 2-ethoxy-4-fluorophenyl],

[BE6384; 2-ethoxy-5-fluorophenyl], [BE 6385; 2-ethoxy-6-fluorophenyl], [BE 6386; 3-chloro-2-ethoxyphenyl], [BE 6387; 4-chloro-2-ethoxyphenyl], [BE 6388 5-chloro-2-ethoxyphenyl], [BE 6389; 6-chloro-2-ethoxyphenyl], [BE 6390; 3-bromo-2-ethoxyphenyl], [BE 6391; 4-bromo-2-ethoxyphenyl], [BE 6392; 5] -bromo-2-ethoxyphenyl], [BE6393; 6-bromo-2-ethoxyphenyl], [BE6394; 2-ethoxy-3-iodophenyl], [BE6395; 2-ethoxy-4-iodophenyl], [BE6396; 2-ethoxy -5-iodophenyl], [BE 6397; 2-ethoxy-6-iodophenyl], [BE 6398; 2,3-diethoxyphenyl], [BE 6399; 2,4-diethoxyphenyl], [BE 6400; 2, 5-diethoxyphenyl], [BE 6401 2,6-diethoxyphenyl], [BE6402; 2-ethoxy-3-methylphenyl], [BE6403; 2-ethoxy-4-methylphenyl], [BE6404; 2-ethoxy-5-methylphenyl], [BE6405; 2-ethoxy; -6-methylphenyl], [BE 6406; 3-ethyl-2-ethoxyphenyl], [BE 6407; 4-ethyl-2-ethoxyphenyl], [BE 6408; 5-ethyl-2-ethoxyphenyl], [BE 6409; 6-ethyl-2 2-ethoxyphenyl], [BE6410; 2-ethoxy-3-trifluoromethoxyphenyl], [BE 6411; 2-ethoxy-4-trifluoromethoxyphenyl], [BE 6412; 2-ethoxy-5-trifluoromethoxyphenyl], [BE 6413; 2-ethoxy-6-trifluoromethoxyphenyl ], [BE 641 4; 2-ethoxy-3-trifluoromethylphenyl], [BE6415; 2-ethoxy-4-trifluoromethylphenyl], [BE6416; 2-ethoxy-5-trifluoromethylphenyl], [BE6417; 2-ethoxy-6-trifluoromethylphenyl], [BE6418; 2-ethoxy-3-methylthiophenyl], [BE6419; 2-ethoxy-4-methylthiophenyl], [BE6420; 2-ethoxy-5-methylthiophenyl], [BE6421; 2-ethoxy-6-methylthiophenyl], [BE6422; 2-ethoxy-4-trifluorothiothiol], [BE 6423; 2-ethoxy-5-trifluorothiothiol], [BE 6425; 2-ethoxy-6-trifluorothiothiol], [BE 6426; 3-ethynyl- 2-ethoxyphenyl], [BE 6427; 4-ethynyl-2-ethoxyphenyl], [BE 6428; 5-ethynyl-2-ethoxyphenyl], [BE 6429; 6-ethynyl-2-ethoxyphenyl], [BE 6430; ethoxyphenyl], [BE6431; 4-cyclopropyl-2-ethoxyphenyl], [BE6432; 5-cyclopropyl-2-ethoxyphenyl], [BE6433; 6-cyclopropyl-2-ethoxyphenyl], [BE 6434; 3-cyclopropyloxy 2-ethoxyphenyl] [BE 6435; 4-cyclopropyloxy-2-ethoxyphenyl], [BE 6436; 5-cyclopropyloxy 2-ethoxyphenyl], [BE 6437; 6-cyclopropyl 2-ethoxyphenyl], [BE 6438; 3-methoxy-2-methylphenyl], BE6439; 4-methoxy-2- methylphenyl], [BE6440; 5-methoxy-2-methylphenyl], [BE6441; 6-methoxy-2-methylphenyl], [BE6442; 3-ethoxy-2-methylphenyl], [BE6443; 4-ethoxy-2-methylphenyl] [BE 644; 5-ethoxy-2-methylphenyl], [BE 6445; 6-ethoxy-2-methylphenyl], [BE 6446; 3-ethyl-2-methylphenyl], [BE 6447; 4-ethyl-2-methylphenyl], [BE 6445; BE6448; 5-ethyl-2-methylphenyl, [BE6449; 6-ethyl-2-methylphenyl], [BE 6450; 3-trifluoromethoxy-2-methylphenyl], [BE 6451; 4-trifluoromethoxy-2-methylphenyl], [BE 6452; 5-trifluoromethoxy-2-methylphenyl], [BE 6453; 6-trifluoromethoxy-2-methylphenyl], [BE 6454; 3-trifluoromethyl-2-methylphenyl], [BE 6455; 4-trifluoromethyl-2-methylphenyl], [BE 6456; trifluoromethyl-2-methylphenyl, [BE 6457; 6-trifluoromethyl-2-methylphenyl], [BE 6458; 3-methylthio-2-methylphenyl], [BE 6459; 4-methylthio-2-methylphenyl], [BE 6460; 5-methylthio- 2-methylphenyl], [BE6461; 6-methylthio-2-methylphenyl], [BE6462; 4-fluoro-2-isopropyloxyphenyl], [BE6463; 4-chloro-2-isopropyloxyphenyl], [BE6464; 4-bromo-2- isopropyloxyphenyl], [BE 6465; 4-iodo-2-isopropyloxyphenyl], [BE 6466; 4-methyl- 2-isopropyloxyphenyl], [BE6467; 4-ethyl-2-isopropyloxyphenyl], [BE6468; 4-methoxy-2-isopropyloxyphenyl], [BE6469; 4-ethoxy-2-isopropyloxyphenyl], [BE6470; 4-trifluoromethyl-2-] isopropyloxyphenyl], [BE6471; 4-trifluoromethoxy-2-isopropyloxyphenyl], [BE6472; 4-methylthio-2-isopropyloxyphenyl], [BE 6473; 4-cyclopropyl-2-isopropyloxyphenyl], [BE 6474; 4-fluoro-2-cyclopropylphenyl] [BE 6475; 4-chloro-2-cyclopropyloxyphenyl], [BE 6476; 4-bromo-2-cyclopropyloxyphenyl], [BE 6477; 4-iodo-2-cyclopropyloxyphenyl], [BE 6478; 4-methyl-2-cyclopropyloxyphenyl], [BE BE6479; 4-ethyl-2-cyclopropyloxyphenyl], [BE 6480; 4-methoxy-2-cyclopropyloxyphenyl], [BE 6481; 4-ethoxy-2-cyclopropyloxyphenyl], [BE 6482; 4-trifluoromethyl-2-cyclopropyloxyphenyl], [BE 6483 4-trifluoromethoxy-2-cyclopropyloxy],

[BE6484; 4-methylthio-2-cyclopropyloxyphenyl], [BE6485; 4-cyclopropyl-2-cyclopropyloxyphenyl], [BE6486; 3,4-difluoro-2-methoxyphenyl], [BE6487; 4,5-difluoro-2-methoxyphenyl] ], [BE6488; 4,6-difluoro-2-methoxyphenyl], [BE 6489; 3,4,5-trifluoro-2-methoxyphenyl], [BE 6490; 3,4,5,6-tetrafluoro-2-methoxyphenyl], [BE6491; 4-chloro-3-fluoro-2-methoxyphenyl], [BE6492; 4-chloro-5-fluoro-2-methoxyphenyl], [BE6493; 4-chloro-6-fluoro-2-methoxyphenyl], [BE6494 4-bromo-3-fluoro-2-methoxyphenyl], [BE6495; 4-bromo-5-fluoro-2-methoxyphenyl], [BE6496; 4-bromo-6-fluoro-2-methoxyphenyl], [BE6497; 3 , 4-difluoro-2-ethoxyphenyl], [BE 6498; 4, 5-difluoro-2-ethoxyphenyl], [BE 6499; 4, 6- difluoro-2-ethoxyphenyl], [BE 6 500; 3, 4, 5-trifluoro-2 -ethoxyphenyl], [BE6501; 3,4,5,6-tetrafluoro-2-ethoxyphenyl], [BE6502; 4-chloro-3-fluoro-2-ethoxyphenyl], [BE6503; 4-chloro-5-fluoro-2 4-ethoxyphenyl], [BE6504; 4-chloro-6-fluoro-2-ethoxyphenyl], [BE6505; 4-bromo-3-fluoro-2-ethoxyphenyl], [BE6506; 4-bromo-5-fluoro-2-ethoxyphenyl ], [BE 6507; 4-bromo-6-fluoro-2-ethoxyphenyl], [BE 6508; 4-difluoro-2-isopropyloxyphenyl], [BE6509; 4,5-difluoro-2-isopropyloxyphenyl], [BE6510; 4,6-difluoro-2-isopropyloxyphenyl], [BE6511; 3,4,5-trifluoro-2- isopropyloxyphenyl], [BE 6512; 3,4,5,6-tetrafluoro-2-isopropyloxyphenyl], [BE 6513; 4-chloro-3-fluoro-2-isopropyloxyphenyl], [BE 6514; 4-chloro-5-fluoro-2- isopropyloxyphenyl], [BE6515; 4-chloro-6-fluoro-2-isopropyloxyphenyl], [BE6516; 4-bromo-3-fluoro-2-isopropyloxyphenyl], [BE6517; 4-bromo-5-fluoro-2-isopropyloxyphenyl] [BE6518; 4-bromo-6-fluoro-2-isopropyloxyphenyl], [BE6519; 3,4-difluoro-2-cyclopropyloxyphenyl], [BE6520; 4,5-difluoro-2-cyclopropyloxyphenyl], [BE 6521; 6-difluoro-2-cyclopropyloxyphenyl], [BE6522; 3,4,5-trifluoro-2-cyclopropyloxyphenyl], [BE6523; 3,4,5,6-tetrafluoro-2-cyclopropyloxyphenyl], [BE6524; 4-chloro- 3-fluoro-2-cyclopropyloxyphenyl], [BE6525; 4-chloro-5-fluoro-2-cyclopropyloxyphenyl], [BE6526; 4-chloro-6-fluoro-2-cyclopropyloxyphenyl], [BE6527; 4-bromo-3- fluoro-2-cyclopropyloxyphenyl], [BE6528; 4-bromo-5-fluoro-2-cyclopropyloxyphenyl], [BE6529; 4-bromo-6 -fluoro-2-cyclopropyloxyphenyl], [BE6530; 3-ethynyl-2-methylphenyl], [BE6531; 4-ethynyl-2-methylphenyl], [BE6532; 5-ethynyl-2-methylphenyl], [BE6533; 6-ethynyl -2-methylphenyl], [BE6534; 3-cyclopropyl-2-methylphenyl], [BE6535; 4-cyclopropyl-2-methylphenyl], [BE6536; 5-cyclopropyl-2-methylphenyl], [BE6537; 6-cyclopropyl-2 -methylphenyl], [BE6538; 3-cyclopropyloxy-2-methylphenyl], [BE6539; 4-cyclopropyloxy-2-methylphenyl], [BE6540; 5-cyclopropyloxy-2-methylphenyl], [BE6541; 6-cyclopropyloxy-2-methylphenyl ], [BE6542; 3-methoxy-2-fluorophenyl], [BE 6543; 4-methoxy-2-fluorophenyl], [BE 6544; 5-methoxy-2-fluorophenyl], [BE6545; 6-methoxy-2-fluorophenyl], [BE6546; 3-ethoxy-2-fluorophenyl], [BE6547; 4-ethoxy-2-fluorophenyl], [BE6548; 5-ethoxy-2-fluorophenyl], [BE6549; 6-ethoxy-2-fluorophenyl], [BE6550 3-ethyl-2-fluorophenyl, [BE6551; 5-ethyl-2-fluorophenyl], [BE6552; 6-ethyl-2-fluorophenyl], [BE6553; 2-fluoro-3-trifluoromethoxyphenyl], [BE6554; 2 -fluoro-4-trifluoromethoxyphenyl], [BE6555; 2-fluoro-5-trifluoromethoxyphenyl], [BE6556; 2-fluoro-6-trif luoromethoxyphenyl], [BE6557; 2-fluoro-3-trifluoromethylphenyl], [BE6558; 2-fluoro-4-trifluoromethylphenyl], [BE6559; 2-fluoro-5-trifluoromethylphenyl], [BE6560; 2-fluoro-6-trifluoromethylphenyl] [BE6561; 2-fluoro-3-fluorothiophenyl], [BE6562; 2-fluoro-4-fluorothiophenyl], [BE6563; 2-fluoro-5-fluorothiophenyl], [BE6564; 2-fluoro-6-fluorothiophenyl], [BE6564; BE6565; 3-ethynyl-2-fluorophenyl], [BE 6566; 4-ethynyl-2-fluorophenyl], [BE6567; 5-ethynyl-2-fluorophenyl], [BE 6568; 6-ethynyl-2-fluorophenyl], [BE6569; 3-cyclopropyl-2-fluorophenyl], [BE6570; 4-cyclopropyl-2-fluorophenyl], [BE6571; 5-cyclopropyl-2-fluorophenyl], [BE6572; 6-cyclopropyl-2-fluorophenyl], [BE6573; 3- cyclopropyloxy-2-fluorophenyl], [BE 6574; 4-cyclopropyloxy 2-fluorophenyl], [BE 6575; 5-cyclopropyloxy 2- fluorophenyl], [BE 6576; 6-cyclopropyloxy 2- fluorophenyl], [BE 6577; 2-ethyl- 3-fluorophenyl], [BE6578; 2-ethyl-4-fluorophenyl], [BE6579; 2-ethyl-5-fluorophenyl], [BE6580; 2-ethyl-6-fluorophenyl], [BE6581; 3-chloro-2-] Ethylphenyl], [BE6582; 4-chloro-2-ethylphenyl], [BE6583; 5-chloro-2-e thylphenyl],

[BE6584; 6-chloro-2-ethylphenyl], [BE6585; 3-bromo-2-ethylphenyl], [BE6586; 4-bromo-2-ethylphenyl], [BE6587; 5-bromo-2-ethylphenyl], [BE6588 6-bromo-2-ethylphenyl], [BE6589; 2-ethyl-3-iodophenyl], [BE6590; 2-ethyl-4-iodophenyl], [BE6591; 2-ethyl-5-iodophenyl], [BE6592; 2 -ethyl-6-iodophenyl], [BE6593; 2-ethyl-3-ethoxyphenyl], [BE6594; 2-ethyl-4-ethoxyphenyl], [BE6595; 2-ethyl-5-ethoxyphenyl], [BE6596; 2-ethyl -6-ethoxyphenyl], [BE6597; 2-ethyl-3-methylphenyl], [BE6598; 2-ethyl-4-methylphenyl], [BE6599; 2-ethyl-5-methylphenyl], [BE6600; 2-ethyl-6 -methylphenyl], [BE6601; 2,3-diethylphenyl], [BE6602; 2,4-diethylphenyl], [BE6603; 2, 5-diethylphenyl], [BE 6604; 2, 6-diethylphenyl], [BE 6605; 2-ethyl -3-trifluoromethoxyphenyl], [BE6606; 2-ethyl-4-trifluoromethoxyphenyl], [BE6607; 2-ethyl-5-trifluoromethoxyphenyl], [BE6608; 2-ethyl-6-trifluoromethoxyphenyl], [BE6609; 2-ethyl-3 -trifluoromethylphenyl, [BE6610; 2-ethyl-4-trifluoromethylphenyl], [BE6611; 2-ethyl-5-trifluoromethylphenyl], [BE6612; 2-ethyl-6-trifluoromethylphenyl], [BE6613; 2-ethyl-3-methylthio] [BE6614; 2-ethyl-4-methylthiophenyl], [BE6615; 2-ethyl-5-methylthiophenyl], [BE6616; 2-ethyl-6-methylthiophenyl], [BE6617; 2-ethyl-3-trifluoromethylthiophenyl] [BE6618; 2-ethyl-4-trifluoromethylthiophenyl], [BE6619; 2-ethyl-5-trifluoromethylthiophenyl], [BE6620; 2-ethyl-6-trifluoromethylthiophenyl], [BE6621; 3-ethynyl-2-ethylphenyl], [BE6621; BE6622; 4-ethynyl-2-ethylphenyl], [BE6623; 5-ethynyl-2-ethylphenyl], [BE6624; 6-ethynyl-2-ethylphenyl], [BE6625; 3-cyclopropyl-2-ethylphenyl], [BE6626; 4-cyclopropyl-2-ethylphenyl], [BE6627; 5-cyclopropyl-2-ethylphenyl], [BE6628; 6-cyclopropyl-2-ethylphenyl], [BE6629; 3-cyclopropyloxy-2-ethylphenyl], [BE6630; cyclopropyloxy-2-ethylphenyl], [BE6631; 5-cyclopropyloxy-2-ethylphenyl], [BE6632; 6-cyclopropyloxy-2-ethylphenyl], [BE6633; 3-fluoro-2-trifluoromethylphenyl], [BE6634; 2-trifluoromethylphenyl], [BE6635; 5-fluoro-2-trifluoromethylphenyl], [BE6636; 6-fluoro-2-trifluoromethylphenyl], [BE6637; 3-chloro-2-trifluoromethylphenyl], [BE6638; 4-chloro-2- trifluoromethylphenyl], [BE 6639; 5-ch loro-2-trifluoromethylphenyl, [BE6640; 6-chloro-2-trifluoromethylphenyl], [BE6641; 3-bromo-2-trifluoromethylphenyl], [BE6642; 4-bromo-2-trifluoromethylphenyl], [BE6643; 5-bromo- 2-trifluoromethylphenyl], [BE6644; 6-bromo-2-trifluoromethylphenyl], [BE6645; 3-iodo-2-trifluoromethylphenyl], [BE6646; 4-iodo-2-trifluoromethylphenyl], [BE6647; 5-iodo-2- 2 trifluoromethylphenyl], [BE6648; 6-iodo-2-trifluoromethylphenyl], [BE6649; 3-ethoxy-2-trifluoromethylphenyl], [BE6650; 4-ethoxy-2-trifluoromethylphenyl], [BE6651; 5-ethoxy-2-trimethylphenyl] [BE6652; 6-ethoxy-2-trifluoromethylphenyl], [BE6653; 3-methyl-2-trifluoromethylphenyl], [BE6654; 4-methyl-2-trifluoromethylphenyl], [BE6655; 5-methyl-2-trifluoromethylphenyl], [BE6654; BE 6656; 6-methyl-2-trifluoromethylphenyl], [BE 6657; 2,3-ditrifluoromethylphenyl], [BE 6658; 2,4-ditrifluoromethylphenyl], [BE 6659; 2, 5-ditrifluoromethylphenyl], [BE 6660; , [BE6661; 2-trifluoromethyl-3- trifluoromethoxyphenyl], [BE6662; 2-trifluoromethyl-4- trifluoromethoxyphenyl], [BE6663; orthomethyl-5-trifluoromethoxyphenyl], [BE6664; 2-trifluoromethyl-6-trifluoromethoxyphenyl], [BE6665; 2-ethyl-3-trifluoromethylphenyl], [BE6666; 2-ethyl-4-trifluoromethylphenyl], [BE6667; 2-ethyl- 5-trifluoromethylphenyl], [BE6668; 2-ethyl-6-trifluoromethylphenyl], [BE6669; 3-methylthio-2-trifluoromethylphenyl], [BE6670; 4-methylthio-2-trifluoromethylphenyl], [BE6671; 5-methylthio-2-] trifluoromethylphenyl], [BE6672; 6-methylthio-2-trifluoromethylphenyl], [BE6673; 2-trifluoromethyl-3- trifluoromethylthiophenyl], [BE6674; 2-trifluoromethyl-4- trifluorothiophenyl], [BE6675; [BE 6667; 2-trifluoromethyl-6-trifluorothiothiol], [BE 6677; 3-ethynyl-2-trifluoromethylphenyl], [BE 6678; 4-ethynyl-2-trifluoromethylphenyl], [BE 6679; 5-ethynyl-2-trifluoromethylphenyl], [BE BE 6680; 6-ethynyl-2-trifluoromethylphenyl, [BE 6681; 3-cyclopropyl-2-trifluoromethylphenyl], [BE 6682; 4-cyclopropyl-2-trifluoromethylphenyl], [BE 6683; 5-cyclopropyl-2-trifluoromethylphenyl],

[BE6684; 6-cyclopropyl-2-trifluoromethylphenyl], [BE6685; 3-cyclopropyloxy-2-trifluoromethylphenyl], [BE6686; 4- cyclopropyloxy-2-trifluoromethylphenyl], [BE6687; 6-cyclopropyloxy-2-trifluoromethylphenyl], [BE6689; 3-methoxynaphthalene-2-yl], [BE6690; 6-chloro-3-methoxynaphthalene-2-yl], [BE6691; 6-fluoro-3-methoxynaphthalene-2]; 7-chloro-3-methoxynaphthalene-2-yl], [BE6692; 7-chloro-3-methoxynaphthalene-2-yl], [BE6694; 8-chloro-3-methoxynaphthalene-2-yl] ], [BE 6695; 8-fluoro-3-methoxynaphthalene-2-yl], [BE 6696; 1-chloro-3-methoxynaphthalene-2-yl], [BE 6697; 1-fluoro-3-methoxynaphthalene-2-yl], [BE6698; 4-chloro-3-methoxynaphthalene-2-yl], [BE 6699; 4-fluoro-3-methoxynaphthalene-2-yl], [BE 6700; 5-chloro-3-methoxynaphthalene-2-yl], [BE6701 5-fluoro-3-methoxynaphthalene-2-yl].

  Further, the present compounds AF1-BF1 to AF360-BF1300 can also be obtained according to the method described above.

The present compounds AF1-BF1 to AF360-BF1300 are compounds represented by the following formula (AFBF).
[Wherein, X ^{61 to} X ⁶⁶ each represent a substituent corresponding to each of the substituent numbers (MF 1) AF 1 to AF 360 shown below, wherein E ¹⁰⁶ is a substituent number (MF 2) BF 1 shown below .About.BF1300. ]
For example, the present compounds AF1-BF1, in the compounds of formula (AFBF), X ⁶¹ ~X ⁶⁶ substituents ID MF1 (X ⁶² ~X ⁶⁴ and X ⁶⁵ is a hydrogen atom, X ⁶¹ and X ⁶⁶ is an oxygen atom And E ¹⁰⁶ represents a compound in which the substituent number (MF 2) is BF 1 (pyrazol-4-yl group), and is represented by the following formula.
[Substituent number (MF1): X ⁶¹ , X ⁶² , X ⁶³ , X ⁶⁴ , X ⁶⁵ , X ⁶⁶ ], [AF 1; O, H, H, H, H, O], [AF 2; O, F, H, H, H, O], [AF 3; O, Cl, H, H, H, O], [AF 4; O, Br, H, H, H, O], [AF 5; O, I, H, O H, H, O], [AF 6; O, Me, H, H, H, O], [AF 7; O, Et, H, H, H, O], [AF 8; O, Pr, H, H, O H, O], [AF 9; O, i-Pr, H, H, H, O], [AF 10; O, CH = CH ₂ , H, H, H, O], [AF 11; O, C (Me ) = CH ₂ , H, H, H, O], [AF 12; O, C≡CH, H, H, H, O], [AF 13; O, C≡ C Me, H, H, H, O], [AF14; O, c-Pr, H, H, H, O], [AF15; O, OMe, H, H, H, O], [AF16; O, OEt, H, H, H, O], [AF17; O, Oi-Pr, H, H, H, O], [AF18; O, SMe, H, H, H, O], [AF19; O, SEt, H, H, H, O], _{[AF20; O, CH 2 F} , H, H, H, O], [AF21; O, CHF 2, H, H, H, O], [AF22; O, CF 3, H, H, H, O ], [AF23; O, OCH 2 F, H, H, H, O], [AF24; O, OCHF 2, H, H, H, O], [AF25; O, OCF 3, H, H, H , O], [AF26; O, SCH ₂ F, H, H, H, O], [AF 27; O, SCHF ₂ , H, H, H, O], [AF 28; O, SCF ₃ , H, H , H, O], [AF 29; O, CN, H, H, H, O], [AF 30; O, NO ₂ , H, H, H, O], [AF 31; O, H, F, H, H, O], [AF 32; O, F, F, H, H, O], [AF 33; O, Cl, F, H, H, O], [AF 34; O, Br, F, H, H, H O], [AF 35; O, I, F, H, H, O], [AF 36; O, Me, F, H, H, O], [AF 37; O, Et, F, H, H, O] , [AF 38; O, Pr, F, H, H, O], [AF 39; O, i-Pr, F, H, H, O], [AF 40; O, CH = CH ₂ , F, H, H, O], [AF 41; O, C (Me) = CH ₂ , F, H, H, O], [AF 42; O, C≡CH, F, H, H, O], [[ AF 43; O, C≡CMe, F, H, H, O], [AF 44; O, c-Pr, F, H, H, O], [AF 45; O, OMe, F, H, H, O] [AF 46; O, OEt, F, H, H, O], [AF 47; O, Oi-Pr, F, H, H, O], [AF 48; O, SMe, F, H, H, O] [AF 49; O, SEt, F, H, H, O], [AF 50; O, CH ₂ F, F, H, H, O], [AF 51; O, CHF ₂ , F, H, H, O ], [AF52; O, CF 3, F, H, H, O], [AF53; O, OCH 2 F, F, H, H, O], [AF54; O, OCHF 2, F, H, H , O], [AF 55; O, OCF ₃ , F, H, H, O], [AF 56; O, SCH ₂ F, F, H, H, O], [AF 57; O, SCHF ₂ , F, H , H, O], [AF 58; O, SCF ₃ , F, H, H, O], [AF 59; O, CN, F, H, H, O], [AF 60; O, NO ₂ , F, H , H, O], [AF 61; O, H, H, F, H, O], [AF 62; O, F, H, F, H, O], [AF 63; O, Cl, H, F, H , O], [AF 64; O, Br, H, F, H, O], [AF 65; O, I, H, F, H, O], [AF 66; O, Me, H, F, H, O ], [AF 67; O, Et, H, F, H, O], [AF 68; O, Pr, H, F, H, O], [AF 69; O, i-Pr, H, F, H, O] ], [AF 70; O, CH = CH ₂ , H, F, H, O], [AF 71; O, C (Me) = CH ₂ , H, F, H, O], [AF 72; O, C≡ CH, H, F, H, O], [AF 73; O, C≡CMe, H, F, H, O], [AF 74; O, c-Pr, H, F, H, O], [AF 75; O, OMe, H, F, H, O], [AF 76; O, OEt, H, F, H, O], [AF 77; O, Oi-Pr, H, F, H, O], [AF 78; O, SMe, H, F, H, O], [AF79; O, SEt, H, F, H, O], [AF80; O, CH 2 F, H, F, H, O], [AF81 _{O, CHF 2, H, F} , H, O], [AF82; O, CF 3, H, F, H, O], [AF83; O, OCH 2 F, H, F, H, O], [ _{AF84; O, OCHF 2, H} , F, H, O], [AF85; O, OCF 3, H, F, H, O], [AF86; O, SCH 2 F, H, F, H, O] [AF 87; O, SCHF ₂ , H, F, H, O], [AF 88; O, SCF ₃ , H, F, H, O], [AF 89; O, CN, H, F, H, O] , [AF 90; O, NO ₂ , H, F, H, O], [AF 91; O, H, H, H, F, O], [AF 92; O, F, H, H, F, O], [AF 93; O, Cl, H, H, F, O], [AF 94; O, Br, H, H, F, O], [AF 95; O, I, H, H, F, O], [AF 96 O, Me, H, H, F, O], [AF 97; O, Et, H, H, F, O], [AF 98; O, Pr, H, H, F, O], [AF 99; O , i-Pr, H, H, F, O], [AF 100; O, CH = CH ₂ , H, H, F, O],

[AF101; O, C (Me ) = CH 2, H, H, F, O], [AF102; O, C≡CH, H, H, F, O], [AF103; O, C≡CMe, H , H, F, O], [AF104; O, c-Pr, H, H, F, O], [AF 105; O, OMe, H, H, F, O], [AF 106; O, OEt, H , H, F, O], [AF 107; O, Oi-Pr, H, H, F, O], [AF 108; O, S Me, H, F, O], [AF 109; O, SE t, H , H, F, O], [AF 110; O, CH ₂ F, H, H, F, O], [AF 111; O, CHF ₂ , H, H, F, O], [AF 112; O, CF ₃ , H, H, F, O ], [AF113; O, OCH 2 F, H, H, F, O], [AF114; O, OCHF 2, H, H, F, O], [AF115; O, _{OCF 3, H, H, F} , O], [AF116; O, SCH 2 F, H, H, F, O], [AF117; O, SCHF 2, H, H, F, O], [AF118; O, SCF ₃ , H, H, F, O], [AF119; O, CN, H, H, F, O], [AF 120; O, NO ₂ , H, H, F, O], [AF 121; S, H, H, H, H, O], [AF 122; S, F, H, H, H, O], [AF 123; S, Cl, H, H, H, O], [AF 124; S, Br, H, H, H, O], [AF 125; S, I, H, H, H, O], [AF 126; S, Me, H, H, H, O], [AF 127; H, H, H, O], [AF 128; S, Pr, H, H, H, O], [AF 129; S, i-Pr, H, H, H, O], [AF 130; S, CH = CH ₂ , H, H, H, O], [AF 131; S, C (Me) = CH ₂ , H, H, H, O], [AF 132; S, C≡CH, H, H, H, O ], [AF133; S, C≡CMe, H, H, H, O], [AF134; S, c-Pr, H, H, H, O], [AF 135; S, OMe, H, H, H] , O], [AF 136; S, OEt, H, H, H, O], [AF 137; S, Oi-Pr, H, H, H, O], [AF 138; S, S Me, H, H, H , O], [AF 139; S, SE t, H, H, H, O], [A F 140; S, CH ₂ F, H, H, H, O], [AF 141; S, CHF ₂ , H, H, H, O], [AF 142; S, CF ₃ , H, H, H, O] _{, [AF143; S, OCH 2} F, H, H, H, O], [AF144; S, OCHF 2, H, H, H, O], [AF145; S, OCF 3, H, H, H, O], [AF 146; S, SCH ₂ F, H, H, H, O], [AF 147; S, SCHF ₂ , H, H, H, O], [AF 148; S, SCF ₃ , H, H, H, O], [AF 149; S, CN, H, H, H, O], [AF 150; S, NO ₂ , H, H, H, O], [AF 151; S, H, F, H, H , O], [AF 152; S, F, F, H, H, O], [AF 153; S, Cl, F, H, H, O], [AF 154; S, Br, F, H, H, O ], [AF 155; S, I, F, H, H, O], [AF 156; S, Me, F, H, H, O], [AF 157; S, Et, F, H, H, O], [AF158; S, Pr, F , H, H, O], [AF159; S, i-Pr, F, H, H, O], [AF160; S, CH = CH 2, F, H, H, O], [AF161; S, C (Me) = CH 2, F, H, H, O], [AF162; S, C≡CH, F, H, H, O], [AF163; S, C≡ CMe, F, H, H, O], [AF 164; S, c-Pr, F, H, H, O], [AF 165; S, OMe, F, H, H, O], [AF 166; S, OEt, F, H, H, O], [AF 167; S, Oi-Pr, F, H, H, O], [AF 168; S, S Me, F, H, H, O], [AF 169; S, SEt, F, H, H, O], [AF 170; S, CH ₂ F, F, H, H, O], [AF 171; S, CHF ₂ , F, H, H, O], [AF 172; S , CF ₃ , F, H, H, O], [AF 173; S, OCH ₂ F, F, H, H, O], [AF 174; S, OCHF ₂ , F, H, H, O], [AF 175 S, OCF ₃ , F, H, H, O], [AF 176; S, SCH ₂ F, F, H, H, O], [AF 177; S, SCHF ₂ , F, H, H, O], [AF 178; S, SCF ₃ , F , H, H, O], [AF 179; S, CN, F, H, H, O], [AF 180; S, NO ₂ , F, H, H, O], [AF 181; S, H, H, H F, H, O], [AF 182; S, F, H, F, H, O], [AF 183; S, Cl, H, F, H, O], [AF 184; S, Br, H, F, H, O], [AF 185; S, I, H, F, H, O], [AF 186; S, Me, H, F, H, O], [AF 187; S, Et, H, F, H, O, [AF 188; S, Pr, H, F, H, O], [AF 189; S, i-Pr, H, F, H, O], [AF 190; S, CH = CH ₂ , H, F , H, O], [AF191 ; S, C (Me) = CH 2, H, F, H, O], [AF192; S, C≡CH, H, F, H, O], [AF193; S , C≡CMe, H, F, H, O], [AF194; S, c-Pr, H, F, H, O], [AF 195; S, OMe, H, F, H, O], [AF 196 S, OEt, H, F, H, O], [AF 197; S, Oi-Pr, H, F, H, O], [AF 198; S, S Me, H, F, H, O], [AF 199 S, SEt, H, F, H, O], [AF ₂₀₀ ; S, CH ₂ F, H, F, H, O],

_{[AF201; S, CHF 2,} H, F, H, O], [AF202; S, CF 3, H, F, H, O], [AF203; S, OCH 2 F, H, F, H, O ], [AF 204; S, OCHF ₂ , H, F, H, O], [AF 205; S, OCF ₃ , H, F, H, O], [AF 206; S, SCH ₂ F, H, F, H] , O], [AF 207; S, SCHF ₂ , H, F, H, O], [AF 208; S, SCF ₃ , H, F, H, O], [AF 209; S, CN, H, F, H , O], [AF210; S , NO 2, H, F, H, O], [AF211; S, H, H, H, F, O], [AF212; S, F, H, H, F, O], [AF 213; S, Cl, H, H, F, O], [AF 214; S, Br, H, H, F, O], [AF 215; S, I, H, H, F, O] , [AF 216; S, Me, H, H, F, O], [AF 217; S, Et, H, H, F, O], [AF 218; S, Pr, H, H, F, O], [[ AF219; S, i-Pr, H, H, F, O], [AF220; S, CH = CH 2, H, H, F, O], [AF221; S, C (Me) = CH 2, H , H, F, O], [AF 222; S, C≡CH, H, H, F, O], [AF 223; S, C ≡ CMe, H, H, F, O], [AF 224; S, c -Pr, H, H, F, O], [AF 225; S, OMe, H, H, F, O], [AF 226; S, OE t, H, H, F, O], [AF 227; S, Oi -Pr, H, H, F, O], [AF 228; S, S Me, H, H, F, O], [AF 229; S, SE t, H, H, F, O], [AF 230; S, CH ₂ F, H, H, F, O], [AF 231; S, CHF ₂ , H, H, F, O], [AF 232; S, CF ₃ , H, H, F, O], [AF 233; S OCH ₂ F, H, H, F, O], [AF234; S, OCHF ₂ , H, H, F, O], [AF 235; S, OCF ₃ , H, H, F, O], [AF 236 S, SCH ₂ F, H, H, F, O], [AF 237; S, SCHF ₂ , H, H, F, O], [AF 238; S, SCF ₃ , H, H, F, O], [AF 239; S, CN, H, H , F, O], [AF 240; S, NO ₂ , H, H, F, O], [AF 241; O, H, H, H, H, S], [AF 242; O, F, H, H, H H, S], [AF 243; O, Cl, H, H, H, S], [AF 244; O, Br, H, H, H, S], [AF 245; O, I, H, H, H, S S], [AF 246; O, Me, H, H, H, S], [AF 247; O, Et, H, H, H, S], [AF 248; O, Pr, H, H, H, S] , [AF249; O, i- Pr, H, H, H, S], [AF250; O, CH = CH 2, H, H, H, S], [AF251; O, C (Me) = CH 2 , H, H, H, S], [AF 252; O, C≡CH, H, H, H, S], [AF 253; O, C ≡ CMe, H, H, H, S], [AF 254; O , c-Pr, H, H, H, S], [AF255; O, OMe, H, H, H, S], [AF 256; O, OEt, H, H, H, S], [AF 257; , Oi-Pr, H, H, H, S], [AF258; O, SMe, H, H, H, S], [AF 259: O, SEt, H, H, H, S], [AF 260; O _{, CH 2 F, H, H} , H, S], [AF261; O, CHF 2, H, H, H, S], [AF262; O, CF 3, H, H, H, S], [AF263 O, OCH ₂ F, H, H, H, S], [AF 264; O, OCHF ₂ , H, H, H, S], [AF 265; O, OCF ₃ , H, H, H, S], [AF 266; O, SCH ₂ F, H, H, H, S], [AF 267; O, SCHF ₂ , H, H, H, S], [AF 268; O, SCF ₃ , H, H, H, S ], [AF 269; O, CN, H, H, H, S], [AF 270; O, NO ₂ , H, H, H, S], [AF 271; O, H, F, H, H, S] [AF 272; O, F, F, H, H, S], [AF 273; O, Cl, F, H, H, S], [AF 274; O, Br, F, H, H, S], [[AF 272; AF 275; O, I, F, H, H, S], [AF 276; O, Me, F, H, H, S], [AF 277; O, Et, F, H, H, S], [AF 278; O, Pr, F, H, H, S], [AF 279; O, i-Pr, F, H, H, S ], [AF280; O, CH = CH 2, F, H, H, S], [AF281; O, C (Me) = CH 2, F, H, H, S], [AF282; O, C≡ CH, F, H, H, S], [AF 283; O, C≡CMe, F, H, H, S], [AF 284; O, c-Pr, F, H, H, S], [AF 285; O, OMe, F, H, H, S], [AF 286; O, OEt, F, H, H, S], [AF 287; O, Oi-Pr, F, H, H, S], [AF 288; O, SMe, F, H, H, S], [AF 289; O, SE t, F, H, H, S], [AF 290; O, CH ₂ F, F, H, H, S], [AF 291; O, CHF ₂ , F, H, H, S], [AF 292; O, CF ₃ , F, H, H, S], [AF 293; O, OCH ₂ F, F, H, H, S], [[ _{AF294; O, OCHF 2, F} , H, H, S], [AF295; O, OCF 3, F, H, H, S], [AF296; O, SCH 2 F, F, H, H, S] [AF 297; O, SCHF ₂ , F, H, H, S], [AF 298; O, SCF ₃ , F, H, H, S], [AF 299; O, CN, F, H, H, S] , [AF 300; O, NO ₂ , F, H, H, S],

[AF301; O, H, H, F, H, S], [AF 302; O, F, H, F, H, S], [AF 303; O, Cl, H, F, H, S], [AF 304 O, Br, H, F, H, S], [AF 305; O, I, H, F, H, S], [AF 306; O, Me, H, F, H, S], [AF 307; O , Et, H, F, H, S], [AF308; O, Pr, H, F, H, S], [AF309; O, i-Pr, H, F, H, S], [AF 310; O _{, CH = CH 2, H,} F, H, S], [AF311; O, C (Me) = CH 2, H, F, H, S], [AF312; O, C≡CH, H, F, H, S], [AF 313; O, C≡CMe, H, F, H, S], [AF 314; O, c-Pr, H, F, H, S], [AF 315; O, OMe, H, F, H, S], [AF 316; O, OEt, H, F, H, S], [AF 317; O, Oi-Pr, H, F, H, S], [AF 318; O, SMe, H, F, H, S], [AF 319; O, SE t, H, F, H, S], [AF 320; O, CH ₂ F, H, F, H, S], [AF 321; O, CHF ₂ , H , F, H, S], [AF 322; O, CF ₃ , H, F, H, S], [AF 323; O, OCH ₂ F, H, F, H, S], [AF 324; O, OCHF ₂ , H, F, H, S ], [AF325; O, OCF 3, H, F, H, S], [AF326; O, SCH 2 F, H, F, H, S], [AF327; O, SCHF ₂ , H, F, H, S], [AF 328; O, SCF ₃ , H, F, H, S], [AF 329: O, CN, H, F, H, S], [AF 330; O, _{NO 2, H, F, H} , S], [AF331; O, H, H, H, F, S], [AF332; O, F, H, H, F, S], [AF333; O, Cl , H, H, F, S], [AF334; O, Br, H, H, F, S], [AF 335; O, I, H, H, F, S], [AF336; O, Me, H] , H, F, S], [AF 337; O, Et, H, H, F, S], [AF 338; O, Pr, H, H, F, S], [AF 339: O, i-Pr, H , H, F, S], [AF340; O, CH = CH 2, H, H, F, S], [ AF 341; O, C (Me) = CH ₂ , H, H, F, S], [AF 342; O, C≡CH, H, H, F, S], [AF 343: O, C Me CMe, H, H, F, S], [AF 344; O, c-Pr, H, H, F, S], [AF 345; O, OMe, H, H, F, S], [AF 346; O, OE t, H, H, F, S], [AF 347; O, Oi-Pr, H, H, F, S], [AF 348; O, SMe, H, H, F, S], [AF 349; O, SE t, H, H, F, S], [ AF350; O, CH 2 F, H, H, F, S], [AF351; O, CHF 2, H, H, F, S], [AF352; O, CF 3, H, H, F, S] , [AF353; O, OCH 2 F, H, H, F, S], [AF354; O, OCHF 2, H, H, F, S], [AF355; O, OCF ₃ , H, H, F, S], [AF 356; O, SCH ₂ F, H, H, F, S], [AF 357; O, SCHF ₂ , H, H, F, S], [AF 358; O SCF ₃ , H, H, F, S], [AF 359; O, CN, H, H, F, S], [AF 360; O, NO ₂ , H, H, F, S].

[Substituent number (MF2); E ¹⁰⁶ ], [BF 1; 1-Ph-PYR-4-yl], [BF 2; 1- (2-F-Ph) PYR-4-yl], [BF 3; 1- (3-F-Ph) PYR-4-yl], [BF4; 1- (4-F-Ph) PYR-4-yl], [BF5; 1- (2-Cl-Ph) PYR-4-yl ], [BF6; 1- (3-Cl-Ph) PYR-4-yl], [BF7; 1- (4-Cl-Ph) PYR-4-yl], [BF8; 1- (2-Br-) Ph) PYR-4-yl], [BF9; 1- (3-Br-Ph) PYR-4-yl], [BF10; 1- (4-Br-Ph) PYR-4-yl], [BF11; 1- (2-Me-Ph) PYR-4-yl], [BF12; 1- (3-Me-Ph) PYR-4-yl], [BF13; 1- (4-Me-Ph) PYR-4 1- (2-Et-Ph) PYR-4-yl], [BF15; 1- (3-Et-Ph) PYR-4-yl], [BF16; 1- (4-) Et-Ph) PYR-4- yl], [BF17; 1- (2-CF 3 -Ph) PYR-4-yl], [BF18; 1- (3-CF 3 -Ph) PYR-4-yl] , [BF19; 1- (4- CF 3 -Ph) PYR-4-yl], [BF20; 1- (2-OMe-Ph) PYR-4-yl], [BF21; 1- (3-OMe- Ph) PYR-4-yl], [BF22; 1- (4-OMe-Ph) PYR-4-yl], [BF23; 1- (2-OEt-Ph) PYR-4-yl], [BF24; 1- (3-OEt-Ph) PYR-4-yl], [BF25; 1- (4-OEt-Ph) PYR-4-yl], [BF26; 1- (4-F-2-F-Ph) ) PYR-4-yl], [BF27; 1- (4-Cl-2-F-Ph) PYR-4-yl], [BF28; 1- (4-Br-2-F-Ph) PYR-4 -yl], [BF29; 1- (4-Me-2-F-Ph) PYR-4-yl], [BF30; 1- (4-Et-2-F-Ph) PYR-4-yl], [BF31; 1- (4-CF 3 -2-F-Ph) PYR-4-yl], [BF32; 1- (4-OMe-2-F-Ph) PYR-4-yl], [BF33; 1- (4-OEt-2-F-Ph) PYR-4-yl], [BF34; 1- (4-F-2-Cl-Ph) PYR-4-yl], [BF35; 4-Cl-2-Cl-Ph) PYR-4-yl], [BF 36; 1- (4-Br-2-Cl-Ph) PYR-4-yl], [BF 37; 1- (4-Me-) 2-Cl-Ph) PYR-4-yl], [BF 38; 1- (4-Et-2-Cl-Ph) PYR-4-yl], [BF 39; 1- (4-CF ₃ -2-Cl] -Ph) PYR-4-yl], [BF40; 1- (4-OMe-2-Cl-Ph) PYR-4-yl], [BF41; 1- (4-OEt-2-Cl-Ph) PYR -4-yl], [BF42; 1- (4-F-2-Me-Ph) PYR-4-yl], [BF43; 1- (4-Cl-2-Me-Ph) PYR-4-yl ], [BF44; 1- (4-Br-2-Me-Ph) PYR-4-yl], [BF45; 1- (4-Me-2-Me-Ph) PYR-4-yl], [BF46] ; 1- (4-Et-2 -Me-Ph) PYR-4-yl], [BF47; 1- (4-CF 3 -2-Me-Ph) PYR-4-yl], [BF48; 1- (4-OMe-2-Me-Ph) PYR-4-yl], [BF49; 1- (4-OEt-2-Me-Ph) PYR-4-yl], [BF50; 1- (4-F) -2-OMe-Ph) PYR-4-yl], [BF51; 1- (4-Cl-2-OMe-Ph) PYR-4-yl], [BF52; 1- (4-Br-2-OMe) -Ph) PYR-4-yl], [BF53; 1- (4-Me-2-OMe-Ph) PYR-4-yl], [BF54; 1- (4-Et-2-OMe-Ph) PYR -4-yl], [BF55; 1- (4-CF 3 -2-OMe-Ph) PYR-4-yl], [BF56; 1- (4-OMe-2-OMe-Ph) PYR-4- yl], [BF57; 1- (4-OEt-2-OMe-Ph) PYR-4-yl], [BF58; 1- (4-F-2-OEt-Ph) PYR-4-yl], [BF4; BF59; 1- (4-Cl-2-OEt-Ph) PYR-4-yl], [BF60; 1- (4-Br-2-OEt-Ph) PYR-4-yl], [BF61; (4-Me-2-OEt-Ph) PYR-4-yl], [BF62; 1- (4-Et-2-OEt-Ph) PYR-4-yl], [BF63; 1- (4-CF) _{3 -2-OEt-Ph) PYR} -4-yl], [BF64; 1- (4-OMe-2-OEt-Ph) PYR-4-yl], [BF65; 1- (4-OEt-2- O Et-Ph) PYR-4-yl], [BF66; 3-Ph-1-Me-PYR-5-yl], [BF67; 3- (2-F-Ph) -1-Me-PYR-5- yl], [BF 68; 3- (3-F-Ph) -1-Me-PYR-5-yl], [BF 69; 3- (4-F-Ph) -1-Me-PYR-5-yl] , [BF70; 3- (2-Cl-Ph) -1-Me-PYR-5-yl], [BF71; 3- (3-Cl-Ph) -1-Me-PYR-5-yl], [BF70; BF 72; 3- (4-Cl-Ph) -1-Me-PYR-5-yl], [BF 73; 3- (2-Br-Ph) -1-Me-PYR-5-yl], [BF 74; 3- (3-Br-Ph) -1-Me-PYR-5-yl], [BF 75; 3- (4-Br-Ph) -1-Me-PYR-5-yl], [BF 76; 3- (2-Me-Ph) -1-Me-PYR-5-yl], [BF 77; 3- (3-Me-Ph) -1-Me-PYR-5-yl], [BF 78; 3- (4) -Me-Ph) -1-Me-PYR-5-yl], [BF 79; 3- (2-Et-Ph) -1-Me-PYR-5-yl], [BF 80; 3- (3-Et) -Ph) -1-Me-PYR- 5-yl], [BF81; 3- (4-Et-Ph) -1-Me-PYR-5-yl], [BF82; 3- (2-CF 3 - Ph) -1-Me-PYR- 5-yl], [BF83; 3- (3-CF 3 -Ph) -1-Me-PYR-5-yl], [BF84; 3- (4-CF 3 - Ph) -1-Me-PYR-5-yl], [BF 85; 3- (2-OMe-Ph) -1-Me-PYR-5-yl], [BF 86; 3- (3-OMe-Ph) -1-Me-PYR-5-yl], [BF 87; 3- (4-OMe-Ph) -1-Me-PYR-5-yl], [BF 88; 3- (2-OEt-Ph) -1 -Me-PYR-5-yl], [BF 89; 3- (3-OEt-Ph) -1-Me-PYR-5-yl], [BF 90; 3- (4-OEt-Ph) -1-Me -PYR-5-yl], [BF 91; 3- (4-F-2-F-Ph) -1-Me-PYR-5-yl], [BF 92; 3- (4-Cl-2-F-) Ph) -1-Me-PYR-5-yl], [BF 93; 3- (4-Br-2-F-Ph) -1-Me-PYR-5-yl], [BF 94; Me-2-F-Ph) -1-Me-PYR-5-yl], [BF 95; 3 - (4-Et-2- F-Ph) -1-Me-PYR-5-yl], [BF96; 3- (4-CF 3 -2-F-Ph) -1-Me-PYR-5- yl], [BF 97; 3- (4-OMe-2-F-Ph) -1-Me-PYR-5-yl], [BF 98; 3- (4-OEt-2-F-Ph) -1-] Me-PYR-5-yl], [BF99; 3- (4-F-2-Cl-Ph) -1-Me-PYR-5-yl], [BF100; 3- (4-Cl-2-Cl) -Ph) -1-Me-PYR-5-yl],

[BF101; 3- (4-Br-2-Cl-Ph) -1-Me-PYR-5-yl], [BF102; 3- (4-Me-2-Cl-Ph) -1-Me-PYR -5-yl], [BF103; 3- (4-Et-2-Cl-Ph) -1-Me-PYR-5-yl], [BF104; 3- (4-CF 3 -2-Cl-Ph )-1-Me-PYR-5-yl], [BF105; 3- (4-OMe-2-Cl-Ph) -1-Me-PYR-5-yl], [BF106; 3- (4-OEt) -2-Cl-Ph) -1-Me-PYR-5-yl], [BF107; 3- (4-F-2-Me-Ph) -1-Me-PYR-5-yl], [BF108; 3- (4-Cl-2-Me-Ph) -1-Me-PYR-5-yl], [BF109; 3- (4-Br-2-Me-Ph) -1-Me-PYR-5- yl], [BF110; 3- (4-Me-2-Me-Ph) -1-Me-PYR-5-yl], [BF111; 3- (4-Et-2-Me-Ph) -1-] Me-PYR-5-yl] , [BF112; 3- (4-CF 3 -2-Me-Ph) -1-Me-PYR-5-yl], [BF113; 3- (4-OMe-2- Me-Ph) -1-Me-PYR-5-yl], [BF 114; 3- (4-OEt-2-Me-Ph) -1-Me-PYR-5-yl], [BF 115; 4-F-2-OMe-Ph) -1-Me-PYR-5-yl], [BF116; 3- (4-Cl-2-OMe-Ph) -1-Me-PYR-5-yl], [BF117; 3- (4-Br-2-OMe-Ph) -1-Me-PYR-5-yl], [BF118; 3- (4-Me-2-OMe-Ph) -1-Me-PYR -5-yl], [BF119; 3- (4-Et-2-OMe-Ph) -1-Me-PYR-5-yl], [BF120; 3- (4-CF 3 -2-OMe-Ph )-1 -Me-PYR-5-yl], [BF121; 3- (4-OMe-2-OMe-Ph) -1-Me-PYR-5-yl], [BF122; 3- (4-OEt) -2-OMe-Ph) -1-Me-PYR-5-yl], [BF 123; 3- (4-F-2-OEt-Ph) -1-Me-PYR-5-yl], [BF 124; 3- (4-Cl-2-OEt-Ph) -1-Me-PYR-5-yl], [BF125; 3- (4-Br-2-OEt-Ph) -1-Me-PYR-5- yl], [B F126; 3- (4-Me-2-OEt-Ph) -1-Me-PYR-5-yl], [BF127; 3- (4-Et-2-OEt-Ph) -1-Me-PYR- 5-yl], [BF128; 3- (4-CF 3 -2-OEt-Ph) -1-Me-PYR-5-yl], [BF129; 3- (4-OMe-2-OEt-Ph) -1-Me-PYR-5-yl], [BF130; 3- (4-OEt-2-OEt-Ph) -1-Me-PYR-5-yl], [BF131; 5-Ph-1-Me -PYR-3-yl], [BF132; 5- (2-F-Ph) -1-Me-PYR-3-yl], [BF133; 5- (3-F-Ph) -1-Me-PYR -3-yl], [BF134; 5- (4-F-Ph) -1-Me-PYR-3-yl], [BF135; 5- (2-Cl-Ph) -1-Me-PYR-3 -yl], [BF136; 5- (3-Cl-Ph) -1-Me-PYR-3-yl], [BF137; 5- (4-Cl-Ph) -1-Me-PYR-3-yl ], [BF 138; 5- (2-Br-Ph) -1-Me-PYR-3-yl], [BF 139; 5- (3-Br-Ph) -1-Me-PYR-3-yl], [BF140; 5- (4-Br-Ph) -1-Me-PYR-3-yl], [BF141; 5- (2-Me-Ph) -1-Me-PYR-3-yl], [BF142 5- (3-Me-Ph) -1-Me-PYR-3-yl], [BF 143; 5- (4-Me-Ph) -1-Me-PYR-3-yl], [BF 144; -(2-Et-Ph) -1-Me-PYR-3-yl], [BF145; 5- (3-Et-Ph) -1-Me-PYR-3-yl], [BF146; 4-Et-Ph) -1-Me-PYR-3-yl], [BF 147; 5- (2-CF ₃ -Ph) -1-Me-PYR-3-yl], [BF 148; 5- (3) _{-CF 3 -Ph) -1-Me-} PYR-3-yl], [BF149; 5- (4-CF 3 -Ph) -1-Me-PYR-3-yl], [BF150; 5- (2 -OMe-Ph) -1-Me-PYR-3-yl], [BF 151; 5- (3-OMe-Ph) -1-Me-PYR-3-yl], [BF 152; 5- (4-OMe) -Ph) -1-Me-PYR-3-yl], [BF153; 5- (2-OEt-Ph) -1-Me-PYR-3-yl], [BF154; OEt-Ph) -1-Me-PYR-3-yl], [BF 155; 5- (4-OEt-Ph) -1-Me-PYR-3-yl], [BF 156; 5- (4-F-) 2-F-Ph) -1-Me-PYR-3-yl], [BF 157; 5- (4-Cl-2-F-Ph) -1-Me-PYR-3-yl], [BF 158; -(4-Br-2-F-Ph) -1-Me-PYR-3-yl], [BF 159; 5- (4-Me-2-F-Ph) -1-Me-PYR-3-yl ], [BF160; 5- (4 -Et-2-F-Ph) -1-Me-PYR-3-yl], [BF161; 5- (4-CF 3 -2-F-Ph) -1- Me-PYR-3-yl], [BF162; 5- (4-OMe-2-F-Ph) -1-Me-PYR-3-yl], [BF163; 5- (4-OEt-2-F) -Ph) -1-Me-PYR-3-yl], [BF 164; 5- (4-F-2-Cl-Ph) -1-Me-PYR-3-yl], [BF 165; 5- (4) -Cl-2-Cl-Ph) -1-Me-PYR-3-yl], [BF166; 5- (4-Br-2-Cl-Ph) -1-Me-PYR-3-yl], [ BF 167; 5- (4-Me-2-Cl-Ph) -1-Me-PYR-3-yl], [BF 168; 5- (4-Et-2-Cl-Ph) -1-Me-PYR- 3-yl], [BF169; 5- (4-CF 3 -2-Cl-Ph) -1-Me-PYR-3-yl], [BF170; 5- (4-OMe-2-Cl-Ph) -1-Me-PYR-3-yl], [BF 171; 5- (4-OEt-2-Cl-Ph) -1-Me-PYR-3-yl], [BF 172; 5- (4-F-) 2-Me-Ph) -1-Me-PYR-3-yl], [BF 173; 5- (4-Cl-2-Me-Ph) -1-Me-PYR-3-yl], [BF 174; -(4-Br-2-Me-Ph) -1-Me-PYR-3-yl], [BF175; 5- (4-Me-2-Me-Ph) -1-Me-PYR-3-yl ], [BF176; 5- (4 -Et-2-Me-Ph) -1-Me-PYR-3-yl], [BF177; 5- (4-CF 3 -2-Me-Ph) -1- Me-PYR-3-yl], [BF 178; 5- (4-OMe-2-Me-Ph) -1-Me-PYR-3-yl], [BF 179; 5- (4-OEt-2-Me) -Ph) -1-Me-PYR-3-yl], [B F180; 5- (4-F-2-OMe-Ph) -1-Me-PYR-3-yl], [BF181; 5- (4-Cl-2-OMe-Ph) -1-Me-PYR- 3-yl], [BF 182; 5- (4-Br-2-OMe-Ph) -1-Me-PYR-3-yl], [BF183; 5- (4-Me-2-OMe-Ph)- 1-Me-PYR-3-yl], [BF 184; 5- (4-Et-2-OMe-Ph) -1-Me-PYR-3-yl], [BF 185; 5- (4-CF _3- 2-OMe-Ph) -1-Me-PYR-3-yl], [BF 186; 5- (4-OMe-2-OMe-Ph) -1-Me-PYR-3-yl], [BF 187; -(4-OEt-2-OMe-Ph) -1-Me-PYR-3-yl], [BF188; 5- (4-F-2-OEt-Ph) -1-Me-PYR-3-yl ], [BF 189; 5- (4-Cl-2-OEt-Ph) -1-Me-PYR-3-yl], [BF190; 5- (4-Br-2-OEt-Ph) -1-Me -PYR-3-yl], [BF191; 5- (4-Me-2-OEt-Ph) -1-Me-PYR-3-yl], [BF192; 5- (4-Et-2-OEt-) Ph) -1-Me-PYR-3-yl], [BF 193; 5- (4-CF ₃ 2-OEt-Ph) -1-Me-PYR-3-yl], [BF 194; 5- (4) -OMe-2-OEt-Ph) -1-Me-PYR-3-yl], [BF195; 5- (4-OEt-2-OEt-Ph) -1-Me-PYR-3-yl], [BF4; BF196; 1-phenyl-1,2,4-TRI-3-yl], [BF197; 1- (2-F-Ph) -1,2,4-TRI-3-yl], [BF198; (3-F-Ph) -1,2,4-TRI-3-yl], [BF 199; 1- (4-F-Ph) -1,2,4-TRI-3-yl], [BF 200; 1- (2-Cl-Ph) -1,2,4-TRI-3-yl],

[BF201; 1- (3-Cl-Ph) -1,2,4-TRI-3-yl], [BF202; 1- (4-Cl-Ph) -1,2,4-TRI-3-yl ], [BF 203; 1- (2-Br-Ph) -1,2,4-TRI-3-yl], [BF 204; 1- (3-Br-Ph) -1,2,4-TRI-3 -yl], [BF205; 1- (4-Br-Ph) -1,2,4-TRI-3-yl], [BF206; 1- (2-Me-Ph) -1,2,4-TRI -3-yl, [BF207; 1- (3-Me-Ph) -1,2,4-TRI-3-yl], [BF208; 1- (4-Me-Ph) -1,2,4 -TRI-3-yl], [BF 209; 1- (2-Et-Ph) -1,2,4-TRI-3-yl], [BF 210; 1- (3-Et-Ph) -1, 2 , 4-TRI-3-yl], [BF211; 1- (4-Et-Ph) -1,2,4-TRI-3-yl], [BF212; 1- (2-CF ₃ -Ph)- 1,2,4-TRI-3-yl], [BF 213; 1- (3-CF ₃ -Ph) -1, 2, 4-TRI-3-yl], [BF 214; 1- (4-CF ₃₎ -Ph) -1,2,4-TRI-3-yl], [BF 215; 1- (2-OMe-Ph) -1, 2, 4-TRI-3-yl], [BF 216; -OMe-Ph) -1,2,4-TRI-3-yl], [BF217; 1- (4-OMe-Ph) -1,2,4-TRI-3-yl], [BF218; 1- (2-OEt-Ph) -1,2,4-TRI-3-yl], [BF 219; 1- (3-OEt-Ph) -1,2,4-TRI-3-yl], [BF 220; 1- (4-OEt-Ph) -1,2,4-TRI-3-yl], [BF221; 1- (4-F-2-F-Ph) -1,2,4-TRI-3- yl], [BF222; 1- (4-Cl-2-F-Ph) -1,2,4-TRI-3-yl], [BF223; 1- (4-Br-2-F-Ph)- 1,2,4-TRI-3-yl], [BF 224; 1- (4-Me-2-F-Ph) -1, 2, 4-TRI-3-yl], [BF 225; 1- (4) -Et-2-F-Ph) -1,2,4-TRI-3-yl], [BF 226; 1- (4-CF ₃ -2-F-Ph) -1,2,4-TRI-3 -yl, [BF 227; 1- (4-OMe-2-F-Ph) -1, 2, 4-TRI-3-yl], [BF 228; (4-OEt-2-F-Ph) -1,2,4-TRI-3-yl], [BF 229; 1- (4-F-2-Cl-Ph) -1,2,4-TRI- 3-yl], [BF 230; 1- (4-Cl-2-Cl-Ph) -1, 2, 4-TRI-3-yl], [BF 231; 1- (4-Br-2-Cl-Ph) ) -1,2,4-TRI-3-yl], [BF 232; 1- (4-Me-2-Cl-Ph) -1, 2, 4-TRI-3-yl], [BF 233; (4-Et-2-Cl-Ph) -1,2,4-TRI-3-yl], [BF 234; 1- (4-CF ₃ -2-Cl-Ph) -1,2,4-TRI -3-yl], [BF235; 1- (4-OMe-2-Cl-Ph) -1,2,4-TRI-3-yl], [BF236; 1- (4-OEt-2-Cl- Ph) -1,2,4-TRI-3-yl], [BF 237; 1- (4-F-2-Me-Ph) -1,2,4-TRI-3-yl], [BF 238; 1 -(4-Cl-2-Me-Ph) -1,2,4-TRI-3-yl], [BF 239; 1- (4-Br-2-Me-Ph) -1,2,4-TRI -3-yl], [BF240; 1- (4-Me-2-Me-Ph) -1,2,4-TRI-3-yl], [BF241; 1- (4-Et-2-Me-) Ph) -1,2,4-TRI-3-yl], [BF 242; 1- (4-CF ₃ -2-Me-Ph) -1,2,4-TRI-3-yl], [BF 243; 1- (4-OMe-2-Me-Ph) -1,2,4-TRI-3-yl], [BF244; 1- (4-OEt-2-Me-Ph) -1,2,4- TRI-3-yl], [BF 245; 1- (4-F-2-OMe-Ph) -1, 2, 4-TRI-3-yl], [BF 246; 1- (4-Cl-2-OMe) -Ph) -1,2,4-TRI-3-yl], [BF 247; 1- (4-Br-2-OMe-Ph) -1,2,4-TRI-3-yl], [BF 248; 1- (4-Me-2-OMe-Ph) -1,2,4-TRI-3-yl], [BF 249; 1- (4-Et-2-OMe-Ph) -1,2,4- TRI-3-yl], [ BF250; 1- (4-CF 3 -2-OMe-Ph) -1,2,4-TRI-3-yl], [BF251; 1- (4-OMe-2- OMe-Ph) -1,2,4-TRI-3-yl], [BF 252; 1- (4-OEt-2-OMe-Ph) -1,2,4 -TRI-3-yl], [BF 253; 1- (4-F-2-OEt-Ph) -1, 2, 4-TRI-3-yl], [BF 254; 1- (4-Cl-2-) OEt-Ph) -1,2,4-TRI-3-yl], [BF255; 1- (4-Br-2-OEt-Ph) -1,2,4-TRI-3-yl], [BF256 1- (4-Me-2-OEt-Ph) -1,2,4-TRI-3-yl], [BF 257; 1- (4-Et-2-OEt-Ph) -1,2,4; -TRI-3-yl], [ BF258; 1- (4-CF 3 -2-OEt-Ph) -1,2,4-TRI-3-yl], [BF259; 1- (4-OMe-2 -OEt-Ph) -1,2,4-TRI-3-yl], [BF 260; 1- (4-OEt-2-OEt-Ph) -1,2,4-TRI-3-yl], BF261; 2-phenyl-1,2,3-TRI-4-yl], [BF262; 2- (2-F-Ph) -1,2,3-TRI-4-yl], [BF263; (3-F-Ph) -1,2,3-TRI-4-yl], [BF 264; 2- (4-F-Ph) -1,2,3-TRI-4-yl], [BF 265; 2- (2-Cl-Ph) -1,2,3-TRI-4-yl], [BF 266; 2- (3-Cl-Ph) -1,2,3-TRI-4-yl], [ BF 267; 2- (4-Cl-Ph) -1,2,3-TRI-4-yl], [BF268; 2- (2-Br-Ph) -1,2,3-TRI-4-yl] , [BF 269; 2- (3-Br-Ph) -1,2,3-TRI-4-yl], [BF 270; 2- (4-Br-Ph) -1,2,3-TRI-4- yl], [BF 271; 2- (2-Me-Ph) -1,2,3-TRI-4-yl], [BF 272; 2- (3-Me-Ph) -1,2,3-TRI- 4-yl], [BF273; 2- (4-Me-Ph) -1,2,3-TRI-4-yl], [BF274; 2- (2-Et-Ph) -1,2,3- TRI-4-yl], [BF275; 2- (3-Et-Ph) -1,2,3-TRI-4-yl], [BF276; 2- (4-Et-Ph) -1,2, 6 3-TRI-4-yl], [BF 277; 2- (2-CF ₃ -Ph) -1,2,3-TRI-4-yl], [BF 278; 2- (3-CF ₃ -Ph)- 1,2,3-TRI-4-yl], [BF 279; 2- (4-CF ₃ -Ph) -1,2,3 -TRI-4-yl], [BF 280; 2- (2-OMe-Ph) -1,2,3-TRI-4-yl], [BF 281; 2- (3-OMe-Ph) -1, 2 , 3-TRI-4-yl], [BF282; 2- (4-OMe-Ph) -1,2,3-TRI-4-yl], [BF283; 2- (2-OEt-Ph) -1 , 2,3-TRI-4-yl], [BF284; 2- (3-OEt-Ph) -1,2,3-TRI-4-yl], [BF285; 2- (4-OEt-Ph) -1,2,3-TRI-4-yl], [BF 286; 2- (4-F-2-F-Ph) -1,2,3-TRI-4-yl], [BF 287; 2- ( 4-Cl-2-F-Ph) -1,2,3-TRI-4-yl], [BF 288; 2- (4-Br-2-F-Ph) -1,2,3-TRI-4 -yl], [BF 289; 2- (4-Me-2-F-Ph) -1,2,3-TRI-4-yl], [BF 290; 2- (4-Et-2-F-Ph) -1,2,3-TRI-4-yl] , [BF291; 2- (4-CF 3 -2-F-Ph) -1,2,3-TRI-4-yl], [BF292; 2- (4-OMe-2-F-Ph) -1,2,3-TRI-4-yl], [BF 293; 2- (4-OEt-2-F-Ph) -1,2,3-TRI- 4-yl], [BF 294; 2- (4-F-2-Cl-Ph) -1,2,3-TRI-4-yl], [BF 295; 2- (4-Cl-2-Cl-Ph) )-1,2,3-TRI-4-yl], [BF 296; 2- (4-Br-2-Cl-Ph) -1,2,3-TRI-4-yl], [BF 297; 2- (4-Me-2-Cl-Ph) -1,2,3-TRI-4-yl], [BF 298; 2- (4-Et-2-Cl-Ph) -1,2,3-TRI- 4-yl], [BF 299; 2- (4-CF3-2-Cl-Ph) -1,2,3-TRI-4-yl], [BF300; 2- (4-OMe-2-Cl-Ph) ) -1,2,3-TRI-4-yl],

[BF301; 2- (4-OEt-2-Cl-Ph) -1,2,3-TRI-4-yl], [BF302; 2- (4-F-2-Me-Ph) -1,2 , 3-TRI-4-yl], [BF 303; 2- (4-Cl-2-Me-Ph) -1,2,3-TRI-4-yl], [BF 304; 2- (4-Br-) 2-Me-Ph) -1,2,3-TRI-4-yl], [BF 305; 2- (4-Me-2-Me-Ph) -1,2,3-TRI-4-yl], [BF306; 2- (4-Et -2-Me-Ph) -1,2,3-TRI-4-yl], [BF307; 2- (4-CF 3 -2-Me-Ph) -1, 2,3-TRI-4-yl], [BF308; 2- (4-OMe-2-Me-Ph) -1,2,3-TRI-4-yl], [BF309; 2- (4-OEt) -2-Me-Ph) -1,2,3-TRI-4-yl], [BF 310; 2- (4-F-2-OMe-Ph) -1,2,3-TRI-4-yl] , [BF 311; 2- (4-Cl-2-OMe-Ph) -1,2,3-TRI-4-yl], [BF312; 2- (4-Br-2-OMe-Ph) -1, 2,3-TRI-4-yl], [BF313; 2- (4-Me-2-OMe-Ph) -1,2,3-TRI-4-yl], [BF314; 2- (4-Et) -2-OMe-Ph) -1,2,3-TRI-4-yl], [BF 315; 2- (4-CF ₃ -2-OMe-Ph) -1,2,3-TRI-4-yl ], [BF316; 2- (4-OMe-2-OMe-Ph) -1,2,3-TRI-4-yl], [BF317; 2- (4-OEt-2-OMe-Ph) -1 , 2,3-TRI-4-yl], [BF 318; 2- (4-F-2-OEt-Ph) -1,2,3-TRI-4-yl], [BF 319; 2- (4-) Cl-2-OEt-Ph) -1,2,3-TRI-4-yl], [BF 320; 2- (4-Br-2-OEt-Ph) -1,2,3-TRI-4-yl ], [BF 321; 2- (4-Me-2-OEt-Ph) -1,2,3-TRI-4-yl], [BF 322; 2- (4-Et-2-OEt-Ph) -1 , 2,3-TRI-4-yl], [BF 323; 2- (4-CF ₃ -2-OEt-Ph) -1,2,3-TRI-4-yl], [BF 324; 2- (4) -OMe-2-OEt-Ph) -1,2,3-TRI-4-yl], [BF 325; 2- (4-O) Et-2-OEt-Ph) -1,2,3-TRI-4-yl], [BF 326; 2-phenylTET-5-yl], [BF 327; 2- (2-F-Ph) TET-5- yl], [BF 328; 2- (3-F-Ph) TET-5-yl], [BF 329; 2- (4-F-Ph) TET-5-yl], [BF 330; 2- (2-Cl) -Ph) TET-5-yl], [BF 331; 2- (3-Cl-Ph) TET-5-yl], [BF332; 2- (4-Cl-Ph) TET-5-yl], [BF333 2- (2-Br-Ph) TET-5-yl], [BF334; 2- (3-Br-Ph) TET-5-yl], [BF335; 2- (4-Br-Ph) TET- 5-yl], [BF336; 2- (2-Me-Ph) TET-5-yl], [BF 337; 2- (3-Me-Ph) TET-5-yl], [BF338; 2- (4) -Me-Ph) TET-5-yl], [BF 339; 2- (2-Et-Ph) TET-5-yl], [BF 340; 2- (3-Et-Ph) TET-5-yl], [BF 341; 2- (4-Et-Ph) TET-5-yl], [BF 342; 2- (2-CF ₃ -Ph) TET-5-yl], [BF 343; 2- (3-CF _3- Ph) TET-5-yl], [BF 344; 2- (4-CF ₃ -Ph) TET-5-yl], [BF 345; 2- (2-OMe-Ph) TET-5-yl], [BF 346 2- (3-OMe-Ph) TET-5-yl], [BF347; 2- (4-OMe-Ph) TET-5-yl], [BF348; 2- (2-OEt-Ph) TET- 5-yl], [BF 349; 2- (3-OEt-Ph) TET-5-yl], [BF 350; 2- (4-OEt-Ph) TET-5-yl], [BF 351; 2- (4) -F-2-F-Ph) TET-5-yl], [BF 352; 2- (4-Cl-2-F-Ph) TET-5-yl], [BF 353; 2- (4-Br-2) -F-Ph) TET-5-yl], [BF 354; 2- (4-Me-2-F-Ph) TET-5-yl], [BF 355; 2- (4-Et-2-F-Ph) ) TET-5-yl], [BF 356; 2- (4-CF3-2-F-Ph) TET-5-yl], [BF357; 2- (4-OMe-2-F-Ph) TET-5] -yl], [BF 358; 2- (4-OEt-2-F-Ph) TET-5-yl], [BF3 59; 2- (4-F-2-Cl-Ph) TET-5-yl], [BF 360; 2- (4-Cl-2-Cl-Ph) TET-5-yl], [BF 361; 2- (4-Br-2-Cl-Ph) TET-5-yl], [BF 362; 2- (4-Me-2-Cl-Ph) TET-5-yl], [BF 363; 2- (4-Et) -2-Cl-Ph) TET-5-yl], [BF 364; 2- (4-CF ₃ -2-Cl-Ph) TET-5-yl], [BF 365; 2- (4-OMe-2-) Cl-Ph) TET-5-yl], [BF 366; 2- (4-OEt-2-Cl-Ph) TET-5-yl], [BF367; 2- (4-F-2-Me-Ph) TET-5-yl], [BF 368; 2- (4-Cl-2-Me-Ph) TET-5-yl], [BF 369; 2- (4-Br-2-Me-Ph) TET-5- yl], [BF370; 2- (4-Me-2-Me-Ph) TET-5-yl], [BF371; 2- (4-Et-2-Me-Ph) TET-5-yl], [ _{BF372; 2- (4-CF 3} -2-Me-Ph) TET-5-yl], [BF373; 2- (4-OMe-2-Me-Ph) TET-5-yl], [BF374; 2 -(4-OEt-2-Me-Ph) TET-5-yl], [BF 375; 2- (4-F-2-OMe-Ph) TET-5-yl], [BF 376; 2- (4-) Cl-2-OMe-Ph) TET-5-yl], [BF 377; 2- (4-Br-2-OMe-Ph) TET-5-yl], [BF 378; 2- (4-Me-2-) OMe-Ph) TET-5-yl], [BF379; 2- (4-Et-2-OMe-Ph) TET-5-yl], [BF380; 2- (4-CF ₃ -2-OMe-Ph] ) TET-5-yl], [BF 381; 2- (4-OMe-2-OMe-Ph) TET-5-yl], [BF 382; 2- (4-OEt-2-OMe-Ph) TET-5] -yl], [BF 383; 2- (4-F-2-OEt-Ph) TET-5-yl], [BF 384; 2- (4-Cl-2-OEt-Ph) TET-5-yl], [BF 385; 2- (4-Br-2-OEt-Ph) TET-5-yl], [BF 386; 2- (4-Me-2-OEt-Ph) TET-5-yl], [BF 387; 2 - (4-Et-2- OEt-Ph) TET-5-yl], [BF388; 2- (4-CF 3 -2-OEt -Ph) TET-5-yl], [BF 389; 2- (4-OMe-2-OEt-Ph) TET-5-yl], [BF390; 2- (4-OEt-2-OEt-Ph) TET -5-yl], [BF 391; 3-phenylTHI-5-yl], [BF 392; 3- (2-F-Ph) THI-5-yl], [BF 393; 3- (3-F-Ph) THI -5-yl], [BF 394; 3- (4-F-Ph) THI-5-yl], [BF 395; 3- (2-Cl-Ph) THI-5-yl], [BF 396; 3-Cl-Ph) THI-5-yl], [BF397; 3- (4-Cl-Ph) THI-5-yl], [BF398; 3- (2-Br-Ph) THI-5-yl] , [BF 399; 3- (3-Br-Ph) THI-5-yl], [BF400; 3- (4-Br-Ph) THI-5-yl],

[BF401; 3- (2-Me-Ph) THI-5-yl], [BF402; 3- (3-Me-Ph) THI-5-yl], [BF403; 3- (4-Me-Ph) THI-5-yl], [BF404; 3- (2-Et-Ph) THI-5-yl], [BF405; 3- (3-Et-Ph) THI-5-yl], [BF406; (4-Et-Ph) THI-5-yl], [BF 407; 3- (2-CF ₃ -Ph) THI 5-yl], [BF 408; 3- (3-CF ₃ -Ph) THI-5 -yl], [BF409; 3- ( 4-CF 3 -Ph) THI-5-yl], [BF410; 3- (2-OMe-Ph) THI-5-yl], [BF411; 3- (3 -OMe-Ph) THI-5-yl], [BF412; 3- (4-OMe-Ph) THI-5-yl], [BF413; 3- (2-OEt-Ph) THI-5-yl], [BF414; 3- (3-OEt-Ph) THI-5-yl], [BF415; 3- (4-OEt-Ph) THI-5-yl], [BF416; 3- (4-F-2-) F-Ph) THI-5-yl], [BF 417; 3- (4-Cl-2-F-Ph) THI-5-yl], [BF418; 3- (4-Br-2-F-Ph) THI-5-yl], [BF 419; 3- (4-Me-2-F-Ph) THI-5-yl], [BF 420; 3- (4-Et-2-F-Ph) THI-5- yl], [BF421; 3- ( 4-CF 3 -2-F-Ph) THI-5-yl], [BF422; 3- (4-OMe-2-F-Ph) THI-5-yl], [BF423; 3- (4-OEt-2-F-Ph) THI-5-yl], [BF424; 3- (4-F-2-Cl-Ph) THI-5-yl], [BF425; 3 -(4-Cl-2-Cl-Ph) THI-5-yl], [BF 426; 3- (4-Br-2-Cl-Ph) THI-5-yl], [BF 427; Me-2-Cl-Ph) THI-5-yl], [BF 428; 3- (4-Et-2-Cl-Ph) THI-5-yl], [BF 429; 3- (4-CF ₃ -2] -Cl-Ph) THI-5-yl], [BF 430; 3- (4-OMe-2-Cl-Ph) THI-5-yl], [BF 431; 3- (4-OEt-2-Cl-Ph) ) THI-5-yl], [BF 432; 3- (4-F-2-Me-Ph) THI-5-yl], [BF 43 3; 3- (4-Cl-2-Me-Ph) THI-5-yl], [BF 434; 3- (4-Br-2-Me-Ph) THI-5-yl], [BF 435; (4-Me-2-Me-Ph) THI-5-yl], [BF 436; 3- (4-Et-2-Me-Ph) THI-5-yl], [BF 437; 3- (4-CF) _{3 -2-Me-Ph) THI} -5-yl], [BF438; 3- (4-OMe-2-Me-Ph) THI-5-yl], [BF439; 3- (4-OEt-2- Me-Ph) THI-5-yl], [BF440; 3- (4-F-2-OMe-Ph) THI-5-yl], [BF441; 3- (4-Cl-2-OMe-Ph) THI-5-yl], [BF 442; 3- (4-Br-2-OMe-Ph) THI-5-yl], [BF 443; 3- (4-Me-2-OMe-Ph) THI-5- yl], [BF444; 3- ( 4-Et-2-OMe-Ph) THI-5-yl], [BF445; 3- (4-CF 3 -2-OMe-Ph) THI-5-yl], [BF446; 3- (4-OMe-2-OMe-Ph) THI-5-yl], [BF 447; 3- (4-OEt-2-OMe-Ph) THI-5-yl], [BF448; -(4-F-2-OEt-Ph) THI-5-yl], [BF 449; 3- (4-Cl-2-OEt-Ph) THI-5-yl], [BF450; Br-2-OEt-Ph) THI-5-yl], [BF 451; 3- (4-Me-2-OEt-Ph) THI-5-yl], [BF 452; 3- (4-Et-2-) OEt-Ph) THI-5-yl], [BF 453; 3- (4-CF ₃ -2-OEt-Ph) THI-5-yl], [BF 454; 3- (4-OMe-2-OEt-Ph) ) THI-5-yl], [BF 455; 3- (4-OEt-2-OEt-Ph) THI-5-yl], [BF 456; 5-phenylTHI-2-yl], [BF 457; 5- (2) -F-Ph) THI-2-yl], [BF 458; 5- (3-F-Ph) THI-2-yl], [BF459; 5- (4-F-Ph) THI-2-yl], [BF 460; 5- (2-Cl-Ph) THI-2-yl], [BF 461; 5- (3-Cl-Ph) THI-2-yl], [BF 462; 5- (4-Cl-Ph) THI-2-yl], [BF 463; 5- (2-Br-Ph) THI-2-yl] , [BF464; 5- (3-Br-Ph) THI-2-yl], [BF465; 5- (4-Br-Ph) THI-2-yl], [BF466; 5- (2-Me-Ph) ) THI-2-yl], [BF 467; 5- (3-Me-Ph) THI-2-yl], [BF 468; 5- (4-Me-Ph) THI-2-yl], [BF 469; -(2-Et-Ph) THI-2-yl], [BF 470; 5- (3-Et-Ph) THI-2-yl], [BF 471; 5- (4-Et-Ph) THI-2- yl], [BF 472; 5- (2-CF ₃ -Ph) THI-2-yl], [BF 473; 5- (3-CF ₃ -Ph) THI-2-yl], [BF 474; 5- (4) _{-CF 3 -Ph) THI-2-} yl], [BF475; 5- (2-OMe-Ph) THI-2-yl], [BF476; 5- (3-OMe-Ph) THI-2-yl] , [BF 477; 5- (4-OMe-Ph) THI-2-yl], [BF 478; 5- (2-OEt-Ph) THI-2-yl], [BF 479; 5- (3-OEt-Ph] ) THI-2-yl], [BF 480; 5- (4-OEt-Ph) THI-2-yl], [BF 481; 5- (4-F-2-F-Ph) THI-2-yl], [BF 482; 5- (4-Cl-2-F-Ph) THI-2-yl], [BF 483; 5- (4-Br-2-F-Ph) THI-2-yl], [BF 484; -(4-Me-2-F-Ph) THI-2-yl], [BF 485; 5- (4-Et-2-F-Ph) THI-2-yl], [BF 486; _{CF 3 -2-F-Ph)} THI-2-yl], [BF487; 5- (4-OMe-2-F-Ph) THI-2-yl], [BF488; 5- (4-OEt-2 -F-Ph) THI-2-yl], [BF 489; 5- (4-F-2-Cl-Ph) THI-2-yl], [BF 490; 5- (4-Cl-2-Cl-Ph) ) THI-2-yl], [BF 491; 5- (4-Br-2-Cl-Ph) THI-2-yl], [BF 492; 5- (4-Me-2-Cl-Ph) THI-2 -yl], [BF493; 5- ( 4-Et-2-Cl-Ph) THI-2-yl], [BF494; 5- (4-CF 3 -2-Cl-Ph) THI-2-yl] , [BF495; 5- (4-OMe-2-Cl-Ph) THI-2-yl], [BF496; 5- (4-OE) t-2-Cl-Ph) THI-2-yl], [BF 497; 5- (4-F-2-Me-Ph) THI-2-yl], [BF 498; 5- (4-Cl-2-) Me-Ph) THI-2-yl], [BF 499; 5- (4-Br-2-Me-Ph) THI-2-yl], [BF500; 5- (4-Me-2-Me-Ph) THI-2-yl],

[BF501; 5- (4-Et -2-Me-Ph) THI-2-yl], [BF502; 5- (4-CF 3 -2-Me-Ph) THI-2-yl], [BF503; 5- (4-OMe-2-Me-Ph) THI-2-yl], [BF 504; 5- (4-OEt-2-Me-Ph) THI-2-yl], [BF 505; 5- (4) -F-2-OMe-Ph) THI-2-yl], [BF 506; 5- (4-Cl-2-OMe-Ph) THI-2-yl], [BF 507; 5- (4-Br-2) -OMe-Ph) THI-2-yl], [BF508; 5- (4-Me-2-OMe-Ph) THI-2-yl], [BF509; 5- (4-Et-2-OMe-Ph) ) THI-2-yl], [BF510; 5- (4-CF 3 -2-OMe-Ph) THI-2-yl], [BF511; 5- (4-OMe-2-OMe-Ph) THI- 2-yl], [BF512; 5- (4-OEt-2-OMe-Ph) THI-2-yl], [BF513; 5- (4-F-2-OEt-Ph) THI-2-yl] , [BF514; 5- (4-Cl-2-OEt-Ph) THI-2-yl], [BF515; 5- (4-Br-2-OEt-Ph) THI-2-yl], [BF516; 5- (4-Me-2-OEt-Ph) THI-2-yl], [BF 517; 5- (4-Et-2-OEt-Ph) THI-2-yl], [BF518; 5- (4) _{-CF 3 -2-OEt-Ph)} THI-2-yl], [BF519; 5- (4-OMe-2-OEt-Ph) THI-2-yl], [BF520; 5- (4-OEt- 2-OEt-Ph) THI-2-yl], [BF521; 5-phenylTHI-3-yl], [BF522; 5- (2-F-Ph) THI-3-yl], [BF523; 3-F-Ph) THI-3-yl], [BF 524; 5- (4-F-Ph) THI-3-yl], [BF 525; 5- (2-Cl-Ph) THI-3-yl] , [BF 526; 5- (3-Cl-Ph) THI-3-yl], [BF 527; 5- (4-Cl-Ph) THI-3-yl], [BF 528; 5- (2-Br-Ph) ) THI-3-yl], [BF 529; 5- (3-Br-Ph) THI-3-yl], [BF 530; 5- (4-Br-Ph) THI-3-yl], [BF 531; 5 -(2-Me-Ph) THI-3-yl], [BF532; 5- (3-Me-Ph) THI-3-yl], [BF533; 5- (4-Me-Ph) THI-3-yl], [BF534; 5- (2-Et-Ph) THI-3-yl ], [BF535; 5- (3 -Et-Ph) THI-3-yl], [BF536; 5- (4-Et-Ph) THI-3-yl], [BF537; 5- (2-CF 3 -Ph) THI-3-yl], [BF 538; 5- (3-CF ₃ -Ph) THI-3-yl], [BF 539; 5- (4-CF ₃ -Ph) THI-3-yl], [BF 540; 5- (2-OMe-Ph) THI-3-yl], [BF 541; 5- (3-OMe-Ph) THI-3-yl], [BF 542; 5- (4-OMe-Ph) THI-3-yl], [BF 543; 5- (2-OEt-Ph) THI-3-yl], [BF 544; 5- (3-OEt-Ph) THI-3-yl], [BF 545; (4-OEt-Ph) THI-3-yl], [BF 546; 5- (4-F-2-F-Ph) THI-3-yl], [BF547; 5- (4-Cl-2-F) -Ph) THI-3-yl], [BF 548; 5- (4-Br-2-F-Ph) THI-3-yl], [BF 549; 5- (4-Me-2-F-Ph) THI -3-yl], [BF 550; 5- (4-Et-2-F-Ph) THI-3-yl], [BF 551; 5- (4-CF ₃ -2-F-Ph) THI-3- yl], [BF 552; 5- (4-OMe-2-F-Ph) THI-3-yl], [BF 553; 5- (4-OEt-2-F-Ph) THI 3- yl], [ BF 554; 5- (4-F-2-Cl-Ph) THI-3-yl], [BF 555; 5- (4-Cl-2-Cl-Ph) THI-3-yl], [BF 556; (4-Br-2-Cl-Ph) THI-3-yl], [BF 557; 5- (4-Me-2-Cl-Ph) THI-3-yl], [BF 558; 5- (4-Et) -2-Cl-Ph) THI-3-yl], [BF 559; 5- (4-CF ₃ -2-Cl-Ph) THI-3-yl], [BF 560; 5- (4-OMe-2-) Cl-Ph) THI-3-yl], [BF 561; 5- (4-OEt-2-Cl-Ph) THI-3-yl], [BF 562; 5- (4-F-2-Me-Ph) THI-3-yl], [BF 563; 5- (4-Cl-2-Me-Ph) THI-3-yl], [BF 564; 5- (4-Br-2-Me-Ph) THI-3-yl], [BF 565; 5- (4-Me-2-Me-Ph) THI-3-yl], [BF 566; 5- (4-Et) -2-Me-Ph) THI-3-yl], [BF 567; 5- (4-CF ₃ -2-Me-Ph) THI-3-yl], [BF 568; 5- (4-OMe-2-) Me-Ph) THI-3-yl], [BF569; 5- (4-OEt-2-Me-Ph) THI-3-yl], [BF570; 5- (4-F-2-OMe-Ph) THI-3-yl], [BF571; 5- (4-Cl-2-OMe-Ph) THI-3-yl], [BF572; 5- (4-Br-2-OMe-Ph) THI-3- yl], [BF 573; 5- (4-Me-2-OMe-Ph) THI-3-yl], [BF 574; 5- (4-Et-2-OMe-Ph) THI-3-yl], [BF4] _{BF575; 5- (4-CF 3} -2-OMe-Ph) THI-3-yl], [BF576; 5- (4-OMe-2-OMe-Ph) THI-3-yl], [BF577; 5 -(4-OEt-2-OMe-Ph) THI-3-yl], [BF578; 5- (4-F-2-OEt-Ph) THI-3-yl], [BF579; Cl-2-OEt-Ph) THI-3-yl], [BF 580; 5- (4-Br-2-OEt-Ph) THI-3-yl], [BF 581; 5- (4-Me-2-) OEt-Ph) THI-3- yl], [BF582; 5- (4-Et-2-OEt-Ph) THI-3-yl], [BF583; 5- (4-CF 3 -2-OEt-Ph ) THI-3-yl], [BF 584; 5- (4-OMe-2-OEt-Ph) THI-3-yl], [BF 585; 5- (4-OEt-2-OEt-Ph) THI-3 -yl], [BF586; 3-phenylFUR-5-yl], [BF587; 3- (2-F-Ph) FUR-5-yl], [BF588; 3- (3-F-Ph) FUR-5 -[yl], [BF 589; 3- (4-F-Ph) FUR-5-yl], [BF 590; 3- (2-Cl-Ph) FUR-5- yl], [BF 591; Cl-Ph) FUR-5-yl], [BF592; 3- (4-Cl-Ph) FUR-5-yl], [BF593; 3- (2-Br-Ph) FUR-5-yl], [BF-59] BF 594; 3- (3-Br-Ph) FUR-5-yl], [BF 595; 3 -(4-Br-Ph) FUR-5-yl], [BF596; 3- (2-Me-Ph) FUR-5-yl], [BF597; 3- (3-Me-Ph) FUR-5- yl], [BF 598; 3- (4-Me-Ph) FUR-5- yl], [BF 599; 3- (2-Et-Ph) FUR-5- yl], [BF 600; -Ph) FUR-5-yl],

[BF601; 3- (4-Et -Ph) FUR-5-yl], [BF602; 3- (2-CF 3 -Ph) FUR-5-yl], [BF603; 3- (3-CF 3 - Ph) FUR-5-yl], [BF 604; 3- (4-CF ₃ -Ph) FUR-5-yl], [BF 605; 3- (2-OMe-Ph) FUR-5-yl], [BF 606 3- (3-OMe-Ph) FUR-5-yl], [BF 607; 3- (4-OMe-Ph) FUR-5-yl], [BF608; 3- (2-OEt-Ph) FUR- 5-yl], [BF609; 3- (3-OEt-Ph) FUR-5-yl], [BF610; 3- (4-OEt-Ph) FUR-5-yl], [BF611; 3- (4) -F-2-F-Ph) FUR-5-yl], [BF612; 3- (4-Cl-2-F-Ph) FUR-5-yl], [BF613; 3- (4-Br-2) -F-Ph) FUR-5-yl], [BF 614; 3- (4-Me-2-F-Ph) FUR-5-yl], [BF 615; 3- (4-Et-2-F-Ph) ) FUR-5-yl], [BF 616; 3- (4-CF ₃ -2-F-Ph) FUR-5-yl], [BF 617; 3- (4-OMe-2-F-Ph) FUR- 5-yl], [BF 618; 3- (4-OEt-2-F-Ph) FUR-5-yl], [BF 619; 3- (4-F-2-Cl-Ph) FUR-5-yl] , [BF620; 3- (4-Cl-2-Cl-Ph) FUR-5-yl], [BF621; 3- (4-Br-2-Cl-Ph) FUR-5-yl], [BF622; 3- (4-Me-2-Cl-Ph) FUR-5-yl], [BF 623; 3- (4-Et-2-Cl-Ph) FUR-5-yl], [BF 624; 3- (4) _{-CF 3 -2-Cl-Ph)} FUR-5-yl], [BF625; 3- (4-OMe-2-Cl-Ph) FUR-5-yl], [BF626; 3- (4-OEt- 2-Cl-Ph) FUR-5-yl], [BF 627; 3- (4-F-2-Me-Ph) FUR-5-yl], [BF 628; 3- (4-Cl-2-Me-) Ph) FUR-5-yl], [BF 629; 3- (4-Br-2-Me-Ph) FUR-5-yl], [BF 630; 3- (4-Me-2-Me-Ph) FUR- 5-yl], [BF 631; 3- (4-Et-2-Me-Ph) FUR-5-yl], [BF 632; 3- (4-C) _{F 3 -2-Me-Ph)} FUR-5-yl], [BF633; 3- (4-OMe-2-Me-Ph) FUR-5-yl], [BF634; 3- (4-OEt-2 -Me-Ph) FUR-5-yl], [BF 635; 3- (4-F-2-OMe-Ph) FUR-5-yl], [BF 636; 3- (4-Cl-2-OMe-Ph) ) FUR-5-yl], [BF 637; 3- (4-Br-2-OMe-Ph) FUR-5-yl], [BF 638; 3- (4-Me-2-OMe-Ph) FUR-5 -yl], [BF639; 3- ( 4-Et-2-OMe-Ph) FUR-5-yl], [BF640; 3- (4-CF 3 -2-OMe-Ph) FUR-5-yl] , [BF641; 3- (4-OMe-2-OMe-Ph) FUR-5-yl], [BF 642; 3- (4-OEt-2-OMe-Ph) FUR-5-yl], [BF643; 3- (4-F-2-OEt-Ph) FUR-5-yl], [BF 644; 3- (4-Cl-2-OEt-Ph) FUR-5-yl], [BF 645; 3- (4) -Br-2-OEt-Ph) FUR-5-yl], [BF 646; 3- (4-Me-2-OEt-Ph) FUR-5-yl], [BF 647; 3- (4-Et-2) -OEt-Ph) FUR-5- yl], [BF648; 3- (4-CF 3 -2-OEt-Ph) FUR-5-yl], [BF649; 3- (4-OMe-2-OEt- Ph) FUR-5-yl], [BF 650; 3- (4-OEt-2-OEt-Ph) FUR-5-yl], [BF 651; 5-phenylFUR-2-yl], [BF 652; 2-F-Ph) FUR-2-yl], [BF653; 5- (3-F-Ph) FUR-2-yl], [BF654; 5- (4-F-Ph) FUR-2-yl] , [BF655; 5- (2-Cl-Ph) FUR-2-yl], [BF 656; 5- (3-Cl-Ph) FUR-2-yl], [BF 657; 5- (4-Cl-Ph) ) FUR-2-yl], [BF 658; 5- (2-Br-Ph) FUR-2-yl], [BF 659; 5- (3-Br-Ph) FUR-2-yl], [BF 660; -(4-Br-Ph) FUR-2-yl], [BF 661; 5- (2-Me-Ph) FUR-2-yl], [BF 662; 5- (3-Me-Ph) FUR-2- yl], [BF 663; 5- (4-Me-Ph) FUR-2-yl] , [BF 664; 5- (2-Et-Ph) FUR-2-yl], [BF 665; 5- (3-Et-Ph) FUR-2-yl], [BF 666; 5- (4-Et-Ph) ) FUR-2-yl], [BF 667; 5- (2-CF ₃ -Ph) FUR-2-yl], [BF 668; 5- (3-CF ₃ -Ph) FUR-2-yl], [BF 669] 5- (4-CF ₃ -Ph) FUR-2-yl], [BF 670; 5- (2-OMe-Ph) FUR-2-yl], [BF 671; 5- (3-OMe-Ph) FUR -2-yl], [BF 672; 5- (4-OMe-Ph) FUR-2-yl], [BF 673; 5- (2-OEt-Ph) FUR-2-yl], [BF 674; 3-OEt-Ph) FUR-2-yl], [BF 675; 5- (4-OEt-Ph) FUR-2-yl], [BF 676; 5- (4-F-2-F-Ph) FUR- 2-yl], [BF677; 5- (4-Cl-2-F-Ph) FUR-2-yl], [BF 678; 5- (4-Br-2-F-Ph) FUR-2-yl] , [BF 679; 5- (4-Me-2-F-Ph) FUR-2-yl], [BF 680; 5- (4-Et-2-F-Ph) FUR-2-yl], [BF 681; _{5- (4-CF 3 -2-} F-Ph) FUR-2-yl], [BF682; 5- (4-OMe-2-F-Ph) FUR-2-yl], [BF683; 5- ( 4-OEt-2-F-Ph) FUR-2-yl], [BF 684; 5- (4-F-2-Cl-Ph) FUR-2-yl], [BF 685; 5- (4-Cl-) 2-Cl-Ph) FUR-2-yl], [BF 686; 5- (4-Br-2-Cl-Ph) FUR-2-yl], [BF 687; 5- (4-Me-2-Cl- Ph) FUR-2-yl], [BF 688; 5- (4-Et-2-Cl-Ph) FUR-2-yl], [BF 689; 5- (4-CF ₃ -2-Cl-Ph) FUR -2-yl], [BF 690; 5- (4-OMe-2-Cl-Ph) FUR-2-yl], [BF 691; 5- (4-OEt-2-Cl-Ph) FUR-2-yl ], [BF692; 5- (4-F-2-Me-Ph) FUR-2-yl], [BF693; 5- (4-Cl-2-Me-Ph) FUR-2-yl], [BF694] 5- (4-Br-2-Me-Ph) FUR-2-yl], [BF 695; 5- (4-Me-2-Me-Ph) ) FUR-2-yl], [BF 696; 5- (4-Et-2-Me-Ph) FUR-2-yl], [BF 697; 5- (4-CF ₃ -2-Me-Ph) FUR- 2-yl], [BF698; 5- (4-OMe-2-Me-Ph) FUR-2-yl], [BF699; 5- (4-OEt-2-Me-Ph) FUR-2-yl] , [BF 700; 5- (4-F-2-OMe-Ph) FUR-2-yl],

[BF 701; 5- (4-Cl-2-OMe-Ph) FUR-2-yl], [BF 702; 5- (4-Br-2-OMe-Ph) FUR-2-yl], [BF 703; -(4-Me-2-OMe-Ph) FUR-2-yl], [BF704; 5- (4-Et-2-OMe-Ph) FUR-2-yl], [BF705; _{CF 3 -2-OMe-Ph)} FUR-2-yl], [BF706; 5- (4-OMe-2-OMe-Ph) FUR-2-yl], [BF707; 5- (4-OEt-2 -OMe-Ph) FUR-2-yl], [BF 708; 5- (4-F-2-OEt-Ph) FUR-2-yl], [BF 709; 5- (4-Cl-2-OEt-Ph) ) FUR-2-yl], [BF 710; 5- (4-Br-2-OEt-Ph) FUR-2-yl], [BF711; 5- (4-Me-2-OEt-Ph) FUR-2 -yl], [BF712; 5- ( 4-Et-2-OEt-Ph) FUR-2-yl], [BF713; 5- (4-CF 3 -2-OEt-Ph) FUR-2-yl] , [BF714; 5- (4-OMe-2-OEt-Ph) FUR-2-yl], [BF715; 5- (4-OEt-2-OEt-Ph) FUR-2-yl], [BF716; 5-phenylFUR-3-yl], [BF717; 5- (2-F-Ph) FUR-3-yl], [BF718; 5- (3-F-Ph) FUR-3-yl], [BF719; 5- (4-F-Ph) FUR-3-yl], [BF720; 5- (2-Cl-Ph) FUR-3-yl], [BF721; 5- (3-Cl-Ph) FUR-3 5- (4-Cl-Ph) FUR-3-yl], [BF 723; 5- (2-Br-Ph) FUR-3-yl], [BF 724; 5- (3-) Br-Ph) FUR-3-yl], [BF 725; 5- (4-Br-Ph) FUR-3-yl], [BF 726; 5- (2-Me-Ph) FUR-3-yl], [BF- BF 727; 5- (3-Me-Ph) FUR-3-yl], [BF 728; 5- (4-Me-Ph) FUR-3-yl], [BF 729; 5- (2-Et-Ph) FUR 5- (3-Et-Ph) FUR-3-yl], [BF731; 5- (4-Et-Ph) FUR-3-yl], [BF732; 2-CF ₃ -Ph) FUR-3-yl], [BF 733; 5 _{- (3-CF 3 -Ph)} FUR-3-yl], [BF734; 5- (4-CF 3 -Ph) FUR-3-yl], [BF735; 5- (2-OMe-Ph) FUR- 3-yl], [BF 736; 5- (3-OMe-Ph) FUR-3-yl], [BF 737; 5- (4-OMe-Ph) FUR-3-yl], [BF 738; 5- (2) -OEt-Ph) FUR-3-yl], [BF739; 5- (3-OEt-Ph) FUR-3-yl], [BF 740; 5- (4-OEt-Ph) FUR-3-yl], [BF 741; 5- (4-F-2-F-Ph) FUR-3-yl], [BF 742; 5- (4-Cl-2-F-Ph) FUR-3-yl], [BF 743; 5 -(4-Br-2-F-Ph) FUR-3-yl], [BF 744; 5- (4-Me-2-F-Ph) FUR-3-yl], [BF 745; Et-2-F-Ph) FUR-3-yl], [BF 746; 5- (4-CF ₃ -2-F-Ph) FUR-3-yl], [BF 747; 5- (4-OMe-2) -F-Ph) FUR-3-yl], [BF 748; 5- (4-OEt-2-F-Ph) FUR-3-yl], [BF 749; 5- (4-F-2-Cl-Ph) ) FUR-3-yl], [BF 750; 5- (4-Cl-2-Cl-Ph) FUR-3-yl], [BF 751; 5- (4-Br-2-Cl-Ph) FUR-3 5- (4-Me-2-Cl-Ph) FUR-3-yl], [BF753; 5- (4-Et-2-Cl-Ph) FUR-3-yl], [BF754; 5- (4-CF 3 -2-Cl-Ph) FUR-3-yl], [BF755; 5- (4-OMe-2-Cl-Ph) FUR-3-yl], [BF756; 5- (4-OEt-2-Cl-Ph) FUR-3-yl], [BF 757; 5- (4-F-2-Me-Ph) FUR-3-yl], [BF 758; 5- (4) -Cl-2-Me-Ph) FUR-3-yl], [BF 759; 5- (4-Br-2-Me-Ph) FUR-3-yl], [BF 760; 5- (4-Me-2) -Me-Ph) FUR-3-yl], [BF 761; 5- (4-Et-2-Me-Ph) FUR-3-yl], [BF 762; 5- (4-CF ₃ -2-Me- Ph) FUR-3-yl], [BF 763; 5- (4-OMe-2-Me-Ph) FUR-3-yl], [BF 764; 4-OEt-2-Me-Ph) FUR-3-yl], [BF 765; 5- (4-F-2-OMe-Ph) FUR-3-yl], [BF 766; 5- (4-Cl-) 2-OMe-Ph) FUR-3-yl], [BF 767; 5- (4-Br-2-OMe-Ph) FUR-3-yl], [BF 768; 5- (4-Me-2-OMe- Ph) FUR-3-yl], [BF 769; 5- (4-Et-2-OMe-Ph) FUR-3-yl], [BF 770; 5- (4-CF ₃ -2-OMe-Ph) FUR -3-yl], [BF 771; 5- (4-OMe-2-OMe-Ph) FUR-3-yl], [BF 772; 5- (4-OEt-2-OMe-Ph) FUR-3-yl ], [BF 773; 5- (4-F-2-OEt-Ph) FUR-3-yl], [BF 774; 5- (4-Cl-2-OEt-Ph) FUR-3-yl], [BF 775] 5- (4-Br-2-OEt-Ph) FUR-3-yl], [BF 776; 5- (4-Me-2-OEt-Ph) FUR-3-yl], [BF 777; 4-Et-2-OEt-Ph) FUR-3-yl], [BF 778; 5- (4-CF ₃ -2-OEt-Ph) FUR-3-yl], [BF 779; 5- (4-OMe) -2-OEt-Ph) FUR-3-yl], [BF 780; 5- (4-OEt-2-OEt-Ph) FUR-3-yl], [BF 781; 2-phenylTHA-4-yl], BF782; 2- (2-F-Ph) THA-4-yl], [BF783; 2- (3-F-Ph) THA-4-yl], [BF784; 2- (4-F-Ph) THA -4-yl], [BF 785; 2- (2-Cl-Ph) THA-4-yl], [BF 786; 2- (3-Cl-Ph) THA-4-yl], [BF 787; 2- ( 4-Cl-Ph) THA-4-yl], [BF 788; 2- (2-Br-Ph) THA-4-yl], [BF 789; 2- (3-Br-Ph) THA-4-yl] , [BF 790; 2- (4-Br-Ph) THA-4-yl], [BF 791; 2- (2-Me-Ph) THA-4-yl], [BF 792; 2- (3-Me-Ph) ) THA-4-yl], [BF 793; 2- (4-Me-Ph) THA-4-yl], [BF 794; 2- (2-Et-Ph) THA-4-yl], [BF795; -(3-Et-Ph) THA-4-yl], [BF796; 2- ( 4-Et-Ph) THA-4-yl], [BF 797; 2- (2-CF ₃ -Ph) THA-4-yl], [BF798; 2- (3-CF ₃ -Ph) THA-4- yl], [BF 799; 2- (4-CF ₃ -Ph) THA-4-yl], [BF 800; 2- (2-OMe-Ph) THA-4-yl],

[BF801; 2- (3-OMe-Ph) THA-4-yl], [BF802; 2- (4-OMe-Ph) THA-4-yl], [BF803; 2- (2-OEt-Ph) THA-4-yl], [BF 804; 2- (3-OEt-Ph) THA-4-yl], [BF 805; 2- (4-OEt-Ph) THA-4-yl], [BF 806; (4-F-2-F-Ph) THA-4-yl], [BF 807; 2- (4-Cl-2-F-Ph) THA-4-yl], [BF 808; 2- (4-Br) -2-F-Ph) THA-4-yl], [BF 809; 2- (4-Me-2-F-Ph) THA-4-yl], [BF 810; 2- (4-Et-2-F) -Ph) THA-4-yl] , [BF811; 2- (4-CF 3 -2-F-Ph) THA-4-yl], [BF812; 2- (4-OMe-2-F-Ph) THA-4-yl], [BF813; 2- (4-OEt-2-F-Ph) THA-4-yl], [BF814; 2- (4-F-2-Cl-Ph) THA-4- yl], [BF 815; 2- (4-Cl-2-Cl-Ph) THA-4-yl], [BF 816; 2- (4-Br-2-Cl-Ph) THA-4-yl], [ BF 817; 2- (4-Me-2-Cl-Ph) THA-4-yl], [BF 818; 2- (4-Et-2-Cl-Ph) THA-4-yl], [BF 819; _{(4-CF 3 -2-Cl} -Ph) THA-4-yl], [BF820; 2- (4-OMe-2-Cl-Ph) THA-4-yl], [BF821; 2- (4- OEt-2-Cl-Ph) THA-4-yl], [BF822; 2- (4-F-2-Me-Ph) THA-4-yl], [BF823; 2- (4-Cl-2-) Me-Ph) THA-4-yl], [BF 824; 2- (4-Br-2-Me-Ph) THA-4-yl], [BF 825; 2- (4-Me-2-Me-Ph) THA-4-yl], [ BF826; 2- (4-Et-2-Me-Ph) THA-4-yl], [BF827; 2- (4-CF 3 -2-Me-Ph) THA-4 -[yl], [BF 828; 2- (4-OMe-2-Me-Ph) THA-4-yl], [BF829; 2- (4-OEt-2-Me-Ph) THA-4-yl], [BF 830; 2- (4-F-2-OMe-Ph) THA-4-yl], [BF 831; 2- (4-Cl-2-OMe-Ph) TH A-4-yl], [BF 832; 2- (4-Br-2-OMe-Ph) THA-4-yl], [BF 833; 2- (4-Me-2-OMe-Ph) THA-4- yl], [BF834; 2- ( 4-Et-2-OMe-Ph) THA-4-yl], [BF835; 2- (4-CF 3 -2-OMe-Ph) THA-4-yl], [BF 836; 2- (4-OMe-2-OMe-Ph) THA-4-yl], [BF 837; 2- (4-OEt-2-OMe-Ph) THA-4-yl], [BF 838; 2 -(4-F-2-OEt-Ph) THA-4-yl], [BF 839; 2- (4-Cl-2-OEt-Ph) THA-4-yl], [BF 840; 2- (4-) Br-2-OEt-Ph) THA-4-yl], [BF 841; 2- (4-Me-2-OEt-Ph) THA-4-yl], [BF 842; 2- (4-Et-2-) OEt-Ph) THA-4- yl], [BF843; 2- (4-CF 3 -2-OEt-Ph) THA-4-yl], [BF844; 2- (4-OMe-2-OEt-Ph ) THA-4-yl], [BF 845; 2- (4-OEt-2-OEt-Ph) THA-4-yl], [BF 846; 2-phenylOXA-4-yl], [BF 847; 2- (2) -F-Ph) OXA-4-yl], [BF 848; 2- (3-F-Ph) OXA-4-yl], [BF849; 2- (4-F-Ph) OXA-4-yl], [BF850; 2- (2-Cl-Ph) OXA-4-yl], [BF 851; 2- (3-Cl-Ph) OXA-4-yl], [BF 852; 2- (4-Cl-Ph) OXA-4-yl], [BF 853; 2- (2-Br-Ph) OXA-4-yl], [BF 854; 2- (3-Br-Ph) OXA-4-yl], [BF 855; (4-Br-Ph) OXA-4-yl], [BF 856; 2- (2-Me-Ph) OXA-4-yl], [BF 857; 2- (3-Me-Ph) OXA-4-yl ], [BF 858; 2- (4-Me-Ph) OXA-4-yl], [BF 859; 2- (2-Et-Ph) OXA-4-yl], [BF 860; 2- (3-Et-) Ph) OXA-4-yl], [BF 861; 2- (4-Et-Ph) OXA-4-yl], [BF 862; 2- (2-CF ₃ -Ph) OXA-4-yl], [BF 863 2- (3-CF ₃ -Ph) OXA-4-yl], [BF _{864; 2- (4-CF 3} -Ph) OXA-4-yl], [BF865; 2- (2-OMe-Ph) OXA-4-yl], [BF866; 2- (3-OMe-Ph) OXA-4-yl], [BF 867; 2- (4-OMe-Ph) OXA-4-yl], [BF 868; 2- (2-OEt-Ph) OXA-4-yl], [BF 869; (3-OEt-Ph) OXA-4-yl], [BF870; 2- (4-OEt-Ph) OXA-4-yl], [BF871; 2- (4-F-2-F-Ph) OXA -4-yl], [BF 872; 2- (4-Cl-2-F-Ph) OXA-4-yl], [BF 873; 2- (4-Br-2-F-Ph) OXA-4-yl ], [BF 874; 2- (4-Me-2-F-Ph) OXA-4-yl], [BF 875; 2- (4-Et-2-F-Ph) OXA-4-yl], [BF 876] _{; 2- (4-CF 3 -2} -F-Ph) OXA-4-yl], [BF877; 2- (4-OMe-2-F-Ph) OXA-4-yl], [BF878; 2- (4-OEt-2-F-Ph) OXA-4-yl], [BF879; 2- (4-F-2-Cl-Ph) OXA-4-yl], [BF 880; 2- (4-Cl) -2-Cl-Ph) OXA-4-yl], [BF 881; 2- (4-Br-2-Cl-Ph) OXA-4-yl], [BF 882; 2- (4-Me-2-Cl) -Ph) OXA-4-yl] , [BF883; 2- (4-Et-2-Cl-Ph) OXA-4-yl], [BF884; 2- (4-CF 3 -2-Cl-Ph) OXA-4-yl], [BF885; 2- (4-OMe-2-Cl-Ph) OXA-4-yl], [BF886; 2- (4-OEt-2-Cl-Ph) OXA-4- yl], [BF 887; 2- (4-F-2-Me-Ph) OXA-4-yl], [BF 888; 2- (4-Cl-2-Me-Ph) OXA-4-yl], [BF4] BF 889; 2- (4-Br-2-Me-Ph) OXA-4-yl], [BF 890; 2- (4-Me-2-Me-Ph) OXA-4-yl], [BF 891; (4-Et-2-Me -Ph) OXA-4-yl], [BF892; 2- (4-CF 3 -2-Me-Ph) OXA-4-yl], [BF893; 2- (4- OMe-2-Me-Ph) OXA-4-yl], [BF 894; 2- (4-OEt-2-Me-Ph) OXA-4-yl], [B F895; 2- (4-F-2-OMe-Ph) OXA-4-yl], [BF896; 2- (4-Cl-2-OMe-Ph) OXA-4-yl], [BF897; (4-Br-2-OMe-Ph) OXA-4-yl], [BF898; 2- (4-Me-2-OMe-Ph) OXA-4-yl], [BF899; 2- (4-Et) -2-OMe-Ph) OXA- 4-yl], [BF900; 2- (4-CF 3 -2-OMe-Ph) OXA-4-yl],

[BF 901; 2- (4-OMe-2-OMe-Ph) OXA-4-yl], [BF 902; 2- (4-OEt-2-OMe-Ph) OXA-4-yl], [BF 903; -(4-F-2-OEt-Ph) OXA-4-yl], [BF 904; 2- (4-Cl-2-OEt-Ph) OXA-4-yl], [BF 905; Br-2-OEt-Ph) OXA-4-yl], [BF 906; 2- (4-Me-2-OEt-Ph) OXA-4-yl], [BF 907; 2- (4-Et-2-) OEt-Ph) OXA-4- yl], [BF908; 2- (4-CF 3 -2-OEt-Ph) OXA-4-yl], [BF909; 2- (4-OMe-2-OEt-Ph ) OXA-4-yl], [BF910; 2- (4-OEt-2-OEt-Ph) OXA-4-yl], [BF911; 4-Ph-1-Me-IMI-2-yl], [BF9] BF 912; 4- (2-F-Ph) -1-Me-IMI-2-yl], [BF 913; 4- (3-F-Ph) -1-Me-IMI-2-yl], [BF 914; 4- (4-F-Ph) -1-Me-IMI-2-yl], [BF 915; 4- (2-Cl-Ph) -1-Me-IMI-2-yl], [BF 916; (3-Cl-Ph) -1-Me-IMI-2-yl], [BF 917; 4- (4-Cl-Ph) -1-Me-IMI-2-yl], [BF 918; 4- (2) -Br-Ph) -1-Me-IMI-2-yl], [BF 919; 4- (3-Br-Ph) -1-Me-IMI-2-yl], [BF 920; 4- (4-Br) -Ph) -1-Me-IMI-2-yl], [BF 921; 4- (2-Me-Ph) -1-Me-IMI-2-yl], [BF 922; 4- (3-Me-Ph) )-[1-Me-IMI-2-yl], [BF 923; 4- (4-Me-Ph) -1-Me-IMI-2-yl], [BF 924; 4- (2-Et-Ph)- 1-Me-IMI-2-yl], [BF 925; 4- (3-Et-Ph) -1-Me-IMI-2-yl], [BF 926; 4- (4-Et-Ph) -1-] Me-IMI-2-yl], [BF 927; 4- (2-CF ₃ -Ph) -1-Me-IMI-2-yl], [BF 928; 4- (3-CF ₃ -Ph) -1-] Me-IMI-2-yl], [BF 929; 4- (4-CF ₃ -Ph) -1-Me-IMI-2-yl], [BF 930; 4- (2-OMe-Ph) -1-Me-IMI-2-yl], [BF 931; 4- (3-OMe-Ph) -1-Me-IMI-2-yl], [BF 932; 4- (4) -OMe-Ph) -1-Me-IMI-2-yl], [BF 933; 4- (2-OEt-Ph) -1-Me-IMI-2-yl], [BF 934; 4- (3-OEt) -Ph) -1-Me-IMI-2-yl], [BF 935; 4- (4-OEt-Ph) -1-Me-IMI-2-yl], [BF 936; 4- (4-F-2) -F-Ph) -1-Me-IMI-2-yl], [BF 937; 4- (4-Cl-2-F-Ph) -1-Me-IMI-2-yl], [BF 938; 4- (4-Br-2-F-Ph) -1-Me-IMI-2-yl], [BF 939; 4- (4-Me-2-F-Ph) -1-Me-IMI-2-yl] , [BF940; 4- (4- Et-2-F-Ph) -1-Me-IMI-2-yl], [BF941; 4- (4-CF 3 -2-F-Ph) -1-Me -IMI-2-yl], [BF 942; 4- (4-OMe-2-F-Ph) -1-Me-IMI-2-yl], [BF 943; 4- (4-OEt-2-F-) Ph) -1-Me-IMI-2-yl], [BF 944; 4- (4-F-2-Cl-Ph) -1-Me-IMI-2-yl], [BF 945; Cl-2-Cl-Ph) -1-Me-IMI-2-yl], [BF 946; 4- (4-Br-2-Cl-Ph) -1-Me-IMI-2-yl], [BF 947 4- (4-Me-2-Cl-Ph) -1-Me-IMI-2-yl], [BF 948; 4- (4-Et-2-Cl-Ph) -1-Me-IMI-2 -yl], [BF949; 4- ( 4-CF 3 -2-Cl-Ph) -1-Me-IMI-2-yl], [BF950; 4- (4-OMe-2-Cl-Ph) - 1-Me-IMI-2-yl], [BF 951; 4- (4-OEt-2-Cl-Ph) -1-Me-IMI-2-yl], [BF 952; 4- (4-F-2) -Me-Ph) -1-Me-IMI-2-yl], [BF953; 4- (4-Cl-2-Me-Ph) -1-Me-IMI-2-yl], [BF954; (4-Br-2-Me-Ph) -1-Me-IMI-2-yl], [BF 955; 4- (4-Me-2-Me-Ph) -1-Me-IMI-2-yl] , [BF 956; 4- (4-Et-2-Me- Ph) -1-Me-IMI- 2-yl], [BF957; 4- (4-CF 3 -2-Me-Ph) -1-Me-IMI-2-yl], [BF958; 4- (4 -OMe-2-Me-Ph) -1-Me-IMI-2-yl], [BF 959; 4- (4-OEt-2-Me-Ph) -1-Me-IMI-2-yl], [ BF 960; 4- (4-F-2-OMe-Ph) -1-Me-IMI-2-yl], [BF 961; 4- (4-Cl-2-OMe-Ph) -1-Me-IMI- 2-yl], [BF 962; 4- (4-Br-2-OMe-Ph) -1-Me-IMI-2-yl], [BF 963; 4- (4-Me-2-OMe-Ph)- 1-Me-IMI-2-yl], [BF 964; 4- (4-Et-2-OMe-Ph) -1-Me-IMI-2-yl], [BF 965; 4- (4-CF _3- 2-OMe-Ph) -1-Me-IMI-2-yl], [BF966; 4- (4-OMe-2-OMe-Ph) -1-Me-IMI-2-yl], [BF967; 4 -(4-OEt-2-OMe-Ph) -1-Me-IMI-2-yl], [BF 968; 4- (4-F-2-OEt-Ph) -1-Me-IMI-2-yl ], [BF969; 4- (4-Cl-2-OEt-Ph) -1-Me-IMI-2-yl], [BF970; 4- (4-Br-2-OEt-Ph) -1-Me -IMI-2-yl], [BF 971; 4- (4-Me-2-OEt-Ph) -1-Me-IMI-2-yl], [BF 972; 4- (4-Et-2-OEt-) Ph) -1-Me-IMI- 2-yl], [BF973; 4- (4-CF 3 -2-OEt-Ph) -1-Me-IMI-2-yl], [BF974; 4- (4 -OMe-2-OEt-Ph) -1-Me-IMI-2-yl], [BF 975; 4- (4-OEt-2-OEt-Ph) -1-Me-IMI-2-yl], BF976; 2-Ph-1-Me-IMI-4-yl], [BF977; 2- (2-F-Ph) -1-Me-IMI-4-yl], [BF978; 2- (3-F) -Ph) -1-Me-IMI-4-yl], [BF 979; 2- (4-F-Ph) -1-Me-IMI-4-yl], [BF 980; 2- (2-Cl-Ph) )-1 -Me-IMI-4-yl], [BF 981; 2- (3-Cl-Ph) -1-Me-IMI-4-yl], [BF 982; 2- (4-Cl-Ph) )-1-Me-IMI-4-yl], [BF 983; 2- (2-Br-Ph) -1-Me-IMI-4-yl], [BF 984; 2- (3-Br-Ph)- 1-Me-IMI-4-yl], [BF985; 2- (4-Br-Ph) -1-Me-IMI-4-yl], [BF986; 2- (2-Me-Ph) -1-] Me-IMI-4-yl], [BF 987; 2- (3-Me-Ph) -1-Me-IMI-4-yl], [BF 988; 2- (4-Me-Ph) -1-Me- IMI-4-yl], [BF 989; 2- (2-Et-Ph) -1-Me-IMI-4-yl], [BF990; 2- (3-Et-Ph) -1-Me-IMI- 4-yl], [BF991; 2- (4-Et-Ph) -1-Me-IMI-4-yl], [BF992; 2- (2-CF ₃ -Ph) -1-Me-IMI-4 -yl], [BF993; 2- ( 3-CF 3 -Ph) -1-Me-IMI-4-yl], [BF994; 2- (4-CF 3 -Ph) -1-Me-IMI-4 -yl, [BF995; 2- (2-OMe-Ph) -1-Me-IMI-4-yl], [BF996; 2- (3-OMe-Ph) -1-Me-IMI-4-yl ], [BF997; 2- (4-OMe-Ph) -1-Me-IMI-4-yl], [BF998; 2- (2-OEt-Ph) -1-Me-IMI-4-yl], [BF 999; 2- (3-OEt-Ph) -1-Me-IMI-4-yl], [BF1000; 2- (4-OEt-Ph) -1-Me-IMI-4-yl],

[BF1001; 2- (4-F-2-F-Ph) -1-Me-IMI-4-yl], [BF1002; 2- (4-Cl-2-F-Ph) -1-Me-IMI -4-yl], [BF1003; 2- (4-Br-2-F-Ph) -1-Me-IMI-4-yl], [BF1004; 2- (4-Me-2-F-Ph) -1-Me-IMI-4-yl], [BF1005; 2- (4-Et-2-F-Ph) -1-Me-IMI-4-yl], [BF1006; 2- (4-CF ₃₎ -2-F-Ph) -1-Me-IMI-4-yl], [BF1007; 2- (4-OMe-2-F-Ph) -1-Me-IMI-4-yl], [BF1008; 2- (4-OEt-2-F-Ph) -1-Me-IMI-4-yl], [BF1009; 2- (4-F-2-Cl-Ph) -1-Me-IMI-4- yl], [BF1010; 2- (4-Cl-2-Cl-Ph) -1-Me-IMI-4-yl], [BF1011; 2- (4-Br-2-Cl-Ph) -1-] Me-IMI-4-yl], [BF1012; 2- (4-Me-2-Cl-Ph) -1-Me-IMI-4-yl], [BF1013; 2- (4-Et-2-Cl) -Ph) -1-Me-IMI- 4-yl], [BF1014; 2- (4-CF 3 -2-Cl-Ph) -1-Me-IMI-4-yl], [BF1015; 2- ( 4-OMe-2-Cl-Ph) -1-Me-IMI-4-yl], [BF1016; 2- (4-OEt-2-Cl-Ph) -1-Me-IMI-4-yl], [BF 1017; 2- (4-F-2-Me-Ph) -1-Me-IMI-4-yl], [BF1018; 2- (4-Cl-2-Me-Ph) -1-Me-IMI -4-yl], [BF1019; 2- (4-Br-2-Me-Ph) -1-Me-IMI-4-yl], [BF1020; 2- (4-Me-2-Me-Ph) -1-Me-IMI-4-yl], [BF 1021; 2- (4-Et-2-Me-Ph) -1-Me-IMI-4-yl], [BF 1022; 2- (4-CF ₃₎ -2-Me-Ph) -1-Me-IMI-4-yl], [BF 1023; 2- (4-OMe-2-Me-Ph) -1-Me-IMI-4-yl], [BF 1024; 2- (4-OEt-2-Me-Ph) -1-Me-IMI-4-yl], [BF1025; 2- (4-F-2-OMe-Ph) -1-Me-IMI-4- yl], [BF1026; 2- (4-Cl-2-OMe-Ph) -1-Me-IMI-4-yl], [BF1027; 2- (4-Br-2-OMe-Ph) -1-] Me-IMI-4-yl], [BF1028; 2- (4-Me-2-OMe-Ph) -1-Me-IMI-4-yl], [BF1029; 2- (4-Et-2-OMe) -Ph) -1-Me-IMI- 4-yl], [BF1030; 2- (4-CF 3 -2-OMe-Ph) -1-Me-IMI-4-yl], [BF1031; 2- ( 4-OMe-2-OMe-Ph) -1-Me-IMI-4-yl], [BF1032; 2- (4-OEt-2-OMe-Ph) -1-Me-IMI-4-yl], [BF1033; 2- (4-F-2-OEt-Ph) -1-Me-IMI-4-yl], [BF1034; 2- (4-Cl-2-OEt-Ph) -1-Me-IMI -4-yl], [BF1035; 2- (4-Br-2-OEt-Ph) -1-Me-IMI-4-yl], [BF1036; 2- (4-Me-2-OEt-Ph) -1-Me-IMI-4-yl], [BF1037; 2- (4-Et-2-OEt-Ph) -1-Me-IMI-4-yl], [BF1038; 2- (4-CF ₃₎ -2-OEt-Ph) -1-Me-IMI-4-yl], [BF1039; 2- (4-OMe-2-OEt-Ph) -1-Me-IMI-4-yl], [BF1040; 2- (4-OEt-2-OEt-Ph) -1-Me-IMI-4-yl] [BF1041; 3-phenylPRL-5-yl], [BF1042; 3- (2-F-Ph) PRL- 5-yl], [BF1043; 3- (3-F-Ph) PRL-5-yl], [BF1044; 3- (4-F-Ph) PRL-5-yl], [BF1045; 3- (2) -Cl-Ph) PRL-5-yl], [BF1046; 3- (3-Cl-Ph) PRL-5-yl], [BF1047; 3- (4-Cl-Ph) PRL-5-yl], [BF1048; 3- (2-Br-Ph) PRL-5-yl], [BF1049; 3- (3-Br-Ph) PRL-5-yl], [BF1050; 3- (4-Br-Ph) PRL-5-yl], [BF1051; 3- (2-Me-Ph) PRL-5-yl], [BF1052; 3- (3-Me-Ph) PRL-5-yl], [BF1053; (4-Me-Ph) PRL-5-yl], [B F1054; 3- (2-Et-Ph) PRL-5-yl], [BF1055; 3- (3-Et-Ph) PRL-5-yl], [BF1056; 3- (4-Et-Ph) PRL -5-yl], [BF1057; 3- (2-CF 3 -Ph) PRL-5-yl], [BF1058; 3- (3-CF 3 -Ph) PRL-5-yl], [BF1059; 3 _{- (4-CF 3 -Ph)} PRL-5-yl], [BF1060; 3- (2-OMe-Ph) PRL-5-yl], [BF1061; 3- (3-OMe-Ph) PRL-5 -yl], [BF1062; 3- (4-OMe-Ph) PRL-5-yl], [BF1063; 3- (2-OEt-Ph) PRL-5-yl], [BF1064; OEt-Ph) PRL-5-yl], [BF1065; 3- (4-OEt-Ph) PRL-5-yl], [BF1066; 3- (4-F-2-F-Ph) PRL-5- yl], [BF1067; 3- (4-Cl-2-F-Ph) PRL-5-yl], [BF1068; 3- (4-Br-2-F-Ph) PRL-5-yl], [ BF1069; 3- (4-Me-2-F-Ph) PRL-5-yl], [BF1070; 3- (4-Et-2-F-Ph) PRL-5-yl], [BF1071; 3- _{(4-CF 3 -2-F} -Ph) PRL-5-yl], [BF1072; 3- (4-OMe-2-F-Ph) PRL-5-yl], [BF1073; 3- (4- OEt-2-F-Ph) PRL-5-yl], [BF1074; 3- (4-F-2-Cl-Ph) PRL-5-yl], [BF1075; 3- (4-Cl-2-) Cl-Ph) PRL-5-yl], [BF1076; 3- (4-Br-2-Cl-Ph) PRL-5-yl], [BF1077; 3- (4-Me-2-Cl-Ph) PRL-5-yl], [ BF1078; 3- (4-Et-2-Cl-Ph) PRL-5-yl], [BF1079; 3- (4-CF 3 -2-Cl-Ph) PRL-5 -yl, [BF1080; 3- (4-OMe-2-Cl-Ph) PRL-5-yl], [BF1081; 3- (4-OEt-2-Cl-Ph) PRL-5-yl], [BF1082; 3- (4-F-2-Me-Ph) PRL-5-yl], [BF1083; 3- (4-Cl-2-Me-Ph) PRL-5-yl], [BF1084; -(4-Br-2-Me-Ph) PRL- 5-yl], [BF1085; 3- (4-Me-2-Me-Ph) PRL-5-yl], [BF1086; 3- (4-Et-2-Me-Ph) PRL-5-yl] , [BF1087; 3- (4- CF 3 -2-Me-Ph) PRL-5-yl], [BF1088; 3- (4-OMe-2-Me-Ph) PRL-5-yl], [BF1089 3- (4-OEt-2-Me-Ph) PRL-5-yl], [BF1090; 3- (4-F-2-OMe-Ph) PRL-5-yl], [BF1091; 4-Cl-2-OMe-Ph) PRL-5-yl], [BF1092; 3- (4-Br-2-OMe-Ph) PRL-5-yl], [BF1093; 3- (4-Me-) 2-OMe-Ph) PRL-5-yl], [BF1094; 3- (4-Et-2-OMe-Ph) PRL-5-yl], [BF1095; 3- (4-CF ₃ -2-OMe] -Ph) PRL-5-yl], [BF1096; 3- (4-OMe-2-OMe-Ph) PRL-5-yl], [BF1097; 3- (4-OEt-2-OMe-Ph) PRL -5-yl], [BF1098; 3- (4-F-2-OEt-Ph) PRL-5-yl], [BF1099; 3- (4-Cl-2-OEt-Ph) PRL-5-yl ], [BF1100; 3- (4-Br-2-OEt-Ph) PRL-5-yl],

[BF 1101; 3- (4-Me-2-OEt-Ph) PRL-5-yl], [BF 1102; 3- (4-Et-2-OEt-Ph) PRL-5-yl], [BF 1103; _{- (4-CF 3 -2-} OEt-Ph) PRL-5-yl], [BF1104; 3- (4-OMe-2-OEt-Ph) PRL-5-yl], [BF1105; 3- (4 -OEt-2-OEt-Ph) PRL-5-yl], [BF1106; 5-phenylPRL-2-yl], [BF1107; 5- (2-F-Ph) PRL-2-yl], [BF1108; 5- (3-F-Ph) PRL-2-yl], [BF1109; 5- (4-F-Ph) PRL-2-yl], [BF1110; 5- (2-Cl-Ph) PRL-2 5- (3-Cl-Ph) PRL-2-yl], [BF1112; 5- (4-Cl-Ph) PRL-2-yl], [BF1113; 5- (2-) Br-Ph) PRL-2-yl], [BF1114; 5- (3-Br-Ph) PRL-2-yl], [BF1115; 5- (4-Br-Ph) PRL-2-yl], BF1116; 5- (2-Me-Ph) PRL-2-yl], [BF1117; 5- (3-Me-Ph) PRL-2-yl], [BF1118; 5- (4-Me-Ph) PRL -2-yl], [BF1 119; 5- (2-Et-Ph) PRL-2-yl], [BF1 120; 5- (3-Et-Ph) PRL-2-yl], [BF1121; 4-Et-Ph) PRL- 2-yl], [BF1122; 5- (2-CF 3 -Ph) PRL-2-yl], [BF1123; 5- (3-CF 3 -Ph) PRL-2- yl], [BF1124; 5- ( 4-CF 3 -Ph) PRL-2-yl], [BF1125; 5- (2-OMe-Ph) PRL-2-yl], [BF1126; 5- (3- OMe-Ph) PRL-2-yl], [BF1127; 5- (4-OMe-Ph) PRL-2-yl], [BF1128; 5- (2-OEt-Ph) PRL-2-yl], BF1129; 5- (3-OEt-Ph) PRL-2-yl], [BF1130; 5- (4-OEt-Ph) PRL-2-yl], [BF1131; 5- (4-F-2-F) -Ph) PRL-2-yl], [BF 1132; 5- (4-Cl-2-F-Ph) PRL-2-yl], [BF 1133; 5- (4-Br-2-FP) h) PRL-2-yl], [BF1 134; 5- (4-Me-2-F-Ph) PRL-2-yl], [BF1 135; 5- (4-Et-2-F-Ph) PRL- 2-yl], [BF1136; 5- (4-CF 3 -2-F-Ph) PRL-2-yl], [BF1137; 5- (4-OMe-2-F-Ph) PRL-2-yl ], [BF1138; 5- (4-OEt-2-F-Ph) PRL-2-yl], [BF1139; 5- (4-F-2-Cl-Ph) PRL-2-yl], [BF1140] 5- (4-Cl-2-Cl-Ph) PRL-2-yl], [BF1141; 5- (4-Br-2-Cl-Ph) PRL-2-yl], [BF1142; 4-Me-2-Cl- Ph) PRL-2-yl], [BF1143; 5- (4-Et-2-Cl-Ph) PRL-2-yl], [BF1144; 5- (4-CF 3 -2-Cl-Ph) PRL-2-yl], [BF1145; 5- (4-OMe-2-Cl-Ph) PRL-2-yl], [BF1146; 5- (4-OEt-2-Cl) -Ph) PRL-2-yl], [BF1147; 5- (4-F-2-Me-Ph) PRL-2-yl], [BF1148; 5- (4-Cl-2-Me-Ph) PRL -2-yl], [BF1149; 5- (4-Br-2-Me-Ph) PRL-2-yl], [BF1150; 5- (4-Me-2-Me-Ph) PRL-2-yl ], [BF1151; 5- (4 -Et-2-Me-Ph) PRL-2-yl], [BF1152; 5- (4-CF 3 -2-Me-Ph) PRL-2-yl], [ BF1153; 5- (4-OMe-2-Me-Ph) PRL-2-yl], [BF1154; 5- (4-OEt-2-Me-Ph) PRL-2-yl], [BF1 155; (4-F-2-OMe-Ph) PRL-2-yl], [BF1156; 5- (4-Cl-2-OMe-Ph) PRL-2-yl], [BF1157; 5- (4-Br -2-OMe-Ph) PRL-2-yl], [BF1158; 5- (4-Me-2-OMe-Ph) PRL-2-yl], [BF1159; 5- (4-Et-2-OMe) -Ph) PRL-2-yl] , [BF1160; 5- (4-CF 3 -2-OMe-Ph) PRL-2-yl], [BF1161; 5- (4-OMe-2-OMe-Ph) PRL-2-yl], [BF1162; 5- (4-OEt-2) -OMe-Ph) PRL-2-yl], [BF1163; 5- (4-F-2-OEt-Ph) PRL-2-yl], [BF1164; 5- (4-Cl-2-OEt-Ph) ) PRL-2-yl], [BF1165; 5- (4-Br-2-OEt-Ph) PRL-2-yl], [BF1166; 5- (4-Me-2-OEt-Ph) PRL-2 -yl], [BF1167; 5- ( 4-Et-2-OEt-Ph) PRL-2-yl], [BF1168; 5- (4-CF 3 -2-OEt-Ph) PRL-2-yl] , [BF1169; 5- (4-OMe-2-OEt-Ph) PRL-2-yl], [BF1170; 5- (4-OEt-2-OEt-Ph) PRL-2-yl], [BF1171; 5-phenylPRL-3-yl], [BF1172; 5- (2-F-Ph) PRL-3-yl], [BF1173; 5- (3-F-Ph) PRL-3-yl], [BF1174; 5- (4-F-Ph) PRL-3-yl], [BF1175; 5- (2-Cl-Ph) PRL-3-yl], [BF1176; 5- (3-Cl-Ph) PRL-3 5- (4-Cl-Ph) PRL-3-yl], [BF1178; 5- (2-Br-Ph) PRL-3-yl], [BF1179; Br-Ph) PRL-3-yl], [BF1180; 5- (4-Br-Ph) PRL-3-yl], [BF1181; 5- (2-Me-Ph) PRL-3-yl], BF1182; 5- (3-Me-Ph) PRL-3-yl], [BF1183; 5- (4-Me-Ph) PRL-3-yl], [BF1184; 5- (2-Et-Ph) PRL 5- (3-Et-Ph) PRL-3-yl], [BF1186; 5- (4-Et-Ph) PRL-3-yl], [BF1187; 2-CF ₃ -Ph) PRL-3-yl], [BF 1188; 5- (3-CF ₃ -Ph) PRL-3-yl], [BF 1189; 5- (4-CF ₃ -Ph) PRL-3 5- (2-OMe-Ph) PRL-3-yl], [BF1191; 5- (3-OMe-Ph) PRL-3-yl], [BF1192; 5- (4-OMe) OMe-Ph) PRL-3-yl], [BF1193; 5- (2-OEt-Ph) PRL-3-yl], [BF1194; 5- (3-OEt-Ph) PRL- 3-yl], [BF 1195; 5- (4-OEt-Ph) PRL-3-yl], [BF 1196; 5- (4-F-2-F-Ph) PRL-3-yl], [BF 1197; 5- (4-Cl-2-F-Ph) PRL-3-yl], [BF1198; 5- (4-Br-2-F-Ph) PRL-3-yl], [BF1 199; 5- (4) -Me-2-F-Ph) PRL-3-yl], [BF1200; 5- (4-Et-2-F-Ph) PRL-3-yl],

[BF1201; 5- (4-CF 3 -2-F-Ph) PRL-3-yl], [BF1202; 5- (4-OMe-2-F-Ph) PRL-3-yl], [BF1203; 5- (4-OEt-2-F-Ph) PRL-3-yl], [BF1204; 5- (4-F-2-Cl-Ph) PRL-3-yl], [BF1205; 5- (4) -Cl-2-Cl-Ph) PRL-3-yl], [BF1206; 5- (4-Br-2-Cl-Ph) PRL-3-yl], [BF1207; 5- (4-Me-2) -Cl-Ph) PRL-3- yl], [BF1208; 5- (4-Et-2-Cl-Ph) PRL-3-yl], [BF1209; 5- (4-CF 3 -2-Cl- Ph) PRL-3-yl], [BF1210; 5- (4-OMe-2-Cl-Ph) PRL-3-yl], [BF1211; 5- (4-OEt-2-Cl-Ph) PRL- 3-yl], [BF1212; 5- (4-F-2-Me-Ph) PRL-3-yl], [BF1213; 5- (4-Cl-2-Me-Ph) PRL-3-yl] , [BF1214; 5- (4-Br-2-Me-Ph) PRL-3-yl], [BF1215; 5- (4-Me-2-Me-Ph) PRL-3-yl], [BF1216; 5- (4-Et-2- Me-Ph) PRL-3-yl], [BF1217; 5- (4-CF 3 -2-Me-Ph) PRL-3-yl], [BF1218; 5- ( 4-OMe-2-Me-Ph) PRL-3-yl], [BF1219; 5- (4-OEt-2-Me-Ph) PRL-3-yl], [BF1220; 5- (4-F-) 2-OMe-Ph) PRL-3-yl], [BF1221; 5- (4-Cl-2-OMe-Ph) PRL-3-yl], [BF1222; 5- (4-Br-2-OMe- Ph) PRL-3-yl], [BF1223; 5- (4-Me-2-OMe-Ph) PRL-3-yl], [BF1224; 5- (4-Et-2-OMe-Ph) PRL- 3-yl], [BF1225; 5- (4-CF 3 -2-OMe-Ph) PRL-3-yl], [BF1226; 5- (4-OMe-2-OMe-Ph) PRL-3-yl ], [BF1227; 5- (4-OEt-2-OMe-Ph) PRL-3-yl], [BF1228; 5- (4-F-2-OEt-Ph) PRL-3-yl], [BF1229] 5- (4-Cl-2-OEt-Ph) P RL-3-yl], [BF1230; 5- (4-Br-2-OEt-Ph) PRL-3-yl], [BF1231; 5- (4-Me-2-OEt-Ph) PRL-3- yl], [BF1232; 5- ( 4-Et-2-OEt-Ph) PRL-3-yl], [BF1233; 5- (4-CF 3 -2-OEt-Ph) PRL-3-yl], [BF 1234; 5- (4-OMe-2-OEt-Ph) PRL-3-yl], [BF1235; 5- (4-OEt-2-OEt-Ph) PRL-3-yl], [BF1236; -phenylTDA-5-yl], [BF1237; 2- (2-F-Ph) TDA-5-yl], [BF1238; 2- (3-F-Ph) TDA-5-yl], [BF1239; 2 -(4-F-Ph) TDA-5-yl], [BF1240; 2- (2-Cl-Ph) TDA-5-yl], [BF1241; 2- (3-Cl-Ph) TDA-5- yl], [BF1242; 2- (4-Cl-Ph) TDA-5-yl], [BF1243; 2- (2-Br-Ph) TDA-5-yl], [BF1244; 2- (3-Br) -Ph) TDA-5-yl], [BF1245; 2- (4-Br-Ph) TDA-5-yl], [BF1246; 2- (2-Me-Ph) TDA-5-yl], [BF1247 2- (3-Me-Ph) TDA-5-yl], [BF1248; 2- (4-Me-Ph) TDA-5-yl], [BF1249; 2- (2-Et-Ph) TDA- 5-yl], [BF1 250; 2- (3-Et-Ph) TDA-5-yl], [BF1251; 2- (4-Et-Ph) TDA-5-yl], [BF1252; 2- (2) _{-CF 3 -Ph) TDA-5-} yl], [BF1253; 2- (3-CF 3 -Ph) TDA-5-yl], [BF1254; 2- (4-CF 3 -Ph) TDA-5- yl], [BF1 255; 2- (2-OMe-Ph) TDA-5-yl], [BF1 256; 2- (3-OMe-Ph) TDA-5-yl], [BF1 257; 2- (4-OMe) -Ph) TDA-5-yl], [BF1258; 2- (2-OEt-Ph) TDA-5-yl], [BF1259; 2- (3-OEt-Ph) TDA-5-yl], [BF1260 2- (4-OEt-Ph) TDA-5-yl], [BF1261; 2- (4-F-2-F-Ph) TDA-5-yl], [BF1262; 2- (4-Cl-2-F-Ph) TDA-5-yl], [BF1263; 2- (4-Br-2-F-Ph) TDA-5-yl], [BF1264; 2- (4-Me) -2-F-Ph) TDA-5-yl], [BF1265; 2- (4-Et-2-F-Ph) TDA-5-yl], [BF1266; 2- (4-CF ₃ -2-) F-Ph) TDA-5-yl], [BF1267; 2- (4-OMe-2-F-Ph) TDA-5-yl], [BF1268; 2- (4-OEt-2-F-Ph) TDA-5-yl], [BF 1269; 2- (4-F-2-Cl-Ph) TDA-5-yl], [BF 1270; 2- (4-Cl-2-Cl-Ph) TDA-5- yl], [BF1271; 2- (4-Br-2-Cl-Ph) TDA-5-yl], [BF1272; 2- (4-Me-2-Cl-Ph) TDA-5-yl], [BF4] BF1273; 2- (4-Et- 2-Cl-Ph) TDA-5-yl], [BF1274; 2- (4-CF 3 -2-Cl-Ph) TDA-5-yl], [BF1275; 2 -(4-OMe-2-Cl-Ph) TDA-5-yl], [BF1276; 2- (4-OEt-2-Cl-Ph) TDA-5-yl], [BF1277; F-2-Me-Ph) TDA-5-yl], [BF1278; 2- (4-Cl-2-Me-Ph) TDA-5-yl], [BF1279; 2- (4-Br-2-) Me-Ph) TDA-5-yl], [BF 1280; 2- (4-Me-2-Me-Ph) TDA-5-yl], [BF1281; 2- (4-Et-2-Me-Ph) TDA-5-yl], [ BF1282; 2- (4-CF 3 -2-Me-Ph) TDA-5-yl], [BF1283; 2- (4-OMe-2-Me-Ph) TDA-5 -yl], [BF1284; 2- (4-OEt-2-Me-Ph) TDA-5-yl], [BF1285; 2- (4-F-2-OMe-Ph) TDA-5-yl], [BF1286; 2- (4-Cl-2-OMe-Ph) TDA-5-yl], [BF1287; 2- (4-Br-2-OMe-Ph) TDA-5-yl], [BF1288; -(4-Me-2-OMe-Ph) TDA-5-yl], [BF1289; 2- (4-Et-2-OMe-Ph) TDA-5-yl], [BF1290; CF ₃ -2-OMe-Ph) TDA-5-yl], [BF 1291; 2- (4-OMe-2-OMe-Ph) TDA-5-yl], [BF1292; 2- (4-OEt-2-OMe-Ph) TDA-5-yl], [BF1293; 2- (4-F) -2-OEt-Ph) TDA-5-yl], [BF1294; 2- (4-Cl-2-OEt-Ph) TDA-5-yl], [BF1295; 2- (4-Br-2-OEt) -Ph) TDA-5-yl], [BF 1296; 2- (4-Me-2-OEt-Ph) TDA-5-yl], [BF 1297; 2- (4-Et-2-OEt-Ph) TDA -5-yl], [BF1298; 2- (4-CF 3 -2-OEt-Ph) TDA-5-yl], [BF1299; 2- (4-OMe-2-OEt-Ph) TDA-5- yl], [BF1300; 2- (4-OEt-2-OEt-Ph) TDA-5-yl]

  Further, the present compounds AG1-BG1 to AG327-BG6699 can also be obtained according to the above-mentioned method.

The present compounds AG1-BG1 to AG327-BG6699 are compounds represented by the following formula (AGBG).

[Wherein, X ^{71 to} X ⁷⁶ each represent a substituent corresponding to each of the substituent numbers (MG1) AG 1 to AG 327 shown below, and in the formula, E ¹⁰⁷ represents a substituent number (MG 2) BG 1 shown below ~ BG 6699. ]
For example, the present compound AG1-BG1, in the compounds of formula (AGBG), X ⁷¹ ~X ⁷⁶ substituents ID ME1 (X ⁷¹ and X ⁷² is a hydrogen atom, X ⁷³ and X ⁷⁶ is an oxygen atom, X ⁷⁴ Is a single bond, X ⁷⁵ is = CH-N = CH-CH =), and E ¹⁰⁷ is a compound in which the substituent number (MG2) is BG1 (pyridin-2-yl group), and is represented by the following formula: Ru.

In X ⁷⁴ of the following substituent number (MF1),-represents a single bond, and = represents a double bond.
[Substituent number (MF1): X ⁷¹ , X ⁷² , X ⁷³ , X ⁷⁴ , X ⁷⁵ , X ⁷⁶ ], [AG 1; H, H, O,-, = CH-N = CH-CH =, O] , [AG2, H, H, O,-, = CF-N = CH-CH =, O], [AG3; H, H, O,-, = CCl-N = CH-CH =, O], [AG2; AG4, H, H, O,-, = CBr-N = CH-CH =, O], [AG5; H, H, O,-, = CI-N = CH-CH =, O], [AG6; H, H, O,-, = C (Me)-N = CH-CH =, O], [AG7; H, H, O,-, = C (Et)-N = CH-CH =, O] , [AG8; H, H, O,-, = C (c-Pr)-N = CH-CH =, O], [AG 9; H, H, O,-, = C (OMe)-N = CH -CH =, O], [AG10; H, H, O,-, = C (OEt)-N = CH-CH =, O], [AG11; H, H, O,-, = C (CH = _{CH 2) -N = CH-CH} =, O], [AG12; H, H, O, -, = C (C≡CH) -N = CH-CH =, O], [AG13; H, H, O,-, = CH-CH = N-CH =, O], [AG14; H, H, O,-, = CF-CH = N-CH =, O], [AG15; H, H, O, -, = CCl-CH = N-CH =, O], [AG16; H, H, O,-, = CBr-CH = N-CH =, O], [AG17; H, H, O,-, = CI-CH = N-CH =, O], [AG18; H, H, O,-, = C (Me) -CH = N-CH =, O], [AG19; H, H, O,- , = C (Et) -CH = N-CH =, O], [AG20; H, H, O,-, = C (c-Pr) -CH = N-CH =, O], [AG21; H , H, O,-, = C (OMe)-CH = N-CH =, O], [AG22; H, H, O,-, = C (OEt)-CH = N-CH =, O], [AG23; H, H, O , -, = C (CH = CH 2) -CH = N-CH =, O], [AG24; H, H, O, -, = C (C≡CH) -CH = N-CH =, O], [AG25; H, H, O,-, = CH-CH = CH-N =, O], [AG26; H, H, O,-, = CF-CH = CH -N =, O], [AG27; H, H, O,-, = CCl-CH = CH-N =, O], [AG28; H, H, O,-, = CBr-CH = CH-N =, O], [AG 29; H, H, O,-, = CI-CH = CH-N =, O], [AG 3 0; H, H, O,-, = C (Me)-CH = CH-N =, O], [AG 31; H, H, O,-, = C (Et)-CH = CH-N =, O], [AG 32; H, H, O,-, = C (c-Pr)-CH = CH-N =, O], [AG 33; H, H, O,-, = C (OMe)-CH = CH-N =, O], [AG34; H, H, O,-, = C (OEt) -CH = CH-N =, O], [AG35; H, H, O,-, = C ( _{CH = CH 2) -CH = CH} -N =, O], [AG36; H, H, O, -, = C (C≡CH) -CH = CH-N =, O], [AG37; H, H, O,-, = CH-CH = NN =, O], [AG 38; H, H, O,-, = CF-CH = N-N =, O], [AG 39; H, H, O, -, = CCl-CH = NN =, O], [AG40; H, H, O,-, = CBr-CH = NN =, O], [AG41; H, H, O,-, = CI-CH = NN =, O], [AG42; H, H, O,-, = C (Me) -CH = NN =, O], [AG43; H, H, O,-, = C (Et) -CH = NN =, O], [AG44; H, H, O,-, = C (c-Pr) -CH = NN =, O], [AG45; H, H, O,-, = C (OMe) -CH = NN =, O], [AG46; H, H, O,-, = C (OEt) -CH = NN =, O], [AG47; H, H, O,-, = C (CH = _{CH 2) -CH = NN =,} O], [AG48; H, H, O, -, = = C (C≡CH) -CH = NN, O], [AG49; H, H, O, -, = CH-N = CH-N =, O], [AG50; H, H, O,-, = CF-N = CH-N =, O], [AG51; H, H, O,-, = CCl -N = CH-N =, O], [AG52; H, H, O,-, = CBr-N = CH-N =, O], [AG53; H, H, O,-, = CI-N = CH-N =, O], [AG54; H, H, O,-, = C (Me) -N = CH-N =, O], [AG55; H, H, O,-, = C ( Et) -N = CH-N =, O], [AG56; H, H, O,-, = C (c-Pr) -N = CH-N =, O], [AG57; H, H, O ,-, = C (OMe)-N = CH-N =, O], [AG 58; H, H, O,-, = C (OEt)-N = CH-N =, O], [AG 59; H , H, O, -, = C (CH = CH 2) -N = CH-N =, O], [AG60; H, H, O, -, = C (C≡CH) -N = CH-N =, O H, H, O,-, = CH-CH = N-CH =, O], [AG 62; H, H, O,-, = CF-N = N-CH =, O], [AG63; H, H, O,-, = CCl-N = N-CH =, O], [AG 64; H, H, O,-, = CBr-N = N-CH =, O], [AG 65 H, H, O,-, = CI-N = N-CH =, O], [AG 66; H, H, O,-, = C (Me)-N = N-CH =, O], [ AG67; H, H, O,-, = C (Et)-N = N-CH =, O], [AG 68; H, H, O,-, = C (c-Pr)-N = N-CH =, O], [AG 69; H, H, O,-, = C (OMe)-N = N-CH =, O], [AG 70; H, H, O,-, = C (OEt)-N = N-CH =, O] , [AG71; H, H, O, -, = C (CH = CH 2) -N = N-CH =, O], [AG72; H, H, O, -, = C (C≡CH) -N = N-CH =, O], [AG 73; H, H, O,-, = CH-N = NN =, O], [AG 74; H, H, O,- , = CF-N = NN =, O], [AG 75; H, H, O,-, = CCl-N = NN =, O], [AG 76; H, H, O,-, = CBr-N = NN =, O], [AG 77; H, H, O,-, = CI-N = NN =, O], [AG 78; H, H, O,-, = C (Me) -N = NN =, O], [AG 79; H, H, O,-, = C (Et)-N = N N =, O], [AG 80; H, H, O,-, = C (c-Pr)-N = N N =, O], [AG 81; H, H, O,-, = C (OMe)-N = NN =, O], [AG 82; H, H, O,-, = C (OEt)-N = NN =, O], [AG 83; H, H, O,-, = C (CH = CH ₂ )-N = NN =, O], [AG 84; H, H, O,-, = C (C≡CH ) -N = NN =, O], [AG85; H, H, O,-, = N-CH = CH-N =, O], [AG86; H, H, O,-, = N-CH = N-CH =, O], [AG 87; H, H, O,-, =, NN = CH-CH =, O], [AG 88; H, H, O,-, = N-CH = NN =, O ], [AG 89; H, H, O,-, = NN = CH-N =, O], [AG 90; H, H, O,-, = NN = N-CH =, O], [AG 91; H , H, O,-, = N-CH = CH-CH =, O], [AG 92; H, H, O, =, -NH-N = CH-, O], [AG 93; H, H, O , =, -N (Me) -N = CH-, O], [AG94; H, H, O, =, -N (Et) -N = CH-, O], [AG95; H, H, O, =, -N (c-Pr) -N = CH -, O], [AG 96; H, H, O, =, -N (i-Pr)-N = CH-, O], [AG 97; H, H, O, =, -N (t-Bu) -N = CH-, O], [ AG98; H, H, O, =, - N (CF 3) -N = CH-, O], [AG99; H, H, O, =, - N (CHF ² ) -N = CH-, O]

[AG100; H, H, O, =, -NH-CH = N-, O], [AG101; H, H, O, =, -N (Me) -CH = N-, O], [AG102; H, H, O, =, -N (Et) -CH = N-, O], [AG103; H, H, O, =, -N (c-Pr) -CH = N-, O], [ AG104; H, H, O, =, -N (i-Pr) -CH = N-, O], [AG105; H, H, O, =, -N (t-Bu) -CH = N-, O], [AG106; H, H, O, =, - N (CF 3) -CH = N-, O], [AG107; H, H, O, =, - N (CHF 2) -CH = N -, O], [AG108; H, H, O, =, -NH-CH = CH-, O], [AG109; H, H, O, =, -N (Me) -CH = CH-, O ], [AG110; H, H, O, =, -N (Et) -CH = CH-, O], [AG111; H, H, O, =, -N (c-Pr) -CH = CH- , O], [AG112; H, H, O, =, -N (i-Pr) -CH = CH-, O], [AG113; H, H, O, =, -N (t-Bu)- CH = CH-, O], [ AG114; H, H, O, =, - N (CF 3) -CH = CH-, O], [AG115; H, H, O, =, - N (CHF 2 ) -CH = CH-, O], [AG116; H, H, O, =, -NH-N = N-, O], [AG117; H, H, O, =, -N (Me) -N = N-, O], [AG118; H, H, O, =, -N (Et) -N = N-, O], [AG119; H, H, O, =, -N (c-Pr) -N = N-, O], [AG120; H, H, O, =, -N (i-Pr) -N = N-, O], [AG121; H, H, O, =, -N ( t-Bu) -N = N-, O], [AG122; H, H, O, =, - N (CF 3) -N = N-, O], [AG123; H, H, O, =, _{-N (CHF 2) -N = N-} , O], [AG124; H, H, O, -, = = CH-O-CH, O], [AG125; H, H, O, -, = CF -O-CH =, O], [AG126; H, H, O,-, = CCl-O-CH =, O], [AG 127; H, H, O,-, = CBr-O-CH =, O], [AG128; H, H, O,-, = CI-O-CH =, O], [AG129; H, H, O,-, = C (Me) -O-CH =, O], [AG130; H, H, O,-, = C (Et)-O-CH =, O], [AG 131; H, H, O,-, = C (c-Pr ) -O-CH =, O], [AG132; H, H, O,-, = C (OMe) -O-CH =, O], [AG133; H, H, O,-, = C (OEt ) -O-CH =, O] , AG134 [; H, H, O, -, = C (CH = CH 2) -O-CH =, O], [AG135; H, H, O, -, = C (C≡CH) -O-CH =, O], [AG 136; H, H, O,-, = CH-ON =, O], [AG 137; H, H, O,-, = CF-ON =, O], [AG 138; H, H, O,-, = CCl-ON =, O], [AG 139; H, H, O,-, = CBr-ON =, O], [AG 140; H, H, O,-, = CI-ON =, O], [AG 141; H, H, O,-, = C (Me)-ON =, O], [AG 142; H, H, O,-, = C (Et) -ON =, O], [AG143; H, H, O,-, = C (c-Pr) -ON =, O], [AG144; H, H, O,-, = C ( OMe) -ON =, O], [AG145; H, H, O, -, = C (OEt) -ON =, O], [AG146; H, H, O, -, = C (CH = CH 2 H) H, H, O,-, = C (C≡CH)-ON =, O], [AG 148; H, H, O,-, = CH-N (Me ) -CH =, O], [AG149; H, H, O,-, = CF-N (Me) -CH =, O], [AG150; H, H, O,-, = CCl-N (Me ) -CH =, O], [AG151; H, H, O,-, = CBr-N (Me) -CH =, O], [AG152; H, H, O,-, = CI-N (Me ) -CH =, O], [AG153; H, H, O,-, = C (Me) -N (Me) -CH =, O], [AG154; H, H, O,-, = C ( Et) -N (Me) -CH =, O], [AG155; H, H, O,-, = C (c-Pr) -N (Me) -CH =, O], [AG156; H, H , O,-, = C (OMe)-N (Me)-CH =, O], [AG 157; H, H, O,-, = C (OEt)-N (Me)-CH =, O], [AG158; H, H, O , -, = C (CH = CH 2) -N (Me) -CH =, O], [AG159; H, H, O, -, = C (C≡CH) - N (Me) -CH =, O], [AG160; H, H, O,-, = CH-N (Me) -N =, O], [AG161; H, H, O,-, = CF- N (Me)-N =, O], [AG 162; H, H, O,-, = CCl-N (Me) -N =, O], [AG163; H, H, O,-, = CBr-N (Me) -N =, O], [AG164; H, H, O,-, = CI-N (Me) -N =, O], [AG165; H, H, O,-, = C (Me) -N (Me) -N =, O], [AG166; H, H, O,-, = C (Et) -N (Me) -N =, O], [AG 167; H, H, O,-, = C (c-Pr) -N (Me) -N =, O], [AG 168; H , H, O,-, = C (OMe)-N (Me)-N =, O], [AG 169; H, H, O,-, = C (OEt)-N (Me)-N =, O H, H, O,-, = C (CH = CH2)-N (Me)-N =, O], [AG 171; H, H, O,-, = C (C≡CH)] -N (Me) -N =, O], [AG172; H, H, O,-, = CH-S-CH =, O], [AG173; H, H, O,-, = CF-S- CH =, O], [AG 174; H, H, O,-, = CCl-S-CH =, O], [AG 175; H, H, O,-, = CBr-S-CH =, O], [AG176; H, H, O,-, = CI-S-CH =, O], [AG 177; H, H, O,-, = C (Me) -S-CH =, O], [AG 178; H, H, O,-, = C (Et)-S-CH =, O], [AG 179; H, H, O,-, = C (c-Pr)-S-CH =, O], [ AG180; H, H, O,-, = C (OMe)-S-CH =, O], [AG 181; H, H, O,-, = C (OEt)-S-CH =, O], [ AG 182; H, H, O,-, = C (CH = CH ₂ )-S-CH =, O], [AG 183; H, H, O,-, = C (C≡CH)-S-CH = H, H, O,-, = CH-SN =, O], [AG 185; H, H, O,-, = CF-SN =, O], [AG 186; H, H] , O,-, = CCl-SN =, O], [AG 187; H, H, O,-, = CBr-SN =, O], [AG 188; H, H, O,-, = CI-SN = , O], [AG 189; H, H, O,-, = C (Me)-SN =, O], [AG 190; H, H, O,-, = C (Et)-SN =, O], [AG191; H, H, O,-, = C (c-Pr)-SN =, O], [AG 192; H, H, O,-, = C (OMe)-SN =, O], [AG 193 H, H, O,-, = C (OEt)-SN =, O], [AG 194; H, H, O,-, = C (CH = C H ₂ ) -SN =, O], [AG 195; H, H, O,-, = C (C≡CH) -SN =, O], [AG 196; H, H, O, =, -CH = CH -O-, O], [AG 197; H, H, O, =, -CF = CH-O-, O], [AG 198; H, H, O, =, -CCl = CH-O-, O] , [AG 199; H, H, O, =, -CBr = CH-O-, O]

[AG200; H, H, O, =, -CI = CH-O-, O], [AG201; H, H, O, =, -C (Me) = CH-O-, O], [AG202; H, H, O, =, -C (Et) = CH-O-, O], [AG 203; H, H, O, =, -C (c-Pr) = CH-O-, O], [ AG 204; H, H, O, =, -C (OMe) = CH-O-, O], [AG 205; H, H, O, =, -C (Oet) = CH-O-, O], [ AG206; H, H, O, =, - C (CH = CH 2) = CH-O-, O], [AG207; H, H, O, =, - C (C≡CH) = CH-O- , O], [AG208; H, H, O, =, -CH = NO-, O], [AG209; H, H, O, =, -CF = NO-, O], [AG210; H, H , O, =, -CCl = NO-, O], [AG211; H, H, O, =, -CBr = NO-, O], [AG 212; H, H, O, =, -CI = NO- , O], [AG213; H, H, O, =, -C (Me) = NO-, O], [AG 214; H, H, O, =, -C (Et) = NO-, O], [AG 215; H, H, O, =, -C (c-Pr) = NO-, O], [AG 216; H, H, O, =, -C (OMe) = NO-, O], [AG 217 H, H, O, =, -C (OEt) = NO-, O], [AG 218; H, H, O, =, -C (CH = CH2) = NO-, O], [AG 219; H , H, O, =, -C (C≡CH) = NO-, O], [AG 220; H, H, O, =, -CH = CH-S-, O], [AG 221; H, H, H O, =, -CF = CH-S-, O], [AG222; H, H, O, =, -CCl = CH-S-, O], [AG 223; H, H, O, =, -CBr = CH-S-, O], [AG224; H, H, O, =, -CI = CH-S-, O], [AG 225; H, H, O, =, -C (Me) = CH- S-, O], [AG 226; H, H, O, =, -C (Et) = CH-S-, O], [AG 227; H, H, O, =, -C (c-Pr) = CH-S-, O], [AG228; H, H, O, =, -C (OMe) = CH-S-, O], [AG 229; H, H, O, =, -C (Oet) = CH-S-, O], [ AG230; H, H, O, =, - C (CH = CH 2) = CH-S-, O], [AG231; H, H, O, =, - C ( C≡CH) = CH-S-, O], [AG 232; H, H, O, =, -CH = NS -, O], [AG233; H, H, O, =, -CF = NS-, O], [AG234; H, H, O, =, -CCl = NS-CH =, O], [AG235; H, H, O, =, -CBr = NS-, O], [AG 236; H, H, O, =, -CI = NS-, O], [AG 237; H, H, O, =, -C (Me) = NS-, O], [AG238; H, H, O, =, -C (Et) = NS-, O], [AG 239: H, H, O, =, -C (c-Pr (c-Pr) H) H, O, =, -C (OMe) = NS-, O], [AG 241; H, H, O, =, -C (OEt) = NS- , O], [AG242; H , H, O, =, - C (CH = CH 2) = NS-, O], [AG243; H, H, O, =, - C (C≡CH) = NS -, O], [AG244; H, H, O, =, -CH = CH-N (Me)-, O], [AG245; H, H, O, =, -CF = CH-N (Me) -CH =, O], [AG246; H, H, O, =, -CCl = CH-N (Me)-, O], [AG247; H, H, O, =, -CBr = CH-N ( Me)-, O], [AG248; H, H, O, =, -CI = CH-N (Me)-, O], [AG249; H, H, O, =, -C (Me) = CH -N (Me)-, O], [AG 250; H, H, O, =, -C (Et) = CH-N (Me)-, O], [AG 251; H, H, O, =,- C (c-Pr) = CH-N (Me)-, O], [AG252; H, H, O, =, -C (OMe) = CH-N (Me)-, O], [AG253; H , H, O, =, - C (Oet) = CH-N (Me) -, O], [AG254; H, H, O, =, - C (CH = CH 2) = CH-N (Me) -, O], [AG 255; H, H, O, =, -C (C≡CH) = CH-N (Me)-, O], [AG 256; H, H, O, =, -CH = NN (Me)-, O], [AG257; H, H, O, =, -CF = NN (Me)-, O], [AG258; H, H, O, =, -CCl = NN (Me)- , O], [AG 259; H, H, O, =, -CBr = N N (Me)-, O], [AG 260; H, H, O, =, -CI = N N (Me)-, O], [AG261; H, H, O, =, -C (Me) = NN (Me)-, O], [AG 262; H, H, O, =, -C (Et) = NN (Me)-, O ], [AG263; H, H, O, =, -C (c-Pr) = NN ( Me)-, O], [AG 264; H, H, O, =, -C (OMe) = NN (Me)-, O], [AG 265; H, H, O, =, -C (OEt) = NN (Me)-, O], [AG 266; H, H, O, =, -C (CH = CH2) = NN (Me)-, O], [AG 267; H, H, O, =,-C (C≡CH) = NN (Me)-, O], [AG 268; H, H, O, =, -O-CH = CH-, O], [AG 269; H, H, O, =, -ON = CH-, O], [AG 270; H, H, O, =, -O-CH = N-, O], [AG 271; H, H, O, =, -ON = N-, O], [ AG 272; H, H, O, =, -S-CH = CH-, O], [AG 273; H, H, O, =, -SN = CH-, O], [AG 274; H, H, O, =, -S-CH = N-, O], [AG 275; H, H, O, =, -SN = N-, O], [AG 276; H, H, O,-, = NO-CH =, O], [AG 277; H, H, O,-, = NO N =, O], [AG 278; H, H, O,-, = NS-CH =, O], [AG 279; H, H, O, -, = NSN =, O], [AG 280; H, H, O, =, -CH = NS-, O], [AG 281; H, H, O, =, -CF = NS-, O], [ AG282; H, H, O, =, -CCl = NS-, O], [AG 283; H, H, O, =, -CBr = NS-, O], [AG 284; H, H, O, =, -CI = NS-, O], [AG 285; H, H, O, =, -C (Me) = NS-, O], [AG 286; H, H, O, =, -C (Et) = NNS -, O], [AG 287; H, H, O, =, -C (c-Pr) = NS-, O], [AG 288; H, H, O, =, -C (OMe) = NS-, O], [AG 289; H, H, O, =, -C (OEt) = NS-, O], [AG 290; H, H, O, =, -C (CH = CH ₂ ) = NS-, O ], [AG291; H, H, O, =, -C (C, CH) = NS-, O], [AG292; H, H, O, =, -CH = CH-N (Me)-, O ], [AG293; H, H, O, =, -CF = CH-N (Me)-, O], [AG 294; H, H, O, =, -CCl = CH-N (Me)-, O ], [AG 295; H, H, O, =, -CBr = CH-N (Me)-, O], [AG 296; H, H, O, =, -CI = CH-N (Me)-, O ], [AG 297; H, H, O, =, -C (Me) = CH-N (Me)-, O], [AG 298; H, H, O, =, -C (Et) = CH-N (Me)-, O], [AG 299; H, H, O, =,-C ( c-Pr) = CH-N (Me)-, O]

[AG300; H, H, O, =, -C (OMe) = CH-N (Me)-, O], [AG 301; H, H, O, =, -C (OEt) = CH-N (Me ), [AG302; H, H, O, =, -C (CH = CH ₂ ) = CH-N (Me)-, O], [AG 303; H, H, O, =, -C (C≡CH) = CH-N (Me)-, O], [AG 304; H, H, O, =, -CH = NN (Me)-, O], [AG 305; H, H, O, = , -CF = NN (Me)-, O], [AG306; H, H, O, =, -CCl = NN (Me)-, O], [AG307; H, H, O, =, -CBr = NN (Me)-, O], [AG308; H, H, O, =, -CI = NN (Me)-, O], [AG 309; H, H, O, =, -C (Me) = NN (Me)-, O], [AG310; H, H, O, =, -C (Et) = NN (Me)-, O], [AG311; H, H, O, =, -C (c- Pr) = NN (Me)-, O], [AG 312; H, H, O, =, -C (OMe) = NN (Me)-, O], [AG 313; H, H, O, =,- C (OEt) = NN (Me ) -, O], [AG314; H, H, O, =, - C (CH = CH 2) = NN (Me) -, O], [AG315; H, H, O, =, -C (C≡CH) = NN (Me)-, O], [AG 316; H, H, O, =, -N = CH-O-, O], [AG 317; H, H, H O, =, -N = NO-, O], [AG 318; H, H, O, =, -N = CH-S-, O], [AG 319; H, H, O, =, -N = NS -, O], [AG 320; H, H, O, =, -N = N-NH-, O], [AG 321; H, H, O, =, -N = NN (Me)-, O], [AG 322; H, H, O, =, -N = CH-NH-, O], [AG 323; H, H, O, =, -N = CH-N (Me)-, O], [AG324; H, H, O,-, = N-NH-CH =, O], [AG 325; H, H, O,-, = NN (Me)-CH =, O], [AG 326; H, H, O ,-, = N-NH-N =, O], [AG 327; H, H, O,-, = NN (Me)-N =, O].

[Substituent number (MG2); E ¹⁰⁷ ], [BG 1: 2 -Py], [BG 2: 3-F-2-Py], [BG 3: 4-Cl-3-F-2-Py], [BG 4 : 5-Cl-3-F-2-Py !, [BG5: 6-Cl-3-F-2-Py], [BG 6: 4-Me-3-F-2-Py], [BG 7: 5] -Me-3-F-2- Py], [BG8: 6-Me-3-F-2-Py], [BG9: 4-CF 3 -3-F-2-Py], [BG10: 5- _{CF 3 -3-F-2-} Py], [BG11: 6-CF 3 -3-F-2-Py], [BG12: 4-CN-3-F-2-Py], [BG13: 5- CN-3-F-2-Py !, [BG14: 6-CN-3-F-2-Py], [BG15: 4-OMe-3-F-2-Py], [BG16: 5-OMe- 3-F-2-Py, [BG17: 6-OMe-3-F-2-Py], [BG18: 4-F-2-Py], [BG19: 3-Cl-4-F-2-] Py], [BG20: 5-Cl-4-F-2-Py], [BG21: 6-Cl-4-F-2-Py], [BG22: 3-Me-4-F-2-Py] , [BG23: 5-Me- 4-F-2-Py], [BG24: 6-Me-4-F-2-Py], [BG25: 3-CF 3 -4-F-2-Py], _{[BG26: 5-CF 3 -4} -F-2-Py], [BG27: 6-CF 3 -4-F-2-Py], [BG28: 3-CN-4-F-2-Py], [BG29: 5-CN-4-F-2-Py], [BG30: 6-CN-4-F-2-Py], [BG31: 3-OMe-4-F-2-Py], [BG32] : 5-OMe-4-F-2-Py], [BG33: 6-OMe-4-F-2-Py], [BG34: 5-F-2-Py], [BG35: 3-Cl-5] -F-2-Py], [BG36: 4-Cl-5-F-2-Py], [BG37: 6-Cl-5-F-2-Py], [BG38: 3-Me-5-F -2-Py], [BG39: 4-Me-5-F-2-Py], [BG40: 6-Me-5-F-2-Py], [BG41: 3-CF ₃ -5-F- 2-Py], [BG42: 4-CF 3 -5-F-2-Py], [BG43: 6-CF 3 -5-F-2-Py], [BG44: 3-CN-5-F- 2-Py], [BG45: 4-CN-5-F-2-Py], [BG46: 6-CN-5-F-2-Py ], [BG47: 3-OMe-5-F-2-Py], [BG48: 4-OMe-5-F-2-Py], [BG49: 6-OMe-5-F-2-Py], [BG50: 6-F-2-Py], [BG51: 3-Cl-6-F-2-Py], [BG52: 4-Cl-6-F-2-Py], [BG53: 5-Cl] -6-F-2-Py], [BG54: 3-Me-6-F-2-Py], [BG55: 4-Me-6-F-2-Py], [BG56: 5-Me-6] -F-2-Py], [ BG57: 3-CF 3 -6-F-2-Py], [BG58: 4-CF 3 -6-F-2-Py], [BG59: 5-CF 3 - 6-F-2-Py], [BG60: 3-CN-6-F-2-Py], [BG61: 4-CN-6-F-2-Py], [BG62: 5-CN-6-] F-2-Py !, [BG63: 3-OMe-6-F-2-Py], [BG64: 4-OMe-6-F-2-Py], [BG65: 5-OMe-6-F-] 2-Py], [BG66: 3-Cl-2-Py], [BG67: 4-Cl-3-Cl-2-Py], [BG 68: 5-Cl-3-Cl-2-Py], [BG BG69: 6-Cl-3-Cl-2-Py, [BG70: 4-Me-3-Cl-2-Py], [BG71: 5-Me-3-Cl-2-Py], [BG72: 6-Me-3-Cl-2-Py !, [BG 73: 4-CF ₃ -3-Cl-2-Py], [BG 74: 5-CF ₃ -3-Cl-2-Py], [BG 75: _{6-CF 3 -3-Cl-} 2-Py], [BG76: 4-CN-3-Cl-2-Py], [BG77: 5-CN-3-Cl-2-Py], [BG78: 6 -CN-3-Cl-2-Py], [BG79: 4-OMe-3-Cl-2-Py], [BG80: 5-OMe-3-Cl-2-Py], [BG 81: 6-OMe] -3-Cl-2-Py !, [BG 82: 4-Cl-2-Py], [BG 83: 3-Cl-4-Cl-2-Py], [BG 84: 5-Cl-4-Cl-2] -Py], [BG85: 6-Cl-4-Cl-2-Py], [BG86: 3-Me-4-Cl-2-Py], [BG87: 5-Me-4-Cl-2-Py] ], [BG88: 6-Me -4-Cl-2-Py], [BG89: 3-CF 3 -4-Cl-2-Py], [BG90: 5-CF 3 -4-Cl-2-Py ], [BG 91: 6-CF ₃ -4-Cl-2-Py], [BG 92: 3-CN-4-Cl-2-Py], [BG93: 5-CN-4-Cl-2-Py], [BG94: 6-CN-4-Cl-2-Py], [BG95: 3- OMe-4-Cl-2-Py], [BG96: 5-OMe-4-Cl-2-Py], [BG97: 6-OMe-4-Cl-2-Py], [BG98: 5-Cl- 2-Py], [BG99: 4-Cl-5-Cl-2-Py], [BG100: 5-Cl-5-Cl-2-Py],

[BG101: 6-Cl-5-Cl-2-Py], [BG102: 4-Me-5-Cl-2-Py], [BG103: 5-Me-5-Cl-2-Py], [BG104 : 6-Me-5-Cl -2-Py], [BG105: 4-CF 3 -5-Cl-2-Py], [BG106: 5-CF 3 -5-Cl-2-Py], [BG107 _{: 6-CF 3 -5-Cl} -2-Py], [BG108: 4-CN-5-Cl-2-Py], [BG109: 3-CN-5-Cl-2-Py], [BG110: 6-CN-5-Cl-2-Py, [BG111: 4-OMe-5-Cl-2-Py], [BG112: 5-OMe-5-Cl-2-Py], [BG113: 6- OMe-5-Cl-2-Py], [BG114: 6-Cl-2-Py], [BG115: 3-Cl-6-Cl-2-Py], [BG116: 4-Cl-6-Cl- 2-Py], [BG117: 5-Cl-6-Cl-2-Py], [BG118: 3-Me-6-Cl-2-Py], [BG119: 4-Me-6-Cl-2-] Py], [BG120: 5- Me-6-Cl-2-Py], [BG121: 3-CF 3 -6-Cl-2-Py], [BG122: 4-CF 3 -6-Cl-2- Py], [BG123: 5- CF 3 -6-Cl-2-Py], [BG124: 3-CN-6-Cl-2-Py], [BG125: 4-CN-6-Cl-2-Py ], [BG126: 5-CN-6-Cl-2-Py], [BG127: 3-OMe-6-Cl-2-Py], [BG128: 4-OMe-6-Cl-2-Py], [BG129: 5-OMe-6-Cl-2-Py], [BG130: 3-Br-2-Py], [BG131: 4-Cl-3-Br-2-Py], [BG132: 5-Cl] -3-Br-2-Py], [BG133: 6-Cl-3-Br-2-Py], [BG134: 4-Me-3-Br-2-Py], [BG135: 5-Me-3] -Br-2-Py], [ BG136: 6-Me-3-Br-2-Py], [BG137: 4-CF 3 -3-Br-2-Py], [BG138: 5-CF 3 -3 -Br-2-Py], [ BG139: 6-CF 3 -3-Br-2-Py], [BG140: 4-CN-3-Br-2-Py], [BG141: 5-CN-3- Br-2-Py, [BG142: 6-CN-3-Br-2-Py], [BG143: 4-OM] e-3-Br-2-Py, [BG144: 5-OMe-3-Br-2-Py], [BG145: 6-OMe-3-Br-2-Py], [BG146: 4-Br- 2-Py], [BG147: 3-Cl-4-Br-2-Py], [BG148: 5-Cl-4-Br-2-Py], [BG149: 6-Cl-4-Br-2-] Py], [BG150: 3-Me-4-Br-2-Py], [BG151: 5-Me-4-Br-2-Py], [BG152: 6-Me-4-Br-2-Py] _{, [BG153: 3-CF 3} -4-Br-2-Py], [BG154: 5-CF 3 -4-Br-2-Py], [BG155: 6-CF 3 -4-Br-2-Py ], [BG156: 3-CN-4-Br-2-Py], [BG157: 5-CN-4-Br-2-Py], [BG158: 6-CN-4-Br-2-Py], [BG159: 3-OMe-4-Br-2-Py], [BG160: 5-OMe-4-Br-2-Py], [BG161: 6-OMe-4-Br-2-Py], [BG162] : 5-Br-2-Py], [BG163: 3-Cl-5-Br-2-Py], [BG164: 4-Cl-5-Br-2-Py], [BG165: 6-Cl-5] -Br-2-Py, [BG166: 3-Me-5-Br-2-Py], [BG167: 4-Me-5-Br-2-Py], [BG168: 6-Me-5-Br -2-Py], [BG169: 3-CF 3 -5-Br-2-Py], [BG170: 4-CF 3 -5-Br-2-Py], [BG171: 6-CF 3 -5- Br-2-Py], [BG172: 3-CN-5-Br-2-Py], [BG173: 4-CN-5-Br-2-Py], [BG174: 6-CN-5-Br- 2-Py], [BG175: 3-OMe-5-Br-2-Py], [BG176: 4-OMe-5-Br-2-Py], [BG177: 6-OMe-5-Br-2-] Py], [BG 178: 6-Br-2-Py], [BG 179: 3-Cl-6-Br-2-Py], [BG 180: 4-Cl-6-Br-2-Py], [BG 181: 5-Cl-6-Br-2-Py], [BG 182: 3-Me-6-Br-2-Py], [BG 183: 4-Me-6-Br-2-Py], [BG 184: 5- Me-6-Br-2- Py], [BG185: 3-CF 3 -6-Br-2-Py], [BG186: _{4-CF 3 -6-Br-} 2-Py], [BG187: 5-CF 3 -6-Br-2-Py], [BG188: 3-CN-6-Br-2-Py], [BG189: 4-CN-6-Br-2-Py], [BG190: 5-CN-6-Br-2-Py], [BG191: 3-OMe-6-Br-2-Py], [BG192: 4-] OMe-6-Br-2-Py], [BG193: 5-OMe-6-Br-2-Py], [BG194: 3-I-2-Py], [BG195: 4-Cl-3-I- 2-Py], [BG196: 5-Cl-3-I-2-Py], [BG 197: 6-Cl-3-I-2-Py], [BG 198: 4-Me-3-I-2-] Py], [BG199: 5-Me-3-I-2-Py], [BG200: 6-Me-3-I-2-Py],

_{[BG201: 4-CF 3 -3} -I-2-Py], [BG202: 5-CF 3 -3-I-2-Py], [BG203: 6-CF 3 -3-I-2-Py] , [BG204: 4-CN-3-I-2-Py], [BG205: 5-CN-3-I-2-Py], [BG206: 6-CN-3-I-2-Py], BG207: 4-OMe-3-I-2-Py, [BG208: 5-OMe-3-I-2-Py], [BG209: 6-OMe-3-I-2-Py], [BG210: 4-I-2-Py, [BG211: 3-Cl-4-I-2-Py], [BG212: 5-Cl-4-I-2-Py], [BG213: 6-Cl-4- I-2-Py], [BG214: 3-Me-4-I-2-Py], [BG215: 5-Me-4-I-2-Py], [BG216: 6-Me-4-I- 2-Py], [BG217: 3-CF 3 -4-I-2-Py], [BG218: 5-CF 3 -4-I-2-Py], [BG219: 6-CF 3 -4-I -2-Py], [BG220: 3-CN-4-I-2-Py], [BG221: 5-CN-4-I-2-Py], [BG222: 6-CN-4-I-2 -Py], [BG223: 3-OMe-4-I-2-Py], [BG224: 5-OMe-4-I-2-Py], [BG225: 6-OMe-4-I-2-Py] ], [BG226: 5-I-2-Py], [BG227: 3-Cl-5-I-2-Py], [BG228: 4-Cl-5-I-2-Py], [BG 229: 6] -Cl-5-I-2-Py], [BG230: 3-Me-5-I-2-Py], [BG231: 4-Me-5-I-2-Py], [BG232: 6-Me -5-I-2-Py] , [BG233: 3-CF 3 -5-I-2-Py], [BG234: 4-CF 3 -5-I-2-Py], [BG235: 6-CF _{3 -5-I-2-Py} ], [BG236: 3-CN-5-I-2-Py], [BG237: 4-CN-5-I-2-Py], [BG238: 6-CN- 5-I-2-Py, [BG239: 3-OMe-5-I-2-Py], [BG240: 4-OMe-5-I-2-Py], [BG241: 6-OMe-5-] I-2-Py !, [BG 242: 6-I-2-Py], [BG 243: 3-Cl-6-I-2-Py], [BG 244: 4-Cl-6-I-2-Py] , [BG245: 5-Cl -6-I-2-Py], [BG246: 3-Me-6-I-2-Py], [BG247: 4-Me-6-I-2-Py], [BG248: 5-Me-6] -I-2-Py, [BG 249: 3-CF ₃ -6-I-2-Py], [BG 250: 4-CF ₃ -6-I-2-Py], [BG 251: 5-CF _3- 6-I-2-Py, [BG252: 3-CN-6-I-2-Py], [BG253: 4-CN-6-I-2-Py], [BG254: 5-CN-6- 6 I-2-Py, [BG255: 3-OMe-6-I-2-Py], [BG256: 4-OMe-6-I-2-Py], [BG257: 5-OMe-6-I- 2-Py], [BG258: 3-Me-2-Py], [BG 259: 4-Cl-3-Me-2-Py], [BG 260: 5-Cl-3-Me-2-Py], [BG BG261: 6-Cl-3-Me-2-Py], [BG262: 4-Me-3-Me-2-Py], [BG263: 5-Me-3-Me-2-Py], [BG264: 6-Me-3-Me- 2-Py], [BG265: 4-CF 3 -3-Me-2-Py], [BG266: 5-CF 3 -3-Me-2-Py], [BG267: _{6-CF 3 -3-Me-} 2-Py], [BG268: 4-CN-3-Me-2-Py], [BG269: 5-CN-3-Me-2-Py], [BG270: 6 -CN-3-Me-2-Py], [BG 271: 4-OMe-3-Me-2-Py], [BG 272: 5-OMe-3-Me-2-Py], [BG 273: 6-OMe] -3-Me-2-Py !, [BG274: 4-Me-2-Py], [BG275: 3-Cl-4-Me-2-Py], [BG276: 5-Cl-4-Me-2] -Py], [BG277: 6-Cl-4-Me-2-Py], [BG278: 3-Me-4-Me-2-Py], [BG279: 5-Me-4-Me-2-Py] ], [BG280: 6-Me -4-Me-2-Py], [BG281: 3-CF 3 -4-Me-2-Py], [BG282: 5-CF 3 -4-Me-2-Py ], [BG 283: 6-CF ₃ -4-Me-2-Py], [BG 284: 3-CN-4-Me-2-Py], [BG 285: 5-CN-4-Me-2-Py] , [BG286: 6-CN-4-Me-2-Py], [BG287: 3-OMe-4-Me-2-Py], [BG288: 5-OM] e-4-Me-2-Py, [BG289: 6-OMe-4-Me-2-Py], [BG290: 5-Me-2-Py], [BG291: 3-Cl-5-Me- 2-Py], [BG292: 4-Cl-5-Me-2-Py], [BG293: 6-Cl-5-Me-2-Py], [BG294: 3-Me-5-Me-2-] Py], [BG295: 4-Me-5-Me-2-Py], [BG 296: 6-Me-5-Me-2-Py], [BG 297: 3-CF ₃ -5-Me-2-Py ], [BG298: 4-CF 3 -5-Me-2-Py], [BG299: 6-CF 3 -5-Me-2-Py], [BG300: 3-CN-5-Me-2-Py ],

[BG301: 4-CN-5-Me-2-Py], [BG302: 6-CN-5-Me-2-Py], [BG303: 3-OMe-5-Me-2-Py], [BG304] : 4-OMe-5-Me-2-Py], [BG305: 6-OMe-5-Me-2-Py], [BG306: 6-Me-2-Py], [BG307: 3-Cl-6] -Me-2-Py], [BG308: 4-Cl-6-Me-2-Py], [BG309: 5-Cl-6-Me-2-Py], [BG310: 3-Me-6-Me -2-Py], [BG311: 4-Me-6-Me-2-Py], [BG312: 5-Me-6-Me-2-Py], [BG313: 3-CF 3 -6-Me- 2-Py], [BG314: 4-CF 3 -6-Me-2-Py], [BG315: 5-CF 3 -6-Me-2-Py], [BG316: 3-CN-6-Me- 2-Py], [BG317: 4-CN-6-Me-2-Py], [BG318: 5-CN-6-Me-2-Py], [BG319: 3-OMe-6-Me-2-] Py], [BG320: 4-OMe-6-Me-2-Py], [BG321: 5-OMe-6-Me-2-Py], [BG322: 3-OMe-2-Py], [BG323: 4-Cl-3-OMe-2-Py !, [BG324: 5-Cl-3-OMe-2-Py], [BG325: 6-Cl-3-OMe-2-Py], [BG326: 4-] Me-3-OMe-2-Py !, [BG 327: 5-Me-3-OMe-2-Py], [BG 328: 6-Me-3-OMe-2-Py], [BG 329: 4-CF _3] -3-OMe-2-Py] , [BG330: 5-CF 3 -3-OMe-2-Py], [BG331: 6-CF 3 -3-OMe-2-Py], [BG332: 4-CN -3-OMe-2-Py !, [BG333: 5-CN-3-OMe-2-Py], [BG334: 6-CN-3-OMe-2-Py], [BG335: 4-OMe-3] -OMe-2-Py], [BG 336: 5-OMe-3-OMe-2-Py], [BG 337: 6-OMe-3-OMe-2-Py], [BG 338: 4-OMe-2-Py] ], [BG339: 3-Cl-4-OMe-2-Py], [BG340: 5-Cl-4-OMe-2-Py], [BG341: 6-Cl-4-OMe-2-Py], [BG 342: 3-Me-4-OMe-2-Py], [BG BG343: 5-Me-4- OMe-2-Py], [BG344: 6-Me-4-OMe-2-Py], [BG345: 3-CF 3 -4-OMe-2-Py], [BG346 _{: 5-CF 3 -4-OMe} -2-Py], [BG347: 6-CF 3 -4-OMe-2-Py], [BG348: 3-CN-4-OMe-2-Py], [BG349 : 5-CN-4-OMe-2-Py], [BG350: 6-CN-4-OMe-2-Py], [BG351: 3-OMe-4-OMe-2-Py], [BG352: 5] -OMe-4-OMe-2-Py], [BG 353: 6-OMe-4-OMe-2-Py], [BG 354: 5-OMe-2-Py], [BG 355: 3-Cl-5-OMe -2-Py !, [BG 356: 4-Cl-5-OMe-2-Py], [BG 357: 6-Cl-5-OMe-2-Py], [BG 358: 3-Me-5-OMe-2] -Py], [BG359: 4- Me-5-OMe-2-Py], [BG360: 6-Me-5-OMe-2-Py], [BG361: 3-CF 3 -5-OMe-2- Py], [BG 362: 4-CF ₃ -5-OMe -2-Py], [BG 363: 6-CF ₃ -5-OMe -2-Py], [BG 3 64: 3-CN -5-OMe -2-] Py], [BG365: 4-CN-5-OMe-2-Py], [BG366: 6-CN-5-OMe-2-Py], [BG367: 3-OMe-5-OMe-2-Py] , [BG368: 4-OMe-5-OMe-2-Py], [BG369: 6-OMe-5-OMe-2-Py], [BG370: 6-OMe-2-Py], [BG371: 3- Cl-6-OMe-2-Py], [BG 372: 4-Cl-6-OMe-2-Py], [BG 373: 5-Cl-6-OMe-2-Py], [BG 374: 3-Me- 6-OMe-2-Py] , [BG375: 4-Me-6-OMe-2-Py], [BG376: 5-Me-6-OMe-2-Py], [BG377: 3-CF 3 -6 -OMe-2-Py], [ BG378: 4-CF 3 -6-OMe-2-Py], [BG379: 5-CF 3 -6-OMe-2-Py], [BG380: 3-CN-6 -OMe-2-Py], [BG 381: 4-CN-6-OMe-2-Py], [BG 382: 5-CN-6-OMe-2-Py], [BG383: 3-OMe-6-OMe] -2-Py !, [BG 384: 4-OMe-6-OMe-2-Py], [BG 385: 5-OMe-6-OMe-2-Py], [BG 386: 3-CF ₃ -2-Py] [BG 387: 4-Cl-3-CF ₃ -2-Py], [BG 388: 5-Cl-3-CF ₃ -2-Py], [BG 389: 6-Cl -3-CF ₃ -2-Py] ], [BG390: 4-Me -3-CF 3 -2-Py], [BG391: 5-Me-3-CF 3 -2-Py], [BG392: 6-Me-3-CF 3 -2- Py], [BG 393: 4-CF ₃ -3-CF ₃ -2-Py], [BG 394: 5-CF ₃ -3-CF ₃ -2-Py], [BG 395: 6-CF ₃ -3-CF ₃ -2-Py !, [BG 396: 4-CN-3-CF ₃ -2-Py], [BG 397: 5-CN-3-CF ₃ -2-Py], [BG 398: 6-CN -3- CF ₃ -2-Py !, [BG 399: 4-OMe-3-CF ₃ -2-Py], [BG 400: 5-OMe -3-CF ₃ -2-Py],

[BG401: 6-OMe-3 -CF 3 -2-Py], [BG402: 4-CF 3 -2-Py], [BG403: 3-Cl-4-CF 3 -2-Py], [BG404: _{5-Cl-4-CF 3} -2-Py], [BG405: 6-Cl-4-CF 3 -2-Py], [BG406: 3-Me-4-CF 3 -2-Py], [BG407 : 5-Me-4-CF 3 -2-Py], [BG408: 6-Me-4-CF 3 -2-Py], [BG409: 3-CF 3 -4-CF 3 -2-Py], [BG410: 5-CF ₃ -4-CF ₃ -2-Py], [BG411: 6-CF ₃ -4-CF ₃ -2-Py], [BG 412: 3-CN -4-CF ₃ -2-] Py], [BG413: 5- CN-4-CF 3 -2-Py], [BG414: 6-CN-4-CF 3 -2-Py], [BG415: 3-OMe-4-CF 3 -2 -Py], [BG416: 5- OMe-4-CF 3 -2-Py], [BG417: 6-OMe-4-CF 3 -2-Py], [BG418: 5-CF 3 -2-Py] , [BG419: 3-Cl- 5-CF 3 -2-Py], [BG420: 4-Cl-5-CF 3 -2-Py], [BG421: 6-Cl-5-CF 3 -2-Py ], [BG422: 3-Me -5-CF 3 -2-Py], [BG423: 4-Me-5-CF 3 -2-Py], [BG424: 6-Me-5-CF 3 -2- Py], [BG 425: 3-CF ₃ -5-CF ₃ -2-Py], [BG 426: 4-CF ₃ -5-CF ₃ -2-Py], [BG 427: 6-CF ₃ -5- CF ₃ -2-Py], [BG 428: 3-CN-5-CF ₃ -2-Py], [BG 429: 4-CN-5-CF ₃ -2-Py], [BG 430: 6-CN -5-] CF ₃ -2-Py !, [BG 431: 3-OMe-5-CF ₃ -2-Py], [BG 432: 4-OMe-5-CF ₃ -2-Py], [BG 433: 6-OMe-5] -CF ₃ -2-Py], [BG 434: 6-CF ₃ -2-Py], [BG 435: 3-Cl-6-CF ₃ -2-Py], [BG 436: 4-Cl 6-CF ₃ -2-Py !, [BG 437: 5-Cl-6-CF ₃ -2-Py], [BG 438: 3-Me-6-CF ₃ -2-Py], [B] G439: 4-Me-6- CF 3 -2-Py], [BG440: 5-Me-6-CF 3 -2-Py], [BG441: 3-CF 3 -6-CF 3 -2-Py] _{, [BG442: 4-CF 3} -6-CF 3 -2-Py], [BG443: 5-CF 3 -6-CF 3 -2-Py], [BG444: 3-CN-6-CF 3 -2 -Py], [BG445: 4- CN-6-CF 3 -2-Py], [BG446: 5-CN-6-CF 3 -2-Py], [BG447: 3-OMe-6-CF 3 - 2-Py], [BG448: 4-OMe-6-CF 3 -2-Py], [BG449: 5-OMe-6-CF 3 -2-Py], [BG450: 3-OCF 3 -2-Py ], [BG 451: 4-Cl-3-OCF ₃ -2-Py], [BG 452: 5-Cl -3-OCF ₃ -2-Py], [BG 453: 6-Cl -3-OCF ₃ -2-] Py], [BG454: 4- Me-3-OCF 3 -2-Py], [BG455: 5-Me-3-OCF 3 -2-Py], [BG456: 6-Me-3-OCF 3 -2 -Py], [BG 457: 4-CF ₃ -3-OCF ₃ -2-Py], [BG 458: 5-CF ₃ -3-OCF ₃ -2-Py], [BG 459: 6-CF ₃ -3-] OCF ₃ -2-Py !, [BG 460: 4-CN-3-OCF ₃ -2-Py], [BG 461: 5-CN-3-OCF ₃ -2-Py], [BG 462: 6-CN-3] _{-OCF 3 -2-Py], [} BG463: 4-OMe-3-OCF 3 -2-Py], [BG464: 5-OMe-3-OCF 3 -2-Py], [BG465: 6-OMe- _{3-OCF 3 -2-Py]} , [BG466: 4-OCF 3 -2-Py], [BG467: 3-Cl-4-OCF 3 -2-Py], [BG468: 5-Cl-4-OCF ₃ -2-Py !, [BG469: 6-Cl-4-OCF ₃ -2-Py], [BG 470: 3-Me-4-OCF ₃ -2-Py], [BG 471: 5-Me-4- 4 OCF ₃ -2-Py !, [BG 472: 6-Me-4-OCF ₃ -2-Py], [BG 473: 3-CF ₃ -4-OCF ₃ -2-Py], [BG 474: 5-CF _3] -4-OCF ₃ -2-Py], [BG 475: 6-CF ₃ -4-OCF ₃ -2-Py !, [BG 476: 3-CN -4-OCF ₃ -2-Py], [BG 477: 5-CN -4-OCF ₃ -2-Py], [BG 478: 6-CN -4- OCF ₃ -2-Py !, [BG 479: 3-OMe -4-OCF ₃ -2-Py], [BG 480: 5-OMe -4-OCF ₃ -2-Py], [BG 481: 6-OMe 4] _{-OCF 3 -2-Py], [} BG482: 5-OCF 3 -2-Py], [BG483: 3-Cl-5-OCF 3 -2-Py], [BG484: 4-Cl-5-OCF 3 -2-Py], [BG 485: 6-Cl-5-OCF ₃ -2-Py], [BG 486: 3-Me-5-OCF ₃ -2-Py], [BG 487: 4-Me-5-OCF] ₃ -2-Py, [BG 488: 6-Me-5-OCF ₃ -2-Py], [BG 489: 3-CF ₃ -5-OCF ₃ -2-Py], [BG 490: 4-CF _{3- 5-OCF 3 -2-Py]} , [BG491: 6-CF 3 -5-OCF 3 -2-Py], [BG492: 3-CN-5-OCF 3 -2-Py], [BG493: 4- _{CN-5-OCF 3 -2-} Py], [BG494: 6-CN-5-OCF 3 -2-Py], [BG495: 3-OMe-5-OCF 3 -2-Py], [BG496: 4 _{-OMe-5-OCF 3 -2-} Py], [BG497: 6-OMe-5-OCF 3 -2-Py], [BG498: 6-OCF 3 -2-Py], [BG499: 3-Cl- _{6-OCF 3 -2-Py]} , [BG500: 4-Cl-6-OCF 3 -2-Py],

[BG501: 5-Cl-6 -OCF 3 -2-Py], [BG502: 3-Me-6-OCF 3 -2-Py], [BG503: 4-Me-6-OCF 3 -2-Py] , [BG504: 5-Me- 6-OCF 3 -2-Py], [BG505: 3-CF 3 -6-OCF 3 -2-Py], [BG506: 4-CF 3 -6-OCF 3 -2 -Py], [BG507: 5- CF 3 -6-OCF 3 -2-Py], [BG508: 3-CN-6-OCF 3 -2-Py], [BG509: 4-CN-6-OCF 3 -2-Py], [BG510: 5-CN-6-OCF 3 -2-Py], [BG511: 3-OMe-6-OCF 3 -2-Py], [BG512: 4-OMe-6-OCF _{3 -2-Py], [BG513} : 5-OMe-6-OCF 3 -2-Py], [BG514: 3-CHF 2 -2-Py], [BG515: 4-Cl-3-CHF 2 -2 -Py], [BG516: 5- Cl-3-CHF 2 -2-Py], [BG517: 6-Cl-3-CHF 2 -2-Py], [BG518: 4-Me-3-CHF 2 - 2-Py], [BG519: 5-Me-3-CHF 2 -2-Py], [BG520: 6-Me-3-CHF 2 -2-Py], [BG521: 4-CF 3 -3-CHF ₂ -2-Py !, [BG 522: 5-CF ₃ -3-CHF ₂ -2-Py], [BG 523: 6-CF ₃ -3-CHF ₂ -2-Py], [BG 524: 4-CN- _{3-CHF 2 -2-Py]} , [BG525: 5-CN-3-CHF 2 -2-Py], [BG526: 6-CN-3-CHF 2 -2-Py], [BG527: 4-OMe _{-3-CHF 2 -2-Py]} , [BG528: 5-OMe-3-CHF 2 -2-Py], [BG529: 6-OMe-3-CHF 2 -2-Py], [BG530: 4- _{CHF 2 -2-Py], [} BG531: 3-Cl-4-CHF 2 -2-Py], [BG532: 5-Cl-4-CHF 2 -2-Py], [BG533: 6-Cl-4 -CHF ₂ -2-Py], [BG 534: 3-Me 4-CHF ₂ -2-Py], [BG 535: 5-Me 4-CHF ₂ 2-Py], [BG 536: 6-Me- 4-CHF ₂ -2-Py], [BG 537: 3-CF ₃ -4-CHF ₂ -2-Py], [BG 538: 5-CF ₃ -4-CHF ₂ -2-Py], [BG 539: 6-CF ₃ -4-CHF ₂ -2-Py], [BG 540: _{3-CN-4-CHF 2} -2-Py], [BG541: 5-CN-4-CHF 2 -2-Py], [BG542: 6-CN-4-CHF 2 -2-Py], [BG543 : 3-OMe-4-CHF 2 -2-Py], [BG544: 5-OMe-4-CHF 2 -2-Py], [BG545: 6-OMe-4-CHF 2 -2-Py], [ _{BG546: 5-CHF 2 -2-} Py], [BG547: 3-Cl-5-CHF 2 -2-Py], [BG548: 4-Cl-5-CHF 2 -2-Py], [BG549: 6 _{-Cl-5-CHF 2 -2-} Py], [BG550: 3-Me-5-CHF 2 -2-Py], [BG551: 4-Me-5-CHF 2 -2-Py], [BG552: 6-Me-5-CHF ₂ -2-Py, [BG553: 3-CF ₃ -5-CHF ₂ -2-Py], [BG 554: 4-CF ₃ -5-CHF ₂ -2-Py], _{[BG555: 6-CF 3 -5} -CHF 2 -2-Py], [BG556: 3-CN-5-CHF 2 -2-Py], [BG557: 4-CN-5-CHF 2 -2-Py ], [BG 558: 6-CN-5-CHF ₂ -2-Py], [BG 559: 3-OMe-5-CHF ₂ -2-Py], [BG 560: 4-OMe-5-CHF ₂ -2-] Py], [BG561: 6- OMe-5-CHF 2 -2-Py], [BG562: 6-CHF 2 -2-Py], [BG563: 3-Cl-6-CHF 2 -2-Py], [BG 564: 4-Cl-6-CHF ₂ -2-Py], [BG 565: 5-Cl 6-CHF ₂ -2-Py], [BG 566: 3-Me-6-CHF ₂ -2-Py] , [BG 567: 4-Me-6-CHF ₂ -2-Py], [BG 568: 5-Me-6-CHF ₂ -2-Py], [BG 569: 3-CF ₃ -6-CHF ₂ -2- Py], [BG570: 4- CF 3 -6-CHF 2 -2-Py], [BG571: 5-CF 3 -6-CHF 2 -2-Py], [BG572: 3-CN-6-CHF 2 -2-Py], [BG 573: 4-CN-6-CHF ₂ -2-Py !, [BG 574: 5-CN-6-CHF ₂ -2-Py], [BG 575: 3-OMe-6-CHF ₂ -2-Py], [BG 576: 4-OMe-6-CHF _{2 -2-Py], [BG577} : 5-OMe-6-CHF 2 -2-Py], [BG578: 3-OCHF 2 -2-Py], [BG579: 4-Cl-3-OCHF 2 -2 -Py], [BG 580: 5-Cl-3-OCHF ₂ -2-Py], [BG 581: 6-Cl-3-OCHF ₂ -2-Py], [BG 582: 4-Me-3-OCHF _2- 2-Py], [BG 583: 5-Me-3-OCHF ₂ -2-Py], [BG 584: 6-Me-3-OCHF ₂ -2-Py], [BG 585: 4-CF ₃ -3-OCHF ₂ -2-Py], [BG 586: 5-CF ₃ -3-OCHF ₂ -2-Py], [BG 587: 6-CF ₃ -3-OCHF ₂ -2-Py], [BG 588: 4-CN- 3-OCHF ₂ -2-Py], [BG 589: 5-CN-3-OCHF ₂ -2-Py], [BG 590: 6-CN -3-OCHF ₂ -2-Py], [BG 59 1: 4-OMe] _{-3-OCHF 2 -2-Py]} , [BG592: 5-OMe-3-OCHF 2 -2-Py], [BG593: 6-OMe-3-OCHF 2 -2-Py], [BG594: 4- _{OCHF 2 -2-Py], [} BG595: 3-Cl-4-OCHF 2 -2-Py], [BG596: 5-Cl-4-OCHF 2 -2-Py], [BG597: 6-Cl-4 _{-OCHF 2 -2-Py], [} BG598: 3-Me-4-OCHF 2 -2-Py], [BG599: 5-Me-4-OCHF 2 -2-Py], [BG600: 6-Me- 4-OCHF ₂ -2-Py],

_{[BG601: 3-CF 3 -4} -OCHF 2 -2-Py], [BG602: 5-CF 3 -4-OCHF 2 -2-Py], [BG603: 6-CF 3 -4-OCHF 2 -2 -Py], [BG604: 3- CN-4-OCHF 2 -2-Py], [BG605: 5-CN-4-OCHF 2 -2-Py], [BG606: 6-CN-4-OCHF 2 - 2-Py], [BG 607: 3-OMe-4-OCHF ₂ -2-Py], [BG 608: 5-OMe-4-OCHF ₂ -2-Py], [BG 609: 6-OMe-4-OCHF ₂ -2-Py], [BG610: 5-OCHF 2 -2-Py], [BG611: 3-Cl-5-OCHF 2 -2-Py], [BG612: 4-Cl-5-OCHF 2 -2- Py], [BG613: 6- Cl-5-OCHF 2 -2-Py], [BG614: 3-Me-5-OCHF 2 -2-Py], [BG615: 4-Me-5-OCHF 2 -2 -Py], [BG 616: 6-Me-5-OCHF ₂ -2-Py], [BG 617: 3-CF ₃ -5-OCHF ₂ -2-Py], [BG 618: 4-CF ₃ -5-OCHF _{2 -2-Py], [BG619} : 6-CF 3 -5-OCHF 2 -2-Py], [BG620: 3-CN-5-OCHF 2 -2-Py], [BG621: 4-CN-5 _{-OCHF 2 -2-Py], [} BG622: 6-CN-5-OCHF 2 -2-Py], [BG623: 3-OMe-5-OCHF 2 -2-Py], [BG624: 4-OMe- 5-OCHF ₂ -2-Py, [BG 625: 6-OMe -5-OCHF ₂ -2-Py], [BG 626: 6-OCHF ₂ -2-Py], [BG 627: 3-Cl -6-OCHF ₂ -2-Py], [BG 628: 4-Cl-6-OCHF ₂ -2-Py], [BG 629: 5-Cl 6-OCHF ₂ -2-Py], [BG 630: 3-Me -6-] OFHF ₂ -2-Py, [BG 631: 4-Me-6-OCHF ₂ -2-Py], [BG 632: 5-Me-6-OCHF ₂ -2-Py], [BG 633: 3-CF _3- 6-OCHF ₂ -2-Py, [BG 634: 4-CF ₃ -6-OCHF ₂ -2-Py], [BG 635: 5-CF ₃ -6-OCHF ₂ -2- P] y], [BG636: 3- CN-6-OCHF 2 -2-Py], [BG637: 4-CN-6-OCHF 2 -2-Py], [BG638: 5-CN-6-OCHF 2 -2 -Py], [BG639: 3- OMe-6-OCHF 2 -2-Py], [BG640: 4-OMe-6-OCHF 2 -2-Py], [BG641: 5-OMe-6-OCHF 2 - 2-Py], [BG 642: 3-Et-2-Py], [BG 643: 4-Cl-3-Et-2-Py], [BG 644: 5-Cl-3-Et-2-Py], [BG BG645: 6-Cl-3-Et-2-Py, [BG646: 4-Me-3-Et-2-Py], [BG647: 5-Me-3-Et-2-Py], [BG 648: 6-Me-3-Et- 2-Py], [BG649: 4-CF 3 -3-Et-2-Py], [BG650: 5-CF 3 -3-Et-2-Py], [BG651: _{6-CF 3 -3-Et-} 2-Py], [BG652: 4-CN-3-Et-2-Py], [BG653: 5-CN-3-Et-2-Py], [BG654: 6 -CN-3-Et-2-Py], [BG655: 4-OMe-3-Et-2-Py], [BG656: 5-OMe-3-Et-2-Py], [BG657: 6-OMe] -3-Et-2-Py, [BG 658: 4-Et-2-Py], [BG 659: 3-Cl-4-Et-2-Py], [BG 660: 5-Cl-4-Et-2 -Py], [BG661: 6-Cl-4-Et-2-Py], [BG662: 3-Me-4-Et-2-Py], [BG663: 5-Me-4-Et-2-Py] ], [BG 664: 6-Me-4-Et-2-Py], [BG 665: 3-CF ₃ -4-Et-2-Py], [BG 666: 5-CF ₃ -4-Et-2-Py] ], [BG 667: 6-CF ₃ -4-Et-2-Py], [BG 668: 3-CN-4-Et-2-Py], [BG 669: 5-CN-4-Et-2-Py] [BG 670: 6-CN-4-Et-2-Py], [BG 671: 3-OMe-4-Et-2-Py], [BG 672: 5-OMe-4-Et-2-Py], [BG 672: 5-OMe BG 673: 6-OMe-4-Et-2-Py], [BG 674: 5-Et-2-Py], [BG 675: 3-Cl-5-Et-2-Py], [BG 676: 4-Cl- 5-Et-2-Py], [BG 677: 6-Cl- 5-Et-2-Py], [BG 678: 3-Me-5-Et-2-Py], [BG 679: 4-Me-5-Et-2-Py], [BG 680: 6-Me-5-] Et-2-Py], [ BG681: 3-CF 3 -5-Et-2-Py], [BG682: 4-CF 3 -5-Et-2-Py], [BG683: 6-CF 3 -5 -Et-2-Py], [BG 684: 3-CN-5-Et-2-Py], [BG 685: 4-CN-5-Et-2-Py], [BG 686: 6-CN-5-Et] -2-Py !, [BG 687: 3-OMe-5-Et-2-Py], [BG 688: 4-OMe-5-Et-2-Py], [BG 689: 6-OMe-5-Et-2] -Py], [BG 690: 6-Et-2-Py], [BG691: 3-Cl-6-Et-2-Py], [BG692: 4-Cl-6-Et-2-Py], [BG693] : 5-Cl-6-Et-2-Py], [BG 694: 3-Me-6-Et-2-Py], [BG 695: 4-Me-6-Et-2-Py], [BG 696: 5] -Me-6-Et-2-Py], [BG 697: 3-CF ₃ -6-Et-2-Py], [BG 698: 4-CF ₃ -6-Et-2-Py], [BG 699: 5] _{-CF 3 -6-Et-2-} Py], [BG700: 3-CN-6-Et-2-Py],

[BG701: 4-CN-6-Et-2-Py], [BG702: 5-CN-6-Et-2-Py], [BG703: 3-OMe-6-Et-2-Py], [BG704] : 4-OMe-6-Et -2-Py], [BG705: 5-OMe-6-Et-2-Py], [BG706: 3-CH 2 CF 3 -2-Py], [BG707: 4- _{Cl-3-CH 2 CF 3} -2-Py], [BG708: 5-Cl-3-CH 2 CF 3 -2-Py], [BG709: 6-Cl-3-CH 2 CF 3 -2-Py ], [BG710: 4-Me -3-CH 2 CF 3 -2-Py], [BG711: 5-Me-3-CH 2 CF 3 -2-Py], [BG712: 6-Me-3-CH ₂ CF ₃ -2-Py, [BG 713: 4-CF ₃ -3-CH ₂ CF ₃ -2-Py], [BG 714: 5-CF ₃ -3-CH ₂ CF ₃ -2-Py], _{BG715: 6-CF 3 -3-} CH 2 CF 3 -2-Py], [BG716: 4-CN-3-CH 2 CF 3 -2-Py], [BG717: 5-CN-3-CH 2 CF ₃ -2-Py !, [BG 718: 6-CN-3-CH ₂ CF ₃ -2-Py], [BG 719: 4-OMe -3-CH ₂ CF ₃ -2-Py], [BG 720: 5-] OMe-3-CH ₂ CF ₃ -2-Py, [BG 721: 6-OMe -3-CH ₂ CF ₃ -2-Py], [BG 72 ₂ : 4-CH ₂ CF ₃ -2-Py], [BG 723] : 3-Cl-4-CH 2 CF 3 -2-Py], [BG724: 5-Cl-4-CH 2 CF 3 -2-Py], [BG725: 6-Cl-4-CH 2 CF 3 - 2-Py], [BG 726: 3-Me-4-CH ₂ CF ₃ -2-Py], [BG 727: 5-Me-4-CH ₂ CF ₃ -2-Py], [BG 728: 6-Me- _{4-CH 2 CF 3 -2-} Py], [BG729: 3-CF 3 -4-CH 2 CF 3 -2-Py], [BG730: 5-CF 3 -4-CH 2 CF 3 -2-Py ], [BG731: 6-CF 3 -4-CH 2 CF 3 -2-Py], [BG732: 3-CN-4-CH 2 CF 3 -2-Py], [BG733: 5-CN-4- CH ₂ CF ₃ -2-Py], [BG 734: 6-CN-4- CH 2 CF 3 -2-Py], [BG735: 3-OMe-4-CH 2 CF 3 -2-Py], [BG736: 5-OMe-4-CH 2 CF 3 -2-Py], [BG 737: 6-OMe-4-CH ₂ CF ₃ -2-Py], [BG 738: 5-CH ₂ CF ₃ -2-Py], [BG 739: 3-Cl-5-CH ₂ CF ₃ -2-Py, [BG 740: 4-Cl-5-CH ₂ CF ₃ -2-Py], [BG 741: 6-Cl-5-CH ₂ CF ₃ -2-Py], [BG 742: _{3-Me-5-CH 2} CF 3 -2-Py], [BG743: 4-Me-5-CH 2 CF 3 -2-Py], [BG744: 6-Me-5-CH 2 CF 3 -2 -Py], [BG 745: 3-CF ₃ -5-CH ₂ CF ₃ -2-Py], [BG 746: 4-CF ₃ -5-CH ₂ CF ₃ -2-Py], [BG 747: 6-CF] _{3 -5-CH 2 CF 3 -2} -Py], [BG748: 3-CN-5-CH 2 CF 3 -2-Py], [BG749: 4-CN-5-CH 2 CF 3 -2-Py ], [BG750: 6-CN -5-CH 2 CF 3 -2-Py], [BG751: 3-OMe-5-CH 2 CF 3 -2-Py], [BG752: 4-OMe-5-CH ₂ CF ₃ -2-Py, [BG 753: 6-OMe-5-CH ₂ CF ₃ -2-Py], [BG 754: 6-CH ₂ CF ₃ -2-Py], [BG 755: 3-Cl- _{6-CH 2 CF 3 -2-} Py], [BG756: 4-Cl-6-CH 2 CF 3 -2-Py], [BG757: 5-Cl-6-CH 2 CF 3 -2-Py], [BG758: 3-Me-6 -CH 2 CF 3 -2-Py], [BG759: 4-Me-6-CH 2 CF 3 -2-Py], [BG760: 5-Me-6-CH 2 CF ₃ -2-Py], [BG 761: 3-CF ₃ -6-CH ₂ CF ₃ -2-Py], [BG 762: 4-CF ₃ -6-CH ₂ CF ₃ -2-Py], [BG 763: _{5-CF 3 -6-CH 2} CF 3 -2-Py], [BG764: 3-CN-6-CH 2 CF 3 -2-Py], [BG765: 4-CN-6-CH 2 CF 3 - 2-P y], [BG766: 5- CN-6-CH 2 CF 3 -2-Py], [BG767: 3-OMe-6-CH 2 CF 3 -2-Py], [BG768: 4-OMe-6- _{CH 2 CF 3 -2-Py]} , [BG769: 5-OMe-6-CH 2 CF 3 -2-Py], [BG770: 3-OEt-2-Py], [BG771: 4-Cl-3- OEt-2-Py, [BG 772: 5-Cl-3-OEt-2-Py], [BG773: 6-Cl-3-OEt-2-Py], [BG 774: 4-Me-3-OEt- 2-Py], [BG 775: 5-Me-3-OEt-2-Py], [BG 776: 6-Me-3-OEt-2-Py], [BG 777: 4-CF ₃ -3-OEt-2 -Py], [BG 778: 5-CF ₃ -3-OEt-2-Py], [BG 779: 6-CF ₃ -3-OEt-2-Py], [BG 780: 4-CN-3-OEt-2 -Py], [BG781: 5-CN-3-OEt-2-Py], [BG 782: 6-CN-3-OEt-2-Py], [BG783: 4-OMe-3-OEt-2-Py] ], [BG 784: 5-OMe-3-OEt-2-Py], [BG 785: 6-OMe-3-OEt-2-Py], [BG 786: 4-OEt-2-Py], [BG 787: 3] -Cl-4-OEt-2-Py], [BG 788: 5-Cl-4-OEt-2-Py], [BG 789: 6-Cl-4-OEt-2-Py], [BG 790: 3-Me -4-OEt-2-Py !, [BG 791: 5-Me-4-OEt-2-Py], [BG 792: 6-Me-4-OEt-2-Py], [BG 793: 3-CF _3- 4-OEt-2-Py !, [BG 794: 5-CF ₃ -4-OEt-2-Py], [BG79 5: 6-CF ₃ -4-OEt-2-Py], [BG 796: 3-CN- 4-OEt-2-Py, [BG 797: 5-CN-4-OEt-2-Py], [BG 798: 6-CN-4-OEt-2-Py], [BG 799: 3-OMe-4-] OEt-2-Py], [BG800: 5-OMe-4-OEt-2-Py],

[BG801: 6-OMe-4-OEt-2-Py], [BG802: 5-OEt-2-Py], [BG803: 3-Cl-5-OEt-2-Py], [BG804: 4-Cl -5-OEt-2-Py !, [BG 805: 6-Cl-5-OEt-2-Py], [BG 806: 3-Me-5-OEt-2-Py], [BG 807: 4-Me-5] -OEt-2-Py], [ BG808: 6-Me-5-OEt-2-Py], [BG809: 3-CF 3 -5-OEt-2-Py], [BG810: 4-CF 3 -5 -OEt-2-Py], [ BG811: 6-CF 3 -5-OEt-2-Py], [BG812: 3-CN-5-OEt-2-Py], [BG813: 4-CN-5- OEt-2-Py, [BG 814: 6-CN-5-OEt-2-Py], [BG 815: 3-OMe-5-OEt-2-Py], [BG 816: 4-OMe-5-OEt- 2-Py], [BG 817: 6-OMe-5-OEt-2-Py], [BG 818: 6-OEt-2-Py], [BG 819: 3-Cl-6-OEt-2-Py], BG 820: 4-Cl-6-OEt-2-Py !, [BG 821: 5-Cl-6-OEt-2-Py], [BG 822: 3-Me-6-OEt-2-Py], [BG 823: 4-Me-6-OEt- 2-Py], [BG824: 5-Me-6-OEt-2-Py], [BG825: 3-CF 3 -6-OEt-2-Py], [BG826: 4 _{-CF 3 -6-OEt-2-} Py], [BG827: 5-CF 3 -6-OEt-2-Py], [BG828: 3-CN-6-OEt-2-Py], [BG829: 4 -CN-6-OEt-2-Py], [BG 830: 5-CN-6-OEt-2-Py], [BG 831: 3-OMe-6-OEt-2-Py], [BG 832: 4-OMe] -6-OEt-2-Py] , [BG833: 5-OMe-6-OEt-2-Py], [BG834: 3-OCH 2 CF 3 -2-Py], [BG835: 4-Cl-3- _{OCH 2 CF 3 -2-Py]} , [BG836: 5-Cl-3-OCH 2 CF 3 -2-Py], [BG837: 6-Cl-3-OCH 2 CF 3 -2-Py], [BG838 : 4-Me-3-OCH 2 CF 3 -2-Py], [BG839: 5-Me-3-OCH 2 CF 3 -2-Py], [BG840 : 6-Me-3-OCH 2 CF 3 -2-Py], [BG841: 4-CF 3 -3-OCH 2 CF 3 -2-Py], [BG842: 5-CF 3 -3-OCH 2 CF ₃ -2-Py, [BG 843: 6-CF ₃ -3-OCH ₂ CF ₃ -2-Py], [BG 844: 4-CN -3-OCH ₂ CF ₃ -2-Py], [BG 845: 5] _{-CN-3-OCH 2 CF 3} -2-Py], [BG846: 6-CN-3-OCH 2 CF 3 -2-Py], [BG847: 4-OMe-3-OCH 2 CF 3 -2- Py], [BG848: 5- OMe-3-OCH 2 CF 3 -2-Py], [BG849: 6-OMe-3-OCH 2 CF 3 -2-Py], [BG850: 4-OCH 2 CF 3 -2-Py !, [BG 851: 3-Cl-4-OCH ₂ CF ₃ -2-Py], [BG 852: 5-Cl 4-OCH ₂ CF ₃ -2-Py], [BG 853: 6-Cl] _{-4-OCH 2 CF 3 -2-} Py], [BG854: 3-Me-4-OCH 2 CF 3 -2-Py], [BG855: 5-Me-4-OCH 2 CF 3 -2-Py] , [BG 856: 6-Me-4-OCH ₂ CF ₃ -2-Py], [BG 857: 3-CF ₃ -4-OCH ₂ CF ₃ -2-Py], [BG 858: 5-CF ₃ -4-] OCH ₂ CF ₃ -2-Py], [BG 859: 6-CF ₃ -4-OCH ₂ CF ₃ -2-Py], [BG 860: 3-CN-4-OCH ₂ CF ₃ -2-Py], BG861: 5-CN-4- OCH 2 CF 3 -2-Py], [BG862: 6-CN-4-OCH 2 CF 3 -2-Py], [BG863: 3-OMe-4-OCH 2 CF 3 -2-Py], [BG864: 5-OMe-4-OCH 2 CF 3 -2-Py], [BG865: 6-OMe-4-OCH 2 CF 3 -2-Py], [BG866: 5-OCH _{2 CF 3 -2-Py],} [BG867: 3-Cl-5-OCH 2 CF 3 -2-Py], [BG868: 4-Cl-5-OCH 2 CF 3 -2-Py], [BG869: _{6-Cl-5-OCH 2} CF 3 -2-Py], [BG870: 3-Me-5-OCH 2 CF 3 -2-Py], [BG 871: 4-Me-5-OCH ₂ CF ₃ -2-Py], [BG 872: 6-Me-5-OCH ₂ CF ₃ -2-Py], [BG 873: 3-CF ₃ -5-OCH ₂ CF ₃ -2-Py !, [BG 874: 4-CF ₃ -5-OCH ₂ CF ₃ -2-Py], [BG 875: 6-CF ₃ -5-OCH ₂ CF ₃ -2-Py], [BG 876] : 3-CN-5-OCH 2 CF 3 -2-Py], [BG877: 4-CN-5-OCH 2 CF 3 -2-Py], [BG878: 6-CN-5-OCH 2 CF 3 - 2-Py], [BG879: 3-OMe-5-OCH 2 CF 3 -2-Py], [BG880: 4-OMe-5-OCH2CF 3 -2-Py], [BG881: 6-OMe-5- _{OCH2CF 3 -2-Py], [} BG882: 6-OCH2CF 3 -2-Py], [BG883: 3-Cl-6-OCH 2 CF 3 -2-Py], [BG884: 4-Cl-6-OCH ₂ CF ₃ -2-Py], [BG 885: 5-Cl-6-OCH ₂ CF ₃ -2-Py], [BG 886: 3-Me-6-OCH ₂ CF ₃ -2-Py], [BG 887: _{4-Me-6-OCH 2} CF 3 -2-Py], [BG888: 5-Me-6-OCH 2 CF 3 -2-Py], [BG889: 3-CF 3 -6-OCH 2 CF 3 - 2-Py], [BG890: 4-CF 3 -6-OCH 2 CF 3 -2-Py], [BG891: 5-CF 3 -6-OCH 2 CF 3 -2-Py], [BG892: 3- _{CN-6-OCH 2 CF 3} -2-Py], [BG893: 4-CN-6-OCH 2 CF 3 -2-Py], [BG894: 5-CN-6-OCH 2 CF 3 -2-Py ], [BG 895: 3-OMe-6-OCH ₂ CF ₃ -2-Py], [BG 896: 4-OMe-6-OCH ₂ CF ₃ -2-Py], [BG 897: 5-OMe -6-OCH ₂ CF ₃ -2-Py, [BG 898: 3-Pr-2-Py], [BG 899: 4-Cl-3-Pr-2-Py], [BG 900: 5-Cl-3-Pr-2-] Py],

[BG901: 6-Cl-3-Pr-2-Py], [BG902: 4-Me-3-Pr-2-Py], [BG 903: 5-Me-3-Pr-2-Py], [BG904] : 6-Me-3-Pr-2-Py], [BG 905: 4-CF ₃ -3-Pr-2-Py], [BG 906: 5-CF ₃ -3-Pr-2-Py], [BG 907] _{: 6-CF 3 -3-Pr} -2-Py], [BG908: 4-CN-3-Pr-2-Py], [BG909: 5-CN-3-Pr-2-Py], [BG910: 6-CN-3-Pr-2-Py, [BG 911: 4-OMe-3-Pr-2-Py], [BG 912: 5-OMe-3-Pr-2-Py], [BG 913: 6- OMe-3-Pr-2-Py], [BG 914: 4-Pr-2-Py], [BG 915: 3-Cl-4-Pr-2-Py], [BG 916: 5-Cl-4-Pr- 2-Py], [BG 917: 6-Cl-4-Pr-2-Py], [BG 918: 3-Me-4-Pr-2-Py], [BG 919: 5-Me-4-Pr-2- Py], [BG920: 6- Me-4-Pr-2-Py], [BG921: 3-CF 3 -4-Pr-2-Py], [BG922: 5-CF 3 -4-Pr-2- Py], [BG 923: 6-CF ₃ -4-Pr-2-Py], [BG 924: 3-CN-4-Pr-2-Py], [BG 925: 5-CN-4-Pr-2-Py ], [BG 926: 6-CN-4-Pr-2-Py], [BG 927: 3-OMe-4-Pr-2-Py], [BG 928: 5-OMe-4-Pr-2-Py], [BG 929: 6-OMe-4-Pr-2-Py], [BG 930: 5-Pr-2-Py], [BG 931: 3-Cl-5-Pr-2-Py], [BG 932: 4-Cl -5-Pr-2-Py, [BG933: 6-Cl-5-Pr-2-Py], [BG 934: 3-Me-5-Pr-2-Py], [BG 935: 4-Me-5] -Pr-2-Py], [ BG936: 6-Me-5-Pr-2-Py], [BG937: 3-CF 3 -5-Pr-2-Py], [BG938: 4-CF 3 -5 -Pr-2-Py], [ BG939: 6-CF 3 -5-Pr-2-Py], [BG940: 3-CN-5-Pr-2-Py], [BG941: 4-CN-5- Pr-2-Py, [BG942: 6-CN-5-Pr-2-Py], [BG943: 3-OM e-5-Pr-2-Py, [BG 944: 4-OMe-5-Pr-2-Py], [BG 945: 6-OMe-5-Pr-2-Py], [BG 946: 6-Pr- 2-Py], [BG 947: 3-Cl-6-Pr-2-Py], [BG 948: 4-Cl-6-Pr-2-Py], [BG 949: 5-Cl-6-Pr-2-] Py], [BG950: 3-Me-6-Pr-2-Py], [BG 951: 4-Me-6-Pr-2-Py], [BG 952: 5-Me-6-Pr-2-Py] _{, [BG953: 3-CF 3} -6-Pr-2-Py], [BG954: 4-CF 3 -6-Pr-2-Py], [BG955: 5-CF 3 -6-Pr-2-Py ], [BG956: 3-CN-6-Pr-2-Py], [BG 957: 4-CN-6-Pr-2-Py], [BG958: 5-CN-6-Pr-2-Py], [BG959: 3-OMe-6-Pr-2-Py], [BG960: 4-OMe-6-Pr-2-Py], [BG961: 5-OMe-6-Pr-2-Py], [BG962] : 3-OPr-2-Py], [BG963: 4-Cl-3-OPr-2-Py], [BG964: 5-Cl-3-OPr-2-Py], [BG965: 6-Cl-3] -OPr-2-Py], [BG966: 4-Me-3-OPr-2-Py], [BG967: 5-Me-3-OPr-2-Py], [BG968: 6-Me-3-OPr -2-Py], [BG969: 4-CF 3 -3-OPr-2-Py], [BG970: 5-CF 3 -3-OPr-2-Py], [BG971: 6-CF 3 -3- OPr-2-Py], [BG 972: 4-CN-3-OPr-2-Py], [BG 973: 5-CN-3-OPr-2-Py], [BG 974: 6-CN-3-OPr- 2-Py], [BG975: 4-OMe-3-OPr-2-Py], [BG976: 5-OMe-3-OPr-2-Py], [BG977: 6-OMe-3-OPr-2-] Py], [BG978: 4-OPr-2-Py], [BG979: 3-Cl-4-OPr-2-Py], [BG 980: 5-Cl-4-OPr-2-Py], [BG981: 6-Cl-4-OPr-2-Py, [BG982: 3-Me-4-OPr-2-Py], [BG983: 5-Me-4-OPr-2-Py], [BG984: 6- Me-4-OPr-2-Py], [BG 985: 3-C _{F 3 -4-OPr-2-} Py], [BG986: 5-CF 3 -4-OPr-2-Py], [BG987: 6-CF 3 -4-OPr-2-Py], [BG988: 3 -CN-4-OPr-2-Py], [BG989: 5-CN-4-OPr-2-Py], [BG990: 6-CN-4-OPr-2-Py], [BG991: 3-OMe] -4-OPr-2-Py, [BG992: 5-OMe-4-OPr-2-Py], [BG993: 6-OMe-4-OPr-2-Py], [BG994: 5-OPr-2 -Py], [BG995: 3-Cl-5-OPr-2-Py], [BG996: 4-Cl-5-OPr-2-Py], [BG997: 6-Cl-5-OPr-2-Py] ], [BG 998: 3-Me-5-OPr-2-Py], [BG 999: 4-Me-5-OPr-2-Py], [BG 1000: 6-Me-5-OPr-2-Py],

_{[BG1001: 3-CF 3 -5} -OPr-2-Py], [BG1002: 4-CF 3 -5-OPr-2-Py], [BG1003: 6-CF 3 -5-OPr-2-Py] , [BG1004: 3-CN-5-OPr-2-Py], [BG1005: 4-CN-5-OPr-2-Py], [BG1006: 6-CN-5-OPr-2-Py], [BG1004: BG1007: 3-OMe-5-OPr-2-Py], [BG1008: 4-OMe-5-OPr-2-Py], [BG1009: 6-OMe-5-OPr-2-Py], [BG1010: 6-OPr-2-Py !, [BG1011: 3-Cl-6-OPr-2-Py], [BG1012: 4-Cl-6-OPr-2-Py], [BG1013: 5-Cl-6-6] OPr-2-Py !, [BG1014: 3-Me-6-OPr-2-Py], [BG1015: 4-Me-6-OPr-2-Py], [BG1016: 5-Me-6-OPr- 2-Py], [BG1017: 3-CF 3 -6-OPr-2-Py], [BG1018: 4-CF 3 -6-OPr-2-Py], [BG1019: 5-CF 3 -6-OPr -2-Py !, [BG1020: 3-CN-6-OPr-2-Py], [BG1021: 4-CN-6-OPr-2-Py], [BG1022: 5-CN-6-OPr-2 -Py], [BG1023: 3-OMe-6-OPr-2-Py], [BG1024: 4-OMe-6-OPr-2-Py], [BG1025: 5-OMe-6-OPr-2-Py] ], [BG1026: 3-SMe-2-Py], [BG1027: 4-Cl-3-SMe-2-Py], [BG1028: 5-Cl-3-SMe-2-Py], [BG1029: 6] -Cl-3-SMe-2-Py], [BG1030: 4-Me-3-SMe-2-Py], [BG1031: 5-Me-3-SMe-2-Py], [BG1032: 6-Me -3-SMe-2-Py] , [BG1033: 4-CF 3 -3-SMe-2-Py], [BG1034: 5-CF 3 -3-SMe-2-Py], [BG1035: 6-CF _{3 -3-SMe-2-Py} ], [BG1036: 4-CN-3-SMe-2-Py], [BG1037: 5-CN-3-SMe-2-Py], [BG1038: 6-CN- 3-SMe-2-Py], [BG1039: 4-OMe-3-SMe-2-Py], [BG BG1040: 5-OMe-3-SMe-2-Py !, [BG1041: 6-OMe-3-SMe-2-Py], [BG1042: 4-SMe-2-Py], [BG1043: 3-Cl- 4-SMe-2-Py !, [BG1044: 5-Cl-4-SMe-2-Py], [BG1045: 6-Cl-4-SMe-2-Py], [BG1046: 3-Me-4-4] SMe-2-Py], [ BG1047: 5-Me-4-SMe-2-Py], [BG1048: 6-Me-4-SMe-2-Py], [BG1049: 3-CF 3 -4-SMe -2-Py], [BG1050: 5-CF 3 -4-SMe-2-Py], [BG1051: 6-CF 3 -4-SMe-2-Py], [BG1052: 3-CN-4-SMe -2-Py !, [BG1053: 5-CN-4-SMe-2-Py], [BG1054: 6-CN-4-SMe-2-Py], [BG1055: 3-OMe-4-SMe-2 -Py], [BG1056: 5-OMe-4-SMe-2-Py], [BG1057: 6-OMe-4-SMe-2-Py], [BG1058: 5-SMe-2-Py], [BG1059] : 3-Cl-5-SMe-2-Py], [BG1060: 4-Cl-5-SMe-2-Py], [BG1061: 6-Cl-5-SMe-2-Py], [BG1062: 3] -Me-5-SMe-2-Py], [BG1063: 4-Me-5-SMe-2-Py], [BG1064: 6-Me-5-SMe-2-Py], [BG1065: 3-CF _{3 -5-SMe-2-Py} ], [BG1066: 4-CF 3 -5-SMe-2-Py], [BG1067: 6-CF 3 -5-SMe-2-Py], [BG1068: 3- CN-5-SMe-2-Py !, [BG1069: 4-CN-5-SMe-2-Py], [BG1070: 6-CN-5-SMe-2-Py], [BG1071: 3-OMe- 5-SMe-2-Py], [BG1072: 4-OMe-5-SMe-2-Py], [BG1073: 6-OMe-5-SMe-2-Py], [BG1074: 6-SMe-2-Py] Py], [BG1075: 3-Cl-6-SMe-2-Py], [BG1076: 4-Cl-6-SMe-2-Py], [BG1077: 5-Cl-6-SMe-2-Py] , [BG1078: 3-Me-6-SMe-2-Py], [BG1079: 4-Me-6-] SMe-2-Py], [ BG1080: 5-Me-6-SMe-2-Py], [BG1081: 3-CF 3 -6-SMe-2-Py], [BG1082: 4-CF 3 -6- SMe-2-Py], [ BG1083: 5-CF 3 -6-SMe-2-Py], [BG1084: 3-CN-6-SMe-2-Py], [BG1085: 4-CN-6-SMe -2-Py], [BG1086: 5-CN-6-SMe-2-Py], [BG1087: 3-OMe-6-SMe-2-Py], [BG1088: 4-OMe-6-SMe-2 -Py], [BG1089: 5- OMe-6-SMe-2-Py], [BG1090: 3-SCF 3 -2-Py], [BG1091: 4-Cl-3-SCF 3 -2-Py], [BG1092: 5-Cl-3 -SCF 3 -2-Py], [BG1093: 6-Cl-3-SCF 3 -2-Py], [BG1094: 4-Me-3-SCF 3 -2-Py] , [BG1095: 5-Me- 3-SCF 3 -2-Py], [BG1096: 6-Me-3-SCF 3 -2-Py], [BG1097: 4-CF 3 -3-SCF 3 -2- Py], [BG1098: 5- CF 3 -3-SCF 3 -2-Py], [BG1099: 6-CF 3 -3-SCF 3 -2-Py], [BG1100: 4-CN-3-SCF 3 -2-Py],

[BG1101: 5-CN-3 -SCF 3 -2-Py], [BG1102: 6-CN-3-SCF 3 -2-Py], [BG1103: 4-OMe-3-SCF 3 -2-Py] , [BG1104: 5-OMe-3-SCF ₃ -2-Py], [BG 1105: 6-OMe-3-SCF ₃ -2-Py], [BG 1106: 4-SCF ₃ -2-Py], [BG 1107] : 3-Cl-4-SCF 3 -2-Py], [BG1108: 5-Cl-4-SCF 3 -2-Py], [BG1109: 6-Cl-4-SCF 3 -2-Py], [ BG1110: 3-Me-4- SCF 3 -2-Py], [BG1111: 5-Me-4-SCF 3 -2-Py], [BG1112: 6-Me-4-SCF 3 -2-Py], _{[BG1113: 3-CF 3 -4} -SCF 3 -2-Py], [BG1114: 5-CF 3 -4-SCF 3 -2-Py], [BG1115: 6-CF 3 -4-SCF 3 -2 -Py], [BG1116: 3- CN-4-SCF 3 -2-Py], [BG1117: 5-CN-4-SCF 3 -2-Py], [BG1118: 6-CN-4-SCF 3 - 2-Py], [BG 1119: 3-OMe-4-SCF ₃ -2-Py], [BG 1 120: 5-OMe-4-SCF ₃ -2-Py], [BG 1121: 6-OMe-4-SCF ₃ -2-Py !, [BG1122: 5-SCF ₃ -2-Py], [BG 1123: 3-Cl-5-SCF ₃ -2-Py], [BG 1 124: 4-Cl-5-SCF ₃ -2-] Py], [BG1125: 6- Cl-5-SCF 3 -2-Py], [BG1126: 3-Me-5-SCF 3 -2-Py], [BG1127: 4-Me-5-SCF 3 -2 -Py], [BG 1128: 6-Me-5-SCF ₃ -2-Py], [BG 1129: 3-CF ₃ -5-SCF ₃ -2-Py], [BG 1130: 4-CF ₃ -5- SCF ₃ -2-Py, [BG1131: 6-CF ₃ -5-SCF ₃ -2-Py], [BG 1132: 3-CN-5-SCF ₃ -2-Py], [BG 1133: 4-CN-5] -SCF ₃ -2-Py], [BG 1134: 6-CN-5-SCF ₃ -2-Py], [BG 1 135: 3-OMe-5-SCF ₃ -2-Py], [BG 11 36: 4-OMe-5-SCF ₃ -2-Py, [BG 1137: 6-OMe-5-SCF ₃ -2-Py], [BG 1138: 6-SCF ₃ -2-Py], [BG 1 139: 3] _{-Cl-6-SCF 3 -2-} Py], [BG1140: 4-Cl-6-SCF 3 -2-Py], [BG1141: 6-Cl-6-SCF 3 -2-Py], [BG1142: 3-Me-6-SCF ₃ -2-Py, [BG1143: 4-Me-6-SCF ₃ -2-Py], [BG 1144: 6-Me-6-SCF ₃ -2-Py], [BG 1 145] : 3-CF ₃ -6-SCF ₃ -2-Py], [BG 1 1 14: 4-CF ₃ -6-SCF ₃ -2-Py], [BG 1147: 6-CF ₃ -6-SCF ₃ -2-Py] ], [BG1148: 3-CN -6-SCF 3 -2-Py], [BG1149: 4-CN-6-SCF 3 -2-Py], [BG1150: 6-CN-6-SCF 3 -2- Py], [BG1151: 3- OMe-6-SCF 3 -2-Py], [BG1152: 4-OMe-6-SCF 3 -2-Py], [BG1153: 6-OMe-6-SCF 3 -2 -Py], [BG1154: 3-S (O) Me-2-Py], [BG 1 155: 4-Cl-3-S (O) Me-2-Py], [BG 1156: 5-Cl-3-S (O) Me-2-Py], [BG 1157: 6-Cl-3-S (O) Me-2-Py], [BG 1158: 4-Me-3-S (O) Me-2-Py], [BG1159: 5-Me-3 -S (O) Me-2-Py], [BG1160: 6-Me-3-S (O) Me-2-Py], [BG1161: 4-CF 3 -3- S (O) Me-2- Py], [BG1162: 5-CF 3 -3-S (O) Me-2-Py], [BG1163: 6-CF 3 -3-S (O) Me-2- Py], [BG1164: 4-CN-3-S (O) Me-2-Py], [BG1165: 5-CN-3-S (O) Me-2-Py], [BG1166: 6-CN- 3-S (O) Me-2-Py], [BG1167: 4-OMe-3-S (O) Me-2-Py], [BG1168: 5-OMe-3-S (O) Me-2-] Py], [BG1169: 6-OMe-3-S (O) Me-2-Py], [BG1170: 4-S (O) Me-2-Py], [BG1171: 3-Cl-4 -S (O) Me-2-Py], [BG1172: 5-Cl-4-S (O) Me-2-Py], [BG1173: 6-Cl-4-S (O) Me-2-Py ], [BG1174: 3-Me-4-S (O) Me-2-Py], [BG1175: 5-Me-4-S (O) Me-2-Py], [BG1176: 6-Me-4] -S (O) Me-2- Py], [BG1177: 3-CF 3 -4-S (O) Me-2-Py], [BG1178: 5-CF 3 -4-S (O) Me-2 -Py], [BG1179: 6- CF 3 -4-S (O) Me-2-Py], [BG1180: 3-CN-4-S (O) Me-2-Py], [BG1181: 5- CN-4-S (O) Me-2-Py], [BG1182: 6-CN-4-S (O) Me-2-Py], [BG1183: 3-OMe-4-S (O) Me- 2-Py], [BG1184: 5-OMe-4-S (O) Me-2-Py], [BG1185: 6-OMe-4-S (O) Me-2-Py], [BG1186: 5-] S (O) Me-2-Py], [BG1187: 3-Cl-5-S (O) Me-2-Py], [BG1188: 4-Cl-5-S (O) Me-2-Py] , [BG1189: 6-Cl-5-S (O) Me-2-Py], [BG1190: 3-Me-5-S (O) Me-2-Py], [BG1191: 4-Me-5-5] S (O) Me-2- Py], [BG1192: 6-Me-5-S (O) Me-2-Py], [BG1193: 3-CF 3 -5-S (O) Me-2-Py ], [BG 1194: 4-CF ₃ -5-S (O) Me-2-Py], [BG 1195: 6-CF ₃ -5- S (O) Me-2-Py], [BG 1 196: 3-CN] -5-S (O) Me-2-Py], [BG 1197: 4-CN-5-S (O) Me-2-Py], [BG1198: 6-CN-5-S (O) Me-2 -Py], [BG1199: 3-OMe-5-S (O) Me-2-Py], [BG1200: 4-OMe-5-S (O) Me-2-Py],

[BG1201: 6-OMe-5-S (O) Me-2-Py], [BG1202: 6-S (O) Me-2-Py], [BG1203: 3-Cl-6-S (O) Me -2-Py !, [BG 1204: 4-Cl-6-S (O) Me-2-Py], [BG 1205: 5-Cl-6-S (O) Me-2-Py], [BG 1206: 3] -Me-6-S (O) Me-2-Py], [BG1207: 4-Me-6-S (O) Me-2-Py], [BG1208: 5-Me-6-S (O) Me -2-Py], [BG1209: 3-CF 3 -6-S (O) Me-2-Py], [BG1210: 4-CF 3 -6-S (O) Me-2-Py], [BG1211 _{: 5-CF 3 -6-S} (O) Me-2-Py], [BG1212: 3-CN-6-S (O) Me-2-Py], [BG1213: 4-CN-6-S ( O) Me-2-Py], [BG1214: 5-CN-6-S (O) Me-2-Py], [BG1215: 3-OMe-6-S (O) Me-2-Py], [BG12 15 BG1216: 4-OMe-6- S (O) Me-2-Py], [BG1217: 5-OMe-6-S (O) Me-2-Py], [BG1218: 3-S (O) CF 3 -2-Py], [BG1219: 4-Cl-3-S (O) CF 3 -2-Py], [BG1220: 5-Cl-3-S (O) CF 3 -2-Py], [BG1221 : 6-Cl-3-S (O) CF 3 -2-Py], [BG1222: 4-Me-3-S (O) CF 3 -2-Py], [BG1223: 5-Me-3-S _{(O) CF 3 -2-Py} ], [BG1224: 6-Me-3-S (O) CF 3 -2-Py], [BG1225: 4-CF 3 -3-S (O) CF 3 -2 -Py], [BG1226: 5- CF 3 -3-S (O) CF 3 -2-Py], [BG1227: 6-CF 3 -3-S (O) CF 3 -2-Py], [BG1228 : 4-CN-3-S (O) CF 3 -2-Py], [BG1229: 5-CN-3-S (O) CF 3 -2-Py], [BG1230: 6-CN-3-S _{(O) CF 3 -2-Py} ], [BG1231: 4-OMe-3-S (O) CF 3 -2-Py], [BG1232: 5-OMe-3-S (O) CF 3 -2- Py], [BG1233: 6- OMe-3-S (O) CF 3 -2-Py], [BG1234: 4-S (O ) CF ₃ -2-Py, [BG 1235: 3-Cl-4-S (O) CF ₃ -2-Py], [BG 1236: 5-Cl-4-S (O) CF ₃ -2-Py] , [BG1237: 6-Cl- 4-S (O) CF 3 -2-Py], [BG1238: 3-Me-4-S (O) CF 3 -2-Py], [BG1239: 5-Me- _{4-S (O) CF 3} -2-Py], [BG1240: 6-Me-4-S (O) CF 3 -2-Py], [BG1241: 3-CF 3 -4-S (O) CF ₃ -2-Py, [BG1242: 5-CF ₃ -4-S (O) CF ₃ -2-Py], [BG 1243: 6-CF ₃ -4-S (O) CF ₃ -2-Py] , [BG1244: 3-CN- 4-S (O) CF 3 -2-Py], [BG1245: 5-CN-4-S (O) CF 3 -2-Py], [BG1246: 6-CN- _{4-S (O) CF 3} -2-Py], [BG1247: 3-OMe-4-S (O) CF 3 -2-Py], [BG1248: 5-OMe-4-S (O) CF 3 -2-Py], [BG1249: 6-OMe-4-S (O) CF 3 -2-Py], [BG1250: 5-S (O) CF 3 -2-Py], [BG1251: 3-Cl _{-5-S (O) CF 3} -2-Py], [BG1252: 4-Cl-5-S (O) CF 3 -2-Py], [BG1253: 6-Cl-5-S (O) CF ₃ -2-Py, [BG1254: 3-Me-5-S (O) CF ₃ -2-Py], [BG 1 255: 4-Me-5-S (O) CF ₃ -2-Py], BG1256: 6-Me-5- S (O) CF 3 -2-Py], [BG1257: 3-CF 3 -5-S (O) CF 3 -2-Py], [BG1258: 4-CF 3 - _{5-S (O) CF 3} -2-Py], [BG1259: 6-CF 3 -5-S (O) CF 3 -2-Py], [BG1260: 3-CN-5-S (O) CF ₃ -2-Py !, [BG 1261: 4-CN-5-S (O) CF ₃ -2-Py], [BG 1262: 6-CN-5-S (O) CF ₃ -2-Py], BG1263: 3-OMe-5- S (O) CF 3 -2-Py], [BG1264: 4-OMe-5-S (O) CF 3 -2-Py], [BG1265: 6-OMe-5- S (O) CF ₃ -2-Py], [BG1266 : 6-S (O) CF 3 -2-Py], [BG1267: 3-Cl-6-S (O) CF 3 -2-Py], [BG1268: 4-Cl-6-S (O) CF ₃ -2-Py !, [BG 1269: 5-Cl-6-S (O) CF ₃ -2-Py], [BG 1270: 3-Me-6-S (O) CF ₃ -2-Py], BG1271: 4-Me-6- S (O) CF 3 -2-Py], [BG1272: 5-Me-6-S (O) CF 3 -2-Py], [BG1273: 3-CF 3 -6 _{-S (O) CF 3 -2-} Py], [BG1274: 4-CF 3 -6-S (O) CF 3 -2-Py], [BG1275: 5-CF 3 -6-S (O) CF ₃ -2-Py !, [BG 1276: 3-CN-6-S (O) CF ₃ -2-Py], [BG 1277: 4-CN-6-S (O) CF ₃ -2-Py], BG1278: 5-CN-6- S (O) CF 3 -2-Py], [BG1279: 3-OMe-6-S (O) CF 3 -2-Py], [BG1280: 4-OMe-6- _{S (O) CF 3 -2-} Py], [BG1281: 5-OMe-6-S (O) CF 3 -2-Py], [BG1282: 3-S (O) 2 Me-2-Py], [BG1283: 4-Cl-3-S (O) 2Me-2-Py], [BG1284: 5-Cl-3-S (O) ₂ Me-2-Py], [BG1285: 6-Cl-3- S (O) ₂ Me-2-Py, [BG1286: 4-Me-3-S (O) ₂ Me-2-Py], [BG1287: 5-Me-3-S (O) ₂ Me-2 -Py], [BG1288: 6- Me-3-S (O) 2 Me-2-Py], [BG1289: 4-CF 3 -3-S (O) 2 Me-2-Py], [BG1290: _{5-CF 3 -3-S (} O) 2 Me-2-Py], [BG1291: 6-CF 3 -3-S (O) 2 Me-2-Py], [BG1292: 4-CN-3- _{S (O) 2 Me-2} -Py], [BG1293: 5-CN-3-S (O) 2 Me-2-Py], [BG1294: 6-CN-3-S (O) 2 Me-2 -Py], [BG1295: 4-OMe-3-S (O) ₂ Me-2-Py], [BG1296: 5-OMe-3-S (O) ₂ Me-2-Py], [BG1297: 6] -OMe-3-S (O) ₂ Me-2-Py], [BG 1298: 4-S (O) 2 Me-2-Py], [BG1299: 3-Cl-4-S (O) 2 Me-2-Py], [BG1300: 5-Cl-4-S (O) ₂ Me-2-Py],

[BG1301: 6-Cl-4 -S (O) 2 Me-2-Py], [BG1302: 3-Me-4-S (O) 2 Me-2-Py], [BG1303: 5-Me-4 _{-S (O) 2 Me-2} -Py], [BG1304: 6-Me-4-S (O) 2 Me-2-Py], [BG1305: 3-CF 3 -4-S (O) 2 Me -2-Py], [BG1306: 5-CF 3 -4-S (O) 2 Me-2-Py], [BG1307: 6-CF 3 -4-S (O) 2 Me-2-Py], [BG1308: 3-CN-4-S (O) ₂ Me-2-Py], [BG1309: 5-CN-4-S (O) ₂ Me-2-Py], [BG1310: 6-CN-4 _{-S (O) 2 Me-2} -Py], [BG1311: 3-OMe-4-S (O) 2 Me-2-Py], [BG1312: 5-OMe-4-S (O) 2 Me- 2-Py], [BG 1313: 6-OMe-4-S (O) ₂ Me-2-Py], [BG 1314: 5-S (O) ₂ Me-2-Py], [BG 1315: 3-Cl- _{5-S (O) 2 Me} -2-Py], [BG1316: 4-Cl-5-S (O) 2 Me-2-Py], [BG1317: 6-Cl-5-S (O) 2 Me -2-Py !, [BG1318: 3-Me-5-S (O) ₂ Me-2-Py], [BG1319: 4-Me-5-S (O) ₂ Me-2-Py], [BG1320] : 6-Me-5-S (O) 2 Me-2-Py], [BG1321: 3-CF 3 -5-S (O) 2 Me-2-Py], [BG1322: 4-CF 3 -5 _{-S (O) 2 Me-2} -Py], [BG1323: 6-CF 3 -5-S (O) 2 Me-2-Py], [BG1324: 3-CN-5-S (O) 2 Me -2-Py !, [BG 1325: 4-CN-5-S (O) ₂ Me-2-Py], [BG 1326: 6-CN-5-S (O) ₂ Me-2-Py], [BG 1327 : 3-OMe-5-S (O) ₂ Me-2-Py], [BG1328: 4-OMe-5-S (O) ₂ Me-2-Py], [BG 1329: 6-OMe-5-S (O) ₂ Me-2-Py, [BG1330: 6-S (O) ₂ Me-2-Py], [BG1331: 3-Cl-6-S (O) ₂ Me-2-Py], BG1332: 4-Cl-6-S (O) ₂ Me- 2-Py], [BG1333: 5-Cl-6-S (O) ₂ Me-2-Py], [BG1334: 3-Me-6-S (O) ₂ Me-2-Py], [BG1335: 4-Me-6-S ( O) 2 Me-2-Py], [BG1336: 5-Me-6-S (O) 2 Me-2-Py], [BG1337: 3-CF 3 -6-S (O) ₂ Me-2-Py, [BG 1338: 4-CF ₃ -6-S (O) ₂ Me-2-Py], [BG 1339: 5-CF ₃ -6-S (O) ₂ Me- 2-Py], [BG1340: 3-CN-6-S (O) ₂ Me-2-Py], [BG1341: 4-CN-6-S (O) ₂ Me-2-Py], [BG1342: 5-CN-6-S ( O) 2 Me-2-Py], [BG1343: 3-OMe-6-S (O) 2 Me-2-Py], [BG1344: 4-OMe-6-S ( O) ₂ Me-2-Py, [BG 1345: 5-OMe-6-S (O) ₂ Me-2-Py], [BG 1346: 3-S (O) ₂ CF ₃ -2-Py], BG1347: 4-Cl-3- S (O) 2 CF 3 -2-Py], [BG1348: 5-Cl-3-S (O) 2 CF 3 -2-Py], [BG1349: 6-Cl- _{3-S (O) 2 CF} 3 -2-Py], [BG1350: 4-Me-3-S (O) 2 CF 3 -2-Py], [BG1351: 5-Me-3-S (O) _{2 CF 3 -2-Py],} [BG1352: 6-Me-3-S (O) 2 CF 3 -2-Py], [BG1353: 4-CF 3 -3-S (O) 2 CF 3 -2 -Py], [BG1354: 5- CF 3 -3-S (O) 2 CF 3 -2-Py], [BG1355: 6-CF 3 -3-S (O) 2 CF 3 -2-Py], [BG1356: 4-CN-3 -S (O) 2 CF 3 -2-Py], [BG1357: 5-CN-3-S (O) 2 CF 3 -2-Py], [BG1358: 6-CN _{-3-S (O) 2 CF} 3 -2-Py], [BG1359: 4-OMe-3-S (O) 2 CF 3 -2-Py], [BG1360: 5-OMe-3-S (O _{) 2 CF 3 -2-Py]} , [BG1361: 6-OMe-3-S (O) 2 CF 3 -2-Py], [BG1362: 4-S (O) 2 CF 3 -2-Py] , [BG1363: 3-Cl- 4-S (O) 2 CF 3 -2-Py], [BG1364: 5-Cl-4-S (O) 2 CF 3 -2-Py], [BG1365: 6- Cl-4-S (O) 2 CF 3 -2-Py], [BG1366: 3-Me-4-S (O) 2 CF 3 -2-Py], [BG1367: 5-Me-4-S ( O) ₂ CF ₃ -2-Py, [BG 1368: 6-Me-4-S (O) ₂ CF ₃ -2-Py], [BG 1 369: 3-CF ₃ -4-S (O) ₂ CF ₃ -2-Py], [BG1370: 5-CF 3 -4-S (O) 2 CF 3 -2-Py], [BG1371: 6-CF 3 -4-S (O) 2 CF 3 -2-Py ], [BG1372: 3-CN -4-S (O) 2 CF 3 -2-Py], [BG1373: 5-CN-4-S (O) 2 CF 3 -2-Py], [BG1374: 6 -CN-4-S (O) 2 CF 3 -2-Py], [BG1375: 3-OMe-4-S (O) 2 CF 3 -2-Py], [BG1376: 5-OMe-4-S _{(O) 2 CF 3 -2-} Py], [BG1377: 6-OMe-4-S (O) 2 CF 3 -2-Py], [BG1378: 5-S (O) 2 CF 3 -2-Py ], [BG1379: 3-Cl -5-S (O) 2 CF 3 -2-Py], [BG1380: 4-Cl-5-S (O) 2 CF 3 -2-Py], [BG1381: 6 -Cl-5-S (O) 2 CF 3 -2-Py], [BG1382: 3-Me-5-S (O) 2 CF 3 -2-Py], [BG1383: 4-Me-5-S (O) ₂ CF ₃ -2-Py, [BG 1384: 6-Me-5-S (O) ₂ CF ₃ -2-Py], [BG 1 385: 3-CF ₃ -5-S (O) ₂ CF ₃ -2-Py, [BG 1 386: 4-CF ₃ -5-S (O) ₂ CF ₃ -2-Py], [BG 1387: 6-CF ₃ -5-S (O) ₂ CF ₃ -2- Py], [BG1388: 3- CN-5-S (O) 2 CF 3 -2-Py], [BG1389: 4-CN-5-S (O) 2 CF 3 -2-Py], [BG1390: 6-CN-5-S ( O) 2 CF 3 -2-Py], [BG1391: 3-OMe-5-S (O) 2 CF 3 -2- Py], [BG1392: 4- OMe-5-S (O) 2 CF 3 -2-Py], [BG1393: 6-OMe-5-S (O) 2 CF 3 -2-Py], [BG1394: _{6-S (O) 2 CF} 3 -2-Py], [BG1395: 3-Cl-6-S (O) 2 CF 3 -2-Py], [BG1396: 4-Cl-6-S (O) ₂ CF ₃ -2-Py, [BG 1397: 5-Cl-6-S (O) ₂ CF ₃ -2-Py], [BG 1398: 3-Me-6-S (O) ₂ CF ₃ -2- Py], [BG1399: 4- Me-6-S (O) 2 CF 3 -2-Py], [BG1400: 5-Me-6-S (O) 2 CF 3 -2-Py],

_{[BG1401: 3-CF 3 -6} -S (O) 2 CF 3 -2-Py], [BG1402: 4-CF 3 -6-S (O) 2 CF 3 -2-Py], [BG1403: 5 _{-CF 3 -6-S (O)} 2 CF 3 -2-Py], [BG1404: 3-CN-6-S (O) 2 CF 3 -2-Py], [BG1405: 4-CN-6- _{S (O) 2 CF 3 -2} -Py], [BG1406: 5-CN-6-S (O) 2 CF 3 -2-Py], [BG1407: 3-OMe-6-S (O) 2 CF ₃ -2-Py, [BG 1408: 4-OMe-6-S (O) ₂ CF ₃ -2-Py], [BG 1409: 5-OMe-6-S (O) ₂ CF ₃ -2-Py] , [BG1410: 3-CN-2-Py], [BG 1411: 4-Cl-3-CN-2-Py], [BG 1412: 5-Cl-3-CN-2-Py], [BG 1413: 6- Cl-3-CN-2-Py !, [BG 1414: 4-Me-3-CN-2-Py], [BG 1415: 5-Me-3-CN-2-Py], [BG 1416: 6-Me- 3-CN-2-Py] , [BG1417: 4-CF 3 -3-CN-2-Py], [BG1418: 5-CF 3 -3-CN-2-Py], [BG1419: 6-CF 3 -3-CN-2-Py !, [BG1420: 4-CN-3-CN-2-Py], [BG1421: 5-CN-3-CN-2-Py], [BG1422: 6-CN-3] -CN-2-Py], [BG1423: 4-OMe-3-CN-2-Py], [BG1424: 5-OMe-3-CN-2-Py], [BG1425: 6-OMe-3-CN] -2-Py], [BG1426: 4-CN-2-Py], [BG1427: 3-Cl-4-CN-2-Py], [BG1428: 5-Cl-4-CN-2-Py], [BG1429: 6-Cl-4-CN-2-Py], [BG1430: 3-Me-4-CN-2-Py], [BG1431: 5-Me-4-CN-2-Py], [BG1432 : 6-Me-4-CN -2-Py], [BG1433: 3-CF 3 -4-CN-2-Py], [BG1434: 5-CF 3 -4-CN-2-Py], [BG1435 _{: 6-CF 3 -4-CN} -2-Py], [BG1436: 3-CN-4-CN-2-Py], [BG1437: 5-CN-4-CN-2-Py] , [BG1438: 6-CN-4-CN-2-Py], [BG1439: 3-OMe-4-CN-2-Py], [BG1440: 5-OMe-4-CN-2-Py], [BG1 940] BG1441: 6-OMe-4-CN-2-Py], [BG1442: 5-CN-2-Py], [BG1443: 3-Cl-5-CN-2-Py], [BG 1444: 4-Cl- 5-CN-2-Py, [BG1445: 6-Cl-5-CN-2-Py], [BG 1446: 3-Me-5-CN-2-Py], [BG1 447: 4-Me-5-] CN-2-Py], [ BG1448: 6-Me-5-CN-2-Py], [BG1449: 3-CF 3 -5-CN-2-Py], [BG1450: 4-CF 3 -5- CN-2-Py], [ BG1451: 6-CF 3 -5-CN-2-Py], [BG1452: 3-CN-5-CN-2-Py], [BG1453: 4-CN-5-CN -2-Py], [BG1454: 6-CN-5-CN-2-Py], [BG1455: 3-OMe-5-CN-2-Py], [BG1456: 4-OMe-5-CN-2] -Py], [BG1457: 6-OMe-5-CN-2-Py], [BG1458: 6-CN-2-Py], [BG1459: 3-Cl-6-CN-2-Py], [BG1460] : 4-Cl-6-CN-2-Py], [BG1461: 5-Cl-6-CN-2-Py], [BG1462: 3-Me-6-CN-2-Py], [BG1463: 4] -Me-6-CN-2- Py], [BG1464: 5-Me-6-CN-2-Py], [BG1465: 3-CF 3 -6-CN-2-Py], [BG1466: 4- _{CF 3 -6-CN-2-} Py], [BG1467: 5-CF 3 -6-CN-2-Py], [BG1468: 3-CN-6-CN-2-Py], [BG1469: 4- CN-6-CN-2-Py !, [BG1470: 5-CN-6-CN-2-Py], [BG1471: 3-OMe-6-CN-2-Py], [BG1472: 4-OMe- 6-CN-2-Py, [BG1473: 5-OMe-6-CN-2-Py], [BG1474: 3-COOMe-2-Py], [BG1475: 4-Cl-3-COOMe-2-] Py], [BG1476: 5-Cl-3-COOMe-2-Py], [BG1477: 6-Cl-3-COOMe-2-Py], [BG1478: 4-Me-3-] COOMe-2-Py], [ BG1479: 5-Me-3-COOMe-2-Py], [BG1480: 6-Me-3-COOMe-2-Py], [BG1481: 4-CF 3 -3-COOMe -2-Py], [BG1482: 5-CF 3 -3-COOMe-2-Py], [BG1483: 6-CF 3 -3-COOMe-2-Py], [BG1484: 4-CN-3-COOMe -2-Py !, [BG1485: 5-CN-3-COOMe-2-Py], [BG1486: 6-CN-3-COOMe-2-Py], [BG1487: 4-OMe-3-COOMe-2] -Py], [BG1488: 5-OMe-3-COOMe-2-Py], [BG1489: 6-OMe-3-COOMe-2-Py], [BG1490: 4-COOMe-2-Py], [BG1491] : 3-Cl-4-COOMe-2-Py], [BG1492: 5-Cl-4-COOMe-2-Py], [BG1493: 6-Cl-4-COOMe-2-Py], [BG1494: 3] -Me-4-COOMe-2-Py], [BG1495: 5-Me-4-COOMe-2-Py], [BG1496: 6-Me-4-COOMe-2-Py], [BG1497: 3-CF _{3 -4-COOMe-2-Py} ], [BG1498: 5-CF 3 -4-COOMe-2-Py], [BG1499: 6-CF 3 -4-COOMe-2-Py], [BG1500: 3- CN-4-COOMe-2-Py],

[BG1501: 5-CN-4-COOMe-2-Py], [BG1502: 6-CN-4-COOMe-2-Py], [BG1503: 3-OMe-4-COOMe-2-Py], [BG1504] : 5-OMe-4-COOMe-2-Py], [BG1505: 6-OMe-4-COOMe-2-Py], [BG1506: 5-COOMe-2-Py], [BG1507: 3-Cl-5] -COOMe-2-Py], [BG1508: 4-Cl-5-COOMe-2-Py], [BG1509: 6-Cl-5-COOMe-2-Py], [BG1510: 3-Me-5-COOMe -2-Py], [BG1511: 4-Me-5-COOMe-2-Py], [BG1512: 6-Me-5-COOMe-2-Py], [BG1513: 3-CF 3 -5-COOMe- 2-Py], [BG1514: 4-CF 3 -5-COOMe-2-Py], [BG1515: 6-CF 3 -5-COOMe-2-Py], [BG1516: 3-CN-5-COOMe- 2-Py], [BG1517: 4-CN-5-COOMe-2-Py], [BG1518: 6-CN-5-COOMe-2-Py], [BG1519: 3-OMe-5-COOMe-2-] Py], [BG1520: 4-OMe-5-COOMe-2-Py], [BG1521: 6-OMe-5-COOMe-2-Py], [BG1522: 6-COOMe-2-Py], [BG1523: 3-Cl-6-COOMe-2-Py], [BG1524: 4-Cl-6-COOMe-2-Py], [BG1525: 5-Cl-6-COOMe-2-Py], [BG1526: 3- Me-6-COOMe-2- Py], [BG1527: 4-Me-6-COOMe-2-Py], [BG1528: 5-Me-6-COOMe-2-Py], [BG1529: 3-CF 3 -6-COOMe-2-Py] , [BG1530: 4-CF 3 -6-COOMe-2-Py], [BG1531: 5-CF 3 -6-COOMe-2-Py], [BG1532: 3-CN -6-COOMe-2-Py !, [BG1533: 4-CN-6-COOMe-2-Py], [BG1534: 5-CN-6-COOMe-2-Py], [BG1535: 3-OMe-6] -COOMe-2-Py], [BG1536: 4-OMe-6-COOMe-2-Py], [BG1537: 5-OM] e-6-COOMe-2- Py], [BG1538: 3-NO 2 -2-Py], [BG1539: 4-Cl-3-NO 2 -2-Py], [BG1540: 5-Cl-3- _{NO 2 -2-Py], [} BG1541: 6-Cl-3-NO 2 -2-Py], [BG1542: 4-Me-3-NO 2 -2-Py], [BG1543: 5-Me-3 _{-NO 2 -2-Py], [} BG1544: 6-Me-3-NO 2 -2-Py], [BG1545: 4-CF 3 -3-NO 2 -2-Py], [BG1546: 5-CF _{3 -3-NO 2 -2-Py} ], [BG1547: 6-CF 3 -3-NO 2 -2-Py], [BG1548: 4-CN-3-NO 2 -2-Py], [BG1549: _{5-CN-3-NO 2} -2-Py], [BG1550: 6-CN-3-NO 2 -2-Py], [BG1551: 4-OMe-3-NO 2 -2-Py], [BG1552 : 5-OMe-3-NO 2 -2-Py], [BG1553: 6-OMe-3-NO 2 -2-Py], [BG1554: 4-NO 2 -2-Py], [BG1555: 3- _{Cl-4-NO 2 -2-} Py], [BG1556: 5-Cl-4-NO 2 -2-Py], [BG1557: 6-Cl-4-NO 2 -2-Py], [BG1558: 3 _{-Me-4-NO 2 -2-} Py], [BG1559: 5-Me-4-NO 2 -2-Py], [BG1560: 6-Me-4-NO 2 -2-Py], [BG1561: _{3-CF 3 -4-NO 2} -2-Py], [BG1562: 5-CF 3 -4-NO 2 -2-Py], [BG1563: 6-CF 3 -4-NO 2 -2-Py] , [BG1564: 3-CN- 4-NO 2 -2-Py], [BG1565: 5-CN-4-NO 2 -2-Py], [BG1566: 6-CN-4-NO 2 -2-Py ], [BG1567: 3-OMe -4-NO 2 -2-Py], [BG1568: 5-OMe-4-NO 2 -2-Py], [BG1569: 6-OMe-4-NO 2 -2- Py], [BG1570: 5- NO 2 -2-Py], [BG1571: 3-Cl-5-NO 2 -2-Py], [BG1572: 4-Cl-5-NO 2 -2-Py], [BG1573: 6-Cl-5 -NO 2 -2-Py], [BG 1574: 3-Me-5- NO 2 -2-Py], [BG1575: 4-Me-5-NO 2 -2-Py], [BG1576: 6-Me-5-NO 2 -2-Py], _{[BG1577: 3-CF 3 -5} -NO 2 -2-Py], [BG1578: 4-CF 3 -5-NO 2 -2-Py], [BG1579: 6-CF 3 -5-NO 2 -2 -Py], [BG1580: 3- CN-5-NO 2 -2-Py], [BG1581: 4-CN-5-NO 2 -2-Py], [BG1582: 6-CN-5-NO 2 - 2-Py], [BG1583: 3-OMe-5-NO 2 -2-Py], [BG1584: 4-OMe-5-NO 2 -2-Py], [BG1585: 6-OMe-5-NO 2 -2-Py], [BG1586: 6-NO 2 -2-Py], [BG1587: 3-Cl-6-NO 2 -2-Py], [BG1588: 4-Cl-6-NO 2 -2- Py], [BG1589: 5- Cl-6-NO 2 -2-Py], [BG1590: 3-Me-6-NO 2 -2-Py], [BG1591: 4-Me-6-NO 2 -2 -Py], [BG1592: 5- Me-6-NO 2 -2-Py], [BG1593: 3-CF 3 -6-NO 2 -2-Py], [BG1594: 4-CF 3 -6-NO ₂ -2-Py], [BG 1595: 5-CF ₃ -6-NO ₂ -2-Py], [BG 1596: 3-CN-6-NO ₂ -2-Py], [BG 1597: 4-CN-6] _{-NO 2 -2-Py], [} BG1598: 5-CN-6-NO 2 -2-Py], [BG1599: 3-OMe-6-NO 2 -2-Py], [BG1600: 4-OMe- 6-NO ₂ -2-Py],

[BG1601: 5-OMe-6 -NO 2 -2-Py], [BG1602: 3-NH 2 -2-Py], [BG1603: 4-Cl-3-NH 2 -2-Py], [BG1604: _{5-Cl-3-NH 2} -2-Py], [BG1605: 6-Cl-3-NH 2 -2-Py], [BG1606: 4-Me-3-NH 2 -2-Py], [BG1607 : 5-Me-3-NH 2 -2-Py], [BG1608: 6-Me-3-NH 2 -2-Py], [BG1609: 4-CF 3 -3-NH 2 -2-Py], _{[BG1610: 5-CF 3 -3} -NH 2 -2-Py], [BG1611: 6-CF 3 -3-NH 2 -2-Py], [BG1612: 4-CN-3-NH 2 -2- Py], [BG1613: 5- CN-3-NH 2 -2-Py], [BG1614: 6-CN-3-NH 2 -2-Py], [BG1615: 4-OMe-3-NH 2 -2 -Py], [BG1616: 5- OMe-3-NH 2 -2-Py], [BG1617: 6-OMe-3-NH 2 -2-Py], [BG1618: 4-NH 2 -2-Py] , [BG1619: 3-Cl- 4-NH 2 -2-Py], [BG1620: 5-Cl-4-NH 2 -2-Py], [BG1621: 6-Cl-4-NH 2 -2-Py ], [BG1622: 3-Me -4-NH 2 -2-Py], [BG1623: 5-Me-4-NH 2 -2-Py], [BG1624: 6-Me-4-NH 2 -2- Py], [BG1625: 3- CF 3 -4-NH 2 -2-Py], [BG1626: 5-CF 3 -4-NH 2 -2-Py], [BG1627: 6-CF 3 -4-NH ₂ -2-Py !, [BG1628: 3-CN-4-NH ₂ -2-Py], [BG 1629: 5-CN-4-NH ₂ -2-Py], [BG 1630: 6-CN -4- _{NH 2 -2-Py], [} BG1631: 3-OMe-4-NH 2 -2-Py], [BG1632: 5-OMe-4-NH 2 -2-Py], [BG1633: 6-OMe-4 _{-NH 2 -2-Py], [} BG1634: 5-NH 2 -2-Py], [BG1635: 3-Cl-5-NH 2 -2-Py], [BG1636: 4-Cl-5-NH 2 -2-Py], [BG1637: 6-Cl-5-NH ₂ -2-Py !, [BG1638: 3-Me-5-NH ₂ -2-Py], [BG1639: 4-Me-5-NH ₂ -2-Py], [BG1640: 6-Me-5-5] _{NH 2 -2-Py], [} BG1641: 3-CF 3 -5-NH 2 -2-Py], [BG1642: 4-CF 3 -5-NH 2 -2-Py], [BG1643: 6-CF _{3 -5-NH 2 -2-Py} ], [BG1644: 3-CN-5-NH 2 -2-Py], [BG1645: 4-CN-5-NH 2 -2-Py], [BG1646: 6 _{-CN-5-NH 2 -2-} Py], [BG1647: 3-OMe-5-NH 2 -2-Py], [BG1648: 4-OMe-5-NH 2 -2-Py], [BG1649: _{6-OMe-5-NH 2} -2-Py], [BG1650: 6-NH 2 -2-Py], [BG1651: 3-Cl-6-NH 2 -2-Py], [BG1652: 4-Cl -6-NH ₂ -2-Py !, [BG1653: 5-Cl-6-NH ₂ -2-Py], [BG 1654: 3-Me-6-NH ₂ -2-Py], [BG 1 655: 4-] _{Me-6-NH 2 -2-} Py], [BG1656: 5-Me-6-NH 2 -2-Py], [BG1657: 3-CF 3 -6-NH 2 -2-Py], [BG1658: _{4-CF 3 -6-NH 2} -2-Py], [BG1659: 5-CF 3 -6-NH 2 -2-Py], [BG1660: 3-CN-6-NH 2 -2-Py], [BG1661: 4-CN-6 -NH 2 -2-Py], [BG1662: 5-CN-6-NH 2 -2-Py], [BG1663: 3-OMe-6-NH 2 -2-Py] , [BG1664: 4-OMe- 6-NH 2 -2-Py], [BG1665: 5-OMe-6-NH 2 -2-Py], [BG1666: 3-NHMe-2-Py], [BG1667: 4-Cl-3-NHMe-2-Py, [BG1668: 5-Cl-3-NHMe-2-Py], [BG1669: 6-Cl-3-NHMe-2-Py], [BG1670: 4-] Me-3-NHMe-2- Py], [BG1671: 5-Me-3-NHMe-2-Py], [BG1672: 6-Me-3-NHMe-2-Py], [BG1673: 4-CF 3 -3-NHMe-2-Py], [BG1674: 5- _{CF 3 -3-NHMe-2-} Py], [BG1675: 6-CF 3 -3-NHMe-2-Py], [BG1676: 4-CN-3-NHMe-2-Py], [BG1677: 5- CN-3-NHMe-2-Py, [BG1678: 6-CN-3-NHMe-2-Py], [BG1679: 4-OMe-3-NHMe-2-Py], [BG1680: 5-OMe- 3-NHMe-2-Py, [BG1681: 6-OMe-3-NHMe-2-Py], [BG1682: 4-NHMe-2-Py], [BG1683: 3-Cl-4-NHMe-2-] Py], [BG1684: 5-Cl-4-NHMe-2-Py], [BG1685: 6-Cl-4-NHMe-2-Py], [BG1686: 3-Me-4-NHMe-2-Py] , [BG1687: 5-Me- 4-NHMe-2-Py], [BG1688: 6-Me-4-NHMe-2-Py], [BG1689: 3-CF 3 -4-NHMe-2-Py], _{[BG1690: 5-CF 3 -4} -NHMe-2-Py], [BG1691: 6-CF 3 -4-NHMe-2-Py], [BG1692: 3-CN-4-NHMe-2-Py], [BG1693: 5-CN-4-NHMe-2-Py], [BG1694: 6-CN-4-NHMe-2-Py], [BG1695: 3-OMe-4-NHMe-2-Py], [BG1696] : 5-OMe-4-NHMe-2-Py], [BG1697: 6-OMe-4-NHMe-2-Py], [BG1698: 5-NHMe-2-Py], [BG1699: 3-Cl-5 -NHMe-2-Py], [BG1700: 4-Cl-5-NHMe-2-Py],

[BG1701: 6-Cl-5-NHMe-2-Py], [BG1702: 3-Me-5-NHMe-2-Py], [BG1703: 4-Me-5-NHMe-2-Py], [BG1704] : 6-Me-5-NHMe -2-Py], [BG1705: 3-CF 3 -5-NHMe-2-Py], [BG1706: 4-CF 3 -5-NHMe-2-Py], [BG1707 _{: 6-CF 3 -5-NHMe} -2-Py], [BG1708: 3-CN-5-NHMe-2-Py], [BG1709: 4-CN-5-NHMe-2-Py], [BG1710: 6-CN-5-NHMe-2-Py], [BG1711: 3-OMe-5-NHMe-2-Py], [BG1712: 4-OMe-5-NHMe-2-Py], [BG1713: 6- OMe-5-NHMe-2-Py !, [BG1714: 6-NHMe-2-Py], [BG1715: 3-Cl-6-NHMe-2-Py], [BG1716: 4-Cl-6-NHMe- 2-Py], [BG1717: 5-Cl-6-NHMe-2-Py], [BG1718: 3-Me-6-NHMe-2-Py], [BG1719: 4-Me-6-NHMe-2-] Py], [BG1720: 5- Me-6-NHMe-2-Py], [BG1721: 3-CF 3 -6-NHMe-2-Py], [BG1722: 4-CF 3 -6-NHMe-2- Py], [BG1723: 5- CF 3 -6-NHMe-2-Py], [BG1724: 3-CN-6-NHMe-2-Py], [BG1725: 4-CN-6-NHMe-2-Py ], [BG1726: 5-CN-6-NHMe-2-Py], [BG1727: 3-OMe-6-NHMe-2-Py], [BG1728: 4-OMe-6-NHMe-2-Py], [BG1729: 5-OMe-6 -NHMe-2-Py], [BG1730: 3-NMe 2 -2-Py], [BG1731: 4-Cl-3-NMe 2 -2-Py], [BG1732: 5 _{-Cl-3-NMe 2 -2-} Py], [BG1733: 6-Cl-3-NMe 2 -2-Py], [BG1734: 4-Me-3-NMe 2 -2-Py], [BG1735: _{5-Me-3-NMe 2} -2-Py], [BG1736: 6-Me-3-NMe 2 -2-Py], [BG1737: 4-CF 3 -3-NMe 2 -2-Py], [ BG17 _{38: 5-CF 3 -3-} NMe 2 -2-Py], [BG1739: 6-CF 3 -3-NMe 2 -2-Py], [BG1740: 4-CN-3-NMe 2 -2-Py ], [BG1741: 5-CN -3-NMe 2 -2-Py], [BG1742: 6-CN-3-NMe 2 -2-Py], [BG1743: 4-OMe-3-NMe 2 -2- Py], [BG1744: 5- OMe-3-NMe 2 -2-Py], [BG1745: 6-OMe-3-NMe 2 -2-Py], [BG1746: 4-NMe 2 -2-Py], [BG1747: 3-Cl-4 -NMe 2 -2-Py], [BG1748: 5-Cl-4-NMe 2 -2-Py], [BG1749: 6-Cl-4-NMe 2 -2-Py] , [BG1750: 3-Me- 4-NMe 2 -2-Py], [BG1751: 5-Me-4-NMe 2 -2-Py], [BG1752: 6-Me-4-NMe 2 -2-Py ], [BG1753: 3-CF 3 -4-NMe 2 -2-Py], [BG1754: 5-CF 3 -4-NMe 2 -2-Py], [BG1755: 6-CF 3 -4-NMe 2 -2-Py !, [BG 1756: 3-CN-4-NMe ₂ -2-Py], [BG 1757: 5-CN-4-NMe ₂ 2-Py], [BG 1758: 6-CN-4-NMe _{2 -2-Py], [BG1759} : 3-OMe-4-NMe 2 -2-Py], [BG1760: 5-OMe-4-NMe 2 -2-Py], [BG1761: 6-OMe-4- _{NMe 2 -2-Py], [} BG1762: 5-NMe 2 -2-Py], [BG1763: 3-Cl-5-NMe 2 -2-Py], [BG1764: 4-Cl-5-NMe 2 - 2-Py], [BG1765: 6-Cl-5-NMe 2 -2-Py], [BG1766: 3-Me-5-NMe 2 -2-Py], [BG1767: 4-Me-5-NMe 2 -2-Py], [BG1768: 6-Me-5-NMe 2 -2-Py], [BG1769: 3-CF 3 -5-NMe 2 -2-Py], [BG1770: 4-CF 3 -5 _{-NMe 2 -2-Py], [} BG1771: 6-CF 3 -5-NMe 2 -2-Py], [BG1772: 3-CN-5-NMe 2 -2-Py], [BG17 73: 4-CN-5- NMe 2 -2-Py], [BG1774: 6-CN-5-NMe 2 -2-Py], [BG1775: 3-OMe-5-NMe 2 -2-Py], [BG1776: 4-OMe-5 -NMe 2 -2-Py], [BG1777: 6-OMe-5-NMe 2 -2-Py], [BG1778: 6-NMe 2 -2-Py], [BG1779: _{3-Cl-6-NMe 2} -2-Py], [BG1780: 4-Cl-6-NMe 2 -2-Py], [BG1781: 5-Cl-6-NMe 2 -2-Py], [BG1782 : 3-Me-6-NMe 2 -2-Py], [BG1783: 4-Me-6-NMe2-2-Py], [BG1784: 5-Me-6-NMe 2 -2-Py], [BG1785 _{: 3-CF 3 -6-NMe} 2 -2-Py], [BG1786: 4-CF 3 -6-NMe 2 -2-Py], [BG1787: 5-CF 3 -6-NMe 2 -2-Py ], [BG 1 788: 3-CN-6-NMe ₂ 2-Py], [BG 1 789: 4-CN-6-NMe ₂ 2-Py], [BG 1 790: 5-CN-6-NMe ₂ -2-] Py], [BG1791: 3- OMe-6-NMe 2 -2-Py], [BG1792: 4-OMe-6-NMe 2 -2-Py], [BG1793: 5-OMe-6-NMe 2 -2 -Py], [BG1794: 3-ACNH-2-Py], [BG1795: 4-Cl-3-ACNH-2-Py], [BG 1796: 5-Cl-3-ACNH-2-Py], [BG1797] : 6-Cl-3-ACNH-2-Py !, [BG1798: 4-Me-3-ACNH-2-Py], [BG1799: 5-Me-3-ACNH-2-Py], [BG1800: 6] -Me-3-ACNH-2-Py],

_{[BG1801: 4-CF 3 -3} -ACNH-2-Py], [BG1802: 5-CF 3 -3-ACNH-2-Py], [BG1803: 6-CF 3 -3-ACNH-2-Py] , [BG1804: 4-CN-3-ACNH-2-Py], [BG1805: 5-CN-3-ACNH-2-Py], [BG1806: 6-CN-3-ACNH-2-Py], [BG1 BG1807: 4-OMe-3-ACNH-2-Py !, [BG1808: 5-OMe-3-ACNH-2-Py], [BG1809: 6-OMe-3-ACNH-2-Py], [BG1810: 4-ACNH-2-Py, [BG 1811: 3-Cl-4-ACNH-2-Py], [BG 1812: 5-Cl-4-ACNH-2-Py], [BG 1813: 6-Cl-4- ACNH-2-Py, [BG1814: 3-Me-4-ACNH-2-Py], [BG1815: 5-Me-4-ACNH-2-Py], [BG1816: 6-Me-4-ACNH- 2-Py], [BG1817: 3-CF 3 -4-ACNH-2-Py], [BG1818: 5-CF 3 -4-ACNH-2-Py], [BG1819: 6-CF 3 -4-ACNH -2-Py !, [BG1820: 3-CN-4-ACNH-2-Py], [BG1821: 5-CN-4-ACNH-2-Py], [BG1822: 6-CN-4-ACNH-2] -Py], [BG1823: 3-OMe-4-ACNH-2-Py], [BG1824: 5-OMe-4-ACNH-2-Py], [BG1825: 6-OMe-4-ACNH-2-Py] ], [BG 1826: 5-ACNH-2-Py], [BG 1827: 3-Cl-5-ACNH-2-Py], [BG 1 828: 4-Cl-5-ACNH-2-Py], [BG 1829: 6] -Cl-5-ACNH-2-Py], [BG1830: 3-Me-5-ACNH-2-Py], [BG1831: 4-Me-5-ACNH-2-Py], [BG1832: 6-Me -5-ACNH-2-Py] , [BG1833: 3-CF 3 -5-ACNH-2-Py], [BG1834: 4-CF 3 -5-ACNH-2-Py], [BG1835: 6-CF _{3 -5-ACNH-2-Py} ], [BG1836: 3-CN-5-ACNH-2-Py], [BG1837: 4-CN-5-ACNH-2-Py], [BG1838: 6-CN- Five- ACNH-2-Py], [BG1839: 3-OMe-5-ACNH-2-Py], [BG1840: 4-OMe-5-ACNH-2-Py], [BG1841: 6-OMe-5-ACNH- 2-Py], [BG1842: 6-ACNH-2-Py], [BG1843: 3-Cl-6-ACNH-2-Py], [BG1844: 4-Cl-6-ACNH-2-Py], [BG BG1845: 5-Cl-6-ACNH-2-Py !, [BG1846: 3-Me-6-ACNH-2-Py], [BG1847: 4-Me-6-ACNH-2-Py], [BG1848: 5-Me-6-ACNH- 2-Py], [BG1849: 3-CF 3 -6-ACNH-2-Py], [BG1850: 4-CF 3 -6-ACNH-2-Py], [BG1851: _{5-CF 3 -6-ACNH-} 2-Py], [BG1852: 3-CN-6-ACNH-2-Py], [BG1853: 4-CN-6-ACNH-2-Py], [BG1854: 5 -CN-6-ACNH-2-Py], [BG1855: 3-OMe-6-ACNH-2-Py], [BG1856: 4-OMe-6-ACNH-2-Py], [BG1857: 5-OMe] -6-ACNH-2-Py], [BG1858: 3- (N (Ac) (Me))-2-Py], [BG1859: 4-Cl-3- (N (Ac) (Me))-2 -Py], [BG1860: 5-Cl-3- (N (Ac) (Me))-2-Py], [BG1861: 6-Cl-3- (N (Ac) (Me))-2-Py ], [BG1862: 4-Me-3- (N (Ac) (Me))-2-Py], [BG1863: 5-Me-3- (N (Ac) (Me))-2-Py], [BG1864: 6-Me-3- (N (Ac) (Me)) - 2-Py], [BG1865: 4-CF 3 -3- (N (Ac) (Me)) - 2-Py], [ _{BG1866: 5-CF 3 -3- (} N (Ac) (Me)) - 2-Py], [BG1867: 6-CF 3 -3- (N (Ac) (Me)) - 2-Py], [ BG1868: 4-CN-3- (N (Ac) (Me))-2-Py], [BG1869: 5-CN-3- (N (Ac) (Me))-2-Py], [BG1870: 6-CN-3- (N (Ac) (Me))-2-Py], [BG1871: 4-OMe-3- (N (Ac) (Me))-2-Py], [BG1872: 5- OMe-3- (N (Ac) (Me))-2-Py], [BG1873: 6-OMe-3- (N (Ac) (Me))-2-Py], [BG1874: 4- (N (Ac) (Me)] )-[2-Py], [BG1875: 3-Cl-4- (N (Ac) (Me))-2-Py], [BG1876: 5-Cl-4- (N (Ac) (Me))- 2-Py], [BG1877: 6-Cl-4- (N (Ac) (Me))-2-Py], [BG1878: 3-Me-4- (N (Ac) (Me))-2-] Py], [BG1879: 5-Me-4- (N (Ac) (Me))-2-Py], [BG1880: 6-Me-4- (N (Ac) (Me))-2-Py] _{, [BG1881: 3-CF 3} -4- (N (Ac) (Me)) - 2-Py], [BG1882: 5-CF 3 -4- (N (Ac) (Me)) - 2-Py] _{, [BG1883: 6-CF 3} -4- (N (Ac) (Me)) - 2-Py], [BG1884: 3-CN-4- (N (Ac) (Me)) - 2-Py], [BG 1885: 5-CN-4- (N (Ac) (Me))-2-Py], [BG 1886: 6-CN-4- (N (Ac) (Me))-2-Py], [BG 1887 : 3-OMe-4- (N (Ac) (Me))-2-Py], [BG1888: 5-OMe-4- (N (Ac) (Me))-2-Py], [BG1889: 6] -OMe-4- (N (Ac) (Me))-2-Py], [BG1890: 5- (N (Ac) (Me))-2-Py], [BG1891: 3-Cl-5- ( N (Ac) (Me))-2-Py], [BG1892: 4-Cl-5- (N (Ac) (Me))-2-Py], [BG1893: 6-Cl-5- (N ( Ac) (Me))-2-Py], [BG 1894: 3-Me-5- (N (Ac) (Me))-2-Py], [BG 1895: 4-Me-5- (N (Ac)) (Me)) - 2-Py ], [BG1896: 6-Me-5- (N (Ac) (Me)) - 2-Py], [BG1897: 3-CF 3 -5- (N (Ac) ( Me)) - 2-Py] , [BG1898: 4-CF 3 -5- (N (Ac) (Me)) - 2-Py], [BG1899: 6-CF 3 -5- (N (Ac) ( Me))-2-Py], [BG 1900: 3-CN-5- (N (Ac) (Me))-2-Py],

[BG1901: 4-CN-5- (N (Ac) (Me))-2-Py], [BG1902: 6-CN-5- (N (Ac) (Me))-2-Py], [BG1903 : 3-OMe-5- (N (Ac) (Me))-2-Py], [BG1904: 4-OMe-5- (N (Ac) (Me))-2-Py], [BG1905: 6 -OMe-5- (N (Ac) (Me))-2-Py], [BG1906: 6- (N (Ac) (Me))-2-Py], [BG1907: 3-Cl-6- ( N (Ac) (Me))-2-Py], [BG1908: 4-Cl-6- (N (Ac) (Me))-2-Py], [BG1909: 5-Cl-6- (N ( Ac) (Me))-2-Py], [BG1910: 3-Me-6- (N (Ac) (Me))-2-Py], [BG1911: 4-Me-6- (N (Ac)) (Me)) - 2-Py ], [BG1912: 5-Me-6- (N (Ac) (Me)) - 2-Py], [BG1913: 3-CF 3 -6- (N (Ac) ( Me)) - 2-Py] , [BG1914: 4-CF 3 -6- (N (Ac) (Me)) - 2-Py], [BG1915: 5-CF 3 -6- (N (Ac) ( Me))-2-Py], [BG1916: 3-CN-6- (N (Ac) (Me))-2-Py], [BG1917: 4-CN-6- (N (Ac) (Me)) )-[2-Py], [BG1918: 5-CN-6- (N (Ac) (Me))-2-Py], [BG1919: 3-OMe-6- (N (Ac) (Me))- 2-Py], [BG1920: 4-OMe-6- (N (Ac) (Me))-2-Py], [BG1921: 5-OMe-6- (N (Ac) (Me))-2-] Py], [BG1922: 3-AC-2-Py], [BG1 923: 4-Cl-3-AC-2-Py], [BG1924: 5-Cl-3-AC-2-Py], [BG1925: 6-Cl-3-AC-2-Py, [BG1926: 4-Me-3-AC-2-Py], [BG1 927: 5-Me-3-AC-2-Py], [BG1 928: 6- Me-3-AC-2- Py], [BG1929: 4-CF 3 -3-AC-2-Py], [BG1930: 5-CF 3 -3-AC-2-Py], [BG1931: 6- CF ₃ -3-AC-2-Py !, [BG1932: 4-CN-3-AC-2-Py], [BG1933: 5-CN-3-AC-2-Py], [BG19] 34: 6-CN-3-AC-2-Py !, [BG1935: 4-OMe-3-AC-2-Py], [BG1936: 5-OMe-3-AC-2-Py], [BG1937: 6-OMe-3-AC-2-Py], [BG1938: 4-AC-2-Py], [BG1939: 3-Cl-4-AC-2-Py], [BG1940: 5-Cl-4- AC-2-Py !, [BG1941: 6-Cl-4-AC-2-Py], [BG1942: 3-Me-4-AC-2-Py], [BG1943: 5-Me-4-AC- 2-Py], [BG1944: 6-Me-4-AC-2-Py], [BG1945: 3-CF 3 -4-AC-2-Py], [BG1946: 5-CF 3 -4-AC- 2-Py], [BG1947: 6-CF 3 -4-AC-2-Py], [BG1948: 3-CN-4-AC-2-Py], [BG1949: 5-CN-4-AC-2 -Py], [BG1950: 6-CN-4-AC-2-Py], [BG1951: 3-OMe-4-AC-2-Py], [BG1952: 5-OMe-4-AC-2-Py] ], [BG1953: 6-OMe-4-AC-2-Py], [BG1954: 5-AC-2-Py], [BG1 955: 3-Cl-5-AC-2-Py], [BG1956: 4] -Cl-5-AC-2-Py], [BG 1957: 6-Cl-5-AC-2-Py], [BG 1958: 3-Me-5-AC-2-Py], [BG 1959: 4-Me -5-AC-2-Py] , [BG1960: 6-Me-5-AC-2-Py], [BG1961: 3-CF 3 -5-AC-2-Py], [BG1962: 4-CF 3 -5-AC-2-Py, [BG 1963: 6-CF ₃ -5-AC-2-Py], [BG 1964: 3-CN-5-AC-2-Py], [BG 1 965: 4-CN- 5-AC-2-Py, [BG1966: 6-CN-5-AC-2-Py], [BG 1967: 3-OMe-5-AC-2-Py], [BG1968: 4-OMe-5-] AC-2-Py], [BG1969: 6-OMe-5-AC-2-Py], [BG1970: 6-AC-2-Py], [BG1971: 3-Cl-6-AC-2-Py] [BG1972: 4-Cl-6-AC-2-Py], [BG1973: 5-Cl-6-AC-2-Py], [BG1974: 3-Me-6-AC-2-Py], BG1975: 4 -Me-6-AC-2-Py], [BG 1976: 5-Me-6-AC-2-Py], [BG 1977: 3-CF ₃ -6-AC-2-Py], [BG 1978: 4- _{CF 3 -6-AC-2-} Py], [BG1979: 5-CF 3 -6-AC-2-Py], [BG1980: 3-CN-6-AC-2-Py], [BG1981: 4- CN-6-AC-2-Py], [BG 1982: 5-CN-6-AC-2-Py], [BG 1983: 3-OMe-6-AC-2-Py], [BG 1984: 4-OMe- 6-AC-2-Py, [BG1985: 5-OMe-6-AC-2-Py], [BG1986: 3-Py], [BG1987: 2-F-3-Py], [BG1988: 4-] Cl-2-F-3-Py !, [BG1989: 5-Cl-2-F-3-Py], [BG1990: 6-Cl-2-F-3-Py], [BG1991: 4-Me- 2-F-3-Py] , [BG1992: 5-Me-2-F-3-Py], [BG1993: 6-Me-2-F-3-Py], [BG1994: 4-CF 3 -2 -F-3-Py], [ BG1995: 5-CF 3 -2-F-3-Py], [BG1996: 6-CF 3 -2-F-3-Py], [BG1997: 4-CN-2 -F-3-Py], [BG1998: 5-CN-2-F-3-Py], [BG1999: 6-CN-2-F-3-Py], [BG2000: 4-OMe-2-F] -3-Py],

[BG2001: 5-OMe-2-F-3-Py], [BG2002: 6-OMe-2-F-3-Py], [BG2003: 4-F-3-Py], [BG2004: 2-Cl] -4-F-3-Py], [BG2005: 5-Cl-4-F-3-Py], [BG2006: 6-Cl-4-F-3-Py], [BG2007: 2-Me-4] -F-3-Py], [BG2008: 5-Me-4-F-3-Py], [BG2009: 6-Me-4-F-3-Py], [BG2010: 2-CF ₃ -4] F-3-Py], [ BG2011: 5-CF 3 -4-F-3-Py], [BG2012: 6-CF 3 -4-F-3-Py], [BG2013: 2-CN-4- F-3-Py], [BG2014: 5-CN-4-F-3-Py], [BG2015: 6-CN-4-F-3-Py], [BG2016: 2-OMe-4-F- 3-Py], [BG2017: 5-OMe-4-F-3-Py], [BG2018: 6-OMe-4-F-3-Py], [BG2019: 5-F-3-Py], BG2020: 2-Cl-5-F-3-Py], [BG2021: 4-Cl-5-F-3-Py], [BG2022: 6-Cl-5-F-3-Py], [BG2023: 2-Me-5-F-3-Py], [BG2024: 4-Me-5-F-3-Py], [BG2025: 6-Me-5-F-3-Py], [BG 2026: 2-] _{CF 3 -5-F-3-} Py], [BG2027: 4-CF 3 -5-F-3-Py], [BG2028: 6-CF 3 -5-F-3-Py], [BG2029: 2 -CN-5-F-3-Py], [BG2030: 4-CN-5-F-3-Py], [BG2031: 6-CN-5-F-3-Py], [BG2032: 2-OMe] -5-F-3-Py !, [BG2033: 4-OMe-5-F-3-Py], [BG2034: 6-OMe-5-F-3-Py], [BG2035: 6-F-3] -Py], [BG2036: 2-Cl-6-F-3-Py], [BG2037: 4-Cl-6-F-3-Py], [BG2038: 5-Cl-6-F-3-Py] ], [BG 2039: 2-Me-6-F-3-Py], [BG 2040: 4-Me-6-F-3-Py], [BG 2041: 5-Me-6-F-3-Py], _{[BG2042: 2-CF 3 -6} -F-3-Py], [BG2043: 4-CF 3 -6-F- 3-Py], [BG2044: 5-CF 3 -6-F-3-Py], [BG2045: 2-CN-6-F-3-Py], [BG2046: 4-CN-6-F-3 -Py], [BG2047: 5-CN-6-F-3-Py], [BG2048: 2-OMe-6-F-3-Py], [BG2049: 4-OMe-6-F-3-Py] ], [BG2050: 5-OMe-6-F-3-Py], [BG2051: 2-Cl-3-Py], [BG2052: 4-Cl-2-Cl-3-Py], [BG2053: 5] -Cl-2-Cl-3-Py, [BG2054: 6-Cl-2-Cl-3-Py], [BG2055: 4-Me-2-Cl-3-Py], [BG 2056: 5-Me -2-Cl-3-Py] , [BG2057: 6-Me-2-Cl-3-Py], [BG2058: 4-CF 3 -2-Cl-3-Py], [BG2059: 5-CF 3 -2-Cl-3-Py] , [BG2060: 6-CF 3 -2-Cl-3-Py], [BG2061: 4-CN-2-Cl-3-Py], [BG2062: 5-CN- 2-Cl-3-Py, [BG2063: 6-CN-2-Cl-3-Py], [BG 2064: 4-OMe-2-Cl-3-Py], [BG 2065: 5-OMe-2-] Cl-3-Py, [BG 2066: 6-OMe-2-Cl-3-Py], [BG 2067: 4-Cl-3-Py], [BG 2068: 2-Cl-4-Cl-3-Py] , [BG2069: 5-Cl-4-Cl-3-Py], [BG2070: 6-Cl-4-Cl-3-Py], [BG2071: 2-Me-4-Cl-3-Py], [BG20 BG2072: 5-Me-4- Cl-3-Py], [BG2073: 6-Me-4-Cl-3-Py], [BG2074: 2-CF 3 -4-Cl-3-Py], [BG2075 : 5-CF ₃ -4-Cl-3-Py !, [BG 2076: 6-CF ₃ -4-Cl-3-Py], [BG 2077: 2-CN-4-Cl-3-Py], [BG 20 78] : 5-CN-4-Cl-3-Py], [BG2079: 6-CN-4-Cl-3-Py], [BG2080: 2-OMe-4-Cl-3-Py], [BG2081: 5] -OMe-4-Cl-3-Py], [BG2082: 6-OMe-4-Cl-3-Py], [BG2083: 5-Cl-3-Py], [BG2084: 4-Cl-5-Cl -3-Py], [B G2085: 5-Cl-5-Cl-3-Py], [BG 2086: 6-Cl-5-Cl-3-Py], [BG 2087: 4-Me-5-Cl-3-Py], [BG 2088: 5-Me-5-Cl- 3-Py], [BG2089: 6-Me-5-Cl-3-Py], [BG2090: 4-CF 3 -5-Cl-3-Py], [BG2091: 5 _{-CF 3 -5-Cl-3-} Py], [BG2092: 6-CF 3 -5-Cl-3-Py], [BG2093: 4-CN-5-Cl-3-Py], [BG2094: 3 -CN-5-Cl-3-Py], [BG2095: 6-CN-5-Cl-3-Py], [BG 2096: 4-OMe-5-Cl-3-Py], [BG 2097: 5-OMe -5-Cl-3-Py, [BG 2098: 6-OMe -5-Cl-3-Py], [BG 2099: 6-Cl-3-Py], [BG 2 100: 2-Cl-6-Cl-3 -Py],

[BG2101: 4-Cl-6-Cl-3-Py], [BG2102: 5-Cl-6-Cl-3-Py], [BG2103: 2-Me-6-Cl-3-Py], [BG2104] : 4-Me-6-Cl -3-Py], [BG2105: 5-Me-6-Cl-3-Py], [BG2106: 2-CF 3 -6-Cl-3-Py], [BG2107: _{4-CF 3 -6-Cl-} 3-Py], [BG2108: 5-CF 3 -6-Cl-3-Py], [BG2109: 2-CN-6-Cl-3-Py], [BG2110: 4-CN-6-Cl-3-Py !, [BG2111: 5-CN-6-Cl-3-Py], [BG2112: 2-OMe-6-Cl-3-Py], [BG2113: 4-] OMe-6-Cl-3-Py, [BG2114: 5-OMe-6-Cl-3-Py], [BG2115: 2-Br-3-Py], [BG2116: 4-Cl-2-Br- 3-Py], [BG2117: 5-Cl-2-Br-3-Py], [BG2118: 6-Cl-2-Br-3-Py], [BG2119: 4-Me-2-Br-3-] Py], [BG2120: 5- Me-2-Br-3-Py], [BG2121: 6-Me-2-Br-3-Py], [BG2122: 4-CF 3 -2-Br-3-Py ], [BG2123: 5-CF 3 -2-Br-3-Py], [BG2124: 6-CF 3 -2-Br-3-Py], [BG2125: 4-CN-2-Br-3-Py ], [BG2126: 5-CN-2-Br-3-Py], [BG2127: 6-CN-2-Br-3-Py], [BG2128: 4-OMe-2-Br-3-Py], [BG 2129: 5-OMe-2-Br-3-Py], [BG 2130: 6-OMe-2-Br-3-Py], [BG 2131: 4-Br-3-Py], [BG 2 132: 2-Cl -4-Br-3-Py !, [BG2133: 5-Cl-4-Br-3-Py], [BG2134: 6-Cl-4-Br-3-Py], [BG2 135: 2-Me-4] -Br-3-Py], [ BG2136: 5-Me-4-Br-3-Py], [BG2137: 6-Me-4-Br-3-Py], [BG2138: 2-CF 3 -4- Br-3-Py], [ BG2139: 5-CF 3 -4-Br-3-Py], [BG2140: 6-CF 3 -4-Br-3-Py], [BG2141: 2-CN-4- Br -3-Py !, [BG2142: 5-CN-4-Br-3-Py], [BG2143: 6-CN-4-Br-3-Py], [BG2144: 2-OMe-4-Br-3] -Py], [BG2145: 5-OMe-4-Br-3-Py], [BG2146: 6-OMe-4-Br-3-Py], [BG2147: 5-Br-3-Py], [BG2148] : [2-Cl-5-Br-3-Py], [BG 2149: 4-Cl-5-Br-3-Py], [BG 2150: 6-Cl-5-Br-3-Py], [BG 2 215: 2] -Me-5-Br-3-Py], [BG2152: 4-Me-5-Br-3-Py], [BG2153: 6-Me-5-Br-3-Py], [BG2154: 2-CF _{3 -5-Br-3-Py} ], [BG2155: 4-CF 3 -5-Br-3-Py], [BG2156: 6-CF 3 -5-Br-3-Py], [BG2157: 2- CN-5-Br-3-Py, [BG2158: 4-CN-5-Br-3-Py], [BG2159: 6-CN-5-Br-3-Py], [BG2160: 2-OMe- 5-Br-3-Py, [BG2161: 4-OMe-5-Br-3-Py], [BG2162: 6-OMe-5-Br-3-Py], [BG2163: 6-Br-3- Py], [BG2164: 2-Cl-6-Br-3-Py], [BG2165: 4-Cl-6-Br-3-Py], [BG2166: 5-Cl-6-Br-3-Py] , [BG2167: 2-Me-6-Br-3-Py], [BG2168: 4-Me-6-Br-3-Py], [BG2169: 5-Me-6-Br-3-Py], [BG2 169: _{BG2170: 2-CF 3 -6-} Br-3-Py], [BG2171: 4-CF 3 -6-Br-3-Py], [BG2172: 5-CF 3 -6-Br-3-Py], [BG2173: 2-CN-6-Br-3-Py], [BG2174: 4-CN-6-Br-3-Py], [BG2175: 5-CN-6-Br-3-Py], [BG2176] : 2-OMe-6-Br-3-Py], [BG2177: 4-OMe-6-Br-3-Py], [BG2178: 5-OMe-6-Br-3-Py], [BG2179: 2] -I-3-Py, [BG2 180: 4-Cl-2-I-3-Py], [BG2181: 5-Cl-2-I-3-Py], [BG2182: 6-Cl-2-I -3-Py], [ BG2183: 4-Me-2-I-3-Py, [BG2184: 5-Me-2-I-3-Py], [BG2185: 6-Me-2-I-3-Py], [BG2186: _{4-CF 3 -2-I-} 3-Py], [BG2187: 5-CF 3 -2-I-3-Py], [BG2188: 6-CF 3 -2-I-3-Py], [BG2189 : 4-CN-2-I-3-Py], [BG2190: 5-CN-2-I-3-Py], [BG2191: 6-CN-2-I-3-Py], [BG2192: 4] -OMe-2-I-3-Py], [BG2193: 5-OMe-2-I-3-Py], [BG2194: 6-OMe-2-I-3-Py], [BG2195: 4-I -3-Py], [BG2196: 2-Cl-4-I-3-Py], [BG2197: 5-Cl-4-I-3-Py], [BG2198: 6-Cl-4-I-3] -Py], [BG2199: 2-Me-4-I-3-Py], [BG2200: 5-Me-4-I-3-Py],

[BG2201: 6-Me-4 -I-3-Py], [BG2202: 2-CF 3 -4-I-3-Py], [BG2203: 5-CF 3 -4-I-3-Py], _{[BG2204: 6-CF 3 -4} -I-3-Py], [BG2205: 2-CN-4-I-3-Py], [BG2206: 5-CN-4-I-3-Py], [ BG2207: 6-CN-4-I-3-Py, [BG2208: 2-OMe-4-I-3-Py], [BG2209: 5-OMe-4-I-3-Py], [BG2210: 6-OMe-4-I-3-Py, [BG2211: 5-I-3-Py], [BG2212: 2-Cl-5-I-3-Py], [BG2213: 4-Cl-5- I-3-Py, [BG2214: 6-Cl-5-I-3-Py], [BG2215: 2-Me-5-I-3-Py], [BG2216: 4-Me-5-I- 3-Py], [BG2217: 6-Me-5-I-3-Py], [BG2218: 2-CF 3 -5-I-3-Py], [BG2219: 4-CF 3 -5-I- 3-Py], [BG2220: 6-CF 3 -5-I-3-Py], [BG2221: 2-CN-5-I-3-Py], [BG2222: 4-CN-5-I-3 -Py], [BG2223: 6-CN-5-I-3-Py], [BG2224: 2-OMe-5-I-3-Py], [BG2225: 4-OMe-5-I-3-Py] ], [BG2226: 6-OMe-5-I-3-Py], [BG2227: 6-I-3-Py], [BG2228: 2-Cl-6-I-3-Py], [BG2229: 4] -Cl-6-I-3-Py], [BG2 230: 5-Cl-6-I-3-Py], [BG2223: 2-Me-6-I-3-Py], [BG2 232: 4-Me -6-I-3-Py] , [BG2233: 5-Me-6-I-3-Py], [BG2234: 2-CF 3 -6-I-3-Py], [BG2235: 4-CF 3 -6-I-3-Py] , [BG2236: 5-CF 3 -6-I-3-Py], [BG2237: 2-CN-6-I-3-Py], [BG2238: 4-CN- 6-I-3-Py, [BG2239: 5-CN-6-I-3-Py], [BG2240: 2-OMe-6-I-3-Py], [BG2241: 4-OMe-6-] I-3-Py, [BG2242: 5-OMe-6-I-3-Py], [BG2243: 2-Me-3-Py !, [BG2244: 4-Cl-2-Me-3-Py], [BG2245: 5-Cl-2-Me-3-Py], [BG2246: 6-Cl-2-] Me-3-Py !, [BG2247: 4-Me-2-Me-3-Py], [BG 2248: 5-Me-2-Me-3-Py], [BG2249: 6-Me-2-Me- 3-Py], [BG2250: 4-CF 3 -2-Me-3-Py], [BG2251: 5-CF 3 -2-Me-3-Py], [BG2252: 6-CF 3 -2-Me -3-Py !, [BG2253: 4-CN-2-Me-3-Py], [BG2254: 5-CN-2-Me-3-Py], [BG2255: 6-CN-2-Me-3] -Py], [BG2256: 4-OMe-2-Me-3-Py], [BG2257: 5-OMe-2-Me-3-Py], [BG2258: 6-OMe-2-Me-3-Py] ], [BG2259: 4-Me-3-Py], [BG2260: 2-Cl-4-Me-3-Py], [BG2261: 5-Cl-4-Me-3-Py], [BG2262: 6] -Cl-4-Me-3-Py], [BG2263: 2-Me-4-Me-3-Py], [BG2264: 5-Me-4-Me-3-Py], [BG2265: 6-Me -4-Me-3-Py] , [BG2266: 2-CF 3 -4-Me-3-Py], [BG2267: 5-CF 3 -4-Me-3-Py], [BG2268: 6-CF ₃ -4-Me-3-Py !, [BG2269: 2-CN-4-Me-3-Py], [BG2270: 5-CN-4-Me-3-Py], [BG2271: 6-CN- 4-Me-3-Py, [BG2272: 2-OMe-4-Me-3-Py], [BG2273: 5-OMe-4-Me-3-Py], [BG2274: 6-OMe-4-4] Me-3-Py], [BG2275: 5-Me-3-Py], [BG2276: 2-Cl-5-Me-3-Py], [BG2277: 4-Cl-5-Me-3-Py] , [BG2278: 6-Cl-5-Me-3-Py], [BG2279: 2-Me-5-Me-3-Py], [BG2280: 4-Me-5-Me-3-Py], [BG2 2 10 BG2281: 6-Me-5- Me-3-Py], [BG2282: 2-CF 3 -5-Me-3-Py], [BG2283: 4-CF 3 -5-Me-3-Py], [ BG 2284: 6 _{-CF 3 -5-Me-3-} Py], [BG2285: 2-CN-5-Me-3-Py], [BG2286: 4-CN-5-Me-3-Py], [BG2287: 6- CN-5-Me-3-Py, [BG2288: 2-OMe-5-Me-3-Py], [BG2289: 4-OMe-5-Me-3-Py], [BG2290: 6-OMe- 5-Me-3-Py, [BG2291: 6-Me-3-Py], [BG2292: 2-Cl-6-Me-3-Py], [BG2293: 4-Cl-6-Me-3-3 Py], [BG2294: 5-Cl-6-Me-3-Py], [BG2295: 2-Me-6-Me-3-Py], [BG2296: 4-Me-6-Me-3-Py] , [BG2297: 5-Me- 6-Me-3-Py], [BG2298: 2-CF 3 -6-Me-3-Py], [BG2299: 4-CF 3 -6-Me-3-Py] [BG 2300: 5-CF ₃ -6-Me-3-Py],

[BG2301: 2-CN-6-Me-3-Py], [BG2302: 4-CN-6-Me-3-Py], [BG2303: 5-CN-6-Me-3-Py], [BG2304] : 2-OMe-6-Me-3-Py], [BG 2305: 4-OMe-6-Me-3-Py], [BG 2306: 5-OMe-6-Me-3-Py], [BG 2307: 2] -OMe-3-Py], [BG2308: 4-Cl-2-OMe-3-Py], [BG2309: 5-Cl-2-OMe-3-Py], [BG2310: 6-Cl-2-OMe] -3-Py !, [BG2311: 4-Me-2-OMe-3-Py], [BG2312: 5-Me-2-OMe-3-Py], [BG2313: 6-Me-2-OMe-3] -Py], [BG2314: 4- CF 3 -2-OMe-3-Py], [BG2315: 5-CF 3 -2-OMe-3-Py], [BG2316: 6-CF 3 -2-OMe- 3-Py], [BG2317: 4-CN-2-OMe-3-Py], [BG2318: 5-CN-2-OMe-3-Py], [BG2319: 6-CN-2-OMe-3-] Py], [BG2320: 4-OMe-2-OMe-3-Py], [BG2321: 5-OMe-2-OMe-3-Py], [BG2322: 6-OMe-2-OMe-3-Py] , [BG2323: 4-OMe-3-Py], [BG2324: 2-Cl-4-OMe-3-Py], [BG2325: 5-Cl-4-OMe-3-Py], [BG2236: 6- Cl-4-OMe-3-Py !, [BG2327: 2-Me-4-OMe-3-Py], [BG2328: 5-Me-4-OMe-3-Py], [BG2329: 6-Me- 4-OMe-3-Py] , [BG2330: 2-CF 3 -4-OMe-3-Py], [BG2331: 5-CF 3 -4-OMe-3-Py], [BG2332: 6-CF 3 -4-OMe-3-Py !, [BG2333: 2-CN-4-OMe-3-Py], [BG2334: 5-CN-4-OMe-3-Py], [BG2335: 6-CN-4] -OMe-3-Py], [BG2336: 2-OMe-4-OMe-3-Py], [BG2337: 5-OMe-4-OMe-3-Py], [BG2338: 6-OMe-4-OMe] -3-Py, [BG2339: 5-OMe-3-Py], [BG2340: 2-Cl-5-OMe- 3-Py], [BG2341: 4-Cl-5-OMe-3-Py], [BG2342: 6-Cl-5-OMe-3-Py], [BG2343: 2-Me-5-OMe-3-3] Py], [BG2344: 4- Me-5-OMe-3-Py], [BG2345: 6-Me-5-OMe-3-Py], [BG2346: 2-CF 3 -5-OMe-3-Py ], [BG2347: 4-CF 3 -5-OMe-3-Py], [BG2348: 6-CF 3 -5-OMe-3-Py], [BG2349: 2-CN-5-OMe-3-Py ], [BG2 350: 4-CN-5-OMe-3-Py], [BG2351: 6-CN-5-OMe-3-Py], [BG2352: 2-OMe-5-OMe-3-Py], [BG2353: 4-OMe-5-OMe-3-Py], [BG2354: 6-OMe-5-OMe-3-Py], [BG2355: 6-OMe-3-Py], [BG2356: 2-Cl] -6-OMe-3-Py !, [BG2357: 4-Cl-6-OMe-3-Py], [BG2358: 5-Cl-6-OMe-3-Py], [BG2359: 2-Me-6] -OMe-3-Py], [ BG2360: 4-Me-6-OMe-3-Py], [BG2361: 5-Me-6-OMe-3-Py], [BG2362: 2-CF 3 -6- OMe-3-Py], [ BG2363: 4-CF 3 -6-OMe-3-Py], [BG2364: 5-CF 3 -6-OMe-3-Py], [BG2365: 2-CN-6- OMe-3-Py, [BG2366: 4-CN-6-OMe-3-Py], [BG2367: 5-CN-6-OMe-3-Py], [BG2368: 2-OMe-6-OMe- 3-Py], [BG2369: 4-OMe-6-OMe-3-Py], [BG2370: 5-OMe-6-OMe-3-Py], [BG2371: 2-CF 3 -3-Py], [BG2372: 4-Cl-2 -CF 3 -3-Py], [BG2373: 5-Cl-2-CF 3 -3-Py], [BG2374: 6-Cl-2-CF 3 -3-Py] , [BG2375: 4-Me- 2-CF 3 -3-Py], [BG2376: 5-Me-2-CF 3 -3-Py], [BG2377: 6-Me-2-CF 3 -3-Py ], [BG 2378: 4-CF ₃ -2-CF ₃ -3-Py], [BG 2379: 5-C] _{F 3 -2-CF 3 -3-} Py], [BG2380: 6-CF 3 -2-CF 3 -3-Py], [BG2381: 4-CN-2-CF 3 -3-Py], [BG2382 : 5-CN-2-CF 3 -3-Py], [BG2383: 6-CN-2-CF 3 -3-Py], [BG2384: 4-OMe-2-CF 3 -3-Py], [ BG2385: 5-OMe-2- CF 3 -3-Py], [BG2386: 6-OMe-2-CF 3 -3-Py], [BG2387: 4-CF 3 -3-Py], [BG2388: 2 _{-Cl-4-CF 3 -3-} Py], [BG2389: 5-Cl-4-CF 3 -3-Py], [BG2390: 6-Cl-4-CF 3 -3-Py], [BG2391: _{2-Me-4-CF 3} -3-Py], [BG2392: 5-Me-4-CF 3 -3-Py], [BG2393: 6-Me-4-CF 3 -3-Py], [BG2394 : 2-CF ₃ -4-CF ₃ -3-Py], [BG 2395: 5-CF ₃ -4-CF ₃ -3-Py], [BG 2 396: 6-CF ₃ -4-CF ₃ -3-Py] ], [BG2397: 2-CN -4-CF 3 -3-Py], [BG2398: 5-CN-4-CF 3 -3-Py], [BG2399: 6-CN-4-CF 3 -3- Py], [BG2400: 2- OMe-4-CF 3 -3-Py],

[BG2401: 5-OMe-4 -CF 3 -3-Py], [BG2402: 6-OMe-4-CF 3 -3-Py], [BG2403: 5-CF 3 -3-Py], [BG2404: _{2-Cl-5-CF 3} -3-Py], [BG2405: 4-Cl-5-CF 3 -3-Py], [BG2406: 6-Cl-5-CF 3 -3-Py], [BG2407 : 2-Me-5-CF 3 -3-Py], [BG2408: 4-Me-5-CF 3 -3-Py], [BG2409: 6-Me-5-CF 3 -3-Py], [ BG 2410: 2-CF ₃ -5-CF ₃ -3-Py], [BG 2411: 4-CF ₃ -5-CF ₃ -3-Py], [BG 2412: 6-CF ₃ -5-CF ₃ -3- CF 3 Py], [BG2413: 2- CN-5-CF 3 -3-Py], [BG2414: 4-CN-5-CF 3 -3-Py], [BG2415: 6-CN-5-CF 3 -3 -Py], [BG2416: 2- OMe-5-CF 3 -3-Py], [BG2417: 4-OMe-5-CF 3 -3-Py], [BG2418: 6-OMe-5-CF 3 - 3-Py], [BG2419: 6-CF 3 -3-Py], [BG2420: 2-Cl-6-CF 3 -3-Py], [BG2421: 4-Cl-6-CF 3 -3-Py ], [BG2422: 5-Cl -6-CF 3 -3-Py], [BG2423: 2-Me-6-CF 3 -3-Py], [BG2424: 4-Me-6-CF 3 -3- Py], [BG2425: 5- Me-6-CF 3 -3-Py], [BG2426: 2-CF 3 -6-CF 3 -3-Py], [BG2427: 4-CF 3 -6-CF 3 -3-Py], [BG2428: 5-CF 3 -6-CF 3 -3-Py], [BG2429: 2-CN-6-CF 3 -3-Py], [BG2430: 4-CN-6- CF ₃ -3-Py !, [BG 2431: 5-CN-6-CF ₃ -3-Py], [BG 2432: 2-OMe-6-CF ₃ -3-Py], [BG 2433: 4-OMe-6] _{-CF 3 -3-Py], [} BG2434: 5-OMe-6-CF 3 -3-Py], [BG2435: 2-OCF 3 -3-Py], [BG2436: 4-Cl-2-OCF 3 -3-Py], [BG 2437: 5-Cl-2- _{OCF 3 -3-Py], [} BG2438: 6-Cl-2-OCF 3 -3-Py], [BG2439: 4-Me-2-OCF 3 -3-Py], [BG2440: 5-Me-2 _{-OCF 3 -3-Py], [} BG2441: 6-Me-2-OCF 3 -3-Py], [BG2442: 4-CF 3 -2-OCF 3 -3-Py], [BG2443: 5-CF _{3 -2-OCF 3 -3-Py} ], [BG2444: 6-CF 3 -2-OCF 3 -3-Py], [BG2445: 4-CN-2-OCF 3 -3-Py], [BG2446: _{5-CN-2-OCF 3} -3-Py], [BG2447: 6-CN-2-OCF 3 -3-Py], [BG2448: 4-OMe-2-OCF 3 -3-Py], [BG2449 : 5-OMe-2-OCF 3 -3-Py], [BG2450: 6-OMe-2-OCF 3 -3-Py], [BG2451: 4-OCF 3 -3-Py], [BG2452: 2- _{Cl-4-OCF 3 -3-} Py], [BG2453: 5-Cl-4-OCF 3 -3-Py], [BG2454: 6-Cl-4-OCF 3 -3-Py], [BG2455: 2 _{-Me-4-OCF 3 -3-} Py], [BG2456: 5-Me-4-OCF 3 -3-Py], [BG2457: 6-Me-4-OCF 3 -3-Py], [BG2458: _{2-CF 3 -4-OCF 3} -3-Py], [BG2459: 5-CF 3 -4-OCF 3 -3-Py], [BG2460: 6-CF 3 -4-OCF 3 -3-Py] , [BG2461: 2-CN- 4-OCF 3 -3-Py], [BG2462: 5-CN-4-OCF 3 -3-Py], [BG2463: 6-CN-4-OCF 3 -3-Py ], [BG2464: 2-OMe -4-OCF 3 -3-Py], [BG2465: 5-OMe-4-OCF 3 -3-Py], [BG2466: 6-OMe-4-OCF 3 -3- Py], [BG2467: 5- OCF 3 -3-Py], [BG2468: 2-Cl-5-OCF 3 -3-Py], [BG2469: 4-Cl-5-OCF 3 -3-Py], [BG2470: 6-Cl-5 -OCF 3 -3-Py], [BG2471: 2-Me-5-OCF 3 -3-Py], [BG2472: 4-Me-5-OCF 3 -3-Py], [BG2473: 6-Me-5-OCF 3 -3-Py], [BG2474: 2-CF 3 -5-OCF 3 -3-Py], [BG2475: 4-CF 3 -5 _{-OCF 3 -3-Py], [} BG2476: 6-CF 3 -5-OCF 3 -3-Py], [BG2477: 2-CN-5-OCF 3 -3-Py], [BG2478: 4-CN _{-5-OCF 3 -3-Py]} , [BG2479: 6-CN-5-OCF 3 -3-Py], [BG2480: 2-OMe-5-OCF 3 -3-Py], [BG2481: 4- _{OMe-5-OCF 3 -3-} Py], [BG2482: 6-OMe-5-OCF 3 -3-Py], [BG2483: 6-OCF 3 -3-Py], [BG2484: 2-Cl-6 _{-OCF 3 -3-Py], [} BG2485: 4-Cl-6-OCF 3 -3-Py], [BG2486: 5-Cl-6-OCF 3 -3-Py], [BG2487: 2-Me- _{6-OCF 3 -3-Py]} , [BG2488: 4-Me-6-OCF 3 -3-Py], [BG2489: 5-Me-6-OCF 3 -3-Py], [BG2490: 2-CF ₃ -6-OCF ₃ -3-Py, [BG2491: 4-CF ₃ -6-OCF ₃ -3-Py], [BG2492: 5-CF ₃ -6-OCF ₃ -3-Py], [BG2493] : 2-CN-6-OCF 3 -3-Py], [BG2494: 4-CN-6-OCF 3 -3-Py], [BG2495: 5-CN-6-OCF 3 -3-Py], [ BG2496: 2-OMe-6- OCF 3 -3-Py], [BG2497: 4-OMe-6-OCF 3 -3-Py], [BG2498: 5-OMe-6-OCF 3 -3-Py], _{[BG2499: 2-CHF 2 -3} -Py], [BG2500: 4-Cl-2-CHF 2 -3-Py],

[BG2501: 5-Cl-2 -CHF 2 -3-Py], [BG2502: 6-Cl-2-CHF 2 -3-Py], [BG2503: 4-Me-2-CHF 2 -3-Py] , [BG2504: 5-Me- 2-CHF 2 -3-Py], [BG2505: 6-Me-2-CHF 2 -3-Py], [BG2506: 4-CF 3 -2-CHF 2 -3- Py], [BG2507: 5- CF 3 -2-CHF 2 -3-Py], [BG2508: 6-CF 3 -2-CHF 2 -3-Py], [BG2509: 4-CN-2-CHF 2 -3-Py], [BG2510: 5-CN-2-CHF 2 -3-Py], [BG2511: 6-CN-2-CHF 2 -3-Py], [BG2512: 4-OMe-2-CHF _{2 -3-Py], [BG2513} : 5-OMe-2-CHF 2 -3-Py], [BG2514: 6-OMe-2-CHF 2 -3-Py], [BG2515: 4-CHF 2 -3 -Py], [BG2516: 2- Cl-4-CHF 2 -3-Py], [BG2517: 5-Cl-4-CHF 2 -3-Py], [BG2518: 6-Cl-4-CHF 2 - 3-Py], [BG2519: 2-Me-4-CHF 2 -3-Py], [BG2520: 5-Me-4-CHF 2 -3-Py], [BG2521: 6-Me-4-CHF 2 -3-Py], [BG2522: 2-CF 3 -4-CHF 2 -3-Py], [BG2523: 5-CF 3 -4-CHF 2 -3-Py], [BG2524: 6-CF 3 - _{4-CHF 2 -3-Py]} , [BG2525: 2-CN-4-CHF 2 -3-Py], [BG2526: 5-CN-4-CHF 2 -3-Py], [BG2527: 6-CN -4-CHF ₂ -3-Py, [BG 2528: 2-OMe 4-CHF ₂ -3-Py], [BG 2529: 5-OMe 4-CHF ₂ -3-Py], [BG 2530: 6- _{OMe-4-CHF 2 -3-} Py], [BG2531: 5-CHF 2 -3-Py], [BG2532: 2-Cl-5-CHF 2 -3-Py], [BG2533: 4-Cl-5 _{-CHF 2 -3-Py], [} BG2534: 6-Cl-5-CHF 2 -3-Py], [BG2535: 2-Me-5-CHF 2 -3-Py], [BG253 6: 4-Me-5- CHF 2 -3-Py], [BG2537: 6-Me-5-CHF 2 -3-Py], [BG2538: 2-CF 3 -5-CHF 2 -3-Py] [BG 2539: 4-CF ₃ -5-CHF ₂ -3-Py], [BG 2540: 6-CF ₃ -5-CHF ₂ -3-Py], [BG 2 54 1: 2 CN 5 CHF _2-3 -Py], [BG2542: 4- CN-5-CHF 2 -3-Py], [BG2543: 6-CN-5-CHF 2 -3-Py], [BG2544: 2-OMe-5-CHF 2 - 3-Py], [BG2545: 4-OMe-5-CHF 2 -3-Py], [BG2546: 6-OMe-5-CHF 2 -3-Py], [BG2547: 6-CHF 2 -3-Py ], [BG2548: 2-Cl -6-CHF 2 -3-Py], [BG2549: 4-Cl-6-CHF 2 -3-Py], [BG2550: 5-Cl-6-CHF 2 -3- Py], [BG2551: 2- Me-6-CHF 2 -3-Py], [BG2552: 4-Me-6-CHF 2 -3-Py], [BG2553: 5-Me-6-CHF 2 -3 -Py], [BG 2554: 2-CF ₃ -6-CHF ₂ -3-Py], [BG ₂ 555: 4-CF ₃ -6-CHF ₂ -3-Py], [BG ₂ 556: 5-CF ₃ -6-] _{CHF 2 -3-Py], [} BG2557: 2-CN-6-CHF 2 -3-Py], [BG2558: 4-CN-6-CHF 2 -3-Py], [BG2559: 5-CN-6 _{-CHF 2 -3-Py], [} BG2560: 2-OMe-6-CHF 2 -3-Py], [BG2561: 4-OMe-6-CHF 2 -3-Py], [BG2562: 5-OMe- _{6-CHF 2 -3-Py]} , [BG2563: 2-OCHF 2 -3-Py], [BG2564: 4-Cl-2-OCHF 2 -3-Py], [BG2565: 5-Cl-2-OCHF _{2 -3-Py], [BG2566} : 6-Cl-2-OCHF 2 -3-Py], [BG2567: 4-Me-2-OCHF 2 -3-Py], [BG2568: 5-Me-2- OCHF ₂ -3-Py, [BG 2569: 6-Me-2-OCHF ₂ -3-Py], [BG 2 570: 4-CF ₃ -2-OCHF ₂ -3-Py], _{BG2571: 5-CF 3 -2-} OCHF 2 -3-Py], [BG2572: 6-CF 3 -2-OCHF 2 -3-Py], [BG2573: 4-CN-2-OCHF 2 -3-Py ], [BG2574: 5-CN -2-OCHF 2 -3-Py], [BG2575: 6-CN-2-OCHF 2 -3-Py], [BG2576: 4-OMe-2-OCHF 2 -3- Py], [BG2577: 5- OMe-2-OCHF 2 -3-Py], [BG2578: 6-OMe-2-OCHF 2 -3-Py], [BG2579: 4-OCHF 2 -3-Py], [BG2580: 2-Cl-4 -OCHF 2 -3-Py], [BG2581: 5-Cl-4-OCHF 2 -3-Py], [BG2582: 6-Cl-4-OCHF 2 -3-Py] , [BG2583: 2-Me- 4-OCHF 2 -3-Py], [BG2584: 5-Me-4-OCHF 2 -3-Py], [BG2585: 6-Me-4-OCHF 2 -3-Py ], [BG 2586: 2-CF ₃ -4-OCHF ₂ -3-Py], [BG 2587: 5-CF ₃ -4-OCHF ₂ -3-Py], [BG 2588: 6-CF ₃ -4-OCHF _2] -3-Py], [BG2589: 2-CN-4-OCHF 2 -3-Py], [BG2590: 5-CN-4-OCHF 2 -3-Py], [BG2591: 6-CN-4-OCHF ₂ -3-Py], [BG2592: 2-OMe-4-OCHF ₂ -3-Py], [BG2593: 5-OMe-4-OCHF ₂ -3-Py], [BG2594: 6-OMe -4-] OCHF _2-3 -Py], [BG 2595: 5-OCHF _2-3 -Py], [BG 2596: 2-Cl-5-OCHF _2-3 -Py], [BG 2597: 4-Cl-5-OCHF _2- 3-Py], [BG2598: 6-Cl-5-OCHF 2 -3-Py], [BG2599: 2-Me-5-OCHF 2 -3-Py], [BG2600: 4-Me-5-OCHF 2 -3-Py],

[BG2601: 6-Me-5-OCHF ₂ -3-Py], [BG 2602: 2-CF ₃ -5-OCHF ₂ -3-Py], [BG 2603: 4-CF ₃ -5-OCHF ₂ -3- ₂ Py], [BG2604: 6- CF 3 -5-OCHF 2 -3-Py], [BG2605: 2-CN-5-OCHF 2 -3-Py], [BG2606: 4-CN-5-OCHF 2 - 3-Py], [BG2607: 6-CN-5-OCHF 2 -3-Py], [BG2608: 2-OMe-5-OCHF 2 -3-Py], [BG2609: 4-OMe-5-OCHF 2 -3-Py, [BG2610: 6-OMe-5-OCHF ₂ -3-Py], [BG 2611: 6-OCHF ₂ -3-Py], [BG 2612: 2-Cl-6-OCHF ₂ -3- Py], [BG2613: 4- Cl-6-OCHF 2 -3-Py], [BG2614: 5-Cl-6-OCHF 2 -3-Py], [BG2615: 2-Me-6-OCHF 2 -3 -Py], [BG2616: 4- Me-6-OCHF 2 -3-Py], [BG2617: 5-Me-6-OCHF 2 -3-Py], [BG2618: 2-CF 3 -6-OCHF 2 -3-Py], [BG2619: 4-CF 3 -6-OCHF 2 -3-Py], [BG2620: 5-CF 3 -6-OCHF 2 -3-Py], [BG2621: 2-CN-6 _{-OCHF 2 -3-Py], [} BG2622: 4-CN-6-OCHF 2 -3-Py], [BG2623: 5-CN-6-OCHF 2 -3-Py], [BG2624: 2-OMe- _{6-OCHF 2 -3-Py]} , [BG2625: 4-OMe-6-OCHF 2 -3-Py], [BG2626: 5-OMe-6-OCHF 2 -3-Py], [BG2627: 2-Et -3-Py !, [BG2628: 4-Cl-2-Et-3-Py], [BG2629: 5-Cl-2-Et-3-Py], [BG 2630: 6-Cl-2-Et-3] -Py], [BG2631: 4-Me-2-Et-3-Py], [BG2632: 5-Me-2-Et-3-Py], [BG2633: 6-Me-2-Et-3-Py] ], [BG2634: 4-CF 3 -2-Et-3-Py], [BG2635: 5-CF 3 -2-Et-3-Py], [BG2636: 6- _{CF 3 -2-Et-3-} Py], [BG2637: 4-CN-2-Et-3-Py], [BG2638: 5-CN-2-Et-3-Py], [BG2639: 6-CN -2-Et-3-Py !, [BG2640: 4-OMe-2-Et-3-Py], [BG2641: 5-OMe-2-Et-3-Py], [BG2642: 6-OMe-2] -Et-3-Py], [BG2643: 4-Et-3-Py], [BG2644: 2-Cl-4-Et-3-Py], [BG2645: 5-Cl-4-Et-3-Py] ], [BG 2 646: 6-Cl-4-Et-3-Py], [BG 2647: 2-Me-4-Et-3-Py], [BG 2648: 5-Me-4-Et-3-Py], [BG2649: 6-Me-4 -Et-3-Py], [BG2650: 2-CF 3 -4-Et-3-Py], [BG2651: 5-CF 3 -4-Et-3-Py], _{[BG2652: 6-CF 3 -4} -Et-3-Py], [BG2653: 2-CN-4-Et-3-Py], [BG2654: 5-CN-4-Et-3-Py], [ BG2655: 6-CN-4-Et-3-Py], [BG2656: 2-OMe-4-Et-3-Py], [BG2657: 5-OMe-4-Et-3-Py], [BG2658: 6-OMe-4-Et-3-Py], [BG2659: 5-Et-3-Py], [BG2660: 2-Cl-5-Et-3-Py], [BG2661: 4-Cl-5- Et-3-Py, [BG2662: 6-Cl-5-Et-3-Py], [BG 2663: 2-Me-5-Et-3-Py], [BG 2664: 4-Me-5-Et- 3-Py], [BG2665: 6-Me-5-Et-3-Py], [BG2666: 2-CF 3 -5-Et-3-Py], [BG2667: 4-CF 3 -5-Et- 3-Py], [BG2668: 6-CF 3 -5-Et-3-Py], [BG2669: 2-CN-5-Et-3-Py], [BG2670: 4-CN-5-Et-3 -Py], [BG2671: 6-CN-5-Et-3-Py], [BG2672: 2-OMe-5-Et-3-Py], [BG 2673: 4-OMe-5-Et-3-Py ], [BG 2674: 6-OMe-5-Et-3-Py], [BG 2 675: 6-Et-3-Py], [BG 2 676: 2-Cl-6-Et-3-Py], [BG 2677: 4] -C l-6-Et-3-Py], [BG2678: 5-Cl-6-Et-3-Py], [BG2679: 2-Me-6-Et-3-Py], [BG2 680: 4-Me- 6-Et-3-Py] , [BG2681: 5-Me-6-Et-3-Py], [BG2682: 2-CF 3 -6-Et-3-Py], [BG2683: 4-CF 3 - 6-Et-3-Py] , [BG2684: 5-CF 3 -6-Et-3-Py], [BG2685: 2-CN-6-Et-3-Py], [BG2686: 4-CN-6 -Et-3-Py], [BG2687: 5-CN-6-Et-3-Py], [BG2688: 2-OMe-6-Et-3-Py], [BG2689: 4-OMe-6-Et] -3-Py], [BG2690: 5-OMe-6-Et-3-Py], [BG2691: 2-CH 2 CF 3 -3-Py], [BG2692: 4-Cl-2-CH 2 CF 3 -3-Py], [BG2693: 5-Cl-2-CH 2 CF 3 -3-Py], [BG2694: 6-Cl-2-CH 2 CF 3 -3-Py], [BG2695: 4-Me _{-2-CH 2 CF 3 -3-} Py], [BG2696: 5-Me-2-CH 2 CF 3 -3-Py], [BG2697: 6-Me-2-CH 2 CF 3 -3-Py] _{, [BG2698: 4-CF 3} -2-CH 2 CF 3 -3-Py], [BG2699: 5-CF 3 -2-CH 2 CF 3 -3-Py], [BG2700: 6-CF 3 -2 -CH ₂ CF ₃ -3-Py],

[BG2701: 4-CN-2 -CH 2 CF 3 -3-Py], [BG2702: 5-CN-2-CH 2 CF 3 -3-Py], [BG2703: 6-CN-2-CH 2 CF ₃ -3-Py, [BG 2704: 4-OMe -2-CH ₂ CF ₃ -3-Py], [BG 2 705: 5-OMe -2-CH ₂ CF ₃ -3-Py], [BG 2706: 6- _{OMe-2-CH 2 CF 3} -3-Py], [BG2707: 4-CH 2 CF 3 -3-Py], [BG2708: 2-Cl-4-CH 2 CF 3 -3-Py], [BG2709 : 5-Cl-4-CH 2 CF 3 -3-Py], [BG2710: 6-Cl-4-CH 2 CF 3 -3-Py], [BG2711: 2-Me-4-CH 2 CF 3 - 3-Py], [BG2712: 5-Me-4-CH 2 CF 3 -3-Py], [BG2713: 6-Me-4-CH 2 CF 3 -3-Py], [BG2714: 2-CF 3 -4-CH ₂ CF ₃ -3-Py, [BG 2715: 5-CF ₃ -4-CH ₂ CF ₃ -3-Py], [BG 2716: 6-CF ₃ -4-CH ₂ CF ₃ -3- Py], [BG2717: 2- CN-4-CH 2 CF 3 -3-Py], [BG2718: 5-CN-4-CH 2 CF 3 -3-Py], [BG2719: 6-CN-4- _{CH 2 CF 3 -3-Py]} , [BG2720: 2-OMe-4-CH 2 CF 3 -3-Py], [BG2721: 5-OMe-4-CH 2 CF 3 -3-Py], [BG2722 : 6-OMe-4-CH 2 CF 3 -3-Py], [BG2723: 5-CH 2 CF 3 -3-Py], [BG2724: 2-Cl-5-CH 2 CF 3 -3-Py] , [BG2725: 4-Cl- 5-CH 2 CF 3 -3-Py], [BG2726: 6-Cl-5-CH 2 CF 3 -3-Py], [BG2727: 2-Me-5-CH 2 CF ₃ -3-Py, [BG ₂ 728: 4-Me-5-CH ₂ CF ₃ -3-Py], [BG ₂ 729: 6-Me-5-CH ₂ CF ₃ -3-Py], [BG 2 730: 2] —CF ₃ -5-CH ₂ CF ₃ -3-Py], [BG 2731: 4-CF ₃ -5-CH ₂ CF ₃ -3-P y], [BG2732: 6- CF 3 -5-CH 2 CF 3 -3-Py], [BG2733: 2-CN-5-CH 2 CF 3 -3-Py], [BG2734: 4-CN-5 _{-CH 2 CF 3 -3-Py]} , [BG2735: 6-CN-5-CH 2 CF 3 -3-Py], [BG2736: 2-OMe-5-CH 2 CF 3 -3-Py], [ BG2737: 4-OMe-5- CH2CF 3 -3-Py], [BG2738: 6-OMe-5-CH2CF 3 -3-Py], [BG2739: 6-CH2CF 3 -3-Py], [BG2740: 2 _{-Cl-6-CH 2 CF 3} -3-Py], [BG2741: 4-Cl-6-CH 2 CF 3 -3-Py], [BG2742: 5-Cl-6-CH 2 CF 3 -3- Py], [BG2743: 2- Me-6-CH 2 CF 3 -3-Py], [BG2744: 4-Me-6-CH 2 CF 3 -3-Py], [BG2745: 5-Me-6- _{CH 2 CF 3 -3-Py]} , [BG2746: 2-CF 3 -6-CH 2 CF 3 -3-Py], [BG2747: 4-CF 3 -6-CH 2 CF 3 -3-Py], _{[BG2748: 5-CF 3 -6} -CH 2 CF 3 -3-Py], [BG2749: 2-CN-6-CH 2 CF 3 -3-Py], [BG2750: 4-CN-6-CH 2 _{CF 3 -3-Py], [} BG2751: 5-CN-6-CH 2 CF 3 -3-Py], [BG2752: 2-OMe-6-CH 2 CF 3 -3-Py], [BG2753: 4 _{-OMe-6-CH 2 CF 3} -3-Py], [BG2754: 5-OMe-6-CH 2 CF 3 -3-Py], [BG2755: 2-OEt-3-Py], [BG2756: 4 -Cl-2-OEt-3-Py], [BG2757: 5-Cl-2-OEt-3-Py], [BG2758: 6-Cl-2-OEt-3-Py], [BG2759: 4-Me -2-OEt-3-Py !, [BG2760: 5-Me-2-OEt-3-Py], [BG2761: 6-Me-2-OEt-3-Py], [BG2762: 4-CF _3- 2-OEt-3-Py] , [BG2763: 5-CF 3 -2-OEt-3-Py], [BG2764: 6-CF 3 -2-OEt-3-Py], [BG2765: 4-CN-2-OEt-3-Py], [BG2766: 5-CN-2-OEt-3-Py], [BG2767: 6-CN-2-OEt-3-Py], [BG2768] : 4-OMe-2-OEt-3-Py], [BG2769: 5-OMe-2-OEt-3-Py], [BG2770: 6-OMe-2-OEt-3-Py], [BG2771: 4] -OEt-3-Py, [BG2772: 2-Cl-4-OEt-3-Py], [BG2773: 5-Cl-4-OEt-3-Py], [BG2774: 6-Cl-4-OEt -3-Py !, [BG2775: 2-Me-4-OEt-3-Py], [BG2776: 5-Me-4-OEt-3-Py], [BG2777: 6-Me-4-OEt-3] -Py], [BG2778: 2- CF 3 -4-OEt-3-Py], [BG2779: 5-CF 3 -4-OEt-3-Py], [BG2780: 6-CF 3 -4-OEt- 3-Py], [BG2781: 2-CN-4-OEt-3-Py], [BG2782: 5-CN-4-OEt-3-Py], [BG2783: 6-CN-4-OEt-3-] Py], [BG2784: 2-OMe-4-OEt-3-Py], [BG2785: 5-OMe-4-OEt-3-Py], [BG2786: 6-OMe-4-OEt-3-Py] [BG 2787: 5-OEt-3-Py], [BG 2 788: 2-Cl-5-OEt-3-Py], [BG 2 789: 4-Cl-5-OEt-3-Py], [BG 2 790: 6- Cl-5-OEt-3-Py, [BG2791: 2-Me-5-OEt-3-Py], [BG2792: 4-Me-5-OEt-3-Py], [BG2793: 6-Me- 5-OEt-3-Py] , [BG2794: 2-CF 3 -5-OEt-3-Py], [BG2795: 4-CF 3 -5-OEt-3-Py], [BG2796: 6-CF 3 -5-OEt-3-Py !, [BG2797: 2-CN-5-OEt-3-Py], [BG2798: 4-CN-5-OEt-3-Py], [BG2799: 6-CN-5] -OEt-3-Py], [BG2800: 2-OMe-5-OEt-3-Py],

[BG2801: 4-OMe-5-OEt-3-Py], [BG2802: 6-OMe-5-OEt-3-Py], [BG2803: 6-OEt-3-Py], [BG2804: 2-Cl] -6-OEt-3-Py !, [BG2805: 4-Cl-6-OEt-3-Py], [BG2806: 5-Cl-6-OEt-3-Py], [BG2807: 2-Me-6] -OEt-3-Py], [BG2808: 4-Me-6-OEt-3-Py], [BG2809: 5-Me-6-OEt-3-Py], [BG 2810: 2-CF ₃ -6-] OEt-3-Py], [ BG2811: 4-CF 3 -6-OEt-3-Py], [BG2812: 5-CF 3 -6-OEt-3-Py], [BG2813: 2-CN-6- OEt-3-Py], [BG2814: 4-CN-6-OEt-3-Py], [BG2815: 5-CN-6-OEt-3-Py], [BG2816: 2-OMe-6-OEt- 3-Py], [BG2817: 4-OMe-6-OEt-3-Py], [BG2818: 5-OMe-6-OEt-3-Py], [BG2819: 2-OCH 2 CF 3 -3-Py ], [BG2820: 4-Cl -2-OCH 2 CF 3 -3-Py], [BG2821: 5-Cl-2-OCH 2 CF 3 -3-Py], [BG2822: 6-Cl-2-OCH _{2 CF 3 -3-Py],} [BG2823: 4-Me-2-OCH 2 CF 3 -3-Py], [BG2824: 5-Me-2-OCH 2 CF 3 -3-Py], [BG2825: _{6-Me-2-OCH 2} CF 3 -3-Py], [BG2826: 4-CF 3 -2-OCH 2 CF 3 -3-Py], [BG2827: 5-CF 3 -2-OCH 2 CF 3 -3-Py], [BG2828: 6-CF 3 -2-OCH 2 CF 3 -3-Py], [BG2829: 4-CN-2-OCH 2 CF 3 -3-Py], [BG2830: 5- _{CN-2-OCH 2 CF 3} -3-Py], [BG2831: 6-CN-2-OCH 2 CF 3 -3-Py], [BG2832: 4-OMe-2-OCH 2 CF 3 -3-Py ], [BG2833: 5-OMe -2-OCH 2 CF 3 -3-Py], [BG2834: 6-OMe-2-OCH 2 CF 3 -3-Py], [BG283 _{5: 4-OCH 2 CF 3} -3-Py], [BG2836: 2-Cl-4-OCH 2 CF 3 -3-Py], [BG2837: 5-Cl-4-OCH 2 CF 3 -3-Py ], [BG2838: 6-Cl -4-OCH 2 CF 3 -3-Py], [BG2839: 2-Me-4-OCH 2 CF 3 -3-Py], [BG2840: 5-Me-4-OCH _{2 CF 3 -3-Py],} [BG2841: 6-Me-4-OCH 2 CF 3 -3-Py], [BG2842: 2-CF 3 -4-OCH 2 CF 3 -3-Py], [BG2843 : 5-CF ₃ -4-OCH ₂ CF ₃ -3-Py], [BG 2844: 6-CF ₃ -4-OCH ₂ CF ₃ -3-Py], [BG 2 845: 2-CN-4-OCH ₂ CF _{3 -3-Py], [BG2846} : 5-CN-4-OCH 2 CF 3 -3-Py], [BG2847: 6-CN-4-OCH 2 CF 3 -3-Py], [BG2848: 2- _{OMe-4-OCH 2 CF 3} -3-Py], [BG2849: 5-OMe-4-OCH 2 CF 3 -3-Py], [BG2850: 6-OMe-4-OCH 2 CF 3 -3-Py ], [BG2851: 5-OCH 2 CF 3 -3-Py], [BG2852: 2-Cl-5-OCH 2 CF 3 -3-Py], [BG2853: 4-Cl-5-OCH 2 CF 3 - 3-Py], [BG2854: 6-Cl-5-OCH 2 CF 3 -3-Py], [BG2855: 2-Me-5-OCH 2 CF 3 -3-Py], [BG2856: 4-Me- _{5-OCH 2 CF 3 -3-} Py], [BG2857: 6-Me-5-OCH 2 CF 3 -3-Py], [BG2858: 2-CF 3 -5-OCH 2 CF 3 -3-Py] [BG 2859: 4-CF ₃ -5-OCH ₂ CF ₃ -3-Py], [BG 2860: 6-CF ₃ -5-OCH ₂ CF ₃ -3-Py], [BG 2 8 1: 2 -CN -5- _{OCH 2 CF 3 -3-Py]} , [BG2862: 4-CN-5-OCH 2 CF 3 -3-Py], [BG2863: 6-CN-5-OCH 2 CF 3 -3-Py], [BG2864 : 2-OMe-5-OCH ₂ CF ₃ -3-Py], [BG2 865: 4-OMe-5- OCH 2 CF 3 -3-Py], [BG2866: 6-OMe-5-OCH 2 CF 3 -3-Py], [BG2867: 6-OCH 2 CF 3 -3-Py ], [BG2868: 2-Cl -6-OCH 2 CF 3 -3-Py], [BG2869: 4-Cl-6-OCH 2 CF 3 -3-Py], [BG2870: 5-Cl-6-OCH _{2 CF 3 -3-Py],} [BG2871: 2-Me-6-OCH 2 CF 3 -3-Py], [BG2872: 4-Me-6-OCH 2 CF 3 -3-Py], [BG2873: _{5-Me-6-OCH 2} CF 3 -3-Py], [BG2874: 2-CF 3 -6-OCH 2 CF 3 -3-Py], [BG2875: 4-CF 3 -6-OCH 2 CF 3 -3-Py], [BG2876: 5-CF 3 -6-OCH 2 CF 3 -3-Py], [BG2877: 2-CN-6-OCH 2 CF 3 -3-Py], [BG2878: 4- _{CN-6-OCH 2 CF 3} -3-Py], [BG2879: 5-CN-6-OCH 2 CF 3 -3-Py], [BG2880: 2-OMe-6-OCH2CF 3 -3-Py], [BG2881: 4-OMe-6 -OCH 2 CF 3 -3-Py], [BG2882: 5-OMe-6-OCH 2 CF 3 -3-Py], [BG2883: 2-Pr-3-Py], [BG2884: 4-Cl-2-Pr-3-Py], [BG2885: 5-Cl-2-Pr-3-Py], [BG2288: 6-Cl-2-Pr-3-Py], [BG 2887] : [4-Me-2-Pr-3-Py], [BG2888: 5-Me-2-Pr-3-Py], [BG2889: 6-Me-2-Pr-3-Py], [BG2890: 4] _{-CF 3 -2-Pr-3-} Py], [BG2891: 5-CF 3 -2-Pr-3-Py], [BG2892: 6-CF 3 -2-Pr-3-Py], [BG2893: 4-CN-2-Pr-3-Py, [BG2894: 5-CN-2-Pr-3-Py], [BG2895: 6-CN-2-Pr-3-Py], [BG2896: 4-] OMe-2-Pr-3-Py, [BG 2897: 5-OMe-2-Pr-3-Py], [BG 2898: 6-OMe-2-Pr-3-Py], [BG 2899: 4-Pr -3-Py], [BG2900: 2-Cl-4-Pr-3-Py],

[BG2901: 5-Cl-4-Pr-3-Py], [BG2902: 6-Cl-4-Pr-3-Py], [BG2903: 2-Me-4-Pr-3-Py], [BG2904] : 5-Me-4-Pr -3-Py], [BG2905: 6-Me-4-Pr-3-Py], [BG2906: 2-CF 3 -4-Pr-3-Py], [BG2907: _{5-CF 3 -4-Pr-} 3-Py], [BG2908: 6-CF 3 -4-Pr-3-Py], [BG2909: 2-CN-4-Pr-3-Py], [BG2910: 5-CN-4-Pr-3-Py, [BG2911: 6-CN-4-Pr-3-Py], [BG2912: 2-OMe-4-Pr-3-Py], [BG2913: 5-] OMe-4-Pr-3-Py, [BG2914: 6-OMe-4-Pr-3-Py], [BG2915: 5-Pr-3-Py], [BG2916: 2-Cl-5-Pr- 3-Py], [BG2917: 4-Cl-5-Pr-3-Py], [BG2918: 6-Cl-5-Pr-3-Py], [BG2919: 2-Me-5-Pr-3- 3 Py], [BG2920: 4- Me-5-Pr-3-Py], [BG2921: 6-Me-5-Pr-3-Py], [BG2922: 2-CF 3 -5-Pr-3-Py ], [BG2923: 4-CF 3 -5-Pr-3-Py], [BG2924: 6-CF 3 -5-Pr-3-Py], [BG2925: 2-CN-5-Pr-3-Py ], [BG 2926: 4-CN-5-Pr-3-Py], [BG 2 927: 6-CN-5-Pr-3-Py], [BG 2 928: 2-OMe-5-Pr-3-Py], [BG2929: 4-OMe-5-Pr-3-Py], [BG2930: 6-OMe-5-Pr-3-Py], [BG2931: 6-Pr-3-Py], [BG2932: 2-Cl -6-Pr-3-Py], [BG 2933: 4-Cl-6-Pr-3-Py], [BG 2 934: 5-Cl-6-Pr-3-Py], [BG 2935: 2-Me-6 -Pr-3-Py], [BG 2 936: 4-Me-6-Pr-3-Py], [BG 2 937: 5-Me-6-Pr-3-Py], [BG 2938: 2-CF ₃ -6- Pr-3-Py], [ BG2939: 4-CF 3 -6-Pr-3-Py], [BG2940: 5-CF 3 -6-Pr-3-Py], [BG2941: 2-CN-6- Pr -3-Py], [BG2942: 4-CN-6-Pr-3-Py], [BG2943: 5-CN-6-Pr-3-Py], [BG2944: 2-OMe-6-Pr-3 -Py], [BG2945: 4-OMe-6-Pr-3-Py], [BG2946: 5-OMe-6-Pr-3-Py], [BG2947: 2-OPr-3-Py], [BG2948] : 4-Cl-2-OPr-3-Py], [BG 2949: 5-Cl-2-OPr-3-Py], [BG 2950: 6-Cl-2-OPr-3-Py], [BG 2 951: 4] -Me-2-OPr-3-Py], [BG2952: 5-Me-2-OPr-3-Py], [BG2953: 6-Me-2-OPr-3-Py], [BG2954: 4-CF _{3 -2-OPr-3-Py} ], [BG2955: 5-CF 3 -2-OPr-3-Py], [BG2956: 6-CF 3 -2-OPr-3-Py], [BG2957: 4- CN-2-OPr-3-Py, [BG2958: 5-CN-2-OPr-3-Py], [BG2959: 6-CN-2-OPr-3-Py], [BG2960: 4-OMe- 2-OPr-3-Py], [BG2961: 5-OMe-2-OPr-3-Py], [BG2962: 6-OMe-2-OPr-3-Py], [BG2963: 4-OPr-3-3] Py], [BG2964: 2-Cl-4-OPr-3-Py], [BG2965: 5-Cl-4-OPr-3-Py], [BG 2966: 6-Cl-4-OPr-3-Py] , [BG2967: 2-Me-4-OPr-3-Py], [BG2968: 5-Me-4-OPr-3-Py], [BG2969: 6-Me-4-OPr-3-Py], _{BG2970: 2-CF 3 -4-} OPr-3-Py], [BG2971: 5-CF 3 -4-OPr-3-Py], [BG2972: 6-CF 3 -4-OPr-3-Py], [BG2 973: 2-CN-4-OPr-3-Py], [BG2 974: 5-CN-4-OPr-3-Py], [BG2 975: 6-CN-4-OPr-3-Py], [BG2976] : 2-OMe-4-OPr-3-Py], [BG2977: 5-OMe-4-OPr-3-Py], [BG2978: 6-OMe-4-OPr-3-Py], [BG2979: 5] -OPr-3-Py], [BG 2 980: 2-Cl-5-OPr-3-Py], [BG 2 981: 4-C] l-5-OPr-3-Py], [BG2982: 6-Cl-5-OPr-3-Py], [BG2983: 2-Me-5-OPr-3-Py], [BG2984: 4-Me- 5-OPr-3-Py] , [BG2985: 6-Me-5-OPr-3-Py], [BG2986: 2-CF 3 -5-OPr-3-Py], [BG2987: 4-CF 3 - 5-OPr-3-Py] , [BG2988: 6-CF 3 -5-OPr-3-Py], [BG2989: 2-CN-5-OPr-3-Py], [BG2990: 4-CN-5 -OPr-3-Py], [BG2991: 6-CN-5-OPr-3-Py], [BG2992: 2-OMe-5-OPr-3-Py], [BG2993: 4-OMe-5-OPr -3-Py !, [BG2994: 6-OMe-5-OPr-3-Py], [BG2995: 6-OPr-3-Py], [BG2996: 2-Cl-6-OPr-3-Py], [BG2997: 4-Cl-6-OPr-3-Py], [BG2998: 5-Cl-6-OPr-3-Py], [BG2999: 2-Me-6-OPr-3-Py], [BG3000] : 4-Me-6-OPr-3-Py],

[BG3001: 5-Me-6 -OPr-3-Py], [BG3002: 2-CF 3 -6-OPr-3-Py], [BG3003: 4-CF 3 -6-OPr-3-Py], _{[BG3004: 5-CF 3 -6} -OPr-3-Py], [BG3005: 2-CN-6-OPr-3-Py], [BG3006: 4-CN-6-OPr-3-Py], [ BG3007: 5-CN-6-OPr-3-Py !, [BG3008: 2-OMe-6-OPr-3-Py], [BG3009: 4-OMe-6-OPr-3-Py], [BG3010: 5-OMe-6-OPr-3-Py], [BG3011: 2-SMe-3-Py], [BG3012: 4-Cl-2-SMe-3-Py], [BG3013: 5-Cl-2-] SMe-3-Py !, [BG3014: 6-Cl-2-SMe-3-Py], [BG3015: 4-Me-2-SMe-3-Py], [BG3016: 5-Me-2-SMe- 3-Py], [BG3017: 6-Me-2-SMe-3-Py], [BG3018: 4-CF 3 -2-SMe-3-Py], [BG3019: 5-CF 3 -2-SMe- 3-Py], [BG3020: 6-CF 3 -2-SMe-3-Py], [BG3021: 4-CN-2-SMe-3-Py], [BG3022: 5-CN-2-SMe-3 -Py], [BG3023: 6-CN-2-SMe-3-Py], [BG3024: 4-OMe-2-SMe-3-Py], [BG3025: 5-OMe-2-SMe-3-Py] ], [BG3026: 6-OMe-2-SMe-3-Py], [BG3027: 4-SMe-3-Py], [BG3028: 2-Cl-4-SMe-3-Py], [BG3029: 5] -Cl-4-SMe-3-Py, [BG3030: 6-Cl-4-SMe-3-Py], [BG3031: 2-Me-4-SMe-3-Py], [BG3032: 5-Me -4-SMe-3-Py] , [BG3033: 6-Me-4-SMe-3-Py], [BG3034: 2-CF 3 -4-SMe-3-Py], [BG3035: 5-CF 3 -4-SMe-3-Py !, [BG 3036: 6-CF ₃ -4-SMe-3-Py], [BG 3037: 2-CN-4-SMe-3-Py], [BG 3038: 5-CN- 4-SMe-3-Py], [BG3039: 6-CN-4-SMe-3-Py], [B G3040: 2-OMe-4-SMe-3-Py], [BG3041: 5-OMe-4-SMe-3-Py], [BG3042: 6-OMe-4-SMe-3-Py], [BG3043: 5-SMe-3-Py !, [BG3044: 2-Cl-5-SMe-3-Py], [BG3045: 4-Cl-5-SMe-3-Py], [BG 3046: 6-Cl-5-] SMe-3-Py, [BG3047: 2-Me-5-SMe-3-Py], [BG3048: 4-Me-5-SMe-3-Py], [BG3049: 6-Me-5-SMe- 3-Py], [BG3050: 2-CF 3 -5-SMe-3-Py], [BG3051: 4-CF 3 -5-SMe-3-Py], [BG3052: 6-CF 3 -5-SMe -3-Py !, [BG3053: 2-CN-5-SMe-3-Py], [BG3054: 4-CN-5-SMe-3-Py], [BG3055: 6-CN-5-SMe-3] -Py], [BG 3056: 2-OMe-5-SMe-3-Py], [BG3057: 4-OMe-5-SMe-3-Py], [BG 3058: 6-OMe-5-SMe-3-Py] ], [BG3059: 6-SMe-3-Py], [BG3060: 2-Cl-6-SMe-3-Py], [BG3061: 4-Cl-6-SMe-3-Py], [BG3062: 5] -Cl-6-SMe-3-Py], [BG3063: 2-Me-6-SMe-3-Py], [BG3064: 4-Me-6-SMe-3-Py], [BG3065: 5-Me -6-SMe-3-Py] , [BG3066: 2-CF 3 -6-SMe-3-Py], [BG3067: 4-CF 3 -6-SMe-3-Py], [BG3068: 5-CF ₃ -6-SMe-3-Py !, [BG3069: 2-CN-6-SMe-3-Py], [BG3070: 4-CN-6-SMe-3-Py], [BG3071: 5-CN- 6-SMe-3-Py], [BG3072: 2-OMe-6-SMe-3-Py], [BG3073: 4-OMe-6-SMe-3-Py], [BG3074: 5-OMe-6-6] SMe-3-Py], [ BG3075: 2-SCF 3 -3-Py], [BG3076: 4-Cl-2-SCF 3 -3-Py], [BG3077: 5-Cl-2-SCF 3 -3 -Py], [BG3078: 6-Cl-2-SCF ₃ -3-Py], [BG 3079: 4-Me-2- SCF 3 -3-Py], [BG3080: 5-Me-2-SCF 3 -3-Py], [BG3081: 6-Me-2-SCF 3 -3-Py], _{[BG3082: 4-CF 3 -2} -SCF 3 -3-Py], [BG3083: 5-CF 3 -2-SCF 3 -3-Py], [BG3084: 6-CF 3 -2-SCF 3 -3 -Py], [BG3085: 4- CN-2-SCF 3 -3-Py], [BG3086: 5-CN-2-SCF 3 -3-Py], [BG3087: 6-CN-2-SCF 3 - 3-Py], [BG3088: 4-OMe-2-SCF 3 -3-Py], [BG3089: 5-OMe-2-SCF 3 -3-Py], [BG3090: 6-OMe-2-SCF 3 -3-Py], [BG3091: 4-SCF 3 -3-Py], [BG3092: 2-Cl-4-SCF 3 -3-Py], [BG3093: 5-Cl-4-SCF 3 -3- Py], [BG3094: 6- Cl-4-SCF 3 -3-Py], [BG3095: 2-Me-4-SCF 3 -3-Py], [BG3096: 5-Me-4-SCF 3 -3 -Py], [BG3097: 6- Me-4-SCF 3 -3-Py], [BG3098: 2-CF 3 -4-SCF 3 -3-Py], [BG3099: 5-CF 3 -4-SCF ₃ -3-Py, [BG ₃ 100: 6-CF ₃ -4-SCF ₃ -3-Py],

[BG3101: 2-CN-4 -SCF 3 -3-Py], [BG3102: 5-CN-4-SCF 3 -3-Py], [BG3103: 6-CN-4-SCF 3 -3-Py] , [BG3104: 2-OMe- 4-SCF 3 -3-Py], [BG3105: 5-OMe-4-SCF 3 -3-Py], [BG3106: 6-OMe-4-SCF 3 -3-Py ], [BG 3107: 5-SCF ₃ -3-Py], [BG 3108: 2-Cl-5-SCF ₃ -3-Py], [BG 3109: 4-Cl-5-SCF ₃ -3-Py], [BG _{3 10 7} BG 3110: 6-Cl-5-SCF ₃ -3-Py, [BG 3 11 1: 2-Me-5-SCF ₃ -3-Py], [BG 3 112: 4-Me-5-SCF ₃ -3-Py], [BG 3113: 6-Me-5-SCF ₃ -3-Py], [BG ₃ 114: 2-CF ₃ -5-SCF ₃ -3-Py], [BG ₃ 115: 4-CF ₃ -5- SCF ₃ -3- Py], [BG3116: 6- CF 3 -5-SCF 3 -3-Py], [BG3117: 2-CN-5-SCF 3 -3-Py], [BG3118: 4-CN-5-SCF 3 - 3-Py], [BG 3119: 6-CN-5-SCF ₃ -3-Py], [BG 3 120: 2-OMe-5-SCF ₃ -3-Py], [BG 3121: 4-OMe-5-SCF ₃ -3-Py, [BG3122: 6-OMe-5-SCF ₃ -3-Py], [BG 3123: 6-SCF ₃ -3-Py], [BG 3124: 2-Cl-6-SCF ₃ -3- Py], [BG3125: 4- Cl-6-SCF 3 -3-Py], [BG3126: 6-Cl-6-SCF 3 -3-Py], [BG3127: 2-Me-6-SCF 3 -3 -Py], [BG3128: 4- Me-6-SCF 3 -3-Py], [BG3129: 6-Me-6-SCF 3 -3-Py], [BG3130: 2-CF 3 -6-SCF 3 -3-Py], [BG3131: 4-CF 3 -6-SCF 3 -3-Py], [BG3132: 6-CF 3 -6-SCF 3 -3-Py], [BG3133: 2-CN-6 -SCF ₃ -3-Py], [BG 3134: 4-CN-6-SCF ₃ -3-Py], [BG 3 135: 6-CN-6-SCF ₃ -3-Py], [BG 313 6: 2-OMe-6- SCF 3 -3-Py], [BG3137: 4-OMe-6-SCF 3 -3-Py], [BG3138: 6-OMe-6-SCF 3 -3-Py], [BG3139: 2-S (O) Me-3-Py], [BG3140: 4-Cl-2-S (O) Me-3-Py], [BG3141: 5-Cl-2-S (O) Me -3-Py !, [BG3142: 6-Cl-2-S (O) Me-3-Py], [BG3143: 4-Me-2-S (O) Me-3-Py], [BG3144: 5] -Me-2-S (O) Me-3-Py], [BG3145: 6-Me-2-S (O) Me-3-Py], [BG3146: 4-CF 3 -2-S (O) Me-3-Py], [ BG3147: 5-CF 3 -2-S (O) Me-3-Py], [BG3148: 6-CF 3 -2-S (O) Me-3-Py], [ BG3149: 4-CN-2-S (O) Me-3-Py], [BG3150: 5-CN-2-S (O) Me-3-Py], [BG3151: 6-CN-2-S ( O) Me-3-Py], [BG3152: 4-OMe-2-S (O) Me-3-Py], [BG3153: 5-OMe-2-S (O) Me-3-Py], [BG3 153] BG3154: 6-OMe-2-S (O) Me-3-Py], [BG3155: 4-S (O) Me-3-Py], [BG3156: 2-Cl-4-S (O) Me- 3-Py], [BG3157: 5-Cl-4-S (O) Me-3-Py], [BG3158: 6-Cl-4-S (O) Me-3-Py], [BG3159: 2- Me-4-S (O) Me-3-Py], [BG3160: 5-Me-4-S (O) Me-3-Py], [BG3161: 6-Me-4-S (O) Me- 3-Py], [BG3162: 2-CF 3 -4-S (O) Me-3-Py], [BG3163: 5-CF 3 -4-S (O) Me-3-Py], [BG3164: _{6-CF 3 -4-S (} O) Me-3-Py], [BG3165: 2-CN-4-S (O) Me-3-Py], [BG3166: 5-CN-4-S (O ) Me-3-Py], [BG3167: 6-CN-4-S (O) Me-3-Py], [BG3168: 2-OMe-4-S (O) Me-3-Py], [BG3169] : 5-OMe-4-S (O) Me-3-Py], [BG3170: 6-OMe-4-S (O) Me-3-Py], [BG3171: 5] -S (O) Me-3-Py], [BG3172: 2-Cl-5-S (O) Me-3-Py], [BG3173: 4-Cl-5-S (O) Me-3-Py ], [BG3174: 6-Cl-5-S (O) Me-3-Py], [BG3175: 2-Me-5-S (O) Me-3-Py], [BG3176: 4-Me-5] -S (O) Me-3- Py], [BG3177: 6-Me-5-S (O) Me-3-Py], [BG3178: 2-CF 3 -5-S (O) Me-3- Py], [BG3179: 4- CF 3 -5-S (O) Me-3-Py], [BG3180: 6-CF 3 -5-S (O) Me-3-Py], [BG3181: 2- CN-5-S (O) Me-3-Py], [BG3182: 4-CN-5-S (O) Me-3-Py], [BG3183: 6-CN-5-S (O) Me- 3-Py], [BG3184: 2-OMe-5-S (O) Me-3-Py], [BG3185: 4-OMe-5-S (O) Me-3-Py], [BG3186: 6- OMe-5-S (O) Me-3-Py], [BG3187: 6-S (O) Me-3-Py], [BG3188: 2-Cl-6-S (O) Me-3-Py] , [BG3189: 4-Cl-6-S (O) Me-3-Py], [BG3190: 5-Cl-6-S (O) Me-3-Py], [BG3191: 2-Me-6- 6 S (O) Me-3-Py], [BG3192: 4-Me-6-S (O) Me-3-Py], [BG3193: 5-Me-6-S (O) Me-3-Py] _{, [BG3194: 2-CF 3} -6-S (O) Me-3-Py], [BG3195: 4-CF 3 -6-S (O) Me-3-Py], [BG3196: 5-CF 3 -6-S (O) Me-3-Py], [BG3197: 2-CN-6-S (O) Me-3-Py], [BG3198: 4-CN-6-S (O) Me-3 -Py], [BG3199: 5-CN-6-S (O) Me-3-Py], [BG3200: 2-OMe-6-S (O) Me-3-Py],

[BG3201: 4-OMe-6-S (O) Me-3-Py], [BG3202: 5-OMe-6-S (O) Me-3-Py], [BG3203: 2-S (O) CF _{3 -3-Py], [BG3204} : 4-Cl-2-S (O) CF 3 -3-Py], [BG3205: 5-Cl-2-S (O) CF 3 -3-Py], [ BG3206: 6-Cl-2- S (O) CF 3 -3-Py], [BG3207: 4-Me-2-S (O) CF 3 -3-Py], [BG3208: 5-Me-2- _{S (O) CF 3 -3-} Py], [BG3209: 6-Me-2-S (O) CF 3 -3-Py], [BG3210: 4-CF 3 -2-S (O) CF 3 - 3-Py], [BG 3211: 5-CF ₃ -2-S (O) CF ₃ -3-Py], [BG 32 12: 6-CF ₃ -2-S (O) CF ₃ -3-Py], [BG 32 1 BG3213: 4-CN-2- S (O) CF 3 -3-Py], [BG3214: 5-CN-2-S (O) CF 3 -3-Py], [BG3215: 6-CN-2- _{S (O) CF 3 -3-} Py], [BG3216: 4-OMe-2-S (O) CF 3 -3-Py], [BG3217: 5-OMe-2-S (O) CF 3 -3 -Py], [BG3218: 6- OMe-2-S (O) CF 3 -3-Py], [BG3219: 4-S (O) CF 3 -3-Py], [BG3220: 2-Cl-4 _{-S (O) CF 3 -3-} Py], [BG3221: 5-Cl-4-S (O) CF 3 -3-Py], [BG3222: 6-Cl-4-S (O) CF 3 - 3-Py], [BG3223: 2-Me-4-S (O) CF 3 -3-Py], [BG3224: 5-Me-4-S (O) CF 3 -3-Py], [BG3225: 6-Me-4-S ( O) CF 3 -3-Py], [BG3226: 2-CF 3 -4-S (O) CF 3 -3-Py], [BG3227: 5-CF 3 -4- _{S (O) CF 3 -3-} Py], [BG3228: 6-CF 3 -4-S (O) CF 3 -3-Py], [BG3229: 2-CN-4-S (O) CF 3 - 3-Py], [BG3230: 5-CN-4-S (O) CF 3 -3-Py], [BG3231: 6-CN-4-S (O) CF 3 -3-Py], [BG3232: 2-OMe-4-S ( O) CF 3 -3-Py], [BG3233: 5-OMe-4 -S (O) CF 3 -3-Py], [BG3234: 6-OMe-4-S (O) CF 3 -3-Py], [BG3235: 5-S (O ) CF ₃ -3-Py !, [BG 3236: 2-Cl-5-S (O) CF ₃ -3-Py], [BG 3237: 4-Cl-5-S (O) CF ₃ -3-Py] , [BG3238: 6-Cl- 5-S (O) CF 3 -3-Py], [BG3239: 2-Me-5-S (O) CF 3 -3-Py], [BG3240: 4-Me- _{5-S (O) CF 3} -3-Py], [BG3241: 6-Me-5-S (O) CF 3 -3-Py], [BG3242: 2-CF 3 -5-S (O) CF _{3 -3-Py], [BG3243} : 4-CF 3 -5-S (O) CF 3 -3-Py], [BG3244: 6-CF 3 -5-S (O) CF 3 -3-Py] [BG 3245: 2-CN-5-S (O) CF ₃ -3-Py], [BG 3246: 4-CN-5-S (O) CF ₃ -3-Py], [BG 3247: 6-CN- _{5-S (O) CF 3} -3-Py], [BG3248: 2-OMe-5-S (O) CF 3 -3-Py], [BG3249: 4-OMe-5-S (O) CF 3 -3-Py !, [BG3 250: 6-OMe-5-S (O) CF ₃ -3-Py], [BG3251: 6-S (O) CF ₃ -3-Py], [BG3252: 2-Cl] _{-6-S (O) CF 3} -3-Py], [BG3253: 4-Cl-6-S (O) CF 3 -3-Py], [BG3254: 5-Cl-6-S (O) CF _{3 -3-Py], [BG3255} : 2-Me-6-S (O) CF 3 -3-Py], [BG3256: 4-Me-6-S (O) CF 3 -3-Py], [ BG3257: 5-Me-6- S (O) CF 3 -3-Py], [BG3258: 2-CF 3 -6-S (O) CF 3 -3-Py], [BG3259: 4-CF 3 - _{6-S (O) CF 3} -3-Py], [BG3260: 5-CF 3 -6-S (O) CF 3 -3-Py], [BG3261: 2-CN-6-S (O) CF _{3 -3-Py], [BG3262} : 4-CN-6-S (O) CF 3 -3-Py], [BG3263: 5-CN-6-S (O) CF 3 -3-Py], [ BG 3264: 2-OMe-6-S (O) CF _3- 3-Py], [BG3265: 4-OMe-6-S (O) CF 3 -3-Py], [BG3266: 5-OMe-6-S (O) CF 3 -3-Py], [BG3267: _{2-S (O) 2 Me} -3-Py], [BG3268: 4-Cl-2-S (O) 2 Me-3-Py], [BG3269: 5-Cl-2-S (O) 2 Me -3-Py !, [BG 3270: 6-Cl-2-S (O) ₂ Me-3-Py], [BG3271: 4-Me-2-S (O) ₂ Me-3-Py], [BG3272 : 5-Me-2-S (O) 2 Me-3-Py], [BG3273: 6-Me-2-S (O) 2 Me-3-Py], [BG3274: 4-CF 3 -2- _{S (O) 2 Me-3} -Py], [BG3275: 5-CF 3 -2-S (O) 2 Me-3-Py], [BG3276: 6-CF 3 -2-S (O) 2 Me -3-Py !, [BG3277: 4-CN-2-S (O) ₂ Me-3-Py], [BG3278: 5-CN-2-S (O) ₂ Me-3-Py], [BG3279] : 6-CN-2-S (O) 2 Me-3-Py], [BG3280: 4-OMe-2-S (O) 2 Me-3-Py], [BG3281: 5-OMe-2-S (O) ₂ Me-3-Py, [BG3282: 6-OMe-2-S (O) ₂ Me-3-Py], [BG 3283: 4-S (O) ₂ Me-3-Py], BG3284: 2-Cl-4- S (O) 2 Me-3-Py], [BG3285: 5-Cl-4-S (O) 2 Me-3-Py], [BG3286: 6-Cl-4- _{S (O) 2 Me-3} -Py], [BG3287: 2-Me-4-S (O) 2 Me-3-Py], [BG3288: 5-Me-4-S (O) 2 Me-3 -Py], [BG3289: 6- Me-4-S (O) 2 Me-3-Py], [BG3290: 2-CF 3 -4-S (O) 2 Me-3-Py], [BG3291: _{5-CF 3 -4-S (} O) 2 Me-3-Py], [BG3292: 6-CF 3 -4-S (O) 2 Me-3-Py], [BG3293: 2-CN-4- _{S (O) 2 Me-3} -Py], [BG3294: 5-CN-4-S (O) 2 Me-3-Py], [BG3295: 6-CN-4-S (O) 2 Me-3 -Py], [BG 3296: 2-OMe-4-S (O) ₂ Me-3-Py, [BG3297: 5-OMe-4-S (O) ₂ Me-3-Py], [BG3298: 6-OMe-4-S (O) ₂ Me-3-Py], [BG 3299: 5-S (O) ₂ Me-3-Py], [BG 3300: 2-Cl-5-S (O) ₂ Me-3-Py],

[BG3301: 4-Cl-5-S (O) ₂ Me-3-Py], [BG3302: 6-Cl-5-S (O) ₂ Me-3-Py], [BG3303: 2-Me-5 _{-S (O) 2 Me-3} -Py], [BG3304: 4-Me-5-S (O) 2 Me-3-Py], [BG3305: 6-Me-5-S (O) 2 Me- 3-Py], [BG3306: 2-CF 3 -5-S (O) 2 Me-3-Py], [BG3307: 4-CF 3 -5-S (O) 2 Me-3-Py], [ _{BG3308: 6-CF 3 -5-} S (O) 2 Me-3-Py], [BG3309: 2-CN-5-S (O) 2 Me-3-Py], [BG3310: 4-CN-5 _{-S (O) 2 Me-3} -Py], [BG3311: 6-CN-5-S (O) 2 Me-3-Py], [BG3312: 2-OMe-5-S (O) 2 Me- 3-Py], [BG3313: 4-OMe-5-S (O) 2 Me-3-Py], [BG3314: 6-OMe-5-S (O) 2 Me-3-Py], [BG3315: _{6-S (O) 2 Me} -3-Py], [BG3316: 2-Cl-6-S (O) 2 Me-3-Py], [BG3317: 4-Cl-6-S (O) 2 Me -3-Py !, [BG3318: 5-Cl-6-S (O) ₂ Me-3-Py], [BG3319: 2-Me-6-S (O) ₂ Me-3-Py], [BG3320] : 4-Me-6-S (O) 2 Me-3-Py], [BG3321: 5-Me-6-S (O) 2 Me-3-Py], [BG3322: 2-CF 3 -6- _{S (O) 2 Me-3} -Py], [BG3323: 4-CF 3 -6-S (O) 2 Me-3-Py], [BG3324: 5-CF 3 -6-S (O) 2 Me -3-Py], [BG3325: 2-CN-6-S (O) ₂ Me-3-Py], [BG3326: 4-CN-6-S (O) ₂ Me-3-Py], [BG3327 : 5-CN-6-S (O) 2 Me-3-Py], [BG3328: 2-OMe-6-S (O) 2 Me-3-Py], [BG3329: 4-OMe-6-S (O) ₂ Me-3-Py, [BG3330: 5-OMe-6-S (O) ₂ Me-3-Py], [BG333 1: 2-S (O) ₂ CF ₃ -3-Py], [BG3332: 4-Cl-2-S (O) _{2 CF 3 -3-Py], [} BG3333: 5-Cl-2-S (O) 2 CF 3 -3-Py], [BG3334: 6-Cl-2-S (O) 2 CF 3 -3-Py ], [BG3335: 4-Me -2-S (O) 2 CF 3 -3-Py], [BG3336: 5-Me-2-S (O) 2 CF 3 -3-Py], [BG3337: 6 -Me-2-S (O) 2 CF 3 -3-Py], [BG3338: 4-CF 3 -2-S (O) 2 CF 3 -3-Py], [BG3339: 5-CF 3 -2 _{-S (O) 2 CF 3 -3} -Py], [BG3340: 6-CF 3 -2-S (O) 2 CF 3 -3-Py], [BG3341: 4-CN-2-S (O) _{2 CF 3 -3-Py],} [BG3342: 5-CN-2-S (O) 2 CF 3 -3-Py], [BG3343: 6-CN-2-S (O) 2 CF 3 -3- Py], [BG3344: 4- OMe-2-S (O) 2 CF 3 -3-Py], [BG3345: 5-OMe-2-S (O) 2 CF 3 -3-Py], [BG3346: 6-OMe-2-S ( O) 2 CF 3 -3-Py], [BG3347: 4-S (O) 2 CF 3 -3-Py], [BG3348: 2-Cl-4-S (O) ₂ CF ₃ -3-Py, [BG 3 349: 5-Cl-4-S (O) ₂ CF ₃ -3-Py], [BG 3 350: 6-Cl-4-S (O) ₂ CF ₃ -3- Py], [BG3351: 2- Me-4-S (O) 2 CF 3 -3-Py], [BG3352: 5-Me-4-S (O) 2 CF 3 -3-Py], [BG3353: 6-Me-4-S ( O) 2 CF 3 -3-Py], [BG3354: 2-CF 3 -4-S (O) 2 CF 3 -3-Py], [BG3355: 5-CF 3 - _{4-S (O) 2 CF} 3 -3-Py], [BG3356: 6-CF 3 -4-S (O) 2 CF 3 -3-Py], [BG3357: 2-CN-4-S (O _{) 2 CF 3 -3-Py]} , [BG3358: 5-CN-4-S (O) 2 CF 3 -3-Py], [BG3359: 6-CN-4-S (O) 2 CF 3 -3 -Py], [BG3360: 2- OMe-4-S (O) 2 CF 3 -3-Py], [BG3361: 5-OMe-4-S (O _{) 2 CF 3 -3-Py]} , [BG3362: 6-OMe-4-S (O) 2 CF 3 -3-Py], [BG3363: 5-S (O) 2 CF 3 -3-Py], [BG3364: 2-Cl-5 -S (O) 2 CF 3 -3-Py], [BG3365: 4-Cl-5-S (O) 2 CF 3 -3-Py], [BG3366: 6-Cl _{-5-S (O) 2 CF} 3 -3-Py], [BG3367: 2-Me-5-S (O) 2 CF 3 -3-Py], [BG3368: 4-Me-5-S (O ) ₂ CF ₃ -3-Py], [BG 3369: 6-Me-5-S (O) ₂ CF ₃ -3-Py], [BG ₃ 370: 2-CF ₃ -5- S (O) ₂ CF _3- 3-Py], [BG3371: 4-CF 3 -5-S (O) 2 CF 3 -3-Py], [BG3372: 6-CF 3 -5-S (O) 2 CF 3 -3-Py] , [BG3373: 2-CN- 5-S (O) 2 CF 3 -3-Py], [BG3374: 4-CN-5-S (O) 2 CF 3 -3-Py], [BG3375: 6- CN-5-S (O) 2 CF 3 -3-Py], [BG3376: 2-OMe-5-S (O) 2 CF 3 -3-Py], [BG3377: 4-OMe-5-S ( O) ₂ CF ₃ -3-Py], [BG 3378: 6-OMe-5-S (O) ₂ CF ₃ -3-Py], [BG 3379: 6-S (O) ₂ CF ₃ -3- Py] , [BG3380: 2-Cl- 6-S (O) 2 CF 3 -3-Py], [BG3381: 4-Cl-6-S (O) 2 CF 3 -3-Py], [BG3382: 5- Cl-6-S (O) 2 CF 3 -3-Py], [BG3383: 2-Me-6-S (O) 2 CF 3 -3-Py], [BG3384: 4-Me-6-S ( O) ₂ CF ₃ -3-Py, [BG 3385: 5-Me-6-S (O) ₂ CF ₃ -3-Py], [BG 3386: 2-CF ₃ -6-S (O) ₂ CF ₃ -3-Py], [BG3387: 4-CF 3 -6-S (O) 2 CF 3 -3-Py], [BG3388: 5-CF 3 -6-S (O) 2 CF 3 -3-Py ], [BG3389: 2-CN -6-S (O) 2 CF 3 -3-Py], [BG3390: 4-CN-6-S (O) _{2 CF 3 -3-Py],} [BG3391: 5-CN-6-S (O) 2 CF 3 -3-Py], [BG3392: 2-OMe-6-S (O) 2 CF 3 -3- Py], [BG3393: 4- OMe-6-S (O) 2 CF 3 -3-Py], [BG3394: 5-OMe-6-S (O) 2 CF 3 -3-Py], [BG3395: 2-CN-3-Py !, [BG 3369: 4-Cl-2-CN-3-Py], [BG 3397: 5-Cl-2-CN-3-Py], [BG 3398: 6-Cl-2-] CN-3-Py !, [BG3399: 4-Me-2-CN-3-Py], [BG3400: 5-Me-2-CN-3-Py],

[BG3401: 6-Me-2 -CN-3-Py], [BG3402: 4-CF 3 -2-CN-3-Py], [BG3403: 5-CF 3 -2-CN-3-Py], _{[BG3404: 6-CF 3 -2} -CN-3-Py], [BG3405: 4-CN-2-CN-3-Py], [BG3406: 5-CN-2-CN-3-Py], [ BG3407: 6-CN-2-CN-3-Py !, [BG3408: 4-OMe-2-CN-3-Py], [BG3409: 5-OMe-2-CN-3-Py], [BG3410: 6-OMe-2-CN-3-Py, [BG 3411: 4-CN-3-Py], [BG 3412: 2-Cl-4-CN-3-Py], [BG 3413: 5-Cl-4- CN-3-Py !, [BG3414: 6-Cl-4-CN-3-Py], [BG3415: 2-Me-4-CN-3-Py], [BG3416: 5-Me-4-CN-] 3-Py], [BG3417: 6-Me-4-CN-3-Py], [BG3418: 2-CF 3 -4-CN-3-Py], [BG3419: 5-CF 3 -4-CN- 3-Py], [BG3420: 6-CF 3 -4-CN-3-Py], [BG3421: 2-CN-4-CN-3-Py], [BG3422: 5-CN-4-CN-3 -Py], [BG3423: 6-CN-4-CN-3-Py], [BG3424: 2-OMe-4-CN-3-Py], [BG3425: 5-OMe-4-CN-3-Py] ], [BG3426: 6-OMe-4-CN-3-Py], [BG3427: 5-CN-3-Py], [BG3428: 2-Cl-5-CN-3-Py], [BG3429: 4] -Cl-5-CN-3-Py], [BG3430: 6-Cl-5-CN-3-Py], [BG3431: 2-Me-5-CN-3-Py], [BG3432: 4-Me -5-CN-3-Py !, [BG 3433: 6-Me-5-CN-3-Py], [BG 3434: 2-CF ₃ -5-CN-3-Py], [BG 3435: 4-CF ₃ -5-CN-3-Py] , [BG3436: 6-CF 3 -5-CN-3-Py], [BG3437: 2-CN-5-CN-3-Py], [BG3438: 4-CN- 5-CN-3-Py, [BG3439: 6-CN-5-CN-3-Py], [BG3440: 2-OMe-5-CN-3-Py], [BG3441: 4-OMe-5-] CN-3-Py !, [BG3442: 6-OMe-5-CN-3-Py], [BG3443: 6-CN-3-Py], [BG3444: 2-Cl-6-CN-3-Py] , [BG3445: 4-Cl-6-CN-3-Py], [BG 3446: 5-Cl-6-CN-3-Py], [BG 3 447: 2-Me-6-CN-3-Py], [BG BG 3448: 4-Me-6-CN-3-Py !, [BG3449: 5-Me-6-CN-3-Py], [BG 3450: 2-CF ₃ -6-CN-3-Py], [BG3451] _{: 4-CF 3 -6-CN} -3-Py], [BG3452: 5-CF 3 -6-CN-3-Py], [BG3453: 2-CN-6-CN-3-Py], [BG3454 : 4-CN-6-CN-3-Py], [BG3455: 5-CN-6-CN-3-Py], [BG3456: 2-OMe-6-CN-3-Py], [BG3457: 4] -OMe-6-CN-3-Py], [BG3458: 5-OMe-6-CN-3-Py], [BG3459: 2-COOMe-3-Py], [BG3460: 4-Cl-2-COOMe -3-Py !, [BG3461: 5-Cl-2-COOMe-3-Py], [BG3462: 6-Cl-2-COOMe-3-Py], [BG3463: 4-Me-2-COOMe-3] -Py], [BG3464: 5- Me-2-COOMe-3-Py], [BG3465: 6-Me-2-COOMe-3-Py], [BG3466: 4-CF 3 -2-COOMe-3- Py], [BG3467: 5- CF 3 -2-COOMe-3-Py], [BG3468: 6-CF 3 -2-COOMe-3-Py], [BG3469: 4-CN-2-COOMe-3- Py], [BG3470: 5-CN-2-COOMe-3-Py], [BG3471: 6-CN-2-COOMe-3-Py], [BG3472: 4-OMe-2-COOMe-3-Py] , [BG3473: 5-OMe-2-COOMe-3-Py], [BG3474: 6-OMe-2-COOMe-3-Py], [BG3475: 4-COOMe-3-Py], [BG3476: 2- Cl-4-COOMe-3-Py], [BG3477: 5-Cl-4-COOMe-3-Py], [BG3478: 6-Cl-4-COOMe-3-Py], [BG3479: 2-Me- 4-COOMe-3-Py], [BG348 0: 5-Me-4- COOMe-3-Py], [BG3481: 6-Me-4-COOMe-3-Py], [BG3482: 2-CF 3 -4-COOMe-3-Py], [BG3483 _{: 5-CF 3 -4-COOMe} -3-Py], [BG3484: 6-CF 3 -4-COOMe-3-Py], [BG3485: 2-CN-4-COOMe-3-Py], [BG3486 : 5-CN-4-COOMe-3-Py], [BG3487: 6-CN-4-COOMe-3-Py], [BG3488: 2-OMe-4-COOMe-3-Py], [BG3489: 5] -OMe-4-COOMe-3-Py], [BG3490: 6-OMe-4-COOMe-3-Py], [BG3491: 5-COOMe-3-Py], [BG3492: 2-Cl-5-COOMe -3-Py], [BG3493: 4-Cl-5-COOMe-3-Py], [BG3494: 6-Cl-5-COOMe-3-Py], [BG3495: 2-Me-5-COOMe-3] -Py], [BG3496: 4- Me-5-COOMe-3-Py], [BG3497: 6-Me-5-COOMe-3-Py], [BG3498: 2-CF 3 -5-COOMe-3- Py], [BG3499: 4- CF 3 -5-COOMe-3-Py], [BG3500: 6-CF 3 -5-COOMe-3-Py],

[BG3501: 2-CN-5-COOMe-3-Py], [BG3502: 4-CN-5-COOMe-3-Py], [BG3503: 6-CN-5-COOMe-3-Py], [BG3504] : 2-OMe-5-COOMe-3-Py], [BG3505: 4-OMe-5-COOMe-3-Py], [BG3506: 6-OMe-5-COOMe-3-Py], [BG3507: 6] -COOMe-3-Py], [BG3508: 2-Cl-6-COOMe-3-Py], [BG3509: 4-Cl-6-COOMe-3-Py], [BG3510: 5-Cl-6-COOMe -3-Py !, [BG 351 1: 2 -Me-6-COOMe-3-Py], [BG3512: 4-Me-6-COOMe-3-Py], [BG3513: 5-Me-6-COOMe-3] -Py], [BG 3514: 2-CF ₃ -6-COOMe-3-Py], [BG 3515: 4-CF ₃ -6-COOMe-3-Py], [BG 3516: 5-CF ₃ -6-COOMe- 3-Py !, [BG3517: 2-CN-6-COOMe-3-Py], [BG3518: 4-CN-6-COOMe-3-Py], [BG3519: 5-CN-6-COOMe-3-] Py], [BG3520: 2-OMe-6-COOMe-3-Py], [BG3521: 4-OMe-6-COOMe-3-Py], [BG3522: 5-OMe-6-COOMe-3-Py] _{, [BG3523: 2-NO 2} -3-Py], [BG3524: 4-Cl-2-NO 2 -3-Py], [BG3525: 5-Cl-2-NO 2 -3-Py], [BG3526 : 6-Cl-2-NO 2 -3-Py], [BG3527: 4-Me-2-NO 2 -3-Py], [BG3528: 5-Me-2-NO 2 -3-Py], [ BG3529: 6-Me-2- NO 2 -3-Py], [BG3530: 4-CF 3 -2-NO 2 -3-Py], [BG3531: 5-CF 3 -2-NO 2 -3-Py ], [BG3532: 6-CF 3 -2-NO 2 -3-Py], [BG3533: 4-CN-2-NO 2 -3-Py], [BG3534: 5-CN-2-NO 2 -3 -Py], [BG3535: 6- CN-2-NO 2 -3-Py], [BG3536: 4-OMe-2-NO 2 -3-Py], [BG3537: 5-OMe _{-2-NO 2 -3-Py]} , [BG3538: 6-OMe-2-NO 2 -3-Py], [BG3539: 4-NO 2 -3-Py], [BG3540: 2-Cl-4- _{NO 2 -3-Py], [} BG3541: 5-Cl-4-NO 2 -3-Py], [BG3542: 6-Cl-4-NO 2 -3-Py], [BG3543: 2-Me-4 _{-NO 2 -3-Py], [} BG3544: 5-Me-4-NO 2 -3-Py], [BG3545: 6-Me-4-NO 2 -3-Py], [BG3546: 2-CF 3 -4-NO ₂ -3-Py, [BG 3547: 5-CF ₃ -4-NO ₂ -3-Py], [BG 3548: 6-CF ₃ -4-NO ₂ -3-Py], [BG 3 549: _{2-CN-4-NO 2} -3-Py], [BG3550: 5-CN-4-NO 2 -3-Py], [BG3551: 6-CN-4-NO 2 -3-Py], [BG3552 : 2-OMe-4-NO 2 -3-Py], [BG3553: 5-OMe-4-NO 2 -3-Py], [BG3554: 6-OMe-4-NO 2 -3-Py], [ _{BG3555: 5-NO 2 -3-} Py], [BG3556: 2-Cl-5-NO 2 -3-Py], [BG3557: 4-Cl-5-NO 2 -3-Py], [BG3558: 6 _{-Cl-5-NO 2 -3-} Py], [BG3559: 2-Me-5-NO 2 -3-Py], [BG3560: 4-Me-5-NO 2 -3-Py], [BG3561: _{6-Me-5-NO 2} -3-Py], [BG3562: 2-CF 3 -5-NO 2 -3-Py], [BG3563: 4-CF 3 -5-NO 2 -3-Py], _{[BG3564: 6-CF 3 -5} -NO 2 -3-Py], [BG3565: 2-CN-5-NO 2 -3-Py], [BG3566: 4-CN-5-NO 2 -3-Py ], [BG3567: 6-CN -5-NO 2 -3-Py], [BG3568: 2-OMe-5-NO 2 -3-Py], [BG3569: 4-OMe-5-NO 2 -3- Py], [BG3570: 6- OMe-5-NO 2 -3-Py], [BG3571: 6-NO 2 -3-Py], [BG3572: 2-Cl-6-NO 2 -3-Py], [BG3573: 4-Cl-6 -NO 2 -3-Py], [BG 3574: 5-Cl-6- NO 2 -3-Py], [BG3575: 2-Me-6-NO 2 -3-Py], [BG3576: 4-Me-6-NO 2 -3-Py], [BG3577: 5-Me-6 -NO 2 -3-Py], [BG3578: 2-CF 3 -6-NO 2 -3-Py], [BG3579: 4-CF 3 -6-NO 2 -3- Py], [BG3580: 5- CF 3 -6-NO 2 -3-Py], [BG3581: 2-CN-6-NO 2 -3-Py], [BG3582: 4-CN-6-NO 2 - 3-Py], [BG3583: 5-CN-6-NO 2 -3-Py], [BG3584: 2-OMe-6-NO 2 -3-Py], [BG3585: 4-OMe-6-NO 2 -3-Py], [BG3586: 5-OMe-6-NO 2 -3-Py], [BG3587: 2-NH 2 -3-Py], [BG3588: 4-Cl-2-NH 2 -3- Py], [BG3589: 5- Cl-2-NH 2 -3-Py], [BG3590: 6-Cl-2-NH 2 -3-Py], [BG3591: 4-Me-2-NH 2 -3 -Py], [BG3592: 5- Me-2-NH 2 -3-Py], [BG3593: 6-Me-2-NH 2 -3-Py], [BG3594: 4-CF 3 -2-NH 2 -3-Py], [BG3595: 5-CF ₃ -2-NH ₂ -3-Py], [BG 359: 6-CF ₃ -2-NH ₂ -3-Py], [BG 3 597: 4-CN-2 _{-NH 2 -3-Py], [} BG3598: 5-CN-2-NH 2 -3-Py], [BG3599: 6-CN-2-NH 2 -3-Py], [BG3600: 4-OMe- 2-NH ₂ -3-Py],

[BG3601: 5-OMe-2 -NH 2 -3-Py], [BG3602: 6-OMe-2-NH 2 -3-Py], [BG3603: 4-NH 2 -3-Py], [BG3604: _{2-Cl-4-NH 2} -3-Py], [BG3605: 5-Cl-4-NH 2 -3-Py], [BG3606: 6-Cl-4-NH 2 -3-Py], [BG3607 : 2-Me-4-NH 2 -3-Py], [BG3608: 5-Me-4-NH 2 -3-Py], [BG3609: 6-Me-4-NH 2 -3-Py], [ _{BG3610: 2-CF 3 -4-} NH 2 -3-Py], [BG3611: 5-CF 3 -4-NH 2 -3-Py], [BG3612: 6-CF 3 -4-NH 2 -3- Py], [BG3613: 2- CN-4-NH 2 -3-Py], [BG3614: 5-CN-4-NH 2 -3-Py], [BG3615: 6-CN-4-NH 2 -3 -Py], [BG3616: 2- OMe-4-NH 2 -3-Py], [BG3617: 5-OMe-4-NH 2 -3-Py], [BG3618: 6-OMe-4-NH 2 - 3-Py], [BG3619: 5-NH 2 -3-Py], [BG3620: 2-Cl-5-NH 2 -3-Py], [BG3621: 4-Cl-5-NH 2 -3-Py ], [BG3622: 6-Cl -5-NH 2 -3-Py], [BG3623: 2-Me-5-NH 2 -3-Py], [BG3624: 4-Me-5-NH 2 -3- Py], [BG3625: 6- Me-5-NH 2 -3-Py], [BG3626: 2-CF 3 -5-NH 2 -3-Py], [BG3627: 4-CF 3 -5-NH 2 -3-Py], [BG3628: 6-CF 3 -5-NH 2 -3-Py], [BG3629: 2-CN-5-NH 2 -3-Py], [BG3630: 4-CN-5- _{NH 2 -3-Py], [} BG3631: 6-CN-5-NH 2 -3-Py], [BG3632: 2-OMe-5-NH 2 -3-Py], [BG3633: 4-OMe-5 _{-NH 2 -3-Py], [} BG3634: 6-OMe-5-NH 2 -3-Py], [BG3635: 6-NH 2 -3-Py], [BG3636: 2-Cl-6-NH 2 -3-Py], [BG3637: 4-Cl-6-NH ₂ -3-Py !, [BG 3638: 5-Cl-6-NH ₂ -3-Py], [BG 3639: 2-Me-6-NH ₂ -3-Py], [BG 3640: 4-Me -6- _{NH 2 -3-Py], [} BG3641: 5-Me-6-NH 2 -3-Py], [BG3642: 2-CF 3 -6-NH 2 -3-Py], [BG3643: 4-CF 3 _{-6-NH 2 -3-Py]} , [BG3644: 5-CF 3 -6-NH 2 -3-Py], [BG3645: 2-CN-6-NH 2 -3-Py], [BG3646: 4 _{-CN-6-NH 2 -3-} Py], [BG3647: 5-CN-6-NH 2 -3-Py], [BG3648: 2-OMe-6-NH 2 -3-Py], [BG3649: _{4-OMe-6-NH 2} -3-Py], [BG3650: 5-OMe-6-NH 2 -3-Py], [BG3651: 2-NHMe-3-Py], [BG3652: 4-Cl- 2-NHMe-3-Py, [BG3653: 5-Cl-2-NHMe-3-Py], [BG3654: 6-Cl-2-NHMe-3-Py], [BG3 655: 4-Me-2-] NHMe-3-Py], [ BG3656: 5-Me-2-NHMe-3-Py], [BG3657: 6-Me-2-NHMe-3-Py], [BG3658: 4-CF 3 -2-NHMe -3-Py], [BG3659: 5-CF 3 -2-NHMe-3-Py], [BG3660: 6-CF 3 -2-NHMe-3-Py], [BG3661: 4-CN-2-NHMe -3-Py !, [BG3662: 5-CN-2-NHMe-3-Py], [BG3663: 6-CN-2-NHMe-3-Py], [BG3664: 4-OMe-2-NHMe-3] -Py], [BG3665: 5-OMe-2-NHMe-3-Py], [BG3666: 6-OMe-2-NHMe-3-Py], [BG3667: 4-NHMe-3-Py], [BG3668] : 2-Cl-4-NHMe-3-Py], [BG3669: 5-Cl-4-NHMe-3-Py], [BG3670: 6-Cl-4-NHMe-3-Py], [BG367 1: 2] -Me-4-NHMe-3-Py], [BG3672: 5-Me-4-NHMe-3-Py], [BG3673: 6-Me-4-NHMe-3-Py], [BG3674: 2-CF ₃ -4-NHMe-3-Py ], [BG3675: 5-CF 3 -4-NHMe-3-Py], [BG3676: 6-CF 3 -4-NHMe-3-Py], [BG3677: 2-CN-4-NHMe-3-Py ], [BG3678: 5-CN-4-NHMe-3-Py], [BG3679: 6-CN-4-NHMe-3-Py], [BG3680: 2-OMe-4-NHMe-3-Py], [BG3681: 5-OMe-4-NHMe-3-Py], [BG3682: 6-OMe-4-NHMe-3-Py], [BG3683: 5-NHMe-3-Py], [BG3684: 2-Cl2 -5-NHMe-3-Py !, [BG 3685: 4-Cl-5-NHMe-3-Py], [BG 3686: 6-Cl-5-NHMe-3-Py], [BG 3687: 2-Me-5] -NHMe-3-Py], [ BG3688: 4-Me-5-NHMe-3-Py], [BG3689: 6-Me-5-NHMe-3-Py], [BG3690: 2-CF 3 -5- NHMe-3-Py], [ BG3691: 4-CF 3 -5-NHMe-3-Py], [BG3692: 6-CF 3 -5-NHMe-3-Py], [BG3693: 2-CN-5- NHMe-3-Py, [BG3694: 4-CN-5-NHMe-3-Py], [BG3695: 6-CN-5-NHMe-3-Py], [BG3696: 2-OMe-5-NHMe- 3-Py], [BG 3697: 4-OMe-5-NHMe-3-Py], [BG 3698: 6-OMe-5-NHMe-3-Py], [BG 3699: 6-NHMe-3-Py], [BG BG 3700: 2-Cl-6-NHMe-3-Py],

[BG3701: 4-Cl-6-NHMe-3-Py], [BG3702: 5-Cl-6-NHMe-3-Py], [BG3703: 2-Me-6-NHMe-3-Py], [BG3704] : 4-Me-6-NHMe -3-Py], [BG3705: 5-Me-6-NHMe-3-Py], [BG3706: 2-CF 3 -6-NHMe-3-Py], [BG3707: _{4-CF 3 -6-NHMe-} 3-Py], [BG3708: 5-CF 3 -6-NHMe-3-Py], [BG3709: 2-CN-6-NHMe-3-Py], [BG3710: 4-CN-6-NHMe-3-Py, [BG3711: 5-CN-6-NHMe-3-Py], [BG3712: 2-OMe-6-NHMe-3-Py], [BG3713: 4- OMe-6-NHMe-3- Py], [BG3714: 5-OMe-6-NHMe-3-Py], [BG3715: 2-NMe 2 -3-Py], [BG3716: 4-Cl-2-NMe _{2 -3-Py], [BG3717} : 5-Cl-2-NMe 2 -3-Py], [BG3718: 6-Cl-2-NMe 2 -3-Py], [BG3719: 4-Me-2- _{NMe 2 -3-Py], [} BG3720: 5-Me-2-NMe2-3-Py], [BG3721: 6-Me-2-NMe2-3-Py], [BG3722: 4-CF 3 -2- NMe2-3-Py], [BG3723: 5-CF 3 -2-NMe 2 -3-Py], [BG3724: 6-CF 3 -2-NMe 2 -3-Py], [BG3725: 4-CN- _{2-NMe 2 -3-Py]} , [BG3726: 5-CN-2-NMe 2 -3-Py], [BG3727: 6-CN-2-NMe 2 -3-Py], [BG3728: 4-OMe _{-2-NMe 2 -3-Py]} , [BG3729: 5-OMe-2-NMe 2 -3-Py], [BG3730: 6-OMe-2-NMe 2 -3-Py], [BG3731: 4- _{NMe 2 -3-Py], [} BG3732: 2-Cl-4-NMe 2 -3-Py], [BG3733: 5-Cl-4-NMe 2 -3-Py], [BG3734: 6-Cl-4 _{-NMe 2 -3-Py], [} BG3735: 2-Me-4-NMe 2 -3-Py], [BG3736: 5-Me-4-NMe 2 -3-Py], [BG3737: 6-Me -4-NMe ₂ -3-Py !, [BG 3738: 2-CF ₃ -4-NMe ₂ -3-Py], [BG 3739: 5-CF ₃ -4-NMe ₂ -3-Py], [BG 3740: _{6-CF 3 -4-NMe 2} -3-Py], [BG3741: 2-CN-4-NMe 2 -3-Py], [BG3742: 5-CN-4-NMe 2 -3-Py], [ BG3743: 6-CN-4- NMe 2 -3-Py], [BG3744: 2-OMe-4-NMe 2 -3-Py], [BG3745: 5-OMe-4-NMe 2 -3-Py], [BG3746: 6-OMe-4 -NMe 2 -3-Py], [BG3747: 5-NMe 2 -3-Py], [BG3748: 2-Cl-5-NMe 2 -3-Py], [BG3749: _{4-Cl-5-NMe 2} -3-Py], [BG3750: 6-Cl-5-NMe 2 -3-Py], [BG3751: 2-Me-5-NMe 2 -3-Py], [BG3752 : 4-Me-5-NMe 2 -3-Py], [BG3753: 6-Me-5-NMe 2 -3-Py], [BG3754: 2-CF 3 -5-NMe 2 -3-Py], _{[BG3755: 4-CF 3 -5} -NMe 2 -3-Py], [BG3756: 6-CF 3 -5-NMe 2 -3-Py], [BG3757: 2-CN-5-NMe 2 -3- Py], [BG 3758: 4-CN-5-NMe ₂ 3-Py], [BG 3759: 6-CN-5-NMe ₂ 3-Py], [BG 3760: 2-OMe-5-NMe _2-3] -Py], [BG3761: 4- OMe-5-NMe 2 -3-Py], [BG3762: 6-OMe-5-NMe 2 -3-Py], [BG3763: 6-NMe 2 -3-Py] , [BG3764: 2-Cl- 6-NMe 2 -3-Py], [BG3765: 4-Cl-6-NMe 2 -3-Py], [BG3766: 5-Cl-6-NMe 2 -3-Py ], [BG3767: 2-Me -6-NMe 2 -3-Py], [BG3768: 4-Me-6-NMe 2 -3-Py], [BG3769: 5-Me-6-NMe 2 -3- Py], [BG3770: 2- CF 3 -6-NMe 2 -3-Py], [BG3771: 4-CF 3 -6-NMe 2 -3-Py], [BG3772: 5-CF _{3 -6-NMe 2 -3-Py} ], [BG3773: 2-CN-6-NMe 2 -3-Py], [BG3774: 4-CN-6-NMe 2 -3-Py], [BG3775: 5 _{-CN-6-NMe 2 -3-} Py], [BG3776: 2-OMe-6-NMe 2 -3-Py], [BG3777: 4-OMe-6-NMe 2 -3-Py], [BG3778: _{5-OMe-6-NMe 2} -3-Py], [BG3779: 2-ACNH-3-Py], [BG3780: 4-Cl-2-ACNH-3-Py], [BG3781: 5-Cl-2 -ACNH-3-Py, [BG3782: 6-Cl-2-ACNH-3-Py], [BG3783: 4-Me-2-ACNH-3-Py], [BG3784: 5-Me-2-ACNH] -3-Py], [BG3785: 6-Me-2-ACNH-3-Py], [BG3786: 4-CF 3 -2-ACNH-3-Py], [BG3787: 5-CF 3 -2-ACNH -3-Py], [BG3788: 6-CF 3 -2-ACNH-3-Py], [BG3789: 4-CN-2-ACNH-3-Py], [BG3790: 5-CN-2-ACNH- 3-Py], [BG3791: 6-CN-2-ACNH-3-Py], [BG3792: 4-OMe-2-ACNH-3-Py], [BG3793: 5-OMe-2-ACNH-3- Py], [BG3794: 6-OMe-2-ACNH-3-Py], [BG3795: 4-ACNH-3-Py], [BG3796: 2-Cl-4-ACNH-3-Py], [BG3797: 5-Cl-4-ACNH-3-Py, [BG3798: 6-Cl-4-ACNH-3-Py], [BG3799: 2-Me-4-ACNH-3-Py], [BG3800: 5-] Me-4-ACNH-3-Py],

[BG3801: 6-Me-4 -ACNH-3-Py], [BG3802: 2-CF 3 -4-ACNH-3-Py], [BG3803: 5-CF 3 -4-ACNH-3-Py], _{[BG3804: 6-CF 3 -4} -ACNH-3-Py], [BG3805: 2-CN-4-ACNH-3-Py], [BG3806: 5-CN-4-ACNH-3-Py], [ BG3807: 6-CN-4-ACNH-3-Py !, [BG3808: 2-OMe-4-ACNH-3-Py], [BG3809: 5-OMe-4-ACNH-3-Py], [BG3810: 6-OMe-4-ACNH-3-Py !, [BG3811: 5-ACNH-3-Py], [BG3812: 2-Cl-5-ACNH-3-Py], [BG3813: 4-Cl-5-] ACNH-3-Py, [BG3814: 6-Cl-5-ACNH-3-Py], [BG3815: 2-Me-5-ACNH-3-Py], [BG3816: 4-Me-5-ACNH- 3-Py], [BG3817: 6-Me-5-ACNH-3-Py], [BG3818: 2-CF 3 -5-ACNH-3-Py], [BG3819: 4-CF 3 -5-ACNH- 3-Py], [BG3820: 6-CF 3 -5-ACNH-3-Py], [BG3821: 2-CN-5-ACNH-3-Py], [BG3822: 4-CN-5-ACNH-3 -Py], [BG3823: 6-CN-5-ACNH-3-Py], [BG3824: 2-OMe-5-ACNH-3-Py], [BG3825: 4-OMe-5-ACNH-3-Py] ], [BG3826: 6-OMe-5-ACNH-3-Py], [BG3827: 6-ACNH-3-Py], [BG3828: 2-Cl-6-ACNH-3-Py], [BG3829: 4] -Cl-6-ACNH-3-Py], [BG3830: 5-Cl-6-ACNH-3-Py], [BG3831: 2-Me-6-ACNH-3-Py], [BG3832: 4-Me -6-ACNH-3-Py] , [BG3833: 5-Me-6-ACNH-3-Py], [BG3834: 2-CF 3 -6-ACNH-3-Py], [BG3835: 4-CF 3 -6-ACNH-3-Py], [BG 3836: 5-CF ₃ -6-ACNH-3-Py], [BG 3837: 2-CN-6-ACNH-3-Py], [BG 3838: 4-CN- 6- ACNH-3-Py, [BG3839: 5-CN-6-ACNH-3-Py], [BG3840: 2-OMe-6-ACNH-3-Py], [BG3841: 4-OMe-6-ACNH- 3-Py], [BG3842: 5-OMe-6-ACNH-3-Py], [BG3843: 2- (N (Ac) (Me))-3-Py], [BG3844: 4-Cl-2-] (N (Ac) (Me))-3-Py], [BG3845: 5-Cl-2- (N (Ac) (Me))-3-Py], [BG 3846: 6-Cl-2- (N) (Ac) (Me))-3-Py], [BG3847: 4-Me-2- (N (Ac) (Me))-3-Py], [BG3848: 5-Me-2- (N (Ac) ) (Me))-3-Py], [BG3849: 6-Me-2- (N (Ac) (Me))-3-Py], [BG3850: 4-CF ₃ -2- (N (Ac)) (Me))-3-Py], [BG3851: 5-CF ₃ -2- (N (Ac) (Me))-3-Py], [BG3852: 6-CF ₃ -2- (N (Ac)) (Me))-3-Py], [BG3853: 4-CN-2- (N (Ac) (Me))-3-Py], [BG3854: 5-CN-2- (N (Ac) (Me) )) [3-Py], [BG3855: 6-CN-2- (N (Ac) (Me))-3-Py], [BG3856: 4-OMe-2- (N (Ac) (Me))] -3-Py], [BG3857: 5-OMe-2- (N (Ac) (Me))-3-Py], [BG3858: 6-OMe-2- (N (Ac) (Me))-3] -Py], [BG 3859: 4- (N (Ac) (Me))-3-Py], [BG3860: 2-Cl-4- (N (Ac) (Me))-3-Py], [BG3861 : 5-Cl-4- (N (Ac) (Me))-3-Py], [BG3862: 6-Cl-4- (N (Ac) (Me))-3-Py], [BG3863: 2] -Me-4- (N (Ac) (Me))-3-Py], [BG3864: 5-Me-4- (N (Ac) (Me))-3-Py], [BG3865: 6-Me -4- (N (Ac) (Me )) - 3-Py], [BG3866: 2-CF 3 -4- (N (Ac) (Me)) - 3-Py], [BG3867: 5-CF 3 -4- (N (Ac) (Me )) - 3-Py], [BG3868: 6-CF 3 -4- (N (Ac) (Me)) - 3-Py], [BG3869: 2-CN- 4- (N (Ac) (Me))-3-Py], [BG3870: 5-CN-4- (N (Ac) (Me))-3-Py], [BG 3871: 6-CN-4- (N (Ac) (Me))-3-Py], [BG3872: 2-OMe-4- (N (Ac) (Me))-3-Py], [BG3873: 5-OMe-4- (N) (Ac) (Me))-3-Py], [BG3874: 6-OMe-4- (N (Ac) (Me))-3-Py], [BG3875: 5- (N (Ac) (Me)] )-[3-Py], [BG3876: 2-Cl-5- (N (Ac) (Me))-3-Py], [BG3877: 4-Cl-5- (N (Ac) (Me))- 3-Py], [BG3878: 6-Cl-5- (N (Ac) (Me))-3-Py], [BG3879: 2-Me-5- (N (Ac) (Me))-3-] Py], [BG3 880: 4-Me-5- (N (Ac) (Me))-3-Py], [BG3881: 6-Me-5- (N (Ac) (Me))-3-Py] _{, [BG3882: 2-CF 3} -5- (N (Ac) (Me)) - 3-Py], [BG3883: 4-CF 3 -5- (N (Ac) (Me)) - 3-Py] [BG 3884: 6-CF ₃ -5- (N (Ac) (Me)) -3-Py], [BG 3885: 2-CN -5- (N (Ac) (Me)) -3-Py], [BG 3886: 4-CN-5- (N (Ac) (Me))-3-Py], [BG3887: 6-CN-5- (N (Ac) (Me))-3-Py], [BG3888 : 2-OMe-5- (N (Ac) (Me))-3-Py], [BG3889: 4-OMe-5- (N (Ac) (Me))-3-Py], [BG 3890: 6 -OMe-5- (N (Ac) (Me))-3-Py], [BG3891: 6- (N (Ac) (Me))-3-Py], [BG3892: 2-Cl-6- ( N (Ac) (Me))-3-Py], [BG3893: 4-Cl-6- (N (Ac) (Me))-3-Py], [BG3894: 5-Cl-6- (N ( Ac) (Me))-3-Py], [BG3895: 2-Me-6- (N (Ac) (Me))-3-Py], [BG3896: 4-Me-6- (N (Ac)) (Me)) - 3-Py ], [BG3897: 5-Me-6- (N (Ac) (Me)) - 3-Py], [BG3898: 2-CF 3 -6- (N (Ac) ( Me))-3-Py], [BG 3899: 4-CF ₃ -6- (N (Ac) (Me))-3-Py], [BG 3900: 5-CF ₃ -6- (N (Ac) (Me))-3-Py],

[BG3901: 2-CN-6- (N (Ac) (Me))-3-Py], [BG3902: 4-CN-6- (N (Ac) (Me))-3-Py], [BG3903 : 5-CN-6- (N (Ac) (Me))-3-Py], [BG 3904: 2-OMe-6- (N (Ac) (Me))-3-Py], [BG 3905: 4] -OMe-6- (N (Ac) (Me))-3-Py], [BG 3906: 5-OMe-6- (N (Ac) (Me))-3-Py], [BG 3907: 2-AC -3-Py], [BG3908: 4-Cl-2-AC-3-Py], [BG3909: 5-Cl-2-AC-3-Py], [BG3910: 6-Cl-2-AC-3] -Py], [BG3911: 4-Me-2-AC-3-Py], [BG3912: 5-Me-2-AC-3-Py], [BG3913: 6-Me-2-AC-3-Py] ], [BG3914: 4-CF 3 -2-AC-3-Py], [BG3915: 5-CF 3 -2-AC-3-Py], [BG3916: 6-CF 3 -2-AC-3- Py], [BG3917: 4-CN-2-AC-3-Py], [BG3918: 5-CN-2-AC-3-Py], [BG3919: 6-CN-2-AC-3-Py] , [BG3920: 4-OMe-2-AC-3-Py], [BG3921: 5-OMe-2-AC-3-Py], [BG3922: 6-OMe-2-AC-3-Py], BG3923: 4-AC-3-Py, [BG3924: 2-Cl-4-AC-3-Py], [BG3925: 5-Cl-4-AC-3-Py], [BG3926: 6-Cl- 4-AC-3-Py, [BG3 927: 2-Me-4-AC-3-Py], [BG3928: 5-Me-4-AC-3-Py], [BG3 929: 6-Me-4-] AC-3-Py], [ BG3930: 2-CF 3 -4-AC-3-Py], [BG3931: 5-CF 3 -4-AC-3-Py], [BG3932: 6-CF 3 -4 -AC-3-Py, [BG3933: 2-CN-4-AC-3-Py], [BG3934: 5-CN-4-AC-3-Py], [BG3935: 6-CN-4-AC -3-Py !, [BG 3936: 2-OMe-4-AC-3-Py], [BG 3937: 5-OMe-4-AC-3-Py], [BG 3938: 6-OMe-4-AC-3] -Py], [BG 3939: 5-AC-3-Py ], [BG3940: 2-Cl-5-AC-3-Py], [BG 3941: 4-Cl-5-AC-3-Py], [BG3942: 6-Cl-5-AC-3-Py], [BG3943: 2-Me-5-AC-3-Py], [BG3944: 4-Me-5-AC-3-Py], [BG3945: 6-Me-5-AC-3-Py], [BG3946] _{: 2-CF 3 -5-AC} -3-Py], [BG3947: 4-CF 3 -5-AC-3-Py], [BG3948: 6-CF 3 -5-AC-3-Py], [ BG3949: 2-CN-5-AC-3-Py, [BG3950: 4-CN-5-AC-3-Py], [BG3951: 6-CN-5-AC-3-Py], [BG3952: 2-OMe-5-AC-3-Py], [BG3953: 4-OMe-5-AC-3-Py], [BG3954: 6-OMe-5-AC-3-Py], [BG3 955: 6- AC-3-Py], [BG 3 965: 2-Cl-6-AC-3-Py], [BG 3 957: 4-Cl-6-AC-3-Py], [BG 39 58: 5-Cl-6-AC- 3-Py], [BG3959: 2-Me-6-AC-3-Py], [BG 3960: 4-Me-6-AC-3-Py], [BG3961: 5-Me-6-AC-3- 3 Py], [BG3962: 2- CF 3 -6-AC-3-Py], [BG3963: 4-CF 3 -6-AC-3-Py], [BG3964: 5-CF 3 -6-AC-3 -Py], [BG3965: 2-CN-6-AC-3-Py], [BG 3966: 4-CN-6-AC-3-Py], [BG3967: 5-CN-6-AC-3-Py] ], [BG 3968: 2-OMe-6-AC-3-Py], [BG 3969: 4-OMe-6-AC-3-Py], [BG 3 970: 5-OMe-6-AC-3-Py], [BG 3971: 4-Py], [BG 3 972: 3-F-4-Py], [BG 3 973: 2-Cl-3-F-4-Py], [BG 3 974: 5-Cl-3-F-4-Py] ], [BG3975: 6-Cl-3-F-4-Py], [BG3976: 2-Me-3-F-4-Py], [BG3977: 5-Me-3-F-4-Py], [BG3978: 6-Me-3 -F-4-Py], [BG3979: 2-CF 3 -3-F-4-Py], [BG3980: 5-CF 3 -3-F-4-Py], [BG 3981: 6-CF ₃ -3-F-4-Py !, [BG3982: 2-CN-3-F-4-Py], [BG3983: 5-CN-3-F-4-Py], [BG3984: 6-CN- 3-F-4-Py, [BG 3985: 2-OMe-3-F-4-Py], [BG 3986: 5-OMe-3-F-4-Py], [BG 3 987: 6-OMe-3- F-4-Py], [BG3988: 2-F-4-Py], [BG3989: 3-Cl-2-F-4-Py], [BG3 990: 5-Cl-2-F-4-Py] , [BG3991: 6-Cl-2-F-4-Py], [BG3992: 3-Me-2-F-4-Py], [BG3993: 5-Me-2-F-4-Py], [BG3993: 5-Me-2-F-4-Py], BG3994: 6-Me-2- F-4-Py], [BG3995: 3-CF 3 -2-F-4-Py], [BG3996: 5-CF 3 -2-F-4-Py], [ BG ₃ 997: 6-CF ₃ -2-F-4-Py !, [BG3998: 3-CN-2-F-4-Py], [BG 3 999: 5-CN-2-F-4-Py], [BG 4000] : 6-CN-2-F-4-Py],

[BG4001: 3-OMe-2-F-4-Py], [BG4002: 5-OMe-2-F-4-Py], [BG4003: 6-OMe-2-F-4-Py], [BG4004] : 5-F-4-Py], [BG4005: 3-Cl-5-F-4-Py], [BG4006: 2-Cl-5-F-4-Py], [BG4007: 6-Cl-5] -F-4-Py], [BG4008: 3-Me-5-F-4-Py], [BG4009: 2-Me-5-F-4-Py], [BG4010: 6-Me-5-F -4-Py], [BG4011: 3-CF 3 -5-F-4-Py], [BG4012: 2-CF 3 -5-F-4-Py], [BG4013: 6-CF 3 -5- F-4-Py !, [BG4014: 3-CN-5-F-4-Py], [BG4015: 2-CN-5-F-4-Py], [BG4016: 6-CN-5-F- 4-Py], [BG4017: 3-OMe-5-F-4-Py], [BG4018: 2-OMe-5-F-4-Py], [BG4019: 6-OMe-5-F-4- 4 Py], [BG4020: 6-F-4-Py], [BG4021: 3-Cl-6-F-4-Py], [BG4022: 2-Cl-6-F-4-Py], [BG4023: 5-Cl-6-F-4-Py], [BG4024: 3-Me-6-F-4-Py], [BG4025: 2-Me-6-F-4-Py], [BG 4026: 5- Me-6-F-4- Py], [BG4027: 3-CF 3 -6-F-4-Py], [BG4028: 2-CF 3 -6-F-4-Py], [BG4029: 5- _{CF 3 -6-F-4-} Py], [BG4030: 3-CN-6-F-4-Py], [BG4031: 2-CN-6-F-4-Py], [BG4032: 5-CN -6-F-4-Py], [BG4033: 3-OMe-6-F-4-Py], [BG4034: 2-OMe-6-F-4-Py], [BG4035: 5-OMe-6] -F-4-Py], [BG4036: 3-Cl-4-Py], [BG4037: 2-Cl-3-Cl-4-Py], [BG4038: 5-Cl-3-Cl-4-Py] ], [BG4039: 6-Cl-3-Cl-4-Py], [BG4040: 2-Me-3-Cl-4-Py], [BG4041: 5-Me-3-Cl-4-Py], [BG4042: 6-Me-3 -Cl-4-Py], [BG4043: 2-CF 3 -3-Cl-4-Py] , [BG4044: 5-CF 3 -3-Cl-4-Py], [BG4045: 6-CF 3 -3-Cl-4-Py], [BG4046: 2-CN -3-Cl-4-Py !, [BG4047: 5-CN-3-Cl-4-Py], [BG4048: 6-CN-3-Cl-4-Py], [BG4049: 2-OMe-3] -Cl-4-Py], [BG4050: 5-OMe-3-Cl-4-Py], [BG4051: 6-OMe-3-Cl-4-Py], [BG4052: 2-Cl-4-Py] ], [BG4053: 3-Cl-2-Cl-4-Py], [BG4054: 5-Cl-2-Cl-4-Py], [BG4055: 6-Cl-2-Cl-4-Py], [BG 4056: 3-Me-2-Cl-4-Py], [BG4057: 5-Me-2-Cl-4-Py], [BG4058: 6-Me-2-Cl-4-Py], [BG4059] _{: 3-CF 3 -2-Cl} -4-Py], [BG4060: 5-CF 3 -2-Cl-4-Py], [BG4061: 6-CF 3 -2-Cl-4-Py], [ BG4062: 3-CN-2-Cl-4-Py, [BG4063: 5-CN-2-Cl-4-Py], [BG4064: 6-CN-2-Cl-4-Py], [BG4065: 3-OMe-2-Cl-4-Py], [BG 4066: 5-OMe-2-Cl-4-Py], [BG4067: 6-OMe-2-Cl-4-Py], [BG 4068: 5-] Cl-4-Py], [BG4069: 2-Cl-5-Cl-4-Py], [BG4070: 5-Cl-5-Cl-4-Py], [BG4071: 6-Cl-5-Cl- 4-Py], [BG4072: 2-Me-5-Cl-4-Py], [BG4073: 5-Me-5-Cl-4-Py], [BG4074: 6-Me-5-Cl-4-] Py], [BG4075: 2- CF 3 -5-Cl-4-Py], [BG4076: 5-CF 3 -5-Cl-4-Py], [BG4077: 6-CF 3 -5-Cl-4 -Py], [BG4078: 2-CN-5-Cl-4-Py], [BG4079: 3-CN-5-Cl-4-Py], [BG4080: 6-CN-5-Cl-4-Py] ], [BG4081: 2-OMe-5-Cl-4-Py], [BG4082: 5-OMe-5-Cl-4-Py], [BG4083: 6-OMe-5-Cl-4-Py], [BG40 84: 6-Cl-4-Py], [BG4085: 3-Cl-6-Cl-4-Py], [BG4086: 2-Cl-6-Cl-4-Py], [BG4087: 5-Cl- 6-Cl-4-Py, [BG4088: 3-Me-6-Cl-4-Py], [BG4089: 2-Me-6-Cl-4-Py], [BG4090: 5-Me-6-6] Cl-4-Py], [ BG4091: 3-CF 3 -6-Cl-4-Py], [BG4092: 2-CF 3 -6-Cl-4-Py], [BG4093: 5-CF 3 -6 -Cl-4-Py], [BG4094: 3-CN-6-Cl-4-Py], [BG4095: 2-CN-6-Cl-4-Py], [BG4096: 5-CN-6-Cl] -4-Py !, [BG4097: 3-OMe-6-Cl-4-Py], [BG4098: 2-OMe-6-Cl-4-Py], [BG4099: 5-OMe-6-Cl-4] -Py], [BG4100: 3-Br-4-Py],

[BG410 1: 2-Cl-3-Br-4-Py], [BG 4102: 5-Cl-3-Br-4-Py], [BG 4103: 6-Cl-3- Br-4-Py], [BG 4 104 : [2-Me-3-Br-4-Py], [BG4105: 5-Me-3-Br-4-Py], [BG4106: 6-Me-3-Br-4-Py], [BG4107: 2] _{-CF 3 -3-Br-4-} Py], [BG4108: 5-CF 3 -3-Br-4-Py], [BG4109: 6-CF 3 -3-Br-4-Py], [BG4110: 2-CN-3-Br-4-Py], [BG4111: 5-CN-3-Br-4-Py], [BG4112: 6-CN-3-Br-4-Py], [BG4113: 2- OMe-3-Br-4-Py], [BG4114: 5-OMe-3-Br-4-Py], [BG4115: 6-OMe-3-Br-4-Py], [BG4116: 2-Br- 4-Py], [BG4117: 3-Cl-2-Br-4-Py], [BG4118: 5-Cl-2-Br-4-Py], [BG4119: 6-Cl-2-Br-4-] Py], [BG 4120: 3-Me-2-Br-4-Py], [BG 4121: 5-Me-2-Br-4-Py], [BG 4122: 6-Me-2-Br-4-Py] _{, [BG4123: 3-CF 3} -2-Br-4-Py], [BG4124: 5-CF 3 -2-Br-4-Py], [BG4125: 6-CF 3 -2-Br-4-Py ], [BG4126: 3-CN-2-Br-4-Py], [BG4127: 5-CN-2-Br-4-Py], [BG4128: 6-CN-2-Br-4-Py], [BG4129: 3-OMe-2-Br-4-Py], [BG4130: 5-OMe-2-Br-4-Py], [BG4131: 6-OMe-2-Br-4-Py], [BG4132] : 5-Br-4-Py], [BG4133: 3-Cl-5-Br-4-Py], [BG4134: 2-Cl-5-Br-4-Py], [BG4135: 6-Cl-5] -Br-4-Py], [BG4136: 3-Me-5-Br-4-Py], [BG4137: 2-Me-5-Br-4-Py], [BG4138: 6-Me-5-Br] -4-Py], [BG4139: 3-CF 3 -5-Br-4-Py], [BG4140: 2-CF 3 -5-Br-4-Py], [BG4141: 6-CF 3 -5- Br -4-Py], [BG4142: 3-CN-5-Br-4-Py], [BG4143: 2-CN-5-Br-4-Py], [BG4144: 6-CN-5-Br-4] -Py], [BG4145: 3-OMe-5-Br-4-Py], [BG4146: 2-OMe-5-Br-4-Py], [BG4147: 6-OMe-5-Br-4-Py] ], [BG4148: 6-Br-4-Py], [BG4149: 3-Cl-6-Br-4-Py], [BG4150: 2-Cl-6-Br-4-Py], [BG4151: 5] -Cl-6-Br-4-Py], [BG4152: 3-Me-6-Br-4-Py], [BG4153: 2-Me-6-Br-4-Py], [BG4154: 5-Me -6-Br-4-Py] , [BG4155: 3-CF 3 -6-Br-4-Py], [BG4156: 2-CF 3 -6-Br-4-Py], [BG4157: 5-CF _{3 -6-Br-4-Py} ], [BG4158: 3-CN-6-Br-4-Py], [BG4159: 2-CN-6-Br-4-Py], [BG4160: 5-CN- 6-Br-4-Py !, [BG4161: 3-OMe-6-Br-4-Py], [BG4162: 2-OMe-6-Br-4-Py], [BG4163: 5-OMe-6-] Br-4-Py], [BG4164: 3-I-4-Py], [BG4165: 2-Cl-3-I-4-Py], [BG4166: 5-Cl-3-I-4-Py] , [BG4167: 6-Cl-3-I-4-Py], [BG4168: 2-Me-3-I-4-Py], [BG4169: 5-Me-3-I-4-Py], [BG BG4170: 6-Me-3- I-4-Py], [BG4171: 2-CF 3 -3-I-4-Py], [BG4172: 5-CF 3 -3-I-4-Py], [ _{BG4173: 6-CF 3 -3-} I-4-Py], [BG4174: 2-CN-3-I-4-Py], [BG4175: 5-CN-3-I-4-Py], [BG4176 : 6-CN-3-I-4-Py], [BG4177: 2-OMe-3-I-4-Py], [BG4178: 5-OMe-3-I-4-Py], [BG4179: 6] -OMe-3-I-4-Py], [BG 4180: 2-I-4-Py], [BG4181: 3-Cl-2-I-4-Py], [BG4182: 5-Cl-2-I -4-Py], [BG4183: 6-Cl-2-I -4-Py !, [BG4184: 3-Me-2-I-4-Py], [BG4185: 5-Me-2-I-4-Py], [BG4186: 6-Me-2-I-4] -Py], [BG4187: 3- CF 3 -2-I-4-Py], [BG4188: 5-CF 3 -2-I-4-Py], [BG4189: 6-CF 3 -2-I- 4-Py], [BG4190: 3-CN-2-I-4-Py], [BG4191: 5-CN-2-I-4-Py], [BG4192: 6-CN-2-I-4- 4 Py], [BG4193: 3-OMe-2-I-4-Py], [BG4194: 5-OMe-2-I-4-Py], [BG4195: 6-OMe-2-I-4-Py] , [BG4196: 5-I-4-Py], [BG4197: 3-Cl-5-I-4-Py], [BG4198: 2-Cl-5-I-4-Py], [BG4199: 6- Cl-5-I-4-Py], [BG4200: 3-Me-5-I-4-Py],

[BG4201: 2-Me-5 -I-4-Py], [BG4202: 6-Me-5-I-4-Py], [BG4203: 3-CF 3 -5-I-4-Py], [ _{BG4204: 2-CF 3 -5-} I-4-Py], [BG4205: 6-CF 3 -5-I-4-Py], [BG4206: 3-CN-5-I-4-Py], [ BG4207: 2-CN-5-I-4-Py, [BG4208: 6-CN-5-I-4-Py], [BG4209: 3-OMe-5-I-4-Py], [BG4210: 2-OMe-5-I-4-Py], [BG4211: 6-OMe-5-I-4-Py], [BG4212: 6-I-4-Py], [BG4213: 3-Cl-6-] I-4-Py], [BG4214: 2-Cl-6-I-4-Py], [BG4215: 5-Cl-6-I-4-Py], [BG4216: 3-Me-6-I- 4-Py], [BG4217: 2-Me-6-I-4-Py], [BG4218: 5-Me-6-I-4-Py], [BG4219: 3-CF 3 -6-I-4 -Py], [BG4220: 2- CF 3 -6-I-4-Py], [BG4221: 5-CF 3 -6-I-4-Py], [BG4222: 3-CN-6-I-4 -Py], [BG4223: 2-CN-6-I-4-Py], [BG4224: 5-CN-6-I-4-Py], [BG4225: 3-OMe-6-I-4-Py] ], [BG4226: 2-OMe-6-I-4-Py], [BG4227: 5-OMe-6-I-4-Py], [BG4228: 3-Me-4-Py], [BG4229: 2] -Cl-3-Me-4-Py], [BG 4230: 5-Cl-3-Me-4-Py], [BG4231: 6-Cl-3-Me-4-Py], [BG4232: 2-Me -3-Me-4-Py !, [BG4233: 5-Me-3-Me-4-Py], [BG4234: 6-Me-3-Me-4-Py], [BG4235: 2-CF _3- 3-Me-4-Py] , [BG4236: 5-CF 3 -3-Me-4-Py], [BG4237: 6-CF 3 -3-Me-4-Py], [BG4238: 2-CN- 3-Me-4-Py !, [BG4239: 5-CN-3-Me-4-Py], [BG4240: 6-CN-3-Me-4-Py], [BG4241: 2-OMe-3-3] Me-4-Py], [BG4242: 5-OMe-3-Me- 4-Py], [BG4243: 6-OMe-3-Me-4-Py], [BG4244: 2-Me-4-Py], [BG4245: 3-Cl-2-Me-4-Py], BG 4246: 5-Cl-2-Me-4-Py !, [BG4247: 6-Cl-2-Me-4-Py], [BG4248: 3-Me-2-Me-4-Py], [BG4249: 5-Me-2-Me- 4-Py], [BG4250: 6-Me-2-Me-4-Py], [BG4251: 3-CF 3 -2-Me-4-Py], [BG4252: 5 _{-CF 3 -2-Me-4-} Py], [BG4253: 6-CF 3 -2-Me-4-Py], [BG4254: 3-CN-2-Me-4-Py], [BG4255: 5 -CN-2-Me-4-Py], [BG4256: 6-CN-2-Me-4-Py], [BG4257: 3-OMe-2-Me-4-Py], [BG4258: 5-OMe] -2-Me-4-Py !, [BG4259: 6-OMe-2-Me-4-Py], [BG4260: 5-Me-4-Py], [BG4261: 3-Cl-5-Me-4] -Py], [BG4262: 2-Cl-5-Me-4-Py], [BG4263: 6-Cl-5-Me-4-Py], [BG4264: 3-Me-5-Me-4-Py ], [BG4265: 2-Me -5-Me-4-Py], [BG4266: 6-Me-5-Me-4-Py], [BG4267: 3-CF 3 -5-Me-4-Py] _{, [BG4268: 2-CF 3} -5-Me-4-Py], [BG4269: 6-CF 3 -5-Me-4-Py], [BG4270: 3-CN-5-Me-4-Py] , [BG4271: 2-CN-5-Me-4-Py], [BG4272: 6-CN-5-Me-4-Py], [BG4273: 3-OMe-5-Me-4-Py], [BG4272: BG4274: 2-OMe-5-Me-4-Py], [BG4275: 6-OMe-5-Me-4-Py], [BG4276: 6-Me-4-Py], [BG4277: 3-Cl- 6-Me-4-Py !, [BG4278: 2-Cl-6-Me-4-Py], [BG4279: 5-Cl-6-Me-4-Py], [BG4280: 3-Me-6-6] Me-4-Py], [ BG4281: 2-Me-6-Me-4-Py], [BG4282: 5-Me-6-Me-4-Py], [BG4283: 3-CF 3 -6-Me -4-P y], [BG4284: 2- CF 3 -6-Me-4-Py], [BG4285: 5-CF 3 -6-Me-4-Py], [BG4286: 3-CN-6-Me-4- Py], [BG4287: 2-CN-6-Me-4-Py], [BG4288: 5-CN-6-Me-4-Py], [BG4289: 3-OMe-6-Me-4-Py] , [BG4290: 2-OMe-6-Me-4-Py], [BG4291: 5-OMe-6-Me-4-Py], [BG4292: 3-OMe-4-Py], [BG4293: 2- Cl-3-OMe-4-Py !, [BG4294: 5-Cl-3-OMe-4-Py], [BG4295: 6-Cl-3-OMe-4-Py], [BG4296: 2-Me- 3-OMe-4-Py], [BG4297: 5-Me-3-OMe-4-Py], [BG4298: 6-Me-3-OMe-4-Py], [BG4299: 2-CF ₃ -3] -OMe-4-Py], [BG 4300: 5-CF ₃ -3-OMe-4-Py],

_{[BG4301: 6-CF 3 -3} -OMe-4-Py], [BG4302: 2-CN-3-OMe-4-Py], [BG4303: 5-CN-3-OMe-4-Py], [ BG4304: 6-CN-3-OMe-4-Py], [BG4305: 2-OMe-3-OMe-4-Py], [BG4306: 5-OMe-3-OMe-4-Py], [BG4307: 6-OMe-3-OMe-4-Py], [BG4308: 2-OMe-4-Py], [BG4309: 3-Cl-2-OMe-4-Py], [BG 4310: 5-Cl-2-] OMe-4-Py], [BG4311: 6-Cl-2-OMe-4-Py], [BG4312: 3-Me-2-OMe-4-Py], [BG4313: 5-Me-2-OMe- 4-Py], [BG4314: 6-Me-2-OMe-4-Py], [BG4315: 3-CF 3 -2-OMe-4-Py], [BG4316: 5-CF 3 -2-OMe- 4-Py], [BG4317: 6-CF 3 -2-OMe-4-Py], [BG4318: 3-CN-2-OMe-4-Py], [BG4319: 5-CN-2-OMe-4 -Py], [BG4320: 6-CN-2-OMe-4-Py], [BG4321: 3-OMe-2-OMe-4-Py], [BG4322: 5-OMe-2-OMe-4-Py] ], [BG 4323: 6-OMe-2-OMe-4-Py], [BG 4324: 5-OMe-4-Py], [BG 4325: 3-Cl-5-OMe-4-Py], [BG 4326: 2] -Cl-5-OMe-4-Py], [BG4327: 6-Cl-5-OMe-4-Py], [BG4328: 3-Me-5-OMe-4-Py], [BG4329: 2-Me -5-OMe-4-Py] , [BG4330: 6-Me-5-OMe-4-Py], [BG4331: 3-CF 3 -5-OMe-4-Py], [BG4332: 2-CF 3 -5-OMe-4-Py] , [BG4333: 6-CF 3 -5-OMe-4-Py], [BG4334: 3-CN-5-OMe-4-Py], [BG4335: 2-CN- 5-OMe-4-Py], [BG4336: 6-CN-5-OMe-4-Py], [BG4337: 3-OMe-5-OMe-4-Py], [BG4338: 2-OMe-5-] OMe-4-Py], [BG4339: 6-OMe-5-OMe-4-Py], [BG43] 40: 6-OMe-4-Py], [BG4341: 3-Cl-6-OMe-4-Py], [BG4342: 2-Cl-6-OMe-4-Py], [BG4343: 5-Cl- 6-OMe-4-Py], [BG4344: 3-Me-6-OMe-4-Py], [BG4345: 2-Me-6-OMe-4-Py], [BG4346: 5-Me-6-6] OMe-4-Py], [ BG4347: 3-CF 3 -6-OMe-4-Py], [BG4348: 2-CF 3 -6-OMe-4-Py], [BG4349: 5-CF 3 -6 -OMe-4-Py], [BG4350: 3-CN-6-OMe-4-Py], [BG4351: 2-CN-6-OMe-4-Py], [BG4352: 5-CN-6-OMe] -4-Py], [BG4353: 3-OMe-6-OMe-4-Py], [BG4354: 2-OMe-6-OMe-4-Py], [BG4355: 5-OMe-6-OMe-4] -Py], [BG 4356: 3-CF ₃ -4-Py], [BG 4 357: 2-Cl-3-CF ₃ -4-Py], [BG 4 358: 5-Cl-3-CF ₃ -4-Py] , [BG4359: 6-Cl- 3-CF 3 -4-Py], [BG4360: 2-Me-3-CF 3 -4-Py], [BG4361: 5-Me-3-CF 3 -4-Py ], [BG4362: 6-Me -3-CF 3 -4-Py], [BG4363: 2-CF 3 -3-CF 3 -4-Py], [BG4364: 5-CF 3 -3-CF 3 - 4-Py], [BG4365: 6-CF 3 -3-CF 3 -4-Py], [BG4366: 2-CN-3-CF 3 -4-Py], [BG4367: 5-CN-3-CF ₃ -4-Py !, [BG 4368: 6-CN-3-CF ₃ -4-Py], [BG 4369: 2-OMe-3-CF ₃ -4-Py], [BG 4370: 5-OMe -3-] _{CF 3 -4-Py], [} BG4371: 6-OMe-3-CF 3 -4-Py], [BG4372: 2-CF 3 -4-Py], [BG4373: 3-Cl-2-CF 3 - 4-Py], [BG4374: 5-Cl-2-CF 3 -4-Py], [BG4375: 6-Cl-2-CF 3 -4-Py], [BG4376: 3-Me-2-CF 3 -4-Py], [BG 4377: 5-Me-2-CF ₃ -4-Py], [B G4378: 6-Me-2- CF 3 -4-Py], [BG4379: 3-CF 3 -2-CF 3 -4-Py], [BG4380: 5-CF 3 -2-CF 3 -4-Py ], [BG4381: 6-CF 3 -2-CF 3 -4-Py], [BG4382: 3-CN-2-CF 3 -4-Py], [BG4383: 5-CN-2-CF 3 -4 -Py], [BG4384: 6- CN-2-CF 3 -4-Py], [BG4385: 3-OMe-2-CF 3 -4-Py], [BG4386: 5-OMe-2-CF 3 - 4-Py], [BG4387: 6-OMe-2-CF 3 -4-Py], [BG4388: 5-CF 3 -4-Py], [BG4389: 3-Cl-5-CF 3 -4-Py ], [BG4390: 2-Cl -5-CF 3 -4-Py], [BG4391: 6-Cl-5-CF 3 -4-Py], [BG4392: 3-Me-5-CF 3 -4- Py], [BG4393: 2- Me-5-CF 3 -4-Py], [BG4394: 6-Me-5-CF 3 -4-Py], [BG4395: 3-CF 3 -5-CF 3 - 4-Py], [BG 4396: 2-CF ₃ -5-CF ₃ -4-Py], [BG 4397: 6-CF ₃ -5-CF ₃ -4-Py], [BG 4 398: 3-CN-5- CF ₃ -4-Py], [BG 4399: 2-CN-5-CF ₃ -4-Py], [BG 4400: 6-CN-5-CF ₃ -4-Py],

[BG4401: 3-OMe-5 -CF 3 -4-Py], [BG4402: 2-OMe-5-CF 3 -4-Py], [BG4403: 6-OMe-5-CF 3 -4-Py] _{, [BG4404: 6-CF 3} -4-Py], [BG4405: 3-Cl-6-CF 3 -4-Py], [BG4406: 2-Cl-6-CF 3 -4-Py], [BG4407 : 5-Cl-6-CF 3 -4-Py], [BG4408: 3-Me-6-CF 3 -4-Py], [BG4409: 2-Me-6-CF 3 -4-Py], [ BG4410: 5-Me-6- CF 3 -4-Py], [BG4411: 3-CF 3 -6-CF 3 -4-Py], [BG4412: 2-CF 3 -6-CF 3 -4-Py ], [BG4413: 5-CF 3 -6-CF 3 -4-Py], [BG4414: 3-CN-6-CF 3 -4-Py], [BG4415: 2-CN-6-CF 3 -4 -Py], [BG4416: 5- CN-6-CF 3 -4-Py], [BG4417: 3-OMe-6-CF 3 -4-Py], [BG4418: 2-OMe-6-CF 3 - 4-Py], [BG4419: 5-OMe-6-CF 3 -4-Py], [BG4420: 3-OCF 3 -4-Py], [BG4421: 2-Cl-3-OCF 3 -4-Py ], [BG4422: 5-Cl -3-OCF 3 -4-Py], [BG4423: 6-Cl-3-OCF 3 -4-Py], [BG4424: 2-Me-3-OCF 3 -4- Py], [BG4425: 5- Me-3-OCF 3 -4-Py], [BG4426: 6-Me-3-OCF 3 -4-Py], [BG4427: 2-CF 3 -3-OCF 3 - 4-Py], [BG4428: 5-CF ₃ -3-OCF ₃ -4-Py], [BG 4429: 6-CF ₃ -3-OCF ₃ -4-Py], [BG 4430: 2-CN-3- 3 _{OCF 3 -4-Py], [} BG4431: 5-CN-3-OCF 3 -4-Py], [BG4432: 6-CN-3-OCF 3 -4-Py], [BG4433: 2-OMe-3 _{-OCF 3 -4-Py], [} BG4434: 5-OMe-3-OCF 3 -4-Py], [BG4435: 6-OMe-3-OCF 3 -4-Py], [BG4436: 2-OCF 3 -4-Py] , [BG4437: 3-Cl- 2-OCF 3 -4-Py], [BG4438: 5-Cl-2-OCF 3 -4-Py], [BG4439: 6-Cl-2-OCF 3 -4-Py ], [BG4440: 3-Me -2-OCF 3 -4-Py], [BG4441: 5-Me-2-OCF 3 -4-Py], [BG4442: 6-Me-2-OCF 3 -4- Py], [BG4443: 3- CF 3 -2-OCF 3 -4-Py], [BG4444: 5-CF 3 -2-OCF 3 -4-Py], [BG4445: 6-CF 3 -2-OCF ₃ -4-Py !, [BG 4446: 3-CN-2-OCF ₃ -4-Py], [BG 4 447: 5-CN-2-OCF ₃ -4-Py], [BG 4448: 6-CN-2-] _{OCF 3 -4-Py], [} BG4449: 3-OMe-2-OCF 3 -4-Py], [BG4450: 5-OMe-2-OCF 3 -4-Py], [BG4451: 6-OMe-2 _{-OCF 3 -4-Py], [} BG4452: 5-OCF 3 -4-Py], [BG4453: 3-Cl-5-OCF 3 -4-Py], [BG4454: 2-Cl-5-OCF 3 -4-Py], [BG4455: 6-Cl-5-OCF 3 -4-Py], [BG4456: 3-Me-5-OCF 3 -4-Py], [BG4457: 2-Me-5-OCF ₃ -4-Py], [BG 4458: 6-Me-5-OCF ₃ -4-Py], [BG 4459: 3-CF ₃ -5-OCF ₃ -4-Py], [BG 4460: 2-CF _{3- 5-OCF 3 -4-Py]} , [BG4461: 6-CF 3 -5-OCF 3 -4-Py], [BG4462: 3-CN-5-OCF 3 -4-Py], [BG4463: 2- _{CN-5-OCF 3 -4-} Py], [BG4464: 6-CN-5-OCF 3 -4-Py], [BG4465: 3-OMe-5-OCF 3 -4-Py], [BG4466: 2 _{-OMe-5-OCF 3 -4-} Py], [BG4467: 6-OMe-5-OCF 3 -4-Py], [BG4468: 6-OCF 3 -4-Py], [BG4469: 3-Cl- _{6-OCF 3 -4-Py]} , [BG4470: 2-Cl-6-OCF 3 -4-Py], [BG4471: 5-Cl-6-OCF 3 -4-Py], [BG44 72: 3-Me-6- OCF 3 -4-Py], [BG4473: 2-Me-6-OCF 3 -4-Py], [BG4474: 5-Me-6-OCF 3 -4-Py], _{[BG4475: 3-CF 3 -6} -OCF 3 -4-Py], [BG4476: 2-CF 3 -6-OCF 3 -4-Py], [BG4477: 5-CF 3 -6-OCF 3 -4 -Py], [BG4478: 3- CN-6-OCF 3 -4-Py], [BG4479: 2-CN-6-OCF 3 -4-Py], [BG4480: 5-CN-6-OCF 3 - 4-Py], [BG4481: 3-OMe-6-OCF 3 -4-Py], [BG4482: 2-OMe-6-OCF 3 -4-Py], [BG4483: 5-OMe-6-OCF 3 -4-Py], [BG4484: 3-CHF 2 -4-Py], [BG4485: 2-Cl-3-CHF 2 -4-Py], [BG4486: 5-Cl-3-CHF 2 -4- Py], [BG4487: 6- Cl-3-CHF 2 -4-Py], [BG4488: 2-Me-3-CHF 2 -4-Py], [BG4489: 5-Me-3-CHF 2 -4 -Py], [BG4490: 6- Me-3-CHF 2 -4-Py], [BG4491: 2-CF 3 -3-CHF 2 -4-Py], [BG4492: 5-CF 3 -3-CHF ₂ -4-Py], [BG4493: 6-CF ₃ -3-CHF ₂ -4-Py], [BG4494: 2-CN-3-CHF ₂ -4-Py], [BG 4495: 5-CN-3] _{-CHF 2 -4-Py], [} BG4496: 6-CN-3-CHF 2 -4-Py], [BG4497: 2-OMe-3-CHF 2 -4-Py], [BG4498: 5-OMe- 3-CHF ₂ -4-Py], [BG 4499: 6-OMe -3-CHF ₂ -4-Py], [BG 4500: 4-CHF ₂ -4-Py],

[BG4501: 3-Cl-4 -CHF 2 -4-Py], [BG4502: 5-Cl-4-CHF 2 -4-Py], [BG4503: 6-Cl-4-CHF 2 -4-Py] , [BG4504: 3-Me- 4-CHF 2 -4-Py], [BG4505: 5-Me-4-CHF 2 -4-Py], [BG4506: 6-Me-4-CHF 2 -4-Py ], [BG4507: 3-CF 3 -4-CHF 2 -4-Py], [BG4508: 5-CF 3 -4-CHF 2 -4-Py], [BG4509: 6-CF 3 -4-CHF 2 -4-Py], [BG4510: 3-CN-4-CHF 2 -4-Py], [BG4511: 5-CN-4-CHF 2 -4-Py], [BG4512: 6-CN-4-CHF ₂ -4-Py !, [BG 4513: 3-OMe -4-CHF ₂ -4-Py], [BG 4514: 5-OMe -4-CHF ₂ -4-Py], [BG 4515: 6-OMe -4-] CHF ₂ -4-Py !, [BG 4516: 5-CHF ₂ -4-Py], [BG 4517: 3-Cl-5-CHF ₂ -4-Py], [BG 4518: 2-Cl-5-CHF _2- 4-Py], [BG4519: 6-Cl-5-CHF ₂ -4-Py], [BG 4520: 3-Me-5-CHF ₂ -4-Py], [BG 4521: 2-Me-5-CHF ₂ -4-Py], [BG4522: 6-Me-5-CHF 2 -4-Py], [BG4523: 3-CF 3 -5-CHF 2 -4-Py], [BG4524: 2-CF 3 -5 -CHF ₂ -4-Py], [BG 4525: 6-CF ₃ -5-CHF ₂ -4-Py], [BG 4526: 3-CN-5-CHF ₂ -4-Py], [BG 4 527: 2-CN -5-CHF ₂ -4-Py], [BG4528: 6-CN-5-CHF ₂ -4-Py], [BG4529: 3-OMe-5-CHF ₂ -4-Py], [BG 4530: 2- _{OMe-5-CHF 2 -4-} Py], [BG4531: 6-OMe-5-CHF 2 -4-Py], [BG4532: 6-CHF 2 -4-Py], [BG4533: 3-Cl-6 _{-CHF 2 -4-Py], [} BG4534: 2-Cl-6-CHF 2 -4-Py], [BG4535: 5-Cl-6-CHF 2 -4-Py], [BG453 6: 3-Me-6- CHF 2 -4-Py], [BG4537: 2-Me-6-CHF 2 -4-Py], [BG4538: 5-Me-6-CHF 2 -4-Py], _{[BG4539: 3-CF 3 -6} -CHF 2 -4-Py], [BG4540: 2-CF 3 -6-CHF 2 -4-Py], [BG4541: 5-CF 3 -6-CHF 2 -4 -Py], [BG4542: 3- CN-6-CHF 2 -4-Py], [BG4543: 2-CN-6-CHF 2 -4-Py], [BG4544: 5-CN-6-CHF 2 - 4-Py], [BG4545: 3-OMe-6-CHF 2 -4-Py], [BG4546: 2-OMe-6-CHF 2 -4-Py], [BG4547: 5-OMe-6-CHF 2 -4-Py], [BG4548: 3-OCHF 2 -4-Py], [BG4549: 2-Cl-3-OCHF 2 -4-Py], [BG4550: 5-Cl-3-OCHF 2 -4- Py], [BG4551: 6- Cl-3-OCHF 2 -4-Py], [BG4552: 2-Me-3-OCHF 2 -4-Py], [BG4553: 5-Me-3-OCHF 2 -4 -Py], [BG4554: 6- Me-3-OCHF 2 -4-Py], [BG4555: 2-CF 3 -3-OCHF 2 -4-Py], [BG4556: 5-CF 3 -3-OCHF _{2 -4-Py], [BG4557} : 6-CF 3 -3-OCHF 2 -4-Py], [BG4558: 2-CN-3-OCHF 2 -4-Py], [BG4559: 5-CN-3 _{-OCHF 2 -4-Py], [} BG4560: 6-CN-3-OCHF 2 -4-Py], [BG4561: 2-OMe-3-OCHF 2 -4-Py], [BG4562: 5-OMe- 3-OCHF ₂ -4-Py], [BG4563: 6-OMe-3-OCHF ₂ -4-Py], [BG4564: 4-OCHF ₂ -4-Py], [BG4 565: 3-Cl-4-OCHF _{2 -4-Py], [BG4566} : 5-Cl-4-OCHF 2 -4-Py], [BG4567: 6-Cl-4-OCHF 2 -4-Py], [BG4568: 3-Me-4- OCHF ₂ -4-Py, [BG 4569: 5-Me 4-OCHF ₂ -4-Py], [BG 4570: 6-Me 4-OCH _{F 2 -4-Py], [} BG4571: 3-CF 3 -4-OCHF 2 -4-Py], [BG4572: 5-CF 3 -4-OCHF 2 -4-Py], [BG4573: 6-CF ₃ -4-OCHF ₂ -4-Py], [BG4574: 3-CN -4-OCHF ₂ -4-Py], [BG 4575: 5-CN -4-OCHF ₂ -4-Py], [BG 4576: 6] _{-CN-4-OCHF 2 -4-} Py], [BG4577: 3-OMe-4-OCHF 2 -4-Py], [BG4578: 5-OMe-4-OCHF 2 -4-Py], [BG4579: _{6-OMe-4-OCHF 2} -4-Py], [BG4580: 5-OCHF 2 -4-Py], [BG4581: 3-Cl-5-OCHF 2 -4-Py], [BG4582: 2-Cl -5-OCHF ₂ -4-Py], [BG4583: 6-Cl-5-OCHF ₂ -4-Py], [BG4584: 3-Me-5-OCHF ₂ -4-Py], [BG4585: 2-] Me-5-OCHF ₂ -4-Py], [BG 4586: 6-Me-5-OCHF ₂ -4-Py], [BG 4587: 3-CF ₃ -5-OCHF ₂ -4-Py], [BG 4588: _{2-CF 3 -5-OCHF 2} -4-Py], [BG4589: 6-CF 3 -5-OCHF 2 -4-Py], [BG4590: 3-CN-5-OCHF 2 -4-Py], [BG4591: 2-CN-5 -OCHF 2 -4-Py], [BG4592: 6-CN-5-OCHF 2 -4-Py], [BG4593: 3-OMe-5-OCHF 2 -4-Py] , [BG 4594: 2-OMe-5-OCHF ₂ -4-Py], [BG 4595: 6-OMe-5-OCHF ₂ -4-Py], [BG 4596: 6-OCHF ₂ -4-Py], [BG 4 597] : 3-Cl-6-OCHF 2 -4-Py], [BG4598: 2-Cl-6-OCHF 2 -4-Py], [BG4599: 5-Cl-6-OCHF 2 -4-Py], [ BG 4600: 3-Me-6-OCHF ₂ -4-Py],

[BG4601: 2-Me-6 -OCHF 2 -4-Py], [BG4602: 5-Me-6-OCHF 2 -4-Py], [BG4603: 3-CF 3 -6-OCHF 2 -4-Py ], [BG4604: 2-CF 3 -6-OCHF 2 -4-Py], [BG4605: 5-CF 3 -6-OCHF 2 -4-Py], [BG4606: 3-CN-6-OCHF 2 - 4-Py], [BG4607: 2-CN-6-OCHF 2 -4-Py], [BG4608: 5-CN-6-OCHF 2 -4-Py], [BG4609: 3-OMe-6-OCHF 2 -4-Py], [BG4610: 2-OMe-6-OCHF 2 -4-Py], [BG4611: 5-OMe-6-OCHF 2 -4-Py], [BG4612: 3-Et-4-Py ], [BG4613: 2-Cl-3-Et-4-Py], [BG4614: 5-Cl-3-Et-4-Py], [BG4615: 6-Cl-3-Et-4-Py], [BG4616: 2-Me-3-Et-4-Py], [BG4617: 5-Me-3-Et-4-Py], [BG4618: 6-Me-3-Et-4-Py], [BG4619 _{: 2-CF 3 -3-Et} -4-Py], [BG4620: 5-CF 3 -3-Et-4-Py], [BG4621: 6-CF 3 -3-Et-4-Py], [ BG4622: 2-CN-3-Et-4-Py !, [BG4623: 5-CN-3-Et-4-Py], [BG4624: 6-CN-3-Et-4-Py], [BG4625: 2-OMe-3-Et-4-Py], [BG4626: 5-OMe-3-Et-4-Py], [BG4627: 6-OMe-3-Et-4-Py], [BG4628: 2- Et-4-Py !, [BG4 629: 3-Cl-2-Et-4-Py], [BG4630: 5-Cl-2-Et-4-Py], [BG 4631: 6-Cl-2-Et- 4-Py], [BG4632: 3-Me-2-Et-4-Py], [BG4633: 5-Me-2-Et-4-Py], [BG4634: 6-Me-2-Et-4-] Py], [BG4635: 3- CF 3 -2-Et-4-Py], [BG4636: 5-CF 3 -2-Et-4-Py], [BG4637: 6-CF 3 -2-Et-4 -Py], [BG4638: 3-CN-2-Et-4-Py], [BG4639: 5-] CN-2-Et-4-Py !, [BG4640: 6-CN-2-Et-4-Py], [BG4641: 3-OMe-2-Et-4-Py], [BG4642: 5-OMe- 2-Et-4-Py], [BG4643: 6-OMe-2-Et-4-Py], [BG4644: 5-Et-4-Py], [BG4645: 3-Cl-5-Et-4- 4 Py], [BG4646: 2-Cl-5-Et-4-Py], [BG4647: 6-Cl-5-Et-4-Py], [BG4648: 3-Me-5-Et-4-Py] [BG 4649: 2-Me-5-Et-4-Py], [BG 4650: 6-Me-5-Et-4-Py], [BG4651: 3-CF ₃ -5-Et-4-Py], _{[BG4652: 2-CF 3 -5} -Et-4-Py], [BG4653: 6-CF 3 -5-Et-4-Py], [BG4654: 3-CN-5-Et-4-Py], [BG 4655: 2-CN-5-Et-4-Py], [BG 4656: 6-CN-5-Et-4-Py], [BG4657: 3-OMe-5-Et-4-Py], [BG4658] : 2-OMe-5-Et-4-Py], [BG4659: 6-OMe-5-Et-4-Py], [BG 4660: 6-Et-4-Py], [BG4661: 3-Cl-6] -Et-4-Py], [BG4662: 2-Cl-6-Et-4-Py], [BG4663: 5-Cl-6-Et-4-Py], [BG4664: 3-Me-6-Et] -4-Py], [BG4665: 2-Me-6-Et-4-Py], [BG4666: 5-Me-6-Et-4-Py], [BG4667: 3-CF ₃ -6-Et- 4-Py], [BG4668: 2-CF 3 -6-Et-4-Py], [BG4669: 5-CF 3 -6-Et-4-Py], [BG4670: 3-CN-6-Et- 4-Py], [BG4671: 2-CN-6-Et-4-Py], [BG4672: 5-CN-6-Et-4-Py], [BG4673: 3-OMe-6-Et-4- 4 Py], [BG 4674: 2-OMe-6-Et-4-Py], [BG 4675: 5-OMe-6-Et-4-Py], [BG 4676: 3-CH ₂ CF ₃ -4-Py], [BG4677: 2-Cl-3 -CH 2 CF 3 -4-Py], [BG4678: 5-Cl-3-CH 2 CF 3 -4-Py], [BG4679: 6-Cl-3 _{-CH 2 CF 3 -4-Py]} , [BG4680: 2-Me-3-CH 2 CF 3 -4-Py], [BG4681: 5-Me-3-CH 2 CF 3 -4-Py], [ BG4682: 6-Me-3- CH 2 CF 3 -4-Py], [BG4683: 2-CF 3 -3-CH 2 CF 3 -4-Py], [BG4684: 5-CF 3 -3-CH 2 CF ₃ -4-Py !, [BG 4685: 6-CF ₃ -3-CH ₂ CF ₃ -4-Py], [BG 4686: 2-CN-3-CH ₂ CF ₃ -4-Py], [BG 4687: _{5-CN-3-CH 2} CF 3 -4-Py], [BG4688: 6-CN-3-CH 2 CF 3 -4-Py], [BG4689: 2-OMe-3-CH 2 CF 3 -4 -Py], [BG4690: 5- OMe-3-CH 2 CF 3 -4-Py], [BG4691: 6-OMe-3-CH 2 CF 3 -4-Py], [BG4692: 2-CH 2 CF _{3 -4-Py], [BG4693} : 3-Cl-2-CH 2 CF 3 -4-Py], [BG4694: 5-Cl-2-CH 2 CF 3 -4-Py], [BG4695: 6- _{Cl-2-CH 2 CF 3} -4-Py], [BG4696: 3-Me-2-CH 2 CF 3 -4-Py], [BG4697: 5-Me-2-CH 2 CF 3 -4-Py ], [BG4698: 6-Me -2-CH 2 CF 3 -4-Py], [BG4699: 3-CF 3 -2-CH 2 CF 3 -4-Py], [BG4700: 5-CF 3 -2 -CH ₂ CF ₃ -4-Py],

_{[BG4701: 6-CF 3 -2} -CH 2 CF 3 -4-Py], [BG4702: 3-CN-2-CH 2 CF 3 -4-Py], [BG4703: 5-CN-2-CH 2 CF ₃ -4-Py !, [BG 4704: 6-CN-2-CH ₂ CF ₃ -4-Py], [BG 4705: 3-OMe-2-CH ₂ CF ₃ -4-Py], [BG 4706: 5] -OMe-2-CH ₂ CF ₃ -4-Py, [BG 4707: 6-OMe-2-CH ₂ CF ₃ -4-Py], [BG 4708: 5-CH ₂ CF ₃ -4-Py], [BG BG4709: 3-Cl-5- CH 2 CF 3 -4-Py], [BG4710: 2-Cl-5-CH 2 CF 3 -4-Py], [BG4711: 6-Cl-5-CH 2 CF 3 -4-Py], [BG4712: 3-Me-5-CH 2 CF 3 -4-Py], [BG4713: 2-Me-5-CH 2 CF 3 -4-Py], [BG4714: 6-Me -5-CH ₂ CF ₃ -4-Py], [BG 4715: 3-CF ₃ -5-CH ₂ CF ₃ -4-Py], [BG 4716: 2-CF ₃ -5-CH ₂ CF ₃ -4- Py], [BG4717: 6- CF 3 -5-CH 2 CF 3 -4-Py], [BG4718: 3-CN-5-CH 2 CF 3 -4-Py], [BG4719: 2-CN-5 _{-CH 2 CF 3 -4-Py]} , [BG4720: 6-CN-5-CH 2 CF 3 -4-Py], [BG4721: 3-OMe-5-CH 2 CF 3 -4-Py], [ BG4722: 2-OMe-5- CH 2 CF 3 -4-Py], [BG4723: 6-OMe-5-CH 2 CF 3 -4-Py], [BG4724: 6-CH 2 CF 3 -4-Py ], [BG4725: 3-Cl -6-CH 2 CF 3 -4-Py], [BG4726: 2-Cl-6-CH 2 CF 3 -4-Py], [BG4727: 5-Cl-6-CH _{2 CF 3 -4-Py],} [BG4728: 3-Me-6-CH 2 CF 3 -4-Py], [BG4729: 2-Me-6-CH 2 CF 3 -4-Py], [BG4730: 5-Me-6-CH ₂ CF ₃ -4-Py], [BG4731: 3-CF ₃ -6-CH ₂ CF ₃ -4-P y], [BG 4732: 2-CF ₃ -6-CH ₂ CF ₃ -4-Py], [BG 4 733: 5-CF ₃ -6-CH ₂ CF ₃ -4-Py], [BG 4 734: 3-CN- _{6-CH 2 CF 3 -4-} Py], [BG4735: 2-CN-6-CH 2 CF 3 -4-Py], [BG4736: 5-CN-6-CH 2 CF 3 -4-Py], [BG4737: 3-OMe-6 -CH 2 CF 3 -4-Py], [BG4738: 2-OMe-6-CH 2 CF 3 -4-Py], [BG4739: 5-OMe-6-CH 2 CF ₃ -4-Py !, [BG4740: 3-OEt-4-Py], [BG4741: 2-Cl-3-OEt-4-Py], [BG4742: 5-Cl-3-OEt-4-Py] [BG4743: 6-Cl-3-OEt-4-Py], [BG4744: 2-Me-3-OEt-4-Py], [BG4745: 5-Me-3-OEt-4-Py], BG4746: 6-Me-3- OEt-4-Py], [BG4747: 2-CF 3 -3-OEt-4-Py], [BG4748: 5-CF 3 -3-OEt-4-Py], [ _{BG4749: 6-CF 3 -3-} OEt-4-Py], [BG4750: 2-CN-3-OEt-4-Py], [BG4751: 5-CN-3-OEt-4-Py], [BG4752 6-CN-3-OEt-4-Py !, [BG4753: 2-OMe-3-OEt-4-Py], [BG4754: 5-OMe-3-OEt-4-Py], [BG4755: 6] -OMe-3-OEt-4-Py], [BG 4756: 2-OEt-4-Py], [BG4757: 3-Cl-2-OEt-4-Py], [BG4758: 5-Cl-2-OEt -4-Py !, [BG4759: 6-Cl-2-OEt-4-Py], [BG 4760: 3-Me-2-OEt-4-Py], [BG4761: 5-Me-2-OEt-4] -Py], [BG4762: 6- Me-2-OEt-4-Py], [BG4763: 3-CF 3 -2-OEt-4-Py], [BG4764: 5-CF 3 -2-OEt-4 -Py], [BG4765: 6- CF 3 -2-OEt-4-Py], [BG4766: 3-CN-2-OEt-4-Py], [BG4767: 5-CN-2-OEt-4- Py], [BG4768: 6-CN-2-OEt-4- Py], [BG4769: 3-OMe-2-OEt-4-Py], [BG4770: 5-OMe-2-OEt-4-Py], [BG4771: 6-OMe-2-OEt-4-Py] , [BG4772: 5-OEt-4-Py], [BG4773: 3-Cl-5-OEt-4-Py], [BG4774: 2-Cl-5-OEt-4-Py], [BG4775: 6- Cl-5-OEt-4-Py], [BG4776: 3-Me-5-OEt-4-Py], [BG4777: 2-Me-5-OEt-4-Py], [BG4778: 6-Me- 5-OEt-4-Py] , [BG4779: 3-CF 3 -5-OEt-4-Py], [BG4780: 2-CF 3 -5-OEt-4-Py], [BG4781: 6-CF 3 -5-OEt-4-Py !, [BG 4782: 3-CN-5-OEt-4-Py], [BG4783: 2-CN-5-OEt-4-Py], [BG 4784: 6-CN-5] -OEt-4-Py], [BG4785: 3-OMe-5-OEt-4-Py], [BG4786: 2-OMe-5-OEt-4-Py], [BG4787: 6-OMe-5-OEt] -4-Py], [BG4788: 6-OEt-4-Py], [BG4789: 3-Cl-6-OEt-4-Py], [BG4790: 2-Cl-6-OEt-4-Py], [BG4791: 5-Cl-6-OEt-4-Py], [BG4792: 3-Me-6-OEt-4-Py], [BG4793: 2-Me-6-OEt-4-Py], [BG4794 : 5-Me-6-OEt -4-Py], [BG4795: 3-CF 3 -6-OEt-4-Py], [BG4796: 2-CF 3 -6-OEt-4-Py], [BG4797 : 5-CF ₃ -6-OEt-4-Py], [BG4798: 3-CN-6-OEt-4-Py], [BG4799: 2-CN-6-OEt-4-Py], [BG4800: 5-CN-6-OEt-4-Py],

[BG4801: 3-OMe-6-OEt-4-Py], [BG4802: 2-OMe-6-OEt-4-Py], [BG4803: 5-OMe-6-OEt-4-Py], [BG4804 _{: 3-OCH 2 CF 3 -4} -Py], [BG4805: 2-Cl-3-OCH 2 CF 3 -4-Py], [BG4806: 5-Cl-3-OCH 2 CF 3 -4-Py] , [BG4807: 6-Cl- 3-OCH 2 CF 3 -4-Py], [BG4808: 2-Me-3-OCH 2 CF 3 -4-Py], [BG4809: 5-Me-3-OCH 2 CF ₃ -4-Py !, [BG 4810: 6-Me-3-OCH ₂ CF ₃ -4-Py], [BG 48 11: 2-CF ₃ -3-OCH ₂ CF ₃ -4-Py], [BG 48 12: 5-CF ₃ -3-OCH ₂ CF ₃ -4-Py], [BG 4813: 6-CF ₃ -3-OCH ₂ CF ₃ -4-Py], [BG 4 814: 2-CN-3-OCH ₂ CF ₃ -4-Py], [BG4815: 5-CN-3-OCH 2 CF 3 -4-Py], [BG4816: 6-CN-3-OCH 2 CF 3 -4-Py], [BG4817: 2-OMe _{-3-OCH 2 CF 3 -4-} Py], [BG4818: 5-OMe-3-OCH 2 CF 3 -4-Py], [BG4819: 6-OMe-3-OCH 2 CF 3 -4-Py] _{, [BG4820: 2-OCH 2} CF 3 -4-Py], [BG4821: 3-Cl-2-OCH 2 CF 3 -4-Py], [BG4822: 5-Cl-2-OCH 2 CF 3 -4 -Py], [BG4823: 6- Cl-2-OCH 2 CF 3 -4-Py], [BG4824: 3-Me-2-OCH 2 CF 3 -4-Py], [BG4825: 5-Me-2 _{-OCH 2 CF 3 -4-Py]} , [BG4826: 6-Me-2-OCH 2 CF 3 -4-Py], [BG4827: 3-CF 3 -2-OCH2CF 3 -4-Py], [BG4828 _{: 5-CF 3 -2-OCH2CF} 3 -4-Py], [BG4829: 6-CF 3 -2-OCH2CF 3 -4-Py], [BG4830: 3-CN-2-OCH 2 CF 3 -4- Py], [BG4831: 5- CN-2-OCH 2 CF 3 -4-Py], [BG4832: 6-CN-2-OCH 2 CF 3 -4-Py], [BG4833: 3-OMe-2-OCH 2 CF 3 -4-Py], [BG4834: 5-OMe _{-2-OCH 2 CF 3 -4-} Py], [BG4835: 6-OMe-2-OCH 2 CF 3 -4-Py], [BG4836: 5-OCH 2 CF 3 -4-Py], [BG4837: _{3-Cl-5-OCH 2} CF 3 -4-Py], [BG4838: 2-Cl-5-OCH 2 CF 3 -4-Py], [BG4839: 6-Cl-5-OCH 2 CF 3 -4 -Py], [BG4840: 3- Me-5-OCH 2 CF 3 -4-Py], [BG4841: 2-Me-5-OCH 2 CF 3 -4-Py], [BG4842: 6-Me-5 -OCH ₂ CF ₃ -4-Py], [BG4843: 3-CF ₃ -5-OCH ₂ CF ₃ -4-Py], [BG4844: 2-CF ₃ -5-OCH ₂ CF ₃ -4-Py] _{, [BG4845: 6-CF 3} -5-OCH 2 CF 3 -4-Py], [BG4846: 3-CN-5-OCH 2 CF 3 -4-Py], [BG4847: 2-CN-5-OCH _{2 CF 3 -4-Py],} [BG4848: 6-CN-5-OCH 2 CF 3 -4-Py], [BG4849: 3-OMe-5-OCH 2 CF 3 -4-Py], [BG4850: _{2-OMe-5-OCH 2} CF 3 -4-Py], [BG4851: 6-OMe-5-OCH 2 CF 3 -4-Py], [BG4852: 6-OCH 2 CF 3 -4-Py], [BG4853: 3-Cl-6 -OCH 2 CF 3 -4-Py], [BG4854: 2-Cl-6-OCH 2 CF 3 -4-Py], [BG4855: 5-Cl-6-OCH 2 CF ₃ -4-Py !, [BG 4856: 3-Me-6-OCH ₂ CF ₃ -4-Py], [BG 4 857: 2-Me-6-OCH ₂ CF ₃ -4-Py], [BG 4 858: 5-] _{Me-6-OCH 2 CF 3} -4-Py], [BG4859: 3-CF 3 -6-OCH 2 CF 3 -4-Py], [BG4860: 2-CF 3 -6-OCH 2 CF 3 -4 -Py], [BG4861: 5-CF ₃ -6-OCH ₂ C _{F 3 -4-Py], [} BG4862: 3-CN-6-OCH 2 CF 3 -4-Py], [BG4863: 2-CN-6-OCH 2 CF 3 -4-Py], [BG4864: 5 _{-CN-6-OCH 2 CF 3} -4-Py], [BG4865: 3-OMe-6-OCH 2 CF 3 -4-Py], [BG4866: 2-OMe-6-OCH 2 CF 3 -4- Py], [BG4867: 5- OMe-6-OCH 2 CF 3 -4-Py], [BG4868: 3-Pr-4-Py], [BG4869: 2-Cl-3-Pr-4-Py], [BG4870: 5-Cl-3-Pr-4-Py], [BG4871: 6-Cl-3-Pr-4-Py], [BG4872: 2-Me-3-Pr-4-Py], [BG4873 : 5-Me-3-Pr -4-Py], [BG4874: 6-Me-3-Pr-4-Py], [BG4875: 2-CF 3 -3-Pr-4-Py], [BG4876: _{5-CF 3 -3-Pr-} 4-Py], [BG4877: 6-CF 3 -3-Pr-4-Py], [BG4878: 2-CN-3-Pr-4-Py], [BG4879: 5-CN-3-Pr-4-Py, [BG4880: 6-CN-3-Pr-4-Py], [BG4881: 2-OMe-3-Pr-4-Py], [BG4882: 5-] OMe-3-Pr-4-Py !, [BG4883: 6-OMe-3-Pr-4-Py], [BG4884: 2-Pr-4-Py], [BG4885: 3-Cl-2-Pr- 4-Py], [BG4886: 5-Cl-2-Pr-4-Py], [BG4887: 6-Cl-2-Pr-4-Py], [BG4888: 3-Me-2-Pr-4- 4 Py], [BG4889: 5- Me-2-Pr-4-Py], [BG4890: 6-Me-2-Pr-4-Py], [BG4891: 3-CF 3 -2-Pr-4-Py ], [BG4892: 5-CF 3 -2-Pr-4-Py], [BG4893: 6-CF 3 -2-Pr-4-Py], [BG4894: 3-CN-2-Pr-4-Py ], [BG4895: 5-CN-2-Pr-4-Py], [BG4896: 6-CN-2-Pr-4-Py], [BG4897: 3-OMe-2-Pr-4-Py], [BG 4898: 5-OMe-2-Pr-4-Py], [BG 4899: 6-OMe-2-Pr-4-Py], [BG 490] 0: 5-Pr-4-Py],

[BG4901: 3-Cl-5-Pr-4-Py], [BG4902: 2-Cl-5-Pr-4-Py], [BG4903: 6-Cl-5-Pr-4-Py], [BG4904] : 3-Me-5-Pr-4-Py], [BG4905: 2-Me-5-Pr-4-Py], [BG4906: 6-Me-5-Pr-4-Py], [BG4907: 3] _{-CF 3 -5-Pr-4-} Py], [BG4908: 2-CF 3 -5-Pr-4-Py], [BG4909: 6-CF 3 -5-Pr-4-Py], [BG4910: 3-CN-5-Pr-4-Py, [BG4911: 2-CN-5-Pr-4-Py], [BG4912: 6-CN-5-Pr-4-Py], [BG4913: 3- OMe-5-Pr-4-Py], [BG4914: 2-OMe-5-Pr-4-Py], [BG4915: 6-OMe-5-Pr-4-Py], [BG4916: 6-Pr- 4-Py], [BG4917: 3-Cl-6-Pr-4-Py], [BG4918: 2-Cl-6-Pr-4-Py], [BG4919: 5-Cl-6-Pr-4- 4 Py], [BG4920: 3-Me-6-Pr-4-Py], [BG4921: 2-Me-6-Pr-4-Py], [BG4922: 5-Me-6-Pr-4-Py] _{, [BG4923: 3-CF 3} -6-Pr-4-Py], [BG4924: 2-CF 3 -6-Pr-4-Py], [BG4925: 5-CF 3 -6-Pr-4-Py ], [BG4926: 3-CN-6-Pr-4-Py], [BG4927: 2-CN-6-Pr-4-Py], [BG 4928: 5-CN-6-Pr-4-Py], [BG4929: 3-OMe-6-Pr-4-Py], [BG4930: 2-OMe-6-Pr-4-Py], [BG4931: 5-OMe-6-Pr-4-Py], [BG4932 : 3-OPr-4-Py], [BG4933: 2-Cl-3-OPr-4-Py], [BG4934: 5-Cl-3-OPr-4-Py], [BG4935: 6-Cl-3] -OPr-4-Py], [BG4936: 2-Me-3-OPr-4-Py], [BG4937: 5-Me-3-OPr-4-Py], [BG4938: 6-Me-3-OPr -4-Py], [BG4939: 2-CF 3 -3-OPr-4-Py], [BG4940: 5-CF 3 -3-OPr-4-Py], [BG4941: 6-C _{F 3 -3-OPr-4-} Py], [BG4942: 2-CN-3-OPr-4-Py], [BG4943: 5-CN-3-OPr-4-Py], [BG4944: 6-CN -3-OPr-4-Py !, [BG 4945: 2-OMe-3-OPr-4-Py], [BG 4946: 5-OMe-3-OPr-4-Py], [BG4947: 6-OMe-3] -OPr-4-Py], [BG4948: 2-OPr-4-Py], [BG4949: 3-Cl-2-OPr-4-Py], [BG4950: 5-Cl-2-OPr-4-Py] ], [BG4951: 6-Cl-2-OPr-4-Py], [BG4952: 3-Me-2-OPr-4-Py], [BG4953: 5-Me-2-OPr-4-Py], [BG4954: 6-Me-2 -OPr-4-Py], [BG4955: 3-CF 3 -2-OPr-4-Py], [BG4956: 5-CF 3 -2-OPr-4-Py], _{[BG4957: 6-CF 3 -2} -OPr-4-Py], [BG4958: 3-CN-2-OPr-4-Py], [BG4959: 5-CN-2-OPr-4-Py], [ BG 4960: 6-CN-2-OPr-4-Py], [BG4961: 3-OMe-2-OPr-4-Py], [BG4962: 5-OMe-2-OPr-4-Py], [BG4963: 6-OMe-2-OPr-4-Py !, [BG 4964: 5-OPr-4-Py], [BG 4965: 3-Cl-5-OPr-4-Py], [BG 4966: 2-Cl-5- OPr-4-Py], [BG4967: 6-Cl-5-OPr-4-Py], [BG4968: 3-Me-5-OPr-4-Py], [BG4969: 2-Me-5-OPr- 4-Py], [BG4970: 6-Me-5-OPr-4-Py], [BG4971: 3-CF 3 -5-OPr-4-Py], [BG4972: 2-CF 3 -5-OPr- 4-Py], [BG 4973: 6-CF ₃ -5-OPr-4-Py], [BG 4974: 3-CN-5-OPr-4-Py], [BG 4 975: 2-CN-5-OPr-4 -Py], [BG4976: 6-CN-5-OPr-4-Py], [BG4977: 3-OMe-5-OPr-4-Py], [BG4978: 2-OMe-5-OPr-4-Py] ], [BG4979: 6-OMe-5-OPr-4-Py], [BG4980: 6-OPr-4- 4 Py], [BG4981: 3-Cl-6-OPr-4-Py], [BG4982: 2-Cl-6-OPr-4-Py], [BG4983: 5-Cl-6-OPr-4-Py] [BG4984: 3-Me-6-OPr-4-Py], [BG4985: 2-Me-6-OPr-4-Py], [BG4986: 5-Me-6-OPr-4-Py], [BG4986: 5-Me-6-OPr-4-Py], _{BG4987: 3-CF 3 -6-} OPr-4-Py], [BG4988: 2-CF 3 -6-OPr-4-Py], [BG4989: 5-CF 3 -6-OPr-4-Py], [BG4990: 3-CN-6-OPr-4-Py], [BG4991: 2-CN-6-OPr-4-Py], [BG4992: 5-CN-6-OPr-4-Py], [BG4993] : 3-OMe-6-OPr-4-Py], [BG4994: 2-OMe-6-OPr-4-Py], [BG4995: 5-OMe-6-OPr-4-Py], [BG4996: 3] -SMe-4-Py], [BG4997: 2-Cl-3-SMe-4-Py], [BG4998: 5-Cl-3-SMe-4-Py], [BG4999: 6-Cl-3-SMe -4-Py], [BG5000: 2-Me-3-SMe-4-Py],

[BG5001: 5-Me-3 -SMe-4-Py], [BG5002: 6-Me-3-SMe-4-Py], [BG5003: 2-CF 3 -3-SMe-4-Py], [ _{BG5004: 5-CF 3 -3-} SMe-4-Py], [BG5005: 6-CF 3 -3-SMe-4-Py], [BG5006: 2-CN-3-SMe-4-Py], [ BG5007: 5-CN-3-SMe-4-Py !, [BG5008: 6-CN-3-SMe-4-Py], [BG5009: 2-OMe-3-SMe-4-Py], [BG5010: 5-OMe-3-SMe-4-Py !, [BG5011: 6-OMe-3-SMe-4-Py], [BG5012: 2-SMe-4-Py], [BG5013: 3-Cl-2- SMe-4-Py !, [BG5014: 5-Cl-2-SMe-4-Py], [BG5015: 6-Cl-2-SMe-4-Py], [BG5016: 3-Me-2-SMe- 4-Py], [BG5017: 5-Me-2-SMe-4-Py], [BG5018: 6-Me-2-SMe-4-Py], [BG5019: 3-CF ₃ -2-SMe-4 -Py], [BG5020: 5- CF 3 -2-SMe-4-Py], [BG5021: 6-CF 3 -2-SMe-4-Py], [BG5022: 3-CN-2-SMe-4 -Py], [BG5023: 5-CN-2-SMe-4-Py], [BG5024: 6-CN-2-SMe-4-Py], [BG5025: 3-OMe-2-SMe-4-Py] ], [BG5026: 5-OMe-2-SMe-4-Py], [BG5027: 6-OMe-2-SMe-4-Py], [BG5028: 5-SMe-4-Py], [BG5029: 3] -Cl-5-SMe-4-Py], [BG5030: 2-Cl-5-SMe-4-Py], [BG5031: 6-Cl-5-SMe-4-Py], [BG5032: 3-Me -5-SMe-4-Py !, [BG5033: 2-Me-5-SMe-4-Py], [BG5034: 6-Me-5-SMe-4-Py], [BG5035: 3-CF _3- 5-SMe-4-Py] , [BG5036: 2-CF 3 -5-SMe-4-Py], [BG5037: 6-CF 3 -5-SMe-4-Py], [BG5038: 3-CN- 5-SMe-4-Py], [BG5039: 2-CN-5-SMe-4-Py], [B G5040: 6-CN-5-SMe-4-Py], [BG5041: 3-OMe-5-SMe-4-Py], [BG5042: 2-OMe-5-SMe-4-Py], [BG5043: 6-OMe-5-SMe-4-Py !, [BG5044: 6-SMe-4-Py], [BG5045: 3-Cl-6-SMe-4-Py], [BG5046: 2-Cl-6-] SMe-4-Py !, [BG5047: 5-Cl-6-SMe-4-Py], [BG5048: 3-Me-6-SMe-4-Py], [BG5049: 2-Me-6-SMe- 4-Py], [BG5050: 5-Me-6-SMe-4-Py], [BG5051: 3-CF 3 -6-SMe-4-Py], [BG5052: 2-CF 3 -6-SMe- 4-Py], [BG5053: 5-CF 3 -6-SMe-4-Py], [BG5054: 3-CN-6-SMe-4-Py], [BG5055: 2-CN-6-SMe-4 -Py], [BG5056: 5-CN-6-SMe-4-Py], [BG5057: 3-OMe-6-SMe-4-Py], [BG5058: 2-OMe-6-SMe-4-Py] ], [BG5059: 5-OMe -6-SMe-4-Py], [BG5060: 3-SCF 3 -4-Py], [BG5061: 2-Cl-3-SCF 3 -4-Py], [BG5062 : 5-Cl-3-SCF 3 -4-Py], [BG5063: 6-Cl-3-SCF 3 -4-Py], [BG5064: 2-Me-3-SCF 3 -4-Py], [ BG5065: 5-Me-3-SCF ₃ -4-Py !, [BG 5066: 6-Me-3-SCF ₃ -4-Py], [BG 50 67: 2-CF ₃ -3-SCF ₃ -4-Py] _{, [BG5068: 5-CF 3} -3-SCF 3 -4-Py], [BG5069: 6-CF 3 -3-SCF 3 -4-Py], [BG5070: 2-CN-3-SCF 3 -4 -Py], [BG5071: 5- CN-3-SCF 3 -4-Py], [BG5072: 6-CN-3-SCF 3 -4-Py], [BG5073: 2-OMe-3-SCF 3 - 4-Py], [BG5074: 5-OMe-3-SCF 3 -4-Py], [BG5075: 6-OMe-3-SCF 3 -4-Py], [BG5076: 2-SCF 3 -4-Py ], [BG5077: 3-Cl-2 -SCF ₃ -4-Py !, [BG5078: 5-Cl-2-SCF ₃ -4-Py], [BG5079: 6-Cl-2-SCF ₃ -4-Py], [BG 5080: 3-Me-] _{2-SCF 3 -4-Py]} , [BG5081: 5-Me-2-SCF 3 -4-Py], [BG5082: 6-Me-2-SCF 3 -4-Py], [BG5083: 3-CF ₃ -2-SCF ₃ -4-Py !, [BG 5084: 5-CF ₃ -2-SCF ₃ -4-Py], [BG 50 85: 6-CF ₃ -2-SCF ₃ -4-Py], [BG 50 86] : 3-CN-2-SCF 3 -4-Py], [BG5087: 5-CN-2-SCF 3 -4-Py], [BG5088: 6-CN-2-SCF 3 -4-Py], [ BG5089: 3-OMe-2- SCF 3 -4-Py], [BG5090: 5-OMe-2-SCF 3 -4-Py], [BG5091: 6-OMe-2-SCF 3 -4-Py], _{[BG5092: 5-SCF 3 -4} -Py], [BG5093: 3-Cl-5-SCF 3 -4-Py], [BG5094: 2-Cl-5-SCF 3 -4-Py], [BG5095: 6-Cl-5-SCF ₃ -4-Py !, [BG5096: 3-Me-5-SCF ₃ -4-Py], [BG5097: 2-Me-5-SCF ₃ -4-Py], [BG5098] : 6-Me-5-SCF 3 -4-Py], [BG5099: 3-CF 3 -5-SCF 3 -4-Py], [BG5100: 2-CF 3 -5-SCF 3 -4-Py] ,

_{[BG5101: 6-CF 3 -5} -SCF 3 -4-Py], [BG5102: 3-CN-5-SCF 3 -4-Py], [BG5103: 2-CN-5-SCF 3 -4-Py ], [BG 5104: 6-CN-5-SCF ₃ -4-Py], [BG 5105: 3-OMe-5-SCF ₃ -4-Py], [BG 5106: 2-OMe-5-SCF ₃ -4-] Py], [BG5107: 6- OMe-5-SCF 3 -4-Py], [BG5108: 6-SCF 3 -4-Py], [BG5109: 3-Cl-6-SCF 3 -4-Py], [BG5110: 2-Cl-6 -SCF 3 -4-Py], [BG5111: 6-Cl-6-SCF 3 -4-Py], [BG5112: 3-Me-6-SCF 3 -4-Py] , [BG5113: 2-Me- 6-SCF 3 -4-Py], [BG5114: 6-Me-6-SCF 3 -4-Py], [BG5115: 3-CF 3 -6-SCF 3 -4- Py], [BG5116: 2- CF 3 -6-SCF 3 -4-Py], [BG5117: 6-CF 3 -6-SCF 3 -4-Py], [BG5118: 3-CN-6-SCF 3 -4-Py], [BG5119: 2-CN-6-SCF 3 -4-Py], [BG5120: 6-CN-6-SCF 3 -4-Py], [BG5121: 3-OMe-6-SCF ₃ -4-Py !, [BG 5122: 2-OMe-6-SCF ₃ -4-Py], [BG 5123: 6-OMe-6-SCF ₃ -4-Py], [BG 5124: 3-S (O)] Me-4-Py !, [BG5125: 2-Cl-3-S (O) Me-4-Py], [BG5126: 5-Cl-3-S (O) Me-4-Py], [BG5127: 6-Cl-3-S (O) Me-4-Py], [BG5128: 2-Me-3-S (O) Me-4-Py], [BG5129: 5-Me-3-S (O) Me-4-Py], [ BG5130: 6-Me-3-S (O) Me-4-Py], [BG5131: 2-CF 3 -3-S (O) Me-4-Py], [BG5132 _{: 5-CF 3 -3-S} (O) Me-4-Py], [BG5133: 6-CF 3 -3-S (O) Me-4-Py], [BG5134: 2-CN-3-S (O) Me-4-Py], [BG5135: 5-CN-3-S (O) Me-4-Py], [BG 5136: 6-CN-3-S (O) Me-4-Py], [BG5137: 2-OMe-3-S (O) Me-4-Py], [BG5138: 5-OMe-3-S ( O) Me-4-Py], [BG5139: 6-OMe-3-S (O) Me-4-Py], [BG5140: 2-S (O) Me-4-Py], [BG5141: 3- Cl-2-S (O) Me-4-Py], [BG5142: 5-Cl-2-S (O) Me-4-Py], [BG5143: 6-Cl-2-S (O) Me- 4-Py !, [BG5144: 3-Me-2-S (O) Me-4-Py], [BG5145: 5-Me-2-S (O) Me-4-Py], [BG5146: 6-] Me-2-S (O) Me-4-Py], [BG5147: 3-CF 3 -2-S (O) Me-4-Py], [BG5148: 5-CF 3 -2-S (O) Me-4-Py], [ BG5149: 6-CF 3 -2-S (O) Me-4-Py], [BG5150: 3-CN-2-S (O) Me-4-Py], [BG5151 : 5-CN-2-S (O) Me-4-Py], [BG5152: 6-CN-2-S (O) Me-4-Py], [BG5153: 3-OMe-2-S (O) ) Me-4-Py], [BG5154: 5-OMe-2-S (O) Me-4-Py], [BG5155: 6-OMe-2-S (O) Me-4-Py], [BG5156] : 5-S (O) Me-4-Py], [BG5157: 3-Cl-5-S (O) Me-4-Py], [BG5158: 2-Cl-5-S (O) Me-4 -Py], [BG5159: 6-Cl-5-S (O) Me-4-Py], [BG5160: 3-Me-5-S (O) Me-4-Py], [BG5161: 2-Me -5-S (O) Me-4-Py], [BG5162: 6-Me-5-S (O) Me-4-Py], [BG5163: 3-CF ₃ -5-S (O) Me- 4-Py], [BG5164: 2-CF 3 -5-S (O) Me-4-Py], [BG5165: 6-CF 3 -5-S (O) Me-4-Py], [BG5166: 3-CN-5-S (O) Me-4-Py], [BG5167: 2-CN-5-S (O) Me-4-Py], [BG5168: 6-CN-5-S (O) Me-4-Py !, [BG5169: 3-OMe-5-S (O) Me-4-Py], [BG5170: 2-OMe-5-S (O) Me-4-Py], [BG5171] : 6-OMe-5-S (O) Me-4-Py], [BG5172: 6-S (O) Me-4-Py], [BG5173: 3-Cl-6-S (O) Me-4 -Py], [BG5174: 2-Cl-6-S (O) Me-4-Py], [BG5175: 5-Cl-6-S (O) Me-4-Py], [BG5176: 3-Me -6-S (O) Me-4-Py], [BG5177: 2-Me-6-S (O) Me-4-Py], [BG5178: 5-Me-6-S (O) Me-4 -Py], [BG5179: 3- CF 3 -6-S (O) Me-4-Py], [BG5180: 2-CF 3 -6-S (O) Me-4-Py], [BG5181: 5 _{-CF 3 -6-S (O)} Me-4-Py], [BG5182: 3-CN-6-S (O) Me-4-Py], [BG5183: 2-CN-6-S (O) Me-4-Py !, [BG5184: 5-CN-6-S (O) Me-4-Py], [BG5185: 3-OMe-6-S (O) Me-4-Py], [BG5186: 2-OMe-6-S ( O) Me-4-Py], [BG5187: 5-OMe-6-S (O) Me-4-Py], [BG5188: 3-S (O) CF 3 -4 -Py], [BG5189: 2- Cl-3-S (O) CF 3 -4-Py], [BG5190: 5-Cl-3-S (O) CF 3 -4-Py], [BG5191: 6 -Cl-3-S (O) CF 3 -4-Py], [BG5192: 2-Me-3-S (O) CF 3 -4-Py], [BG5193: 5-Me-3-S (O ) CF ₃ -4-Py !, [BG 5194: 6-Me-3-S (O) CF ₃ -4-Py], [BG 5195: 2-CF ₃ -3-S (O) CF ₃ -4-Py] ], [BG5196: 5-CF 3 -3-S (O) CF 3 -4-Py], [BG5197: 6-CF 3 -3-S (O) CF 3 -4-Py], [BG5198: 2 -CN-3-S (O) CF 3 -4-Py], [BG5199: 5-CN-3-S (O) CF 3 -4-Py], [BG5200: 6-CN-3-S (O ) CF ₃ -4-Py],

[BG5201: 2-OMe-3 -S (O) CF 3 -4-Py], [BG5202: 5-OMe-3-S (O) CF 3 -4-Py], [BG5203: 6-OMe-3 _{-S (O) CF 3 -4-} Py], [BG5204: 2-S (O) CF 3 -4-Py], [BG5205: 3-Cl-2-S (O) CF 3 -4-Py] , [BG5206: 5-Cl- 2-S (O) CF 3 -4-Py], [BG5207: 6-Cl-2-S (O) CF 3 -4-Py], [BG5208: 3-Me- _{2-S (O) CF 3} -4-Py], [BG5209: 5-Me-2-S (O) CF 3 -4-Py], [BG5210: 6-Me-2-S (O) CF 3 -4-Py], [BG5211: 3-CF 3 -2-S (O) CF 3 -4-Py], [BG5212: 5-CF 3 -2-S (O) CF 3 -4-Py], _{[BG5213: 6-CF 3 -2} -S (O) CF 3 -4-Py], [BG5214: 3-CN-2-S (O) CF 3 -4-Py], [BG5215: 5-CN- _{2-S (O) CF 3} -4-Py], [BG5216: 6-CN-2-S (O) CF 3 -4-Py], [BG5217: 3-OMe-2-S (O) CF 3 -4-Py], [BG5218: 5-OMe-2-S (O) CF 3 -4-Py], [BG5219: 6-OMe-2-S (O) CF 3 -4-Py], [BG5220 : 5-S (O) CF 3 -4-Py], [BG5221: 3-Cl-5-S (O) CF 3 -4-Py], [BG5222: 2-Cl-5-S (O) CF _{3 -4-Py], [BG5223} : 6-Cl-5-S (O) CF 3 -4-Py], [BG5224: 3-Me-5-S (O) CF 3 -4-Py], [ BG5225: 2-Me-5- S (O) CF 3 -4-Py], [BG5226: 6-Me-5-S (O) CF 3 -4-Py], [BG5227: 3-CF 3 -5 _{-S (O) CF 3 -4-} Py], [BG5228: 2-CF 3 -5-S (O) CF 3 -4-Py], [BG5229: 6-CF 3 -5-S (O) CF _{3 -4-Py], [BG5230} : 3-CN-5-S (O) CF 3 -4-Py], [BG5231: 2-CN-5-S (O) CF 3 -4-Py], [ BG5232: 6-CN-5-S (O) CF _3- 4-Py], [BG5233: 3-OMe-5-S (O) CF 3 -4-Py], [BG5234: 2-OMe-5-S (O) CF 3 -4-Py], [BG5235: 6-OMe-5-S ( O) CF 3 -4-Py], [BG5236: 6-S (O) CF 3 -4-Py], [BG5237: 3-Cl-6-S (O) CF 3 -4-Py], [BG5238: 2-Cl-6-S (O) CF 3 -4-Py], [BG5239: 5-Cl-6-S (O) CF 3 -4-Py], [BG5240 : 3-Me-6-S (O) CF 3 -4-Py], [BG5241: 2-Me-6-S (O) CF 3 -4-Py], [BG5242: 5-Me-6-S _{(O) CF 3 -4-Py} ], [BG5243: 3-CF 3 -6-S (O) CF 3 -4-Py], [BG5244: 2-CF 3 -6-S (O) CF 3 - 4-Py], [BG5245: 5-CF 3 -6-S (O) CF 3 -4-Py], [BG5246: 3-CN-6-S (O) CF 3 -4-Py], [BG5247 : 2-CN-6-S (O) CF 3 -4-Py], [BG5248: 5-CN-6-S (O) CF 3 -4-Py], [BG5249: 3-OMe-6-S _{(O) CF 3 -4-Py} ], [BG5250: 2-OMe-6-S (O) CF 3 -4-Py], [BG5251: 5-OMe-6-S (O) CF 3 -4- Py], [BG5252: 3-S (O) ₂ Me-4-Py], [BG5253: 2-Cl-3-S (O) ₂ Me-4-Py], [BG5254: 5-Cl-3- _{S (O) 2 Me-4} -Py], [BG5255: 6-Cl-3-S (O) 2 Me-4-Py], [BG5256: 2-Me-3-S (O) 2 Me-4 -Py], [BG5257: 5-Me-3-S (O) ₂ Me-4-Py], [BG5258: 6-Me-3-S (O) ₂ Me-4-Py], [BG5259: 2] _{-CF 3 -3-S (O)} 2 Me-4-Py], [BG5260: 5-CF 3 -3-S (O) 2 Me-4-Py], [BG5261: 6-CF 3 -3- _{S (O) 2 Me-4} -Py], [BG5262: 2-CN-3-S (O) 2 Me-4-Py], [BG5263: 5-CN-3-S (O) 2 Me-4 -Py], [BG5264: 6-CN-3-S (O) ₂ Me-4-Py], [BG5265: 2-OMe-3-S (O) ₂ Me-4-Py], [BG5266: 5-OMe-3-S (O) ₂ Me-4-Py], [BG5267: 6-OMe-3 -S (O) 2 Me-4-Py], [BG5268: 2-S (O) 2 Me-4-Py], [BG5269: 3-Cl-2-S (O ) ₂ Me-4-Py], [BG5270: 5-Cl-2-S (O) ₂ Me-4-Py], [BG5271: 6-Cl-2-S (O) ₂ Me-4-Py] , [BG5272: 3-Me- 2-S (O) 2 Me-4-Py], [BG5273: 5-Me-2-S (O) 2 Me-4-Py], [BG5274: 6-Me- _{2-S (O) 2 Me} -4-Py], [BG5275: 3-CF 3 -2-S (O) 2 Me-4-Py], [BG5276: 5-CF 3 -2-S (O) _{2 Me-4-Py],} [BG5277: 6-CF 3 -2-S (O) 2 Me-4-Py], [BG5278: 3-CN-2-S (O) 2 Me-4-Py] , [BG5279: 5-CN- 2-S (O) 2 Me-4-Py], [BG5280: 6-CN-2-S (O) 2 Me-4-Py], [BG5281: 3-OMe- _{2-S (O) 2 Me} -4-Py], [BG5282: 5-OMe-2-S (O) 2 Me-4-Py], [BG5283: 6-OMe-2-S (O) 2 Me -4-Py !, [BG 5284: 5-S (O) ₂ Me-4-Py], [BG 5285: 3-Cl-5-S (O) ₂ Me-4-Py], [BG 5286: 2-Cl] _{-5-S (O) 2 Me} -4-Py], [BG5287: 6-Cl-5-S (O) 2 Me-4-Py], [BG5288: 3-Me-5-S (O) 2 Me-4-Py], [BG5289: 2-Me-5-S (O) ₂ Me-4-Py], [BG5290: 6-Me-5-S (O) ₂ Me-4-Py], _{BG5291: 3-CF 3 -5-} S (O) 2 Me-4-Py], [BG5292: 2-CF 3 -5-S (O) 2 Me-4-Py], [BG5293: 6-CF 3 _{-5-S (O) 2 Me} -4-Py], [BG5294: 3-CN-5-S (O) 2 Me-4-Py], [BG5295: 2-CN-5-S (O) 2 Me-4-Py], [BG5296: 6-CN- _{5-S (O) 2 Me} -4-Py], [BG5297: 3-OMe-5-S (O) 2 Me-4-Py], [BG5298: 2-OMe-5-S (O) 2 Me -4-Py], [BG5299: 6-OMe-5-S (O) ₂ Me-4-Py], [BG5300: 6-S (O) ₂ Me-4-Py],

[BG5301: 3-Cl-6 -S (O) 2 Me-4-Py], [BG5302: 2-Cl-6-S (O) 2 Me-4-Py], [BG5303: 5-Cl-6 _{-S (O) 2 Me-4} -Py], [BG5304: 3-Me-6-S (O) 2 Me-4-Py], [BG5305: 2-Me-6-S (O) 2 Me- 4-Py], [BG5306: 5-Me-6-S (O) 2 Me-4-Py], [BG5307: 3-CF 3 -6-S (O) 2 Me-4-Py], [BG5308 _{: 2-CF 3 -6-S} (O) 2 Me-4-Py], [BG5309: 5-CF 3 -6-S (O) 2 Me-4-Py], [BG5310: 3-CN-6 _{-S (O) 2 Me-4} -Py], [BG5311: 2-CN-6-S (O) 2 Me-4-Py], [BG5312: 5-CN-6-S (O) 2 Me- 4-Py], [BG5313: 3-OMe-6-S (O) ₂ Me-4-Py], [BG5314: 2-OMe-6-S (O) ₂ Me-4-Py], [BG5315: 5-OMe-6-S ( O) 2 Me-4-Py], [BG5316: 3-S (O) 2 CF 3 -4-Py], [BG5317: 2-Cl-3-S (O) 2 _{CF 3 -4-Py], [} BG5318: 5-Cl-3-S (O) 2 CF 3 -4-Py], [BG5319: 6-Cl-3-S (O) 2 CF 3 -4-Py ], [BG5320: 2-Me -3-S (O) 2 CF 3 -4-Py], [BG5321: 5-Me-3-S (O) 2 CF 3 -4-Py], [BG5322: 6 -Me-3-S (O) 2 CF 3 -4-Py], [BG5323: 2-CF 3 -3-S (O) 2 CF 3 -4-Py], [BG5324: 5-CF 3 -3 _{-S (O) 2 CF 3 -4} -Py], [BG5325: 6-CF 3 -3-S (O) 2 CF 3 -4-Py], [BG5326: 2-CN-3-S (O) ₂ CF ₃ -4-Py, [BG 5327: 5-CN-3-S (O) ₂ CF ₃ -4-Py], [BG 5328: 6-CN-3-S (O) ₂ CF ₃ -4- Py], [BG 5329: 2-OMe-3-S (O) ₂ CF ₃ -4-Py], [BG 5330: 5-OMe-3-S (O) ₂ CF ₃ -4-Py], [BG 5 33 1 : 6-OMe-3-S (O) 2 CF 3 -4-Py], [BG5332: 2-S (O) 2 CF 3 -4-Py], [BG5333: 3-Cl-2-S (O _{) 2 CF 3 -4-Py]} , [BG5334: 5-Cl-2-S (O) 2 CF 3 -4-Py], [BG5335: 6-Cl-2-S (O) 2 CF 3 -4 -Py], [BG 5336: 3-Me-2-S (O) ₂ CF ₃ -4-Py], [BG 5337: 5-Me-2-S (O) ₂ CF ₃ -4-Py], [BG 5 338] : 6-Me-2-S (O) 2 CF 3 -4-Py], [BG5339: 3-CF 3 -2-S (O) 2 CF 3 -4-Py], [BG5340: 5-CF 3 _{-2-S (O) 2 CF} 3 -4-Py], [BG5341: 6-CF 3 -2-S (O) 2 CF 3 -4-Py], [BG5342: 3-CN-2-S ( O) ₂ CF ₃ -4-Py, [BG 5343: 5-CN-2-S (O) ₂ CF ₃ -4-Py], [BG 5344: 6-CN-2-S (O) ₂ CF _3- 4-Py], [BG 5345: 3-OMe-2-S (O) ₂ CF ₃ -4-Py], [BG 5346: 5-OMe-2-S (O) ₂ CF ₃ -4-Py], BG5347: 6-OMe-2- S (O) 2 CF 3 -4-Py], [BG5348: 5-S (O) 2 CF 3 -4-Py], [BG5349: 3-Cl-5-S ( O) ₂ CF ₃ -4-Py], [BG 5350: 2-Cl-5-S (O) ₂ CF ₃ -4-Py], [BG 5351: 6-Cl-5-S (O) ₂ CF _3- 4-Py], [BG5352: 3-Me-5-S (O) 2 CF 3 -4-Py], [BG5353: 2-Me-5-S (O) 2 CF 3 -4-Py], [ BG 5354: 6-Me-5-S (O) ₂ CF ₃ -4-Py, [BG 5 355: 3-CF ₃ -5- S (O) ₂ CF ₃ -4-Py], [BG 5356: 2-CF _{3 -5-S (O) 2} CF 3 -4-Py], [BG5357: 6-CF 3 -5-S (O) 2 CF 3 -4-Py], [BG5358: 3-CN-5-S _{(O) 2 CF 3 -4-} Py], [BG5359: 2-CN-5-S (O) 2 CF 3 -4-Py], [BG5360: 6 -CN-5-S (O) 2 CF 3 -4-Py], [BG5361: 3-OMe-5-S (O) 2 CF 3 -4-Py], [BG5362: 2-OMe-5-S _{(O) 2 CF 3 -4-} Py], [BG5363: 6-OMe-5-S (O) 2 CF 3 -4-Py], [BG5364: 6-S (O) 2 CF 3 -4-Py ], [BG5365: 3-Cl -6-S (O) 2 CF 3 -4-Py], [BG5366: 2-Cl-6-S (O) 2 CF 3 -4-Py], [BG5367: 5 -Cl-6-S (O) 2 CF 3 -4-Py], [BG5368: 3-Me-6-S (O) 2 CF 3 -4-Py], [BG5369: 2-Me-6-S _{(O) 2 CF 3 -4-} Py], [BG5370: 5-Me-6-S (O) 2 CF 3 -4-Py], [BG5371: 3-CF 3 -6-S (O) 2 CF ₃ -4-Py], [BG5372: 2-CF ₃ -6-S (O) ₂ CF ₃ -4-Py], [BG5373: 5-CF ₃ -6-S (O) ₂ CF ₃ -4- Py], [BG5374: 3- CN-6-S (O) 2 CF 3 -4-Py], [BG5375: 2-CN-6-S (O) 2 CF 3 -4-Py], [BG5376: 5-CN-6-S ( O) 2 CF 3 -4-Py], [BG5377: 3-OMe-6-S (O) 2 CF 3 -4-Py], [BG5378: 2-OMe-6- _{S (O) 2 CF 3 -4} -Py], [BG5379: 5-OMe-6-S (O) 2 CF 3 -4-Py], [BG5380: 3-CN-4-Py], [BG5381: 2-Cl-3-CN-4-Py !, [BG5382: 5-Cl-3-CN-4-Py], [BG5383: 6-Cl-3-CN-4-Py], [BG5384: 2-] Me-3-CN-4- Py], [BG5385: 5-Me-3-CN-4-Py], [BG5386: 6-Me-3-CN-4-Py], [BG5387: 2-CF 3 -3-CN-4-Py] , [BG5388: 5-CF 3 -3-CN-4-Py], [BG5389: 6-CF 3 -3-CN-4-Py], [BG5390: 2-CN -3-CN-4-Py !, [BG5391: 5-CN-3-CN-4-Py], [BG5392: 6-CN-3-CN-4-Py], [BG 5393: 2-OMe-3-CN-4-Py !, [BG5394: 5-OMe-3-CN-4-Py], [BG5395: 6-OMe-3-CN-4-Py], [BG5396: 2-CN-4-Py], [BG5397: 3-Cl-2-CN-4-Py], [BG5398: 5-Cl-2-CN-4-Py], [BG5399: 6-Cl-2-] CN-4-Py], [BG5400: 3-Me-2-CN-4-Py],

[BG5401: 5-Me-2-CN-4-Py], [BG5402: 6-Me-2-CN-4-Py], [BG5403: 3-CF ₃ -2-CN-4-Py], [BG _{BG5404: 5-CF 3 -2-} CN-4-Py], [BG5405: 6-CF 3 -2-CN-4-Py], [BG5406: 3-CN-2-CN-4-Py], [ BG5407: 5-CN-2-CN-4-Py, [BG5408: 6-CN-2-CN-4-Py], [BG5409: 3-OMe-2-CN-4-Py], [BG5410: 5-OMe-2-CN-4-Py, [BG5411: 6-OMe-2-CN-4-Py], [BG5412: 5-CN-4-Py], [BG5413: 3-Cl-5- CN-4-Py !, [BG5414: 2-Cl-5-CN-4-Py], [BG5415: 6-Cl-5-CN-4-Py], [BG5416: 3-Me-5-CN-] 4-Py], [BG5417: 2-Me-5-CN-4-Py], [BG5418: 6-Me-5-CN-4-Py], [BG5419: 3-CF 3 -5-CN-4 -Py], [BG5420: 2- CF 3 -5-CN-4-Py], [BG5421: 6-CF 3 -5-CN-4-Py], [BG5422: 3-CN-5-CN-4 -Py], [BG5423: 2-CN-5-CN-4-Py], [BG5424: 6-CN-5-CN-4-Py], [BG5425: 3-OMe-5-CN-4-Py] ], [BG5426: 2-OMe-5-CN-4-Py], [BG5427: 6-OMe-5-CN-4-Py], [BG5428: 6-CN-4-Py], [BG5429: 3] -Cl-6-CN-4-Py], [BG5430: 2-Cl-6-CN-4-Py], [BG5431: 5-Cl-6-CN-4-Py], [BG5432: 3-Me -6-CN-4-Py !, [BG5433: 2-Me-6-CN-4-Py], [BG5434: 5-Me-6-CN-4-Py], [BG5435: 3-CF _3- 6-CN-4-Py], [BG 5436: 2-CF ₃ -6-CN-4-Py], [BG 5437: 5-CF ₃ -6-CN-4-Py], [BG 5438: 3-CN- 6-CN-4-Py], [BG5439: 2-CN-6-CN-4-Py], [BG5440: 5-CN-6-CN-4-Py], [BG5441: 3-OMe-6-] C N-4-Py], [BG5442: 2-OMe-6-CN-4-Py], [BG5443: 5-OMe-6-CN-4-Py], [BG5444: 3-COOMe-4-Py] [BG5445: 2-Cl-3-COOMe-4-Py], [BG5446: 5-Cl-3-COOMe-4-Py], [BG5447: 6-Cl-3-COOMe-4-Py], [BG5 445: BG5448: 2-Me-3-COOMe-4-Py], [BG5449: 5-Me-3-COOMe-4-Py], [BG5450: 6-Me-3-COOMe-4-Py], [BG5451: _{2-CF 3 -3-COOMe-} 4-Py], [BG5452: 5-CF 3 -3-COOMe-4-Py], [BG5453: 6-CF 3 -3-COOMe-4-Py], [BG5454 : 2-CN-3-COOMe-4-Py], [BG5455: 5-CN-3-COOMe-4-Py], [BG5456: 6-CN-3-COOMe-4-Py], [BG5457: 2] -OMe-3-COOMe-4-Py], [BG5458: 5-OMe-3-COOMe-4-Py], [BG5459: 6-OMe-3-COOMe-4-Py], [BG5460: 2-COOMe -4-Py !, [BG5461: 3-Cl-2-COOMe-4-Py], [BG5462: 5-Cl-2-COOMe-4-Py], [BG5463: 6-Cl-2-COOMe-4] -Py], [BG5464: 3-Me-2-COOMe-4-Py], [BG5465: 5-Me-2-COOMe-4-Py], [BG5466: 6-Me-2-COOMe-4-Py] ], [BG5467: 3-CF 3 -2-COOMe-4-Py], [BG5468: 5-CF 3 -2-COOMe-4-Py], [BG5469: 6-CF 3 -2-COOMe-4- Py], [BG5470: 3-CN-2-COOMe-4-Py], [BG5471: 5-CN-2-COOMe-4-Py], [BG5472: 6-CN-2-COOMe-4-Py] [BG5473: 3-OMe-2-COOMe-4-Py], [BG5474: 5-OMe-2-COOMe-4-Py], [BG5475: 6-OMe-2-COOMe-4-Py], [BG5 475: BG 5476: 5-COOMe-4-Py], [BG5477: 3-Cl-5-COOMe-4-Py], [BG5478: 2-Cl-5- COOMe-4-Py !, [BG5479: 6-Cl-5-COOMe-4-Py], [BG5480: 3-Me-5-COOMe-4-Py], [BG5481: 2-Me-5-COOMe- 4-Py], [BG5482: 6-Me-5-COOMe-4-Py], [BG5483: 3-CF 3 -5-COOMe-4-Py], [BG5484: 2-CF 3 -5-COOMe- 4-Py], [BG5485: 6-CF 3 -5-COOMe-4-Py], [BG5486: 3-CN-5-COOMe-4-Py], [BG5487: 2-CN-5-COOMe-4 -Py], [BG5488: 6-CN-5-COOMe-4-Py], [BG5489: 3-OMe-5-COOMe-4-Py], [BG5490: 2-OMe-5-COOMe-4-Py] ], [BG5491: 6-OMe-5-COOMe-4-Py], [BG5492: 6-COOMe-4-Py], [BG5493: 3-Cl-6-COOMe-4-Py], [BG5494: 2] -Cl-6-COOMe-4-Py], [BG5495: 5-Cl-6-COOMe-4-Py], [BG5496: 3-Me-6-COOMe-4-Py], [BG5497: 2-Me -6-COOMe-4-Py] , [BG5498: 5-Me-6-COOMe-4-Py], [BG5499: 3-CF 3 -6-COOMe-4-Py], [BG5500: 2-CF 3 -6-COOMe-4-Py],

_{[BG5501: 5-CF 3 -6} -COOMe-4-Py], [BG5502: 3-CN-6-COOMe-4-Py], [BG5503: 2-CN-6-COOMe-4-Py], [ BG5504: 5-CN-6-COOMe-4-Py !, [BG5505: 3-OMe-6-COOMe-4-Py], [BG5506: 2-OMe-6-COOMe-4-Py], [BG5507: 5-OMe-6-COOMe- 4-Py], [BG5508: 3-NO 2 -4-Py], [BG5509: 2-Cl-3-NO 2 -4-Py], [BG5510: 5-Cl- 3-NO ₂ -4-Py], [BG5511: 6-Cl-3-NO ₂ -4-Py], [BG5512: 2-Me-3-NO ₂ -4-Py], [BG5513: 5-Me -3-NO ₂ -4-Py !, [BG5514: 6-Me-3-NO ₂ -4-Py], [BG5515: 2-CF ₃ -3-NO ₂ -4-Py], [BG 5516: 5] _{-CF 3 -3-NO 2 -4-} Py], [BG5517: 6-CF 3 -3-NO 2 -4-Py], [BG5518: 2-CN-3-NO 2 -4-Py], [ BG5519: 5-CN-3- NO 2 -4-Py], [BG5520: 6-CN-3-NO 2 -4-Py], [BG5521: 2-OMe-3-NO 2 -4-Py], [BG5522: 5-OMe-3 -NO 2 -4-Py], [BG5523: 6-OMe-3-NO 2 -4-Py], [BG5524: 2-NO 2 -4-Py], [BG5525: 3-Cl-2-NO ₂ -4-Py !, [BG 5526: 5-Cl 2-NO ₂ -4-Py], [BG 5527: 6-Cl 2-NO ₂ -4-Py], [BG 5528] : 3-Me-2-NO 2 -4-Py], [BG5529: 5-Me-2-NO 2 -4-Py], [BG5530: 6-Me-2-NO 2 -4-Py], [ _{BG5531: 3-CF 3 -2-} NO 2 -4-Py], [BG5532: 5-CF 3 -2-NO 2 -4-Py], [BG5533: 6-CF 3 -2-NO 2 -4- Py], [BG5534: 3- CN-2-NO 2 -4-Py], [BG5535: 5-CN-2-NO 2 -4-Py], [BG5536: 6-CN-2-NO 2 -4 -Py], [BG5537: 3-O _{Me-2-NO 2 -4-} Py], [BG5538: 5-OMe-2-NO 2 -4-Py], [BG5539: 6-OMe-2-NO 2 -4-Py], [BG5540: 5 _{-NO 2 -4-Py], [} BG5541: 3-Cl-5-NO 2 -4-Py], [BG5542: 2-Cl-5-NO 2 -4-Py], [BG5543: 6-Cl- _{5-NO 2 -4-Py]} , [BG5544: 3-Me-5-NO 2 -4-Py], [BG5545: 2-Me-5-NO 2 -4-Py], [BG5546: 6-Me -5-NO ₂ -4-Py], [BG5547: 3-CF ₃ -5-NO ₂ -4-Py], [BG 5548: 2-CF ₃ -5-NO ₂ -4-Py], [BG 5549: _{6-CF 3 -5-NO 2} -4-Py], [BG5550: 3-CN-5-NO 2 -4-Py], [BG5551: 2-CN-5-NO 2 -4-Py], [ BG5552: 6-CN-5- NO 2 -4-Py], [BG5553: 3-OMe-5-NO 2 -4-Py], [BG5554: 2-OMe-5-NO 2 -4-Py], [BG5555: 6-OMe-5 -NO 2 -4-Py], [BG5556: 6-NO 2 -4-Py], [BG5557: 3-Cl-6-NO 2 -4-Py], [BG5558: _{2-Cl-6-NO 2} -4-Py], [BG5559: 5-Cl-6-NO 2 -4-Py], [BG5560: 3-Me-6-NO 2 -4-Py], [BG5561 : 2-Me-6-NO 2 -4-Py], [BG5562: 5-Me-6-NO 2 -4-Py], [BG5563: 3-CF 3 -6-NO 2 -4-Py], _{[BG5564: 2-CF 3 -6} -NO 2 -4-Py], [BG5565: 5-CF 3 -6-NO 2 -4-Py], [BG5566: 3-CN-6-NO 2 -4- Py], [BG5567: 2- CN-6-NO 2 -4-Py], [BG5568: 5-CN-6-NO 2 -4-Py], [BG5569: 3-OMe-6-NO 2 -4 -Py], [BG5570: 2- OMe-6-NO 2 -4-Py], [BG5571: 5-OMe-6-NO 2 -4-Py], [BG5572: 3-NH 2 -4-Py] [BG5573: 2-Cl-3-NH ₂ -4-Py], [BG5574: 5-Cl-3 -NH 2 -4-Py], [BG5575: 6-Cl-3-NH 2 -4-Py], [BG5576: 2-Me-3-NH 2 -4-Py] , [BG5577: 5-Me- 3-NH 2 -4-Py], [BG5578: 6-Me-3-NH 2 -4-Py], [BG5579: 2-CF 3 -3-NH 2 -4- Py], [BG5580: 5- CF 3 -3-NH 2 -4-Py], [BG5581: 6-CF 3 -3-NH 2 -4-Py], [BG5582: 2-CN-3-NH 2 -4-Py], [BG5583: 5-CN-3-NH 2 -4-Py], [BG5584: 6-CN-3-NH 2 -4-Py], [BG5585: 2-OMe-3-NH _{2 -4-Py], [BG5586} : 5-OMe-3-NH 2 -4-Py], [BG5587: 6-OMe-3-NH 2 -4-Py], [BG5588: 2-NH 2 -4 -Py], [BG5589: 3- Cl-2-NH 2 -4-Py], [BG5590: 5-Cl-2-NH 2 -4-Py], [BG5591: 6-Cl-2-NH 2 - 4-Py], [BG5592: 3-Me-2-NH 2 -4-Py], [BG5593: 5-Me-2-NH 2 -4-Py], [BG5594: 6-Me-2-NH 2 -4-Py], [BG5595: 3-CF ₃ -2-NH ₂ -4-Py], [BG5596: 5-CF ₃ -2-NH ₂ -4-Py], [BG 5597: 6-CF _{3- 2-NH 2 -4-Py]} , [BG5598: 3-CN-2-NH 2 -4-Py], [BG5599: 5-CN-2-NH 2 -4-Py], [BG5600: 6-CN -2-NH ₂ -4-Py],

[BG5601: 3-OMe-2 -NH 2 -4-Py], [BG5602: 5-OMe-2-NH 2 -4-Py], [BG5603: 6-OMe-2-NH 2 -4-Py] _{, [BG5604: 5-NH 2} -4-Py], [BG5605: 3-Cl-5-NH 2 -4-Py], [BG5606: 2-Cl-5-NH 2 -4-Py], [BG5607 : 6-Cl-5-NH 2 -4-Py], [BG5608: 3-Me-5-NH 2 -4-Py], [BG5609: 2-Me-5-NH 2 -4-Py], [ BG5610: 6-Me-5- NH 2 -4-Py], [BG5611: 3-CF 3 -5-NH 2 -4-Py], [BG5612: 2-CF 3 -5-NH 2 -4-Py ], [BG5613: 6-CF 3 -5-NH 2 -4-Py], [BG5614: 3-CN-5-NH 2 -4-Py], [BG5615: 2-CN-5-NH 2 -4 -Py], [BG5616: 6- CN-5-NH 2 -4-Py], [BG5617: 3-OMe-5-NH 2 -4-Py], [BG5618: 2-OMe-5-NH 2 - 4-Py], [BG5619: 6-OMe-5-NH 2 -4-Py], [BG5620: 6-NH 2 -4-Py], [BG5621: 3-Cl-6-NH 2 -4-Py ], [BG5622: 2-Cl -6-NH 2 -4-Py], [BG5623: 5-Cl-6-NH 2 -4-Py], [BG5624: 3-Me-6-NH 2 -4- Py], [BG5625: 2- Me-6-NH 2 -4-Py], [BG5626: 5-Me-6-NH 2 -4-Py], [BG5627: 3-CF 3 -6-NH 2 - 4-Py], [BG5628: 2-CF 3 -6-NH 2 -4-Py], [BG5629: 5-CF 3 -6-NH 2 -4-Py], [BG5630: 3-CN-6- _{NH 2 -4-Py], [} BG5631: 2-CN-6-NH 2 -4-Py], [BG5632: 5-CN-6-NH 2 -4-Py], [BG5633: 3-OMe-6 _{-NH 2 -4-Py], [} BG5634: 2-OMe-6-NH 2 -4-Py], [BG5635: 5-OMe-6-NH 2 -4-Py], [BG5636: 3-NHMe- 4-Py], [BG5637: 2-Cl-3-NH Me-4-Py !, [BG5638: 5-Cl-3-NHMe-4-Py], [BG5639: 6-Cl-3-NHMe-4-Py], [BG5640: 2-Me-3-NHMe- 4-Py], [BG5641: 5-Me-3-NHMe-4-Py], [BG5642: 6-Me-3-NHMe-4-Py], [BG5643: 2-CF 3 -3-NHMe-4 -Py], [BG5644: 5- CF 3 -3-NHMe-4-Py], [BG5645: 6-CF 3 -3-NHMe-4-Py], [BG5646: 2-CN-3-NHMe-4 -Py], [BG5647: 5-CN-3-NHMe-4-Py], [BG5648: 6-CN-3-NHMe-4-Py], [BG5649: 2-OMe-3-NHMe-4-Py] ], [BG5650: 5-OMe-3-NHMe-4-Py], [BG5651: 6-OMe-3-NHMe-4-Py], [BG5652: 2-NHMe-4-Py], [BG5653: 3] -Cl-2-NHMe-4-Py], [BG5654: 5-Cl-2-NHMe-4-Py], [BG5655: 6-Cl-2-NHMe-4-Py], [BG5656: 3-Me -2-NHMe-4-Py !, [BG5657: 5-Me-2-NHMe-4-Py], [BG5658: 6-Me-2-NHMe-4-Py], [BG5659: 3-CF _3- 2-NHMe-4-Py], [BG 5660: 5-CF ₃ -2-NHMe 4-Py], [BG 566 1: 6-CF ₃ 2-NHMe 4-Py], [BG 566 2: 3-CN- 2-NHMe-4-Py], [BG5663: 5-CN-2-NHMe-4-Py], [BG5664: 6-CN-2-NHMe-4-Py], [BG5665: 3-OMe-2-] NHMe-4-Py], [BG5666: 5-OMe-2-NHMe-4-Py], [BG5667: 6-OMe-2-NHMe-4-Py], [BG5668: 5-NHMe-4-Py] , [BG5669: 3-Cl-5-NHMe-4-Py], [BG 5670: 2-Cl-5-NHMe-4-Py], [BG5671: 6-Cl-5-NHMe-4-Py], BG5672: 3-Me-5-NHMe-4-Py], [BG5673: 2-Me-5-NHMe-4-Py], [BG5674: 6-Me-5-NHMe-4-Py], [BG5675: 3-CF ₃ -5-NHMe-4-Py !, [BG 5676: 2-CF ₃ -5-NHMe-4-Py], [BG 5677: 6-CF ₃ -5-NHMe-4-Py], [BG 5 678: 3-CN] -5-NHMe-4-Py !, [BG5679: 2-CN-5-NHMe-4-Py], [BG5680: 6-CN-5-NHMe-4-Py], [BG5681: 3-OMe-5] -NHMe-4-Py], [BG5682: 2-OMe-5-NHMe-4-Py], [BG5683: 6-OMe-5-NHMe-4-Py], [BG5684: 6-NHMe-4-Py] ], [BG5685: 3-Cl-6-NHMe-4-Py], [BG5686: 2-Cl-6-NHMe-4-Py], [BG5687: 5-Cl-6-NHMe-4-Py], [BG5688: 3-Me-6-NHMe-4-Py], [BG5689: 2-Me-6-NHMe-4-Py], [BG5690: 5-Me-6-NHMe-4-Py], [BG5691] _{: 3-CF 3 -6-NHMe} -4-Py], [BG5692: 2-CF 3 -6-NHMe-4-Py], [BG5693: 5-CF 3 -6-NHMe-4-Py], [ BG5694: 3-CN-6-NHMe-4-Py], [BG5695: 2-CN-6-NHMe-4-Py], [BG5696: 5-CN-6-NHMe-4-Py], [BG5697: 3-OMe-6-NHMe-4-Py], [BG5698: 2-OMe-6-NHMe-4-Py], [BG5699: 5-OMe-6-NHMe-4-Py], [BG5700: 3- NMe ₂ -4-Py],

[BG5701: 2-Cl-3 -NMe 2 -4-Py], [BG5702: 5-Cl-3-NMe 2 -4-Py], [BG5703: 6-Cl-3-NMe 2 -4-Py] , [BG5704: 2-Me- 3-NMe 2 -4-Py], [BG5705: 5-Me-3-NMe 2 -4-Py], [BG5706: 6-Me-3-NMe 2 -4-Py ], [BG5707: 2-CF 3 -3-NMe 2 -4-Py], [BG5708: 5-CF 3 -3-NMe 2 -4-Py], [BG5709: 6-CF 3 -3-NMe 2 -4-Py], [BG5710: 2-CN-3-NMe 2 -4-Py], [BG5711: 5-CN-3-NMe 2 -4-Py], [BG5712: 6-CN-3-NMe _{2 -4-Py], [BG5713} : 2-OMe-3-NMe 2 -4-Py], [BG5714: 5-OMe-3-NMe 2 -4-Py], [BG5715: 6-OMe-3- _{NMe 2 -4-Py], [} BG5716: 4-NMe 2 -4-Py], [BG5717: 3-Cl-4-NMe 2 -4-Py], [BG5718: 5-Cl-4-NMe 2 - 4-Py], [BG5719: 6-Cl-4-NMe 2 -4-Py], [BG5720: 3-Me-4-NMe 2 -4-Py], [BG5721: 5-Me-4-NMe 2 -4-Py], [BG5722: 6-Me-4-NMe 2 -4-Py], [BG5723: 3-CF 3 -4-NMe 2 -4-Py], [BG5724: 5-CF 3 -4 _{-NMe 2 -4-Py], [} BG5725: 6-CF 3 -4-NMe 2 -4-Py], [BG5726: 3-CN-4-NMe 2 -4-Py], [BG5727: 5-CN -4-NMe ₂ -4-Py !, [BG 5728: 6-CN -4-NMe ₂ -4-Py], [BG 5729: 3-OMe -4-NMe ₂ -4-Py], [BG 5730: 5- 5 _{OMe-4-NMe 2 -4-} Py], [BG5731: 6-OMe-4-NMe 2 -4-Py], [BG5732: 5-NMe 2 -4-Py], [BG5733: 3-Cl-5 _{-NMe 2 -4-Py], [} BG5734: 2-Cl-5-NMe 2 -4-Py], [BG5735: 6-Cl-5-NMe 2 -4-Py], [BG573 6: 3-Me-5- NMe 2 -4-Py], [BG5737: 2-Me-5-NMe 2 -4-Py], [BG5738: 6-Me-5-NMe 2 -4-Py], _{[BG5739: 3-CF 3 -5} -NMe 2 -4-Py], [BG5740: 2-CF 3 -5-NMe 2 -4-Py], [BG5741: 6-CF 3 -5-NMe 2 -4 -Py], [BG5742: 3- CN-5-NMe 2 -4-Py], [BG5743: 2-CN-5-NMe 2 -4-Py], [BG5744: 6-CN-5-NMe 2 - 4-Py], [BG5745: 3-OMe-5-NMe 2 -4-Py], [BG5746: 2-OMe-5-NMe 2 -4-Py], [BG5747: 6-OMe-5-NMe 2 -4-Py], [BG5748: 6-NMe 2 -4-Py], [BG5749: 3-Cl-6-NMe 2 -4-Py], [BG5750: 2-Cl-6-NMe 2 -4- Py], [BG5751: 5- Cl-6-NMe 2 -4-Py], [BG5752: 3-Me-6-NMe 2 -4-Py], [BG5753: 2-Me-6-NMe 2 -4 -Py], [BG5754: 5- Me-6-NMe 2 -4-Py], [BG5755: 3-CF 3 -6-NMe 2 -4-Py], [BG5756: 2-CF 3 -6-NMe _{2 -4-Py], [BG5757} : 5-CF 3 -6-NMe 2 -4-Py], [BG5758: 3-CN-6-NMe 2 -4-Py], [BG5759: 2-CN-6 _{-NMe 2 -4-Py], [} BG5760: 5-CN-6-NMe 2 -4-Py], [BG5761: 3-OMe-6-NMe 2 -4-Py], [BG5762: 2-OMe- _{6-NMe 2 -4-Py]} , [BG5763: 5-OMe-6-NMe 2 -4-Py], [BG5764: 3-ACNH-4-Py], [BG5765: 2-Cl-3-ACNH- 4-Py], [BG 5766: 5-Cl-3-ACNH-4-Py], [BG 5767: 6-Cl-3-ACNH-4-Py], [BG5 768: 2-Me-3-ACNH-4-] Py], [BG5769: 5- Me-3-ACNH-4-Py], [BG5770: 6-Me-3-ACNH-4-Py], [BG5771: 2-CF 3 -3-ACNH-4-P y], [BG5772: 5- CF 3 -3-ACNH-4-Py], [BG5773: 6-CF 3 -3-ACNH-4-Py], [BG5774: 2-CN-3-ACNH-4- Py], [BG5775: 5-CN-3-ACNH-4-Py], [BG5776: 6-CN-3-ACNH-4-Py], [BG5777: 2-OMe-3-ACNH-4-Py] , [BG5778: 5-OMe-3-ACNH-4-Py], [BG5779: 6-OMe-3-ACNH-4-Py], [BG5780: 2-ACNH-4-Py], [BG5781: 3- Cl-2-ACNH-4-Py], [BG5782: 5-Cl-2-ACNH-4-Py], [BG5783: 6-Cl-2-ACNH-4-Py], [BG5784: 3-Me- 2-ACNH-4-Py] , [BG5785: 5-Me-2-ACNH-4-Py], [BG5786: 6-Me-2-ACNH-4-Py], [BG5787: 3-CF 3 -2 -ACNH-4-Py], [ BG5788: 5-CF 3 -2-ACNH-4-Py], [BG5789: 6-CF 3 -2-ACNH-4-Py], [BG5790: 3-CN-2 -ACNH-4-Py], [BG5791: 5-CN-2-ACNH-4-Py], [BG5792: 6-CN-2-ACNH-4-Py], [BG5793: 3-OMe-2-ACNH] -4-Py], [BG5794: 5-OMe-2-ACNH-4-Py], [BG5795: 6-OMe-2-ACNH-4-Py], [BG5796: 5-ACNH-4-Py], [BG5797: 3-Cl-5-ACNH-4-Py], [BG5798: 2-Cl-5-ACNH-4-Py], [BG5799: 6-Cl-5-ACNH-4-Py], [BG5800] : 3-Me-5-ACNH-4-Py],

[BG5801: 2-Me-5-ACNH-4-Py], [BG5802: 6-Me-5-ACNH-4-Py], [BG5803: 3-CF ₃ -5-ACNH-4-Py], _{BG5804: 2-CF 3 -5-} ACNH-4-Py], [BG5805: 6-CF 3 -5-ACNH-4-Py], [BG5806: 3-CN-5-ACNH-4-Py], [ BG5807: 2-CN-5-ACNH-4-Py], [BG5808: 6-CN-5-ACNH-4-Py], [BG5809: 3-OMe-5-ACNH-4-Py], [BG5810: 2-OMe-5-ACNH-4-Py], [BG5811: 6-OMe-5-ACNH-4-Py], [BG5812: 6-ACNH-4-Py], [BG5813: 3-Cl-6-] ACNH-4-Py !, [BG5814: 2-Cl-6-ACNH-4-Py], [BG5815: 5-Cl-6-ACNH-4-Py], [BG5816: 3-Me-6-ACNH- 4-Py], [BG5817: 2-Me-6-ACNH-4-Py], [BG5818: 5-Me-6-ACNH-4-Py], [BG5819: 3-CF 3 -6-ACNH-4 -Py], [BG5820: 2- CF 3 -6-ACNH-4-Py], [BG5821: 5-CF 3 -6-ACNH-4-Py], [BG5822: 3-CN-6-ACNH-4 -Py], [BG 5823: 2-CN-6-ACNH-4-Py], [BG 5824: 5-CN-6-ACNH-4-Py], [BG 5825: 3-OMe-6-ACNH-4-Py ], [BG5826: 2-OMe-6-ACNH-4-Py], [BG5827: 5-OMe-6-ACNH-4-Py], [BG5828: 3- (N (Ac) (Me))-4] -Py], [BG5829: 2-Cl-3- (N (Ac) (Me))-4-Py], [BG5830: 5-Cl-3- (N (Ac) (Me))-4-Py ], [BG5831: 6-Cl-3- (N (Ac) (Me))-4-Py], [BG5832: 2-Me-3- (N (Ac) (Me))-4-Py], [BG5833: 5-Me-3- (N (Ac) (Me))-4-Py], [BG5834: 6-Me-3- (N (Ac) (Me))-4-Py], [BG5835 _{: 2-CF 3 -3- (N} (Ac) (Me)) - 4-Py], [BG5836: 5-CF 3 -3 - (N (Ac) (Me )) - 4-Py], [BG5837: 6-CF 3 -3- (N (Ac) (Me)) - 4-Py], [BG5838: 2-CN-3- (N (Ac) (Me))-4-Py], [BG5839: 5-CN-3- (N (Ac) (Me))-4-Py], [BG5840: 6-CN-3- (N) (Ac) (Me))-4-Py], [BG5841: 2-OMe-3- (N (Ac) (Me))-4-Py], [BG5842: 5-OMe-3- (N (Ac) ) (Me))-4-Py], [BG5843: 6-OMe-3- (N (Ac) (Me))-4-Py], [BG5844: 2- (N (Ac) (Me))-] 4-Py], [BG 5845: 3-Cl-2- (N (Ac) (Me))-4-Py], [BG 5846: 5-Cl-2- (N (Ac) (Me))-4-] Py], [BG5 847: 6-Cl-2- (N (Ac) (Me))-4-Py], [BG5848: 3-Me-2- (N (Ac) (Me))-4-Py] , [BG5849: 5-Me-2- (N (Ac) (Me))-4-Py], [BG5850: 6-Me-2- (N (Ac) (Me))-4-Py], [BG _{BG5851: 3-CF 3 -2- (} N (Ac) (Me)) - 4-Py], [BG5852: 5-CF 3 -2- (N (Ac) (Me)) - 4-Py], [ _{BG5853: 6-CF 3 -2- (} N (Ac) (Me)) - 4-Py], [BG5854: 3-CN-2- (N (Ac) (Me)) - 4-Py], [BG5855 : 5-CN-2- (N (Ac) (Me))-4-Py], [BG5856: 6-CN-2- (N (Ac) (Me))-4-Py], [BG5857: 3] -OMe-2- (N (Ac) (Me))-4-Py], [BG5858: 5-OMe-2- (N (Ac) (Me))-4-Py], [BG5859: 6-OMe -2- (N (Ac) (Me))-4-Py], [BG 5860: 5- (N (Ac) (Me))-4-Py], [BG 586 1: 3-Cl-5- (N ( Ac) (Me))-4-Py], [BG5862: 2-Cl-5- (N (Ac) (Me))-4-Py], [BG5863: 6-Cl-5- (N (Ac)) (Me))-4-Py], [BG5864: 3-Me-5- (N (Ac) (Me))-4-Py], [BG5865: 2-Me-5- (N (Ac) (Me) ))-4-Py], [BG 5866: 6-Me-5- ( N (Ac) (Me)) - 4-Py], [BG5867: 3-CF 3 -5- (N (Ac) (Me)) - 4-Py], [BG5868: 2-CF 3 -5- ( N (Ac) (Me)) - 4-Py], [BG5869: 6-CF 3 -5- (N (Ac) (Me)) - 4-Py], [BG5870: 3-CN-5- (N (Ac) (Me))-4-Py], [BG 587: 2 -CN-5- (N (Ac) (Me))-4-Py], [BG 5872: 6-CN-5- (N (Ac) ) (Me))-4-Py], [BG5873: 3-OMe-5- (N (Ac) (Me))-4-Py], [BG5874: 2-OMe-5- (N (Ac) ( Me))-4-Py], [BG5875: 6-OMe-5- (N (Ac) (Me))-4-Py], [BG5876: 6- (N (Ac) (Me))-4-] Py], [BG5877: 3-Cl-6- (N (Ac) (Me))-4-Py], [BG5878: 2-Cl-6- (N (Ac) (Me))-4-Py] [BG5879: 5-Cl-6- (N (Ac) (Me))-4-Py], [BG5880: 3-Me-6- (N (Ac) (Me))-4-Py], [BG5879: BG 581: 2-Me-6- (N (Ac) (Me))-4-Py], [BG5882: 5-Me-6- (N (Ac) (Me))-4-Py], [BG 5883: _{3-CF 3 -6- (N (} Ac) (Me)) - 4-Py], [BG5884: 2-CF 3 -6- (N (Ac) (Me)) - 4-Py], [BG5885: 5-CF ₃ -6- (N (Ac) (Me))-4-Py], [BG5886: 3-CN-6- (N (Ac) (Me))-4-Py], [BG5887: 2 -CN-6- (N (Ac) (Me))-4-Py], [BG5888: 5-CN-6- (N (Ac) (Me))-4-Py], [BG5889: 3-OMe -6- (N (Ac) (Me))-4-Py], [BG5890: 2-OMe-6- (N (Ac) (Me))-4-Py], [BG5891: 5-OMe-6 -(N (Ac) (Me))-4-Py], [BG5892: 3-AC-4-Py], [BG5893: 2-Cl-3-AC-4-Py], [BG5894: 5-Cl] -3-AC-4-Py, [BG5895: 6-Cl-3-AC-4-Py], [BG 5896: 2-Me-3-AC-4-Py], [BG5897: 5-Me-3] -AC-4-Py], [BG5898: 6-Me-3 -AC-4-Py], [BG5899: 2-CF 3 -3-AC-4-Py], [BG5900: 5-CF 3 -3-AC-4-Py],

_{[BG5901: 6-CF 3 -3} -AC-4-Py], [BG5902: 2-CN-3-AC-4-Py], [BG5903: 5-CN-3-AC-4-Py], [ BG5904: 6-CN-3-AC-4-Py !, [BG5905: 2-OMe-3-AC-4-Py], [BG5906: 5-OMe-3-AC-4-Py], [BG5907: 6-OMe-3-AC-4-Py], [BG5908: 2-AC-4-Py], [BG5909: 3-Cl-2-AC-4-Py], [BG5910: 5-Cl-2-] AC-4-Py !, [BG5911: 6-Cl-2-AC-4-Py], [BG5912: 3-Me-2-AC-4-Py], [BG5913: 5-Me-2-AC-] 4-Py], [BG5914: 6-Me-2-AC-4-Py], [BG5915: 3-CF 3 -2-AC-4-Py], [BG5916: 5-CF 3 -2-AC- 4-Py], [BG5917: 6-CF 3 -2-AC-4-Py], [BG5918: 3-CN-2-AC-4-Py], [BG5919: 5-CN-2-AC-4 -Py], [BG5920: 6-CN-2-AC-4-Py], [BG5921: 3-OMe-2-AC-4-Py], [BG5922: 5-OMe-2-AC-4-Py] ], [BG5923: 6-OMe-2-AC-4-Py], [BG5924: 5-AC-4-Py], [BG5925: 3-Cl-5-AC-4-Py], [BG5926: 2] -Cl-5-AC-4-Py], [BG5927: 6-Cl-5-AC-4-Py], [BG5928: 3-Me-5-AC-4-Py], [BG5929: 2-Me -5-AC-4-Py] , [BG5930: 6-Me-5-AC-4-Py], [BG5931: 3-CF 3 -5-AC-4-Py], [BG5932: 2-CF 3 -5-AC-4-Py, [BG 5933: 6-CF ₃ -5-AC-4-Py], [BG 5934: 3-CN-5-AC-4-Py], [BG 59 35: 2-CN- 5-AC-4-Py, [BG5936: 6-CN-5-AC-4-Py], [BG5937: 3-OMe-5-AC-4-Py], [BG5938: 2-OMe-5-] AC-4-Py], [BG5939: 6-OMe-5-AC-4-Py], [BG5940: 6-AC-4-Py], [BG5941: 3-Cl-6-AC-4-Py] , [ BG5942: 2-Cl-6-AC-4-Py], [BG5943: 5-Cl-6-AC-4-Py], [BG5944: 3-Me-6-AC-4-Py], [BG5945: 2-Me-6-AC- 4-Py], [BG5946: 5-Me-6-AC-4-Py], [BG5947: 3-CF 3 -6-AC-4-Py], [BG5948: 2 _{-CF 3 -6-AC-4-} Py], [BG5949: 5-CF 3 -6-AC-4-Py], [BG5950: 3-CN-6-AC-4-Py], [BG5951: 2 -CN-6-AC-4-Py], [BG5952: 5-CN-6-AC-4-Py], [BG5953: 3-OMe-6-AC-4-Py], [BG5954: 2-OMe] -6-AC-4-Py !, [BG5 955: 5-OMe-6-AC-4-Py], [BG5956: 1,2- (methylenedioxy) phenyl-4-yl], [BG5957: 2, 3-dihydrobenzofuran-5-yl], [BG5958: 2,3-dihydrobenzofuran-6-yl], [BG5959: 1,3-dihydroisobenzofuran-5-yl], [BG 5960: benzofuran-5-yl] , [BG5961: benzofuran-6-yl], [BG5962: 2,3-dihydrobenzothiophen-5-yl], [BG5963: 2,3-dihydrobenzothiophen-6-yl], [BG5964: 1,3-] Dihydroisobenzothiophen-5-yl], [BG5965: benzothiophen-5-yl], [BG5966: benzothiophen-6-yl], [BG5967: benzodioxane-4-yl], [BG5968: chroman-6- ], [BG5969: Roman-7-yl], [BG5970: isochroman-6-yl], [BG5971: isochroman-7-yl], [BG5972: phenyl], [BG5973: 2-fluorophenyl], [BG5974: 3-fluorophenyl] [BG5975: 4-fluorophenyl], [BG5976: 2,4-difluorophenyl], [BG5977: 2,4,6-trifluorophenyl], [BG5978: 2,3,4,5,6-pentafluoro] Phenyl], [BG5979: 2,3-difluorophenyl], [BG5 980: 2-chlorophenyl], [BG5981: 3-chlorophenyl], [BG5982: 4-chlorophenyl], [BG5983: 2,3-dichlorophenyl], [BG5984 2,4-dichlorophenyl], [BG5985: 2,5-dichlorophenyl], [BG5986: 2,6-dichlorophenyl], [BG5987: 3,4-dichlorophenyl], [BG5988: 3,5-dichlorophenyl], [BG5989 : 2,3,4-Trichlorophenyl], [BG5990: 2,3,5-Trichlorophenyl], [BG5991: 2,3,6-Trichlorophenyl], [BG5992: 2,4,5-Trichlorophenyl], [BG5993: 2,4,6-trichlorophenyl], [BG5994: 3,4,5-trichlorophenyl], [BG5995: 2 , 3,4,6-Tetrachlorophenyl], [BG5996: 2,3,5,6-Tetrachlorophenyl], [BG5997: 2,3,4,5,6-pentachlorophenyl], [BG5998: 2-bromophenyl ], [BG5999: 3-bromophenyl], [BG6000: 4-bromophenyl],

[BG6001: 2,4-dibromophenyl], [BG6002: 2,5-dibromophenyl], [BG6003: 2, 6-dibromophenyl], [BG6004: 2, 4, 6-tribromophenyl], [BG6005: 2,3,4,5,6-pentabromophenyl], [BG6006: 2-iodophenyl], [BG6007: 3-iodophenyl], [BG6008: 4-iodophenyl], [BG6009: 2, 4-di] Iodophenyl], [BG6010: 2-chloro-3-fluorophenyl], [BG6011: 2-chloro-4-fluorophenyl], [BG6012: 2-chloro-5-fluorophenyl], [BG6013: 2-chloro- 6-fluorophenyl], [BG6014: 2-chloro-3-bromophenyl], [BG6015: 2-chloro-4-bromophenyl], [BG6016: 2-chloro-5-bromophenyl], [BG6017: 2- Chloro-6-bromophenyl], [BG6018: 2-bromo-3-chlorophenyl], [BG6019: 2-bromo-4-chlorophenyl], [BG6020: 2-bromo-5-chlorophenyl], [BG6021: 2-bromo -3-Fluorophenyl], [BG6022: 2-bromo-4-fluorophenyl], [BG6023: 2-bromo-5-fluorophenyl], [BG60 24: 2-bromo-6-fluorophenyl], [BG6025: 2-fluoro-3-chlorophenyl], [BG6026: 2-fluoro-4-chlorophenyl], [BG6027: 2-fluoro-5-chlorophenyl], [BG6028 : [2-fluoro-4-bromophenyl], [BG6029: 3-chloro-4-fluorophenyl], [BG6030: 3-chloro-5-fluorophenyl], [BG6031: 3-chloro-4-bromophenyl], [BG6032: 3-chloro-5-bromophenyl], [BG6033: 3-fluoro-4-chlorophenyl], [BG6034: 3-fluoro-4-bromophenyl], [BG6035: 3-bromo-4-chlorophenyl], [BG 6036: 3-bromo-4-fluorophenyl], [BG 6037: 2, 6-dichloro-4-bromophenyl], [BG 6038: 2,3-difluoro-4-chlorophenyl], [BG 60 39: 2, 6-difluoro -4-Chlorophenyl], [BG6040: 2,5-difluoro-4-chlorophenyl], [BG6041: 3,5-difluoro-4-chlorophenyl], [BG6042: 2,3,5-trifluoro-4-chlorophenyl] , [BG6043: 2,3,6-trifluoro-4-chlorophenyl], [BG6044: 2,3, 5,6-Tetrafluoro-4-chlorophenyl], [BG 6045: 2-fluoro-4-bromophenyl], [BG 6046: 2,3-difluoro-4-bromophenyl], [BG 6047: 2, 6-difluoro-4] -Bromophenyl], [BG6048: 2,5-difluoro-4-bromophenyl], [BG6049: 3,5-difluoro-4-bromophenyl], [BG6050: 2,3,5-trifluoro-4-bromo Phenyl], [BG6051: 2,3,6-trifluoro-4-bromophenyl], [BG6052: 2,3,5,6-tetrafluoro-4-bromophenyl], [BG6053: 2-fluoro-4- Iodophenyl], [BG6054: 3-fluoro-4-iodophenyl], [BG6055: 2,3-difluoro-4-iodophenyl], [BG6056: 2, 6-difluoro-4-iodophenyl], [BG6057: 2,5-Difluoro-4-iodophenyl], [BG 6058: 3,5-Difluoro-4-iodophenyl], [BG 6059: 2, 3, 5-trifluoro-4-iodophenyl], [BG 6060: 2, 3,6-Trifluoro-4-iodophenyl], [BG6061: 2,3,5,6-tetrafluoro-4-iodophenyl], [BG6062: 2-methylflo] Nyl], [BG6063: 3-methylphenyl], [BG6064: 4-methylphenyl], [BG6065: 2,3-dimethylphenyl], [BG6066: 2,4-dimethylphenyl], [BG6067: 2, 5- Dimethylphenyl], [BG 6068: 2, 6-dimethylphenyl], [BG 6069: 3,4-dimethylphenyl], [BG 6070: 3,5-dimethylphenyl], [BG 607 1: 2, 3,5-trimethylphenyl], [BG6072: 2, 3, 4-trimethylphenyl], [BG6073: 2, 3, 6-trimethylphenyl], [BG607 4: 2, 4, 5-trimethylphenyl], [BG 6075: 2, 4, 6-trimethylphenyl] ], [BG6076: 3,4,5-trimethylphenyl], [BG6077: 2,3,4,6- tetramethylphenyl], [BG6078: 2,3,5,6-tetramethylphenyl], [BG6079: 2,3,4,5,6-pentamethylphenyl], [BG6080: 2-ethylphenyl], [BG6081: 3-ethylphenyl], [BG6082: 4-ethylphenyl], [BG6083: 2,4-diethyl] Phenyl], [BG6084: 2, 6-diethylphenyl], [BG 6085: 3,5-diethylphenyl], [BG 60 8: 2, 4, 6-triethylphenyl], [BG 6087: 2-n-propylpheny] ], [BG 6088: 3-n-propylphenyl], [BG 6089: 4-n-propylphenyl], [BG 6090: 2-isopropylphenyl], [BG6091: 3-isopropylphenyl], [BG6092: 4-isopropylphenyl] , [BG6093: 2,4-diisopropylphenyl], [BG6094: 2, 6-diisopropylphenyl], [BG 6095: 3,5-diisopropylphenyl], [BG 6096: 2-s-butylphenyl], [BG 6097: 3- s-Butylphenyl], [BG6098: 4-s-butylphenyl], [BG6099: 2-t-butylphenyl], [BG6100: 3-t-butylphenyl],

[BG 6101: 4-t-butylphenyl], [BG 6102: 4-n-butylphenyl], [BG 6103: 4-n-nonylphenyl], [BG 6104: 2-methyl-4-t-butylphenyl], [BG 6 105 : 2-Methyl-6-t-butylphenyl], [BG6106: 2-methyl-4-isopropylphenyl], [BG6107: 2-methyl-5-isopropylphenyl], [BG6108: 3-methyl-4-isopropylphenyl] ], [BG 6109: 2-cyclohexylphenyl], [BG 6110: 3-cyclohexylphenyl], [BG 6111: 4-cyclohexylphenyl], [BG 6112: 4-cyclopropylphenyl], [BG 6113: 4-cyclobutylphenyl], [BG 6113: BG6114: 4-cyclopentylphenyl], [BG6115: 2-chloro-4-phenylphenyl], [BG6116: 2-bromo-4-phenylphenyl], [BG6117: 4-hydroxyphenyl], [BG6118: 2-methoxyphenyl] ], [BG6119: 3-methoxyphenyl], [BG6120: 4-methoxyphenyl], [BG6121: 2-ethoxyphenyl], [BG6122: 3-ethoxyphenyl], [BG6123: 4-ethoxyphenyl], [BG6124: 2-n-propyloxyphenyl], [BG 6125: 3-n-propyloxyphenyl], [BG 6126: 4-n-propyloxyphenyl], [BG 6127: 2-isopropyloxyphenyl], [BG 6128: 3-isopropyloxy Phenyl], [BG 6129: 4-isopropyloxyphenyl], [BG 6130: 2-n-hexyloxyphenyl], [BG 6131: 3-n-hexyloxyphenyl], [BG 6132: 4-n-hexyloxyphenyl], [BG BG6133: 2-benzyloxyphenyl], [BG 6134: 3-benzyloxyphenyl], [BG 6135: 4-benzyloxyphenyl], [BG 6136: 2,3-dimethoxyphenyl], [BG 6137: 2,4-dimethoxyphenyl] , [BG6138: 2,5-dimethoxyphenyl], [BG6139: 2,6-dimethoxyphenyl], [BG6140: 3,4-dimethoxyphenyl], [BG6141: 3,5-dimethoxyphenyl], [BG6142: 2- t-Butoxyphenyl], [BG6143: 3-t-butoxyphenyl], [BG6144: 4-t-butoxyphenyl], [BG6145: 3- (3-chlorophenyl) phenyl], [BG6146 : 4- (4-chlorophenyl) phenyl], [BG6147: 2-phenoxyphenyl], [BG6148: 3-phenoxyphenyl], [BG6149: 4-phenoxyphenyl], [BG6150: 2- (2-fluorophenoxy) phenyl] ], [BG6151: 3- (3-chlorophenoxy) phenyl], [BG6152: 4- (4-chlorophenoxy) phenyl], [BG6153: 2,3,6-trimethyl-4-fluorophenyl], [BG6154: 2,3,6-trimethyl-4-chlorophenyl], [BG6155: 2,3,6-trimethyl-4-bromophenyl], [BG6156: 2,4-dimethyl-6-fluorophenyl], [BG6157: 2, 4-dimethyl-6-chlorophenyl], [BG 6158: 2,4-dimethyl-6-bromophenyl], [BG 6159: 2-isopropyl-4-chloro-5-methylphenyl], [BG 6160: 2-chloro-4- Nitrophenyl], [BG6161: 2-nitro-4-chlorophenyl], [BG6162: 2-methoxy-5-nitrophenyl], [BG6163: 2,4-dichloro-5-nitrophenyl], [BG6164: 2,4 -Dichloro-6-nitrophenyl], [BG 6165: 2, 6-dichloro-4-nitrof [BG 6166: 2,6-dibromo-4-nitrophenyl], [BG 6167: 2, 6-diiodo-4-nitrophenyl], [BG 6168: 2-methyl-5-isopropyl-4-chlorophenyl], [BG BG 6169: 2-methoxycarbonylphenyl], [BG 6170: 3-methoxycarbonylphenyl], [BG6171: 4-methoxycarbonylphenyl], [BG6172: 4-acetoxyphenyl], [BG6173: 2-methoxymethylphenyl], [BG6174 : 3-methoxymethylphenyl], [BG 6175: 4-methoxymethylphenyl], [BG 6176: 2-phenylphenyl], [BG 6177: 3-phenylphenyl], [BG 6178: 4-phenylphenyl], [BG 6179: 2- (2-fluorophenyl) phenyl], [BG6180: 2-methyl-5-bromophenyl], [BG6181: 2-methyl-6-bromophenyl], [BG6182: 2-chloro-3-methylphenyl], [BG6183 : 2-chloro-4-methylphenyl], [BG6184: 2-chloro-5-methylphenyl], [BG6185: 2-fluoro-3-methylphenyl], [BG 6186: 2-fluoro-4-methylphenyl], [BG 6187: 2-f Luoro-5-methylphenyl], [BG 6188: 2-bromo-3-methylphenyl], [BG 6189: 2-bromo-4-methylphenyl], [BG 6190: 2-bromo-5-methylphenyl], [BG6191: 3-Methyl-4-chlorophenyl], [BG6192: 3-methyl-5-chlorophenyl], [BG6193: 3-methyl-4-fluorophenyl], [BG6194: 3-methyl-5-fluorophenyl], [BG6195: 3-Methyl-4-bromophenyl], [BG 6196: 3-methyl-5-bromophenyl], [BG 6197: 3-fluoro-4-methylphenyl], [BG 6198: 3-chloro-4-methylphenyl], [BG BG 6199: 3-bromo-4-methylphenyl], [BG 6200: 2-chloro-4, 5-dimethylphenyl],

[BG6201: 2-bromo-4,5-dimethylphenyl], [BG6202: 2-chloro-3,5-dimethylphenyl], [BG6203: 2-bromo-3,5-dimethylphenyl], [BG6204: 2, 6-dibromo-4-methylphenyl], [BG 6205: 2,4-dichloro-6-methylphenyl], [BG 6206: 2,4-difluoro-6-methylphenyl], [BG 6207: 2,4-dibromo-6. -Methylphenyl], [BG 6208: 2, 6-Dimethyl-4-fluorophenyl], [BG 6209: 2, 6-Dimethyl-4-chlorophenyl], [BG 6210: 2, 6-Dimethyl-4-bromophenyl], [BG BG6211: 3,5-dimethyl-4-fluorophenyl], [BG6212: 3,5-dimethyl-4-chlorophenyl], [BG6213: 3,5-dimethyl-4-bromophenyl], [BG6214: 2, 3- Difluoro-4-methylphenyl], [BG6215: 2,5-difluoro-4-methylphenyl], [BG6216: 3,5-difluoro-4-methylphenyl], [BG6217: 2,3,5-trifluoro- 4-Methylphenyl], [BG6218: 2,3,6-trifluoro-4-methylphenyl], [BG6219: 2,3,5,6-tetrafluoro-4-methylphenyl], [BG 6220: 2-fluoro-4-ethylphenyl], [BG6221: 3-fluoro-4-ethylphenyl], [BG6222: 2,3-difluoro-4-ethylphenyl], [BG6223: 2, 6-difluoro-4] -Ethylphenyl], [BG 6224: 2, 5-difluoro-4-ethylphenyl], [BG 6 225: 3,5-difluoro-4-ethylphenyl], [BG 6226: 2, 3, 5-trifluoro-4-ethyl] Phenyl], [BG6227: 2,3, 6-trifluoro-4-ethylphenyl], [BG6228: 2, 3, 5, 6- tetrafluoro-4-ethylphenyl], [BG 6229: 2- trifluoromethylphenyl ], [BG 6230: 3-trifluoromethylphenyl], [BG6231: 4- trifluoromethylphenyl], [BG6232: 4- (2, 2, 2- trifluoro- 1 -trifluoromethyl-ethyl) phenyl], [BG6233: 2-trifluoromethoxyphenyl], [BG6234: 3-trifluoromethoxyphenyl], [BG6235: 4-trifluoromethoxyphenyl], [BG6236: 4- (2,2-difluoroethoxy) phenyl], [BG6234: BG 6237: 4- (2, 2, 2- trifluoro ethyl ketone B) phenyl], [BG6238: 2-nitrophenyl], [BG 6239: 3-nitrophenyl], [BG 6240: 4-nitrophenyl], [BG6241: 2-cyanophenyl], [BG6242: 3-cyanophenyl], [BG6243: 4-cyanophenyl], [BG6244: 2-methyl-3-chlorophenyl], [BG6245: 2-methyl-4-chlorophenyl], [BG6246: 2-methyl-5-chlorophenyl], [BG6247: 2- Methyl-6-chlorophenyl], [BG6248: 2-methyl-3-fluorophenyl], [BG6249: 2-methyl-4-fluorophenyl], [BG6250: 2-methyl-5-fluorophenyl], [BG6251: 2 -Methyl-6-fluorophenyl], [BG6252: 2-methyl-3-bromophenyl], [BG6253: 2-methyl-4-bromophenyl], [BG6254: 4-methylthiophenyl], [BG6255: 4-methyl] Sulfonylphenyl], [BG6256: 4-methylsulfinylphenyl], [BG6257: 4-trifluoromethylthiophenyl], [BG6258: 4-ethynylphenyl], [BG6259: 4- (1-propynyl) phenyl], [BG6260: 4-vinylphenyl], [BG6261: 4 -(2,2-dichlorovinyl) phenyl], [BG6262: 4- (2, 2-difluorovinyl) phenyl], [BG6263: cyclohexyl], [BG6264: 2-chlorocyclohexyl], [BG6265: 3-chlorocyclohexyl ], [BG 6266: 4-chlorocyclohexyl], [BG 6267: 4, 4-dichlorocyclohexyl], [BG 6268: 2-bromocyclohexyl], [BG 6269: 3-bromocyclohexyl], [BG 6270: 4-bromocyclohexyl], [BG BG6271: 4, 4-dibromocyclohexyl], [BG6272: 2-iodocyclohexyl], [BG6273: 3-iodocyclohexyl], [BG6274: 4-iodocyclohexyl], [BG6275: 2-fluorocyclohexyl], [BG6276: 3 -Fluorocyclohexyl], [BG6277: 4-fluorocyclohexyl], [BG6278: 4, 4-difluorocyclohexyl], [BG6279: 4-methylcyclohexyl], [BG6280: 4-ethylcyclohexyl], [BG6281: 1-cyclohexenyl] ], [BG6282: 2-cyclohexenyl], [BG6283: 3-cyclohexenyl], [BG6284: 2-chloro] Ro-1-cyclohexenyl], [BG6285: 3-chloro-1-cyclohexenyl], [BG6286: 4-chloro-1-cyclohexenyl], [BG6287: 5-chloro-1-cyclohexenyl], [BG6288: 6-chloro-1-cyclohexenyl], [BG 6289: 1-chloro-2-cyclohexenyl], [BG 6290: 2-chloro-2-cyclohexenyl], [BG 6291: 3-chloro-2-cyclohexenyl], [BG BG 6292: 4-chloro-2-cyclohexenyl], [BG 6293: 5-chloro-2-cyclohexenyl], [BG 6294: 6-chloro-2-cyclohexenyl], [BG 6295: 1-chloro-3-cyclohexenyl] [BG 629: 2-chloro-3-cyclohexenyl], [BG 6297: 3-chloro-3-cyclohexenyl], [BG 6298: 4-chloro-3-cyclohexenyl], [BG 6 299: 5-chloro-3-cyclophenyl] Hexenyl], [BG 6300: 6-chloro-3-cyclohexenyl],

[BG6301: 4-bromo-1-cyclohexenyl], [BG6302: 4-bromo-2-cyclohexenyl], [BG6303: 4-bromo-3-cyclohexenyl], [BG 6304: 4-methyl-1-cyclohexenyl] ], [BG 6305: 4-methyl-2-cyclohexenyl], [BG 6306: 4-methyl-3-cyclohexenyl], [BG 6307: 4-ethyl-1-cyclohexenyl], [BG 6308: 4-ethyl-2-cyclohexenyl] Cyclohexenyl], [BG6309: 4-ethyl-3-cyclohexenyl], [BG6310: trifluoromethyl], [BG6311: tert-butyl], [BG6312: 3-fluoro-2-methoxyphenyl], [BG6313: 4 -Fluoro-2-methoxyphenyl], [BG6314: 5-fluoro-2-methoxyphenyl], [BG6315: 6-fluoro-2-methoxyphenyl], [BG6316: 3-chloro-2-methoxyphenyl], [BG6317 : 4-chloro-2-methoxyphenyl], [BG6318: 5-chloro-2-methoxyphenyl], [BG6319: 6-chloro-2-methoxyphenyl], [BG6320: 3-bromo-2-methoxyphenyl], [BG6321: 4-bromo-2-methoxyphenyl], [BG6322 : 5-bromo-2-methoxyphenyl], [BG6323: 6-bromo-2-methoxyphenyl], [BG6324: 3-iodo-2-methoxyphenyl], [BG6325: 4-iodo-2-methoxyphenyl], [BG6326: 5-iodo-2-methoxyphenyl], [BG6327: 6-iodo-2-methoxyphenyl], [BG6328: 2,3-dimethoxyphenyl], [BG6329: 2,4-dimethoxyphenyl], [BG6330 2,5-Dimethoxyphenyl], [BG6331: 2,6-Dimethoxyphenyl], [BG6332: 3-Methyl-2-methoxyphenyl], [BG6333: 4-Methyl-2-methoxyphenyl], [BG6334: 5 -Methyl-2-methoxyphenyl], [BG6335: 6-methyl-2-methoxyphenyl], [BG 6336: 3-ethyl-2-methoxyphenyl], [BG 6337: 4-ethyl-2-methoxyphenyl], [BG 6338 : 5-ethyl-2-methoxyphenyl], [BG6339: 6-ethyl-2-methoxyphenyl], [BG6340: 3-trifluoromethoxy-2-methoxyphenyl], [BG6341: 4-trifluoromethoxy-2-] Methoxyphenyl], [BG6342: 5-trifluorome Xyl-2-methoxyphenyl], [BG6343: 6-trifluoromethoxy-2-methoxyphenyl], [BG6344: 3-trifluoromethyl-2-methoxyphenyl], [BG 6345: 4-trifluoromethyl-2-methoxy] Phenyl], [BG 6346: 5-trifluoromethyl-2-methoxyphenyl], [BG 6347: 6-trifluoromethyl-2-methoxyphenyl], [BG 6348: 3-methylthio-2-methoxyphenyl], [BG 6 349: 4 -Methylthio-2-methoxyphenyl], [BG6350: 5-methylthio-2-methoxyphenyl], [BG6351: 6-methylthio-2-methoxyphenyl], [BG6352: 3-trifluoromethylthio-2-methoxyphenyl], [BG6353: 4-trifluoromethylthio-2-methoxyphenyl], [BG6354: 5-trifluoromethylthio-2-methoxyphenyl], [BG6355: 6-trifluoromethylthio-2-methoxyphenyl], [BG6356: 3- Ethynyl-2-methoxyphenyl], [BG 6357: 4-ethynyl-2-methoxyphenyl], [BG 6358: 5-ethynyl-2-] Methoxyphenyl], [BG6359: 6-ethynyl-2-methoxyphenyl], [BG 6360: 3-cyclopropyl-2-methoxyphenyl], [BG6361: 4-cyclopropyl-2-methoxyphenyl], [BG6362: 5- Cyclopropyl-2-methoxyphenyl], [BG6363: 6-cyclopropyl-2-methoxyphenyl], [BG6364: 3-cyclopropyloxy-2-methoxyphenyl], [BG6365: 4-cyclopropyloxy-2-methoxy Phenyl], [BG 6366: 5-Cyclopropyloxy 2-methoxyphenyl], [BG 6367: 6-Cyclopropyloxy 2-methoxyphenyl], [BG 6368: 2-Ethoxy-3-fluorophenyl], [BG 6369: 2 -Ethoxy-4-fluorophenyl], [BG6370: 2-ethoxy-5-fluorophenyl], [BG6371-2-ethoxy-6-fluorophenyl], [BG6372: 3-chloro-2-ethoxyphenyl], [BG6373 : 4-chloro-2-ethoxyphenyl], [BG6374: 5-chloro-2-ethoxyphenyl], [BG6375: 6-chloro-2-ethoxyphenyl], [BG 6376: 3- Lomo-2-ethoxyphenyl], [BG6377: 4-bromo-2-ethoxyphenyl], [BG6378: 5-bromo-2-ethoxyphenyl], [BG6379: 6-bromo-2-ethoxyphenyl], [BG6380: 2-ethoxy-3-iodophenyl], [BG6381: 2-ethoxy-4-iodophenyl], [BG6382: 2-ethoxy-5-iodophenyl], [BG6383: 2-ethoxy-6-iodophenyl], BG6384: 2,3-diethoxyphenyl], [BG6385: 2,4-diethoxyphenyl], [BG6386: 2,5-diethoxyphenyl], [BG6387: 2,6-diethoxyphenyl], [BG6388: 2-Ethoxy-3-methylphenyl], [BG 6389: 2-ethoxy-4-methylphenyl], [BG 6390: 2-ethoxy-5-methylphenyl], [BG 6 39 1: 2-ethoxy-6-methylphenyl], [BG BG6392: 3-ethyl-2-ethoxyphenyl], [BG6393: 4-ethyl-2-ethoxyphenyl], [BG6394: 5-ethyl-2-ethoxyphenyl], [BG6395: 6-ethyl-2-ethoxyphenyl] , [BG 6396: 2-ethoxy-3-trifluoromethoxyphenyl], [BG 6397: 2- Ethoxy-4-trifluoromethoxyphenyl], [BG6398: 2-ethoxy-5-trifluoromethoxyphenyl], [BG 6399: 2-ethoxy-6-trifluoromethoxyphenyl], [BG 6400: 2-ethoxy-3-triful Fluoromethylphenyl],

[BG6401: 2-Ethoxy-4-trifluoromethylphenyl], [BG6402: 2-ethoxy-5-trifluoromethylphenyl], [BG6403: 2-ethoxy-6-trifluoromethylphenyl], [BG6404: 2- Ethoxy-3-methylthiophenyl], [BG6405: 2-ethoxy-4-methylthiophenyl], [BG6406: 2-ethoxy-5-methylthiophenyl], [BG6407: 2-ethoxy-6-methylthiophenyl], [BG6408: 2-Ethoxy-3-trifluoromethylthiophenyl], [BG 6409: 2-ethoxy-4-trifluoromethylthiophenyl], [BG 6410: 2-ethoxy-5-trifluoromethylthiophenyl], [BG 6411: 2-ethoxy-6 -Trifluoromethylthiophenyl], [BG6412: 3-ethynyl-2-ethoxyphenyl], [BG6413: 4-ethynyl-2-ethoxyphenyl], [BG6414: 5-ethynyl-2-ethoxyphenyl], [BG6415: 6 -Ethynyl-2-ethoxyphenyl], [BG6416: 3-cyclopropyl-2-ethoxyphenyl], [BG6417: 4-cyclopropyl-2-] Ethoxyphenyl], [BG6418: 5-cyclopropyl-2-ethoxyphenyl], [BG6419: 6-cyclopropyl-2-ethoxyphenyl], [BG6420: 3-cyclopropyloxy-2-ethoxyphenyl], [BG6421: 4-cyclopropyloxy-2-ethoxyphenyl], [BG6422: 5-cyclopropyloxy-2-ethoxyphenyl], [BG6423: 6-cyclopropyloxy-2-ethoxyphenyl], [BG6424: 3-methoxy-2 -Methylphenyl], [BG 6425: 4-methoxy-2-methylphenyl], [BG 6426: 5-methoxy-2-methylphenyl], [BG 6427: 6-methoxy-2-methylphenyl], [BG 6428: 3-ethoxy] -2-Methylphenyl], [BG6429: 4-ethoxy-2-methylphenyl], [BG6430: 5-ethoxy-2-methylphenyl], [BG6431: 6-ethoxy-2-methylphenyl], [BG6432: 3] -Ethyl-2-methylphenyl], [BG6433: 4-ethyl-2-methylphenyl], [BG6434: 5-ethyl-2-methylphenyl], [BG6435: 6-ethyl-2-methylphenyl], [BG6436 : 3-T Fluoromethoxy-2-methylphenyl], [BG 6437: 4-trifluoromethoxy-2-methylphenyl], [BG 6438: 5-trifluoromethoxy-2-methylphenyl], [BG 6439: 6-trifluoromethoxy-2-] Methylphenyl], [BG 6440: 3-trifluoromethyl-2-methylphenyl], [BG6441: 4-trifluoromethyl-2-methylphenyl], [BG6442: 5-trifluoromethyl-2-methylphenyl], [BG BG6443: 6-trifluoromethyl-2-methylphenyl], [BG6444: 3-methylthio-2-methylphenyl], [BG6445: 4-methylthio-2-methylphenyl], [BG6446: 5-methylthio-2-methyl] Phenyl], [BG 6447: 6-methylthio-2-methylphenyl], [BG 6448: 4-fluoro-2-isopropyloxyphenyl], [BG 6449: 4-chloro-2-isopropyloxyphenyl], [BG 6450: 4-bromo -2-isopropyloxyphenyl], [BG6451: 4-iodo-2-isopropyloxyphenyl], [BG6452: 4-methyl-2-isopropyl] Oxyphenyl], [BG6453: 4-ethyl-2-isopropyloxyphenyl], [BG6454: 4-methoxy-2-isopropyloxyphenyl], [BG6455: 4-ethoxy-2-isopropyloxyphenyl], [BG645: 4 -Trifluoromethyl-2-isopropyloxyphenyl], [BG 6457: 4-trifluoromethoxy-2-isopropyloxyphenyl], [BG 6458: 4-methylthio-2-isopropyloxyphenyl], [BG 6459: 4-cyclopropyl- 2-isopropyloxyphenyl], [BG 6460: 4-fluoro-2-cyclopropyloxyphenyl], [BG6461: 4-chloro-2-cyclopropyloxyphenyl], [BG6462: 4-bromo-2-cyclopropyloxyphenyl] ], [BG6463: 4-iodo-2-cyclopropyloxyphenyl], [BG6464: 4-methyl-2-cyclopropyloxyphenyl], [BG6465: 4-ethyl-2-cyclopropyloxyphenyl], [BG6466: 4-Methoxy-2-cyclopropyloxyphenyl], [BG6 467: 4-ethoxy-2-cyclopropyloxyphenyl], [BG 6468: 4-trifluoromethyl-2-cyclopropyloxyphenyl], [BG 6469: 4-trifluoromethoxy-2-cyclopropyloxyphenyl], [BG 6470 : 4-methylthio-2-cyclopropyloxyphenyl], [BG6471: 4-cyclopropyl-2-cyclopropyloxyphenyl], [BG6472: 3,4-difluoro-2-methoxyphenyl], [BG6473: 4, 5 -Difluoro-2-methoxyphenyl], [BG 4474: 4, 6-difluoro-2-methoxyphenyl], [BG 6475: 3, 4, 5-trifluoro-2-methoxyphenyl], [BG 6476: 3, 4, 5 , 6-Tetrafluoro-2-methoxyphenyl], [BG6477: 4-chloro-3-fluoro-2-methoxyphenyl], [BG6478: 4-chloro-5-fluoro-2-methoxyphenyl], [BG 6479: 4 -Chloro-6-fluoro-2-methoxyphenyl], [BG 6480: 4-bromo-3-fluoro-2-methoxyphenyl], [BG 6481: 4-bromo-5-fluoro-2-methoxyphenyl], [BG 6 482: 4-bromo-6-fluoro-2-methoxyphenyl], [BG6483: 3,4-difluoro-2-ethoxyphenyl], [BG6484: 4, 5-difluoro-2-ethoxyphenyl], [BG 6485: 4 , 6-Difluoro-2-ethoxyphenyl], [BG6486: 3,4,5-trifluoro-2-ethoxyphenyl], [BG6487: 3,4,5,6-tetrafluoro-2-ethoxyphenyl], [ BG 6488: 4-chloro-3-fluoro-2-ethoxyphenyl], [BG 6489: 4-chloro-5-fluoro-2-ethoxyphenyl], [BG6490: 4-chloro-6-fluoro-2-ethoxyphenyl], [BG6491: 4-bromo-3-fluoro-2-ethoxyphenyl], [BG6492: 4-bromo-5-fluoro-2-ethoxyphenyl], [BG6493: 4-bromo-6-fluoro-2-ethoxyphenyl] [BG6494: 3,4-difluoro-2-isopropyloxyphenyl], [BG 6495: 4, 5-difluoro-2-isopropyloxyphenyl], [BG 6496: 4, 6-difluoro-2-isopropyloxyphenyl], [BG BG6497: 3,4,5-trifluoro-2-isopropyl Xyphenyl], [BG 6498: 3, 4, 5, 6-tetrafluoro-2-isopropyloxyphenyl], [BG 6499: 4-chloro-3-fluoro-2-isopropyloxyphenyl], [BG 6500: 4-chloro-5 -Fluoro-2-isopropyloxyphenyl],

[BG6501: 4-chloro-6-fluoro-2-isopropyloxyphenyl], [BG6502: 4-bromo-3-fluoro-2-isopropyloxyphenyl], [BG6503: 4-bromo-5-fluoro-2-isopropyl] Oxyphenyl], [BG6504: 4-bromo-6-fluoro-2-isopropyloxyphenyl], [BG6505: 3,4-difluoro-2-cyclopropyloxyphenyl], [BG650: 4, 5-difluoro-2-] Cyclopropyloxyphenyl], [BG6507: 4, 6-difluoro-2-cyclopropyloxyphenyl], [BG 6508: 3, 4, 5-trifluoro-2-cyclopropyloxyphenyl], [BG 6 509: 3, 4, 6 5,6-tetrafluoro-2-cyclopropyloxyphenyl], [BG6510: 4-chloro-3-fluoro-2-cyclopropyloxyphenyl], [BG6511: 4-chloro-5-fluoro-2-cyclopropyloxy Phenyl], [BG 6512: 4-chloro-6-fluoro-2-cyclopropyloxyphenyl], [BG 6513: 4-bromo-3-fluoro-2-cyclopropyl Xyphenyl], [BG6514: 4-bromo-5-fluoro-2-cyclopropyloxyphenyl], [BG6515: 4-bromo-6-fluoro-2-cyclopropyloxyphenyl], [BG6516: 3-ethynyl-2-] Methylphenyl], [BG6517: 4-ethynyl-2-methylphenyl], [BG6518: 5-ethynyl-2-methylphenyl], [BG6519: 6-ethynyl-2-methylphenyl], [BG6520: 3-cyclopropyl] -2-Methylphenyl], [BG6521: 4-cyclopropyl-2-methylphenyl], [BG6522: 5-cyclopropyl-2-methylphenyl], [BG6523: 6-cyclopropyl-2-methylphenyl], [BG6523: BG6524: 3-cyclopropyloxy-2-methylphenyl], [BG6525: 4-cyclopropyloxy-2-methylphenyl], [BG6526: 5-cyclopropyloxy-2-methylphenyl], [BG6527: 6-cyclo Propyloxy-2-methylphenyl], [BG6528: 3-methoxy-2-fluorophenyl], [BG6529: 4-methoxy-2-fluorophenyl], [BG6530: 5-methoxy-2-ful] Orophenyl], [BG6531: 6-methoxy-2-fluorophenyl], [BG6532: 3-ethoxy-2-fluorophenyl], [BG6533: 4-ethoxy-2-fluorophenyl], [BG6534: 5-ethoxy-2 -Fluorophenyl], [BG6535: 6-ethoxy-2-fluorophenyl], [BG6536: 3-ethyl-2-fluorophenyl], [BG6537: 5-ethyl-2-fluorophenyl], [BG6538: 6-ethyl -2-Fluorophenyl], [BG6539: 2-fluoro-3-trifluoromethoxyphenyl], [BG6540: 2-fluoro-4-trifluoromethoxyphenyl], [BG6541: 2-fluoro-5-trifluoromethoxyphenyl ], [BG 6542: 2-fluoro-6-trifluoromethoxyphenyl], [BG 6543: 2-fluoro-3-trifluoromethylphenyl], [BG 6544: 2-fluoro-4-trifluoromethylphenyl], [BG 6545: 2-Fluoro-5-trifluoromethylphenyl], [BG 6546: 2-fluoro-6-trifluoromethylphenyl], [BG6547: 2-fluoro-3-fluorophenyl Nyl], [BG6548: 2-fluoro-4-fluorophenyl], [BG6549: 2-fluoro-5-fluorophenyl], [BG6550: 2-fluoro-6-fluorophenyl], [BG6551: 3-ethynyl-2 -Fluorophenyl], [BG6552: 4-ethynyl-2-fluorophenyl], [BG6553: 5-ethynyl-2-fluorophenyl], [BG6554: 6-ethynyl-2-fluorophenyl], [BG6555: 3-cyclo Propyl-2-fluorophenyl], [BG6556: 4-cyclopropyl-2-fluorophenyl], [BG6557: 5-cyclopropyl-2-fluorophenyl], [BG6558: 6-cyclopropyl-2-fluorophenyl], [BG6559: 3-cyclopropyloxy-2-fluorophenyl], [BG6560: 4-cyclopropyloxy-2-fluorophenyl], [BG6561: 5-cyclopropyloxy-2-fluorophenyl], [BG6562: 6- Cyclopropyloxy-2-fluorophenyl], [BG6563: 2-ethyl-3-fluorophenyl], [BG6564: 2-ethyl-4-fluorophenyl], [BG6565: 2-ethyl-5 -Fluorophenyl], [BG6566: 2-ethyl-6-fluorophenyl], [BG6567: 3-chloro-2-ethylphenyl], [BG6568: 4-chloro-2-ethylphenyl], [BG6569: 5-chloro -2-ethylphenyl], [BG6570: 6-chloro-2-ethylphenyl], [BG6571: 3-bromo-2-ethylphenyl], [BG6572: 4-bromo-2-ethylphenyl], [BG6573: 5] -Bromo-2-ethylphenyl], [BG6574: 6-bromo-2-ethylphenyl], [BG6575: 2-ethyl-3-iodophenyl], [BG6576: 2-ethyl-4-iodophenyl], [BG6577 : [2-ethyl-5-iodophenyl], [BG6578: 2-ethyl-6-iodophenyl], [BG6579: 2-ethyl-3-ethoxyphenyl], [BG6580: 2-ethyl-4-ethoxyphenyl], [BG6581: 2-ethyl-5-ethoxyphenyl], [BG6582: 2-ethyl-6-ethoxyphenyl], [BG6583: 2-ethyl-3-methylphenyl], [BG6584: 2-ethyl-4-methylphenyl ], [BG6585: 2-ethyl-5-methylphenyl], [BG6586: 2-ethyl-6-methylphenyl], [BG6587: 2, 3- Ethylphenyl], [BG6588: 2,4-diethylphenyl], [BG6589: 2,5-diethylphenyl], [BG6590: 2, 6-diethylphenyl], [BG6591: 2-ethyl-3-trifluoromethoxyphenyl] ], [BG6592: 2-ethyl-4-trifluoromethoxyphenyl], [BG6593: 2-ethyl-5-trifluoromethoxyphenyl], [BG6594: 2-ethyl-6-trifluoromethoxyphenyl], [BG6595: 2-ethyl-3-trifluoromethylphenyl], [BG6596: 2-ethyl-4-trifluoromethylphenyl], [BG6597: 2-ethyl-5-trifluoromethylphenyl], [BG6598: 2-ethyl-6 -Trifluoromethylphenyl], [BG6599: 2-ethyl-3-methylthiophenyl], [BG6600: 2-ethyl-4-methylthiophenyl],

[BG6601: 2-ethyl-5-methylthiophenyl], [BG6602: 2-ethyl-6-methylthiophenyl], [BG6603: 2-ethyl-3-trifluoromethylthiophenyl], [BG6604: 2-ethyl-4- 4 Trifluoromethylthiophenyl], [BG 6605: 2-ethyl-5-trifluoromethylthiophenyl], [BG 6606: 2-ethyl-6-trifluoromethylthiophenyl], [BG 6607: 3-ethynyl-2-ethylphenyl], [ BG6608: 4-ethynyl-2-ethylphenyl], [BG6609: 5-ethynyl-2-ethylphenyl], [BG6610: 6-ethynyl-2-ethylphenyl], [BG6611: 3-cyclopropyl-2-ethylphenyl ], [BG6612: 4-cyclopropyl-2-ethylphenyl], [BG6613: 5-cyclopropyl-2-ethylphenyl], [BG6614: 6-cyclopropyl-2-ethylphenyl], [BG6615: 3-cyclo Propyloxy-2-ethylphenyl], [BG6616: 4-cyclopropyloxy-2-ethylphenyl], [BG6617: 5-cyclopropyloxy-2-ethylphenyl], [BG6 618: 6-Cyclopropyloxy-2-ethylphenyl], [BG 6619: 3-fluoro-2-trifluoromethylphenyl], [BG6620: 4-fluoro-2-trifluoromethylphenyl], [BG 6621: 5-fluoro -2-Trifluoromethylphenyl], [BG6622: 6-fluoro-2-trifluoromethylphenyl], [BG 6623: 3-chloro-2-trifluoromethylphenyl], [BG 6624: 4-chloro-2-trifluoro] Methylphenyl], [BG 6625: 5-chloro-2-trifluoromethylphenyl], [BG 6626: 6-chloro-2-trifluoromethylphenyl], [BG 6627: 3-bromo-2-trifluoromethylphenyl], [BG BG6628: 4-bromo-2-trifluoromethylphenyl], [BG6629: 5-bromo-2-trifluoromethylphenyl], [BG6630: 6-bromo-2-trifluoromethylphenyl], [BG6631: 3-iodo -2-trifluoromethylphenyl], [BG6632: 4-iodo-2-trifluoromethylphenyl], [BG6633: 5-iodo-2-trifluoromeme [Phenylphenyl], [BG6634: 6-iodo-2-trifluoromethylphenyl], [BG6635: 3-ethoxy-2-trifluoromethylphenyl], [BG 6636: 4-ethoxy-2-trifluoromethylphenyl], [BG 6637 : 5-ethoxy-2-trifluoromethylphenyl], [BG 6638: 6-ethoxy-2-trifluoromethylphenyl], [BG 6639: 3-methyl-2-trifluoromethylphenyl], [BG 6640: 4-methyl- 2-trifluoromethylphenyl], [BG6641: 5-methyl-2-trifluoromethylphenyl], [BG6642: 6-methyl-2-trifluoromethylphenyl], [BG6643: 2,3-bistrifluoromethylphenyl] [BG6644: 2,4-bistrifluoromethylphenyl], [BG 6645: 2,5-bistrifluoromethylphenyl], [BG 6646: 2, 6-bistrifluoromethylphenyl], [BG 6647: 2-trifluoromethyl-3] -Trifluoromethoxyphenyl], [BG 6648: 2-trifluoromethyl-4-trifluoromethoxyphenyl ], [BG 6649: 2-trifluoromethyl-5-trifluoromethoxyphenyl], [BG 6650: 2-trifluoromethyl-6-trifluoromethoxyphenyl], [BG6651: 2-ethyl-3-trifluoromethylphenyl] [BG6652: 2-ethyl-4-trifluoromethylphenyl], [BG6653: 2-ethyl-5-trifluoromethylphenyl], [BG6654: 2-ethyl-6-trifluoromethylphenyl], [BG6655: 3 -Methylthio-2-trifluoromethylphenyl], [BG6665: 4-methylthio-2-trifluoromethylphenyl], [BG6657: 5-methylthio-2-trifluoromethylphenyl], [BG6658: 6-methylthio-2-] Trifluoromethylphenyl], [BG6659: 2-trifluoromethyl-3-trifluoromethylthiophenyl], [BG6660: 2-trifluoromethyl-4-trifluoromethylthiophenyl], [BG6661: 2-trifluoromethyl-5] -Trifluoromethylthiophenyl], [BG6662: 2-trifluoromethyl-6- Fluoromethylthiophenyl], [BG6663: 3-ethynyl-2-trifluoromethylphenyl], [BG6664: 4-ethynyl-2-trifluoromethylphenyl], [BG6665: 5-ethynyl-2-trifluoromethylphenyl] [BG6666: 6-ethynyl-2-trifluoromethylphenyl], [BG6667: 3-cyclopropyl-2-trifluoromethylphenyl], [BG6668: 4-cyclopropyl-2-trifluoromethylphenyl], [BG6669 : 5-cyclopropyl-2-trifluoromethylphenyl], [BG 6670: 6-cyclopropyl-2-trifluoromethylphenyl], [BG6671: 3-cyclopropyloxy-2-trifluoromethylphenyl], [BG6672: 4-cyclopropyloxy-2-trifluoromethylphenyl], [BG6673: 5-cyclopropyloxy-2-trifluoromethylphenyl], [BG6674: 6-cyclopropyloxy-2-trifluoromethylphenyl], [BG6675 : 3-methoxynaphthalen-2-yl], [BG 667] 6: 6-chloro-3-methoxynaphthalen-2-yl], [BG 6677: 6-fluoro-3-methoxynaphthalen-2-yl], [BG 6678: 7-chloro-3-methoxynaphthalen-2-yl], [BG 6679: 7-Fluoro-3-methoxynaphthalen-2-yl], [BG 6680: 8-Chloro-3-methoxynaphthalen-2-yl], [BG 6681: 8-Fluoro-3-methoxynaphthalen-2-yl] [BG 6682: 1-chloro-3-methoxynaphthalen-2-yl], [BG6683: 1-fluoro-3-methoxynaphthalen-2-yl], [BG6684: 4-chloro-3-methoxynaphthalen-2-yl ], [BG6685: 4-fluoro-3-methoxynaphthalen-2-yl], [BG6686: 5-chloro-3-methoxynaphthalen-2-yl], [BG6687: 5-fluoro-3-methoxynaphthalene-2-yl] [BG 6688: 2-naphthyl], [BG 6690: adamantan-1-yl], [BG6691: 3-methyladamantan-1-yl], [BG6692: 5-methyladamantane-] 1-yl], [BG6693: 5,7-dimethyladamantan-1-yl], [BG6694: 3,5-dimethyladama] Tan-1-yl], [BG6695: 3,5,7-trimethyladamantan-1-yl], [BG6696: 5-methyladamantan-1-yl], [BG6697: 5,7-dimethyladamantan-1-yl] ], [BG6698: 3,5-dimethyladamantan-1-yl], [BG6699: 3,5,7-trimethyladamantan-1-yl].

  In addition, the present compounds AH1-BH1 to AH3780-BH4501 can also be obtained according to the method described above.

The present compounds AH1-BH1 to AH3780-BH4501 are compounds represented by the following formula (AHBH).
[Wherein, X ^{80 to} X ⁸⁹ each represent a substituent corresponding to each of the substituent numbers (MH1) AH 1 to AH 3780 shown below, and in the formula, E ¹⁰⁸ represents a substituent number (MG 2) BH 1 shown below ~ BH4501. ]
For example, the present compound AH1-BH1 is a compound represented by the formula (AHBH) in which X ^{80 to} X ⁸⁹ have a substituent number MH 1 (X ⁸⁰ has a carbon atom, X ⁸¹ has -CH = CH-, X ⁸² has -C (CH ₃ ) =, X ⁸³ is CH ₂ , X ⁸⁴ and X ⁸⁹ are oxygen atoms, X ^{85 to} X ⁸⁴⁷ and X ⁸⁸ are hydrogen atoms, E ¹⁰⁸ is a substituent number (MH 2) is BH 1 (thiazole) Represents a compound which is a -2-yl group) and is represented by the following formula.

[Substituent number (MH1); X ⁸⁰ , X ⁸¹ , X ⁸² , X ⁸³ , X ⁸⁴ , X ⁸⁵ , X ⁸⁶ , X ⁸⁷ , X ⁸⁸ , X ⁸⁹ ], [AH 1; C, -CH = CH-, = CH-C (Me) = , CH 2, O, H, H, H, H, O], [AH2; C, -CH = CH -, = CH-C (Me) =, CH 2, O, Cl, H, H, H, O], [AH3; C, -CH = CH -, = CH-C (Me) =, CH 2, O, Br, H, H, H, O], [AH4; C, -CH = CH -, = CH-C (Me) =, CH 2, O, CF 3, H, H, H, O], [AH5; C, -CH = CH -, = CH-C ( _{Me) =, CH 2, O} , Me, H, H, H, O], [AH6; C, -CH = CH -, = CH-C (Me) =, CH 2, O, Et, H, H , H, O], [AH7 ; C, -CH = CH -, = CH-C (Me) =, CH 2, O, c-Pr, H, H, H, O], [AH8; C, - CH = CH -, = CH- C (Me) =, CH 2, O, OMe, H, H, H, O], [AH9; C, -CH = CF -, = CH-C (Me) =, _{CH 2, O, H, H} , H, H, O], [AH10; C, -CH = CF -, = CH-C (Me) =, CH 2, O, Cl, H, H, H, O ], [AH11; C, -CH = CF -, = CH-C (Me) =, CH 2, O, Br, H, H, H, O], [AH12; C, -CH = CF -, = CH-C (Me) =, CH 2, O, CF 3, H, H, H, O], [AH13; C, -CH = CF -, = CH-C (Me) =, CH 2, O, Me, H, H, H, O], [AH14; C, -CH = CF -, = CH-C (Me) =, CH 2, O, Et, H, H, H, O], [AH15; C, -CH = CF -, = CH-C (Me) =, CH 2, O, c-Pr, H, H, H, O], [AH16; C, -CH = CF -, = CH-C _{(Me) =, CH 2,} O, OMe, H, H, H, O], [AH17; C, -CF = CH -, = CH-C (Me) =, CH 2, O, H, H, H, H, O], [ AH18; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Cl, H, H, H, O], [AH19; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Br, H, H, H, O], [AH20; C, -CF = CH -, = CH-C (Me ), = CH ₂ , O, CF ₃ , H, H, H, O], [AH 21; C, -CF = CH-, = CH-C (Me) =, CH ₂ , O, Me, H, H , H, O], [AH22 ; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Et, H, H, H, O], [AH23; C, -CF = CH -, = CH-C ( Me) =, CH 2, O, c-Pr, H, H, H, O], [AH24; C, -CF = CH -, = CH-C (Me) =, _{CH 2, O, OMe, H} , H, H, O], [AH25; C, -CF = CH -, = CH-C (Me) =, CH 2, O, H, H, H, H, O ], [AH26; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Cl, H, H, H, O], [AH27; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Br, H, H, H, O], [AH28; C, -CF = CH -, = CH-C (Me) =, CH 2, O, CF _{3, H, H, H,} O], [AH29; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Me, H, H, H, O], [AH30; C, -CF = CH -, = CH-C (Me) =, CH 2, O, Et, H, H, H, O], [AH31; C, -CF = CH -, = CH-C (Me ), = CH ₂ , O, c-Pr, H, H, H, O], [AH 32; C, -CF = CH-, = CH-C (Me) =, CH ₂ , O, OMe, H, H, H, O], [ AH33; C, -CH = CH -, = CF-C (Me) =, CH 2, O, H, H, H, H, O], [AH34; C, -CH = CH -, = CF-C (Me) =, CH 2, O, Cl, H, H, H, O], [AH35; C, -CH = CH -, = CF-C (Me) =, CH _{2, O, Br, H,} H, H, O], [AH36; C, -CH = CH -, = CF-C (Me) =, CH 2, O, CF 3, H, H, H, O ], [AH37; C, -CH = CH -, = CF-C (Me) =, CH 2, O, Me, H, H, H, O], [AH38; C, -CH = CH -, = CF-C (Me) =, CH 2, O, Et, H, H, H, O], [AH39; C, -CH = CH -, = CF-C (Me) =, CH 2, O, c -Pr, H, H, H, O], [AH40; C, -CH = CH -, = CF-C (Me) =, CH 2, O, OMe, H, H, H, O], [AH41 C, -CH = CH-, = CH-C _{Br =, CH 2, O,} H, H, H, H, O], [AH42; C, -CH = CH -, = CH-CBr =, CH 2, O, Cl, H, H, H, O ], [AH43; C, -CH = CH -, = CH-CBr =, CH 2, O, Br, H, H, H, O], [AH44; C, -CH = CH -, = CH-CBr =, CH ₂ , O, CF ₃ , H, H, H, O], [AH 45; C, -CH = CH-, = CH-CBr =, CH ₂ , O, Me, H, H, H, O ], [AH46; C, -CH = CH -, = CH-CBr =, CH 2, O, Et, H, H, H, O], [AH47; C, -CH = CH -, = CH-CBr _{=, CH 2, O, c} -Pr, H, H, H, O], [AH48; C, -CH = CH -, = CH-CBr =, CH 2, O, OMe, H, H, H, O], [AH49; C, -CH = CH -, = CH-CCl =, CH 2, O, H, H, H, H, O], [AH50; C, -CH = CH -, = CH- _{CCl =, CH 2, O,} Cl, H, H, H, O], [AH51; C, -CH = CH -, = CH-CCl =, CH 2, O, Br, H, H, H, O ], [AH52; C, -CH = CH -, = CH-CCl =, CH 2, O, CF 3, H, H, H, O], [AH53; C, -CH = CH -, = CH- _{CCl =, CH 2, O,} Me, H, H, H, O], [AH54; C, -CH = CH -, = CH-CCl =, CH 2, O, Et, H, H, H, O ], [AH55; C, -CH = CH -, = CH-CCl =, CH 2, O, c-Pr, H, H, H, O], [AH56; C, -CH = CH -, = CH _{-CCl =, CH 2, O,} OMe, H, H, H, O], [AH57; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, O, H, H, H, H, O] , [AH58; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, O, Cl, H, H, H, O], [AH59 ; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, O, Br, H, H, H, O], [AH60; C, -C (Me) = CH- , = CH-C (Me) =, CH ₂ , O, CF ₃ , H, H, H, O], [AH 61; C, -C (Me) = CH-, = CH-C (Me) =, _{CH 2, O, Me, H} , H, H, O], [AH62; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, O, E t, H, H, H, O], [AH63; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, O, c-Pr, H, H, H, O ], [AH64; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, O, OMe, H, H, H, O], [AH65; C, -CH = CH -, = CH-C (CF 3) =, CH 2, O, H, H, H, H, O], [AH66; C, -CH = CH -, = CH-C (CF 3) =, CH _{2, O, Cl, H,} H, H, O], [AH67; C, -CH = CH -, = CH-C (CF 3) =, CH 2, O, Br, H, H, H, O ], [AH68; C, -CH = CH -, = CH-C (CF 3) =, CH 2, O, CF 3, H, H, H, O], [AH69; C, -CH = CH- _{, = CH-C (CF 3} ) =, CH 2, O, Me, H, H, H, O], [AH70; C, -CH = CH -, = CH-C (CF 3) =, CH 2 , O, Et, H, H, H, O, [AH 71; C, -CH = CH-, = CH-C (CF ₃ ) =, CH ₂ , O, c-Pr, H, H, H, H O], [AH 72; C, -CH = CH-, = CH-C (CF ₃ ) =, CH ₂ , O, OMe, H, H, H, O], [AH 73; C, -CH = CH- , = CH-C (Et) =, CH ₂ , O, H, H, H, H, O], [AH 74; C,-CH = CH-, = CH-C (Et) =, CH ₂ , O , Cl, H, H, H , O], [AH75; C, -CH = CH -, = CH-C (Et) =, CH 2, O, Br, H, H, H, O], [AH76 ; C, -CH = CH -, = CH-C (Et) =, CH 2, O, CF 3, H, H, H, O], [AH77; C, -CH = CH -, = CH-C _{(Et) =, CH 2,} O, Me, H, H, H, O], [AH78; C, -CH = CH -, = CH-C (Et) =, CH 2, O, Et, H, H, H, O], [ AH79; C, -CH = CH -, = CH-C (Et) =, CH 2, O, c-Pr, H, H, H, O], [AH80; C, -CH = CH -, = CH- C (Et) =, CH 2, O, OMe, H, H, H, O], [AH81; C, -CH = CH -, = CH-C (c-Pr ), = CH ₂ , O, H, H, H, H, O, [AH 82; C, -CH = CH-, = CH-C (c-Pr) =, CH ₂ , O, Cl, H, H, H, O], [AH 83; C, -CH = CH - , = CH-C (c-Pr) =, CH 2, O, Br, H, H, H, O], [AH84; C, -CH = CH -, = CH -C (c-Pr) =, CH 2, O, CF 3, H, H, H, O], [AH85; C, -CH = CH -, = CH-C (c-Pr) =, CH 2 , O, Me, H, H , H, O], [AH86; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, O, Et, H, H, H, O ], [AH 87; C, -CH = CH-, = CH-C (c-Pr) =, CH ₂ , O, c-Pr, H, H, H, O], [AH 88; C, -CH = CH -, = CH-C ( c-Pr) =, CH 2, O, OMe, H, H, H, O], [AH89; N, -CH = CH -, - N =, CH 2, O, H, H, H, H, O], [AH90; N, -CH = CH -, - N =, CH 2, O, F, H, H, H, O], [AH91; N, -CH = CH -, - N =, CH 2, O, Cl, H, H, H, O], [AH92; N, -CH = CH -, - N =, CH 2, O, Br, H, H, H , O], [AH93; N , -CH = CH -, - N =, CH 2, O, Me, H, H, H, O], [AH94; N, -CH = CH -, - N =, _{CH 2, O, Et, H} , H, H, O], [AH95; N, -CH = CH -, - N =, CH 2, O, Pr, H, H, H, O], [AH96; N, -CH = CH -, - N =, CH 2, O, i-Pr, H, H, H, O], [AH97; N, -CH = CH -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH98; N, -CH = CH -, - N =, CH 2, O, c-Bu, H, H, H, O], [AH99; N , -CH = CH -, - N =, CH 2, O, OMe, H, H, H, O], [AH100; N, -CH = CH -, - N =, CH 2, O, Oi-Pr , H, H, H, O],

[AH101; N, -CH = CH -, - N =, CH 2, O, SMe, H, H, H, O], [AH102; N, -CH = CH -, - N =, CH 2, O , Set, H, H, H , O], [AH103; N, -CH = CH -, - N =, CH 2, O, CF 3, H, H, H, O], [AH104; N, - CH = CH -, - N = , CH 2, O, CHF 2, H, H, H, O], [AH105; N, -CH = CH -, - N =, CH 2, O, OCF 3, H , H, H, O], [AH106; N, -CH = CH -, - N =, CH 2, O, OCHF 2, H, H, H, O], [AH107; N, -CH = CH- _{, -N =, CH 2, O} , CH = CH 2, H, H, H, O], [AH108; N, -CH = CH -, - N =, CH 2, O, C (Me) = CH _{2, H, H, H,} O], [AH109; N, -CH = CH -, - N =, CH 2, O, CH = CHMe, H, H, H, O], [AH110; N, - CH = CH -, - N = , CH 2, O, C≡CH, H, H, H, O], [AH111; N, -CH = CH -, - N =, CH 2, O, C≡CMe , H, H, H, O ], [AH112; N, -CH = CH -, - N =, CH 2, O, CN, H, H, H, O], [AH113; N, -CH = CF _{-, - N =, CH 2} , O, H, H, H, H, O], [AH114; N, -CH = CF -, - N =, CH 2, O, Cl, H, H, H, O], [AH115; N, -CH = CF -, - N =, CH 2, O, Br, H, H, H, O], [AH116; N, -CH = CF -, - N =, CH _{2, O, CF 3, H} , H, H, O], [AH117; N, -CH = CF -, - N =, CH 2, O, Me, H, H, H, O], [AH118; N, -CH = CF -, - N =, CH 2, O, Et, H, H, H, O], [AH119; N, -CH = CF -, - N =, CH 2, O, c- Pr, H, H, H, O], [AH120; N, -CH = CF -, - N =, CH 2, O, OMe, H, H, H, O], [AH121; N, -CF = CH -, - N =, CH 2, O, H, H, H, H, O], [AH122; N, -CF = CH -, - N =, CH 2, O, Cl, H, H, H , O], [AH123; N , -CF = CH -, - N =, CH 2, O, Br, H, H, H, O], [AH124 ; N, -CF = CH -, - N =, CH 2, O, CF 3, H, H, H, O], [AH125; N, -CF = CH -, - N =, CH 2, O, Me, H, H, H, O], [AH126; N, -CF = CH -, - N =, CH 2, O, Et, H, H, H, O], [AH127; N, -CF = CH -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH128; N, -CF = CH -, - N =, CH 2, O, OMe, H, H , H, O], [AH129 ; N, -CH = CCl -, - N =, CH 2, O, H, H, H, H, O], [AH130; N, -CH = CCl -, - N =, CH ₂ , O, Cl, H, H, H, O], [AH 131; N, -CH = CCl-, -N =, CH ₂ , O, Br, H, H, H, O], [[ AH132; N, -CH = CCl - , - N =, CH 2, O, CF 3, H, H, H, O], [AH133; N, -CH = CCl -, - N =, CH 2, O , Me, H, H, H , O], [AH134; N, -CH = CCl -, - N =, CH 2, O, Et, H, H, H, O], [AH135; N, -CH = CCl -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH136; N, -CH = CCl -, - N =, CH 2, O, OMe, H, H, H, O], [ AH137; N, -CCl = CH -, - N =, CH 2, O, H, H, H, H, O], [AH138; N, -CCl = CH -, - _{N =, CH 2, O,} Cl, H, H, H, O], [AH139; N, -CCl = CH -, - N =, CH 2, O, Br, H, H, H, O], [AH140; N, -CCl = CH -, - N =, CH 2, O, CF 3, H, H, H, O], [AH141; N, -CCl = CH -, - N =, CH 2, O, Me, H, H, H, O], [AH142; N, -CCl = CH -, - N =, CH 2, O, Et, H, H, H, O], [AH143; N, - CCl = CH -, - N = , CH 2, O, c-Pr, H, H, H, O], [AH144; N, -CCl = CH -, - N =, CH 2, O, OMe, H , H, H, O], [AH145; N, -CH = C (Me) -, - N =, CH 2, O, H, H, H, H, O], [AH146; N, -CH = C (Me) -, - N =, CH 2, O, Cl, H, H, H, O], [AH147; N, -CH = C (Me) -, _{-N =, CH 2, O,} Br, H, H, H, O], [AH148; N, -CH = C (Me) -, - N =, CH 2, O, CF 3, H, H, H, O], [AH149; N, -CH = C (Me) -, - N =, CH 2, O, Me, H, H, H, O], [AH150; N, -CH = C (Me ), -N =, CH ₂ , O, Et, H, H, H, O], [AH 151; N, -CH = C (Me)-, -N =, CH ₂ , O, c-Pr, H, H, H, O] , [AH152; N, -CH = C (Me) -, - N =, CH 2, O, OMe, H, H, H, O], [AH153; N, -C (Me) = CH -, - N =, CH 2, O, H, H, H, H, O], [AH154; N, -C (Me) = CH -, - N =, CH 2, O, Cl, H, H, H, O], [AH155; N, -C (Me) = CH -, - N =, CH 2, O, Br, H, H, H, O], [AH156; N, -C (Me) = CH -, - N =, CH 2, O, CF 3, H, H, H, O], [AH157; N, -C (Me) = CH -, - N =, CH 2 , O, Me, H, H , H, O], [AH158; N, -C (Me) = CH -, - N =, CH 2, O, Et, H, H, H, O], [AH159 ; N, -C (Me) = CH -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH160; N, -C (Me) = CH -, - N _{=, CH 2, O, OMe} , H, H, H, O], [AH161; N, -CH = CH -, - N =, CH 2, O, H, F, H, H, O], [ AH162; N, -CH = CH - , - N =, CH 2, O, Cl, F, H, H, O], [AH163; N, -CH = CH -, - N =, CH 2, O, br, F, H, H, O], [AH164; N, -CH = CH -, - N =, CH 2, O, CF 3, F, H, H, O], [AH165; N, -CH = CH -, - N =, CH 2, O, Me, F, H, H, O], [AH166; N, -CH = CH -, - N =, CH 2, O, Et, F, H, H, O], [AH167; N, -CH = CH -, - N =, CH 2, O, c-Pr, F, H, H, O], [AH168; N, -CH = CH -, - _{N =, CH 2, O,} OMe, F, H, H, O], [AH169; N, -CH = CH -, - N =, CH 2, O, H, H, F , H, O], [AH170 ; N, -CH = CH -, - N =, CH 2, O, Cl, H, F, H, O], [AH171; N, -CH = CH -, - N =, CH ₂ , O, Br, H, F, H, O], [AH 172; N, -CH = CH-, -N =, CH ₂ , O, CF ₃ , H, F, H, O], [AH173; N, -CH = CH -, - N =, CH 2, O, Me, H, F, H, O], [AH174; N, -CH = CH -, - N =, CH 2, O , Et, H, F, H , O], [AH175; N, -CH = CH -, - N =, CH 2, O, c-Pr, H, F, H, O], [AH176; N, -CH = CH -, - N = , CH 2, O, OMe, H, F, H, O], [AH177; N, -CH = CH -, - N =, CH 2, O, H, H, H, F, O], [ AH178; N, -CH = CH -, - N =, CH 2, O, Cl, H, H, F, O], [AH179; N, -CH = CH -, - _{N =, CH 2, O,} Br, H, H, F, O], [AH180; N, -CH = CH -, - N =, CH 2, O, CF 3, H, H, F, O] , [AH181; N, -CH = CH -, - N =, CH 2, O, Me, H, H, F, O], [AH182; N, -CH = CH -, - N =, CH 2, O, Et, H, H, F, O], [AH183; N, -CH = CH -, - N =, CH 2, O, c-Pr, H, H, F, O], [AH184; N , -CH = CH -, - N =, CH 2, O, OMe, H, H, F, O], [AH185; C, = CH-S -, - N =, CH 2, O, H, H , H, H, O], [AH186; C, = CH-S -, - N =, CH 2, O, F, H, H, H, O], [AH187; C, = CH-S-, _{-N =, CH 2, O,} Cl, H, H, H, O], [AH188; C, = CH-S -, - N =, CH 2, O, Br, H, H, H, O] , [AH189; C, = CH -S -, - N =, CH 2, O, Me, H, H, H, O], [AH190; C, = CH-S -, - N =, CH 2, O, Et, H, H, H, O], [AH191; C, = CH-S -, - N =, CH 2, O, Pr, H, H, H, O], [AH192; C, = CH-S -, - N = , CH 2, O, i-Pr, H, H, H, O], [AH193; C, = CH-S -, - N =, CH 2, O, c-Pr , H, H, H, O], [AH194 ; C, = CH-S - , - N =, CH 2, O, c-Bu, H, H, H, O], [AH195; C, = CH-S -, - N =, CH 2, O , OMe, H, H, H , O], [AH196; C, = CH-S -, - N =, CH 2, O, Oi-Pr, H, H, H, O], [AH197; C, = CH-S -, - N =, CH 2, O, SMe, H, H, H, O], [AH198; C, = CH-S -, - N =, CH 2, O, Set, H, H, H, O], [ AH199; C, = CH-S -, - N =, CH 2, O, CF 3, H, H, H, O], [AH200; C, = CH-S-, _{-N =, CH 2, O,} CHF 2 H, H, H, O],

[AH201; C, = CH- S -, - N =, CH 2, O, OCF 3, H, H, H, O], [AH202; C, = CH-S -, - N =, CH 2, _{O, OCHF 2 H, H,} H, O], [AH203; C, = CH-S -, - N =, CH 2, O, CH = CH 2, H, H, H, O], [AH204; C, = CH-S -, - N =, CH 2, O, C (Me) = CH 2, H, H, H, O], [AH205; C, = CH-S -, - N =, CH ₂ , O, CH = CHMe, H, H, H, O], [AH 206; C, = CH-S-, -N =, CH ₂ , O, C≡CH, H, H, H, O], [AH207; C, = CH- S -, - N =, CH 2, O, C≡CMe, H, H, H, O], [AH208; C, = C (CF 3) -S -, - N =, CH ₂ , O, H, H, H, H, H, O], [AH 209; C, = C (CF ₃ ) -S-, -N =, CH ₂ , O, Cl, H, H, H, H O], [AH210; C, = C (CF 3) -S -, - N =, CH 2, O, Br, H, H, H, O], [AH211; C, = C (CF 3) - S -, - N =, CH 2, O, CF 3, H, H, H, O], [AH212; C, = C (CF 3) -S -, - N =, CH 2, O, Me, H, H, H, O] , [AH213; C, = C (CF 3) -S -, - N =, CH 2, O, Et, H, H, H, O], [AH214; C, = _{C (CF 3) -S -,} - N =, CH 2, O, c-Pr, H, H, H, O], [AH215; C, = C (CF 3) -S -, - N =, _{CH 2, O, OMe, H} , H, H, O], [AH216; C, = CF-S -, - N =, CH 2, O, H, H, H, H, O], [AH217; C, = CF-S -, - N =, CH 2, O, Cl, H, H, H, O], [AH218; C, = CF-S -, - N =, CH 2, O, Br, H, H, H, O] , [AH219; C, = CF-S -, - N =, CH 2, O, CF 3, H, H, H, O], [AH220; C, = CF-S _{-, - N =, CH 2} , O, Me, H, H, H, O], [AH221; C, = CF-S -, - N =, CH 2, O, Et, H, H, H, O], [AH222; C, = CF-S -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH223; C, = CF-S -, - N = , CH ₂ , O, OMe, H, H, H, O], [AH224; C, = CCl-S -, - N =, CH 2, O, H, H, H, H, O], [AH225; C, = CCl-S -, - N = , CH 2, O, Cl, H, H, H, O], [AH226; C, = CCl-S -, - N =, CH 2, O, Br, H, H , H, O], [AH227 ; C, = CCl-S -, - N =, CH 2, O, CF 3, H, H, H, O], [AH228; C, = CCl-S -, - _{N =, CH 2, O,} Me, H, H, H, O], [AH229; C, = CCl-S -, - N =, CH 2, O, Et, H, H, H, O], [AH230; C, = CCl- S -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH231; C, = CCl-S -, - N =, CH 2 , O, OMe, H, H, H, O], [AH 232; C, = C (Me)-S-,-N =, CH ₂ , O, H, H, H, H, O], [AH 233 ; C, = C (Me) -S -, - N =, CH 2, O, Cl, H, H, H, O], [AH234; C, = C (Me) -S -, - N =, _{CH 2, O, Br, H} , H, H, O], [AH235; C, = C (Me) -S -, - N =, CH 2, O, CF 3, H, H, H, O] , [AH 236; C, = C (Me)-S-,-N =, CH ₂ , O, Me, H, H, H, O], [AH 237; C, = C (Me)-S-,- _{N =, CH 2, O,} Et, H, H, H, O], [AH238; C, = C (Me) -S -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH239; C, = C (Me) -S -, - N =, CH 2, O, OMe, H, H, H, O], [AH240; C, = CH-S-, _{-N =, CH 2, O,} H, F, H, H, O], [AH241; C, = CH-S -, - N =, CH 2, O, Cl, F, H, H, O] , [AH 242; C, = CH-S-, -N =, CH ₂ , O, Br, F, H, H, O], [AH 243; C, = CH-S-, -N =, CH ₂ , _{O, CF 3, F, H} , H, O], [AH244; C, = CH-S -, - N =, CH 2, O, Me, F, H, H, O], [AH245; C, = CH-S -, - N =, CH 2, O, Et, F, H, H, O], [AH246; C, = CH-S -, - N =, CH 2, O, c-Pr, F, H, H, O], [AH 247; C, = CH-S-, -N = _{, CH 2, O, OMe,} F, H, H, O], [AH248; C, = CH-S -, - N =, CH 2, O, H, H, F, H, O], [AH249 ; C, = CH-S - , - N =, CH 2, O, Cl, H, F, H, O], [AH250; C, = CH-S -, - N =, CH 2, O, Br , H, F, H, O ], [AH251; C, = CH-S -, - N =, CH 2, O, CF 3, H, F, H, O], [AH252; C, = CH- S -, - N =, CH 2, O, Me, H, F, H, O], [AH253; C, = CH-S -, - N =, CH 2, O, Et, H, F, H , O], [AH254; C , = CH-S -, - N =, CH 2, O, c-Pr, H, F, H, O], [AH255; C, = CH-S -, - N =, CH ₂ , O, OMe, H, F, H, O], [AH 256; C, = CH-S-, -N =, CH ₂ , O, H, H, H, F, O], [[ AH257; C, = CH-S -, - N =, CH 2, O, Cl, H, H, F, O], [AH258; C, = CH-S -, - N =, CH 2, O, Br, H, H, F, O], [AH 259; C, = CH-S-,-N =, CH ₂ , O, CF ₃ , H, H, F, O], [AH 260; C, = CH -S -, - N =, CH 2, O, Me, H, H, F, O], [AH261; C, = CH-S -, - N =, CH 2, O, Et, H, H, F, O], [AH262; C, = CH-S -, - N =, CH 2, O, c-Pr, H, H, F, O], [AH263; C, = CH-S -, - _{N =, CH 2, O,} OMe, H, H, F, O], [AH264; C, = CH-O -, - N =, CH 2, O, H, H, H, H, O], [AH265; C, = CH- O -, - N =, CH 2, O, F, H, H, H, O], [AH266; C, = CH-O -, - N =, CH 2, O , Cl, H, H, H, O], [AH 267; C, = CH-O-,-N =, CH ₂ , O, Br, H, H, H, O], [AH 268; C, = CH -O -, - N =, CH 2, O, Me, H, H, H, O], [AH269; C, = CH-O -, - N =, CH 2, O, Et, H, H, H, O], [AH270; C, = CH-O -, - N =, CH 2, O, Pr, H, H, H, O], [AH271; C, = CH-O -, - N = , CH ₂ , O, i-Pr, H, H, H, O], [AH 272; C , = CH-O -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH273; C, = CH-O -, - N =, CH 2, O, c -Bu, H, H, H, O], [AH274; C, = CH-O -, - N =, CH 2, O, OMe, H, H, H, O], [AH275; C, = CH -O -, - N =, CH 2, O, Oi-Pr, H, H, H, O], [AH276; C, = CH-O -, - N =, CH 2, O, SMe, H, H, H, O], [AH 277; C, = CH-O-,-N =, CH ₂ , O, Set, H, H, H, O], [AH 278; C, = CH-O-,- _{N =, CH 2, O,} CF 3, H, H, H, O], [AH279; C, = CH-O -, - N =, CH 2, O, CHF 2 H, H, H, O] , [AH280; C, = CH -O -, - N =, CH 2, O, OCF 3, H, H, H, O], [AH281; C, = CH-O -, - N =, CH 2 _{, O, OCHF 2, H,} H, H, O], [AH282; C, = CH-O -, - N =, CH 2, O, CH = CH 2, H, H, H, O], [ AH283; C, = CH-O -, - N =, CH 2, O, C (Me) = CH 2, H, H, H, O], [AH284; C, = CH-O -, - N = _{, CH 2, O, CH =} CHMe, H, H, H, O], [AH285; C, = CH-O -, - N =, CH 2, O, C≡CH, H, H, H, O ], [AH286; C, = CH-O -, - N =, CH 2, O, C≡CMe, H, H, H, O], [AH287; C, = C (CF 3) -O-, _{-N =, CH 2, O,} H, H, H, H, O], [AH288; C, = C (CF 3) -O -, - N =, CH 2, O, Cl, H, H, H, O], [AH289; C, = C (CF 3) -O -, - N =, CH 2, O, Br, H, H, H, O], [AH290; C, = C (CF 3 ) -O-, -N =, CH ₂ , O, CF ₃ , H, H, H, O], [AH 291; C, = C (CF ₃ ) -O-, -N =, CH ₂ , O, Me, H, H, H, O], [AH292; C, = C (CF 3) -O -, - N =, CH 2, O, Et, H, H, H, O], [AH293; C _{, = C (CF 3) -O} -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH294; C, = C (CF 3) -O -, - N =, CH _{2, O, OMe, H,} H, H, O], [AH295; C, = CF-O -, - N =, CH 2, O, H, H, H, H, O], [AH296; C , = CF-O -, - N =, CH 2, O, Cl, H, H, H, O], [AH297; C, = CF-O -, - N =, CH 2, O, Br, H , H, H, O], [AH 298; C, = CF-O-,-N =, CH ₂ , O, CF ₃ , H, H, H, O], [AH 299; C, = CF-O- _{, -N =, CH 2, O} , Me, H, H, H, O], [AH300; C, = CF-O -, - N =, CH 2, O, Et, H, H, H, O ],

[AH301; C, = CF- O -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH302; C, = CF-O -, - N =, CH 2 , O, OMe, H, H , H, O], [AH303; C, = CCl-O -, - N =, CH 2, O, H, H, H, H, O], [AH304; C, = CCl-O -, - N =, CH 2, O, Cl, H, H, H, O], [AH305; C, = CCl-O -, - N =, CH 2, O, Br, H, H, H, O], [ AH306; C, = CCl-O -, - N =, CH 2, O, CF 3, H, H, H, O], [AH307; C, = CCl-O-, _{-N =, CH 2, O,} Me, H, H, H, O], [AH308; C, = CCl-O -, - N =, CH 2, O, Et, H, H, H, O] , [AH309; C, = CCl -O -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH310; C, = CCl-O -, - N =, CH ₂ , O, OMe, H, H, H, O], [AH 311; C, = C (Me)-O-,-N =, CH ₂ , O, H, H, H, H, O], [[ AH312; C, = C (Me ) -O -, - N =, CH 2, O, Cl, H, H, H, O], [AH313; C, = C (Me) -O -, - N = _{, CH 2, O, Br,} H, H, H, O], [AH314; C, = C (Me) -O -, - N =, CH 2, O, CF 3, H, H, H, O ], [AH315; C, = C (Me) -O -, - N =, CH 2, O, Me, H, H, H, O], [AH316; C, = C (Me) -O-, _{-N =, CH 2, O,} Et, H, H, H, O], [AH317; C, = C (Me) -O -, - N =, CH 2, O, c-Pr, H, H , H, O], [AH318 ; C, = C (Me) -O -, - N =, CH 2, O, OMe, H, H, H, O], [AH319; C, = CH-O- _{, -N =, CH 2, O} , H, F, H, H, O], [AH320; C, = CH-O -, - N =, CH 2, O, Cl, F, H, H, O ], [AH 321; C, = CH-O-, -N =, CH ₂ , O, Br, F, H, H, O], [AH 322; C, = CH-O-, -N =, CH _{2 , O, CF 3, F,} H, H, O], [AH323; C, = CH-O -, - N =, CH 2, O, Me, F, H, H, O], [AH324; C , = CH-O-, -N =, CH ₂ , O, Et, F, H, H, O], [AH 325; C, = CH-O-,-N =, CH ₂ , O, c-Pr, F, H, H, O], [AH 326; C, = CH-O- _{, -N =, CH 2, O} , OMe, F, H, H, O], [AH327; C, = CH-O -, - N =, CH 2, O, H, H, F, H, O ], [AH328; C, = CH-O -, - N =, CH 2, O, Cl, H, F, H, O], [AH329; C, = CH-O -, - N =, CH 2 , O, Br, H, F , H, O], [AH330; C, = CH-O -, - N =, CH 2, O, CF 3, H, F, H, O], [AH331; C , = CH-O -, - N =, CH 2, O, Me, H, F, H, O], [AH332; C, = CH-O -, - N =, CH 2, O, Et, H , F, H, O], [AH333; C, = CH-O -, - N =, CH 2, O, c-Pr, H, F, H, O], [AH334; C, = CH-O _{-, - N =, CH 2} , O, OMe, H, F, H, O], [AH335; C, = CH-O -, - N =, CH 2, O, H, H, H, F, O], [AH336; C, = CH-O -, - N =, CH 2, O, Cl, H, H, F, O], [AH337; C, = CH-O -, - N =, CH _{2, O, Br, H,} H, F, O], [AH338; C, = CH-O -, - N =, CH 2, O, CF 3, H, H, F, O], [AH339; C, = CH-O -, - N =, CH 2, O, Me, H, H, F, O], [AH340; C, = CH-O -, - N =, CH 2, O, Et, H, H, F, O] , [AH341; C, = CH-O -, - N =, CH 2, O, c-Pr, H, H, F, O], [AH342; C, = CH- O -, - N =, CH 2, O, OMe, H, H, F, O], [AH343; C, = CH-O -, - N =, CH 2, O, H, H, H, H , O], [AH344; C , = CH-O -, - N =, CH 2, O, Cl, H, H, H, O], [AH345; C, = CH-O -, - N =, _{CH 2, O, Br, H} , H, H, O], [AH346; C, = CH-O -, - N =, CH 2, O, CF 3, H, H, H, O], [AH347 ; C, = CH-O - , - N =, CH 2, O, Me, H, H, H, O], [AH348; C, = CH-O -, - N =, CH 2, O, Et , H, H, H, O], [AH 349; C, = CH-O-,-N _{=, CH 2, O, c} -Pr, H, H, H, O], [AH350; C, = CH-O -, - N =, CH 2, O, OMe, H, H, H, O] , [AH 351; C, = CH-O-, -CH =, CH ₂ , O, H, H, H, H, O], [AH 352; C, = CH-O-, -CH =, CH ₂ , O, F, H, H, H, O], [AH353; C, = CH-O -, - CH =, CH 2, O, Cl, H, H, H, O], [AH354; C, = CH-O -, - CH = , CH 2, O, Br, H, H, H, O], [AH355; C, = CH-O -, - CH =, CH 2, O, Me, H, H , H, O], [AH356 ; C, = CH-O -, - CH =, CH 2, O, Et, H, H, H, O], [AH357; C, = CH-O -, - CH _{=, CH 2, O, Pr} , H, H, H, O], [AH358; C, = CH-O -, - CH =, CH 2, O, i-Pr, H, H, H, O] , [AH359; C, = CH -O -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH360; C, = CH-O -, - CH =, CH _{2, O, c-Bu,} H, H, H, O], [AH361; C, = CH-O -, - CH =, CH 2, O, OMe, H, H, H, O], [AH362 ; C, = CH-O - , - CH =, CH 2, O, Oi-Pr, H, H, H, O], [AH363; C, = CH-O -, - CH =, CH 2, O , SMe, H, H, H , O], [AH364; C, = CH-O -, - CH =, CH 2, O, Set, H, H, H, O], [AH365; C, = CH -O -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH366; C, = CH-O -, - CH =, CH 2, O, CHF 2, H, H, H, O], [ AH367; C, = CH-O -, - CH =, CH 2, O, OCF 3, H, H, H, O], [AH368; C, = CH-O-, _{-CH =, CH 2, O,} OCHF 2, H, H, H, O], [AH369; C, = CH-O -, - CH =, CH 2, O, CH = CH 2, H, H, H, O], [AH370; C, = CH-O -, - CH =, CH 2, O, C (Me) = CH 2, H, H, H, O], [AH371; C, = CH- O -, - CH =, CH 2, O, CH = CHMe, H, H, H, O], [AH372; C, = CH-O -, - CH =, CH 2, O , C≡CH, H, H, H, O], [AH 373; C, CHCH—O—, —CH =, CH ₂ , O, C≡CMe, H, H, H, O], [AH 374; _{C, = C (CF 3)} -O -, - CH =, CH 2, O, H, H, H, H, O], [AH375; C, = C (CF 3) -O -, - CH = _{, CH 2, O, Cl,} H, H, H, O], [AH376; C, = C (CF 3) -O -, - CH =, CH 2, O, Br, H, H, H, O ], [AH377; C, = C (CF 3) -O -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH378; C, = C (CF 3) - O -, - CH =, CH 2, O, Me, H, H, H, O], [AH379; C, = C (CF 3) -O -, - CH =, CH 2, O, Et, H , H, H, O], [AH380; C, = C (CF 3) -O -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH381; C, _{= C (CF 3) -O -} , - CH =, CH 2, O, OMe, H, H, H, O], [AH382; C, = CF-O -, - CH =, CH 2, O, H, H, H, H, O], [AH383; C, = CF-O -, - CH =, CH 2, O, Cl, H, H, H, O], [AH384; C, = CF- O -, - CH =, CH 2, O, Br, H, H, H, O], [AH385; C, = CF-O -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH386; C, = CF-O -, - CH =, CH 2, O, Me, H, H, H, O], [AH387; C, = CF-O -, - CH = _{, CH 2, O, Et,} H, H, H, O], [AH388; C, = CF-O -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH389; C, = CF- O -, - CH =, CH 2, O, OMe, H, H, H, O], [AH390; C, = CCl-O -, - CH =, CH 2, O , H, H, H, H , O], [AH391; C, = CCl-O -, - CH =, CH 2, O, Cl, H, H, H, O], [AH392; C, = CCl -O -, - CH =, CH 2, O, Br, H, H, H, O], [AH393; C, = CCl-O -, - CH =, CH 2, O, CF 3, H, H , H, O], [AH394 ; C, = CCl-O -, - CH =, CH 2, O, Me, H, H, H, O], [AH395; C, = C Cl-O -, - CH = , CH 2, O, Et, H, H, H, O], [AH396; C, = CCl-O -, - CH =, CH 2, O, c-Pr, H , H, H, O], [AH 397; C, = CCl-O-, -CH =, CH ₂ , O, OMe, H, H, H, O], [AH 398; C, = C (Me)- O -, - CH =, CH 2, O, H, H, H, H, O], [AH399; C, = C (Me) -O -, - CH =, CH 2, O, Cl, H, H, H, O], [AH 400; C, C C (Me) -O-, -CH =, CH ₂ , O, Br, H, H, H, O],

[AH401; C, = C ( Me) -O -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH402; C, = C (Me) -O -, - _{CH =, CH 2, O,} Me, H, H, H, O], [AH403; C, = C (Me) -O -, - CH =, CH 2, O, Et, H, H, H, O], [AH404; C, = C (Me) -O -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH405; C, = C (Me) - O -, - CH =, CH 2, O, OMe, H, H, H, O], [AH406; C, = CH-O -, - CH =, CH 2, O, H, F, H, H , O], [AH407; C , = CH-O -, - CH =, CH 2, O, Cl, F, H, H, O], [AH408; C, = CH-O -, - CH =, _{CH 2, O, Br, F} , H, H, O], [AH409; C, = CH-O -, - CH =, CH 2, O, CF 3, F, H, H, O], [AH410 ; C, = CH-O - , - CH =, CH 2, O, Me, F, H, H, O], [AH411; C, = CH-O -, - CH =, CH 2, O, Et , F, H, H, O ], [AH412; C, = CH-O -, - CH =, CH 2, O, c-Pr, F, H, H, O], [AH413; C, = CH -O -, - CH =, CH 2, O, OMe, F, H, H, O], [AH414; C, = CH-O -, - CH =, CH 2, O, H, H, F, H, O], [AH415; C, = CH-O -, - CH =, CH 2, O, Cl, H, F, H, O], [AH416; C, = CH-O -, - CH = _{, CH 2, O, Br,} H, F, H, O], [AH417; C, = CH-O -, - CH =, CH 2, O, CF 3, H, F, H, O], [ AH418; C, = CH-O -, - CH =, CH 2, O, Me, H, F, H, O], [AH419; C, = CH-O -, - CH =, CH 2, O, Et, H, F, H, O], [AH420; C, = CH-O -, - CH =, CH 2, O, c-Pr, H, F, H, O], [AH421; C, = CH-O -, - CH = , CH 2, O, OMe, H, F, H, O], [AH422; C, = CH-O -, - CH =, CH 2, O, H, H, H , F, O], [AH423 ; C, = CH-O -, - CH =, CH 2, O, Cl, H, H, F, O], [AH424; C, = CH-O -, - CH =, CH ₂ , O, Br, H, H, F, O], [AH425; C, = CH-O -, - CH =, CH 2, O, CF 3, H, H, F, O], [AH426; C, = CH-O -, - CH =, CH 2, O, Me, H, H, F, O], [AH427; C, = CH-O -, - CH =, CH 2, O, Et, H, H, F, O], [ AH428; C, = CH-O -, - CH =, CH 2, O, c-Pr, H, H, F, O], [AH429; C, = CH-O- _{, -CH =, CH 2, O} , OMe, H, H, F, O], [AH430; C, = CH-O -, - CH =, CH 2, O, H, H, H, H, O ], [AH431; C, = CH-O -, - CH =, CH 2, O, Cl, H, H, H, O], [AH432; C, = CH-O -, - CH =, CH 2 , O, Br, H, H , H, O], [AH433; C, = CH-O -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH434; C , = CH-O -, - CH =, CH 2, O, Me, H, H, H, O], [AH435; C, = CH-O -, - CH =, CH 2, O, Et, H , H, H, O], [AH436; C, = CH-O -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH437; C, = CH-O _{-, - CH =, CH 2} , O, OMe, H, H, H, O], [AH438; C, = CH-CH =, - O-, CH 2, O, H, H, H, H, O], [AH439; C, = CH-CH =, - O-, CH 2, O, F, H, H, H, O], [AH440; C, = CH-CH =, - O-, CH ₂ , O, Cl, H, H, H, O, [AH 441; C, = CH-CH =, -O-, CH ₂ , O, Br, H, H, O], [AH 442: C , = CH-CH =, - O-, CH 2, O, Me, H, H, H, O], [AH443; C, = CH-CH =, - O-, CH 2, O, Et, H , H, H, O], [AH444; C, = CH-CH =, - O-, CH 2, O, Pr, H, H, H, O], [AH445; C, = CH-CH =, _{-O-, CH 2, O, i} -Pr, H, H, H, O], [AH446; C, = CH-CH =, - O-, CH 2, O, c-Pr, H, H, H, O], [AH447; C, = CH-CH =, - O-, CH 2, O, c-Bu, H, H, H, O], [AH448; C, = CH-CH =, - O-, CH ₂ , O , OMe, H, H, H , O], [AH449; C, = CH-CH =, - O-, CH 2, O, Oi-Pr, H, H, H, O], [AH450; C, = CH-CH =, - O- , CH 2, O, SMe, H, H, H, O], [AH451; C, = CH-CH =, - O-, CH 2, O, Set, H, H, H, O], [ AH452; C, = CH-CH =, - O-, CH 2, O, CF 3, H, H, H, O], [AH453; C, = CH-CH =, _{-O-, CH 2, O, CHF} 2, H, H, H, O], [AH454; C, = CH-CH =, - O-, CH 2, O, OCF 3, H, H, H, O], [AH455; C, = CH-CH =, - O-, CH 2, O, OCHF 2, H, H, H, O], [AH456; C, = CH-CH =, - O-, _{CH 2, O, CH = CH} 2, H, H, H, O], [AH457; C, = CH-CH =, - O-, CH 2, O, C (Me) = CH 2, H, H , H, O], [AH458 ; C, = CH-CH =, - O-, CH 2, O, CH = CHMe, H, H, H, O], [AH459; C, = CH-CH =, _{-O-, CH 2, O, C≡CH} , H, H, H, O], [AH460; C, = CH-CH =, - O-, CH 2, O, C≡CMe, H, H, H, O], [AH461; C, = C (CF 3) -CH =, - O-, CH 2, O, H, H, H, H, O], [AH462; C, = C (CF 3 ) -CH =, -O-, CH ₂ , O, Cl, H, H, H, O], [AH 463; C, = C (CF ₃ ) -CH =, -O-, CH ₂ , O, Br , H, H, H, O ], [AH464; C, = C (CF 3) -CH =, - O-, CH 2, O, CF 3, H, H, H, O], [AH465; C _{, = C (CF 3) -CH} =, - O-, CH 2, O, Me, H, H, H, O], [AH466; C, = C (CF 3) -CH =, - O-, _{CH 2, O, Et, H} , H, H, O], [AH467; C, = C (CF 3) -CH =, - O-, CH 2, O, c-Pr, H, H, H, O], [AH468; C, = C (CF 3) -CH =, - O-, CH 2, O, OMe, H, H, H, O], [AH469; C, = CF-CH =, - _{O-, CH 2, O, H} , H, H, H, O], [AH470; C, = CF-CH =, - O-, CH _{2, O, Cl, H,} H, H, O], [AH471; C, = CF-CH =, - O-, CH 2, O, Br, H, H, H, O], [AH472; C , = CF-CH =, - O-, CH 2, O, CF 3, H, H, H, O], [AH473; C, = CF-CH =, - O-, CH 2, O, Me, H, H, H, O] , [AH474; C, = CF-CH =, - O-, CH 2, O, Et, H, H, H, O], [AH475; C, = CF-CH = _{, -O-, CH 2, O,} c-Pr, H, H, H, O], [AH476; C, = CF-CH =, - O-, CH 2, O, OMe, H, H, H , O], [AH477; C , = CCl-CH =, - O-, CH 2, O, H, H, H, H, O], [AH478; C, = CCl-CH =, - O-, _{CH 2, O, Cl, H} , H, H, O], [AH479; C, = CCl-CH =, - O-, CH 2, O, Br, H, H, H, O], [AH480; C, = CCl-CH =, - O-, CH 2, O, CF 3, H, H, H, O], [AH481; C, = CCl-CH =, - O-, CH 2, O, Me , H, H, H, O ], [AH482; C, = CCl-CH =, - O-, CH 2, O, Et, H, H, H, O], [AH483; C, = CCl-CH _{=, - O-, CH 2,} O, c-Pr, H, H, H, O], [AH484; C, = CCl-CH =, - O-, CH 2, O, OMe, H, H, H, O], [AH485; C, = C (Me) -CH =, - O-, CH 2, O, H, H, H, H, O], [AH486; C, = C (Me) - _{CH =, - O-, CH 2} , O, Cl, H, H, H, O], [AH487; C, = C (Me) -CH =, - O-, CH 2, O, Br, H, H, H, O], [ AH488; C, = C (Me) -CH =, - O-, CH 2, O, CF 3, H, H, H, O], [AH489; C, = C ( Me) -CH =, - O-, CH 2, O, Me, H, H, H, O], [AH490; C, = C (Me) -CH =, - O-, CH 2, O, Et , H, H, H, O], [AH 491; C, = C (Me) -CH =, -O-, CH ₂ , O, c-Pr, H, H, H, O], [AH 492; C , = = C (Me) -CH , - O-, CH 2, O, OMe, H, H, H, O], [AH493; C, = CH-CH =, - O-, CH 2, O, H, F , H, H, O], [AH 494; C, = CH-CH =, -O-, CH ₂ , O, Cl, F, H, H, O], [AH 495; C, = CH-CH =, _{-O-, CH 2, O, Br} , F, H, H, O], [AH496; C, = CH-CH =, - O-, CH 2, O, CF 3, F, H, H, O ], [AH497; C, = CH-CH =, - O-, CH 2, O, Me, F, H, H, O], [AH498; C, = CH-CH =, - O-, CH 2 , O, Et, F, H , H, O], [AH499; C, = CH-CH =, - O-, CH 2, O, c-Pr, F, H, H, O], [AH500; C, = CH-CH =, - O-, CH 2, O, OMe, F, H, H, O],

[AH501; C, = CH- CH =, - O-, CH 2, O, H, H, F, H, O], [AH502; C, = CH-CH =, - O-, CH 2, O , Cl, H, F, H , O], [AH503; C, = CH-CH =, - O-, CH 2, O, Br, H, F, H, O], [AH504; C, = CH _{-CH =, - O-, CH 2} , O, CF 3, H, F, H, O], [AH505; C, = CH-CH =, - O-, CH 2, O, Me, H, F , H, O], [AH506 ; C, = CH-CH =, - O-, CH 2, O, Et, H, F, H, O], [AH507; C, = CH-CH =, - O _{-, CH 2, O, c} -Pr, H, F, H, O], [AH508; C, = CH-CH =, - O-, CH 2, O, OMe, H, F, H, O] , [AH 509; C, = CH-CH =, -O-, CH ₂ , O ₂ , H, H, H, F, O], [AH 510; C, = CH-CH =, -O-, CH ₂ , O, Cl, H, H, F, O], [AH511; C, = CH-CH =, - O-, CH 2, O, Br, H, H, F, O], [AH512; C, = CH-CH =, - O-, CH 2, O, CF 3, H, H, F, O], [AH513; C, = CH-CH =, - O-, CH 2, O, Me, H, H, F, O], [ AH514; C, = CH-CH =, - O-, CH 2, O, Et, H, H, F, O], [AH515; C, = CH-CH =, - _{O-, CH 2, O, c} -Pr, H, H, F, O], [AH516; C, = CH-CH =, - O-, CH 2, O, OMe, H, H, F, O ], [AH517; C, = CH-CH =, - O-, CH 2, O, H, H, H, H, O], [AH518; C, = CH-CH =, - O-, CH 2 , O, Cl, H, H, H, O, [AH 519; C, = CH-CH =, -O-, CH ₂ , O, Br, H, H, H, O], [AH 520; C, = CH-CH =, - O- , CH 2, O, CF 3, H, H, H, O], [AH521; C, = CH-CH =, - O-, CH 2, O, Me, H , H, H, O], [AH522; C, = CH-CH =, - O-, CH 2, O, Et, H, H, H, O], [AH523; C, = CH-CH =, _{-O-, CH 2, O, c} -Pr, H, H, H, O], [AH524; C, = CH-CH =, - O-, CH 2, O, OMe, H, H, H, O], [ AH525; C, = CH-CH =, - S-, CH 2, O, H, H, H, H, O], [AH526; C, = CH-CH =, - S-, CH 2, O, F, H, H, H, O], [AH527; C, = CH-CH =, - S-, CH 2, O, Cl, H, H, H, O], [AH528; C, = CH- _{CH =, - S-, CH 2} , O, Br, H, H, H, O], [AH529; C, = CH-CH =, - S-, CH 2, O, Me, H, H, H , O], [AH530; C , = CH-CH =, - S-, CH 2, O, Et, H, H, H, O], [AH531; C, = CH-CH =, - S-, _{CH 2, O, Pr, H} , H, H, O], [AH532; C, = CH-CH =, - S-, CH 2, O, i-Pr, H, H, H, O], [ AH533; C, = CH-CH =, - S-, CH 2, O, c-Pr, H, H, H, O], [AH534; C, = CH-CH =, - S-, CH 2, O, c-Bu, H, H, H, O], [AH535; C, = CH-CH =, - S-, CH 2, O, OMe, H, H, H, O], [AH536; C , = CH-CH =, - S-, CH 2, O, Oi-Pr, H, H, H, O], [AH537; C, = CH-CH =, - S-, CH 2, O, SMe , H, H, H, O ], [AH538; C, = CH-CH =, - S-, CH 2, O, Set, H, H, H, O], [AH539; C, = CH-CH _{=, - S-, CH 2,} O, CF 3, H, H, H, O], [AH540; C, = CH-CH =, - S-, CH 2, O, CHF 2, H, H, H, O], [AH541; C, = CH-CH =, - S-, CH 2, O, OCF 3, H, H, H, O], [AH542; C, = CH-CH =, - S _{-, CH 2, O, OCHF} 2, H, H, H, O], [AH543; C, = CH-CH =, - S-, CH 2, O, CH = CH 2, H, H, H, O], [AH544; C, = CH-CH =, - S-, CH 2, O, C (Me) = CH 2, H, H, H, O], [AH545; C, = CH-CH = _{, -S-, CH 2, O,} CH = CHMe, H, H, H, O], [AH546; C, = CH-CH =, - S-, CH 2, O, C≡CH, H, H , H, O], [AH547 ; C, = CH-CH =, - S-, CH 2, O, C≡CMe, H, H, H, O], [AH 548; C, = C (CF 3) -CH =, - S-, CH 2, O, H, H, H, H, O], [AH549; C, = C (CF 3) -CH =, - _{S-, CH 2, O, Cl} , H, H, H, O], [AH550; C, = C (CF 3) -CH =, - S-, CH 2, O, Br, H, H, H , O], [AH551; C , = C (CF 3) -CH =, - S-, CH 2, O, CF 3, H, H, H, O], [AH552; C, = C (CF 3 ) -CH =, - S-, CH 2, O, Me, H, H, H, O], [AH553; C, = C (CF 3) -CH =, - S-, CH 2, O, Et , H, H, H, O ], [AH554; C, = C (CF 3) -CH =, - S-, CH 2, O, c-Pr, H, H, H, O], [AH555; _{C, = C (CF 3)} -CH =, - S-, CH 2, O, OMe, H, H, H, O], [AH556; C, = CF-CH =, - S-, CH 2, O, H, H, H, H, O, [AH 557; C, = CF-CH =, -S-, CH ₂ , O, Cl, H, H, H, O], [AH 558; C, = CF-CH =, - S-, CH 2, O, Br, H, H, H, O], [AH559; C, = CF-CH =, - S-, CH 2, O, CF 3, H, H, H, O], [ AH560; C, = CF-CH =, - S-, CH 2, O, Me, H, H, H, O], [AH561; C, = CF-CH =, - _{S-, CH 2, O, Et} , H, H, H, O], [AH562; C, = CF-CH =, - S-, CH 2, O, c-Pr, H, H, H, O ], [AH563; C, = CF-CH =, - S-, CH 2, O, OMe, H, H, H, O], [AH564; C, = CCl-CH =, - S-, CH 2 , O, H, H, H , H, O], [AH565; C, = CCl-CH =, - S-, CH 2, O, Cl, H, H, H, O], [AH566; C, = CCl-CH =, - S- , CH 2, O, Br, H, H, H, O], [AH567; C, = CCl-CH =, - S-, CH 2, O, CF 3, H , H, H, O], [AH568; C, = CCl-CH =, - S-, CH 2, O, Me, H, H, H, O], [AH569; C, = CCl-CH =, _{-S-, CH 2, O, Et} , H, H, H, O], [AH570; C, = CCl-CH =, - S-, CH 2, O, c-Pr, H, H, H, O] , [AH571; C, = CCl-CH =, - S-, CH 2, O, OMe, H, H, H, O], [AH572; C, = C (Me) _{-CH =, - S-, CH 2} , O, H, H, H, H, O], [AH573; C, = C (Me) -CH =, - S-, CH 2, O, Cl, H , H, H, O], [AH574; C, = C (Me) -CH =, - S-, CH 2, O, Br, H, H, H, O], [AH575; C, = C ( Me) -CH =, - S-, CH 2, O, CF 3, H, H, H, O], [AH576; C, = C (Me) -CH =, - S-, CH 2, O, Me, H, H, H, O], [AH577; C, = C (Me) -CH =, - S-, CH 2, O, Et, H, H, H, O], [AH578; C, = C (Me) -CH =, - S-, CH 2, O, c-Pr, H, H, H, O], [AH579; C, = C (Me) -CH =, - S-, CH _{2, O, OMe, H,} H, H, O], [AH580; C, = CH-CH =, - S-, CH 2, O, H, F, H, H, O], [AH581; C , = CH-CH =, - S-, CH 2, O, Cl, F, H, H, O], [AH582; C, = CH-CH =, - S-, CH 2, O, Br, F , H, H, O], [AH583; C, = CH-CH =, - S-, CH 2, O, CF 3, F, H, H, O], [AH584; C, = CH-CH = _{, -S-, CH 2, O,} Me, F, H, H, O], [AH585; C, = CH-CH =, - S-, CH 2, O, Et, F, H, H, O ], [AH586; C, = CH-CH =, - S-, CH 2, O, c-Pr, F, H, H, O], [AH587; C, = CH-CH =, - S-, _{CH 2, O, OMe, F} , H, H, O], [AH588; C, = CH-CH =, - S-, CH 2, O, H, H, F, H, O], [AH589; C, = CH-CH =, - S-, CH 2, O, Cl, H, F, H, O], [AH590; C, = CH-CH =, - S-, CH 2, O, Br, H, F, H, O] , [AH591; C, = CH-CH =, - S-, CH 2, O, CF 3, H, F, H, O], [AH592; C, = CH-CH _{=, - S-, CH 2,} O, Me, H, F, H, O], [AH593; C, = CH-CH =, - S-, CH 2, O, Et, H, F, H, O], [AH 594; C, = CH-CH =, - S-, CH 2, O, c-Pr, H, F, H, O], [AH595; C, = CH-CH =, - S-, CH 2, O, OMe, H , F, H, O], [AH596; C, = CH-CH =, - S-, CH 2, O, H, H, H, F, O], [AH597; C, = CH-CH =, _{-S-, CH 2, O, Cl} , H, H, F, O], [AH598; C, = CH-CH =, - S-, CH 2, O, Br, H, H, F, O] , [AH599; C, = CH -CH =, - S-, CH 2, O, CF 3, H, H, F, O], [AH600; C, = CH-CH =, - S-, CH 2 , O, Me, H, H, F, O],

[AH601; C, = CH- CH =, - S-, CH 2, O, Et, H, H, F, O], [AH602; C, = CH-CH =, - S-, CH 2, O , c-Pr, H, H , F, O], [AH603; C, = = CH-CH, - S-, CH 2, O, OMe, H, H, F, O], [AH604; C, = CH-CH =, - S- , CH 2, O, H, H, H, H, O], [AH605; C, = CH-CH =, - S-, CH 2, O, Cl, H, H, H, O], [ AH606; C, = CH-CH =, - S-, CH 2, O, Br, H, H, H, O], [AH607; C, = CH-CH =, - _{S-, CH 2, O, CF} 3, H, H, H, O], [AH608; C, = CH-CH =, - S-, CH 2, O, Me, H, H, H, O] , [AH609; C, = CH -CH =, - S-, CH 2, O, Et, H, H, H, O], [AH610; C, = CH-CH =, - S-, CH 2, O, c-Pr, H, H, H, O], [AH611; C, = CH-CH =, - S-, CH 2, O, OMe, H, H, H, O], [AH612; C , = CH-S -, - CH =, CH 2, O, H, H, H, H, O], [AH613; C, = CH-S -, - CH =, CH 2, O, F, H , H, H, O], [AH614; C, = CH-S -, - CH =, CH 2, O, Cl, H, H, H, O], [AH615; C, = CH-S-, _{-CH =, CH 2, O,} Br, H, H, H, O], [AH616; C, = CH-S -, - CH =, CH 2, O, Me, H, H, H, O] , [AH617; C, = CH -S -, - CH =, CH 2, O, Et, H, H, H, O], [AH618; C, = CH-S -, - CH =, CH 2, O, Pr, H, H, H, O], [AH619; C, = CH-S -, - CH =, CH 2, O, i-Pr, H, H, H, O], [AH620; C , = CH-S -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH621; C, = CH-S -, - CH =, CH 2, O, c -Bu, H, H, H, O], [AH 622; C, = CH-S-, -CH =, CH ₂ , O, OMe, H, H, H, O], [AH 623; C, = CH -S -, - CH =, CH 2, O, Oi-Pr, H, H, H, O], [AH624; C, = CH-S -, - CH =, CH 2, O, SMe, H, H, H, O] , [AH625; C, = CH -S -, - CH =, CH 2, O, Set, H, H, H, O], [AH626; C, = CH-S -, - CH =, CH 2, _{O, CF 3, H, H} , H, O], [AH627; C, = CH-S -, - CH =, CH 2, O, CHF 2, H, H, H, O], [AH628; C , = CH-S -, - CH =, CH 2, O, OCF 3, H, H, H, O], [AH629; C, = CH-S -, - CH =, CH 2, O, OCHF 2 , H, H, H, O ], [AH630; C, = CH-S -, - CH =, CH 2, O, CH = CH 2, H, H, H, O], [AH631; C, = CH-S -, - CH = , CH 2, O, C (Me) = CH 2, H, H, H, O], [AH632; C, = CH-S -, - CH =, CH 2, O , CH = CHMe, H, H , H, O], [AH633; C, = CH-S -, - CH =, CH 2, O, C≡CH, H, H, H, O], [AH634; C, = CH-S -, - CH =, CH 2, O, C≡CMe, H, H, H, O], [AH635; C, = C (CF 3) -S -, - CH =, CH _{2, O, H, H,} H, H, O], [AH636; C, = C (CF 3) -S -, - CH =, CH 2, O, Cl, H, H, H, O], [AH637; C, = C ( CF 3) -S -, - CH =, CH 2, O, Br, H, H, H, O], [AH638; C, = C (CF 3) -S-, _{-CH =, CH 2, O,} CF 3, H, H, H, O], [AH639; C, = C (CF 3) -S -, - CH =, CH 2, O, Me, H, H , H, O], [AH640 ; C, = C (CF 3) -S -, - CH =, CH 2, O, Et, H, H, H, O], [AH641; C, = C (CF _{3) -S -, - CH =} , CH 2, O, c-Pr, H, H, H, O], [AH642; C, = C (CF 3) -S -, - CH =, CH 2, O, OMe, H, H, H, O], [AH643; C, = CF-S -, - CH =, CH 2, O, H, H, H, H, O], [AH644; C, = CF-S -, - CH = , CH 2, O, Cl, H, H, H, O], [AH645; C, = CF-S -, - CH =, CH 2, O, Br, H, H , H, O], [AH646 ; C, = CF-S -, - CH =, CH 2, O, CF 3, H, H, H , O], [AH647; C , = CF-S -, - CH =, CH 2, O, Me, H, H, H, O], [AH648; C, = CF-S -, - CH =, _{CH 2, O, Et, H} , H, H, O], [AH649; C, = CF-S -, - CH =, CH 2, O, c-Pr, H, H, H, O], [ AH650; C, = CF-S -, - CH =, CH 2, O, OMe, H, H, H, O], [AH651; C, = CCl-S -, - CH =, CH 2, O, H, H, H, H, O], [AH652; C, = CCl-S -, - CH =, CH 2, O, Cl, H, H, H, O], [AH653; C, = CCl- S -, - CH =, CH 2, O, Br, H, H, H, O], [AH654; C, = CCl-S -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH655; C, = CCl-S -, - CH =, CH 2, O, Me, H, H, H, O], [AH656; C, = CCl-S -, - CH = _{, CH 2, O, Et,} H, H, H, O], [AH657; C, = CCl-S -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH658; C, = CCl- S -, - CH =, CH 2, O, OMe, H, H, H, O], [AH659; C, = C (Me) -S -, - CH =, CH ₂ , O, H, H, H, H, H, O], [AH 660; C, = C (Me)-S-, -CH =, CH ₂ , O, Cl, H, H, H, O], [[ AH661; C, = C (Me ) -S -, - CH =, CH 2, O, Br, H, H, H, O], [AH662; C, = C (Me) -S -, - CH = _{, CH 2, O, CF 3} , H, H, H, O], [AH663; C, = C (Me) -S -, - CH =, CH 2, O, Me, H, H, H, O ], [AH664; C, = C (Me) -S -, - CH =, CH 2, O, Et, H, H, H, O], [AH665; C, = C (Me) -S-, _{-CH =, CH 2, O,} c-Pr, H, H, H, O], [AH666; C, = C (Me) -S -, - CH =, CH 2, O, OMe, H, H , H, O], [AH667 ; C, = CH-S -, - CH =, CH 2, O, H, F, H, H, O], [AH668; C, = CH-S -, - CH =, CH ₂ , O, Cl, F, H, H, O], [AH 669; C, = CH-S-, -CH =, CH ₂ , O, Br, F, H, H, O], [[ AH 670; C, = CH-S -, - CH =, CH 2, O, CF 3, F, H, H, O], [AH671; C, = CH-S -, - CH =, CH 2, O, Me, F , H, H, O], [AH 672; C, = CH-S-, -CH =, CH ₂ , O, Et, F, H, H, O], [AH 673; C, = CH-S-, _{-CH =, CH 2, O,} c-Pr, F, H, H, O], [AH674; C, = CH-S -, - CH =, CH 2, O, OMe, F, H, H, O], [AH675; C, = CH-S -, - CH =, CH 2, O, H, H, F, H, O], [AH676; C, = CH-S -, - CH =, CH _{2, O, Cl, H,} F, H, O], [AH677; C, = CH-S -, - CH =, CH 2, O, Br, H, F, H, O], [AH678; C , = CH-S -, - CH =, CH 2, O, CF 3, H, F, H, O], [AH679; C, = CH-S -, - CH =, CH 2, O, Me, H, F, H, O] , [AH680; C, = CH-S -, - CH =, CH 2, O, Et, H, F, H, O], [AH681; C, = CH-S- _{, -CH =, CH 2, O} , c-Pr, H, F, H, O], [AH682; C, = CH-S -, - CH =, CH 2, O, OMe, H, F, H , O], [AH683; C , = CH-S -, - CH =, CH 2, O, H, H, H, F, O], [AH684; C, = CH-S -, - CH =, _{CH 2, O, Cl, H} , H, F, O], [AH685; C, = CH-S -, - CH =, CH 2, O, Br, H, H, F, O], [AH686; C, = CH-S -, - CH =, CH 2, O, CF 3, H, H, F, O], [AH687; C, = CH-S -, - CH =, CH 2, O, Me , H, H, F, O ], [AH688; C, = CH-S -, - CH =, CH 2, O, Et, H, H, F, O], [AH689; C, = CH-S _{-, - CH =, CH 2} , O, c-Pr, H, H, F, O], [AH690; C, = CH-S -, - CH =, CH 2, O, OMe, H, H, F, O], [AH691; C, = CH-S -, - CH =, CH 2, O, H, H, H, H, O], [AH692; C, = CH-S -, - CH = _{, CH 2, O, Cl,} H, H, H, O], [AH693; C, = CH-S -, - CH =, CH 2, O, Br, H, H, H, O], [AH694 C, = CH-S -, - CH = , CH 2, O, CF 3, H, H, H, O], [AH695; C, = CH-S -, - CH =, CH 2, O, Me, H, H, H, O], [AH 696; C, = CH-S-, -CH =, CH ₂ , O, Et, H, H, H, O], [AH 697; C, = CH-S-,- _{CH =, CH 2, O,} c-Pr, H, H, H, O], [AH698; C, = CH-S -, - CH =, CH 2, O, OMe, H, H, H, O ], [AH699; C, -CH = CH -, = CH-N =, CH 2, O, H, H, H, H, O], [AH700; C, -CH = CH -, = CH-N =, CH ₂ , O, Cl, H, H, H, O],

[AH701; C, -CH = CH -, = CH-N =, CH 2, O, Br, H, H, H, O], [AH702; C, -CH = CH -, = CH-N =, _{CH 2, O, CF 3,} H, H, H, O], [AH703; C, -CH = CH -, = CH-N =, CH 2, O, Me, H, H, H, O], [AH704; C, -CH = CH -, = CH-N =, CH 2, O, Et, H, H, H, O], [AH705; C, -CH = CH -, = CH-N =, _{CH 2, O, c-Pr} , H, H, H, O], [AH706; C, -CH = CH -, = CH-N =, CH 2, O, OMe, H, H, H, O] , [AH707; C, -CH = CF -, = CH-N =, CH 2, O, H, H, H, H, O], [AH708; C, -CH = CF -, = CH-N = _{, CH 2, O, Cl,} H, H, H, O], [AH709; C, -CH = CF -, = CH-N =, CH 2, O, Br, H, H, H, O], [AH710; C, -CH = CF -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [AH711; C, -CH = CF -, = CH-N = _{, CH 2, O, Me,} H, H, H, O], [AH712; C, -CH = CF -, = CH-N =, CH 2, O, Et, H, H, H, O], [AH713; C, -CH = CF -, = CH-N =, CH 2, O, c-Pr, H, H, H, O], [AH714; C, -CH = CF -, = CH-N _{=, CH 2, O, OMe} , H, H, H, O], [AH715; C, -CF = CH -, = CH-N =, CH 2, O, H, H, H, H, O] , [AH716; C, -CF = CH -, = CH-N =, CH 2, O, Cl, H, H, H, O], [AH717; C, -CF = CH -, = CH-N = _{, CH 2, O, Br,} H, H, H, O], [AH718; C, -CF = CH -, = CH-N =, CH 2, O, CF 3, H, H, H, O] , [AH719; C, -CF = CH -, = CH-N =, CH 2, O, Me, H, H, H, O], [AH720; C, -CF = CH -, = CH-N = _{, CH 2, O, Et,} H, H, H, O], [AH721; C, -CF = CH -, = CH-N =, CH 2, O, c-Pr, H, H, H, O ], [AH722; C, -CF = CH -, = CH-N =, CH 2, O, OMe, H, H, H, O], [AH723; C, -CH = CH- , = CF-N =, CH 2, O, H, H, H, H, O], [AH724; C, -CH = CH -, = CF-N =, CH 2, O, Cl, H, H , H, O], [AH725 ; C, -CH = CH -, = CF-N =, CH 2, O, Br, H, H, H, O], [AH726; C, -CH = CH-, _{= CF-N =, CH 2} , O, CF 3, H, H, H, O], [AH727; C, -CH = CH -, = CF-N =, CH 2, O, Me, H, H , H, O], [AH728 ; C, -CH = CH -, = CF-N =, CH 2, O, Et, H, H, H, O], [AH729; C, -CH = CH-, _{= CF-N =, CH 2} , O, c-Pr, H, H, H, O], [AH730; C, -CH = CH -, = CF-N =, CH 2, O, OMe, H, H, H, O], [ AH731; C, -CH = CCl -, = CH-N =, CH 2, O, H, H, H, H, O], [AH732; C, -CH = CCl- , = CH-N =, CH 2, O, Cl, H, H, H, O], [AH733; C, -CH = CCl -, = CH-N =, CH 2, O, Br, H, H , H, O], [AH734 ; C, -CH = CCl -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [AH735; C, -CH = CCl- , = CH-N =, CH 2, O, Me, H, H, H, O], [AH736; C, -CH = CCl -, = CH-N =, CH 2, O, Et, H, H , H, O], [AH737 ; C, -CH = CCl -, = CH-N =, CH 2, O, c-Pr, H, H, H, O], [AH738; C, -CH = CCl -, = CH-N =, CH 2, O, OMe, H, H, H, O], [AH739; C, -CCl = CH -, = CH-N =, CH 2, O, H, H, H, H, O], [ AH740; C, -CCl = CH -, = CH-N =, CH 2, O, Cl, H, H, H, O], [AH741; C, -CCl = CH- , = = CH-N, CH 2, O, Br, H, H, H, O], [AH742; C, -CCl = CH -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [ AH743; C, -CCl = CH -, = = CH-N, CH 2, O, Me, H, H, H, O], [AH744; C, -CCl = CH- , = CH-N =, CH ₂ , O, Et, H, H, H, O], [AH 745; C, -CCl = CH-, = CH- _{N =, CH 2, O,} c-Pr, H, H, H, O], [AH746; C, -CCl = CH -, = CH-N =, CH 2, O, OMe, H, H, H , O], [AH747; C , -CH = CH -, = CCl-N =, CH 2, O, H, H, H, H, O], [AH748; C, -CH = CH -, = CCl _{-N =, CH 2, O,} Cl, H, H, H, O], [AH749; C, -CH = CH -, = CCl-N =, CH 2, O, Br, H, H, H, O], [AH750; C, -CH = CH -, = CCl-N =, CH 2, O, CF 3, H, H, H, O], [AH751; C, -CH = CH -, = CCl _{-N =, CH 2, O,} Me, H, H, H, O], [AH752; C, -CH = CH -, = CCl-N =, CH 2, O, Et, H, H, H, O], [AH753; C, -CH = CH -, = CCl-N =, CH 2, O, c-Pr, H, H, H, O], [AH754; C, -CH = CH -, = _{CCl-N =, CH 2,} O, OMe, H, H, H, O], [AH755; C, -CH = C (Me) -, = CH-N =, CH 2, O, H, H, H, H, O], [ AH756; C, -CH = C (Me) -, = CH-N =, CH 2, O, Cl, H, H, H, O], [AH757; C, -CH = C (Me) -, = CH-N =, CH 2, O, Br, H, H, H, O], [AH758; C, -CH = C (Me) -, = CH-N =, CH _{2, O, CF 3, H} , H, H, O], [AH759; C, -CH = C (Me) -, = CH-N =, CH 2, O, Me, H, H, H, O ], [AH760; C, -CH = C (Me) -, = CH-N =, CH 2, O, Et, H, H, H, O], [AH761; C, -CH = C (Me) -, = CH-N =, CH 2, O, c-Pr, H, H, H, O], [AH762; C, -CH = C (Me) -, = CH-N =, CH 2, O , OMe, H, H, H , O], [AH763; C, -C (Me) = CH -, = CH-N =, CH 2, O, H, H, H, H, O], [AH764 ; C, -C (Me) = CH -, = CH-N =, CH 2, O, Cl, H, H, H, O], [AH765; C, -C (Me) = CH -, = CH _{-N =, CH 2, O,} Br, H, H, H, O], [AH766; C, -C (Me) = CH -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [ AH767; C, -C (Me) = CH -, = CH-N =, CH 2, O, Me, H, H, H, O], [AH768; C, -C (Me) = CH -, = CH-N =, CH 2, O, Et, H, H, H, O], [AH769; C, -C (Me) = CH -, = CH-N =, CH _{2, O, c-Pr,} H, H, H, O], [AH770; C, -C (Me) = CH -, = CH-N =, CH 2, O, OMe, H, H, H, O], [AH771; C, -CH = CH -, = C (Me) -N =, CH 2, O, H, H, H, H, O], [AH772; C, -CH = CH-, = C (Me) -N =, CH 2, O, Cl, H, H, H, O], [AH773; C, -CH = CH -, = C (Me) -N =, CH 2, O, br, H, H, H, O], [AH774; C, -CH = CH -, = C (Me) -N =, CH 2, O, CF 3, H, H, H, O], [AH775 ; C, -CH = CH -, = C (Me) -N =, CH 2, O, Me, H, H, H, O], [AH776; C, -CH = CH -, = C (Me) _{-N =, CH 2, O,} Et, H, H, H, O], [AH777; C, -CH = CH -, = C (Me) -N =, CH 2, O, c-Pr, H , H, H, O], [AH778; C, -CH = CH -, = C (Me) -N =, CH 2, O, OMe, H, H, H, O], [AH779; C, - _{CH = C (CF 3) -} , = CH-N =, CH 2, O, H, H, H, H, O], [AH780; C, -CH = C (CF 3) -, = CH-N =, CH ₂ , O, Cl, H, H, H, O], [AH 781; C, -CH = C (CF ₃ )-, = CH-N =, CH ₂ , O, Br, H, H, H H, O], [AH782; C, -CH = C (CF 3) -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [AH783; C, -CH _{= C (CF 3) -,} = CH-N =, CH 2, O, Me, H, H, H, O], [AH784; C, -CH = C (CF 3) -, = CH-N = _{, CH 2, O, Et,} H, H, H, O], [AH785; C, -CH = C (CF 3) -, = CH-N =, CH 2, O, c-Pr, H, H , H, O], [AH786 ; C, -CH = C (CF 3) -, = CH-N =, CH 2, O, OMe, H, H, H, O], [AH787; C, -C (CF ₃ ) = CH-, = CH-N =, CH ₂ , O, H, H, H, H, O], [AH 788; C,-C (CF ₃ ) = CH-, = CH-N =, CH ₂ , O, Cl, H, H , H, O], [AH789; C, -C (CF 3) = CH -, = CH-N =, CH 2, O, Br, H, H, H, O] , [AH790; C, -C ( CF 3) = CH -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [AH791; C, -C (CF 3) = CH -, = CH-N =, CH 2, O, Me, H, H, H, O], [AH792; C, -C (CF 3) = CH -, = CH-N =, CH 2, O, Et, H, H, H, O], [AH793; C, -C (CF 3) = CH -, = CH-N =, CH 2, O, c-Pr, H, H, H, O ], [AH794; C, -C (CF 3) = CH -, = = CH-N, CH 2, O, OMe, H, H, H, O], [AH795; C, -CH = CH-, _{= C (CF 3) -N =} , CH 2, O, H, H, H, H, O], [AH796; C, -CH = CH -, = C (CF 3) -N =, CH 2, O, Cl, H, H, H, O], [AH797; C, -CH = CH -, = C (CF 3) -N =, CH 2, O, Br, H, H, H, O], [AH798; C, -CH = CH -, = C (CF 3) -N =, CH 2, O, CF 3, H, H, H, O], [AH799; C, -CH = CH -, = _{C (CF 3) -N =,} CH 2, O, Me, H, H, H, O], [AH800; C, -CH = CH -, = C (CF 3) -N =, CH 2, O , Et, H, H, H, O],

[AH801; C, -CH = CH -, = C (CF 3) -N =, CH 2, O, c-Pr, H, H, H, O], [AH802; C, -CH = CH-, _{= C (CF 3) -N =} , CH 2, O, OMe, H, H, H, O], [AH803; C, = CH-CH = CH -, - C (Me) =, CH 2, O , H, H, H, H, O], [AH 804; C, = CH-CH = CH-,-C (Me) =, CH ₂ , O, Cl, H, H, H, O], [AH 805 ; C, = CH-CH = CH -, - C (Me) =, CH 2, O, Br, H, H, H, O], [AH806; C, = CH-CH = CH -, - C ( _{Me) =, CH 2, O} , CF 3, H, H, H, O], [AH807; C, = CH-CH = CH -, - C (Me) =, CH 2, O, Me, H, H, H, O], [AH 808; C, = CH-CH = CH-, -C (Me) =, CH ₂ , O, Et, H, H, H, O], [AH 809; C, = CH -CH = CH -, - C ( Me) =, CH 2, O, c-Pr, H, H, H, O], [AH810; C, = CH-CH = CH -, - C (Me) = _{, CH 2, O, OMe,} H, H, H, O], [AH811; C, = CH-CH = CF -, - C (Me) =, CH 2, O, H, H, H, H, O], [AH812; C, = CH-CH = CF -, - C (Me) =, CH 2, O, Cl, H, H, H, O], [AH813; C, = CH-CH = CF -, - C (Me) = , CH 2, O, Br, H, H, H, O], [AH814; C, = CH-CH = CF -, - C (Me) =, CH 2, O, _{CF 3, H, H, H} , O], [AH815; C, = CH-CH = CF -, - C (Me) =, CH 2, O, Me, H, H, H, O], [AH816 ; C, = CH-CH = CF -, - C (Me) =, CH 2, O, Et, H, H, H, O], [AH817; C, = CH-CH = CF -, - C ( _{Me) =, CH 2, O} , c-Pr, H, H, H, O], [AH818; C, = CH-CH = CF -, - C (Me) =, CH 2, O, OMe, H , H, H, O], [AH 819; C, = CH-CF = CH-, -C (Me) =, CH ₂ , O, H, H, H, H, O], [AH 820; C, = CH-CF = CH -, - C (Me) =, CH 2, O, Cl, H, H, H, O], [AH821; C, = CH-CF = CH -, - C (M _{e) =, CH 2, O} , Br, H, H, H, O], [AH822; C, = CH-CF = CH -, - C (Me) =, CH 2, O, CF 3, H, H, H, O], [AH 823; C, = CH-CF = CH-, -C (Me) =, CH ₂ , O, Me, H, H, H, O], [AH 824; C, = CH -CF = CH -, - C ( Me) =, CH 2, O, Et, H, H, H, O], [AH825; C, = CH-CF = CH -, - C (Me) =, CH ₂ , O, c-Pr, H, H, H, O], [AH 826; C, = CH-CF = CH-,-C (Me) =, CH ₂ , O, OMe, H, H, H, H O], [AH 827; C, = CF-CH = CH-, -C (Me) =, CH ₂ , O, H, H, H, H, O], [AH 828; C, = CF-CH = CH -, - C (Me) = , CH 2, O, Cl, H, H, H, O], [AH829; C, = CF-CH = CH -, - C (Me) =, CH 2, O, br, H, H, H, O], [AH830; C, = CF-CH = CH -, - C (Me) =, CH 2, O, CF 3, H, H, H, O], [AH831 ; C, = CF-CH = CH -, - C (Me) =, CH 2, O, Me, H, H, H, O], [AH832; C, = CF-CH = CH -, - C ( _{Me) =, CH 2, O} , Et, H, H, H, O], [AH833; C, = CF-CH = CH -, - C (Me) =, CH 2, O, c-Pr, H , H, H, O], [AH834; C, = CF-CH = CH -, - C (Me) =, CH 2, O, OMe, H, H, H, O], [AH835; C, = CH-CH = CH -, - C (Br) =, CH 2, O, H, H, H, H, O], [AH836; C, = CH-CH = CH -, - C (Br) =, _{CH 2, O, Cl, H} , H, H, O], [AH837; C, = CH-CH = CH -, - C (Br) =, CH 2, O, Br, H, H, H, O ], [AH838; C, = CH-CH = CH -, - C (Br) =, CH 2, O, CF 3, H, H, H, O], [AH839; C, = CH-CH = CH -, - C (Br) = , CH 2, O, Me, H, H, H, O], [AH840; C, = CH-CH = CH -, - C (Br) =, CH 2, O, Et, H, H, H, O], [AH841; C, = CH-CH = CH -, - C (Br) =, CH 2, O, c-Pr, H, H, H, O], [ AH842; C, = CH-CH = CH -, - C (Br) =, CH 2, O, OMe, H, H, H, O], [AH843; C, = CH-CH = CH -, - C _{(Cl) =, CH 2,} O, H, H, H, H, O], [AH844; C, = CH-CH = CH -, - C (Cl) =, CH 2, O, Cl, H, H, H, O], [AH 845; C, = CH-CH = CH-,-C (Cl) =, CH ₂ , O, Br, H, H, H, O], [AH 846; C, = CH -CH = CH -, - C ( Cl) =, CH 2, O, CF 3, H, H, H, O], [AH847; C, = CH-CH = CH -, - C (Cl) =, CH ₂ , O, Me, H, H, H, O, [AH 848; C, = CH-CH = CH-, -C (Cl) =, CH ₂ , O, Et, H, H, H, O ], [AH849; C, = CH-CH = CH -, - C (Cl) =, CH 2, O, c-Pr, H, H, H, O], [AH850; C, = CH-CH = CH -, - C (Cl) =, CH 2, O, OMe, H, H, H, O], [AH851; C, = CH-C (Me) = CH -, - C (Me) =, CH _{2, O, H, H,} H, H, O], [AH852; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, O, Cl, H, H, H , O], [AH853; C , = CH-C (Me) = CH -, - C (Me) =, CH 2, O, Br, H, H, H, O], [AH854; C, = CH -C (Me) = CH -, - C (Me) =, CH 2, O, CF 3, H, H, H, O], [AH855; C, = CH-C (Me) = CH -, - _{C (Me) =, CH 2} , O, Me, H, H, H, O], [AH856; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, O, Et, H, H, H, O], [AH 857; C, = CH-C (Me) = CH-,-C (Me) =, CH ₂ , O, c-Pr, H, H, H, O ], [AH858; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, O, OMe, H, H, H, O], [AH859; C, = CH-CH = CH -, - C (CF 3) =, CH 2, O, H, H, H, H, O], [AH860; C, = CH-CH = CH -, - C (CF 3) =, CH _{2, O, Cl, H,} H, H, O], [AH861; C, = CH-CH = CH -, - C (CF 3) =, CH 2, O, Br, H, H, H, O ], [AH862; C, = CH-CH = CH -, - C (CF 3) =, CH 2, O, CF 3, H, H, H, O], [AH863; C, = CH-CH = _{CH -, - C (CF 3} ) =, CH 2, O, Me, H, H, H, O], [AH864; C, = CH-CH = CH -, - C (CF 3) =, CH 2 , O, Et, H, H , H, O], [AH865; C, = CH-CH = CH -, - C (CF 3) =, CH 2, O, c-Pr, H, H, H, O], [AH866; C, = CH-CH = CH -, - C (CF 3) =, CH 2, O, OMe, H, H, H, O], [AH867; C, -CH = CH- , = CH-N =, CH 2, O, H, H, H, H, O], [AH868; C, -CH = CH -, = CH-N =, CH 2, O, Cl, H, H , H, O], [AH869 ; C, -CH = CH -, = = CH-N, CH 2, O, Br, H, H, H, O], [AH870; C, -CH = CH-, _{= CH-N =, CH 2} , O, CF 3, H, H, H, O], [AH871; C, -CH = CH -, = CH-N =, CH 2, O, Me, H, H , H, O], [AH872 ; C, -CH = CH -, = = CH-N, CH 2, O, Et, H, H, H, O], [AH873; C, -CH = CH-, _{= CH-N =, CH 2} , O, c-Pr, H, H, H, O], [AH874; C, -CH = CH -, = CH-N =, CH 2, O, OMe, H, H, H, O], [ AH875; C, -CH = CF -, = CH-N =, CH 2, O, H, H, H, H, O], [AH876; C, -CH = CF- , = CH-N =, CH 2, O, Cl, H, H, H, O], [AH877; C, -CH = CF -, = CH-N =, CH 2, O, Br, H, H , H, O], [AH878 ; C, -CH = CF -, = CH-N =, CH 2, O, CF 3, H, H, H, O], [AH879; C, -CH = CF- , = CH-N =, CH 2, O, Me, H, H, H, O], [AH880; C, -CH = CF -, = CH-N =, CH 2, O, Et, H, H , H, O], [AH881 ; C, -CH = CF -, = CH-N =, CH 2, O, c-Pr, H, H, H, O], [AH882; C, -CF = CH -, = CH-N =, CH 2, O, H, H, H, H, O], [AH883; C, -CF = CH -, = CH-N =, C _{H 2, O, Cl, H} , H, H, O], [AH884; C, -CF = CH -, = CH-N =, CH 2, O, Br, H, H, H, O], [ AH885; C, -CF = CH - , = CH-N =, CH 2, O, CF 3, H, H, H, O], [AH886; C, -CF = CH -, = CH-N =, _{CH 2, O, Me, H} , H, H, O], [AH887; C, -CF = CH -, = CH-N =, CH 2, O, Et, H, H, H, O], [ AH888; C, -CF = CH - , = CH-N =, CH 2, O, c-Pr, H, H, H, O], [AH889; C, -CF = CH -, = CH-N = _{, CH 2, O, OMe,} H, H, H, O], [AH890; C, -CH = CH -, = CF-N =, CH 2, O, H, H, H, H, O], [AH891; C, -CH = CH -, = CF-N =, CH 2, O, Cl, H, H, H, O], [AH892; C, -CH = CH -, = CF-N =, _{CH 2, O, Br, H} , H, H, O], [AH893; C, -CH = CH -, = CF-N =, CH 2, O, CF 3, H, H, H, O], [AH894; C, -CH = CH -, = CF-N =, CH 2, O, Me, H, H, H, O], [AH895; C, -CH = CH -, = CF-N =, _{CH 2, O, Et, H} , H, H, O], [AH896; C, -CH = CH -, = CF-N =, CH 2, O, c-Pr, H, H, H, O] , [AH897; C, -CH = CH -, = CF-N =, CH 2, O, OMe, H, H, H, O], [AH898; C, = CH-CH = CH -, - CH = , CH ₂ , O, H, H, H, H, H, O], [AH 899; C, = CH-CH = CH-, -CH =, CH ₂ , O, Cl, H, H, H, O], [AH900; C, = CH- CH = CH -, - CH =, CH 2, O, Br, H, H, H, O],

[AH901; C, = CH- CH = CH -, - CH =, CH 2, O, CF 3, H, H, H, O], [AH902; C, = CH-CH = CH -, - CH = _{, CH 2, O, Me,} H, H, H, O], [AH903; C, = CH-CH = CH -, - CH =, CH 2, O, Et, H, H, H, O], [AH904; C, = CH- CH = CH -, - CH =, CH 2, O, c-Pr, H, H, H, O], [AH905; C, = CH-CH = CH -, - CH _{=, CH 2, O, OMe} , H, H, H, O], [AH906; C, = CH-CH = CH -, - N =, CH 2, O, H, H, H, H, O] , [AH907; C, = CH -CH = CH -, - N =, CH 2, O, Cl, H, H, H, O], [AH908; C, = CH-CH = CH -, - N = _{, CH 2, O, Br,} H, H, H, O], [AH909; C, = CH-CH = CH -, - N =, CH 2, O, CF 3, H, H, H, O] , [AH910; C, = CH -CH = CH -, - N =, CH 2, O, Me, H, H, H, O], [AH911; C, = CH-CH = CH -, - N = _{, CH 2, O, Et,} H, H, H, O], [AH912; C, = CH-CH = CH -, - N =, CH 2, O, c-Pr, H, H, H, O ], [AH913; C, = CH-CH = CH -, - N =, CH 2, O, OMe, H, H, H, O], [AH914; C, = CH-C (Me) = CH- _{, -N =, CH 2, O} , H, H, H, H, O], [AH915; C, = CH-C (Me) = CH -, - N =, CH 2, O, Cl, H, H, H, O], [ AH916; C, = CH-C (Me) = CH -, - N =, CH 2, O, Br, H, H, H, O], [AH917; C, = CH -C (Me) = CH -, - N =, CH 2, O, CF 3, H, H, H, O], [AH918; C, = CH-C (Me) = CH -, - N =, _{CH 2, O, Me, H} , H, H, O], [AH919; C, = CH-C (Me) = CH -, - N =, CH 2, O, Et, H, H, H, O ], [AH920; C, = CH-C (Me) = CH -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH921; C, = CH-C ( Me) = CH -, - N =, CH 2, O, OMe, H, H, H, O], [AH922; C, = C (Me) -CH = CH -, - N =, CH 2 , O, H, H, H , H, O], [AH923; C, = C (Me) -CH = CH -, - N =, CH 2, O, Cl, H, H, H, O], [AH924; C, = C ( Me) -CH = CH -, - N =, CH 2, O, Br, H, H, H, O], [AH925; C, = C (Me) -CH = CH _{-, - N =, CH 2} , O, CF 3, H, H, H, O], [AH926; C, = C (Me) -CH = CH -, - N =, CH 2, O, Me, H, H, H, O] , [AH927; C, = C (Me) -CH = CH -, - N =, CH 2, O, Et, H, H, H, O], [AH928; C, = C (Me) -CH = CH -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH929; C, = C (Me) -CH = CH -, - _{N =, CH 2, O,} OMe, H, H, H, O], [AH930; C, = CH-C (CF 3) = CH -, - N =, CH 2, O, H, H, H , H, O], [AH931 ; C, = CH-C (CF 3) = CH -, - N =, CH 2, O, Cl, H, H, H, O], [AH932; C, = CH _{-C (CF 3) = CH -} , - N =, CH 2, O, Br, H, H, H, O], [AH933; C, = CH-C (CF 3) = CH -, - N = _{, CH 2, O, CF 3} , H, H, H, O], [AH934; C, = CH-C (CF 3) = CH -, - N =, CH 2, O, Me, H, H, H, O], [AH935; C, = CH-C (CF 3) = CH -, - N =, CH 2, O, Et, H, H, H, O], [AH936; C, = CH- _{C (CF 3) = CH -} , - N =, CH 2, O, c-Pr, H, H, H, O], [AH937; C, = CH-C (CF 3) = CH -, - N =, CH ₂ , O, OMe, H, H, H, O], [AH 938; C, = C (CF ₃ ) -CH = CH-, -N =, CH ₂ , O, H, H, H, H H, O], [AH939; C, = C (CF 3) -CH = CH -, - N =, CH 2, O, Cl, H, H, H, O], [AH940; C, = C ( _{CF 3) -CH = CH -,} - N =, CH 2, O, Br, H, H, H, O], [AH941; C, = C (CF 3) -CH = CH -, - N =, _{CH 2, O, CF 3,} H, H, H, O], [AH942; C, = C (CF 3) -CH = CH -, - N =, CH 2, O, Me, H, H, H, O], [ AH943; C, = C (CF 3) -CH = CH -, - N =, CH 2, O, Et, H, H, H, O], [AH944; C, = _{C (CF 3) -CH = CH} -, - N =, CH 2, O, c-Pr, H, H, H, O], [AH945; C, = C (CF 3) -CH = CH-, _{-N =, CH 2, O,} OMe, H, H, H, O], [AH946; C, -CH = CH -, = CH-C (Me) =, CH 2, S, H, H, H , H, O], [AH947 ; C, -CH = CH -, = CH-C (Me) =, CH 2, S, Cl, H, H, H, O], [AH948; C, -CH = CH -, = CH-C ( Me) =, CH 2, S, Br, H, H, H, O], [AH949; C, -CH = CH -, = CH-C (Me) =, CH 2 _{, S, CF 3, H,} H, H, O], [AH950; C, -CH = CH -, = CH-C (Me) =, CH 2, S, Me, H, H, H, O] , [AH 951; C, -CH = CH-, = CH-C (Me) =, CH ₂ , S, Et, H, H, H, O], [AH 952; C, -CH = CH-, = CH _{-C (Me) =, CH 2} , S, c-Pr, H, H, H, O], [AH953; C, -CH = CH -, = CH-C (Me) =, CH 2, S, OMe, H, H, H, O], [AH954; C, -CH = CF -, = CH-C (Me) =, CH 2, S, H, H, H, H, O], [AH955; C, -CH = CF -, = CH-C (Me) =, CH 2, S, Cl, H, H, H, O], [AH956; C, -CH = CF -, = CH-C (Me ), = CH ₂ , S, Br, H, H, H, O], [AH 957; C,-CH = CF-, = CH-C (Me) =, CH ₂ , S, CF ₃ , H, H , H, O], [AH958 ; C, -CH = CF -, = CH-C (Me) =, CH 2, S, Me, H, H, H, O], [AH959; C, -CH = CF -, = CH-C ( Me) =, CH 2, S, Et, H, H, H, O], [AH960; C, -CH = CF -, = CH-C (Me) =, CH 2 , S, c-Pr, H , H, H, O], [AH961; C, -CH = CF -, = CH-C (Me) =, CH 2, S, OMe, H, H, H, O ], [AH962; C, -CF = CH -, = CH-C (Me) =, CH 2, S, H, H, H, H, O], [AH963; C, -CF = CH -, = CH-C (Me ) =, CH 2, S, Cl, H, H, H, O], [AH964; C, -CF = CH -, = CH-C (Me) =, CH 2, S, Br, H, H, H, O], [AH965; C, -CF = CH -, = CH-C (Me) =, CH 2, S, CF 3, H, H, H, O], [AH966; C, -CF = CH -, = CH-C (Me) =, CH 2, S, Me, H, H, H, O], [AH967; C, -CF = CH -, = CH- _{C (Me) =, CH 2} , S, Et, H, H, H, O], [AH968; C, -CF = CH -, = CH-C (Me) =, CH 2, S, c-Pr , H, H, H, O ], [AH969; C, -CF = CH -, = CH-C (Me) =, CH 2, S, OMe, H, H, H, O], [AH970; C , -CF = CH -, = CH -C (Me) =, CH 2, S, H, H, H, H, O], [AH971; C, -CF = CH -, = CH-C (Me) _{=, CH 2, S, Cl} , H, H, H, O], [AH972; C, -CF = CH -, = CH-C (Me) =, CH 2, S, Br, H, H, H , O], [AH973; C , -CF = CH -, = CH-C (Me) =, CH 2, S, CF 3, H, H, H, O], [AH974; C, -CF = CH -, = CH-C (Me ) =, CH 2, S, Me, H, H, H, O], [AH975; C, -CF = CH -, = CH-C (Me) =, CH 2, S, Et, H, H, H, O], [AH976; C, -CF = CH -, = CH-C (Me) =, CH 2, S, c-Pr, H, H, H, O] , [AH977; C, -CF = CH -, = CH-C (Me) =, CH 2, S, OMe, H, H, H, O], [AH978; C, -CH = CH -, = CF _{-C (Me) =, CH 2} , S, H, H, H, H, O], [AH979; C, -CH = CH -, = CF-C (Me) =, CH 2, S, Cl, H, H, H, O] , [AH980; C, -CH = CH -, = CF-C (Me) =, CH 2, S, Br, H, H, H, O], [AH981; C, -CH = CH -, = CF- C (Me) =, CH 2, S, CF 3, H, H, H, O], [AH982; C, -CH = CH -, = CF-C (Me) _{=, CH 2, S, Me} , H, H, H, O], [AH983; C, -CH = CH -, = CF-C (Me) =, CH 2, S, Et, H, H , H, O], [AH984 ; C, -CH = CH -, = CF-C (Me) =, CH 2, S, c-Pr, H, H, H, O], [AH985; C, - CH = CH -, = CF- C (Me) =, CH 2, S, OMe, H, H, H, O], [AH986; C, -CH = CH -, = CH-CBr =, CH 2, S, H, H, H, H, O], [AH987; C, -CH = CH -, = CH-CBr =, CH 2, S, Cl, H, H, H, O], [AH988; C , -CH = CH -, = CH -CBr =, CH 2, S, Br, H, H, H, O], [AH989; C, -CH = CH -, = CH-CBr =, CH 2, S _{, CF 3, H, H,} H, O], [AH990; C, -CH = CH -, = CH-CBr =, CH 2, S, Me, H, H, H, O], [AH991; C , -CH = CH -, = CH -CBr =, CH 2, S, Et, H, H, H, O], [AH992; C, -CH = CH -, = CH-CBr =, CH 2, S , c-Pr, H, H , H, O], [AH993; C, -CH = CH -, = CH-CBr =, CH 2, S, OMe, H, H, H, O], [AH994; C, -CH = CH -, = CH-CCl =, CH 2, S, H, H, H, H, O], [AH995; C, -CH = CH -, = CH-CCl =, CH 2, S, Cl, H, H, H, O], [AH996; C, -CH = CH -, = CH-CCl =, CH 2, S, Br, H, H, H, O], [AH997; C , -CH = CH -, = CH -CCl =, CH 2, S, CF 3, H, H, H, O], [AH998; C, -CH = CH -, = CH-CCl =, CH 2, S, Me, H, H, H, O], [AH999; C, -CH = CH -, = CH-CCl =, CH 2, S, Et, H, H, H, O], [AH1000; C , -CH = CH -, = CH -CCl =, CH 2, S, c-Pr, H, H, H, O],

[AH1001; C, -CH = CH -, = CH-CCl =, CH 2, S, OMe, H, H, H, O], [AH1002; C, -C (Me) = CH -, = CH- _{C (Me) =, CH 2} , S, H, H, H, H, O], [AH1003; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, S, Cl, H, H, H, O], [AH1004; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, S, Br, H, H, H, O], [AH1005; C, -C (Me ) = CH -, = CH-C (Me) =, CH 2, S, CF 3, H, H, H, O], [AH1006; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, S, Me, H, H, H, O], [AH1007; C, -C (Me) = CH -, = CH-C (Me) =, CH ₂ , S, Et, H, H, H, O], [AH 1008; C, -C (Me) = CH-, = CH-C (Me) =, CH ₂ , S, c-Pr, H, H, H, O] , [AH1009; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, S, OMe, H, H, H, O], [AH1010 ; C, -CH = CH -, = CH-C (CF 3) =, CH 2, S, H, H, H, H, O], [AH1011; C, -CH = CH -, = CH-C _{(CF 3) =, CH 2} , S, Cl, H, H, H, O], [AH1012; C, -CH = CH -, = CH-C (CF 3) =, CH 2, S, Br, H, H, H, O] , [AH1013; C, -CH = CH -, = CH-C (CF 3) =, CH 2, S, CF 3, H, H, H, O], [AH1014; C, -CH = CH -, = CH-C (CF 3) =, CH 2, S, Me, H, H, H, O], [AH1015; C, -CH = CH -, = CH-C ( CF ₃ ) =, CH ₂ , S, Et, H, H, H, O], [AH 1016; C, -CH = CH-, = CH-C (CF ₃ ) =, CH ₂ , S, c-Pr , H, H, H, O ], [AH1017; C, -CH = CH -, = CH-C (CF 3) =, CH 2, S, OMe, H, H, H, O], [AH1018; C, -CH = CH -, = CH-C (Et) =, CH 2, S, H, H, H, H, O], [AH1019; C, -CH = CH -, = CH-C (Et ), CH ₂ , S, Cl, H, H, H, O], [AH 1020; C, -CH = CH -, = CH-C (Et) =, CH 2, S, Br, H, H, H, O], [AH1021; C, -CH = CH -, = CH-C (Et) =, CH ₂ , S, CF ₃ , H, H, H, O], [AH 1022; C, -CH = CH-, = CH-C (Et) =, CH ₂ , S, Me, H, H, H, O ], [AH1023; C, -CH = CH -, = CH-C (Et) =, CH 2, S, Et, H, H, H, O], [AH1024; C, -CH = CH -, = CH-C (Et) =, CH 2, S, c-Pr, H, H, H, O], [AH1025; C, -CH = CH -, = CH-C (Et) =, CH 2, S , OMe, H, H, H , O], [AH1026; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, S, H, H, H, H, O], [AH1027; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, S, Cl, H, H, H, O], [AH1028; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, S, Br, H, H, H, O], [AH1029; C, -CH = CH -, = CH-C (c-Pr) =, CH 2 , S, CF ₃ , H, H, H, O], [AH 1030; C, -CH = CH-, = CH-C (c-Pr) =, CH ₂ , S, Me, H, H, H, H O], [AH1031; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, S, Et, H, H, H, O], [AH1032; C, -CH = CH -, = CH-C (c -Pr) =, CH 2, S, c-Pr, H, H, H, O], [AH1033; C, -CH = CH -, = CH-C (c-Pr ), = CH ₂ , S, OMe, H, H, H, O], [AH 1034; N, -CH = CH-, -N =, CH ₂ , S, H, H, H, H, O], [AH1035; N, -CH = CH -, - N =, CH 2, S, F, H, H, H, O], [AH1036; N, -CH = CH -, - N =, CH 2, S , Cl, H, H, H , O], [AH1037; N, -CH = CH -, - N =, CH 2, S, Br, H, H, H, O], [AH1038; N, -CH = CH -, - N =, CH 2, S, Me, H, H, H, O], [AH1039; N, -CH = CH -, - N =, CH 2, S, Et, H, H, H, O], [AH1040; N, -CH = CH -, - N =, CH 2, S, Pr, H, H, H, O], [AH1041; N, -CH = CH -, - N =, CH 2, S, i-Pr, H, H, H, O], [AH1042; N, -CH = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1043; N, -CH = CH -, - N =, CH 2, S, c-Bu, H, H, H, O], [AH1044; N , -CH = CH -, - N =, CH 2, S, OMe, H, H, H, O], [AH1045; N, -CH = CH -, - N =, CH 2, S, Oi-Pr , H, H, H, O ], [AH1046; N, -CH = CH -, - N =, CH 2, S, SMe, H, H, H, O], [AH1047; N, -CH = CH _{-, - N =, CH 2} , S, Set, H, H, H, O], [AH1048; N, -CH = CH -, - N =, CH 2, S, CF 3, H, H, H , O], [AH1049; N , -CH = CH -, - N =, CH 2, S, CHF 2, H, H, H, O], [AH1050; N, -CH = CH -, - N = _{, CH 2, S, OCF 3} , H, H, H, O], [AH1051; N, -CH = CH -, - N =, CH 2, S, OCHF 2, H, H, H, O], [AH1052; N, -CH = CH -, - N =, CH 2, S, CH = CH 2, H, H, H, O], [AH1053; N, -CH = CH -, - N =, CH _{2, S, C (Me)} = CH 2, H, H, H, O], [AH1054; N, -CH = CH -, - N =, CH 2, S, CH = CHMe, H, H, H , O], [AH1055; N , -CH = CH -, - N =, CH 2, S, C≡CH, H, H, H, O], [AH1056; N, -CH = CH -, - N _{=, CH 2, S, C≡CMe} , H, H, H, O], [AH1057; N, -CH = CH -, - N =, CH 2, S, CN, H, H, H, O] , [AH1058; N, -CH = CF -, - N =, CH 2, S, H, H, H, H, O], [AH1059; N, -CH = CF -, - N =, CH 2, S, Cl, H, H, H, O], [AH1060; N, -CH = CF -, - N =, CH 2, S, Br, H, H, H, O], [AH1061; N, - CH = CF -, - N = , CH 2, S, CF 3, H, H, H, O], [AH1062; N, -CH = CF -, - N =, CH 2, S, Me, H, H, H, O], [AH 1063; N, -CH = CF-, -N =, CH _{2, S, Et, H,} H, H, O], [AH1064; N, -CH = CF -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1065 ; N, -CH = CF -, - N =, CH 2, S, OMe, H, H, H, O], [AH1066; N, -CF = CH -, - N =, CH 2, S, H , H, H, H, O ], [AH1067; N, -CF = CH -, - N =, CH 2, S, Cl, H, H, H, O], [AH1068; N, -CF = CH _{-, - N =, CH 2} , S, Br, H, H, H, O], [AH1069; N, -CF = CH -, - N =, CH 2, S, CF 3, H, H, H , O], [AH1070; N , -CF = CH -, - N =, CH 2, S, Me, H, H, H, O], [AH1071; N, -CF = CH -, - N =, _{CH 2, S, Et, H} , H, H, O], [AH1072; N, -CF = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [ AH1073; N, -CF = CH - , - N =, CH 2, S, OMe, H, H, H, O], [AH1074; N, -CH = CCl -, - N =, CH 2, S, H, H, H, H, O], [AH1075; N, -CH = CCl -, - N =, CH 2, S, Cl, H, H, H, O], [AH1076; N, -CH = CCl -, - N =, CH 2, S, Br, H, H, H, O], [AH1077; N, -CH = CCl -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1078; N, -CH = CCl -, - N =, CH 2, S, Me, H, H, H, O], [AH1079; N, -CH = CCl -, - N = _{, CH 2, S, Et,} H, H, H, O], [AH1080; N, -CH = CCl -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1081; N, -CH = CCl -, - N =, CH 2, S, OMe, H, H, H, O], [AH1082; N, -CCl = CH -, - N =, CH 2, S , H, H, H, H , O], [AH1083; N, -CCl = CH -, - N =, CH 2, S, Cl, H, H, H, O], [AH1084; N, -CCl = CH -, - N =, CH 2, S, Br, H, H, H, O], [AH1085; N, -CCl = CH -, - N =, CH 2, S, CF 3, H, H , H, O], [AH1086 ; N, -CCl = CH -, - N =, CH 2, S, M e, H, H, H, O], [AH1087; N, -CCl = CH -, - N =, CH 2, S, Et, H, H, H, O], [AH1088; N, -CCl = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1089; N, -CCl = CH -, - N =, CH 2, S, OMe, H, H , H, O], [AH1090 ; N, -CH = C (Me) -, - N =, CH 2, S, H, H, H, H, O], [AH1091; N, -CH = C ( Me) -, - N =, CH 2, S, Cl, H, H, H, O], [AH1092; N, -CH = C (Me) -, - N =, CH 2, S, Br, H , H, H, O], [AH1093; N, -CH = C (Me) -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1094; N, -CH = C (Me) -, - N =, CH 2, S, Me, H, H, H, O], [AH1095; N, -CH = C (Me) -, - N =, CH 2, S, Et, H, H, H, O], [AH1096; N, -CH = C (Me) -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1097; N, -CH = C (Me) -, - N =, CH 2, S, OMe, H, H, H, O], [AH1098; N, -C (Me) = CH -, - N =, CH _{2, S, H, H,} H, H, O], [AH1099; N, -C (Me) = CH -, - N =, CH 2, S, Cl, H, H, H, O], [ AH1100; N, -C (Me) = CH -, - N =, CH 2, S, Br, H, H, H, O],

[AH1101; N, -C (Me ) = CH -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1102; N, -C (Me) = CH -, - _{N =, CH 2, S,} Me, H, H, H, O], [AH1103; N, -C (Me) = CH -, - N =, CH 2, S, Et, H, H, H, O], [AH1104; N, -C (Me) = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1105; N, -C (Me) = CH -, - N =, CH 2, S, OMe, H, H, H, O], [AH1106; N, -CH = CH -, - N =, CH 2, S, H, F, H, H , O], [AH1107; N , -CH = CH -, - N =, CH 2, S, Cl, F, H, H, O], [AH1108; N, -CH = CH -, - N =, _{CH 2, S, Br, F} , H, H, O], [AH1109; N, -CH = CH -, - N =, CH 2, S, CF 3, F, H, H, O], [AH1110 ; N, -CH = CH -, - N =, CH 2, S, Me, F, H, H, O], [AH1111; N, -CH = CH -, - N =, CH 2, S, Et , F, H, H, O ], [AH1112; N, -CH = CH -, - N =, CH 2, S, c-Pr, F, H, H, O], [AH1113; N, -CH = CH -, - N =, CH 2, S, OMe, F, H, H, O], [AH1114; N, -CH = CH -, - N =, CH 2, S, H, H, F, H, O], [AH1115; N, -CH = CH -, - N =, CH 2, S, Cl, H, F, H, O], [AH1116; N, -CH = CH -, - N = _{, CH 2, S, Br,} H, F, H, O], [AH1117; N, -CH = CH -, - N =, CH 2, S, CF 3, H, F, H, O], [ AH1118; N, -CH = CH - , - N =, CH 2, S, Me, H, F, H, O], [AH1119; N, -CH = CH -, - N =, CH 2, S, Et, H, F, H, O], [AH1120; N, -CH = CH -, - N =, CH 2, S, c-Pr, H, F, H, O], [AH1121; N, - CH = CH -, - N = , CH 2, S, OMe, H, F, H, O], [AH1122; N, -CH = CH -, - N =, CH 2, S, H, H, H , F, O], [AH1123 ; N, -CH = CH -, - N =, CH 2, S, Cl, H, H , F, O], [AH1124 ; N, -CH = CH -, - N =, CH 2, S, Br, H, H, F, O], [AH1125; N, -CH = CH -, - N _{=, CH 2, S, CF} 3, H, H, F, O], [AH1126; N, -CH = CH -, - N =, CH 2, S, Me, H, H, F, O], [AH1127; N, -CH = CH -, - N =, CH 2, S, Et, H, H, F, O], [AH1128; N, -CH = CH -, - N =, CH 2, S , c-Pr, H, H , F, O], [AH1129; N, -CH = CH -, - N =, CH 2, S, OMe, H, H, F, O], [AH1130; C, = CH-S -, - N =, CH 2, S, H, H, H, H, O], [AH1131; C, = CH-S -, - N =, CH 2, S, F, H, H, H, O], [ AH1132; C, = CH-S -, - N =, CH 2, S, Cl, H, H, H, O], [AH1133; C, = CH-S -, - _{N =, CH 2, S,} Br, H, H, H, O], [AH1134; C, = CH-S -, - N =, CH 2, S, Me, H, H, H, O], [AH1135; C, = CH- S -, - N =, CH 2, S, Et, H, H, H, O], [AH1136; C, = CH-S -, - N =, CH 2, S , Pr, H, H, H , O], [AH1137; C, = CH-S -, - N =, CH 2, S, i-Pr, H, H, H, O], [AH1138; C, = CH-S -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1139; C, = CH-S -, - N =, CH 2, S, c- Bu, H, H, H, O], [AH1140; C, = CH-S -, - N =, CH 2, S, OMe, H, H, H, O], [AH1141; C, = CH- S -, - N =, CH 2, S, Oi-Pr, H, H, H, O], [AH1142; C, = CH-S -, - N =, CH 2, S, SMe, H, H , H, O], [AH1143 ; C, = CH-S -, - N =, CH 2, S, Set, H, H, H, O], [AH1144; C, = CH-S -, - N _{=, CH 2, S, CF} 3, H, H, H, O], [AH1145; C, = CH-S -, - N =, CH 2, S, CHF 2, H, H, H, O] , [AH1146; C, = CH -S -, - N =, CH 2, S, OCF 3, H, H, H, O], [AH1147; C, = CH-S -, - _{N =, CH 2, S,} OCHF 2, H, H, H, O], [AH1148; C, = CH-S -, - N =, CH 2, S, CH = CH 2, H, H, H , O], [AH1149; C , = CH-S -, - N =, CH 2, S, C (Me) = CH 2, H, H, H, O], [AH1150; C, = CH-S _{-, - N =, CH 2} , S, CH = CHMe, H, H, H, O], [AH1151; C, = CH-S -, - N =, CH 2, S, C≡CH, H, H, H, O], [AH 1152; C, = CH-S-,-N =, CH ₂ , S, C≡CMe, H, H, H, O], [AH 1153; C, = C (CF ₃ ) -S -, - N =, CH 2, S, H, H, H, H, O], [AH1154; C, = C (CF 3) -S -, - N =, CH 2, S, Cl , H, H, H, O ], [AH1155; C, = C (CF 3) -S -, - N =, CH 2, S, Br, H, H, H, O], [AH1156; C, _{= C (CF 3) -S -} , - N =, CH 2, S, CF 3, H, H, H, O], [AH1157; C, = C (CF 3) -S -, - N =, _{CH 2, S, Me, H} , H, H, O], [AH1158; C, = C (CF 3) -S -, - N =, CH 2, S, Et, H, H, H, O] , [AH1159; C, = C (CF 3) -S -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1160; C, = C (CF 3) - S -, - N =, CH 2, S, OMe, H, H, H, O], [AH1161; C, = CF-S -, - N =, CH 2, S, H, H, H, H , O], [AH1162; C , = CF-S -, - N =, CH 2, S, Cl, H, H, H, O], [AH1163; C, = CF-S -, - N =, _{CH 2, S, Br, H} , H, H, O], [AH1164; C, = CF-S -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1165 ; C, = CF-S - , - N =, CH 2, S, Me, H, H, H, O], [AH1166; C, = CF-S -, - N =, CH 2, S, Et , H, H, H, O ], [AH1167; C, = CF-S -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1168; C, = CF -S -, - N =, CH 2, S, OMe, H, H, H, O], [AH1169; C, = CCl-S -, - N =, CH _{2, S, H, H,} H, H, O], [AH1170; C, = CCl-S -, - N =, CH 2, S, Cl, H, H, H, O], [AH1171; C , = CCl-S -, - N =, CH 2, S, Br, H, H, H, O], [AH1172; C, = CCl-S -, - N =, CH 2, S, CF 3, H, H, H, O] , [AH1173; C, = CCl-S -, - N =, CH 2, S, Me, H, H, H, O], [AH1174; C, = CCl-S- _{, -N =, CH 2, S} , Et, H, H, H, O], [AH1175; C, = CCl-S -, - N =, CH 2, S, c-Pr, H, H, H , O], [AH1176; C , = CCl-S -, - N =, CH 2, S, OMe, H, H, H, O], [AH1177; C, = C (Me) -S -, - _{N =, CH 2, S,} H, H, H, H, O], [AH1178; C, = C (Me) -S -, - N =, CH 2, S, Cl, H, H, H, O], [AH1179; C, = C (Me) -S -, - N =, CH 2, S, Br, H, H, H, O], [AH1180; C, = C (Me) -S- _{, -N =, CH 2, S} , CF 3, H, H, H, O], [AH1181; C, = C (Me) -S -, - N =, CH 2, S, Me, H, H , H, O], [AH1182 ; C, = C (Me) -S -, - N =, CH 2, S, Et, H, H, H, O], [AH1183; C, = C (Me) -S -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1184; C, = C (Me) -S -, - N =, CH 2, S, OMe , H, H, H, O ], [AH1185; C, = CH-S -, - N =, CH 2, S, H, F, H, H, O], [AH1186; C, = CH-S _{-, - N =, CH 2} , S, Cl, F, H, H, O], [AH1187; C, = CH-S -, - N =, CH 2, S, Br, F, H, H, O], [AH1188; C, = CH-S -, - N =, CH 2, S, CF 3, F, H, H, O], [AH1189; C, = CH-S -, - N =, _{CH 2, S, Me, F} , H, H, O], [AH1190; C, = CH-S -, - N =, CH 2, S, Et, F, H, H, O], [AH1191; C, = CH-S -, - N =, CH 2, S, c-Pr, F, H, H, O], [AH1192; C, = CH-S -, - N =, CH 2, S, OMe, F, H, H, O], [ AH1193; C, = CH-S -, - N =, CH 2, S, H, H, F, H, O], [AH1194; C, = CH-S -, - _{N =, CH 2, S,} Cl, H, F, H, O], [AH1195; C, = CH-S -, - N =, CH 2, S, Br, H, F, H, O], [AH1196; C, = CH- S -, - N =, CH 2, S, CF 3, H, F, H, O], [AH1197; C, = CH-S -, - N =, CH 2, S, Me, H, F, H, O], [AH1198; C, = CH-S -, - N =, CH 2, S, Et, H, F, H, O], [AH1199; C, = CH-S -, - N = , CH 2, S, c-Pr, H, F, H, O], [AH1200; C, = CH-S -, - N =, CH 2, S, OMe, H , F, H, O],

[AH1201; C, = CH- S -, - N =, CH 2, S, H, H, H, F, O], [AH1202; C, = CH-S -, - N =, CH 2, S , Cl, H, H, F , O], [AH1203; C, = CH-S -, - N =, CH 2, S, Br, H, H, F, O], [AH1204; C, = CH -S -, - N =, CH 2, S, CF 3, H, H, F, O], [AH1205; C, = CH-S -, - N =, CH 2, S, Me, H, H , F, O], [AH1206 ; C, = CH-S -, - N =, CH 2, S, Et, H, H, F, O], [AH1207; C, = CH-S -, - N _{=, CH 2, S, c} -Pr, H, H, F, O], [AH1208; C, = CH-S -, - N =, CH 2, S, OMe, H, H, F, O] , [AH1209; C, = CH -O -, - N =, CH 2, S, H, H, H, H, O], [AH1210; C, = CH-O -, - N =, CH 2, S, F, H, H, H, O], [AH1211; C, = CH-O -, - N =, CH 2, S, Cl, H, H, H, O], [AH1212; C, = CH-O -, - N = , CH 2, S, Br, H, H, H, O], [AH1213; C, = CH-O -, - N =, CH 2, S, Me, H, H , H, O], [AH1214 ; C, = CH-O -, - N =, CH 2, S, Et, H, H, H, O], [AH1215; C, = CH-O -, - N _{=, CH 2, S, Pr} , H, H, H, O], [AH1216; C, = CH-O -, - N =, CH 2, S, i-Pr, H, H, H, O] , [AH1217; C, = CH -O -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1218; C, = CH-O -, - N =, CH _{2, S, c-Bu,} H, H, H, O], [AH1219; C, = CH-O -, - N =, CH 2, S, OMe, H, H, H, O], [AH1220 ; C, = CH-O - , - N =, CH 2, S, Oi-Pr, H, H, H, O], [AH1221; C, = CH-O -, - N =, CH 2, S , SMe, H, H, H , O], [AH1222; C, = CH-O -, - N =, CH 2, S, Set, H, H, H, O], [AH1223; C, = CH -O -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1224; C, = CH-O -, - N =, CH 2, S, CHF 2, H, H , H, O], [AH 1225; C, = CH-O-, -N =, CH ₂ , S, OCF ₃ , H, H, H, O], [AH 1226; C, = CH-O-,- _{N =, CH 2, S,} OCHF 2, H, H, H, O], [AH1227; C, = CH-O -, - N =, CH 2, S, CH = CH 2, H, H, H , O], [AH1228; C , = CH-O -, - N =, CH 2, S, C (Me) = CH 2, H, H, H, O], [AH1229; C, = CH-O _{-, - N =, CH 2} , S, CH = CHMe, H, H, H, O], [AH1230; C, = CH-O -, - N =, CH 2, S, C≡CH, H, H, H, O], [AH 1231; C, = CH-O-,-N =, CH ₂ , S, C≡CMe, H, H, H, O], [AH 1232; C, = C (CF ₃ ) -O -, - N =, CH 2, S, H, H, H, H, O], [AH1233; C, = C (CF 3) -O -, - N =, CH 2, S, Cl , H, H, H, O ], [AH1234; C, = C (CF 3) -O -, - N =, CH 2, S, Br, H, H, H, O], [AH1235; C, _{= C (CF 3) -O -} , - N =, CH 2, S, CF 3, H, H, H, O], [AH1236; C, = C (CF 3) -O -, - N =, _{CH 2, S, Me, H} , H, H, O], [AH1237; C, = C (CF 3) -O -, - N =, CH 2, S, Et, H, H, H, O] , [AH1238; C, = C (CF 3) -O -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1239; C, = C (CF 3) - O -, - N =, CH 2, S, OMe, H, H, H, O], [AH1240; C, = CF-O -, - N =, CH 2, S, H, H, H, H , O], [AH1241; C , = CF-O -, - N =, CH 2, S, Cl, H, H, H, O], [AH1242; C, = CF-O -, - N =, _{CH 2, S, Br, H} , H, H, O], [AH1243; C, = CF-O -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1244 ; C, = CF-O - , - N =, CH 2, S, Me, H, H, H, O], [AH1245; C, = CF-O -, - N =, CH 2, S, Et , H, H, H, O ], [AH1246; C, = CF-O -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1247; C, = CF-O -, - N =, CH 2, S, OMe, H, H, H, O], [AH1248; C, = CCl-O -, - N =, CH _{2, S, H, H,} H, H, O], [AH1249; C, = CCl-O -, - N =, CH 2, S, Cl, H, H, H, O], [AH1250; C , = CCl-O -, - N =, CH 2, S, Br, H, H, H, O], [AH1251; C, = CCl-O -, - N =, CH 2, S, CF 3, H, H, H, O] , [AH1252; C, = CCl-O -, - N =, CH 2, S, Me, H, H, H, O], [AH1253; C, = CCl-O- _{, -N =, CH 2, S} , Et, H, H, H, O], [AH1254; C, = CCl-O -, - N =, CH 2, S, c-Pr, H, H, H , O], [AH1255; C , = CCl-O -, - N =, CH 2, S, OMe, H, H, H, O], [AH1256; C, = C (Me) -O -, - _{N =, CH 2, S,} H, H, H, H, O], [AH1257; C, = C (Me) -O -, - N =, CH 2, S, Cl, H, H, H, O], [AH1258; C, = C (Me) -O -, - N =, CH 2, S, Br, H, H, H, O], [AH1259; C, = C (Me) -O- _{, -N =, CH 2, S} , CF 3, H, H, H, O], [AH1260; C, = C (Me) -O -, - N =, CH 2, S, Me, H, H , H, O], [AH1261 ; C, = C (Me) -O -, - N =, CH 2, S, Et, H, H, H, O], [AH1262; C, = C (Me) -O -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1263; C, = C (Me) -O -, - N =, CH 2, S, OMe , H, H, H, O ], [AH1264; C, = CH-O -, - N =, CH 2, S, H, F, H, H, O], [AH1265; C, = CH-O _{-, - N =, CH 2} , S, Cl, F, H, H, O], [AH1266; C, = CH-O -, - N =, CH 2, S, Br, F, H, H, O], [AH1267; C, = CH-O -, - N =, CH 2, S, CF 3, F, H, H, O], [AH1268; C, = CH-O -, - N =, _{CH 2, S, Me, F} , H, H, O], [AH1269; C, = CH-O -, - N =, CH 2, S, Et, F, H, H, O], [AH1270; C , = CH-O -, - N =, CH 2, S, c-Pr, F, H, H, O], [AH1271; C, = CH-O -, - N =, CH 2, S, OMe , F, H, H, O ], [AH1272; C, = CH-O -, - N =, CH 2, S, H, H, F, H, O], [AH1273; C, = CH-O _{-, - N =, CH 2} , S, Cl, H, F, H, O], [AH1274; C, = CH-O -, - N =, CH 2, S, Br, H, F, H, O], [AH1275; C, = CH-O -, - N =, CH 2, S, CF 3, H, F, H, O], [AH1276; C, = CH-O -, - N =, _{CH 2, S, Me, H} , F, H, O], [AH1277; C, = CH-O -, - N =, CH 2, S, Et, H, F, H, O], [AH1278; C, = CH-O -, - N =, CH 2, S, c-Pr, H, F, H, O], [AH1279; C, = CH-O -, - N =, CH 2, S, OMe, H, F, H, O], [AH1280; C, = CH-O -, - N =, CH 2, S, H, H, H, F, O], [AH1281; C, = CH- O -, - N =, CH 2, S, Cl, H, H, F, O], [AH1282; C, = CH-O -, - N =, CH 2, S, Br, H, H, F , O], [AH1283; C , = CH-O -, - N =, CH 2, S, CF 3, H, H, F, O], [AH1284; C, = CH-O -, - N = _{, CH 2, S, Me,} H, H, F, O], [AH1285; C, = CH-O -, - N =, CH 2, S, Et, H, H, F, O], [AH1286 ; C, = CH-O - , - N =, CH 2, S, c-Pr, H, H, F, O], [AH1287; C, = CH-O -, - N =, CH 2, S , OMe, H, H, F, O], [AH 1 288; C, = CH-O-,-N =, CH ₂ , S, H, H, H, H, O], [AH 1 289; C, = CH -O -, - N =, CH 2, S, Cl, H, H, H, O], [AH1290; C, = CH-O -, - N =, CH 2, S, Br, H, H, H, O], [AH1291; C, = CH-O -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1292; C, = CH-O -, - N _{=, CH 2, S, Me} , H, H, H, O], [AH1293; C, = CH-O -, - N =, CH 2, S, Et, H, H, H, O], [ AH 1294; C, = CH-O -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1295; C, = CH-O -, - N =, CH 2, S, OMe, H, H, H, O] , [AH1296; C, = CH-O -, - CH =, CH 2, S, H, H, H, H, O], [AH1297; C, = CH-O- _{, -CH =, CH 2, S} , F, H, H, H, O], [AH1298; C, = CH-O -, - CH =, CH 2, S, Cl, H, H, H, O ], [AH1299; C, = CH-O -, - CH =, CH 2, S, Br, H, H, H, O], [AH1300; C, = CH-O -, - CH =, CH 2 , S, Me, H, H, H, O],

[AH1301; C, = CH- O -, - CH =, CH 2, S, Et, H, H, H, O], [AH1302; C, = CH-O -, - CH =, CH 2, S , Pr, H, H, H , O], [AH1303; C, = CH-O -, - CH =, CH 2, S, i-Pr, H, H, H, O], [AH1304; C, = CH-O -, - CH =, CH 2, S, c-Pr, H, H, H, O], [AH1305; C, = CH-O -, - CH =, CH 2, S, c- Bu, H, H, H, O], [AH1306; C, = CH-O -, - CH =, CH 2, S, OMe, H, H, H, O], [AH1307; C, = CH- O -, - CH =, CH 2, S, Oi-Pr, H, H, H, O], [AH1308; C, = CH-O -, - CH =, CH 2, S, SMe, H, H , H, O], [AH 1309; C, = CH-O-, -CH =, CH ₂ , S, Set, H, H, H, O], [AH 1310; C, = CH-O-,-CH _{=, CH 2, S, CF} 3, H, H, H, O], [AH1311; C, = CH-O -, - CH =, CH 2, S, CHF 2, H, H, H, O] , [AH1312; C, = CH -O -, - CH =, CH 2, S, OCF 3, H, H, H, O], [AH1313; C, = CH-O -, - CH =, CH 2 , S, OCHF ₂ , H, H, H, O], [AH 1314; C, = CH-O-, -CH =, CH ₂ , S, CH = CH ₂ , H, H, H, O], [[ AH1315; C, = CH-O -, - CH =, CH 2, S, C (Me) = CH 2, H, H, H, O], [AH1316; C, = CH-O -, - CH = _{, CH 2, S, CH =} CHMe, H, H, H, O], [AH1317; C, = CH-O -, - CH =, CH 2, S, C≡CH, H, H, H, O ], [AH1318; C, = CH-O -, - CH =, CH 2, S, C≡CMe, H, H, H, O], [AH1319; C, = C (CF 3) -O-, _{-CH =, CH 2, S,} H, H, H, H, O], [AH1320; C, = C (CF 3) -O -, - CH =, CH 2, S, Cl, H, H, H, O], [AH1321; C, = C (CF 3) -O -, - CH =, CH 2, S, Br, H, H, H, O], [AH1322; C, = C (CF 3 ) -O-, -CH =, CH ₂ , S, CF ₃ , H, H, H, O], [ AH1323; C, = C (CF 3) -O -, - CH =, CH 2, S, Me, H, H, H, O], [AH1324; C, = C ( _{CF 3) -O -, - CH} =, CH 2, S, Et, H, H, H, O], [AH1325; C, = C (CF 3) -O -, - CH =, CH 2, S , c-Pr, H, H , H, O], [AH1326; C, = C (CF 3) -O -, - CH =, CH 2, S, OMe, H, H, H, O], [ AH1327; C, = CF-O -, - CH =, CH 2, S, H, H, H, H, O], [AH1328; C, = CF-O -, - CH =, CH 2, S, Cl, H, H, H, O], [AH1329; C, = CF-O -, - CH =, CH 2, S, Br, H, H, H, O], [AH1330; C, = CF- O -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1331; C, = CF-O -, - CH =, CH 2, S, Me, H, H, H, O], [AH1332; C, = CF-O -, - CH =, CH 2, S, Et, H, H, H, O], [AH1333; C, = CF-O -, - CH = _{, CH 2, S, c-} Pr, H, H, H, O], [AH1334; C, = CF-O -, - CH =, CH 2, S, OMe, H, H, H, O], [AH1335; C, = CCl- O -, - CH =, CH 2, S, H, H, H, H, O], [AH1336; C, = CCl-O -, - CH =, CH 2, S , Cl, H, H, H , O], [AH1337; C, = CCl-O -, - CH =, CH 2, S, Br, H, H, H, O], [AH1338; C, = CCl -O -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1339; C, = CCl-O -, - CH =, CH 2, S, Me, H, H , H, O], [AH1340 ; C, = CCl-O -, - CH =, CH 2, S, Et, H, H, H, O], [AH1341; C, = CCl-O -, - CH _{=, CH 2, S, c} -Pr, H, H, H, O], [AH1342; C, = CCl-O -, - CH =, CH 2, S, OMe, H, H, H, O] , [AH1343; C, = C (Me) -O -, - CH =, CH 2, S, H, H, H, H, O], [AH1344; C, = C (Me) -O -, - _{CH =, CH 2, S,} Cl, H, H, H, O], [AH1345; C, = C (Me) -O- _{, -CH =, CH 2, S} , Br, H, H, H, O], [AH1346; C, = C (Me) -O -, - CH =, CH 2, S, CF 3, H, H , H, O], [AH1347 ; C, = C (Me) -O -, - CH =, CH 2, S, Me, H, H, H, O], [AH1348; C, = C (Me) -O -, - CH =, CH 2, S, Et, H, H, H, O], [AH1349; C, = C (Me) -O -, - CH =, CH 2, S, c-Pr , H, H, H, O ], [AH1350; C, = C (Me) -O -, - CH =, CH 2, S, OMe, H, H, H, O], [AH1351; C, = CH-O -, - CH = , CH 2, S, H, F, H, H, O], [AH1352; C, = CH-O -, - CH =, CH 2, S, Cl, F, H , H, O], [AH1353 ; C, = CH-O -, - CH =, CH 2, S, Br, F, H, H, O], [AH1354; C, = CH-O -, - CH _{=, CH 2, S, CF} 3, F, H, H, O], [AH1355; C, = CH-O -, - CH =, CH 2, S, Me, F, H, H, O], [AH1356; C, = CH- O -, - CH =, CH 2, S, Et, F, H, H, O], [AH1357; C, = CH-O -, - CH =, CH 2, S , c-Pr, F, H , H, O], [AH1358; C, = CH-O -, - CH =, CH 2, S, OMe, F, H, H, O], [AH1359; C, = CH-O -, - CH =, CH 2, S, H, H, F, H, O], [AH1360; C, = CH-O -, - CH =, CH 2, S, Cl, H, F, H, O], [ AH1361; C, = CH-O -, - CH =, CH 2, S, Br, H, F, H, O], [AH1362; C, = CH-O -, - _{CH =, CH 2, S,} CF 3, H, F, H, O], [AH1363; C, = CH-O -, - CH =, CH 2, S, Me, H, F, H, O] , [AH1364; C, = CH -O -, - CH =, CH 2, S, Et, H, F, H, O], [AH1365; C, = CH-O -, - CH =, CH 2, S, c-Pr, H, F, H, O], [AH1366; C, = CH-O -, - CH =, CH 2, S, OMe, H, F, H, O], [AH1367; C , = CH-O -, - CH =, CH 2, S, H, H, H, F, O], [AH1368; C, = CH-O -, - CH =, CH ₂ , S, Cl, H, H, F, O], [AH 1369; C, = CH-O-, -CH =, CH ₂ , S, Br, H, H, F, O], [[ AH1370; C, = CH-O -, - CH =, CH 2, S, CF 3, H, H, F, O], [AH1371; C, = CH-O -, - CH =, CH 2, S , Me, H, H, F , O], [AH1372; C, = CH-O -, - CH =, CH 2, S, Et, H, H, F, O], [AH1373; C, = CH -O -, - CH =, CH 2, S, c-Pr, H, H, F, O], [AH1374; C, = CH-O -, - CH =, CH 2, S, OMe, H, H, F, O], [ AH1375; C, = CH-O -, - CH =, CH 2, S, H, H, H, H, O], [AH1376; C, = CH-O -, - _{CH =, CH 2, S,} Cl, H, H, H, O], [AH1377; C, = CH-O -, - CH =, CH 2, S, Br, H, H, H, O], [AH1378; C, = CH- O -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1379; C, = CH-O -, - CH =, CH 2, S, Me, H, H, H, O], [AH 1 380; C, = CH-O-, -CH =, CH ₂ , S, Et, H, H, H, O], [AH 1381; C, = CH-O -, - CH = , CH 2, S, c-Pr, H, H, H, O], [AH1382; C, = CH-O -, - CH =, CH 2, S, OMe, H , H, H, O], [AH1383; C, = CH-CH =, - O-, CH 2, S, H, H, H, H, O], [AH1384; C, = CH-CH =, _{-O-, CH 2, S, F} , H, H, H, O], [AH1385; C, = CH-CH =, - O-, CH 2, S, Cl, H, H, H, O] , [AH1386; C, = CH -CH =, - O-, CH 2, S, Br, H, H, H, O], [AH1387; C, = CH-CH =, - O-, CH 2, S, Me, H, H, H, O], [AH 1388; C, = CH-CH =, -O-, CH ₂ , S, Et, H, H, H, O], [AH 1389; C, = CH-CH =, - O-, CH 2, S, Pr, H, H, H, O], [AH1390; C, = CH-CH =, - O-, CH 2, S, i-Pr, H , H, H, O], [AH1391; C, = CH-CH =, - O-, CH 2, S, c-Pr, H, H, H, O] , [AH1392; C, = CH -CH =, - O-, CH 2, S, c-Bu, H, H, H, O], [AH1393; C, = CH-CH =, - O-, CH _{2, S, OMe, H,} H, H, O], [AH1394; C, = CH-CH =, - O-, CH 2, S, Oi-Pr, H, H, H, O], [AH1395 ; C, = CH-CH = , - O-, CH 2, S, SMe, H, H, H, O], [AH1396; C, = CH-CH =, - O-, CH 2, S, Set , H, H, H, O ], [AH1397; C, = CH-CH =, - O-, CH 2, S, CF 3, H, H, H, O], [AH1398; C, = CH- _{CH =, - O-, CH 2} , S, CHF 2, H, H, H, O], [AH1399; C, = CH-CH =, - O-, CH 2, S, OCF 3, H, H , H, O], [AH1400 ; C, = CH-CH =, - O-, CH 2, S, OCHF 2, H, H, H, O],

[AH1401; C, = CH- CH =, - O-, CH 2, S, CH = CH 2, H, H, H, O], [AH1402; C, = CH-CH =, - O-, CH _{2, S, C (Me)} = CH 2, H, H, H, O], [AH1403; C, = CH-CH =, - O-, CH 2, S, CH = CHMe, H, H, H , O], [AH1404; C , = CH-CH =, - O-, CH 2, S, C≡CH, H, H, H, O], [AH1405; C, = CH-CH =, - O _{-, CH 2, S, C≡CMe} , H, H, H, O], [AH1406; C, = C (CF 3) -CH =, - O-, CH 2, S, H, H, H, H, O], [AH1407; C, = = C (CF 3) -CH, - O-, CH 2, S, Cl, H, H, H, O], [AH1408; C, = C (CF 3 ) -CH =, - O-, CH 2, S, Br, H, H, H, O], [AH1409; C, = C (CF 3) -CH =, - O-, CH 2, S, CF ₃ , H, H, H, O], [AH 1410; C, = C (CF ₃ ) -CH =, -O-, CH ₂ , S, Me, H, H, O], [AH 1411; C _{, = C (CF 3) -CH} =, - O-, CH 2, S, Et, H, H, H, O], [AH1412; C, = C (CF 3) -CH =, - O-, _{CH 2, S, c-Pr} , H, H, H, O], [AH1413; C, = C (CF 3) -CH =, - O-, CH 2, S, OMe, H, H, H, O], [AH1414; C, = CF-CH =, - O-, CH 2, S, H, H, H, H, O], [AH1415; C, = CF-CH =, - O-, CH ₂ , S, Cl, H, H, H, O, [AH 1416; C, = CF-CH =, -O-, CH ₂ , S, Br, H, H, O], [AH 1417; C , = CF-CH =, - O-, CH 2, S, CF 3, H, H, H, O], [AH1418; C, = CF-CH =, - O-, CH 2, S, Me, H, H, H, O] , [AH1419; C, = CF-CH =, - O-, CH 2, S, Et, H, H, H, O], [AH1420; C, = CF-CH = _{, -O-, CH 2, S,} c-Pr, H, H, H, O], [AH1421; C, = CF-CH =, - O-, CH 2, S, OMe, H, H, H , O], [AH1422; C , = CCl-CH =, - O-, CH 2, S, H, H, H, H, O], [AH1423; C, = CCl-CH =, - O-, CH 2, S, Cl, H, H, H, O], [AH1424; C, = CCl- _{CH =, - O-, CH 2} , S, Br, H, H, H, O], [AH1425; C, = CCl-CH =, - O-, CH 2, S, CF 3, H, H, H, O], [AH1426; C, = CCl-CH =, - O-, CH 2, S, Me, H, H, H, O], [AH1427; C, = CCl-CH =, - O- _{, CH 2, S, Et,} H, H, H, O], [AH1428; C, = CCl-CH =, - O-, CH 2, S, c-Pr, H, H, H, O], [AH1429; C, = CCl- CH =, - O-, CH 2, S, OMe, H, H, H, O], [AH1430; C, = C (Me) -CH =, - O-, CH _{2, S, H, H,} H, H, O], [AH1431; C, = C (Me) -CH =, - O-, CH 2, S, Cl, H, H, H, O], [ AH1432; C, = C (Me ) -CH =, - O-, CH 2, S, Br, H, H, H, O], [AH1433; C, = C (Me) -CH =, - O- _{, CH 2, S, CF 3} , H, H, H, O], [AH1434; C, = C (Me) -CH =, - O-, CH 2, S, Me, H, H, H, O ], [AH 1435; C, = C (Me) -CH =, -O-, CH ₂ , S, Et, H, H, H, O], [AH 1436; C, = C (Me) -CH =, _{-O-, CH 2, S, c} -Pr, H, H, H, O], [AH1437; C, = C (Me) -CH =, - O-, CH 2, S, OMe, H, H , H, O], [AH1438 ; C, = CH-CH =, - O-, CH 2, S, H, F, H, H, O], [AH1439; C, = CH-CH =, - O _{-, CH 2, S, Cl} , F, H, H, O], [AH1440; C, = CH-CH =, - O-, CH 2, S, Br, F, H, H, O], [ AH1441; C, = CH-CH =, - O-, CH 2, S, CF 3, F, H, H, O], [AH1442; C, = CH-CH =, - O-, CH 2, S , Me, F, H, H, O], [AH 1443; C, = CH-CH =, -O-, CH ₂ , S, Et, F, H, H, O], [AH 1444; C, = CH _{-CH =, - O-, CH 2} , S, c-Pr, F, H, H, O], [AH1445; C, = CH-CH =, - _{O-, CH 2, S, OMe} , F, H, H, O], [AH1446; C, = CH-CH =, - O-, CH 2, S, H, H, F, H, O], [AH1447; C, = CH- CH =, - O-, CH 2, S, Cl, H, F, H, O], [AH1448; C, = CH-CH =, - O-, CH 2, S , Br, H, F, H , O], [AH1449; C, = CH-CH =, - O-, CH 2, S, CF 3, H, F, H, O], [AH1450; C, = CH-CH =, - O-, CH 2, S, Me, H, F, H, O], [AH1451; C, = CH-CH =, - O-, CH 2, S, Et, H, F , H, O], [AH1452 ; C, = CH-CH =, - O-, CH 2, S, c-Pr, H, F, H, O], [AH1453; C, = CH-CH =, _{-O-, CH 2, S, OMe} , H, F, H, O], [AH1454; C, = CH-CH =, - O-, CH 2, S, H, H, H, F, O] , [AH1455; C, = CH -CH =, - O-, CH 2, S, Cl, H, H, F, O], [AH1456; C, = CH-CH =, - O-, CH 2, S, Br, H, H, F, O], [AH1457; C, = CH-CH =, - O-, CH 2, S, CF 3, H, H, F, O], [AH1458; C, = CH-CH =, - O- , CH 2, S, Me, H, H, F, O], [AH1459; C, = CH-CH =, - O-, CH 2, S, Et, H, H, F, O], [ AH1460; C, = CH-CH =, - O-, CH 2, S, c-Pr, H, H, F, O], [AH1461; C, = CH-CH = _{, -O-, CH 2, S,} OMe, H, H, F, O], [AH1462; C, = CH-CH =, - O-, CH 2, S, H, H, H, H, O ], [AH1463; C, = CH-CH =, - O-, CH 2, S, Cl, H, H, H, O], [AH1464; C, = CH-CH =, - O-, CH 2 , S, Br, H, H, H, O], [AH 1465; C, = CH-CH =, -O-, CH ₂ , S, CF ₃ , H, H, O], [AH 1466; C , = CH-CH =, - O-, CH 2, S, Me, H, H, H, O], [AH1467; C, = CH-CH =, - O-, CH 2, S, Et, H , H, H, O], [AH1468; C, = CH-CH =, - O-, CH 2, S, c-Pr, H, H, H , O], [AH1469; C , = CH-CH =, - O-, CH 2, S, OMe, H, H, H, O], [AH1470; C, = CH-CH =, - S-, _{CH 2, S, H, H} , H, H, O], [AH1471; C, = CH-CH =, - S-, CH 2, S, F, H, H, H, O], [AH1472; C, = CH-CH =, - S-, CH 2, S, Cl, H, H, H, O], [AH1473; C, = CH-CH =, - S-, CH 2, S, Br, H, H, H, O] , [AH1474; C, = CH-CH =, - S-, CH 2, S, Me, H, H, H, O], [AH1475; C, = CH-CH = _{, -S-, CH 2, S,} Et, H, H, H, O], [AH1476; C, = CH-CH =, - S-, CH 2, S, Pr, H, H, H, O ], [AH1477; C, = CH-CH =, - S-, CH 2, S, i-Pr, H, H, H, O], [AH1478; C, = CH-CH =, - S-, _{CH 2, S, c-Pr} , H, H, H, O], [AH1479; C, = CH-CH =, - S-, CH 2, S, c-Bu, H, H, H, O] , [AH1480; C, = CH -CH =, - S-, CH 2, S, OMe, H, H, H, O], [AH1481; C, = CH-CH =, - S-, CH 2, S, Oi-Pr, H, H, H, O], [AH1482; C, = CH-CH =, - S-, CH 2, S, SMe, H, H, H, O], [AH1483; C , = CH-CH =, - S-, CH 2, S, Set, H, H, H, O], [AH1484; C, = CH-CH =, - S-, CH 2, S, CF 3, H, H, H, O] , [AH1485; C, = CH-CH =, - S-, CH 2, S, CHF 2, H, H, H, O], [AH1486; C, = CH-CH =, -S-, CH ₂ , S, OCF ₃ , H, H, H, O], [AH 1487; C, = CH-CH =, -S-, CH ₂ , S, OCHF ₂ , H, H, H, O], [AH1488; C, = CH-CH =, - S-, CH 2, S, CH = CH 2, H, H, H, O], [AH1489; C, = CH-CH =, _{-S-, CH 2, S, C} (Me) = CH 2, H, H, H, O], [AH1490; C, = CH-CH =, - S-, CH 2, S, CH = CHMe, H, H, H, O], [AH1491; C, = CH-CH =, -S-, CH _{2, S, C≡CH, H,} H, H, O], [AH1492; C, = CH-CH =, - S-, CH 2, S, C≡CMe, H, H, H, O], [AH1493; C, = C ( CF 3) -CH =, - S-, CH 2, S, H, H, H, H, O], [AH1494; C, = C (CF 3) -CH =, _{-S-, CH 2, S, Cl} , H, H, H, O], [AH1495; C, = C (CF 3) -CH =, - S-, CH 2, S, Br, H, H, H, O], [AH1496; C, = C (CF 3) -CH =, - S-, CH 2, S, CF 3, H, H, H, O], [AH1497; C, = C (CF _{3) -CH =, - S-,} CH 2, S, Me, H, H, H, O], [AH1498; C, = C (CF 3) -CH =, - S-, CH 2, S, Et, H, H, H, O], [AH1499; C, = C (CF 3) -CH =, - S-, CH 2, S, c-Pr, H, H, H, O], [AH1500 _{; C, = C (CF 3} ) -CH =, - S-, CH 2, S, OMe, H, H, H, O],

[AH1501; C, = CF- CH =, - S-, CH 2, S, H, H, H, H, O], [AH1502; C, = CF-CH =, - S-, CH 2, S , Cl, H, H, H, O], [AH 1503; C, = CF-CH =, -S-, CH ₂ , S, Br, H, H, O, [AH 1504; C, = CF _{-CH =, - S-, CH 2} , S, CF 3, H, H, H, O], [AH1505; C, = CF-CH =, - S-, CH 2, S, Me, H, H , H, O], [AH1506 ; C, = CF-CH =, - S-, CH 2, S, Et, H, H, H, O], [AH1507; C, = CF-CH =, - S _{-, CH 2, S, c} -Pr, H, H, H, O], [AH1508; C, = CF-CH =, - S-, CH 2, S, OMe, H, H, H, O] , [AH1509; C, = CCl -CH =, - S-, CH 2, S, H, H, H, H, O], [AH1510; C, = CCl-CH =, - S-, CH 2, S, Cl, H, H, H, O], [AH1511; C, = CCl-CH =, - S-, CH 2, S, Br, H, H, H, O], [AH1512; C, = CCl-CH =, - S-, CH 2, S, CF 3, H, H, H, O], [AH1513; C, = CCl-CH =, - S-, CH 2, S, Me, H, H, H, O], [ AH1514; C, = CCl-CH =, - S-, CH 2, S, Et, H, H, H, O], [AH1515; C, = CCl-CH =, - _{S-, CH 2, S, c} -Pr, H, H, H, O], [AH1516; C, = CCl-CH =, - S-, CH 2, S, OMe, H, H, H, O ], [AH1517; C, = C (Me) -CH =, - S-, CH 2, S, H, H, H, H, O], [AH1518; C, = C (Me) -CH =, _{-S-, CH 2, S, Cl} , H, H, H, O], [AH1519; C, = C (Me) -CH =, - S-, CH 2, S, Br, H, H, H , O], [AH 1520; C, = C (Me) -CH =, -S-, CH ₂ , S, CF ₃ , H, H, H, O], [AH 1521; C, = C (Me)- _{CH =, - S-, CH 2} , S, Me, H, H, H, O], [AH1522; C, = C (Me) -CH =, - S-, CH 2, S, Et, H, H, H, O], [ AH1523; C, = C (Me) -CH =, - S-, CH 2, S, c-Pr, H, H, H, O] , [AH1524; C, = C (Me) -CH =, - S-, CH 2, S, OMe, H, H, H, O], [AH1525; C, = CH _{-CH =, - S-, CH 2} , S, H, F, H, H, O], [AH1526; C, = CH-CH =, - S-, CH 2, S, Cl, F, H, H, O], [AH1527; C, = CH-CH =, - S-, CH 2, S, Br, F, H, H, O], [AH1528; C, = CH-CH =, - S- _{, CH 2, S, CF 3} , F, H, H, O], [AH1529; C, = CH-CH =, - S-, CH 2, S, Me, F, H, H, O], [ AH1530; C, = CH-CH =, - S-, CH 2, S, Et, F, H, H, O], [AH1531; C, = CH-CH =, - S-, CH 2, S, c-Pr, F, H, H, O], [AH1532; C, = CH-CH =, - S-, CH 2, S, OMe, F, H, H, O], [AH1533; C, = CH-CH =, - S-, CH 2, S, H, H, F, H, O], [AH1534; C, = CH-CH =, - S-, CH 2, S, Cl, H, F , H, O], [AH1535 ; C, = CH-CH =, - S-, CH 2, S, Br, H, F, H, O], [AH1536; C, = CH-CH =, - S _{-, CH 2, S, CF} 3, H, F, H, O], [AH1537; C, = CH-CH =, - S-, CH 2, S, Me, H, F, H, O], [AH1538; C, = CH- CH =, - S-, CH 2, S, Et, H, F, H, O], [AH1539; C, = CH-CH =, - S-, CH 2, S , c-Pr, H, F , H, O], [AH1540; C, = CH-CH =, - S-, CH 2, S, OMe, H, F, H, O], [AH1541; C, = CH-CH =, - S- , CH 2, S, H, H, H, F, O], [AH1542; C, = CH-CH =, - S-, CH 2, S, Cl, H, H, F, O], [ AH1543; C, = CH-CH =, - S-, CH 2, S, Br, H, H, F, O], [AH1544; C, = CH-CH =, - _{S-, CH 2, S, CF} 3, H, H, F, O], [AH1545; C, = CH-CH =, - S-, CH 2, S, Me, H, H, F, O] , [AH1546; C, = CH -CH =, - S-, CH 2, S, Et, H, H, F, O], [AH1547; C , = CH-CH =, - S-, CH 2, S, c-Pr, H, H, F, O], [AH1548; C, = CH-CH =, - S-, CH 2, S, OMe , H, H, F, O], [AH 1 549; C, = CH-CH =, -S-, CH ₂ , S, H, H, H, H, O], [AH 1550; C, = CH-CH _{=, - S-, CH 2,} S, Cl, H, H, H, O], [AH1551; C, = CH-CH =, - S-, CH 2, S, Br, H, H, H, O], [AH1552; C, = CH-CH =, - S-, CH 2, S, CF 3, H, H, H, O], [AH1553; C, = CH-CH =, - S-, _{CH 2, S, Me, H} , H, H, O], [AH1554; C, = CH-CH =, - S-, CH 2, S, Et, H, H, H, O], [AH1555; C, = CH-CH =, - S-, CH 2, S, c-Pr, H, H, H, O], [AH1556; C, = CH-CH =, - S-, CH 2, S, OMe, H, H, H, O], [AH1557; C, = CH-S -, - CH =, CH 2, S, H, H, H, H, O], [AH1558; C, = CH- S -, - CH =, CH 2, S, F, H, H, H, O], [AH1559; C, = CH-S -, - CH =, CH 2, S, Cl, H, H, H , O], [AH1560; C , = CH-S -, - CH =, CH 2, S, Br, H, H, H, O], [AH1561; C, = CH-S -, - CH =, _{CH 2, S, Me, H} , H, H, O], [AH1562; C, = CH-S -, - CH =, CH 2, S, Et, H, H, H, O], [AH1563; C, = CH-S -, - CH =, CH 2, S, Pr, H, H, H, O], [AH1564; C, = CH-S -, - CH =, CH 2, S, i- Pr, H, H, H, O], [AH1565; C, = CH-S -, - CH =, CH 2, S, c-Pr, H, H, H, O], [AH1566; C, = CH-S -, - CH = , CH 2, S, c-Bu, H, H, H, O], [AH1567; C, = CH-S -, - CH =, CH 2, S, OMe, H , H, H, O], [AH1568; C, = CH-S -, - CH =, CH 2, S, Oi-Pr, H, H, H, O], [AH1569; C, = CH-S _{-, - CH =, CH 2} , S, SMe, H, H, H, O], [AH1570; C, = CH-S -, - CH =, CH 2 , S, Set, H, H, H, O], [AH 1571; C, = CH-S-, -CH =, CH ₂ , S, CF ₃ , H, H, O], [AH 1572; C , = CH-S -, - CH =, CH 2, S, CHF 2, H, H, H, O], [AH1573; C, = CH-S -, - CH =, CH 2, S, OCF 3 , H, H, H, O ], [AH1574; C, = CH-S -, - CH =, CH 2, S, OCHF 2, H, H, H, O], [AH1575; C, = CH- S -, - CH =, CH 2, S, CH = CH 2, H, H, H, O], [AH1576; C, = CH-S -, - CH =, CH 2, S, C (Me) _{= CH 2, H, H,} H, O], [AH1577; C, = CH-S -, - CH =, CH 2, S, CH = CHMe, H, H, H, O], [AH1578; C , = CH-S -, - CH =, CH 2, S, C≡CH, H, H, H, O], [AH1579; C, = CH-S -, - CH =, CH 2, S, C ≡CMe, H, H, H, O], [AH 1580; C, = C (CF ₃ ) -S-, -CH =, CH ₂ , S, H, H, H, H, O], [AH 1581; _{C, = C (CF 3)} -S -, - CH =, CH 2, S, Cl, H, H, H, O], [AH1582; C, = C (CF 3) -S -, - CH = _{, CH 2, S, Br,} H, H, H, O], [AH1583; C, = C (CF 3) -S -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1584; C, = C (CF 3) -S -, - CH =, CH 2, S, Me, H, H, H, O], [AH1585; C, = C (CF 3) - S -, - CH =, CH 2, S, Et, H, H, H, O], [AH1586; C, = C (CF 3) -S -, - CH =, CH 2, S, c-Pr , H, H, H, O ], [AH1587; C, = C (CF 3) -S -, - CH =, CH 2, S, OMe, H, H, H, O], [AH1588; C, = CF-S -, - CH =, CH 2, S, H, H, H, H, O], [AH1589; C, = CF-S -, - CH =, CH 2, S, Cl, H, H, H, O], [ AH1590; C, = CF-S -, - CH =, CH 2, S, Br, H, H, H, O], [AH1591; C, = CF-S -, - CH =, CH ₂ , S, CF ₃ , H, H, H, O], [ AH1592; C, = CF-S -, - CH =, CH 2, S, Me, H, H, H, O], [AH1593; C, = CF-S -, - CH =, CH 2, S, Et, H, H, H, O], [AH1594; C, = CF-S -, - CH =, CH 2, S, c-Pr, H, H, H, O], [AH1595; C, = CF-S -, - CH = , CH 2, S, OMe, H, H, H, O], [AH1596; C, = CCl-S -, - CH =, CH 2, S, H, H, H , H, O], [AH1597 ; C, = CCl-S -, - CH =, CH 2, S, Cl, H, H, H, O], [AH1598; C, = CCl-S -, - CH _{=, CH 2, S, Br} , H, H, H, O], [AH1599; C, = CCl-S -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1600; C, = CCl- S -, - CH =, CH 2, S, Me, H, H, H, O],

[AH1601; C, = CCl- S -, - CH =, CH 2, S, Et, H, H, H, O], [AH1602; C, = CCl-S -, - CH =, CH 2, S , c-Pr, H, H , H, O], [AH1603; C, = CCl-S -, - CH =, CH 2, S, OMe, H, H, H, O], [AH1604; C, = C (Me) -S -, - CH =, CH 2, S, H, H, H, H, O], [AH1605; C, = C (Me) -S -, - CH =, CH 2, S, Cl, H, H, H, O], [AH1606; C, = C (Me) -S -, - CH =, CH 2, S, Br, H, H, H, O], [AH1607; C, = C (Me) -S -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1608; C, = C (Me) -S -, - CH =, _{CH 2, S, Me, H} , H, H, O], [AH1609; C, = C (Me) -S -, - CH =, CH 2, S, Et, H, H, H, O], [AH 1610; C, = C (Me)-S-, -CH =, CH ₂ , S, c-Pr, H, H, H, O], [AH 1611; C, = C (Me)-S-, _{-CH =, CH 2, S,} OMe, H, H, H, O], [AH1612; C, = CH-S -, - CH =, CH 2, S, H, F, H, H, O] , [AH1613; C, = CH -S -, - CH =, CH 2, S, Cl, F, H, H, O], [AH1614; C, = CH-S -, - CH =, CH 2, S, Br, F, H, H, O], [AH1615; C, = CH-S -, - CH =, CH 2, S, CF 3, F, H, H, O], [AH1616; C, = CH-S -, - CH =, CH 2, S, Me, F, H, H, O], [AH1617; C, = CH-S -, - CH =, CH 2, S, Et, F, H, H, O], [ AH1618; C, = CH-S -, - CH =, CH 2, S, c-Pr, F, H, H, O], [AH1619; C, = CH-S- _{, -CH =, CH 2, S} , OMe, F, H, H, O], [AH1620; C, = CH-S -, - CH =, CH 2, S, H, H, F, H, O ], [AH1621; C, = CH-S -, - CH =, CH 2, S, Cl, H, F, H, O], [AH1622; C, = CH-S -, - CH =, CH 2 , S, Br, H, F , H, O], [AH1623; C, = CH-S -, - CH =, CH 2, S, CF 3, H , F, H, O], [AH1624; C, = CH-S -, - CH =, CH 2, S, Me, H, F, H, O], [AH1625; C, = CH-S-, _{-CH =, CH 2, S,} Et, H, F, H, O], [AH1626; C, = CH-S -, - CH =, CH 2, S, c-Pr, H, F, H, O], [AH1627; C, = CH-S -, - CH =, CH 2, S, OMe, H, F, H, O], [AH1628; C, = CH-S -, - CH =, CH ₂ , S, H, H, H, F, O], [AH 1629; C, = CH-S-, -CH =, CH ₂ , S, Cl, H, H, F, O], [AH 1630; C , = CH-S -, - CH =, CH 2, S, Br, H, H, F, O], [AH1631; C, = CH-S -, - CH =, CH 2, S, CF 3, H, H, F, O] , [AH1632; C, = CH-S -, - CH =, CH 2, S, Me, H, H, F, O], [AH1633; C, = CH-S- _{, -CH =, CH 2, S} , Et, H, H, F, O], [AH1634; C, = CH-S -, - CH =, CH 2, S, c-Pr, H, H, F , O], [AH1635; C , = CH-S -, - CH =, CH 2, S, OMe, H, H, F, O], [AH1636; C, = CH-S -, - CH =, _{CH 2, S, H, H} , H, H, O], [AH1637; C, = CH-S -, - CH =, CH 2, S, Cl, H, H, H, O], [AH1638; C, = CH-S -, - CH =, CH 2, S, Br, H, H, H, O], [AH1639; C, = CH-S -, - CH =, CH 2, S, CF 3 , H, H, H, O ], [AH1640; C, = CH-S -, - CH =, CH 2, S, Me, H, H, H, O], [AH1641; C, = CH-S _{-, - CH =, CH 2} , S, Et, H, H, H, O], [AH1642; C, = CH-S -, - CH =, CH 2, S, c-Pr, H, H, H, O], [AH1643; C, = CH-S -, - CH =, CH 2, S, OMe, H, H, H, O], [AH1644; C, -CH = CH -, = CH- _{N =, CH 2, S,} H, H, H, H, O], [AH1645; C, -CH = CH -, = CH-N =, CH 2, S, Cl, H, H, H, O ], [AH 1646; C, -CH = CH-, = CH-N =, CH ₂ , S, Br, H, H, H, O], [AH 16 47; C, -CH = CH - , = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1648; C, -CH = CH -, = CH-N =, _{CH 2, S, Me, H} , H, H, O], [AH1649; C, -CH = CH -, = CH-N =, CH 2, S, Et, H, H, H, O], [ AH1650; C, -CH = CH - , = CH-N =, CH 2, S, c-Pr, H, H, H, O], [AH1651; C, -CH = CH -, = CH-N = _{, CH 2, S, OMe,} H, H, H, O], [AH1652; C, -CH = CF -, = CH-N =, CH 2, S, H, H, H, H, O], [AH1653; C, -CH = CF -, = CH-N =, CH 2, S, Cl, H, H, H, O], [AH1654; C, -CH = CF -, = CH-N =, _{CH 2, S, Br, H} , H, H, O], [AH1655; C, -CH = CF -, = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1656; C, -CH = CF -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1657; C, -CH = CF -, = CH-N =, _{CH 2, S, Et, H} , H, H, O], [AH1658; C, -CH = CF -, = CH-N =, CH 2, S, c-Pr, H, H, H, O] , [AH1659; C, -CH = CF -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1660; C, -CF = CH -, = CH-N = _{, CH 2, S, H,} H, H, H, O], [AH1661; C, -CF = CH -, = CH-N =, CH 2, S, Cl, H, H, H, O], [AH1662; C, -CF = CH -, = CH-N =, CH 2, S, Br, H, H, H, O], [AH1663; C, -CF = CH -, = CH-N =, _{CH 2, S, CF 3,} H, H, H, O], [AH1664; C, -CF = CH -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1665; C, -CF = CH -, = CH-N =, CH 2, S, Et, H, H, H, O], [AH1666; C, -CF = CH -, = CH-N =, _{CH 2, S, c-Pr} , H, H, H, O], [AH1667; C, -CF = CH -, = CH-N =, CH 2, S, OMe, H, H, H, O] , [AH1668; C, -CH = CH -, = CF-N =, CH 2, S, H, H, H, H, O], [AH1669; C, -CH = CH -, = CF-N =, CH 2, S, Cl, H, H, H, O], [AH1670; C, -CH = CH -, = CF-N =, _{CH 2, S, Br, H} , H, H, O], [AH1671; C, -CH = CH -, = CF-N =, CH 2, S, CF 3, H, H, H, O], [AH1672; C, -CH = CH -, = CF-N =, CH 2, S, Me, H, H, H, O], [AH1673; C, -CH = CH -, = CF-N =, _{CH 2, S, Et, H} , H, H, O], [AH1674; C, -CH = CH -, = CF-N =, CH 2, S, c-Pr, H, H, H, O] , [AH1675; C, -CH = CH -, = CF-N =, CH 2, S, OMe, H, H, H, O], [AH1676; C, -CH = CCl -, = CH-N = _{, CH 2, S, H,} H, H, H, O], [AH1677; C, -CH = CCl -, = CH-N =, CH 2, S, Cl, H, H, H, O], [AH1678; C, -CH = CCl -, = CH-N =, CH 2, S, Br, H, H, H, O], [AH1679; C, -CH = CCl -, = CH-N =, _{CH 2, S, CF 3,} H, H, H, O], [AH1680; C, -CH = CCl -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1681; C, -CH = CCl -, = CH-N =, CH 2, S, Et, H, H, H, O], [AH1682; C, -CH = CCl -, = CH-N =, _{CH 2, S, c-Pr} , H, H, H, O], [AH1683; C, -CH = CCl -, = CH-N =, CH 2, S, OMe, H, H, H, O] , [AH1684; C, -CCl = CH -, = CH-N =, CH 2, S, H, H, H, H, O], [AH1685; C, -CCl = CH -, = CH-N = _{, CH 2, S, Cl,} H, H, H, O], [AH1686; C, -CCl = CH -, = CH-N =, CH 2, S, Br, H, H, H, O], [AH1687; C, -CCl = CH -, = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1688; C, -CCl = CH -, = CH-N = _{, CH 2, S, Me,} H, H, H, O], [AH1689; C, -CCl = CH -, = CH-N =, CH 2, S, Et, H, H, H, O], [AH 1690; C, -CCl = CH-, = CH-N =, CH _{2, S, c-Pr,} H, H, H, O], [AH1691; C, -CCl = CH -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1692; C, -CH = CH -, = CCl-N =, CH 2, S, H, H, H, H, O], [AH1693; C, -CH = CH -, = CCl-N =, _{CH 2, S, Cl, H} , H, H, O], [AH1694; C, -CH = CH -, = CCl-N =, CH 2, S, Br, H, H, H, O], [ AH1695; C, -CH = CH - , = CCl-N =, CH 2, S, CF 3, H, H, H, O], [AH1696; C, -CH = CH -, = CCl-N =, _{CH 2, S, Me, H} , H, H, O], [AH1697; C, -CH = CH -, = CCl-N =, CH 2, S, Et, H, H, H, O], [ AH1698; C, -CH = CH - , = CCl-N =, CH 2, S, c-Pr, H, H, H, O], [AH1699; C, -CH = CH -, = CCl-N = _{, CH 2, S, OMe,} H, H, H, O], [AH1700; C, -CH = C (Me) -, = CH-N =, CH 2, S, H, H, H, H, O],

[AH1701; C, -CH = C (Me) -, = = CH-N, CH 2, S, Cl, H, H, H, O], [AH1702; C, -CH = C (Me) -, _{= CH-N =, CH 2} , S, Br, H, H, H, O], [AH1703; C, -CH = C (Me) -, = CH-N =, CH 2, S, CF 3, H, H, H, O] , [AH1704; C, -CH = C (Me) -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1705; C, -CH = C (Me) -, = CH-N =, CH 2, S, Et, H, H, H, O], [AH1706; C, -CH = C (Me) -, = CH-N = _{, CH 2, S, c-} Pr, H, H, H, O], [AH1707; C, -CH = C (Me) -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1708; C, -C (Me) = CH -, = CH-N =, CH 2, S, H, H, H, H, O], [AH1709; C, -C (Me ) = CH-, = CH-N =, CH ₂ , S, Cl, H, H, H, O], [AH 1710; C,-C (Me) = CH-, = CH-N =, CH ₂ , S, Br, H, H, H, O], [AH1711; C, -C (Me) = CH -, = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1712; C, -C (Me ) = CH -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1713; C, -C (Me) = CH-, _{= CH-N =, CH 2} , S, Et, H, H, H, O], [AH1714; C, -C (Me) = CH -, = CH-N =, CH 2, S, c-Pr , H, H, H, O ], [AH1715; C, -C (Me) = CH -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1716; C , -CH = CH -, = C (Me) -N =, CH 2, S, H, H, H, H, O], [AH1717; C, -CH = CH -, = C (Me) -N _{=, CH 2, S, Cl} , H, H, H, O], [AH1718; C, -CH = CH -, = C (Me) -N =, CH 2, S, Br, H, H, H , O], [AH1719; C , -CH = CH -, = C (Me) -N =, CH 2, S, CF 3, H, H, H, O], [AH1720; C, -CH = CH -, = C (Me) -N =, CH 2, S, Me, H, H, H, O], [AH1721; C, -CH = CH -, = C (Me) -N = _{, CH 2, S, Et,} H, H, H, O], [AH1722; C, -CH = CH -, = C (Me) -N =, CH 2, S, c-Pr, H, H, H, O], [AH1723; C, -CH = CH -, = C (Me) -N =, CH 2, S, OMe, H, H, H, O], [AH1724; C, -CH = C _{(CF 3) -, = CH} -N =, CH 2, S, H, H, H, H, O], [AH1725; C, -CH = C (CF 3) -, = CH-N =, CH _{2, S, Cl, H,} H, H, O], [AH1726; C, -CH = C (CF 3) -, = CH-N =, CH 2, S, Br, H, H, H, O ], [AH1727; C, -CH = C (CF 3) -, = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1728; C, -CH = C ( _{CF 3) -, = CH-} N =, CH 2, S, Me, H, H, H, O], [AH1729; C, -CH = C (CF 3) -, = CH-N =, CH 2 , S, Et, H, H , H, O], [AH1730; C, -CH = C (CF 3) -, = CH-N =, CH 2, S, c-Pr, H, H, H, O], [AH1731; C, -CH = C (CF 3) -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1732; C, -C (CF 3 ) = CH-, = CH-N =, CH ₂ , S, H, H, H, H, O], [AH 1733; C,-C (CF ₃ ) = CH-, = CH-N =, CH ₂ , S, Cl, H, H, H, O], [AH 1734; C, -C (CF ₃ ) = CH-, = CH-N =, CH ₂ , S, Br, H, H, H, O] , [AH1735; C, -C ( CF 3) = CH -, = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1736; C, -C (CF 3) = CH -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1737; C, -C (CF 3) = CH -, = CH-N =, CH 2, S, Et, H, H, H, O], [AH1738; C, -C (CF 3) = CH -, = CH-N =, CH 2, S, c-Pr, H, H, H, O ], [AH1739; C, -C (CF 3) = CH -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1740; C, -CH = CH-, _{= C (CF 3) -N =} , CH 2, S, H, H, H, H, O], [AH1 741; C, -CH = CH - , = C (CF 3) -N =, CH 2, S, Cl, H, H, H, O], [AH1742; C, -CH = CH -, = C ( _{CF 3) -N =, CH 2} , S, Br, H, H, H, O], [AH1743; C, -CH = CH -, = C (CF 3) -N =, CH 2, S, CF ₃ , H, H, H, O], [AH 1 744; C, -CH = CH-, = C (CF ₃ ) -N =, CH ₂ , S, Me, H, H, H, O], [AH 1 745 ; C, -CH = CH -, = C (CF 3) -N =, CH 2, S, Et, H, H, H, O], [AH1746; C, -CH = CH -, = C (CF _{3) -N =, CH 2,} S, c-Pr, H, H, H, O], [AH1747; C, -CH = CH -, = C (CF 3) -N =, CH 2, S, OMe, H, H, H, O], [AH1748; C, = CH-CH = CH -, - C (Me) =, CH 2, S, H, H, H, H, O], [AH1749; C, = CH-CH = CH -, - C (Me) =, CH 2, S, Cl, H, H, H, O], [AH1750; C, = CH-CH = CH -, - C (Me _{) =, CH 2, S,} Br, H, H, H, O], [AH1751; C, = CH-CH = CH -, - C (Me) =, CH 2, S, CF 3, H, H , H, O], [AH1752 ; C, = CH-CH = CH -, - C (Me) =, CH 2, S, Me, H, H, H, O], [AH1753; C, = CH- CH = CH -, - C ( Me) =, CH 2, S, Et, H, H, H, O], [AH1754; C, = CH-CH = CH -, - C (Me) =, CH 2 , S, c-Pr, H , H, H, O], [AH1755; C, = CH-CH = CH -, - C (Me) =, CH 2, S, OMe, H, H, H, O ], [AH1756; C, = CH-CH = CF -, - C (Me) =, CH 2, S, H, H, H, H, O], [AH1757; C, = CH-CH = CF- , -C (Me) =, CH 2, S, Cl, H, H, H, O], [AH1758; C, = CH-CH = CF -, - C (Me) =, CH 2, S, Br , H, H, H, O ], [AH1759; C, = CH-CH = CF -, - C (Me) =, CH 2, S, CF 3, H, H, H, O], [AH1760; C, = CH-CH = CF -, - C (Me) =, CH 2, S, Me, H, H, H, O], [AH1761; C, = CH-CH = CF -, - C (Me) =, CH 2, S, Et, H, H, H, O], [AH1762; C, = CH-CH = CF -, - C (Me) = , CH 2, S, c-Pr, H, H, H, O], [AH1763; C, = CH-CH = CF -, - C (Me) =, CH 2, S, OMe, H, H, H, O], [AH 1764; C, = CH-CF = CH-, -C (Me) =, CH ₂ , S, H, H, H, H, O], [[ AH1765; C, = CH-CF = CH -, - C (Me) =, CH 2, S, Cl, H, H, H, O], [AH1766; C, = CH-CF = CH -, - C _{(Me) =, CH 2,} S, Br, H, H, H, O], [AH1767; C, = CH-CF = CH -, - C (Me) =, CH 2, S, CF 3, H , H, H, O], [AH1768; C, = CH-CF = CH -, - C (Me) =, CH 2, S, Me, H, H, H, O], [AH1769; C, = CH-CF = CH -, - C (Me) =, CH 2, S, Et, H, H, H, O], [AH1770; C, = CH-CF = CH -, - C (Me) =, _{CH 2, S, c-Pr} , H, H, H, O], [AH1771; C, = CH-CF = CH -, - C (Me) =, CH 2, S, OMe, H, H, H , O], [AH1772; C , = CF-CH = CH -, - C (Me) =, CH 2, S, H, H, H, H, O], [AH1773; C, = CF-CH = CH -, - C (Me) =, CH 2, S, Cl, H, H, H, O], [AH1774; C, = CF-CH = CH -, - C (Me) =, CH 2, S , Br, H, H, H, O], [AH 1 775; C, = CF-CH = CH-, -C (Me) =, CH ₂ , S, CF ₃ , H, H, H, O], [[ AH1776; C, = CF-CH = CH -, - C (Me) =, CH 2, S, Me, H, H, H, O], [AH1777; C, = CF-CH = CH -, - C _{(Me) =, CH 2,} S, Et, H, H, H, O], [AH1778; C, = CF-CH = CH -, - C (Me) =, CH 2, S, c-Pr, H, H, H, O] , [AH1779; C, = CF-CH = CH -, - C (Me) =, CH 2, S, OMe, H, H, H, O], [AH1780; C, = CH-CH = CH -, - C (Br) =, CH 2, S, H, H, H, H, O], [AH17 81; C, = CH-CH = CH -, - C (Br) =, CH 2, S, Cl, H, H, H, O], [AH1782; C, = CH-CH = CH -, - C _{(Br) =, CH 2,} S, Br, H, H, H, O], [AH1783; C, = CH-CH = CH -, - C (Br) =, CH 2, S, CF 3, H , H, H, O], [AH 1784; C, = CH-CH = CH-, -C (Br) =, CH ₂ , S, Me, H, H, H, O], [AH 1 785; C, = CH-CH = CH -, - C (Br) =, CH 2, S, Et, H, H, H, O], [AH1786; C, = CH-CH = CH -, - C (Br) =, _{CH 2, S, c-Pr} , H, H, H, O], [AH1787; C, = CH-CH = CH -, - C (Br) =, CH 2, S, OMe, H, H, H , O], [AH1788; C , = CH-CH = CH -, - C (Cl) =, CH 2, S, H, H, H, H, O], [AH1789; C, = CH-CH = CH -, - C (Cl) =, CH 2, S, Cl, H, H, H, O], [AH1790; C, = CH-CH = CH -, - C (Cl) =, CH 2, S , Br, H, H, H , O], [AH1791; C, = CH-CH = CH -, - C (Cl) =, CH 2, S, CF 3, H, H, H, O], [ AH1792; C, = CH-CH = CH -, - C (Cl) =, CH 2, S, Me, H, H, H, O], [AH1793; C, = CH-CH = CH -, - C _{(Cl) =, CH 2,} S, Et, H, H, H, O], [AH1794; C, = CH-CH = CH -, - C (Cl) =, CH 2, S, c-Pr, H, H, H, O] , [AH1795; C, = CH-CH = CH -, - C (Cl) =, CH 2, S, OMe, H, H, H, O], [AH1796; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, S, H, H, H, H, O], [AH1797; C, = CH-C (Me) = CH-, _{-C (Me) =, CH 2} , S, Cl, H, H, H, O], [AH1798; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, S , Br, H, H, H , O], [AH1799; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, S, CF 3, H, H, H, O ], [AH1800; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, S, Me, H, H, H, O],

[AH1801; C, = CH- C (Me) = CH -, - C (Me) =, CH 2, S, Et, H, H, H, O], [AH1802; C, = CH-C (Me ) = CH -, - C ( Me) =, CH 2, S, c-Pr, H, H, H, O], [AH1803; C, = CH-C (Me) = CH -, - C (Me _{) =, CH 2, S,} OMe, H, H, H, O], [AH1804; C, = CH-CH = CH -, - C (CF 3) =, CH 2, S, H, H, H , H, O], [AH1805 ; C, = CH-CH = CH -, - C (CF 3) =, CH 2, S, Cl, H, H, H, O], [AH1806; C, = CH -CH = CH -, - C ( CF 3) =, CH 2, S, Br, H, H, H, O], [AH1807; C, = CH-CH = CH -, - C (CF 3) = _{, CH 2, S, CF 3} , H, H, H, O], [AH1808; C, = CH-CH = CH -, - C (CF 3) =, CH 2, S, Me, H, H, H, O], [AH 1809; C, = CH-CH = CH-, -C (CF ₃ ) =, CH ₂ , S, Et, H, H, H, O], [AH 1810; C, = CH- CH = CH -, - C ( CF 3) =, CH 2, S, c-Pr, H, H, H, O], [AH1811; C, = CH-CH = CH -, - C (CF 3) _{=, CH 2, S, OMe} , H, H, H, O], [AH1812; C, -CH = CH -, = CH-N =, CH 2, S, H, H, H, H, O] , [AH1813; C, -CH = CH -, = CH-N =, CH 2, S, Cl, H, H, H, O], [AH1814; C, -CH = CH -, = CH-N = _{, CH 2, S, Br,} H, H, H, O], [AH1815; C, -CH = CH -, = CH-N =, CH 2, S, CF 3, H, H, H, O] , [AH1816; C, -CH = CH -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1817; C, -CH = CH -, = CH-N = _{, CH 2, S, Et,} H, H, H, O], [AH1818; C, -CH = CH -, = CH-N =, CH 2, S, c-Pr, H, H, H, O ], [AH1819; C, -CH = CH -, = CH-N =, CH 2, S, OMe, H, H, H, O], [AH1820; C, -CH = CF -, = CH-N =, CH ₂ , S, H, H, H, H, O], [AH 1821; C,- CH = CF -, = CH- N =, CH 2, S, Cl, H, H, H, O], [AH1822; C, -CH = CF -, = CH-N =, CH 2, S, Br , H, H, H, O ], [AH1823; C, -CH = CF -, = CH-N =, CH 2, S, CF 3, H, H, H, O], [AH1824; C, - CH = CF -, = CH- N =, CH 2, S, Me, H, H, H, O], [AH1825; C, -CH = CF -, = CH-N =, CH 2, S, Et , H, H, H, O ], [AH1826; C, -CH = CF -, = CH-N =, CH 2, S, c-Pr, H, H, H, O], [AH1827; C, -CF = CH -, = CH- N =, CH 2, S, H, H, H, H, O], [AH1828; C, -CF = CH -, = CH-N =, CH 2, S, Cl, H, H, H, O], [AH1829; C, -CF = CH -, = CH-N =, CH 2, S, Br, H, H, H, O], [AH1830; C, - CF = CH -, = CH- N =, CH 2, S, CF 3, H, H, H, O], [AH1831; C, -CF = CH -, = CH-N =, CH 2, S, Me, H, H, H, O], [AH1832; C, -CF = CH -, = CH-N =, CH 2, S, Et, H, H, H, O], [AH1833; C, - CF = CH -, = CH- N =, CH 2, S, c-Pr, H, H, H, O], [AH1834; C, -CF = CH -, = CH-N =, CH 2, S , OMe, H, H, H , O], [AH1835; C, -CH = CH -, = CF-N =, CH 2, S, H, H, H, H, O], [AH1836; C, -CH = CH -, = CF- N =, CH 2, S, Cl, H, H, H, O], [AH1837; C, -CH = CH -, = CF-N =, CH 2, S, br, H, H, H, O], [AH1838; C, -CH = CH -, = CF-N =, CH 2, S, CF 3, H, H, H, O], [AH1839; C, -CH = CH -, = CF- N =, CH 2, S, Me, H, H, H, O], [AH1840; C, -CH = CH -, = CF-N =, CH 2, S, Et, H, H, H, O], [AH1841; C, -CH = CH -, = CF-N =, CH 2, S, c-Pr, H, H, H, O], [AH1842; C , -CH = CH -, = CF -N =, CH 2, S, OMe, H, H, H, O], [AH184 3; C, = CH-CH = CH -, - CH =, CH 2, S, H, H, H, H, O], [AH1844; C, = CH-CH = CH -, - CH =, CH _{2, S, Cl, H,} H, H, O], [AH1845; C, = CH-CH = CH -, - CH =, CH 2, S, Br, H, H, H, O], [AH1846 ; C, = CH-CH = CH -, - CH =, CH 2, S, CF 3, H, H, H, O], [AH1847; C, = CH-CH = CH -, - CH =, CH _{2, S, Me, H,} H, H, O], [AH1848; C, = CH-CH = CH -, - CH =, CH 2, S, Et, H, H, H, O], [AH1849 ; C, = CH-CH = CH -, - CH =, CH 2, S, c-Pr, H, H, H, O], [AH1850; C, = CH-CH = CH -, - CH =, _{CH 2, S, OMe, H} , H, H, O], [AH1851; C, = CH-CH = CH -, - N =, CH 2, S, H, H, H, H, O], [ AH1852; C, = CH-CH = CH -, - N =, CH 2, S, Cl, H, H, H, O], [AH1853; C, = CH-CH = CH -, - N =, CH _{2, S, Br, H,} H, H, O], [AH1854; C, = CH-CH = CH -, - N =, CH 2, S, CF 3, H, H, H, O], [ AH1855; C, = CH-CH = CH -, - N =, CH 2, S, Me, H, H, H, O], [AH1856; C, = CH-CH = CH -, - N =, CH _{2, S, Et, H,} H, H, O], [AH1857; C, = CH-CH = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1858; C, = CH- CH = CH -, - N =, CH 2, S, OMe, H, H, H, O], [AH1859; C, = CH-C (Me) = CH -, - _{N =, CH 2, S,} H, H, H, H, O], [AH1860; C, = CH-C (Me) = CH -, - N =, CH 2, S, Cl, H, H, H, O], [AH1861; C, = CH-C (Me) = CH -, - N =, CH 2, S, Br, H, H, H, O], [AH1862; C, = CH-C (Me) = CH -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1863; C, = CH-C (Me) = CH -, - N =, CH 2 , S, Me, H, H, H, O], [AH 1864; C, = CH-C (Me) = CH-,-N _{=, CH 2, S, Et} , H, H, H, O], [AH1865; C, = CH-C (Me) = CH -, - N =, CH 2, S, c-Pr, H, H , H, O], [AH 1866; C, = CH-C (Me) = CH-,-N =, CH ₂ , S, OMe, H, H, H, O], [AH 1867; C, = C ( Me) -CH = CH -, - N =, CH 2, S, H, H, H, H, O], [AH1868; C, = C (Me) -CH = CH -, - N =, CH 2 , S, Cl, H, H , H, O], [AH1869; C, = C (Me) -CH = CH -, - N =, CH 2, S, Br, H, H, H, O], [AH1870; C, = C ( Me) -CH = CH -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1871; C, = C (Me) -CH = CH -, - N =, CH 2, S, Me, H, H, H, O], [AH1872; C, = C (Me) -CH = CH -, - N =, CH 2, S, Et, H, H, H, O] , [AH1873; C, = C (Me) -CH = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1874; C, = C (Me) -CH = CH -, - N =, CH 2, S, OMe, H, H, H, O], [AH1875; C, = CH-C (CF 3) = CH-, _{-N =, CH 2, S,} H, H, H, H, O], [AH1876; C, = CH-C (CF 3) = CH -, - N =, CH 2, S, Cl, H, H, H, O], [ AH1877; C, = CH-C (CF 3) = CH -, - N =, CH 2, S, Br, H, H, H, O], [AH1878; C, = _{CH-C (CF 3) =} CH -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1879; C, = CH-C (CF 3) = CH -, - _{N =, CH 2, S,} Me, H, H, H, O], [AH1880; C, = CH-C (CF 3) = CH -, - N =, CH 2, S, Et, H, H , H, O], [AH1881 ; C, = CH-C (CF 3) = CH -, - N =, CH 2, S, c-Pr, H, H, H, O], [AH1882; C, _{= CH-C (CF 3)} = CH -, - N =, CH 2, S, OMe, H, H, H, O], [AH1883; C, = C (CF 3) -CH = CH -, - _{N =, CH 2, S,} H, H, H, H, O], [AH1884; C, = C (CF 3) -CH = CH-, _{-N =, CH 2, S,} Cl, H, H, H, O], [AH1885; C, = C (CF 3) -CH = CH -, - N =, CH 2, S, Br, H, H, H, O], [ AH1886; C, = C (CF 3) -CH = CH -, - N =, CH 2, S, CF 3, H, H, H, O], [AH1887; C, _{= C (CF 3) -CH =} CH -, - N =, CH 2, S, Me, H, H, H, O], [AH1888; C, = C (CF 3) -CH = CH -, - _{N =, CH 2, S,} Et, H, H, H, O], [AH1889; C, = C (CF 3) -CH = CH -, - N =, CH 2, S, c-Pr, H , H, H, O], [AH1890; C, = C (CF 3) -CH = CH -, - N =, CH 2, S, OMe, H, H, H, O], [AH1891; C, -CH = CH -, = CH- C (Me) =, CH 2, NMe, H, H, H, H, O], [AH1892; C, -CH = CH -, = CH-C (Me) = _{, CH 2, NMe, Cl,} H, H, H, O], [AH1893; C, -CH = CH -, = CH-C (Me) =, CH 2, NMe, Br, H, H, H, O], [AH1894; C, -CH = CH -, = CH-C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH1895; C, -CH = CH- , = CH-C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH1896; C, -CH = CH -, = CH-C (Me) =, CH 2, NMe , Et, H, H, H , O], [AH1897; C, -CH = CH -, = CH-C (Me) =, CH 2, NMe, c-Pr, H, H, H, O], [AH1898; C, -CH = CH -, = CH-C (Me) =, CH 2, NMe, OMe, H, H, H, O], [AH1899; C, -CH = CF -, = CH- _{C (Me) =, CH 2} , NMe, H, H, H, H, O], [AH1900; C, -CH = CF -, = CH-C (Me) =, CH 2, NMe, Cl, H , H, H, O],

[AH1901; C, -CH = CF -, = CH-C (Me) =, CH 2, NMe, Br, H, H, H, O], [AH1902; C, -CH = CF -, = CH- _{C (Me) =, CH 2} , NMe, CF 3, H, H, H, O], [AH1903; C, -CH = CF -, = CH-C (Me) =, CH 2, NMe, Me, H, H, H, O] , [AH1904; C, -CH = CF -, = CH-C (Me) =, CH 2, NMe, Et, H, H, H, O], [AH1905; C, -CH = CF -, = CH- C (Me) =, CH 2, NMe, c-Pr, H, H, H, O], [AH1906; C, -CH = CF -, = CH-C (Me _{) =, CH 2, NMe,} OMe, H, H, H, O], [AH1907; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, H, H, H, H, O], [AH1908; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, Cl, H, H, H, O], [AH1909; C, -CF = CH -, = CH-C (Me ) =, CH 2, NMe, Br, H, H, H, O], [AH1910; C, -CF = CH -, = CH-C (Me) =, CH 2, _{NMe, CF 3, H, H} , H, O], [AH1911; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH1912; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, Et, H, H, H, O], [AH1913; C, -CF = CH -, = CH- _{C (Me) =, CH 2} , NMe, c-Pr, H, H, H, O], [AH1914; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, OMe , H, H, H, O ], [AH1915; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, H, H, H, H, O], [AH1916; C , -CF = CH -, = CH -C (Me) =, CH 2, NMe, Cl, H, H, H, O], [AH1917; C, -CF = CH -, = CH-C (Me) _{=, CH 2, NMe, Br} , H, H, H, O], [AH1918; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH1919; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH1920; C, -CF = CH -, = CH-C (Me) = , CH 2, NMe, Et, H, H, H, O], [AH1921; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, c-Pr, H, H, H, O], [AH1922; C, -CF = CH -, = CH-C (Me) =, CH 2, NMe, OMe, H, H, H, O], [ AH1923; C, -CH = CH - , = CF-C (Me) =, CH 2, NMe, H, H, H, H, O], [AH1924; C, -CH = CH -, = CF-C _{(Me) =, CH 2,} NMe, Cl, H, H, H, O], [AH1925; C, -CH = CH -, = CF-C (Me) =, CH 2, NMe, Br, H, H, H, O], [ AH1926; C, -CH = CH -, = CF-C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH1927; C, - CH = CH -, = CF- C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH1928; C, -CH = CH -, = CF-C (Me) =, _{CH 2, NMe, Et, H} , H, H, O], [AH1929; C, -CH = CH -, = CF-C (Me) =, CH 2, NMe, c-Pr, H, H, H , O], [AH1930; C , -CH = CH -, = CF-C (Me) =, CH 2, NMe, OMe, H, H, H, O], [AH1931; C, -CH = CH- , = CH-CBr =, CH 2, NMe, H, H, H, H, O], [AH1932; C, -CH = CH -, = CH-CBr =, CH 2, NMe, Cl, H, H , H, O], [AH1933 ; C, -CH = CH -, = CH-CBr =, CH 2, NMe, Br, H, H, H, O], [AH1934; C, -CH = CH-, _{= CH-CBr =, CH 2} , NMe, CF 3, H, H, H, O], [AH1935; C, -CH = CH -, = CH-CBr =, CH 2, NMe, Me, H, H , H, O], [AH 1936; C, -CH = CH-, = CH-CBr =, CH ₂ , NMe, Et, H, H, H, O], [AH 1937; C, -CH = CH-, _{= CH-CBr =, CH 2} , NMe, c-Pr, H, H, H, O], [AH1938; C, -CH = CH -, = CH-CBr =, CH 2, NMe, OMe, H, H, H, O], [ AH1939; C, -CH = CH -, = CH-CCl =, CH 2, NMe, H, H, H, H, O], [AH1 940; C, -CH = CH - , = CH-CCl =, CH 2, NMe, Cl, H, H, H, O], [AH1941; C, -CH = CH -, = CH-CCl =, CH _{2, NMe, Br, H,} H, H, O], [AH1942; C, -CH = CH -, = CH-CCl =, CH 2, NMe, CF 3, H, H, H, O], [ AH1943; C, -CH = CH - , = CH-CCl =, CH 2, NMe, Me, H, H, H, O], [AH1944; C, -CH = CH -, = CH-CCl =, CH _{2, NMe, Et, H,} H, H, O], [AH1945; C, -CH = CH -, = CH-CCl =, CH 2, NMe, c-Pr, H, H, H, O], [AH1946; C, -CH = CH -, = CH-CCl =, CH 2, NMe, OMe, H, H, H, O], [AH1947; C, -C (Me) = CH -, = CH- _{C (Me) =, CH 2} , NMe, H, H, H, H, O], [AH1948; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, NMe, Cl, H, H, H, O], [AH1949; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, NMe, Br, H, H, H, O], [AH1950; C, -C (Me ) = CH -, = CH-C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH1951; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH1952; C, -C (Me) = CH -, = CH-C (Me) _{=, CH 2, NMe, Et} , H, H, H, O], [AH1953; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, NMe, c-Pr, H, H, H, O] , [AH1954; C, -C (Me) = CH -, = CH-C (Me) =, CH 2, NMe, OMe, H, H, H, O], [AH1955 ; C, -CH = CH -, = CH-C (CF 3) =, CH 2, NMe, H, H, H, H, O], [AH1956; C, -CH = CH -, = CH-C _{(CF 3) =, CH 2} , NMe, Cl, H, H, H, O], [AH1957; C, -CH = CH -, = CH-C (CF 3) =, CH 2, NMe, Br, H, H, H, O] , [AH1958; C, -CH = CH -, = CH-C (CF 3) =, CH 2, NMe, CF 3, H, H, H, O], [AH1959; C, -CH = CH -, = CH-C (CF 3) =, CH 2, NMe, Me, H, H, H, O], [AH1960; C, -CH = CH -, = CH _{-C (CF 3) =, CH} 2, NMe, Et, H, H, H, O], [AH1961; C, -CH = CH -, = CH-C (CF 3) =, CH 2, NMe, c-Pr, H, H, H, O], [AH1962; C, -CH = CH -, = CH-C (CF 3) =, CH 2, NMe, OMe, H, H, H, O], [AH1963; C, -CH = CH -, = CH-C (Et) =, CH 2, NMe, H, H, H, H, O], [AH1964; C, -CH = CH -, = CH- _{C (Et) =, CH 2} , NMe, Cl, H, H, H, O], [AH1965; C, -CH = CH -, = CH-C (Et) =, CH 2, NMe, Br, H , H, H, O], [AH1966; C, -CH = CH -, = CH-C (Et) =, CH 2, NMe, CF 3, H, H, H, O], [AH1967; C, -CH = CH -, = CH- C (Et) =, CH 2, NMe, Me, H, H, H, O], [AH1968; C, -CH = CH -, = CH-C (Et) = _{, CH 2, NMe, Et,} H, H, H, O], [AH1969; C, -CH = CH -, = CH-C (Et) =, CH 2, NMe, c-Pr, H, H, H, O], [AH1970; C, -CH = CH -, = CH-C (Et) =, CH 2, NMe, OMe, H, H, H, O], [AH1971; C, -CH = CH -, = CH-C (c -Pr) =, CH 2, NMe, H, H, H, H, O], [AH1972; C, -CH = CH -, = CH-C (c-Pr) = _{, CH 2, NMe, Cl,} H, H, H, O], [AH1973; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, NMe, Br, H, H, H, O], [AH1974; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, NMe, CF 3, H, H, H, O], [AH1975; C, - CH = CH -, = CH- C (c-Pr) =, CH 2, NMe, Me, H, H, H, O], [AH1976; C, -CH = CH -, = CH-C (c- _{Pr) =, CH 2, NMe} , Et, H, H, H, O], [AH1977; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, NMe, c-Pr , H, H, H, O], [ AH1978; C, -CH = CH -, = CH-C (c-Pr) =, CH 2, NMe, OMe, H, H, H, O], [AH1979; N, -CH = CH -, - N = , CH 2, NMe, H, H, H, H, O], [AH1980; N, -CH = CH -, - N =, CH 2, NMe, F, H, H, H, O], [ AH1981; N, -CH = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH1982; N, -CH = CH -, - _{N =, CH 2, NMe,} Br, H, H, H, O], [AH1983; N, -CH = CH -, - N =, CH 2, NMe, Me, H, H, H, O], [AH1984; N, -CH = CH -, - N =, CH 2, NMe, Et, H, H, H, O], [AH1985; N, -CH = CH -, - N =, CH 2, NMe , Pr, H, H, H , O], [AH1986; N, -CH = CH -, - N =, CH 2, NMe, i-Pr, H, H, H, O], [AH1987; N, -CH = CH -, - N = , CH 2, NMe, c-Pr, H, H, H, O], [AH1988; N, -CH = CH -, - N =, CH 2, NMe, c- Bu, H, H, H, O], [AH1989; N, -CH = CH -, - N =, CH 2, NMe, OMe, H, H, H, O], [AH1990; N, -CH = CH -, - N =, CH 2, NMe, Oi-Pr, H, H, H, O], [AH1991; N, -CH = CH -, - N =, CH 2, NMe, SMe, H, H , H, O], [AH1992 ; N, -CH = CH -, - N =, CH 2, NMe, Set, H, H, H, O], [AH1993; N, -CH = CH -, - N _{=, CH 2, NMe, CF} 3, H, H, H, O], [AH1994; N, -CH = CH -, - N =, CH 2, NMe, CHF 2, H, H, H, O] , [AH1995; N, -CH = CH -, - N =, CH 2, NMe, OCF 3, H, H, H, O], [AH1996; N, -CH = CH -, - N =, CH 2 _{, NMe, OCHF 2, H,} H, H, O], [AH1997; N, -CH = CH -, - N =, CH 2, NMe, CH = CH 2, H, H, H, O], [ AH1998; N, -CH = CH - , - N =, CH 2, NMe, C (Me) = CH 2, H, H, H, O], [AH1999; N, -CH = CH-, _{-N =, CH 2, NMe,} CH = CHMe, H, H, H, O], [AH2000; N, -CH = CH -, - N =, CH 2, NMe, C≡CH, H, H, H, O],

[AH2001; N, -CH = CH -, - N =, CH 2, NMe, C≡CMe, H, H, H, O], [AH2002; N, -CH = CH -, - N =, CH 2 , NMe, CN, H, H , H, O], [AH2003; N, -CH = CF -, - N =, CH 2, NMe, H, H, H, H, O], [AH2004; N, -CH = CF -, - N = , CH 2, NMe, Cl, H, H, H, O], [AH2005; N, -CH = CF -, - N =, CH 2, NMe, Br, H, H, H, O], [ AH2006; N, -CH = CF -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2007; N, -CH = CF-, _{-N =, CH 2, NMe,} Me, H, H, H, O], [AH2008; N, -CH = CF -, - N =, CH 2, NMe, Et, H, H, H, O] , [AH2009; N, -CH = CF -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2010; N, -CH = CF -, - N =, CH _{2, NMe, OMe, H,} H, H, O], [AH2011; N, -CF = CH -, - N =, CH 2, NMe, H, H, H, H, O], [AH2012; N , -CF = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2013; N, -CF = CH -, - N =, CH 2, NMe, Br, H , H, H, O], [AH2014; N, -CF = CH -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2015; N, -CF = CH- _{, -N =, CH 2, NMe} , Me, H, H, H, O], [AH2016; N, -CF = CH -, - N =, CH 2, NMe, Et, H, H, H, O ], [AH2017; N, -CF = CH -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2018; N, -CF = CH -, - N =, _{CH 2, NMe, OMe, H} , H, H, O], [AH2019; N, -CH = CCl -, - N =, CH 2, NMe, H, H, H, H, O], [AH2020; N, -CH = CCl -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2021; N, -CH = CCl -, - N =, CH 2, NMe, Br, H, H, H, O] , [AH2022; N, -CH = CCl -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2023; N, - CH = CCl -, - N = , CH 2, NMe, Me, H, H, H, O], [AH2024; N, -CH = CCl -, - N =, CH 2, NMe, Et, H, H , H, O], [AH2025 ; N, -CH = CCl -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2026; N, -CH = CCl-, _{-N =, CH 2, NMe,} OMe, H, H, H, O], [AH2027; N, -CCl = CH -, - N =, CH 2, NMe, H, H, H, H, O] , [AH2028; N, -CCl = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2029; N, -CCl = CH -, - N =, CH 2, NMe, Br, H, H, H, O], [AH2030; N, -CCl = CH -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2031; N, -CCl = CH -, - N = , CH 2, NMe, Me, H, H, H, O], [AH2032; N, -CCl = CH -, - N =, CH 2, NMe, Et, H, H, H, O], [ AH2033; N, -CCl = CH -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2034; N, -CCl = CH- _{, -N =, CH 2, NMe} , OMe, H, H, H, O], [AH2035; N, -CH = C (Me) -, - N =, CH 2, NMe, H, H, H, H, O], [AH2036; N, -CH = C (Me) -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2037; N, -CH = C (Me ) -, - N =, CH 2, NMe, Br, H, H, H, O], [AH2038; N, -CH = C (Me) -, - N =, CH 2, NMe, CF 3, H , H, H, O], [AH2039; N, -CH = C (Me) -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2040; N, -CH = C (Me) -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2041; N, -CH = C (Me) -, - N =, CH 2, NMe, c -Pr, H, H, H, O], [AH2042; N, -CH = C (Me) -, - N =, CH 2, NMe, OMe, H, H, H, O], [AH2043; N , -C (Me) = CH - , - N =, CH 2, NMe, H, H, H, H, O], [AH2044; N, -C (Me) = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2045; N, -C (Me) = CH -, - N =, CH 2, NMe, Br, H , H, H, O], [AH2046; N, -C (Me) = CH -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2047; N, -C (Me) = CH -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2048; N, -C (Me) = CH -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2049; N, -C (Me) = CH -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2050; N, -C (Me) = CH -, - N =, CH 2, NMe, OMe, H, H, H, O], [AH2051; N, -CH = CH -, - N =, CH 2, NMe , H, F, H, H , O], [AH2052; N, -CH = CH -, - N =, CH 2, NMe, Cl, F, H, H, O], [AH2053; N, -CH = CH -, - N =, CH 2, NMe, Br, F, H, H, O], [AH2054; N, -CH = CH -, - N =, CH 2, NMe, CF 3, F, H , H, O], [AH2055 ; N, -CH = CH -, - N =, CH 2, NMe, Me, F, H, H, O], [AH2056; N, -CH = CH -, - N _{=, CH 2, NMe, Et} , F, H, H, O], [AH2057; N, -CH = CH -, - N =, CH 2, NMe, c-Pr, F, H, H, O] , [AH2058; N, -CH = CH -, - N =, CH 2, NMe, OMe, F, H, H, O], [AH2059; N, -CH = CH -, - N =, CH 2, NMe, H, H, F, H, O], [AH2060; N, -CH = CH -, - N =, CH 2, NMe, Cl, H, F, H, O], [AH2061; N, - CH = CH -, - N = , CH 2, NMe, Br, H, F, H, O], [AH2062; N, -CH = CH -, - N =, CH 2, NMe, CF 3, H, F, H, O], [ AH2063; N, -CH = CH -, - N =, CH 2, NMe, Me, H, F, H, O], [AH2064; N, -CH = CH -, - _{N =, CH 2, NMe,} Et, H, F, H, O], [AH2065; N, -CH = CH -, - N =, CH 2, NMe, c-Pr, H, F, H, O ], [AH2066; N, -CH = CH -, - N =, CH 2, NMe, OMe, H, F, H, O], [AH2067; N, -CH = CH -, - N =, CH 2, NMe , H, H, H, F , O], [AH2068; N, -CH = CH -, - N =, CH 2, NMe, Cl, H, H, F, O], [AH2069; N, -CH = CH -, - N =, CH 2, NMe, Br, H, H, F, O], [AH2070; N, -CH = CH -, - N =, CH 2, NMe, CF 3, H, H , F, O], [AH2071 ; N, -CH = CH -, - N =, CH 2, NMe, Me, H, H, F, O], [AH2072; N, -CH = CH -, - N _{=, CH 2, NMe, Et} , H, H, F, O], [AH2073; N, -CH = CH -, - N =, CH 2, NMe, c-Pr, H, H, F, O] , [AH2074; N, -CH = CH -, - N =, CH 2, NMe, OMe, H, H, F, O], [AH2075; C, = CH-S -, - N =, CH 2, NMe, H, H, H, H, O], [AH2076; C, = CH-S -, - N =, CH 2, NMe, F, H, H, H, O], [AH2077; C, = CH-S -, - N = , CH 2, NMe, Cl, H, H, H, O], [AH2078; C, = CH-S -, - N =, CH 2, NMe, Br, H, H , H, O], [AH 2079; C, = CH-S-, -N =, CH ₂ , N Me, H, H, H, O], [AH 2080; C, = CH-S-,-N _{=, CH 2, NMe, Et} , H, H, H, O], [AH2081; C, = CH-S -, - N =, CH 2, NMe, Pr, H, H, H, O], [ AH2082; C, = CH-S -, - N =, CH 2, NMe, i-Pr, H, H, H, O], [AH2083; C, = CH-S -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2084; C, = CH-S -, - N =, CH 2, NMe, c-Bu, H, H, H, O], [AH2085 ; C, = CH-S - , - N =, CH 2, NMe, OMe, H, H, H, O], [AH2086; C, = CH-S -, - N =, CH 2, NMe, Oi -Pr, H, H, H, O], [AH 2087; C, = CH-S-,-N =, CH ₂ , N Me, S Me, H, H, H, O], [AH 2088; C, = CH -S-, -N =, CH ₂ , N Me , Set, H, H, H, O], [AH 2089; C, = CH-S-,-N =, CH ₂ , N Me, CF ₃ , H, H, O], [AH 2090; C, = CH-S -, - N = , CH 2, NMe, CHF 2, H, H, H, O], [AH2091; C, = CH-S -, - N =, CH 2, NMe, OCF 3, H , H, H, O], [AH 2092; C, = CH-S-,-N =, CH ₂ , N Me, OCHF ₂ , H, H, H, O], [AH 2093; C, = CH-S- _{, -N =, CH 2, NMe} , CH = CH 2, H, H, H, O], [AH2094; C, = CH-S -, - N =, CH 2, NMe, C (Me) = CH ₂ , H, H, H, O], [AH 2095; C, = CH-S-, -N =, CH ₂ , N Me, CH = CH Me, H, H, H, O], [AH 2096; C, = CH-S -, - N = , CH 2, NMe, C≡CH, H, H, H, O], [AH2097; C, = CH-S -, - N =, CH 2, NMe, C≡CMe , H, H, H, O ], [AH2098; C, = C (CF 3) -S -, - N =, CH 2, NMe, H, H, H, H, O], [AH2099; C, _{= C (CF 3) -S -} , - N =, CH 2, NMe, Cl, H, H, H, O], [AH2100; C, = C (CF 3) -S -, - N =, CH ₂ , NMe, Br, H, H, H, O],

[AH2101; C, = C ( CF 3) -S -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2102; C, = C (CF 3) -S- _{, -N =, CH 2, NMe} , Me, H, H, H, O], [AH2103; C, = C (CF 3) -S -, - N =, CH 2, NMe, Et, H, H , H, O], [AH2104 ; C, = C (CF 3) -S -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2105; C, = C _{(CF 3) -S -, -} N =, CH 2, NMe, OMe, H, H, H, O], [AH2106; C, = CF-S -, - N =, CH 2, NMe, H, H, H, H, O], [AH 2107; C, = CF-S-,-N =, CH ₂ , N Me, Cl, H, H, H, O], [AH 2 108; C, = CF-S- _{, -N =, CH 2, NMe} , Br, H, H, H, O], [AH2109; C, = CF-S -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2110; C, = CF-S -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2111; C, = CF-S -, - N =, CH ₂ , N Me, Et, H, H, H, O], [AH 2 112; C, = CF-S-,-N =, CH ₂ , N Me, c-Pr, H, H, H, O], [AH 2 113 ; C, = CF-S - , - N =, CH 2, NMe, OMe, H, H, H, O], [AH2114; C, = CCl-S -, - N =, CH 2, NMe, H , H, H, H, O ], [AH2115; C, = CCl-S -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2116; C, = CCl-S _{-, - N =, CH 2} , NMe, Br, H, H, H, O], [AH2117; C, = CCl-S -, - N =, CH 2, NMe, CF 3, H, H, H , O], [AH2118; C , = CCl-S -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2119; C, = CCl-S -, - N =, _{CH 2, NMe, Et, H} , H, H, O], [AH2120; C, = CCl-S -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [ AH2121; C, = CCl-S -, - N =, CH 2, NMe, OMe, H, H, H, O], [AH2122; C, = C (Me) -S -, - N =, CH 2 , NMe, H, H, H, H, O ], [AH 2123; C, = C (Me)-S-,-N =, CH ₂ , N Me, Cl, H, H, H, O], [AH 2 124; C, = C (Me)-S-, _{-N =, CH 2, NMe,} Br, H, H, H, O], [AH2125; C, = C (Me) -S -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2126; C, = C (Me) -S -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2127; C, = C (Me) - S -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2128; C, = C (Me) -S -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH 2 129; C, = C (Me)-S-,-N =, CH ₂ , N Me, OMe, H, H, H, O], [AH 2 130; C, = CH -S -, - N =, CH 2, NMe, H, F, H, H, O], [AH2131; C, = CH-S -, - N =, CH 2, NMe, Cl, F, H, H, O], [AH2132; C, = CH-S -, - N =, CH 2, NMe, Br, F, H, H, O], [AH2133; C, = CH-S -, - N = , CH ₂ , NMe, CF ₃ , F, H, H, O], [AH 2 134; C, = CH-S-, -N =, CH ₂ , NMe, Me, F, H, H, O], [[ AH2135; C, = CH-S -, - N =, CH 2, NMe, Et, F, H, H, O], [AH2136; C, = CH-S -, - N =, CH 2, NMe, c-Pr, F, H, H, O], [AH 2 137; C, = CH-S-,-N =, CH ₂ , N Me, OMe, F, H, H, O], [AH 2 138; C, = CH-S -, - N = , CH 2, NMe, H, H, F, H, O], [AH2139; C, = CH-S -, - N =, CH 2, NMe, Cl, H, F , H, O], [AH 2 140; C, = CH-S-,-N =, CH ₂ , N Me, Br, H, F, H, O], [AH 2141; C, = CH-S-,-N _{=, CH 2, NMe, CF} 3, H, F, H, O], [AH2142; C, = CH-S -, - N =, CH 2, NMe, Me, H, F, H, O], [AH2143; C, = CH- S -, - N =, CH 2, NMe, Et, H, F, H, O], [AH2144; C, = CH-S -, - N =, CH 2, NMe , c-Pr, H, F, H, O], [AH 2145; C, = CH-S- _{, -N =, CH 2, NMe} , OMe, H, F, H, O], [AH2146; C, = CH-S -, - N =, CH 2, NMe, H, H, H, F, O ], [AH2147; C, = CH-S -, - N =, CH 2, NMe, Cl, H, H, F, O], [AH2148; C, = CH-S -, - N =, CH 2 , NMe, Br, H, H , F, O], [AH2149; C, = CH-S -, - N =, CH 2, NMe, CF 3, H, H, F, O], [AH2150; C , = CH-S -, - N =, CH 2, NMe, Me, H, H, F, O], [AH2151; C, = CH-S -, - N =, CH 2, NMe, Et, H , H, F, O], [AH2152; C, = CH-S-,-N =, CH ₂ , N Me, c-Pr, H, H, F, O], [AH 2 153; C, = CH-S _{-, - N =, CH 2} , NMe, OMe, H, H, F, O], [AH2154; C, = CH-O -, - N =, CH 2, NMe, H, H, H, H, O], [AH2155; C, = CH-O -, - N =, CH 2, NMe, F, H, H, H, O], [AH2156; C, = CH-O -, - N =, CH _{2, NMe, Cl, H,} H, H, O], [AH2157; C, = CH-O -, - N =, CH 2, NMe, Br, H, H, H, O], [AH2158; C , = CH-O -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2159; C, = CH-O -, - N =, CH 2, NMe, Et, H , H, H, O], [AH 2 160; C, = CH-O-,-N =, CH ₂ , N Me, Pr, H, H, H, O], [AH 2161; C, = CH-O-, _{-N =, CH 2, NMe,} i-Pr, H, H, H, O], [AH2162; C, = CH-O -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH 2 163; C, = CH-O-,-N =, CH ₂ , N Me, c-Bu, H, H, H, O], [AH 2 164; C, = CH-O-,- _{N =, CH 2, NMe,} OMe, H, H, H, O], [AH2165; C, = CH-O -, - N =, CH 2, NMe, Oi-Pr, H, H, H, O ], [AH2166; C, = CH-O -, - N =, CH 2, NMe, SMe, H, H, H, O], [AH2167; C, = CH-O -, - N =, CH 2 , NMe, Set, H, H, H, O], [AH 2 168; C, = CH-O -, - N = , CH 2, NMe, CF 3, H, H, H, O], [AH2169; C, = CH-O -, - N =, CH 2, NMe, CHF 2, H , H, H, O], [AH 2170; C, = CH-O-,-N =, CH ₂ , NMe, OCF ₃ , H, H, H, O], [AH 2171; C, = CH-O- _{, -N =, CH 2, NMe} , OCHF 2, H, H, H, O], [AH2172; C, = CH-O -, - N =, CH 2, NMe, CH = CH 2, H, H , H, O], [AH 2 173; C, = CH-O-,-N =, CH ₂ , N Me, C (Me) = CH ₂ , H, H, H, O], [AH 2 174; C, = CH -O -, - N =, CH 2, NMe, CH = CHMe, H, H, H, O], [AH2175; C, = CH-O -, - N =, CH 2, NMe, C≡CH, H, H, H, O], [AH 2176; C, = CH-O-,-N =, CH ₂ , NMe, C≡CMe, H, H, H, O], [AH 2177; C, = C ( _{CF 3) -O -, - N} =, CH 2, NMe, H, H, H, H, O], [AH2178; C, = C (CF 3) -O -, - N =, CH 2, NMe , Cl, H, H, H, O], [AH 2179; C, = C (CF ₃ ) -O-, -N =, CH ₂ , N Me, Br, H, H, H, O], [AH 2 180; _{C, = C (CF 3)} -O -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2181; C, = C (CF 3) -O -, - N _{=, CH 2, NMe, Me} , H, H, H, O], [AH2182; C, = C (CF 3) -O -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2183; C, = C (CF 3) -O -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2184; C, = C (CF 3 ) -O-, -N =, CH ₂ , NMe, OMe, H, H, H, O], [AH 2 185; C, = CF-O-, -N =, CH ₂ , NMe, H, H, H , H, O], [AH2186 ; C, = CF-O -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2187; C, = CF-O -, - N _{=, CH 2, NMe, Br} , H, H, H, O], [AH2188; C, = CF-O -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH 2189; C, = CF-O -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2190; C, = CF-O -, - N =, CH 2, NMe, Et, H, H, H, O] , [AH2191; C, = CF-O -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2192; C, = CF- O -, - N =, CH 2, NMe, OMe, H, H, H, O], [AH2193; C, = CCl-O -, - N =, CH 2, NMe, H, H, H, H , O], [AH2194; C , = CCl-O -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2195; C, = CCl-O -, - N =, _{CH 2, NMe, Br, H} , H, H, O], [AH2196; C, = CCl-O -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2197 ; C, = CCl-O - , - N =, CH 2, NMe, Me, H, H, H, O], [AH2198; C, = CCl-O -, - N =, CH 2, NMe, Et , H, H, H, O ], [AH2199; C, = CCl-O -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2200; C, = CCl -O -, - N =, CH 2, NMe, OMe, H, H, H, O],

[AH2201; C, = C ( Me) -O -, - N =, CH 2, NMe, H, H, H, H, O], [AH2202; C, = C (Me) -O -, - N _{=, CH 2, NMe, Cl} , H, H, H, O], [AH2203; C, = C (Me) -O -, - N =, CH 2, NMe, Br, H, H, H, O ], [AH2204; C, = C (Me) -O -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2205; C, = C (Me) -O- _{, -N =, CH 2, NMe} , Me, H, H, H, O], [AH2206; C, = C (Me) -O -, - N =, CH 2, NMe, Et, H, H, H, O], [AH 2 207; C, = C (Me)-O-,-N =, CH ₂ , N Me, c-Pr, H, H, H, O], [AH 2 208; C, = C (Me ) -O-, -N =, CH ₂ , NMe, OMe, H, H, H, O], [AH 2209; C, = CH-O-, -N =, CH ₂ , NMe, H, F, H , H, O], [AH2210 ; C, = CH-O -, - N =, CH 2, NMe, Cl, F, H, H, O], [AH2211; C, = CH-O -, - N _{=, CH 2, NMe, Br} , F, H, H, O], [AH2212; C, = CH-O -, - N =, CH 2, NMe, CF 3, F, H, H, O], [AH2213; C, = CH- O -, - N =, CH 2, NMe, Me, F, H, H, O], [AH2214; C, = CH-O -, - N =, CH 2, NMe , Et, F, H, H , O], [AH2215; C, = CH-O -, - N =, CH 2, NMe, c-Pr, F, H, H, O], [AH2216; C, = CH-O -, - N =, CH 2, NMe, OMe, F, H, H, O], [AH2217; C, = CH-O -, - N =, CH 2, NMe, H, H, F, H, O], [ AH2218; C, = CH-O -, - N =, CH 2, NMe, Cl, H, F, H, O], [AH2219; C, = CH-O -, - _{N =, CH 2, NMe,} Br, H, F, H, O], [AH2220; C, = CH-O -, - N =, CH 2, NMe, CF 3, H, F, H, O] , [AH2221; C, = CH -O -, - N =, CH 2, NMe, Me, H, F, H, O], [AH2222; C, = CH-O -, - N =, CH 2, NMe, Et, H, F, H, O], [AH 2223; C, = CH-O-,- _{N =, CH 2, NMe,} c-Pr, H, F, H, O], [AH2224; C, = CH-O -, - N =, CH 2, NMe, OMe, H, F, H, O ], [AH2225; C, = CH-O -, - N =, CH 2, NMe, H, H, H, F, O], [AH2226; C, = CH-O -, - N =, CH 2 , NMe, Cl, H, H, F, O], [AH 2 227; C, = CH-O-, -N =, CH ₂ , N Me, Br, H, H, F, O], [AH 2 228; C, = CH-O -, - N =, CH 2, NMe, CF 3, H, H, F, O], [AH2229; C, = CH-O -, - N =, CH 2, NMe, Me, H , H, F, O], [AH 2 230; C, = CH-O-,-N =, CH ₂ , N Me, Et, H, H, F, O], [AH 2 231; C, = CH-O-, _{-N =, CH 2, NMe,} c-Pr, H, H, F, O], [AH2232; C, = CH-O -, - N =, CH 2, NMe, OMe, H, H, F, O], [AH2233; C, = CH-O -, - N =, CH 2, NMe, H, H, H, H, O], [AH2234; C, = CH-O -, - N =, CH _{2, NMe, Cl, H,} H, H, O], [AH2235; C, = CH-O -, - N =, CH 2, NMe, Br, H, H, H, O], [AH2236; C , = CH-O -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2237; C, = CH-O -, - N =, CH 2, NMe, Me, H, H, H, O] , [AH2238; C, = CH-O -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2239; C, = CH-O- _{, -N =, CH 2, NMe} , c-Pr, H, H, H, O], [AH2240; C, = CH-O -, - N =, CH 2, NMe, OMe, H, H, H , O], [AH2241; C , = CH-O -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2242; C, = CH-O -, - CH =, _{CH 2, NMe, F, H} , H, H, O], [AH2243; C, = CH-O -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2244; C, = CH-O -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2245; C, = CH-O -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH 2246; C, = CH -O -, - CH =, CH 2, NMe, Et, H, H, H, O], [AH2247; C, = CH-O -, - CH =, CH 2, NMe, Pr, H, H, H, O], [AH 2248; C, = CH-O-, -CH =, CH ₂ , NMe, i-Pr, H, H, H, O], [AH 2249; C, = CH-O-,- _{CH =, CH 2, NMe,} c-Pr, H, H, H, O], [AH2250; C, = CH-O -, - CH =, CH 2, NMe, c-Bu, H, H, H , O], [AH2251; C , = CH-O -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2252; C, = CH-O -, - CH =, _{CH 2, NMe, Oi-Pr} , H, H, H, O], [AH2253; C, = CH-O -, - CH =, CH 2, NMe, SMe, H, H, H, O], [ AH2254; C, = CH-O -, - CH =, CH 2, NMe, Set, H, H, H, O], [AH2255; C, = CH-O -, - CH =, CH 2, NMe, _{CF 3, H, H, H} , O], [AH2256; C, = CH-O -, - CH =, CH 2, NMe, CHF 2, H, H, H, O], [AH2257; C, = CH-O -, - CH = , CH 2, NMe, OCF 3, H, H, H, O], [AH2258; C, = CH-O -, - CH =, CH 2, NMe, OCHF 2, H , H, H, O], [AH 2259; C, = CH-O-, -CH =, CH ₂ , NMe, CH = CH ₂ , H, H, H, O], [AH 2 260; C, = CH- O -, - CH =, CH 2, NMe, C (Me) = CH 2, H, H, H, O], [AH2261; C, = CH-O -, - CH =, CH 2, NMe, CH = CHMe, H, H, H , O], [AH2262; C, = CH-O -, - CH =, CH 2, NMe, C≡CH, H, H, H, O], [AH2263; C, = CH-O -, - CH =, CH 2, NMe, C≡CMe, H, H, H, O], [AH2264; C, = C (CF 3) -O -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2265; C, = C (CF 3) -O -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2266 _{; C, = C (CF 3} ) -O -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2267; C, = C (CF _{3) -O -, - CH =} , CH 2, NMe, CF 3, H, H, H, O], [AH2268; C, = C (CF 3) -O -, - CH =, CH 2, NMe , Me, H, H, H , O], [AH2269; C, = C (CF 3) -O -, - CH =, CH 2, NMe, Et, H, H, H, O], [AH2270; _{C, = C (CF 3)} -O -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2271; C, = C (CF 3) -O -, - _{CH =, CH 2, NMe,} OMe, H, H, H, O], [AH2272; C, = CF-O -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2273; C, = CF- O -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2274; C, = CF-O -, - CH =, CH 2, NMe , Br, H, H, H , O], [AH2275; C, = CF-O -, - CH =, CH 2, NMe, CF 3, H, H, H, O], [AH2276; C, = CF-O -, - CH = , CH 2, NMe, Me, H, H, H, O], [AH2277; C, = CF-O -, - CH =, CH 2, NMe, Et, H, H , H, O], [AH 2278; C, = CF-O-, -CH =, CH ₂ , NMe, c-Pr, H, H, H, O], [AH 2279; C, = CF-O-, _{-CH =, CH 2, NMe,} OMe, H, H, H, O], [AH2280; C, = CCl-O -, - CH =, CH 2, NMe, H, H, H, H, O] , [AH2281; C, = CCl -O -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2282; C, = CCl-O -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2283; C, = CCl-O -, - CH =, CH 2, NMe, CF 3, H, H, H, O], [AH2284; C, = CCl-O -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH2285; C, = CCl-O -, - CH =, CH 2, NMe, Et, H, H, H, O], [ AH2286; C, = CCl-O -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2287; C, = CCl-O- _{, -CH =, CH 2, NMe} , OMe, H, H, H, O], [AH2288; C, = C (Me) -O -, - CH =, CH 2, NMe, H, H, H, H, O], [AH 2 289; C, = C (Me)-O-, -CH =, CH ₂ , N Me, Cl, H, H, H, O], [AH 2 290; C, = C (Me) -O -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2291; C, = C (Me) -O -, - CH =, CH 2, NMe, _{CF 3, H, H, H} , O], [AH2292; C, = C (Me) -O -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH2293; C , = C (Me) -O - , - CH =, CH 2, NMe, Et, H, H, H, O], [AH2294; C, = C (Me) -O -, - CH =, CH 2 , NMe, c-Pr, H , H, H, O], [AH2295; C, = C (Me) -O -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2296; C, = CH- O -, - CH =, CH 2, NMe, H, F, H, H, O], [AH2297; C, = CH-O -, - CH =, CH 2, NMe , Cl, F, H, H , O], [AH2298; C, = CH-O -, - CH =, CH 2, NMe, Br, F, H, H, O], [AH2299; C, = CH -O -, - CH =, CH 2, NMe, CF 3, F, H, H, O], [AH2300; C, = CH-O -, - CH =, CH 2, NMe, Me, F, H , H, O],

[AH2301; C, = CH- O -, - CH =, CH 2, NMe, Et, F, H, H, O], [AH2302; C, = CH-O -, - CH =, CH 2, NMe , c-Pr, F, H , H, O], [AH2303; C, = CH-O -, - CH =, CH 2, NMe, OMe, F, H, H, O], [AH2304; C, = CH-O -, - CH =, CH 2, NMe, H, H, F, H, O], [AH2305; C, = CH-O -, - CH =, CH 2, NMe, Cl, H, F, H, O], [AH 2306; C, = CH-O-, -CH =, CH ₂ , NMe, Br, H, F, H, O], [AH 2307; C, = CH-O-,- _{CH =, CH 2, NMe,} CF 3, H, F, H, O], [AH2308; C, = CH-O -, - CH =, CH 2, NMe, Me, H, F, H, O] , [AH2309; C, = CH -O -, - CH =, CH 2, NMe, Et, H, F, H, O], [AH2310; C, = CH-O -, - CH =, CH 2, NMe, c-Pr, H, F, H, O], [AH2311; C, = CH-O -, - CH =, CH 2, NMe, OMe, H, F, H, O], [AH2312; C , = CH-O -, - CH =, CH 2, NMe, H, H, H, F, O], [AH2313; C, = CH-O -, - CH =, CH 2, NMe, Cl, H , H, F, O], [AH2314; C, = CH-O -, - CH =, CH 2, NMe, Br, H, H, F, O], [AH2315; C, = CH-O-, _{-CH =, CH 2, NMe,} CF 3, H, H, F, O], [AH2316; C, = CH-O -, - CH =, CH 2, NMe, Me, H, H, F, O ], [AH2317; C, = CH-O -, - CH =, CH 2, NMe, Et, H, H, F, O], [AH2318; C, = CH-O -, - CH =, CH 2 , NMe, c-Pr, H , H, F, O], [AH2319; C, = CH-O -, - CH =, CH 2, NMe, OMe, H, H, F, O], [AH2320; C, = CH-O -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2321; C, = CH-O -, - CH =, CH 2, NMe, Cl, H, H, H, O] , [AH2322; C, = CH-O -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2323; C, = CH-O- , -CH _{=, CH 2, NMe, CF} 3, H, H, H, O], [AH2324; C, = CH-O -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH2325; C, = CH- O -, - CH =, CH 2, NMe, Et, H, H, H, O], [AH2326; C, = CH-O -, - CH =, CH 2, NMe , c-Pr, H, H , H, O], [AH2327; C, = CH-O -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2328; C, = CH-CH =, - O- , CH 2, NMe, H, H, H, H, O], [AH2329; C, = CH-CH =, - O-, CH 2, NMe, F, H, H, H, O], [AH 2 330; C, = CH-CH =, -O-, CH ₂ , N Me, Cl, H, H, H, O], [AH 2331; C, = CH-CH =,- _{O-, CH 2, NMe, Br} , H, H, H, O], [AH2332; C, = CH-CH =, - O-, CH 2, NMe, Me, H, H, H, O], [AH2333; C, = CH- CH =, - O-, CH 2, NMe, Et, H, H, H, O], [AH2334; C, = CH-CH =, - O-, CH 2, NMe , Pr, H, H, H, O], [AH 2 335; C, = CH-CH =, -O-, CH ₂ , NMe, i-Pr, H, H, H, O], [AH 2336; C, = CH-CH =, - O- , CH 2, NMe, c-Pr, H, H, H, O], [AH2337; C, = CH-CH =, - O-, CH 2, NMe, c- Bu, H, H, H, O], [AH 2338; C, = CH-CH =, -O-, CH ₂ , NMe, OMe, H, H, H, O], [AH 2339; C, = CH- _{CH =, - O-, CH 2} , NMe, Oi-Pr, H, H, H, O], [AH2340; C, = CH-CH =, - O-, CH 2, NMe, SMe, H, H , H, O], [AH2341 ; C, = CH-CH =, - O-, CH 2, NMe, Set, H, H, H, O], [AH2342; C, = CH-CH =, - O _{-, CH 2, NMe, CF} 3, H, H, H, O], [AH2343; C, = CH-CH =, - O-, CH 2, NMe, CHF 2, H, H, H, O] , [AH2344; C, = CH -CH =, - O-, CH 2, NMe, OCF 3, H, H, H, O], [AH2345; C, = CH-CH =, - O-, CH _{2, NMe, OCHF 2, H} , H, H, O], [AH2346; C, = CH-CH =, - O-, CH 2, NMe, CH = CH 2, H, H, H, O], [AH2347; C, = CH- CH =, - O-, CH 2, NMe, C (Me) = CH 2, H, H, H, O], [AH2348; C, = CH-CH =, - O _{-, CH 2, NMe, CH} = CHMe, H, H, H, O], [AH2349; C, = CH-CH =, - O-, CH 2, NMe, C≡CH, H, H, H, O], [AH2350; C, = CH-CH =, - O-, CH 2, NMe, C≡CMe, H, H, H, O], [AH2351; C, = C (CF 3) -CH = _{, -O-, CH 2, NMe,} H, H, H, H, O], [AH2352; C, = C (CF 3) -CH =, - O-, CH 2, NMe, Cl, H, H , H, O], [AH2353 ; C, = = C (CF 3) -CH, - O-, CH 2, NMe, Br, H, H, H, O], [AH2354; C, = C (CF _{3) -CH =, - O-,} CH 2, NMe, CF 3, H, H, H, O], [AH2355; C, = C (CF 3) -CH =, - O-, CH 2, NMe , Me, H, H, H, O], [AH 2 356; C, = C (CF ₃ ) -CH =, -O-, CH ₂ , N Me, Et, H, H, H, O], [AH 2 357; _{C, = = C (CF 3} ) -CH, - O-, CH 2, NMe, c-Pr, H, H, H, O], [AH2358; C, = C (CF 3) -CH =, - _{O-, CH 2, NMe, OMe} , H, H, H, O], [AH2359; C, = CF-CH =, - O-, CH 2, NMe, H, H, H, H, O], [AH2360; C, = CF- CH =, - O-, CH 2, NMe, Cl, H, H, H, O], [AH2361; C, = CF-CH =, - O-, CH 2, NMe , Br, H, H, H , O], [AH2362; C, = CF-CH =, - O-, CH 2, NMe, CF 3, H, H, H, O], [AH2363; C, = CF-CH =, - O-, CH 2, NMe, Me, H, H, H, O], [AH2364; C, = CF-CH =, - O-, CH 2, NMe, Et, H, H , H, O], [AH 2 365; C, = CF-CH =, -O-, CH ₂ , N Me, c-Pr, H, H, H, O], [AH 2 366; C, = CF-CH =, - O- , CH 2, NMe, OMe, H, H, H, O], [AH2367; C, = CCl-CH =, - O-, CH 2, NMe, H, H, H, H, O], [AH 2368; C, = CCl-CH =, -O-, CH ₂ , N Me, Cl, H, H, H, O], [AH 2369; C, = CCl-CH =,- _{O-, CH 2, NMe, Br} , H, H, H, O], [AH2370; C, = CCl-CH =, - O-, CH 2, NMe, CF 3, H, H, H, O] , [AH2371; C, = CCl -CH =, - O-, CH 2, NMe, Me, H, H, H, O], [AH2372; C, = CCl-CH =, - O-, CH 2, NMe, Et, H, H, H, O], [AH2373; C, = CCl-CH =, - O-, CH 2, NMe, c-Pr, H, H, H, O], [AH2374; C , = CCl-CH =, -O-, CH ₂ , NMe, OMe, H, H, H, O], [AH 2 375; C, = C (Me) -CH =, -O-, CH ₂ , NMe, H, H, H, H, H, O], [AH 2376; C, = C (Me) -CH =, -O-, CH ₂ , N Me, H, H, H, O], [AH 2 377; C, = C (Me) -CH =, - O-, CH 2, NMe, Br, H, H, H, O], [AH2378; C, = C (Me) -CH =, - O-, CH 2, _{NMe, CF 3, H, H} , H, O], [AH2379; C, = C (Me) -CH =, - O-, CH 2, NMe, Me, H, H, H, O], [AH2380 ; C, = C (Me) -CH =, - O-, CH 2, NMe, Et, H, H, H, O], [AH2381; C, = C (Me) -CH =, - O-, _{CH 2, NMe, c-Pr} , H, H, H, O], [AH2382; C, = C (Me) -CH =, - O-, CH 2, NMe, OMe, H, H, H, O ], [AH2383; C, = CH-CH =, - O-, CH 2, NMe, H, F, H, H, O], [AH2384; C, = CH-CH =, - O-, CH 2 , NMe, Cl, F, H, H, O], [AH 2385; C, = CH-CH =, -O-, CH ₂ , NMe, Br, F, H, H, O], [AH 2386; C, = CH-CH =, - O- , CH 2, NMe, CF 3, F, H, H, O], [AH2387; C, = CH-CH =, - O-, CH 2, NMe, Me, F , H, H, O], [AH2388; C, = CH-CH =, - O-, CH 2, NMe, Et, F, H, H, O], [AH2389; C, = CH-CH =, - O-, CH _{2, NMe, c-Pr,} F, H, H, O], [AH2390; C, = CH-CH =, - O-, CH 2, NMe, OMe, F, H, H, O], [AH2391 ; C, = CH-CH = , - O-, CH 2, NMe, H, H, F, H, O], [AH2392; C, = CH-CH =, - O-, CH 2, NMe, Cl , H, F, H, O ], [AH2393; C, = CH-CH =, - O-, CH 2, NMe, Br, H, F, H, O], [AH2394; C, = CH-CH _{=, - O-, CH 2,} NMe, CF 3, H, F, H, O], [AH2395; C, = CH-CH =, - O-, CH 2, NMe, Me, H, F, H , O], [AH2396; C , = CH-CH =, - O-, CH 2, NMe, Et, H, F, H, O], [AH2397; C, = CH-CH =, - O-, _{CH 2, NMe, c-Pr} , H, F, H, O], [AH2398; C, = CH-CH =, - O-, CH 2, NMe, OMe, H, F, H, O], [ AH2399; C, = CH-CH =, - O-, CH 2, NMe, H, H, H, F, O], [AH2400; C, = CH-CH =, - O-, CH 2, NMe, Cl, H, H, F, O],

[AH2401; C, = CH- CH =, - O-, CH 2, NMe, Br, H, H, F, O], [AH2402; C, = CH-CH =, - O-, CH 2, NMe , CF ₃ , H, H, F, O], [AH 2403; C, = CH-CH =, -O-, CH ₂ , NMe, Me, H, F, O], [AH 2404; C, = CH-CH =, - O-, CH 2, NMe, Et, H, H, F, O], [AH2405; C, = CH-CH =, - O-, CH 2, NMe, c-Pr, H , H, F, O], [AH 2406; C, = CH-CH =, -O-, CH ₂ , NMe, OMe, H, F, O], [AH 2407; C, = CH-CH =, _{-O-, CH 2, NMe, H} , H, H, H, O], [AH2408; C, = CH-CH =, - O-, CH 2, NMe, Cl, H, H, H, O] , [AH2409; C, = CH -CH =, - O-, CH 2, NMe, Br, H, H, H, O], [AH2410; C, = CH-CH =, - O-, CH 2, _{NMe, CF 3, H, H} , H, O], [AH2411; C, = CH-CH =, - O-, CH 2, NMe, Me, H, H, H, O], [AH2412; C, = CH-CH =, - O- , CH 2, NMe, Et, H, H, H, O], [AH2413; C, = CH-CH =, - O-, CH 2, NMe, c-Pr, H, H, H, O] , [AH2414; C, = CH-CH =, - O-, CH 2, NMe, OMe, H, H, H, O], [AH2415; C, = CH-CH = _{, -S-, CH 2, NMe,} H, H, H, H, O], [AH2416; C, = CH-CH =, - S-, CH 2, NMe, F, H, H, H, O ], [AH2417; C, = CH-CH =, - S-, CH 2, NMe, Cl, H, H, H, O], [AH2418; C, = CH-CH =, - S-, CH 2 , NMe, Br, H, H , H, O], [AH2419; C, = CH-CH =, - S-, CH 2, NMe, Me, H, H, H, O], [AH2420; C, = CH-CH =, - S- , CH 2, NMe, Et, H, H, H, O], [AH2421; C, = CH-CH =, - S-, CH 2, NMe, Pr, H, H, H, O], [ AH2422; C, = CH-CH =, - S-, CH 2, NMe, i-Pr, H, H, H, O], [AH2423; C, = CH-CH = , -S- _{, CH 2, NMe, c-} Pr, H, H, H, O], [AH2424; C, = CH-CH =, - S-, CH 2, NMe, c-Bu, H, H, H, O ], [AH2425; C, = CH-CH =, - S-, CH 2, NMe, OMe, H, H, H, O], [AH2426; C, = CH-CH =, - S-, CH 2 , NMe, Oi-Pr, H , H, H, O], [AH2427; C, = CH-CH =, - S-, CH 2, NMe, SMe, H, H, H, O], [AH2428; C, = CH-CH =, - S-, CH 2, NMe, Set, H, H, H, O], [AH2429; C, = CH-CH =, - S-, CH 2, NMe, CF 3 , H, H, H, O ], [AH2430; C, = CH-CH =, - S-, CH 2, NMe, CHF 2, H, H, H, O], [AH2431; C, = CH- _{CH =, - S-, CH 2} , NMe, OCF 3, H, H, H, O], [AH2432; C, = CH-CH =, - S-, CH 2, NMe, OCHF 2, H, H , H, O], [AH2433 ; C, = CH-CH =, - S-, CH 2, NMe, CH = CH 2, H, H, H, O], [AH2434; C, = CH-CH = _{, -S-, CH 2, NMe,} C (Me) = CH 2, H, H, H, O], [AH2435; C, = CH-CH =, - S-, CH 2, NMe, CH = CHMe , H, H, H, O ], [AH2436; C, = CH-CH =, - S-, CH 2, NMe, C≡CH, H, H, H, O], [AH2437; C, = CH _{-CH =, - S-, CH 2} , NMe, C≡CMe, H, H, H, O], [AH2438; C, = C (CF 3) -CH =, - S-, CH 2, NMe, H, H, H, H, O], [AH2439; C, = C (CF 3) -CH =, - S-, CH 2, NMe, Cl, H, H, H, O], [AH2440; C _{, = = C (CF 3)} -CH, - S-, CH 2, NMe, Br, H, H, H, O], [AH2441; C, = C (CF 3) -CH =, - S-, _{CH 2, NMe, CF 3,} H, H, H, O], [AH2442; C, = C (CF 3) -CH =, - S-, CH 2, NMe, Me, H, H, H, O ], [AH2443; C, = C (CF 3) -CH =, - S-, CH 2, NMe, Et, H, H, H, O], [AH2 444; C, = C (CF 3) -CH =, - S-, CH 2, NMe, c-Pr, H, H, H, O], [AH2445; C, = C (CF 3) -CH = _{, -S-, CH 2, NMe,} OMe, H, H, H, O], [AH2446; C, = CF-CH =, - S-, CH 2, NMe, H, H, H, H, O ], [AH2447; C, = CF-CH =, - S-, CH 2, NMe, Cl, H, H, H, O], [AH2448; C, = CF-CH =, - S-, CH 2 , NMe, Br, H, H , H, O], [AH2449; C, = CF-CH =, - S-, CH 2, NMe, CF 3, H, H, H, O], [AH2450; C , = CF-CH =, - S-, CH 2, NMe, Me, H, H, H, O], [AH2451; C, = CF-CH =, - S-, CH 2, NMe, Et, H , H, H, O], [AH2452; C, = CF-CH =, - S-, CH 2, NMe, c-Pr, H, H, H, O], [AH2453; C, = CF-CH _{=, - S-, CH 2,} NMe, OMe, H, H, H, O], [AH2454; C, = CCl-CH =, - S-, CH 2, NMe, H, H, H, H, O], [AH2455; C, = CCl-CH =, - S-, CH 2, NMe, Cl, H, H, H, O], [AH2456; C, = CCl-CH =, - S-, CH _{2, NMe, Br, H,} H, H, O], [AH2457; C, = CCl-CH =, - S-, CH 2, NMe, CF 3, H, H, H, O], [AH2458; C, = = CCl-CH, - S-, CH 2, NMe, Me, H, H, H, O], [AH2459; C, = CCl-CH =, - S-, CH 2, NMe, Et, H, H, H, O] , [AH2460; C, = CCl-CH =, - S-, CH 2, NMe, c-Pr, H, H, H, O], [AH2461; C, = CCl- _{CH =, - S-, CH 2} , NMe, OMe, H, H, H, O], [AH2462; C, = C (Me) -CH =, - S-, CH 2, NMe, H, H, H, H, O], [ AH2463; C, = C (Me) -CH =, - S-, CH 2, NMe, Cl, H, H, H, O], [AH2464; C, = C (Me ) -CH =, - S-, CH 2, NMe, Br, H, H, H, O], [AH2465; C, = C (Me) -CH =, - S-, CH 2, NMe, CF 3 , H, H, H, O], [AH 2466; C, = C (Me) -CH =, -S-, CH ₂ , N Me, H, H, H, O], [AH 2467; C, = C (Me) -CH =, - S-, CH 2, NMe, Et, H, H, H, O], [AH2468; C, = C (Me) -CH =, - S-, CH 2, NMe , c-Pr, H, H, H, O], [AH 2469; C, = C (Me) -CH =, -S-, CH ₂ , N Me, OMe, H, H, H, O], [AH 2 470 ; C, = CH-CH = , - S-, CH 2, NMe, H, F, H, H, O], [AH2471; C, = CH-CH =, - S-, CH 2, NMe, Cl , F, H, H, O ], [AH2472; C, = CH-CH =, - S-, CH 2, NMe, Br, F, H, H, O], [AH2473; C, = CH-CH _{=, - S-, CH 2,} NMe, CF 3, F, H, H, O], [AH2474; C, = CH-CH =, - S-, CH 2, NMe, Me, F, H, H , O], [AH2475; C , = CH-CH =, - S-, CH 2, NMe, Et, F, H, H, O], [AH2476; C, = CH-CH =, - S-, _{CH 2, NMe, c-Pr} , F, H, H, O], [AH2477; C, = CH-CH =, - S-, CH 2, NMe, OMe, F, H, H, O], [ AH2478; C, = CH-CH =, - S-, CH 2, NMe, H, H, F, H, O], [AH2479; C, = CH-CH =, - S-, CH 2, NMe, Cl, H, F, H, O], [AH2480; C, = CH-CH =, - S-, CH 2, NMe, Br, H, F, H, O], [AH2481; C, = CH- _{CH =, - S-, CH 2} , NMe, CF 3, H, F, H, O], [AH2482; C, = CH-CH =, - S-, CH 2, NMe, Me, H, F, H, O], [AH2483; C, = CH-CH =, - S-, CH 2, NMe, Et, H, F, H, O], [AH2484; C, = CH-CH =, - S- , CH ₂ , NMe, c-Pr, H, F, H, O], [AH 2485; C, = CH-CH =, -S-, CH ₂ , NMe, OMe, H, F, H, O], [AH2486; C, = CH- CH =, - S-, CH 2, NMe, H, H, H, F, O], [AH2487; C, = CH-CH =, - S-, CH 2, NMe , Cl, H, H, F, O], [AH2488; C, = CH-CH =, - S-, CH 2, NMe, Br, H, H, F, O], [AH2489; C, = CH-CH =, - S-, CH _{2, NMe, CF 3, H} , H, F, O], [AH2490; C, = CH-CH =, - S-, CH 2, NMe, Me, H, H, F, O], [AH2491; C, = CH-CH =, - S-, CH 2, NMe, Et, H, H, F, O], [AH2492; C, = CH-CH =, - S-, CH 2, NMe, c- Pr, H, H, F, O], [AH2493; C, = CH-CH =, - S-, CH 2, NMe, OMe, H, H, F, O], [AH2494; C, = CH- _{CH =, - S-, CH 2} , NMe, H, H, H, H, O], [AH2495; C, = CH-CH =, - S-, CH 2, NMe, Cl, H, H, H , O], [AH2496; C , = CH-CH =, - S-, CH 2, NMe, Br, H, H, H, O], [AH2497; C, = CH-CH =, - S-, _{CH 2, NMe, CF 3,} H, H, H, O], [AH2498; C, = CH-CH =, - S-, CH 2, NMe, Me, H, H, H, O], [AH2499 ; C, = CH-CH = , - S-, CH 2, NMe, Et, H, H, H, O], [AH2500; C, = CH-CH =, - S-, CH 2, NMe, c -Pr, H, H, H, O],

[AH2501; C, = CH- CH =, - S-, CH 2, NMe, OMe, H, H, H, O], [AH2502; C, = CH-S -, - CH =, CH 2, NMe , H, H, H, H, O], [AH 2503; C, = CH-S-, -CH =, CH ₂ , N Me, F, H, H, H, O], [AH 2504; C, = CH -S -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2505; C, = CH-S -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2506; C, = CH-S -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH2507; C, = CH-S -, - CH = , CH ₂ , NMe, Et, H, H, H, O], [AH 2508; C, = CH-S-, -CH =, CH ₂ , NMe, Pr, H, H, H, O], [AH 2509 ; C, = CH-S - , - CH =, CH 2, NMe, i-Pr, H, H, H, O], [AH2510; C, = CH-S -, - CH =, CH 2, NMe , c-Pr, H, H , H, O], [AH2511; C, = CH-S -, - CH =, CH 2, NMe, c-Bu, H, H, H, O], [AH2512; C, = CH-S -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2513; C, = CH-S -, - CH =, CH 2, NMe, Oi- Pr, H, H, H, O], [AH2514; C, = CH-S -, - CH =, CH 2, NMe, SMe, H, H, H, O], [AH2515; C, = CH- S -, - CH =, CH 2, NMe, Set, H, H, H, O], [AH2516; C, = CH-S -, - CH =, CH 2, NMe, CF 3, H, H, H, O], [AH2517; C, = CH-S -, - CH =, CH 2, NMe, CHF 2, H, H, H, O], [AH2518; C, = CH-S -, - CH _{=, CH 2, NMe, OCF} 3, H, H, H, O], [AH2519; C, = CH-S -, - CH =, CH 2, NMe, OCHF 2, H, H, H, O] , [AH2520; C, = CH -S -, - CH =, CH 2, NMe, CH = CH 2, H, H, H, O], [AH2521; C, = CH-S -, - CH =, _{CH 2, NMe, C (Me} ) = CH 2, H, H, H, O], [AH2522; C, = CH-S -, - CH =, CH 2, NMe, CH = CHMe, H, H, H , O], [AH2523; C, = CH-S -, - CH =, CH 2, NMe, C≡CH, H, H, H, O], [AH2524; C, = CH-S -, - CH =, CH 2, NMe, C≡CMe, H, H, H, O], [AH2525; C, = C (CF 3) -S -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2526; C, = C (CF 3) -S -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2527 _{; C, = C (CF 3} ) -S -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2528; C, = C (CF 3) -S -, - CH _{=, CH 2, NMe, CF} 3, H, H, H, O], [AH2529; C, = C (CF 3) -S -, - CH =, CH 2, NMe, Me, H, H, H , O], [AH2530; C , = C (CF 3) -S -, - CH =, CH 2, NMe, Et, H, H, H, O], [AH2531; C, = C (CF 3) -S -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2532; C, = C (CF 3) -S -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2533; C, = CF-S -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2534; C, = CF- S -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2535; C, = CF-S -, - CH =, CH 2, NMe, Br, H, H, H , O], [AH 2536; C, = CF-S-, -CH =, CH ₂ , NMe, CF ₃ , H, H, H, O], [AH 2537; C, = CF-S-, -CH = _{, CH 2, NMe, Me,} H, H, H, O], [AH2538; C, = CF-S -, - CH =, CH 2, NMe, Et, H, H, H, O], [AH2539 ; C, = CF-S - , - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2540; C, = CF-S -, - CH =, CH 2, NMe , OMe, H, H, H , O], [AH2541; C, = CCl-S -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2542; C, = CCl -S -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2543; C, = CCl-S -, - CH =, CH 2, NMe, Br, H , H, H, O], [AH2544; C, = CCl-S -, - CH =, CH 2, NMe, CF 3, H, H, H, O], [AH2545; C, = CCl-S- _{, -CH =, CH 2, NMe} , Me, H, H, H, O], [AH2546; C, = CCl-S -, - CH =, CH 2, NMe, Et, H, H, H, O ], [AH2547; C, = CCl-S -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2548; C, = CCl-S -, - CH =, _{CH 2, NMe, OMe, H} , H, H, O], [AH2549; C, = C (Me) -S -, - CH =, CH 2, NMe, H, H, H, H, O], [AH2550; C, = C ( Me) -S -, - CH =, CH 2, NMe, Cl, H, H, H, O], [AH2551; C, = C (Me) -S -, - CH _{=, CH 2, NMe, Br} , H, H, H, O], [AH2552; C, = C (Me) -S -, - CH =, CH 2, NMe, CF 3, H, H, H, O], [AH2553; C, = C (Me) -S -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH2554; C, = C (Me) -S- _{, -CH =, CH 2, NMe} , Et, H, H, H, O], [AH2555; C, = C (Me) -S -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [ AH2556; C, = C (Me) -S -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2557; C, = CH-S _{-, - CH =, CH 2} , NMe, H, F, H, H, O], [AH2558; C, = CH-S -, - CH =, CH 2, NMe, Cl, F, H, H, O], [AH2559; C, = CH-S -, - CH =, CH 2, NMe, Br, F, H, H, O], [AH2560; C, = CH-S -, - CH =, CH _{2, NMe, CF 3, F} , H, H, O], [AH2561; C, = CH-S -, - CH =, CH 2, NMe, Me, F, H, H, O], [AH2562; C, = CH-S -, - CH =, CH 2, NMe, Et, F, H, H, O], [AH2563; C, = CH-S -, - CH =, CH 2, NMe, c- Pr, F, H, H, O], [AH2564; C, = CH-S -, - CH =, CH 2, NMe, OMe, F, H, H, O], [AH2565; C, = CH- S-, -CH =, C _{H 2, NMe, H, H} , F, H, O], [AH2566; C, = CH-S -, - CH =, CH 2, NMe, Cl, H, F, H, O], [AH2567; C, = CH-S -, - CH =, CH 2, NMe, Br, H, F, H, O], [AH2568; C, = CH-S -, - CH =, CH 2, NMe, CF 3 , H, F, H, O], [AH 2569; C, = CH-S-, -CH =, CH ₂ , NMe, Me, H, F, H, O], [AH 2570; C, = CH-S _{-, - CH =, CH 2} , NMe, Et, H, F, H, O], [AH2571; C, = CH-S -, - CH =, CH 2, NMe, c-Pr, H, F, H, O], [AH2572; C, = CH-S -, - CH =, CH 2, NMe, OMe, H, F, H, O], [AH2573; C, = CH-S -, - CH = , CH ₂ , NMe, H, H, H, F, O], [AH 2574; C, = CH-S-, -CH =, CH ₂ , NMe, Cl, H, H, F, O], [AH 2575 ; C, = CH-S - , - CH =, CH 2, NMe, Br, H, H, F, O], [AH2576; C, = CH-S -, - CH =, CH 2, NMe, CF ₃ , H, H, F, O], [AH 2577; C, = CH-S-, -CH =, CH ₂ , NMe, Me, H, F, O], [AH 2578; C, = CH- S -, - CH =, CH 2, NMe, Et, H, H, F, O], [AH2579; C, = CH-S -, - CH =, CH 2, NMe, c-Pr, H, H , F, O], [AH 2580; C, = CH-S-, -CH =, CH ₂ , N Me, OMe, H, F, O], [AH 2581; C, = CH-S-,-CH =, CH ₂ , NMe, H, H, H, H, H, O], [AH 2582; C, = CH-S-, -CH =, CH ₂ , N Me, Cl, H, H, H, O], [[ AH2583; C, = CH-S -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2584; C, = CH-S -, - CH =, CH 2, NMe, _{CF 3, H, H, H} , O], [AH2585; C, = CH-S -, - CH =, CH 2, NMe, Me, H, H, H, O], [AH2586; C, = CH -S -, - CH =, CH 2, NMe, Et, H, H, H, O], [AH2587; C, = CH-S -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2588; C, = CH-S -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH2589; C, -CH = CH -, = CH-N = _{, CH 2, NMe, H,} H, H, H, O], [AH2590; C, -CH = CH -, = CH-N =, CH 2, NMe, Cl, H, H, H, O], [AH2591; C, -CH = CH -, = CH-N =, CH 2, NMe, Br, H, H, H, O], [AH2592; C, -CH = CH -, = CH-N =, _{CH 2, NMe, CF 3,} H, H, H, O], [AH2593; C, -CH = CH -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2594; C, -CH = CH -, = CH-N =, CH 2, NMe, Et, H, H, H, O], [AH2595; C, -CH = CH -, = CH-N =, _{CH 2, NMe, c-Pr} , H, H, H, O], [AH2596; C, -CH = CH -, = CH-N =, CH 2, NMe, OMe, H, H, H, O] , [AH2597; C, -CH = CF -, = CH-N =, CH 2, NMe, H, H, H, H, O], [AH2598; C, -CH = CF -, = CH-N = _{, CH 2, NMe, Cl,} H, H, H, O], [AH2599; C, -CH = CF -, = = CH-N, CH 2, NMe, Br, H, H, H, O], [AH2600; C, -CH = CF -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O],

[AH2601; C, -CH = CF -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2602; C, -CH = CF -, = CH-N =, _{CH 2, NMe, Et, H} , H, H, O], [AH2603; C, -CH = CF -, = CH-N =, CH 2, NMe, c-Pr, H, H, H, O] , [AH2604; C, -CH = CF -, = CH-N =, CH 2, NMe, OMe, H, H, H, O], [AH2605; C, -CF = CH -, = CH-N = _{, CH 2, NMe, H,} H, H, H, O], [AH2606; C, -CF = CH -, = CH-N =, CH 2, NMe, Cl, H, H, H, O], [AH2607; C, -CF = CH -, = CH-N =, CH 2, NMe, Br, H, H, H, O], [AH2608; C, -CF = CH -, = CH-N =, _{CH 2, NMe, CF 3,} H, H, H, O], [AH2609; C, -CF = CH -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2610; C, -CF = CH -, = CH-N =, CH 2, NMe, Et, H, H, H, O], [AH2611; C, -CF = CH -, = CH-N =, _{CH 2, NMe, c-Pr} , H, H, H, O], [AH2612; C, -CF = CH -, = CH-N =, CH 2, NMe, OMe, H, H, H, O] , [AH2613; C, -CH = CH -, = CF-N =, CH 2, NMe, H, H, H, H, O], [AH2614; C, -CH = CH -, = CF-N = _{, CH 2, NMe, Cl,} H, H, H, O], [AH2615; C, -CH = CH -, = = CF-N, CH 2, NMe, Br, H, H, H, O], [AH2616; C, -CH = CH -, = CF-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2617; C, -CH = CH -, = CF-N = _{, CH 2, NMe, Me,} H, H, H, O], [AH2618; C, -CH = CH -, = = CF-N, CH 2, NMe, Et, H, H, H, O], [AH2619; C, -CH = CH -, = CF-N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2620; C, -CH = CH -, = CF-N _{=, CH 2, NMe, OMe} , H, H, H, O], [AH2621; C, -CH = CCl -, = CH-N =, CH 2, NMe, H, H, H, H, O] , [AH2622; C, -CH = CCl -, = CH-N =, CH 2, NMe, Cl, H, H, H, O], [AH2623; C, -CH = CCl -, = CH-N =, _{CH 2, NMe, Br, H} , H, H, O], [AH2624; C, -CH = CCl -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2625; C, -CH = CCl -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2626; C, -CH = CCl -, = CH-N =, _{CH 2, NMe, Et, H} , H, H, O], [AH2627; C, -CH = CCl -, = CH-N =, CH 2, NMe, c-Pr, H, H, H, O] , [AH2628; C, -CH = CCl -, = CH-N =, CH 2, NMe, OMe, H, H, H, O], [AH2629; C, -CCl = CH -, = CH-N = _{, CH 2, NMe, H,} H, H, H, O], [AH2630; C, -CCl = CH -, = CH-N =, CH 2, NMe, Cl, H, H, H, O], [AH2631; C, -CCl = CH -, = CH-N =, CH 2, NMe, Br, H, H, H, O], [AH2632; C, -CCl = CH -, = CH-N =, _{CH 2, NMe, CF 3,} H, H, H, O], [AH2633; C, -CCl = CH -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2634; C, -CCl = CH -, = CH-N =, CH 2, NMe, Et, H, H, H, O], [AH2635; C, -CCl = CH -, = CH-N =, _{CH 2, NMe, c-Pr} , H, H, H, O], [AH2636; C, -CCl = CH -, = CH-N =, CH 2, NMe, OMe, H, H, H, O] , [AH2637; C, -CH = CH -, = CCl-N =, CH 2, NMe, H, H, H, H, O], [AH2638; C, -CH = CH -, = CCl-N = _{, CH 2, NMe, Cl,} H, H, H, O], [AH2639; C, -CH = CH -, = = CCl-N, CH 2, NMe, Br, H, H, H, O], [AH2640; C, -CH = CH -, = CCl-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2641; C, -CH = CH -, = CCl-N = _{, CH 2, NMe, Me,} H, H, H, O], [AH2642; C, -CH = CH -, = CCl-N =, C _{H 2, NMe, Et, H} , H, H, O], [AH2643; C, -CH = CH -, = CCl-N =, CH 2, NMe, c-Pr, H, H, H, O] , [AH2644; C, -CH = CH -, = CCl-N =, CH 2, NMe, OMe, H, H, H, O], [AH2645; C, -CH = C (Me) -, = CH _{-N =, CH 2, NMe,} H, H, H, H, O], [AH2646; C, -CH = C (Me) -, = CH-N =, CH 2, NMe, Cl, H, H , H, O], [AH2647 ; C, -CH = C (Me) -, = = CH-N, CH 2, NMe, Br, H, H, H, O], [AH2648; C, -CH = C (Me) -, = CH -N =, CH 2, NMe, CF 3, H, H, H, O], [AH2649; C, -CH = C (Me) -, = CH-N =, CH _{2, NMe, Me, H,} H, H, O], [AH2650; C, -CH = C (Me) -, = = CH-N, CH 2, NMe, Et, H, H, H, O] , [AH2651; C, -CH = C (Me) -, = CH-N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2652; C, -CH = C (Me ) -, = CH-N = , CH 2, NMe, OMe, H, H, H, O], [AH2653; C, -C (Me) = CH -, = CH-N =, CH 2, NMe, H, H, H, H, O], [AH2654; C, -C (Me) = CH -, = = CH-N, CH 2, NMe, Cl, H, H, H, O], [AH2655; C, -C (Me) = CH -, = CH-N =, CH 2, NMe, Br, H, H, H, O], [AH2656; C, -C (Me) = CH -, = CH- _{N =, CH 2, NMe,} CF 3, H, H, H, O], [AH2657; C, -C (Me) = CH -, = CH-N =, CH 2, NMe, Me, H, H , H, O], [AH2658 ; C, -C (Me) = CH -, = CH-N =, CH 2, NMe, Et, H, H, H, O], [AH2659; C, -C ( Me) = CH -, = CH -N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2660; C, -C (Me) = CH -, = CH-N =, _{CH 2, NMe, OMe, H} , H, H, O], [AH2661; C, -CH = CH -, = C (Me) -N =, CH 2, NMe, H, H, H, H, O ], [AH2662; C, -CH = CH-, = C ( _{Me) -N =, CH 2,} NMe, Cl, H, H, H, O], [AH2663; C, -CH = CH -, = C (Me) -N =, CH 2, NMe, Br, H , H, H, O], [AH2664; C, -CH = CH -, = C (Me) -N =, CH 2, NMe, CF 3, H, H, H, O], [AH2665; C, -CH = CH -, = C ( Me) -N =, CH 2, NMe, Me, H, H, H, O], [AH2666; C, -CH = CH -, = C (Me) -N = , CH ₂ , NMe, Et, H, H, H, O], [AH 2667; C, -CH = CH-, = C (Me) -N =, CH ₂ , NMe, c-Pr, H, H, H, O], [AH2668; C, -CH = CH -, = C (Me) -N =, CH 2, NMe, OMe, H, H, H, O], [AH2669; C, -CH = C _{(CF 3) -, = CH} -N =, CH 2, NMe, H, H, H, H, O], [AH2670; C, -CH = C (CF 3) -, = CH-N =, CH _{2, NMe, Cl, H,} H, H, O], [AH2671; C, -CH = C (CF 3) -, = CH-N =, CH 2, NMe, Br, H, H, H, O ], [AH2672; C, -CH = C (CF 3) -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2673; C, -CH = C ( _{CF 3) -, = CH-} N =, CH 2, NMe, Me, H, H, H, O], [AH2674; C, -CH = C (CF 3) -, = CH-N =, CH 2 , NMe, Et, H, H , H, O], [AH2675; C, -CH = C (CF 3) -, = CH-N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2676; C, -CH = C (CF 3) -, = CH-N =, CH 2, NMe, OMe, H, H, H, O], [AH2677; C, -C (CF 3 ) = CH -, = CH- N =, CH 2, NMe, H, H, H, H, O], [AH2678; C, -C (CF 3) = CH -, = CH-N =, CH 2 , NMe, Cl, H, H , H, O], [AH2679; C, -C (CF 3) = CH -, = = CH-N, CH 2, NMe, Br, H, H, H, O] , [AH2680; C, -C ( CF 3) = CH -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2681; C, -C (CF 3) = CH -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2682; C, -C (CF 3) = CH -, = CH-N =, CH 2, NMe, Et, H, H, H, O], [AH2683; C, -C (CF 3) = CH -, = = CH-N, CH 2, NMe, c-Pr, H, H, H, O], [AH2684; C, -C (CF 3) = CH -, = CH-N =, CH 2, NMe, OMe, H, H, H, O], [AH2685; C, -CH = CH -, = C _{(CF 3) -N =, CH} 2, NMe, H, H, H, H, O], [AH2686; C, -CH = CH -, = C (CF 3) -N =, CH 2, NMe, Cl, H, H, H, O], [AH2687; C, -CH = CH -, = C (CF 3) -N =, CH 2, NMe, Br, H, H, H, O], [AH2688 ; C, -CH = CH -, = = C (CF 3) -N, CH 2, NMe, CF 3, H, H, H, O], [AH2689; C, -CH = CH -, = C ( _{CF 3) -N =, CH 2} , NMe, Me, H, H, H, O], [AH2690; C, -CH = CH -, = C (CF 3) -N =, CH 2, NMe, Et , H, H, H, O ], [AH2691; C, -CH = CH -, = C (CF 3) -N =, CH 2, NMe, c-Pr, H, H, H, O], [ AH2692; C, -CH = CH - , = C (CF 3) -N =, CH 2, NMe, OMe, H, H, H, O], [AH2693; C, = CH-CH = CH -, - _{C (Me) =, CH 2} , NMe, H, H, H, H, O], [AH2694; C, = CH-CH = CH -, - C (Me) =, CH 2, NMe, Cl, H , H, H, O], [AH2695; C, = CH-CH = CH -, - C (Me) =, CH 2, NMe, Br, H, H, H, O], [AH2696; C, = CH-CH = CH -, - C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH2697; C, = CH-CH = CH -, - C (Me) = , CH ₂ , NMe, Me, H, H, H, O, [AH 2698; C, = CH-CH = CH-, -C (Me) =, CH ₂ , NMe, Et, H, H, H, H, O], [AH2699; C, = CH-CH = CH -, - C (Me) =, CH 2, NMe, c-Pr, H, H, H, O], [AH2700; C, = CH-CH = CH -, - C (Me) =, CH 2, NMe, OMe, H, H, H, O],

[AH 2701; C, = CH-CH = CF-, -C (Me) =, CH ₂ , N Me, H, H, H, H, O], [AH 2702; C, = CH-CH = CF-,- _{C (Me) =, CH 2} , NMe, Cl, H, H, H, O], [AH2703; C, = CH-CH = CF -, - C (Me) =, CH 2, NMe, Br, H , H, H, O], [AH 2704; C, = CH-CH = CF-, -C (Me) =, CH ₂ , N Me, CF ₃ , H, H, H, O], [AH 2 705; C, = CH-CH = CF -, - C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH2706; C, = CH-CH = CF -, - C (Me) = , CH ₂ , NMe, Et, H, H, H, O], [AH 2707; C, = CH-CH = CF-, -C (Me) =, CH ₂ , NMe, c-Pr, H, H, H, O], [AH 2 708; C, = CH-CH = CF-, -C (Me) =, CH ₂ , N Me, OMe, H, H, H, O], [AH 2709; C, = CH-CF = CH -, - C (Me ) =, CH 2, NMe, H, H, H, H, O], [AH2710; C, = CH-CF = CH -, - C (Me) =, CH 2, NMe, Cl, H, H, H, O], [AH2711; C, = CH-CF = CH -, - C (Me) =, CH 2, NMe, Br, H, H, H, O], [ AH2712; C, = CH-CF = CH -, - C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH2713; C, = CH-CF = CH -, - _{C (Me) =, CH 2} , NMe, Me, H, H, H, O], [AH2714; C, = CH-CF = CH -, - C (Me) =, CH 2, NMe, Et, H , H, H, O], [AH2715; C, = CH-CF = CH -, - C (Me) =, CH 2, NMe, c-Pr, H, H, H, O], [AH2716; C , = CH-CF = CH - , - C (Me) =, CH 2, NMe, OMe, H, H, H, O], [AH2717; C, = CF-CH = CH -, - C (Me) _{=, CH 2, NMe, H} , H, H, H, O], [AH2718; C, = CF-CH = CH -, - C (Me) =, CH 2, NMe, Cl, H, H, H , O], [AH2719; C , = CF-CH = CH -, - C (Me) =, CH 2, NMe, Br, H, H, H, O], [AH2720; C, = CF-CH = CH-,- _{C (Me) =, CH 2} , NMe, CF 3, H, H, H, O], [AH2721; C, = CF-CH = CH -, - C (Me) =, CH 2, NMe, Me, H, H, H, O] , [AH2722; C, = CF-CH = CH -, - C (Me) =, CH 2, NMe, Et, H, H, H, O], [AH2723; C, = CF-CH = CH -, - C (Me) =, CH 2, NMe, c-Pr, H, H, H, O], [AH2724; C, = CF-CH = CH -, - C (Me _{) =, CH 2, NMe,} OMe, H, H, H, O], [AH2725; C, = CH-CH = CH -, - C (Br) =, CH 2, NMe, H, H, H, H, O], [AH2726; C, = CH-CH = CH -, - C (Br) =, CH 2, NMe, Cl, H, H, H, O], [AH2727; C, = CH-CH = CH -, - C (Br ) =, CH 2, NMe, Br, H, H, H, O], [AH2728; C, = CH-CH = CH -, - C (Br) =, CH 2, _{NMe, CF 3, H, H} , H, O], [AH2729; C, = CH-CH = CH -, - C (Br) =, CH 2, NMe, Me, H, H, H, O], [AH2730; C, = CH- CH = CH -, - C (Br) =, CH 2, NMe, Et, H, H, H, O], [AH2731; C, = CH-CH = CH -, - _{C (Br) =, CH 2} , NMe, c-Pr, H, H, H, O], [AH2732; C, = CH-CH = CH -, - C (Br) =, CH 2, NMe, OMe , H, H, H, O], [AH 2733; C, = CH-CH = CH-, -C (Cl) =, CH ₂ , N Me, H, H, H, H, O], [AH 2734; C , = CH-CH = CH - , - C (Cl) =, CH 2, NMe, Cl, H, H, H, O], [AH2735; C, = CH-CH = CH -, - C (Cl) _{=, CH 2, NMe, Br} , H, H, H, O], [AH2736; C, = CH-CH = CH -, - C (Cl) =, CH 2, NMe, CF 3, H, H, H, O], [AH 2 737; C, = CH-CH = CH-, -C (Cl) =, CH ₂ , NMe, Me, H, H, H, O], [AH 2738; C, = CH-CH = CH -, - C (Cl ) =, CH 2, NMe, Et, H, H, H, O], [AH2739; C, = CH-CH = CH -, - C (Cl) =, CH 2, NMe, c -Pr, H, H, H, O], [AH 2740; C, = CH-CH = CH-,-C (Cl) =, CH ₂ , N Me, OMe, H, H, H, O], [AH 274 1 ; C, = CH-C ( Me) = CH -, - C (Me) =, CH 2, NMe, H, H, H, H, O], [AH2742; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, NMe, Cl, H, H, H, O], [AH2743; C, = CH-C (Me) = CH -, - C (Me) =, CH _{2, NMe, Br, H,} H, H, O], [AH2744; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, NMe, CF 3, H, H, H, O], [AH2745; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, NMe, Me, H, H, H, O], [AH2746; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, NMe, Et, H, H, H, O], [AH2747; C, = CH-C (Me) = CH -, - _{C (Me) =, CH 2} , NMe, c-Pr, H, H, H, O], [AH2748; C, = CH-C (Me) = CH -, - C (Me) =, CH 2, NMe, OMe, H, H, H, O], [AH2749; C, = CH-CH = CH -, - C (CF 3) =, CH 2, NMe, H, H, H, H, O], [AH2750; C, = CH- CH = CH -, - C (CF 3) =, CH 2, NMe, Cl, H, H, H, O], [AH2751; C, = CH-CH = CH-, _{-C (CF 3) =, CH} 2, NMe, Br, H, H, H, O], [AH2752; C, = CH-CH = CH -, - C (CF 3) =, CH 2, NMe, _{CF 3, H, H, H} , O], [AH2753; C, = CH-CH = CH -, - C (CF 3) =, CH 2, NMe, Me, H, H, H, O], [ AH2754; C, = CH-CH = CH -, - C (CF 3) =, CH 2, NMe, Et, H, H, H, O], [AH2755; C, = CH-CH = CH -, - _{C (CF 3) =, CH} 2, NMe, c-Pr, H, H, H, O], [AH2756; C, = CH-CH = CH -, - C (CF 3) =, CH 2, NMe , OMe, H, H, H , O], [AH2757; C, -CH = CH -, = CH-N =, CH 2, NMe, H, H, H, H, O], [AH2758; C, -CH = C H -, = CH-N = , CH 2, NMe, Cl, H, H, H, O], [AH2759; C, -CH = CH -, = CH-N =, CH 2, NMe, Br, H , H, H, O], [AH2760; C, -CH = CH -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2761; C, -CH = CH -, = CH-N = , CH 2, NMe, Me, H, H, H, O], [AH2762; C, -CH = CH -, = CH-N =, CH 2, NMe, Et, H , H, H, O], [AH2763; C, -CH = CH -, = CH-N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2764; C, -CH = CH -, = CH-N =, CH 2, NMe, OMe, H, H, H, O], [AH2765; C, -CH = CF -, = CH-N =, CH 2, NMe, H, H, H, H, O] , [AH2766; C, -CH = CF -, = = CH-N, CH 2, NMe, Cl, H, H, H, O], [AH2767; C, -CH = CF -, = = CH-N , CH 2, NMe, Br, H, H, H, O], [AH2768; C, -CH = CF -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O] , [AH2769; C, -CH = CF -, = = CH-N, CH 2, NMe, Me, H, H, H, O], [AH2770; C, -CH = CF -, = CH-N = , CH 2, NMe, Et, H, H, H, O], [AH2771; C, -CH = CF -, = CH-N =, CH 2, NMe, c-Pr , H, H, H, O ], [AH2772; C, -CF = CH -, = CH-N =, CH 2, NMe, H, H, H, H, O], [AH2773; C, -CF = CH -, = CH-N =, CH 2, NMe, Cl, H, H, H, O], [AH2774; C, -CF = CH -, = CH-N =, CH 2, NMe, Br, H, H, H, O] , [AH2775; C, -CF = CH -, = CH-N =, CH 2, NMe, CF 3, H, H, H, O], [AH2776; C, -CF = CH -, = CH-N =, CH 2, NMe, Me, H, H, H, O], [AH2777; C, -CF = CH -, = CH-N =, CH 2, NMe, Et, H, H, H, O] , [AH2778; C, -CF = CH -, = CH-N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2779; C, - CF = CH -, = CH-N = , CH 2, NMe, OMe, H, H, H, O], [AH2780; C, -CH = CH -, = CF-N =, CH 2, NMe, H, H , H, H, O], [AH2781; C, -CH = CH -, = CF-N =, CH 2, NMe, Cl, H, H, H, O], [AH2782; C, -CH = CH -, = CF-N =, CH 2, NMe, Br, H, H, H, O], [AH2783; C, -CH = CH -, = CF-N =, CH 2, NMe, CF 3, H , H, H, O], [AH2784; C, -CH = CH -, = CF-N =, CH 2, NMe, Me, H, H, H, O], [AH2785; C, -CH = CH -, = CF-N =, CH 2, NMe, Et, H, H, H, O], [AH2786; C, -CH = CH -, = CF-N =, CH 2, NMe, c-Pr, H, H, H, O] , [AH2787; C, -CH = CH -, = CF-N =, CH 2, NMe, OMe, H, H, H, O], [AH2788; C, = CH- CH = CH -, - CH = , CH 2, NMe, H, H, H, H, O], [AH2789; C, = CH-CH = CH -, - CH =, CH 2, NMe, Cl, H , H, H, O], [AH2790; C, = CH-CH = CH -, - CH =, CH 2, NMe, Br, H, H, H, O], [AH2791; C, = CH-CH = CH -, - CH =, CH 2, NMe, CF 3, H, H, H, O], [AH2792; C, = CH-CH = CH -, - CH =, CH 2, NMe, Me, H , H, H, O], [AH 2793; C, = CH-CH = CH-, -CH =, CH ₂ , NMe, Et, H, H, H, O], [AH 2794; C, = CH-CH = CH -, - CH =, CH 2, NMe, c-Pr, H, H, H, O], [AH2795; C, = CH-CH = CH -, - CH =, CH 2, NMe, OMe, H, H, H, O], [AH 2796; C, = CH-CH = CH-,-N =, CH ₂ , N Me, H, H, H, H, O], [AH 2 797; C, = CH- CH = CH -, - N = , CH 2, NMe, Cl, H, H, H, O], [AH2798; C, = CH-CH = CH -, - N =, CH 2, NMe, Br, H , H, H, O], [AH2799; C, = CH-CH = CH -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH280 0; C, = CH-CH = CH -, - N =, CH 2, NMe, Me, H, H, H, O],

[AH2801; C, = CH- CH = CH -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2802; C, = CH-CH = CH -, - N =, _{CH 2, NMe, c-Pr} , H, H, H, O], [AH2803; C, = CH-CH = CH -, - N =, CH 2, NMe, OMe, H, H, H, O] , [AH2804; C, = CH -C (Me) = CH -, - N =, CH 2, NMe, H, H, H, H, O], [AH2805; C, = CH-C (Me) = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2806; C, = CH-C (Me) = CH -, - N =, CH 2, NMe, Br, H, H, H, O], [AH 2 807; C, = CH-C (Me) = CH-,-N =, CH ₂ , N Me, CF ₃ , H, H, O, [AH 2 808; C , = CH-C (Me) = CH -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2809; C, = CH-C (Me) = CH -, - N _{=, CH 2, NMe, Et} , H, H, H, O], [AH2810; C, = CH-C (Me) = CH -, - N =, CH 2, NMe, c-Pr, H, H , H, O], [AH 2811; C, = CH-C (Me) = CH-,-N =, CH ₂ , N Me, OMe, H, H, H, O], [AH 2812; Me) -CH = CH -, - N =, CH 2, NMe, H, H, H, H, O], [AH2813; C, = C (Me) -CH = CH -, - N =, CH 2 , NMe, Cl, H, H , H, O], [AH2814; C, = C (Me) -CH = CH -, - N =, CH 2, NMe, Br, H, H, H, O], [AH2815; C, = C ( Me) -CH = CH -, - N =, CH 2, NMe, CF 3, H, H, H, O], [AH2816; C, = C (Me) -CH = CH -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2817; C, = C (Me) -CH = CH -, - N =, CH 2, NMe, Et, H, H, H, O] , [AH2818; C, = C (Me) -CH = CH -, - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2819; C, = C (Me) -CH = CH -, - N =, CH 2, NMe, OMe, H, H, H, O], [AH2820; C, = CH-C (CF 3) = CH-, _{-N =, CH 2, NMe,} H, H, H , H, O], [AH2821 ; C, = CH-C (CF 3) = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2822; C, = CH _{-C (CF 3) = CH -} , - N =, CH 2, NMe, Br, H, H, H, O], [AH2823; C, = CH-C (CF 3) = CH -, - N = _{, CH 2, NMe, CF 3} , H, H, H, O], [AH2824; C, = CH-C (CF 3) = CH -, - N =, CH 2, NMe, Me, H, H, H, O], [AH2825; C, = CH-C (CF 3) = CH -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2826; C, = CH- _{C (CF 3) = CH -} , - N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2827; C, = CH-C (CF 3) = CH -, - N _{=, CH 2, NMe, OMe} , H, H, H, O], [AH2828; C, = C (CF 3) -CH = CH -, - N =, CH 2, NMe, H, H, H, H, O], [AH2829; C, = C (CF 3) -CH = CH -, - N =, CH 2, NMe, Cl, H, H, H, O], [AH2830; C, = C ( _{CF 3) -CH = CH -,} - N =, CH 2, NMe, Br, H, H, H, O], [AH2831; C, = C (CF 3) -CH = CH -, - N =, _{CH 2, NMe, CF 3,} H, H, H, O], [AH2832; C, = C (CF 3) -CH = CH -, - N =, CH 2, NMe, Me, H, H, H , O], [AH2833; C , = C (CF 3) -CH = CH -, - N =, CH 2, NMe, Et, H, H, H, O], [AH2834; C, = C (CF _{3) -CH = CH -, -} N =, CH 2, NMe, c-Pr, H, H, H, O], [AH2835; C, = C (CF 3) -CH = CH -, - N = , CH ₂ , NMe, OMe, H, H, H, O], [AH 2836; C, -CH = CH-, = CH-C (Me) =, -CH = CH-,-, H, H, H , H, O], [AH 2837; C, -CH = CH-, = CH-C (Me) =, -CH = CH-,-, Cl, H, H, H, O], [AH 2838; C, -CH = CH-, = CH-C (Me) =, -CH = CH-,-, Br, H, H, H, O], [AH2839; C, -CH = CH-, = CH-C ( Me) =, -CH = CH- _{, -, CF 3, H,} H, H, O], [AH2840; C, -CH = CH -, = CH-C (Me) =, - CH = CH -, -, Me, H, H, H , O], [AH2841; C, -CH = CH-, = CH-C (Me) =, -CH = CH-,-, Et, H, H, H, O], [AH2842; C, -CH = CH-, = CH-C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 2843; C, -CH = CH-, = CH-C ( Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH 2844; C, -CH = CF-, = CH-C (Me) =, -CH = CH-,- , H, H, H, H, O], [AH 2845; C, -CH = CF-, = CH-C (Me) =, -CH = CH-,-, Cl, H, H, H, O] , [AH2846; C, -CH = CF-, = CH-C (Me) =, -CH = CH-,-, Br, H, H, H, O], [AH 2847; C, -CH = CF- , = CH-C (Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH2848; C, -CH = CF -, = CH-C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH 2849; C, -CH = CF-, = CH-C (Me) =, -CH = CH-,-, Et, H , H, H, O], [AH 2850; C, -CH = CF-, = CH-C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [[ C, -CH = CF-, = CH-C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH2852; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, H, H, H, H, O], [AH2853; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, Cl, H, H, H, H, O], [AH 2 854; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, Br, H, H, H, O], [AH2855; C, -CF = CH -, = CH-C (Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH2856; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH 2857; C, -CF = CH-, = CH-C ( Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 2858; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,- , c-Pr, H, H, H, O], [ AH 2859; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH 2860; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, H, H, H, H, O], [AH2861; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, Cl, H, H, H, H, O], [AH2862; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, Br, H, H, H, O], [AH2863; C, -CF = CH -, = CH-C (Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH2864; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH 2865; C, -CF = CH-, = CH-C ( Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 2866; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,- , c-Pr, H, H, H, O], [AH 2867; C, -CF = CH-, = CH-C (Me) =, -CH = CH-,-, OMe, H, H, H, H O], [AH 2868; C, -CH = CH-, = CF-C (Me) =, -CH = CH-,-, H, H, H, H, O], [AH 2869; C, -CH = CH-, = CF-C (Me) =, -CH = CH-,-, Cl, H, H, H, O], [AH 2870; C, -CH = CH-, = CF-C (Me) = , -CH = CH -, -, Br, H, H, H, O], [AH2871; C, -CH = CH -, = CF-C (Me) =, - CH = CH -, -, CF 3 , H, H, H, O], [AH2872; C, -CH = CH-, = CF-C (Me) =, -CH = CH-,-, Me, H, H, H, O], [[ C, -CH = CH-, = CF-C (Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 2874; C, -CH = CH-, = CF-C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 2875; C, -CH = CH-, = CF-C (Me) =,- CH = CH-,-, OMe, H, H, H, O], [AH 2876; C, -CH = CH-, = CH-CBr =, -CH = CH-,-, H, H, H, H C, -CH = CH-, = CH-CBr =, -CH = CH-,-, Cl, H, H, H, O], [AH 2878; C, -CH = CH- , = CH-CBr = , -CH = CH-,-, Br, H, H, H, O], [AH 2879; C, -CH = CH-, = CH-CBr =, -CH = CH-,-, CF ₃ , H, H, H, O], [AH 2 880; C, -CH = CH-, = CH-CBr =, -CH = CH-,-, Me, H, H, H, O], [AH2881; C, -CH = CH-, = CH-CBr =, -CH = CH-,-, Et, H, H, H, O], [AH2882; C, -CH = CH-, = CH-CBr =, -CH = CH -,-, c-Pr, H, H, H, O], [AH2883; C, -CH = CH-, = CH-CBr =, -CH = CH-,-, OMe, H, H, H, O], [AH2884; C, -CH = CH-, = CH-CCl =, -CH = CH-,-, H, H, H, H, O], [AH2885; C, -CH = CH-, = CH-CCl =, -CH = CH-,-, Cl, H, H, H, O], [AH2886; C, -CH = CH-, = CH-CCl =, -CH = CH-,-, br, H, H, H, O], [AH2887; C, -CH = CH -, = CH-CCl =, - CH = CH -, -, CF 3, H, H, H, O], [AH2888 C, -CH = CH-, = CH-CCl =, -CH = CH-,-, Me, H, H, H, O], [AH2889; C, -CH = CH-, = CH-CCl = , -CH = CH-,-, Et, H, H, H, O], [AH 2890; C, -CH = CH-, = CH-CCl =, -CH = CH-,-, c-Pr, H , H, H, O], [AH2891; C, -CH = CH-, = CH-CCl =, -CH = CH-,-, OMe, H, H, H, O], [AH2892; C,- C (Me) = CH-, = CH-C (Me) =, -CH = CH-,-, H, H, H, H, O], [AH 2893; C, -C (Me) = CH-, = CH-C (Me) =, -CH = CH-,-, Cl, H, H, H, O], [AH 2894; C, -C (Me) = CH-, = CH-C (Me) = , -CH = CH-,-, Br, H, H, H, O], [AH 2895; C, -C (Me) = CH-, = CH-C (Me) =, -CH = CH-,- _{, CF 3, H, H,} H, O], [AH2896; C, -C (Me) = CH -, = CH-C (Me) =, - CH = CH -, -, Me, H, H, H, O], [AH 2897; C, -C (Me) = CH-, = CH-C (Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 2898; C, -C (Me) = CH-, = CH-C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH2899; C, -C (Me) = CH-, = CH-C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH 2900; C, -CH = CH-, = CH-C (CF ₃ ) =, -CH = CH-,-, H, H, H, H, O],

[AH2901; C, -CH = CH -, = CH-C (CF 3) =, - CH = CH -, -, Cl, H, H, H, O], [AH2902; C, -CH = CH- _{, = CH-C (CF 3} ) =, - CH = CH -, -, Br, H, H, H, O], [AH2903; C, -CH = CH -, = CH-C (CF 3) = , -CH = CH -, -, CF 3, H, H, H, O], [AH2904; C, -CH = CH -, = CH-C (CF 3) =, - CH = CH -, -, Me, H, H, H, O], [AH2905; C, -CH = CH -, = CH-C (CF 3) =, - CH = CH -, -, Et, H, H, H, O] , [AH 2906; C, -CH = CH-, = CH-C (CF ₃ ) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 2907; C, -CH = CH-, = CH-C (CF ₃ ) =, -CH = CH-,-, OMe, H, H, H, O], [AH 2908; C, -CH = CH-, = CH-C (Et ) =, -CH = CH-,-, H, H, H, H, O], [AH 2909; C, -CH = CH-, = CH-C (Et) =, -CH = CH-,-, Cl, H, H, H, O], [AH 2910; C, -CH = CH-, = CH-C (Et) =, -CH = CH-,-, Br, H, H, H, O], [AH2911; C, -CH = CH -, = = CH-C (Et), - CH = CH -, -, CF 3, H, H, H, O], [AH2912; C, -CH = CH- , = CH-C (Et) =, -CH = CH-,-, Me, H, H, H, O], [AH 2913; C, -CH = CH-, = CH-C (Et) =,- CH = CH-,-, Et, H, H, H, O], [AH 2914; C, -CH = CH-, = CH-C (Et) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 2915; C, -CH = CH-, = CH-C (Et) =, -CH = CH-,-, OMe, H, H, H, O], [AH 2916 C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, H, H, H, H, O], [AH 2917; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, Cl, H, H, H, O], [AH 2918; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, Br, H, H, H, O], [AH 2919; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,- , CF ₃ , H, H, H, O], [AH 2920; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, Me, H, H, H, O] , [AH 2921; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, Et, H, H, H, O], [AH 2922; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 2923; C, -CH = CH-, = CH-C (c-Pr) =, -CH = CH-,-, OMe, H, H, H, O], [AH 2924; N, -CH = CH-, -N =, -CH = CH-,-, H , H, H, H, O], [AH 2925; N, -CH = CH-, -N =, -CH = CH-,-, F, H, H, H, O], [AH 2926; N,- CH = CH-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 2927; N, -CH = CH-, -N =, -CH = CH-,- , Br, H, H, H, O], [AH 2 928; N, -CH = CH-, -N =, -CH = CH-,-, Me, H, H, H] O, [AH 2 929; N , -CH = CH-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 2930; N, -CH = CH-, -N =, -CH = CH- ,-, Pr, H, H, H, O, [AH2931; N, -CH = CH-, -N =, -CH = CH-,-, i-Pr, H, H, H, O], [AH2932; N, -CH = CH-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH2933; N, -CH = CH-, -N = , -CH = CH-,-, c-Bu, H, H, H, O], [AH 2934; N, -CH = CH-, -N =, -CH = CH-,-, OMe, H, H , H, O], [AH 2935; N, -CH = CH-, -N =, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH 2936; N, -CH = CH-, -N =, -CH = CH-,-, SMe, H, H, H, O], [AH 2937; N, -CH = CH-, -N =, -CH = CH-,-, Set , H, H, H, O ], [AH2938; N, -CH = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH2939; N, -CH = CH -, - N = , - CH = CH -, -, CHF 2, H, H, H, O], [AH2940; N, -CH = CH -, - N =, - CH = CH- ,-, OCF ₃ , H, H, H, O], [AH 29 41; N, -CH = CH - , - N =, - CH = CH -, -, OCHF 2, H, H, H, O], [AH2942; N, -CH = CH -, - N =, - CH = CH -, -, CH = CH 2, H, H, H, O], [AH2943; N, -CH = CH -, - N =, - CH = CH -, -, C (Me) = CH ₂ , H, H, H, O], [AH2944; N, -CH = CH-, -N =, -CH = CH-,-, CH = CHMe, H, H, H, O], [AH 2945; N, -CH = CH-, -N =, -CH = CH-,-, C≡CH, H, H, H, O], [AH 2946; N, -CH = CH-, -N =, -CH = CH-,-, C≡CMe, H, H, H, O], [AH2947; N, -CH = CH-, -N =, -CH = CH-,-, CN, H, H, H, H O, [AH2948; N, -CH = CF-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 2949; N, -CH = CF-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 2950; N, -CH = CF-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH2951; N, -CH = CF -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH2952; N, -CH = CF- , -N =, -CH = CH-,-, Me, H, H, H, O], [AH 2953; N, -CH = CF-, -N =, -CH = CH-,-, Et, H , H, H, O], [AH 2 954; N, -CH = CF-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 2 955; N,- CH = CF-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH2956; N, -CF = CH-, -N =, -CH = CH-,- , H, H, H, H, O], [AH 2957; N, -CF = CH-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH2958; N , -CF = CH-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH2959; N, -CF = CH-, -N =, -CH = CH- _{, -, CF 3, H,} H, H, O], [AH2960; N, -CF = CH -, - N =, - CH = CH -, -, Me, H, H, H, O], [ AH 2961; N, -CF = CH-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH2962; N, -CF = CH-, -N =, -CH = CH-,-, c-Pr, H, H , H, O], [AH2963; N, -CF = CH-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH2964; N, -CH = CCl- , -N =, -CH = CH-,-, H, H, H, H, O], [AH 2965; N, -CH = CCl-, -N =, -CH = CH-,-, Cl, H , H, H, O], [AH 2966; N, -CH = CCl-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH 2967; N, -CH = CCl -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH2968; N, -CH = CCl -, - N =, - CH = CH -, -, Me, H, H, H, O], [AH2969; N, -CH = CCl-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 2970; N, -CH = CCl-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH2971; N, -CH = CCl-, -N =, -CH = CH -,-, OMe, H, H, H, O], [AH 2972; N, -CCl = CH-, -N =, -CH = CH-,-, H, H, H, H, O], [[ AH 2 973; N, -CCl = CH-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 2974; N, -CCl = CH-, -N =, -CH = CH -, -, Br, H, H, H, O], [AH2975; N, -CCl = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O N, -CCl = CH-, -N =, -CH = CH-,-, Me, H, H, H, O], [AH2977; N, -CCl = CH-, -N =] , -CH = CH-,-, Et, H, H, H, O], [AH2978; N, -CCl = CH-, -N =, -CH = CH-,-, c-Pr, H, H , H, O], [AH2979; N, -CCl = CH-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 2980; N, -CH = C ( Me)-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 2981; N, -CH = C (Me)-, -N =, -CH = CH- ,-, Cl, H, H, H, O, [AH2982; N, -CH = C (Me)-, -N =, -CH = CH-,-, Br, H, H, H, O] , [AH2983; N, -CH = C (Me) -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH2984; N, -CH = C (Me ) -, -N =, -CH = CH-,-, Me, H, H, H, O], [AH 2985; N, -CH = C (Me)-, -N =, -CH = CH-,- , Et, H, H, H, O], [AH2986; N, -CH = C (Me)-, -N =, -CH = CH-,-, c-Pr, H, H, H, O] , [AH2987; N, -CH = C (Me)-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH2988; N, -C (Me) = CH -, -N =, -CH = CH-,-, H, H, H, H, O], [AH2989; N, -C (Me) = CH-, -N =, -CH = CH-,- , Cl, H, H, H, O], [AH 2 990; N, -C (Me) = CH-, -N =, -CH = CH-,-, Br, H, H, H, O], [[ AH 299 1; N, -C (Me) = CH-, -N =, -CH = CH-,-, CF ₃ , H, H, H, O], [AH 299 2; N, -C (Me) = CH- , -N =, -CH = CH-,-, Me, H, H, H, O], [AH2993; N, -C (Me) = CH-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 2994; N, -C (Me) = CH-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH2995; N, -C (Me) = CH-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH2996; N, -CH = CH-, -N =, -CH = CH-,-, H, F, H, H, O], [AH 2997; N, -CH = CH-, -N =, -CH = CH-,-, Cl, F, H, H, O], [AH2998; N, -CH = CH-, -N =, -CH = CH-,-, Br, F, H, H, O], [AH 2999; N, -CH = CH-, -N =, - CH = CH - , -, CF 3, F, H, H, O], [AH3000; N, -CH = CH -, - N =, - CH = CH -, -, Me, F , H, H, O],

[AH 3001; N, -CH = CH-, -N =, -CH = CH-,-, Et, F, H, H, O], [AH3002; N, -CH = CH-, -N =,- CH = CH-,-, c-Pr, F, H, H, O], [AH 3003; N, -CH = CH-, -N =, -CH = CH-,-, OMe, F, H, H , O], [AH3004; N, -CH = CH-, -N =, -CH = CH-,-, H, H, F, H, O], [AH3005; N, -CH = CH-,- N =, -CH = CH-,-, Cl, H, F, H, O], [AH 3006; N, -CH = CH-, -N =, -CH = CH-,-, Br, H, F , H, O], [AH3007 ; N, -CH = CH -, - N =, - CH = CH -, -, CF 3, H, F, H, O], [AH3008; N, -CH = CH -, -N =, -CH = CH-,-, Me, H, F, H, O], [AH 3009; N, -CH = CH-, -N =, -CH = CH-,-, Et, H, F, H, O], [AH 3010; N, -CH = CH-, -N =, -CH = CH-,-, c-Pr, H, F, H, O], [AH 3011; N, -CH = CH-, -N =, -CH = CH-,-, OMe, H, F, H, O], [AH 3012; N, -CH = CH-, -N =, -CH = CH-, -, H, H, H, F, O], [AH 3013; N, -CH = CH-, -N =, -CH = CH-,-, Cl, H, H, F, O], [AH 3014; N, -CH = CH-, -N =, -CH = CH-,-, Br, H, H, F, O], [AH 3015; N, -CH = CH-, -N =, -CH = CH _{-, -, CF 3, H} , H, F, O], [AH3016; N, -CH = CH -, - N =, - CH = CH -, -, Me, H, H, F, O], [AH3017; N, -CH = CH-, -N =, -CH = CH-,-, Et, H, H, F, O], [AH3018; N, -CH = CH-, -N =,- CH = CH-,-, c-Pr, H, H, F, O], [AH 3019; N, -CH = CH-, -N =, -CH = CH-,-, OMe, H, H, F , O], [AH 3020; C, = CH-S-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 3021; C, = CH-S-,- N =, -CH = CH-,-, F, H, H, H, O], [AH3022; C, = CH-S-, -N =, -CH = CH-,-, Cl, H, H , H, O], [AH 3023; C, = CH-S-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH 3024; C, = CH-S-, -N =, -CH = CH-,-, Me, H, H, H, O] , [AH3025; C, = CH-S-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH3026; C, = CH-S-, -N =, -CH = CH-,-, Pr, H, H, H, O], [AH3027; C, = CH-S-, -N =, -CH = CH-,-, i-Pr, H, H, H H, O], [AH3028; C, = CH-S-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3029; C, = CH-S -, -N =, -CH = CH-,-, c-Bu, H, H, H, O], [AH3030; C, = CH-S-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3031; C, = CH-S-, -N =, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH 3032; C, = CH-S-, -N =, -CH = CH-,-, SMe, H, H, H, O], [AH 3033; C, = CH-S-, -N =, -CH = CH -, -, Set, H, H, H, O], [AH3034; C, = CH-S -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3035; C, = CH- S -, - N =, - CH = CH -, -, CHF 2, H, H, H, O], [AH3036; C, = CH-S -, - N =, -CH = CH -, -, OCF 3, H, H, H, O], [AH3037; C, = CH-S -, - N =, - CH = CH -, -, OCHF 2, H, H, H, O], [AH3038; C, = CH-S -, - N =, - CH = CH -, -, CH = CH 2, H, H, H, O], [AH3039; C, = CH- S -, - N =, - CH = CH -, -, C (Me) = CH 2, H, H, H, O], [AH3040; C, = CH-S -, - N =, - CH = CH-,-, CH = CHMe, H, H, H, O], [AH3041; C, = CH-S-, -N =, -CH = CH-,-, C≡CH, H, H, H , O], [AH3042; C, = CH-S-, -N =, -CH = CH-,-, C≡CMe, H, H, H, O], [AH3043; C, = C (CF ₃ ) -S-, -N =, -CH = CH-,-, H, H, H, H, O], [AH3044; C, = C (CF ₃ ) -S-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3045; C, _{= C (CF 3) -S -} , - N =, - CH = CH -, -, Br, H, H, H, O], [AH3046; C, = C (CF 3) -S -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3047; C, = C (CF 3) -S -, - N =, - CH = CH -, -, Me , H, H, H, O ], [AH3048; C, = C (CF 3) -S -, - N =, - CH = CH -, -, Et, H, H, H, O], [AH3049 _{; C, = C (CF 3} ) -S -, - N =, - CH = CH -, -, c-Pr, H, H, H, O], [AH3050; C, = C (CF 3) - S-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH3051; C, = CF-S-, -N =, -CH = CH-,-, H , H, H, H, O], [AH3052; C, = CF-S-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH3053; C, = CF-S-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH3054; C, = CF-S-, -N =, -CH = CH-,- _{, CF 3, H, H,} H, O], [AH3055; C, = CF-S -, - N =, - CH = CH -, -, Me, H, H, H, O], [AH3056; C, = CF-S-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH3057; C, = CF-S-, -N =, -CH = CH -,-, c-Pr, H, H, H, O], [AH3058; C, = CF-S-, -N =, -CH = CH-,-, OMe, H, H, H, O] , [AH3059; C, = CCl-S-, -N =, -CH = CH-,-, H, H, H, H, O], [AH3060; C, = CCl-S-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH3061; C, = CCl-S-, -N =, -CH = CH-,-, Br, H, H, H, H O], [AH3062; C, = CCl-S -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3063; C, = CCl-S -, - N =, -CH = CH-,-, Me, H, H, H, O], [AH 3064; C, = CCl-S-, -N =, -CH = CH-,-, Et, H, H , H, O], [AH 3065; C, = CCl-S-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3066; C, = CCl- S-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH3 C, = C (Me) -S-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 3068; C, = C (Me) -S-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH3069; C, = C (Me) -S-, -N =, -CH = CH-,-, Br , H, H, H, O ], [AH3070; C, = C (Me) -S -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3071 C, = C (Me) -S-, -N =, -CH = CH-,-, Me, H, H, H, O], [AH3072; C, = C (Me) -S-,- N =, -CH = CH-,-, Et, H, H, H, O], [AH3073; C, = C (Me) -S-, -N =, -CH = CH-,-, c- Pr, H, H, H, O], [AH 3074; C, = C (Me)-S-,-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3075 C, = CH-S-, -N =, -CH = CH-,-, H, F, H, H, O], [AH3076; C, = CH-S-, -N =, -CH = CH-,-, Cl, F, H, H, O], [AH3077; C, = CH-S-, -N =, -CH = CH-,-, Br, F, H, H, O], [AH3078; C, = CH- S -, - N =, - CH = CH -, -, CF 3, F, H, H, O], [AH3079; C, = CH-S -, - N =, -CH = CH-,-, Me, F, H, H, O], [AH 3080; C, = CH-S-, -N =, -CH = CH-,-, Et, F, H, H, H O], [AH3081; C, = CH-S-, -N =, -CH = CH-,-, c-Pr, F, H, H, O], [AH3082; C, = CH-S-, -N =, -CH = CH-,-, OMe, F, H, H, O], [AH3083; C, = CH-S-, -N =, -CH = CH-,-, H, H, H F, H, O], [AH3084; C, = CH-S-, -N =, -CH = CH-,-, Cl, H, F, H, O], [AH 3085; C, = CH-S -, -N =, -CH = CH-,-, Br, H, F, H, O], [AH3086; C, = CH-S-, -N =, -CH = CH-,-, CF ₃ , H, F, H, O], [AH3087; C, = CH-S-, -N =, -CH = CH-,-, Me, H, F, H, O], [AH3088; C, = CH-S-, -N =, -CH = CH-,-, Et, H, F, H, O], [AH3089; C, = CH-S-, -N =,- CH = CH-,-, c-Pr, H, F, H, O], [AH 3090; C, = CH-S-, -N =, -CH = CH-,-, OMe, H, F, H , O], [AH3091; C, = CH-S-, -N =, -CH = CH-,-, H, H, H, F, O], [AH3092; C, = CH-S-,- N =, -CH = CH-,-, Cl, H, H, F, O], [AH 3093; C, = CH-S-, -N =, -CH = CH-,-, Br, H, H , F, O], [AH3094 ; C, = CH-S -, - N =, - CH = CH -, -, CF 3, H, H, F, O], [AH3095; C, = CH-S -, -N =, -CH = CH-,-, Me, H, H, F, O], [AH3096; C, = CH-S-, -N =, -CH = CH-,-, Et, H, H, F, O], [AH3097; C, = CH-S-, -N =, -CH = CH-,-, c-Pr, H, H, F, O], [AH3098; C, = CH-S-, -N =, -CH = CH-,-, OMe, H, H, F, O], [AH3099; C, = CH-O-, -N =, -CH = CH-, -, H, H, H, H, O], [AH 3 100; C, = CH-O-, -N =, -CH = CH-,-, F, H, H, H, O],

[AH 3 101; C, = CH-O-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3102; C, = CH-O-, -N =,- CH = CH-,-, Br, H, H, H, O], [AH 3103; C, = CH-O-, -N =, -CH = CH-,-, Me, H, H, H, O ], [AH 3104; C, = CH-O-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 3105; C, = CH-O-, -N = , -CH = CH-,-, Pr, H, H, H, O], [AH 3106; C, = CH-O-, -N =, -CH = CH-,-, i-Pr, H, H , H, O], [AH 3107; C, = CH-O-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3108; C, = CH- O-, -N =, -CH = CH-,-, c-Bu, H, H, H, O], [AH 3109; C, = CH-O-, -N =, -CH = CH-,- , OMe, H, H, H, O], [AH 3110; C, = CH-O-, -N =, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH 3 111 C, = CH-O-, -N =, -CH = CH-,-, SMe, H, H, H, O], [AH 3112; C, = CH-O-, -N =, -CH = CH -, -, Set, H , H, H, O], [AH3113; C, = CH-O -, - N =, - CH = CH -, -, CF 3, H, H, H, O] , [AH3114; C, = CH -O -, - N =, - CH = CH -, -, CHF 2, H, H, H, O], [AH3115; C, = CH-O -, - N = , -CH = CH -, -, OCF 3, H, H, H, O], [AH3116; C, = CH-O -, - N =, - CH = CH -, -, OCHF 2, H, H , H, O], [AH3117 ; C, = CH-O -, - N =, - CH = CH -, -, CH = CH 2, H, H, H, O], [AH3118; C, = CH -O -, - N =, - CH = CH -, -, C (Me) = CH 2, H, H, H, O], [AH3119; C, = CH-O -, - N =, - CH = CH-,-, CH = CHMe, H, H, H, O], [AH 3 120; C, = CH-O-, -N =, -CH = CH-,-, C≡CH, H, H, H, O], [AH 3121; C, = CH-O-, -N =, -CH = CH-,-, C≡CMe, H, H, H, O], [AH 3122; C, = C (CF ₃ ) -O-, -N =, -CH = CH-,-, H, H , H, H, O], [AH ₃ 123; C, = C (CF3)-O-,-N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3 124; C , = C (CF ₃ ) -O-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH ₃ 125; C, = C (CF ₃ ) -O-,- N =, - CH = CH - , -, CF 3, H, H, H, O], [AH3126; C, = C (CF 3) -O -, - N =, - CH = CH -, -, Me, H, H, H, O], [AH ₃ 127; C, = C (CF3)-O-, -N =, -CH = CH-,-, Et, H, H, H, O], [[ AH3128; C, = C (CF 3) -O -, - N =, - CH = CH -, -, c-Pr, H, H, H, O], [AH3129; C, = C (CF 3) -O-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3130; C, = CF-O-, -N =, -CH = CH-,-, H, H, H, H, H, O], [AH3 131; C, = CF-O-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3132; C, = CF-O-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH3133; C, = CF-O-, -N =, -CH = CH-, _{-, CF 3, H, H} , H, O], [AH3134; C, = CF-O -, - N =, - CH = CH -, -, Me, H, H, H, O], [AH3135 C, = CF-O-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 3136; C, = CF-O-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3137; C, = CF-O-, -N =, -CH = CH-,-, OMe, H, H, H, O ], [AH 3138; C, = CCl-O-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 3139; C, = CCl-O-, -N = , -CH = CH-,-, Cl, H, H, H, O], [AH 3140; C, = CCl-O-, -N =, -CH = CH-,-, Br, H, H, H , O], [AH3141; C , = CCl-O -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3142; C, = CCl-O-, -N =, -CH = CH-,-, Me, H, H, H, O], [AH3143; C, = CCl-O-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 3 144; C, = CCl-O-, -N =, -CH = CH -,-, c-Pr, H, H, H, O], [AH 3 145; C, = CCl-O-, -N =, -CH = CH-,-, OMe, H, H, H, O] , [AH 3146; C, = C (Me)-O-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 3147; C, = C (Me)-O -, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3148; C, = C (Me) -O-, -N =, -CH = CH-,- , Br, H, H, H , O], [AH3149; C, = C (Me) -O -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH 3 150; C, = C (Me)-O-, -N =, -CH = CH-,-, Me, H, H, H, O], [AH 3151; C, = C (Me)-O- , -N =, -CH = CH-,-, Et, H, H, H, O], [AH3152; C, = C (Me) -O-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3 153; C, = C (Me)-O-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3 154; C, = CH-O-, -N =, -CH = CH-,-, H, F, H, H, O], [AH 3 155; C, = CH-O-, -N =,- CH = CH-,-, Cl, F, H, H, O], [AH 3156; C, = CH-O-, -N =, -CH = CH-,-, Br, F, H, H, O ], [AH3157; C, = CH-O -, - N =, - CH = CH -, -, CF 3, F, H, H, O], [AH3158; C, = CH-O -, - N =, -CH = CH-,-, Me, F, H, H, O], [AH 3 159; C, = CH-O-, -N =, -CH = CH-,-, Et, F, H, H, O], [AH 3 160; C, = CH-O-, -N =, -CH = CH-,-, c-Pr, F, H, H, O], [AH3161; C, = CH-O -, -N =, -CH = CH-,-, OMe, F, H, H, O], [AH3162; C, = CH-O-, -N =, -CH = CH-,-, H, H, F, H, O], [AH 3163; C, = CH-O-,-N =, -CH = CH-,-, Cl, H, F, H, O], [AH 3 164; C, = CH -O-, -N =, -CH = CH-,-, Br, H, F, H, O], [AH 3165; C, = CH-O-, -N =, -CH = CH-,-, CF ₃ , H, F, H, O], [AH 3166; C, = CH-O-, -N =, -CH = CH-,-, Me, H, F, H, O ], [AH 3 167; C, = CH-O-, -N =, -CH = CH-,-, Et, H, F, H, O], [AH 3168; C, = CH-O-, -N = , -CH = CH-,-, c-Pr, H, F, H, O], [AH 3169; C, = CH-O-, -N =, -CH = CH-,-, OMe, H, F , H, O], [AH 3170; C, = CH-O-, -N =, -CH = CH-,-, H, H, H, F, O], [AH3171; C, = CH-O- , -N =, -CH = CH-,-, Cl, H, H, F, O], [AH 3172; C, = CH-O-, -N =, -CH = CH-,-, Br, H , H, F, O], [AH3173; C, = CH-O -, - N =, - CH = CH -, -, CF 3, H, H, F, O], [AH3174; C, = CH -O-, -N =, -CH = CH-,-, Me, H, H, F, O], [AH 3175; C, = CH-O-, -N =, -CH = CH-,-, Et, H, H, F, O], [AH 3176; C, = CH-O-, -N =, -CH = CH-,-, c-Pr, H, H, F, O], [AH 3177; C, = CH-O-, -N =, -CH = CH-,-, OMe, H, H, F, O], [AH 3178; C, = CH-O-, -N =, -CH = CH -,-, H, H, H, H, H, O], [AH 3179; C, = CH-O-, -N =, -CH = CH-,-, Cl, H, H, H, O], [[ AH 3180; C, = CH-O-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH3181; C, = CH-O-, -N =, -CH _{= CH -, -, CF 3} , H, H, H, O], [AH3182; C, = CH-O -, - N =, - CH = CH -, -, Me, H, H, H, O ], [AH3183; C, = CH-O-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 3184; C, = CH-O-, -N = , -CH = CH-,-, c-Pr, H, H, H, O], [AH 3 185; C, = CH-O-, -N =, -CH = CH-,-, OMe, H, H , H, O], [AH 3186; C, = CH-O-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3187; C, = CH-O- , -CH =, -CH = CH-,-, F, H, H, H, O], [AH 3188; C, = CH-O-, -CH =, -CH = CH-,-, Cl, H , H, H, O], [AH 3189; C, = CH-O-, -CH =, -CH = CH-,-, Br, H, H , H, O], [AH 3190; C, = CH-O-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH3191; C, = CH-O- , -CH =, -CH = CH-,-, Et, H, H, H, O], [AH 3192; C, = CH-O-, -CH =, -CH = CH-,-, Pr, H , H, H, O], [AH3193; C, = CH-O-, -CH =, -CH = CH-,-, i-Pr, H, H, H, O], [AH 3194; C, = CH-O-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3195; C, = CH-O-, -CH =, -CH = CH- ,-, c-Bu, H, H, H, O, [AH 3 196; C, = CH-O-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH 3 197; C, = CH-O-, -CH =, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH 3198; C, = CH-O-, -CH = , -CH = CH-,-, SMe, H, H, H, O], [AH 3199; C, = CH-O-, -CH =, -CH = CH-,-, Set, H, H, H , O], [AH3200; C , = CH-O -, - CH =, - CH = CH -, -, CF 3, H, H, H, O],

[AH3201; C, = CH- O -, - CH =, - CH = CH -, -, CHF 2, H, H, H, O], [AH3202; C, = CH-O -, - CH =, -CH = CH -, -, OCF 3, H, H, H, O], [AH3203; C, = CH-O -, - CH =, - CH = CH -, -, OCHF 2, H, H, H, O], [AH3204; C, = CH-O -, - CH =, - CH = CH -, -, CH = CH 2, H, H, H, O], [AH3205; C, = CH- O -, - CH =, - CH = CH -, -, C (Me) = CH 2, H, H, H, O], [AH3206; C, = CH-O -, - CH =, - CH = CH-,-, CH = CHMe, H, H, H, O], [AH 3207; C, = CH-O-, -CH =, -CH = CH-,-, C≡CH, H, H, H , O], [AH 3208; C, = CH-O-, -CH =, -CH = CH-,-, C, CMe, H, H, H, O], [AH 3209; C, = C (CF ₃ ) -O-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3210; C, = C (CF ₃ ) -O-, -CH =, -CH = CH -, -, Cl, H , H, H, O], [AH3211; C, = C (CF 3) -O -, - CH =, - CH = CH -, -, Br, H, H, H , O], [AH3212; C , = C (CF 3) -O -, - CH =, - CH = CH -, -, CF 3, H, H, H, O], [AH3213; C, = C _{(CF 3) -O -, -} CH =, - CH = CH -, -, Me, H, H, H, O], [AH3214; C, = C (CF 3) -O -, - CH =, -CH = CH-,-, Et, H, H, H, O], [AH 3215; C, = C (CF ₃ ) -O-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O] , [AH3216; C, = C (CF 3) -O -, - CH =, - CH = CH -, -, OMe, H, H, H, O], [AH3217; C, = CF-O-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3218; C, = CF-O-, -CH =, -CH = CH -,-, Cl, H, H, H, O, [AH 3219; C, = CF-O-, -CH =, -CH = CH-,-, Br, H, H, H, O], [[ AH3220; C, = CF-O -, - CH =, - CH = CH -, -, CF 3, H, H, H, O], [AH3221; C, = CF-O -, - CH =, - CH = CH-,-, Me, H, H, H, O], [AH 3222; C, = CF-O-, -CH =, -CH = CH-,-, Et, H, H, H, O ], [AH 3223; C, = CF-O-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3224; C, = CF-O-,- CH =, -CH = CH-,-, OMe, H, H, H, O], [AH 3225; C, = CCl-O-, -CH =, -CH = CH-,-, H, H, H , H, O], [AH 3226; C, = CCl-O-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH 3227; C, = CCl-O- , -CH =, -CH = CH-,-, Br, H, H, H, O], [AH 3228; C, = CCl-O-, -CH =, -CH = CH-,-, CF ₃ , H, H, H, O], [AH3229; C, = CCl-O-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH 3230; C, = CCl -O-, -CH =, -CH = CH-,-, Et, H, H, H, O], [AH3231; C, = CCl-O-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3232; C, = CCl-O-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH3233; C, = C (Me) -O-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH3234; C, = C (Me) -O-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH3235; C, = C (Me) -O-, -CH =, -CH = CH-,-, Br, H , H, H, O], [AH3236; C, = C (Me) -O -, - CH =, - CH = CH -, -, CF 3, H, H, H, O], [AH3237; C , = C (Me) -O-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH 3238; C, = C (Me) -O-, -CH = , -CH = CH-,-, Et, H, H, H, O], [AH 3239; C, = C (Me) -O-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3240; C, = C (Me)-O-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH3241; C , = CH-O-, -CH =, -CH = CH-,-, H, F, H, H, O], [AH3242; C, = CH-O-, -CH =, -CH = CH- ,-, Cl, F, H, H, O], [AH3243; C, = CH-O-, -CH =, -CH = CH-,-, Br, F, H, H, O], [AH 3244; C, = CH-O-, -CH =, -CH = CH-,- , CF ₃ , F, H, H, O], [AH 3245; C, = CH-O-, -CH =, -CH = CH-,-, Me, F, H, H, O], [AH 3246; C, = CH-O-, -CH =, -CH = CH-,-, Et, F, H, H, O], [AH 3247; C, = CH-O-, -CH =, -CH = CH -,-, c-Pr, F, H, H, O], [AH 3248; C, = CH-O-, -CH =, -CH = CH-,-, OMe, F, H, H, O] , [AH 3249; C, = CH-O-, -CH =, -CH = CH-,-, H, H, F, H, O], [AH 3250; C, = CH-O-, -CH =, -CH = CH-,-, Cl, H, F, H, O], [AH3251; C, = CH-O-, -CH =, -CH = CH-,-, Br, H, F, H, O], [AH3252; C, = CH-O -, - CH =, - CH = CH -, -, CF 3, H, F, H, O], [AH3253; C, = CH-O -, - CH =, -CH = CH-,-, Me, H, F, H, O], [AH 3 254; C, = CH-O-, -CH =, -CH = CH-,-, Et, H, F , H, O], [AH 3 255; C, = CH-O-, -CH =, -CH = CH-,-, c-Pr, H, F, H, O], [AH 3 256; C, = CH- O-, -CH =, -CH = CH-,-, OMe, H, F, H, O], [AH 3257; C, = CH-O-, -CH =, -CH = CH-,-, H , H, H, F, O], [AH3258; C, = CH-O-, -CH =, -CH = CH-,-, Cl, H, H, F, O], [AH 3259; C, = CH-O-, -CH =, -CH = CH-,-, Br, H, H, F, O], [AH 3 260; C, = CH-O-, -CH =, -CH = CH-,- _{, CF 3, H, H,} F, O], [AH3261; C, = CH-O -, - CH =, - CH = CH -, -, Me, H, H, F, O], [AH3262; C, = CH-O-, -CH =, -CH = CH-,-, Et, H, H, F, O], [AH 3263; C, = CH-O-, -CH =, -CH = CH -,-, c-Pr, H, H, F, O], [AH 3 264; C, = CH-O-, -CH =, -CH = CH-,-, OMe, H, H, F, O] , [AH3265; C, = CH-O-, -CH =, -CH = C H-,-, H, H, H, H, H, O], [AH 3 266; C, = CH-O-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH 3 267; C, = CH-O-, -CH =, -CH = CH-,-, Br, H, H, H, O], [AH 3268; C, = CH-O-, -CH =,- CH = CH -, -, CF 3, H, H, H, O], [AH3269; C, = CH-O -, - CH =, - CH = CH -, -, Me, H, H, H, O], [AH 3270; C, = CH-O-, -CH =, -CH = CH-,-, Et, H, H, H, O], [AH3271; C, = CH-O-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3272; C, = CH-O-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH3273; C, = CH-CH =, -O-, -CH = CH-,-, H, H, H, H, O], [AH 3274; C, = CH-CH =, -O-, -CH = CH-,-, F, H, H, H, O], [AH 3275; C, = CH-CH =, -O-, -CH = CH-,-, Cl, H, H, H, O], [AH3276; C, = CH-CH =, -O-, -CH = CH-,-, Br, H, H, H, O], [AH 3277; C, = CH -CH =, -O-, -CH = CH-,-, Me, H, H, H, O], [AH 3278; C, = CH-CH =, -O-, -CH = CH-,-, Et, H, H, H, O], [AH 3279; C, = CH-CH =, -O-, -CH = CH-,-, Pr, H, H, H, O], [AH 3280; C, = CH-CH =, -O-, -CH = CH-,-, i-Pr, H, H, H, O], [AH3281; C, = CH-CH =, -O-, -CH = CH -,-, c-Pr, H, H, H, O], [AH3282; C, = CH-CH =, -O-, -CH = CH-,-, c-Bu, H, H, H, H O], [AH3283; C, = CH-CH =, -O-, -CH = CH-,-, OMe, H, H, H, O], [AH3284; C, = CH-CH =, -O -, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH 3285; C, = CH-CH =, -O-, -CH = CH-,-, SMe, H, H, H, O], [AH 3286; C, = CH-CH =, -O-, -CH = CH-,-, Set, H, H, H, O], [AH 3287; C, = CH-CH =, - O -, - CH = CH -, -, CF 3, H, H, H, O], [AH3288; C, = CH-CH =, - O -, - CH = CH -, -, CHF 2, H, H, H, O], [AH3289; C, = CH-CH =, - O -, - CH = CH - , -, OCF 3, H, H, H, O], [AH3290; C, = CH-CH =, - O -, - CH = CH -, -, OCHF 2, H , H, H, O], [AH3291; C, = CH-CH =, - O -, - CH = CH -, -, CH = CH 2, H, H, H, O], [AH3292; C, = CH-CH =, - O -, - CH = CH -, -, C (Me) = CH 2, H, H, H, O], [AH3293; C, = CH-CH =, - O-, -CH = CH-,-, CH = CHMe, H, H, H, O], [AH 3294; C, = CH-CH =, -O-, -CH = CH-,-, C≡CH, H, H, H, O], [AH 3295; C, = CH-CH =, -O-, -CH = CH-,-, C≡CMe, H, H, H, O], [AH 3296; C, = C _{(CF 3) -CH =, -} O -, - CH = CH -, -, H, H, H, H, O], [AH3297; C, = C (CF 3) -CH =, - O-, -CH = CH -, -, Cl , H, H, H, O], [AH3298; C, = C (CF 3) -CH =, - O -, - CH = CH -, -, Br, H, H, H, O], [ AH3299; C, = C (CF 3) -CH =, - O -, - CH = CH -, -, CF 3, H, H, H, O], [AH3300; C , = C (CF ₃ ) -CH =, -O-, -CH = CH-,-, Me, H, H, H, O],

[AH3301; C, = C ( CF 3) -CH =, - O -, - CH = CH -, -, Et, H, H, H, O], [AH3302; C, = C (CF 3) - CH =, - O -, - CH = CH -, -, c-Pr, H, H, H, O], [AH3303; C, = C (CF 3) -CH =, - O -, - CH = CH-,-, OMe, H, H, H, H, O], [AH 3 304; C, = CF-CH =, -O-, -CH = CH-,-, H, H, H, H, O], [AH 3 305; C, = CF-CH =, -O-, -CH = CH-,-, Cl, H, H, H, O], [AH 3306; C, = CF-CH =, -O-,- CH = CH -, -, Br , H, H, H, O], [AH3307; C, = CF-CH =, - O -, - CH = CH -, -, CF 3, H, H, H, O], [AH 3308; C, = CF-CH =, -O-, -CH = CH-,-, Me, H, H, H, O], [AH 3309; C, = CF-CH =, -O -, -CH = CH-,-, Et, H, H, H, O], [AH3310; C, = CF-CH =, -O-, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3311; C, = CF-CH =, -O-, -CH = CH-,-, OMe, H, H, H, O], [AH3312; C, = CCl-CH =, -O-, -CH = CH-,-, H, H, H, H, O], [AH3313; C, = CCl-CH =, -O-, -CH = CH-,-, Cl, H, H, H, O], [AH3314; C, = CCl-CH =, -O-, -CH = CH-,-, Br, H, H, H, O], [AH3315; C, = CCl -CH =, - O -, - CH = CH -, -, CF 3, H, H, H, O], [AH3316; C, = CCl-CH =, - O -, - CH = CH -, - , Me, H, H, H, O], [AH3317; C, = CCl-CH =, -O-, -CH = CH-,-, Et, H, H, H, O], [AH3318; C , = CCl-CH =, -O-, -CH = CH-,-, c-Pr, H, H, H, O], [AH3319; C, = CCl-CH =, -O-, -CH = CH-,-, OMe, H, H, H, O, [AH 3320; C, = C (Me)-CH =, -O-, -CH = CH-,-, H, H, H, H, H, O], [AH3321; C, = C (Me) -CH =, -O-, -CH = CH-,-, Cl, H, H, H, O], [AH3322; C, = C (Me) -CH =, -O-, -CH = CH- , -, Br, H, H , H, O], [AH3323; C, = C (Me) -CH =, - O -, - CH = CH -, -, CF 3, H, H, H, O ], [AH 3324; C, = C (Me) -CH =, -O-, -CH = CH-,-, Me, H, H, H, O], [AH 3325; C, = C (Me)- CH =, -O-, -CH = CH-,-, Et, H, H, H, O], [AH3326; C, = C (Me) -CH =, -O-, -CH = CH-, -, c-Pr, H, H, H, O], [AH 3327; C, = C (Me)-CH =, -O-, -CH = CH-,-, OMe, H, H, H, O ], [AH 3328; C, = CH-CH =, -O-, -CH = CH-,-, H, F, H, H, O], [AH 3329; C, = CH-CH =, -O- , -CH = CH-,-, Cl, F, H, H, O], [AH3330; C, = CH-CH =, -O-, -CH = CH-,-, Br, F, H, H , O], [AH3331; C , = CH-CH =, - O -, - CH = CH -, -, CF 3, F, H, H, O], [AH3332; C, = CH-CH =, -O-, -CH = CH-,-, Me, F, H, H, O], [AH3333; C, = CH-CH =, -O-, -CH = CH-,-, Et, F, H, H, O], [AH3334; C, = CH-CH =, -O-, -CH = CH-,-, c-Pr, F, H, H, O], [AH3335; C, = CH -CH =, -O-, -CH = CH-,-, OMe, F, H, H, O], [AH 3336; C, = CH-CH =, -O-, -CH = CH-,-, H, H, F, H, O], [AH 3337; C, = CH-CH =, -O-, -CH = CH-,-, Cl, H, F, H, O], [AH 3338; C, = CH-CH =, -O-, -CH = CH-,-, Br, H, F, H, O], [AH3339; C, = CH-CH =, -O-, -CH = CH-, _{-, CF 3, H, F} , H, O], [AH3340; C, = CH-CH =, - O -, - CH = CH -, -, Me, H, F, H, O], [AH3341 C, = CH-CH =, -O-, -CH = CH-,-, Et, H, F, H, O], [AH3342; C, = CH-CH =, -O-, -CH = CH-,-, c-Pr, H, F, H, O], [AH 3343; C, = CH-CH =, -O-, -CH = CH-,-, OMe, H, F, H, O ], [AH 3344; C, = CH-CH =, -O-, -CH = CH-, -, H, H, H, F, O], [AH3345; C, = CH-CH =, -O-, -CH = CH-,-, Cl, H, H, F, O], [AH3346; C, = CH-CH =, -O-, -CH = CH-,-, Br, H, H, F, O], [AH 3347; C, = CH-CH =, -O-, -CH = CH _{-, -, CF 3, H} , H, F, O], [AH3348; C, = CH-CH =, - O -, - CH = CH -, -, Me, H, H, F, O], [AH 3349; C, = CH-CH =, -O-, -CH = CH-,-, Et, H, H, F, O], [AH 3 350; C, = CH-CH =, -O-,- CH = CH-,-, c-Pr, H, H, F, O], [AH 3351; C, = CH-CH =, -O-, -CH = CH-,-, OMe, H, H, F , O], [AH 3352; C, = CH-CH =, -O-, -CH = CH-,-, H, H, H, H, O], [AH 3353; C, = CH-CH =,- O-, -CH = CH-,-, Cl, H, H, H, O], [AH 3354; C, = CH-CH =, -O-, -CH = CH-,-, Br, H, H , H, O], [AH 3 355; C, = CH-CH =, -O-, -CH = CH-,-, CF ₃ , H, H, H, O], [AH 3356; C, = CH-CH =, -O-, -CH = CH-,-, Me, H, H, H, O], [AH 3357; C, = CH-CH =, -O-, -CH = CH-,-, Et, H, H, H, O], [AH3358; C, = CH-CH =, -O-, -CH = CH-,-, c-Pr, H, H, H, O], [AH3359; C, = CH-CH =, -O-, -CH = CH-,-, OMe, H, H, H, O], [AH 3360; C, = CH-CH =, -S-, -CH = CH-, -, H, H, H, H, H, O], [AH3361; C, = CH-CH =, -S-, -CH = CH-,-, F, H, H, H, O], [AH3362; C, = CH-CH =, -S-, -CH = CH-,-, Cl, H, H, H, O], [AH3363; C, = CH-CH =, -S-, -CH = CH -,-, Br, H, H, H, O], [AH 3364; C, = CH-CH =, -S-, -CH = CH-,-, Me, H, H, H, O], [[ AH 3365; C, = CH-CH =, -S-, -CH = CH-,-, Et, H, H, H, O], [AH 3366; C, = CH-CH =, -S-, -CH = CH-,-, Pr, H, H, H, O], [AH 3367; C, = CH-CH =, -S-, -CH = CH-,-, i-Pr, H, H, H, O], [AH 3368; C, = CH-CH =, -S-, -CH = CH -,-, c-Pr, H, H, H, O], [AH 3369; C, = CH-CH =, -S-, -CH = CH-,-, c-Bu, H, H, H, H O], [AH 3370; C, = CH-CH =, -S-, -CH = CH-,-, OMe, H, H, H, O], [AH3371; C, = CH-CH =, -S -, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH3372; C, = CH-CH =, -S-, -CH = CH-,-, SMe, H, H, H, O], [AH 3373; C, = CH-CH =, -S-, -CH = CH-,-, Set, H, H, H, O], [AH 3374; C, = CH-CH =, - S -, - CH = CH -, -, CF 3, H, H, H, O], [AH3375; C, = CH-CH =, - S -, - CH = CH -, -, CHF ₂ , H, H, H, O], [AH 3376; C, = CH-CH =, -S-, -CH = CH-,-, OCF ₃ , H, H, H, O], [AH 3377; C , = CH-CH =, -S-, -CH = CH-,-, OCHF ₂ , H, H, H, O], [AH 3378; C, = CH-CH =, -S-, -CH = CH _{-, -, CH = CH 2} , H, H, H, O], [AH3379; C, = CH-CH =, - S -, - CH = CH -, -, C (Me) = CH 2, H , H, H, O], [AH 3 380; C, = CH-CH =, -S-, -CH = CH-,-, CH = CHMe, H, H, H, O], [AH3381; C, = CH-CH =, -S-, -CH = CH-,-, C≡CH, H, H, H, O], [AH3382; C, = CH-CH =, -S-, -CH = CH- ,-, C≡CMe, H, H, H, O], [AH 3383; C, = C (CF ₃ ) -CH =, -S-, -CH = CH-,-, H, H, H, H , O], [AH3384; C , = C (CF 3) -CH =, - S -, - CH = CH -, -, Cl, H, H, H, O], [AH3385; C, = C ( _{CF 3) -CH =, - S} -, - CH = CH -, -, Br, H, H, H, O], [AH3386; C, = C (CF 3) -CH =, - S -, - CH = CH -, -, CF 3, H, H, H, O], [AH3387; C, = C (CF 3) -CH =, - S -, - CH = CH -, -, Me, H, H, H, O], [AH3388; C, = C (CF 3) -CH =, - S -, - CH = CH -, -, Et, H, H, H, O], [AH3389; C, = C (CF ₃ ) -CH =, -S-, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3390; C, = C (CF ₃ ) -CH =, -S-, -CH = CH-,-, OMe, H, H, H, O], [AH3391; C, = CF-CH =, -S-, -CH = CH-,-, H, H, H, H, H O], [AH3392; C, = CF-CH =, -S-, -CH = CH-,-, Cl, H, H, H, O], [AH3393; C, = CF-CH =, -S -, - CH = CH -, -, Br, H, H, H, O], [AH3394; C, = CF-CH =, - S -, - CH = CH -, -, CF 3, H, H , H, O], [AH3395; C, = CF-CH =, -S-, -CH = CH-,-, Me, H, H, H, O], [AH3396; C, = CF-CH = , -S-, -CH = CH-,-, Et, H, H, H, O], [AH 3397; C, = CF-CH =, -S-, -CH = CH-,-, c-Pr , H, H, H, O], [AH3398; C, = CF-CH =, -S-, -CH = CH-,-, OMe, H, H, H, O], [AH3399; C, = CCl-CH =, -S-, -CH = CH-,-, H, H, H, H, O], [AH 3400; C, = CCl-CH =, -S-, -CH = CH-,- , Cl, H, H, H, O],

[AH3401; C, = CCl-CH =, -S-, -CH = CH-,-, Br, H, H, H, O], [AH3402; C, = CCl-CH =, -S-,- CH = CH -, -, CF 3, H, H, H, O], [AH3403; C, = CCl-CH =, - S -, - CH = CH -, -, Me, H, H, H, O], [AH3404; C, = CCl-CH =, -S-, -CH = CH-,-, Et, H, H, H, O], [AH 3405; C, = CCl-CH =, -S -, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3406; C, = CCl-CH =, -S-, -CH = CH-,-, OMe, H, H, H, O], [AH3407; C, = C (Me) -CH =, -S-, -CH = CH-,-, H, H, H, H, O], [AH 3408; C, = C (Me) -CH =, -S-, -CH = CH-,-, Cl, H, H, H, O], [AH 3409; C, = C (Me) -CH =, -S-,- CH = CH -, -, Br , H, H, H, O], [AH3410; C, = C (Me) -CH =, - S -, - CH = CH -, -, CF 3, H, H , H, O], [AH 3411; C, = C (Me) -CH =, -S-, -CH = CH-,-, Me, H, H, H, O], [AH 3412; C, = C (Me) -CH =, -S-, -CH = CH-,-, Et, H, H, H, O], [AH 3413; C, = C (Me) -CH =, -S-, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3414; C, = C (Me) -CH =, -S-, -CH = CH-,-, OMe, H, H , H, O], [AH3415; C, = CH-CH =, -S-, -CH = CH-,-, H, F, H, H, O], [AH3416; C, = CH-CH = , -S-, -CH = CH-,-, Cl, F, H, H, O], [AH 3417; C, = CH-CH =, -S-, -CH = CH-,-, Br, F , H, H, O], [AH3418; C, = CH-CH =, - S -, - CH = CH -, -, CF 3, F, H, H, O], [AH3419; C, = CH -CH =, -S-, -CH = CH-,-, Me, F, H, H, O], [AH 3420; C, = CH-CH =, -S-, -CH = CH-,-, Et, F, H, H, O], [AH 3421; C, = CH-CH =, -S-, -CH = CH-,-, c-Pr, F, H, H, O], [AH 3422; C, = CH-CH =, -S-, -CH = CH-,- , OMe, F, H, H, O], [AH 3423; C, = CH-CH =, -S-, -CH = CH-,-, H, H, F, H, O], [AH 3424; C , = CH-CH =, -S-, -CH = CH-,-, Cl, H, F, H, O], [AH 3425; C, = CH-CH =, -S-, -CH = CH- , -, Br, H, F , H, O], [AH3426; C, = CH-CH =, - S -, - CH = CH -, -, CF 3, H, F, H, O], [ AH 3427; C, = CH-CH =, -S-, -CH = CH-,-, Me, H, F, H, O], [AH 3428; C, = CH-CH =, -S-, -CH = CH-,-, Et, H, F, H, O], [AH 3429; C, = CH-CH =, -S-, -CH = CH-,-, c-Pr, H, F, H, O], [AH 3430; C, = CH-CH =, -S-, -CH = CH-,-, OMe, H, F, H, O], [AH3431; C, = CH-CH =, -S -, -CH = CH-,-, H, H, H, F, O], [AH3432; C, = CH-CH =, -S-, -CH = CH-,-, Cl, H, H, H F, O], [AH 3433; C, = CH-CH =, -S-, -CH = CH-,-, Br, H, H, F, O], [AH 3434; C, = CH-CH =, -S -, - CH = CH - , -, CF 3, H, H, F, O], [AH3435; C, = CH-CH =, - S -, - CH = CH -, -, Me, H , H, F, O], [AH 3436; C, = CH-CH =, -S-, -CH = CH-,-, Et, H, H, F, O], [AH 3437; C, = CH- CH =, -S-, -CH = CH-,-, c-Pr, H, H, F, O], [AH3438; C, = CH-CH =, -S-, -CH = CH-,- , OMe, H, H, F, O], [AH 3439; C, = CH-CH =, -S-, -CH = CH-,-, H, H, H, H, O], [AH 3440; C , = CH-CH =, -S-, -CH = CH-,-, Cl, H, H, H, O], [AH3441; C, = CH-CH =, -S-, -CH = CH- , -, Br, H, H , H, O], [AH3442; C, = CH-CH =, - S -, - CH = CH -, -, CF 3, H, H, H, O], [ AH 3443; C, = CH-CH =, -S-, -CH = CH-,-, Me, H, H, H, O], [AH 3444; C, = CH-CH =, -S-, -CH = CH-,-, Et, H, H, H, O], [AH 344 5; C, = CH-CH =, -S-, -CH = CH-,-, c-Pr, H, H, H, O], [AH3446; C, = CH-CH =, -S-, -CH = CH-,-, OMe, H, H, H, O], [AH 3447; C, = CH-S-, -CH =, -CH = CH-,-, H, H, H, H, H O], [AH 3448; C, = CH-S-, -CH =, -CH = CH-,-, F, H, H, H, O], [AH 3449; C, = CH-S-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH 3450; C, = CH-S-, -CH =, -CH = CH-,-, Br, H, H, H, O], [AH3451; C, = CH-S-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH3452; C, = CH-S-, -CH =, -CH = CH-,-, Et, H, H, H, O], [AH3453; C, = CH-S-, -CH =, -CH = CH-,-, Pr, H, H, H, O], [AH 3454; C, = CH-S-, -CH =, -CH = CH-,-, i-Pr, H, H, H, O], [AH 3455; C, = CH -S-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3456; C, = CH-S-, -CH =, -CH = CH-, -, c-Bu, H, H, H, O], [AH 3457; C, = CH-S-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [[ AH 3458; C, = CH-S-, -CH =, -CH = CH-,-, Oi-Pr, H, H, H, O], [AH 3459; C, = CH-S-, -CH =, -CH = CH-,-, SMe, H, H, H, O], [AH 3460; C, = CH-S-, -CH =, -CH = CH-,-, Set, H, H, H, H O], [AH3461; C, = CH-S -, - CH =, - CH = CH -, -, CF 3, H, H, H, O], [AH3462; C, = CH-S -, - CH =, - CH = CH - , -, CHF 2, H, H, H, O], [AH3463; C, = CH-S -, - CH =, - CH = CH -, -, OCF 3, H , H, H, O], [AH 3464; C, = CH-S-, -CH =, -CH = CH-,-, OCHF ₂ , H, H, H, O], [AH 3 465; C, = CH -S -, - CH =, - CH = CH -, -, CH = CH 2, H, H, H, O], [AH3466; C, = CH-S -, - CH =, - CH = CH- , -, C (Me) = CH 2, H, H , H, O], [AH 3467; C, = CH-S-, -CH =, -CH = CH-,-, CH = CHMe, H, H, H, O], [AH 3468; C, = CH- S-, -CH =, -CH = CH-,-, C≡CH, H, H, H, O], [AH 3469; C, = CH-S-, -CH =, -CH = CH-,- , C≡CMe, H, H, H, O], [AH ₃ 470; C, C C (CF ₃ ) -S-, -CH =, -CH = CH-,-, H, H, H, H, O ], [AH3471; C, = C (CF 3) -S -, - CH =, - CH = CH -, -, Cl, H, H, H, O], [AH3472; C, = C (CF 3 ) -S-, -CH =, -CH = CH-,-, Br, H, H, H, O], [AH 3473; C, = C (CF ₃ ) -S-, -CH =, -CH = _{CH -, -, CF 3,} H, H, H, O], [AH3474; C, = C (CF 3) -S -, - CH =, - CH = CH -, -, Me, H, H, H, O], [AH3475; C, = C (CF 3) -S -, - CH =, - CH = CH -, -, Et, H, H, H, O], [AH3476; C, = C _{(CF 3) -S -, -} CH =, - CH = CH -, -, c-Pr, H, H, H, O], [AH3477; C, = C (CF 3) -S -, - CH =, -CH = CH-,-, OMe, H, H, H, O], [AH3478; C, = CF-S-, -CH =, -CH = CH-,-, H, H, H, H H, O], [AH 3479; C, = CF-S-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH 3480; C, = CF-S-, -CH =, - CH = CH - , -, Br, H, H, H, O], [AH3481; C, = CF-S -, - CH =, - CH = CH -, -, CF 3, H , H, H, O], [AH3482; C, = CF-S-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH3483; C, = CF- S-, -CH =, -CH = CH-,-, Et, H, H, H, O], [AH 3484; C, = CF-S-, -CH =, -CH = CH-,-, c -Pr, H, H, H, O], [AH 3485; C, = CF-S-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH 3486; C , = CCl-S-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3487; C, = CCl-S-, -CH =, -CH = CH- ,-, Cl, H, H, H, O], [AH 3488; C, = CCl-S-, -CH =, -CH = CH-,-, Br, H, H, H, O], [AH 3489; C, = CCl-S-, -CH =, - CH = CH -, -, CF 3, H, H, H, O], [AH3490; C, = CCl-S -, - CH =, - CH = CH -, -, Me, H, H , H, O], [AH3491; C, = CCl-S-, -CH =, -CH = CH-,-, Et, H, H, H, O], [AH3492; C, = CCl-S- , -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3493; C, = CCl-S-, -CH =, -CH = CH-,-, OMe , H, H, H, O], [AH 3494; C, = C (Me)-S-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3495; C, = C (Me) -S-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH3496; C, = C (Me) -S-, -CH =, -CH = CH-,-, Br, H, H, H, O], [AH 3497; C, = C (Me) -S-, -CH =, -CH = CH-,-, CF ₃ , H, H, H, O], [AH 3498; C, = C (Me)-S-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH 3499; C , = C (Me) -S-, -CH =, -CH = CH-,-, Et, H, H, H, O], [AH 3500; C, = C (Me) -S-, -CH = , -CH = CH-,-, c-Pr, H, H, H, O],

[AH 3501; C, = C (Me)-S-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH 3502; C, = CH-S-, -CH =, -CH = CH-,-, H, F, H, H, O], [AH 3503; C, = CH-S-, -CH =, -CH = CH-,-, Cl, F, H, H, O], [AH 3504; C, = CH-S-, -CH =, -CH = CH-,-, Br, F, H, H, O], [AH 3505; C, = CH-S-, -CH =, - CH = CH - , -, CF 3, F, H, H, O], [AH3506; C, = CH-S -, - CH =, - CH = CH -, -, Me, F , H, H, O], [AH3507; C, = CH-S-, -CH =, -CH = CH-,-, Et, F, H, H, O], [AH 3508; C, = CH- S-, -CH =, -CH = CH-,-, c-Pr, F, H, H, O], [AH 3509; C, = CH-S-, -CH =, -CH = CH-,- , OMe, F, H, H, O], [AH 3510; C, = CH-S-, -CH =, -CH = CH-,-, H, H, F, H, O], [AH 3511; C , = CH-S-, -CH =, -CH = CH-,-, Cl, H, F, H, O], [AH 3512; C, = CH-S-, -CH =, -CH = CH- , -, Br, H, F , H, O], [AH3513; C, = CH-S -, - CH =, - CH = CH -, -, CF 3, H, F, H, O], [ AH 3514; C, = CH-S-, -CH =, -CH = CH-,-, Me, H, F, H, O], [AH 3515; C, = CH-S-, -CH =, -CH = CH-,-, Et, H, F, H, O], [AH 3516; C, = CH-S-, -CH =, -CH = CH-,-, c-Pr, H, F, H, O], [AH 3517; C, = CH-S-, -CH =, -CH = CH-,-, OMe, H, F, H, O], [AH 3518; C, = CH-S-, -CH =, -CH = CH-,-, H, H, H, F, O], [AH 3519; C, = CH-S-, -CH =, -CH = CH-,-, Cl, H, H, F, O], [AH 3520; C, = CH-S-, -CH =, -CH = CH-,-, Br, H, H, F, O], [AH 3521; C, = CH-S-, -CH =, - CH = CH - , -, CF 3, H, H, F, O], [AH3522; C, = CH-S -, - CH =, - CH = CH -, -, Me, H , H, F, O], [AH 3523; C, = CH-S- , -CH =, -CH = CH-,-, Et, H, H, F, O], [AH 3524; C, = CH-S-, -CH =, -CH = CH-,-, c-Pr , H, H, F, O], [AH 3525; C, = CH-S-, -CH =, -CH = CH-,-, OMe, H, H, F, O], [AH 3526; C, = CH-S-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3527; C, = CH-S-, -CH =, -CH = CH-,- , Cl, H, H, H, O], [AH 3528; C, = CH-S-, -CH =, -CH = CH-,-, Br, H, H, H, O], [AH 3529; C , = CH-S -, - CH =, - CH = CH -, -, CF 3, H, H, H, O], [AH3530; C, = CH-S -, - CH =, - CH = CH -,-, Me, H, H, H, O], [AH 3531; C, = CH-S-, -CH =, -CH = CH-,-, Et, H, H, H, O], [[ AH 3532; C, = CH-S-, -CH =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3533; C, = CH-S-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH 3534; C, -CH = CH-, = CH-N =, -CH = CH-,-, H, H, H, H, O], [AH 3 535; C, -CH = CH-, = CH-N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3536; C, -CH = CH -, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [AH 3537; C, -CH = CH-, = CH-N =, -CH = CH-, _{-, CF 3, H, H} , H, O], [AH3538; C, -CH = CH -, = CH-N =, - CH = CH -, -, Me, H, H, H, O], [AH 3539; C, -CH = CH-, = CH-N =, -CH = CH-,-, Et, H, H, H, O], [AH 3540; C, -CH = CH-, = CH- N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3541; C, -CH = CH-, = CH-N =, -CH = CH-,-, OMe , H, H, H, O], [AH3542; C, -CH = CF-, = CH-N =, -CH = CH-,-, H, H, H, H, O], [AH3543; C , -CH = CF-, = CH-N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3544; C, -CH = CF-, = CH-N =,- CH = CH-,-, Br, H, H, H, O], [AH 3545; C, -CH = CF - , = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3546; C, -CH = CF -, = CH- N =, -CH = CH-,-, Me, H, H, H, O], [AH 3547; C, -CH = CF-, = CH-N =, -CH = CH-,-, Et, H , H, H, O], [AH 3548; C, -CH = CF-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3549; C , -CH = CF-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3550; C, -CF = CH-, = CH-N =,- CH = CH-,-, H, H, H, H, H, O], [AH3551; C, -CF = CH-, = CH-N =, -CH = CH-,-, Cl, H, H, H , O], [AH3552; C, -CF = CH-, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [AH 3553; C, -CF = CH- , = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3554; C, -CF = CH -, = CH-N =, - CH = CH-, -, Me, H, H, H, O], [AH 3 555; C, -CF = CH-, = CH-N =, -CH = CH-,-, Et, H, H, H, O], [[ AH 3556; C, -CF = CH-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3557; C, -CF = CH-, = CH -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3558; C, -CH = CH-, = CF-N =, -CH = CH-,-, H, H, H, H, O], [AH 3559; C, -CH = CH-, = CF-N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3560; C, -CH = CH-, = CF-N =, -CH = CH-,-, Br, H, H, H, O], [AH3561; C, -CH = CH-, = CF-N =, -CH _{= CH -, -, CF 3} , H, H, H, O], [AH3562; C, -CH = CH -, = CF-N =, - CH = CH -, -, Me, H, H, H , O], [AH 3563; C, -CH = CH-, = CF-N =, -CH = CH-,-, Et, H, H, H, O], [AH 3564; C, -CH = CH- , = CF-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3565; C, -CH = CH-, = CF-N =, -CH = CH- ,-, OMe, H, H, H, O], [AH 3 566; C, -CH = CCl-, = CH-N =, -CH = CH-,-, H, H, H, H, O], [AH3567; C, -CH = CCl-, = CH- N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3568; C, -CH = CCl-, = CH-N =, -CH = CH-,-, Br, H , H, H, O], [AH3569; C, -CH = CCl -, = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3570; C, -CH = CCl-, = CH-N =, -CH = CH-,-, Me, H, H, H, O], [AH3571; C, -CH = CCl-, = CH-N =, -CH = CH-,-, Et, H, H, H, O, [AH3572; C, -CH = CCl-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H H, O], [AH3573; C, -CH = CCl-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH3574; C, -CCl = CH -, = CH-N =, -CH = CH-,-, H, H, H, H, O], [AH3575; C, -CCl = CH-, = CH-N =, -CH = CH-, -, Cl, H, H, H, O], [AH 3576; C, -CCl = CH-, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [[ AH3577; C, -CCl = CH - , = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3578; C, -CCl = CH -, = CH- N =, -CH = CH-,-, Me, H, H, H, O], [AH3579; C, -CCl = CH-, = CH-N =, -CH = CH-,-, Et, H , H, H, O], [AH3580; C, -CCl = CH-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3581; C , -CCl = CH-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH3582; C, -CH = CH-, = CCl-N =,- CH = CH-,-, H, H, H, H, H, O], [AH 3583; C, -CH = CH-, = CCl-N =, -CH = CH-,-, Cl, H, H, H , O], [AH 3584; C, -CH = CH-, = CCl-N =, -CH = CH-,-, Br, H, H, H, O], [AH 3585; C, -CH = CH- , = CCl-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3586; C, -CH = CH -, = CCl-N =, - C H = CH-,-, Me, H, H, H, O, [AH 3587; C, -CH = CH-, = CCl-N =, -CH = CH-,-, Et, H, H, H , O], [AH 3588; C, -CH = CH-, = CCl-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3589; C, -CH = CH-, = CCl-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3 590; C, -CH = C (Me)-, = CH-N =, -CH = CH-,-, H, H, H, H, H, O], [AH3591; C, -CH = C (Me)-, = CH-N =, -CH = CH-,-, Cl, H, H , H, O], [AH 3592; C, -CH = C (Me)-, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [AH 3 5 5 3 C; -CH = C (Me) -, = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3594; C, -CH = C (Me) -, = CH-N =, -CH = CH-,-, Me, H, H, H, O], [AH3595; C, -CH = C (Me)-, = CH-N =, -CH = CH-, -, Et, H, H, H, O, [AH 3596; C, -CH = C (Me)-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H , O], [AH 3597; C, -CH = C (Me)-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3598; C, -C (Me) = CH-, = CH-N =, -CH = CH-,-, H, H, H, H, O], [AH3599; C, -C (Me) = CH-, = CH-N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3600; C, -C (Me) = CH-, = CH-N =, -CH = CH-,-, Br , H, H, H, O],

[AH3601; C, -C (Me ) = CH -, = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3602; C, -C (Me) = CH-, = CH-N =, -CH = CH-,-, Me, H, H, H, O], [AH3603; C, -C (Me) = CH-, = CH-N =,- CH = CH-,-, Et, H, H, H, O], [AH3604; C, -C (Me) = CH-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3605; C, -C (Me) = CH-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3606 C, -CH = CH-, = C (Me) -N =, -CH = CH-,-, H, H, H, H, O], [AH 3607; C, -CH = CH-, = C (Me) -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3608; C, -CH = CH-, = C (Me) -N =, -CH = CH -, -, Br, H, H, H, O], [AH3609; C, -CH = CH -, = C (Me) -N =, - CH = CH -, -, CF 3, H, H, H, O], [AH 3610; C, -CH = CH-, = C (Me) -N =, -CH = CH-,-, Me, H, H, H, O], [AH 3611; C,- CH = CH-, = C (Me) -N =, -CH = CH-,-, Et, H, H, H, O], [AH 3612; C, -CH = CH-, = C (Me)- N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3613; C, -CH = CH-, = C (Me) -N =, -CH = CH-, -, OMe, H, H, H, O], [AH3614; C, -CH = C (CF 3) -, = CH-N =, - CH = CH -, -, H, H, H, H, O], [AH3615; C, -CH = C (CF 3) -, = CH-N =, - CH = CH -, -, Cl, H, H, H, O], [AH3616; C, -CH _{= C (CF 3) -,} = CH-N =, - CH = CH -, -, Br, H, H, H, O], [AH3617; C, -CH = C (CF 3) -, = CH -N =, - CH = CH - , -, CF 3, H, H, H, O], [AH3618; C, -CH = C (CF 3) -, = CH-N =, - CH = CH- , -, Me, H, H , H, O], [AH3619; C, -CH = C (CF 3) -, = CH-N =, - CH = CH -, -, Et, H, H, H , O], [AH 3620; C, -CH = C (CF ₃ )-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3621; C, -CH = C (CF ₃ )-, = CH-N =, - CH = CH -, -, OMe, H, H, H, O], [AH3622; C, -C (CF 3) = CH -, = = CH-N, - CH = CH -, -, H, H, H, H, O], [AH3623; C, -C (CF 3) = CH -, = CH-N =, - CH = CH -, -, Cl, H, H, H, O] , [AH3624; C, -C ( CF 3) = CH -, = CH-N =, - CH = CH -, -, Br, H, H, H, O], [AH3625; C, -C (CF _{3) = CH -, = CH} -N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3626; C, -C (CF 3) = CH -, = CH- N =, - CH = CH - , -, Me, H, H, H, O], [AH3627; C, -C (CF 3) = CH -, = CH-N =, - CH = CH -, - , Et, H, H, H , O], [AH3628; C, -C (CF 3) = CH -, = CH-N =, - CH = CH -, -, c-Pr, H, H, H , O], [AH 3629; C, -C (CF ₃ ) = CH-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3630; C,- CH = CH -, = C ( CF 3) -N =, - CH = CH -, -, H, H, H, H, O], [AH3631; C, -CH = CH -, = C (CF 3 ) -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3632; C, -CH = CH-, = C (CF ₃ ) -N =, -CH = CH- , -, Br, H, H , H, O], [AH3633; C, -CH = CH -, = C (CF 3) -N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3634; C, -CH = CH -, = C (CF 3) -N =, - CH = CH -, -, Me, H, H, H, O], [AH3635; C, -CH = CH -, = C ( CF 3) -N =, - CH = CH -, -, Et, H, H, H, O], [AH3636; C, -CH = CH -, = C (CF _{3) -N =, - CH =} CH -, -, c-Pr, H, H, H, O], [AH3637; C, -CH = CH -, = C (CF 3) -N =, - CH = CH-,-, OMe, H, H, H, O], [AH 3638; C, = CH-CH = CH-, -C (Me) =, -CH = CH-,-, H, H, H , H, O], [A H 3639; C, = CH-CH = CH-, -C (Me) =, -CH = CH-,-, Cl, H, H, H, O], [AH 3640; C, = CH-CH = CH- , -C (Me) =, -CH = CH-,-, Br, H, H, H, O], [AH3641; C, = CH-CH = CH-, -C (Me) =, -CH = _{CH -, -, CF 3,} H, H, H, O], [AH3642; C, = CH-CH = CH -, - C (Me) =, - CH = CH -, -, Me, H, H , H, O], [AH3643; C, = CH-CH = CH-, -C (Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 3644; C, = CH-CH = CH-, -C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3645; C, = CH-CH = CH-,- C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH 3646; C, = CH-CH = CF-, -C (Me) =, -CH = CH- ,-, H, H, H, H, O, [AH 3647; C, = CH-CH = CF-,-C (Me) =, -CH = CH-,-, Cl, H, H, H, H O, [AH 3648; C, = CH-CH = CF-, -C (Me) =, -CH = CH-,-, Br, H, H, H, O], [AH 3649; C, = CH- CH = CF -, - C ( Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH3650; C, = CH-CH = CF -, - C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH3651; C, = CH-CH = CF-, -C (Me) =, -CH = CH-,-, Et , H, H, H, O], [AH3652; C, = CH-CH = CF-, -C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O] , [AH3653; C, = CH-CH = CF-, -C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH3654; C, = CH-CF = CH-, -C (Me) =, -CH = CH-,-, H, H, H, H, O], [AH 3655; C, = CH-CF = CH-, -C (Me) =,- CH = CH-,-, Cl, H, H, H, O], [AH 3656; C, = CH-CF = CH-, -C (Me) =, -CH = CH-,-, Br, H, H, H, O], [ AH3657; C, = CH-CF = CH -, - C (Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH3658; C, = CH-CF = CH- , -C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH3659; C, = CH-CF = CH-, -C (Me) =, -CH = CH-,-, Et, H, H, H, H, O], [AH 3660; C, = CH-CF = CH-, -C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3661; C, = CH-CF = CH-, -C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH3662; C , = CF-CH = CH-, -C (Me) =, -CH = CH-,-, H, H, H, H, O], [AH3663; C, = CF-CH = CH-, -C (Me) =, -CH = CH-,-, Cl, H, H, H, O], [AH3664; C, = CF-CH = CH-, -C (Me) =, -CH = CH-, -, Br, H, H, H, O], [AH3665; C, = CF-CH = CH -, - C (Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH3666; C, = CF-CH = CH-, -C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH3667; C, = CF- CH = CH-, -C (Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 3668; C, = CF-CH = CH-, -C (Me) = , -CH = CH-,-, c-Pr, H, H, H, O], [AH3669; C, = CF-CH = CH-, -C (Me) =, -CH = CH-,-, OMe, H, H, H, O], [AH 3 670; C, = CH-CH = CH-, -C (Br) =, -CH = CH-,-, H, H, H, H, O], [AH 3671; C, = CH-CH = CH-, -C (Br) =, -CH = CH-,-, Cl, H, H, H, O], [AH 3672; C, = CH-CH = CH -, -C (Br) =, -CH = CH-,-, Br, H, H, H, O], [AH 3673; C, = CH-CH = CH-, -C (Br) =, -CH _{= CH -, -, CF 3} , H, H, H, O], [AH3674; C, = CH-CH = CH -, - C (Br) =, - CH = CH -, -, Me, H, H, H, O], [AH 3 675; C, = CH-CH = CH-, -C (Br) =, -CH = CH-,-, Et, H, H, H, O], [AH 3 676; C , = CH-CH = CH-, -C (Br) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3677; C, = CH-CH = CH-, -C (Br) =, -CH = CH-,-, OMe, H, H, H, O], [AH3678; C, = CH-CH = CH-, -C (Cl) =, -CH = CH-,-, H, H, H, H, O], [AH 3679; C, = CH-CH = CH-, -C (Cl) =, -CH = CH-,-, Cl, H, H, H, O], [AH 3 680; C, = CH-CH = CH -, -C (Cl) =, -CH = CH-,-, Br, H, H, H, O], [AH3681; C, = CH-CH = CH-, -C (Cl) =, -CH _{= CH -, -, CF 3} , H, H, H, O], [AH3682; C, = CH-CH = CH -, - C (Cl) =, - CH = CH -, -, Me, H, H, H, O], [AH3683; C, = CH-CH = CH-, -C (Cl) =, -CH = CH-,-, Et, H, H, H, O], [AH3684; C , = CH-CH = CH-, -C (Cl) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3685; C, = CH-CH = CH-, -C (Cl) =, -CH = CH-,-, OMe, H, H, H, O], [AH 3686; C, = CH-C (Me) = CH-, -C (Me) =,- CH = CH-,-, H, H, H, H, H, O], [AH 3687; C, = CH-C (Me) = CH-, -C (Me) =, -CH = CH-,-, Cl , H, H, H, O], [AH 3688; C, = CH-C (Me) = CH-,-C (Me) =, -CH = CH-,-, Br, H, H, H, O ], [AH3689; C, = CH-C (Me) = CH -, - C (Me) =, - CH = CH -, -, CF 3, H, H, H, O], [AH3690; C, = CH-C (Me) = CH-, -C (Me) =, -CH = CH-,-, Me, H, H, H, O], [AH3691; C, = CH-C (Me) = CH-, -C (Me) =, -CH = CH-,-, Et, H, H, H, O], [AH 3692; C, = CH-C (Me) = CH-, -C (Me) =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3693; C, = CH-C (Me) = CH-, -C (Me) =, -CH = CH -,-, OMe, H, H, H, O], [AH 3694; C, = CH-CH = CH-, -C (CF ₃ ) =, -CH = CH-,-, H, H, H, H, O], [AH3695; C, = CH-CH = CH -, - C (CF 3) =, - CH = CH -, -, Cl, H, H, H, O], [AH3696; C, = CH-CH = CH-,-C (CF ₃ ) =, -CH = CH-,-, Br, H, H, H, O], [AH 3697; C, = CH-CH = CH-, -C (CF ₃ ) =, -CH = CH-,-, _{CF 3, H, H, H} , O], [AH3698; C, = CH-CH = CH -, - C (CF 3) =, - CH = CH -, -, Me, H, H, H, O ], [AH3699; C, = CH-CH = CH -, - C (CF 3) =, - CH = CH -, -, Et, H, H, H, O], [AH3700; C, = CH- CH = CH -, - C ( CF 3) =, - CH = CH -, -, c-Pr, H, H, H, O],

[AH3701; C, = CH- CH = CH -, - C (CF 3) =, - CH = CH -, -, OMe, H, H, H, O], [AH3702; C, -CH = CH- , = CH-N =, -CH = CH-,-, H, H, H, H, O], [AH 3703; C, -CH = CH-, = CH-N =, -CH = CH-,- , Cl, H, H, H, O], [AH 3704; C, -CH = CH-, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [AH 3705 ; C, -CH = CH -, = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3706; C, -CH = CH -, = CH-N =, -CH = CH-,-, Me, H, H, H, O], [AH3707; C, -CH = CH-, = CH-N =, -CH = CH-,-, Et, H, H, H, O], [AH3708; C, -CH = CH-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3709; C, -CH = CH-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3710; C, -CH = CF-, = CH-N =, -CH = CH-,-, H, H, H, H, H, O], [AH 3711; C, -CH = CF-, = CH-N =, -CH = CH-,-, Cl, H, H, H, H O, [AH 3712; C, -CH = CF-, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [AH3713; C, -CH = CF-, = CH-N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3714; C, -CH = CF -, = CH-N =, - CH = CH -, - , Me, H, H, H, O], [AH3715; C, -CH = CF-, = CH-N =, -CH = CH-,-, Et, H, H, H, O], [AH3716 C, -CH = CF-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3717; C, -CF = CH-, = CH- N =, -CH = CH-,-, H, H, H, H, O], [AH3718; C, -CF = CH-, = CH-N =, -CH = CH-,-, Cl, H , H, H, O], [AH3719; C, -CF = CH-, = CH-N =, -CH = CH-,-, Br, H, H, H, O], [AH3720; C,- CF = CH -, = CH- N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3721; C, -CF = CH -, = CH-N =, - CH = CH-,-, Me, H, H , H, O], [AH 3722; C, -CF = CH-, = CH-N =, -CH = CH-,-, Et, H, H, H, O], [AH 3723; C, -CF = CH-, = CH-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3724; C, -CF = CH-, = CH-N =, -CH = CH-,-, OMe, H, H, H, O], [AH3725; C, -CH = CH-, = CF-N =, -CH = CH-,-, H, H, H, H, O ], [AH 3726; C, -CH = CH-, = CF-N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3727; C, -CH = CH-, = CF-N =, -CH = CH-,-, Br, H, H, H, O], [AH3728; C, -CH = CH-, = CF-N =, -CH = CH-,-, CF ₃ , H, H, H, O], [AH3729; C, -CH = CH-, = CF-N =, -CH = CH-,-, Me, H, H, H, O], [AH3730; C, -CH = CH-, = CF-N =, -CH = CH-,-, Et, H, H, H, O], [AH3731; C, -CH = CH-, = CF-N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH3732; C, -CH = CH-, = CF-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3733; C, = CH-CH = CH-, -CH =, -CH = CH-,-, H, H, H, H, O], [AH 3734; C, = CH -CH = CH-, -CH =, -CH = CH-,-, Cl, H, H, H, O], [AH3735; C, = CH-CH = CH-, -CH =, -CH = CH -, -, Br, H, H, H, O], [AH3736; C, = CH-CH = CH -, - CH =, - CH = CH -, -, CF 3, H, H, H, O ], [AH 3737; C, = CH-CH = CH-, -CH =, -CH = CH-,-, Me, H, H, H, O], [AH 3738; C, = CH-CH = CH- , -CH =, -CH = CH-,-, Et, H, H, H, O], [AH 3739; C, = CH-CH = CH-, -CH =, -CH = CH-,-, c -Pr, H, H, H, O], [AH3740; C, = CH-CH = CH-, -CH =, -CH = CH-,-, OMe, H, H, H, O], [AH3741 C, = CH-CH = CH-, -N =, -CH = CH-,-, H, H, H, H, O], [AH3742; C, = CH-CH = CH-, -N = , -CH = CH-,- , Cl, H, H, H, O], [AH 3743; C, = CH-CH = CH-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH 3744 ; C, = CH-CH = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3745; C, = CH-CH = CH -, - N =, -CH = CH-,-, Me, H, H, H, O], [AH 3746; C, = CH-CH = CH-, -N =, -CH = CH-,-, Et, H, H, H, O], [AH 3747; C, = CH-CH = CH-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3748; C, = CH-CH = CH-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3749; C, = CH-C (Me) = CH-, -N = , -CH = CH-,-, H, H, H, H, O, [AH 3750; C, = CH-C (Me) = CH-, -N =, -CH = CH-,-, Cl, H, H, H, O], [AH3751; C, = CH-C (Me) = CH-, -N =, -CH = CH-,-, Br, H, H, H, O], [AH3752 ; C, = CH-C ( Me) = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3753; C, = CH-C (Me) = CH-, -N =, -CH = CH-,-, Me, H, H, H, O], [AH 3754; C, = CH-C (Me) = CH-, -N =, -CH = CH-,-, Et, H, H, H, H, O], [AH 3755; C, = CH-C (Me) = CH-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3756; C, = CH-C (Me) = CH-,-N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3757; C , = C (Me) -CH = CH-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 3758; C, = C (Me) -CH = CH- , -N =, -CH = CH-,-, Cl, H, H, H, O], [AH 3759; C, = C (Me) -CH = CH-, -N =, -CH = CH-, -, Br, H, H, H, O], [AH3760; C, = C (Me) -CH = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3761; C, = C (Me) -CH = CH-, -N =, -CH = CH-,-, Me, H, H, H, O], [AH3762; C, = C ( Me) -CH = CH-, -N =, -CH = CH-,-, Et, H , H, H, O], [AH3763; C, = C (Me) -CH = CH-, -N =, -CH = CH-,-, c-Pr, H, H, H, O], [[ AH 3764; C, = C (Me) -CH = CH-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH 3765; C, = CH-C (CF ₃ ) = CH-, -N =, -CH = CH-,-, H, H, H, H, O], [AH 3766; C, = CH-C (CF ₃ ) = CH-, -N =,- CH = CH-,-, Cl, H, H, H, O], [AH 3767; C, = CH-C (CF ₃ ) = CH-, -N =, -CH = CH-,-, Br, H , H, H, O], [AH3768; C, = CH-C (CF 3) = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [ AH3769; C, = CH-C (CF 3) = CH -, - N =, - CH = CH -, -, Me, H, H, H, O], [AH3770; C, = CH-C (CF _{3) = CH -, - N} =, - CH = CH -, -, Et, H, H, H, O], [AH3771; C, = CH-C (CF 3) = CH -, - N =, -CH = CH-,-, c-Pr, H, H, H, O], [AH 3772; C, = CH-C (CF ₃ ) = CH-, -N =, -CH = CH-,-, OMe, H, H, H, O], [AH3773; C, = C (CF 3) -CH = CH -, - N =, - CH = CH -, -, H, H, H, H, O] , [AH3774; C, = C (CF 3) -CH = CH -, - N =, - CH = CH -, -, Cl, H, H, H, O], [AH3775; C, = C (CF _{3) -CH = CH -, -} N =, - CH = CH -, -, Br, H, H, H, O], [AH3776; C, = C (CF 3) -CH = CH -, - N =, - CH = CH -, -, CF 3, H, H, H, O], [AH3777; C, = C (CF 3) -CH = CH -, - N =, - CH = CH -, - , Me, H, H, H , O], [AH3778; C, = C (CF 3) -CH = CH -, - N =, - CH = CH -, -, Et, H, H, H, O ], [AH3779; C, = C (CF 3) -CH = CH -, - N =, - CH = CH -, -, c-Pr, H, H, H, O], [AH3780; C, = _{C (CF 3) -CH = CH} -, - N =, - CH = CH -, -, OMe, H, H, H, O].

[Substituent group number ^{(MH2); E 108]:} [BH1; 2-THA], [BH2; 4-F-2-THA], [BH3; 4-Cl-2-THA], [BH4; 4-Br -2-THA, [BH5; 4-I-2-THA], [BH6; 4-Me-2-THA], [BH7; 4-Et-2-THA], [BH8; 4-Pr-2 -THA], [BH9; 4- i-Pr-2-THA], [BH10; 4-CF 3 -2-THA], [BH11; 4-CHF 2 -2-THA], [BH12; 4-OMe -2-THA], [BH13; 4-OEt-2-THA], [BH14; 4-OCF 3 -2-THA], [BH15; 4-OCHF 2 -2-THA], [BH16; 4-CN -2-THA, [BH17; 4-SMe-2-THA], [BH18; 4-SEt-2-THA], [BH19; 4-c-Pr-2-THA], [BH20; 5-F -2-THA], [BH21; 5-Cl-2-THA], [BH22; 5-Br-2-THA], [BH23; 5-I-2-THA], [BH24; -THA], [BH25; 5-Et-2-THA], [BH26; 5-Pr-2-THA], [BH27; 5-i-Pr-2-THA], [BH28; 5-CF _3- 2-THA], [BH29; 5-CHF 2 -2-THA], [BH30; 5-OMe-2-THA], [BH31; 5-OEt-2-THA], [BH32; 5-OCF 3 - 2-THA], [BH33; 5-OCHF 2 -2-THA], [BH34; 5-CN-2-THA], [BH35; 5-SMe-2-THA], [BH36; 5-SEt-2 -THA], [BH37; 5-c-Pr-2-THA], [BH38; 4-F-5-F-2-THA], [BH39; 4-F-5-Cl-2-THA], [BH40; 4-F-5-Br-2-THA], [BH41; 4-F-5-I-2-THA], [BH42; 4-F-5-Me-2-THA], [BH43] 4-F-5-Et-2-THA], [BH44; 4-F-5-Pr-2-THA], [BH45; 4-F-5-i-Pr-2-THA], [BH46] ; 4-F-5-CF 3 -2-THA], [BH47; 4-F-5-CHF 2 -2-THA], [BH48; 4-F-5-OMe-2-THA], [BH49 4-F-5-OEt-2-T HA], [BH50; 4- F-5-OCF 3 -2-THA], [BH51; 4-F-5-OCHF 2 -2-THA], [BH52; 4-F-5-CN-2- THA], [BH53; 4-F-5-SMe-2-THA], [BH54; 4-F-5-SEt-2-THA], [BH55; 4-F-5-c-Pr-2-] THA], [BH56; 4-Cl-5-F-2-THA], [BH57; 4-Cl-5-Cl-2-THA], [BH58; 4-Cl-5-Br-2-THA] [BH59; 4-Cl-5-I-2-THA], [BH60; 4-Cl-5-Me-2-THA], [BH61; 4-Cl-5-Et-2-THA], [BH60; BH62; 4-Cl-5- Pr-2-THA], [BH63; 4-Cl-5-i-Pr-2-THA], [BH64; 4-Cl-5-CF 3 -2-THA], [BH65; 4-Cl-5 -CHF 2 -2-THA], [BH66; 4-Cl-5-OMe-2-THA], [BH67; 4-Cl-5-OEt-2-THA], [ BH68; 4-Cl-5- OCF 3 -2-THA], [BH69; 4-Cl-5-OCHF 2 -2-THA], [BH70; 4-Cl-5-CN-2-THA], [ BH71; 4-Cl-5-SMe-2-THA], [BH72; 4-Cl-5-SEt-2-THA], [BH73; 4-Cl-5-c-Pr-2-THA], [BH 73; BH74; 4-Me-5-F-2-THA], [BH75; 4-Me-5-Cl-2-THA], [BH76; 4-Me-5-Br-2-THA], [BH77; 4-Me-5-I-2-THA], [BH 78; 4-Me-5-Me-2-THA], [BH 79; 4-Me-5-Et-2-THA], [BH 80; Me-5-Pr-2- THA], [BH81; 4-Me-5-i-Pr-2-THA], [BH82; 4-Me-5-CF 3 -2-THA], [BH83; 4 _{-Me-5-CHF 2 -2-} THA], [BH84; 4-Me-5-OMe-2-THA], [BH85; 4-Me-5-OEt-2-THA], [BH86; 4- _{Me-5-OCF 3 -2-} THA], [BH87; 4-Me-5-OCHF 2 -2-THA], [BH88; 4-Me-5-CN-2-THA], [BH89; 4- Me-5-SMe-2-THA], [BH90; 4-Me-5-SEt-2-THA], [BH9 1; 4-Me-5-c-Pr-2-THA], [BH92; 4-Et-5-F-2-THA], [BH93; 4-Et-5-Cl-2-THA], [B. BH94; 4-Et-5-Br-2-THA], [BH95; 4-Et-5-I-2-THA], [BH96; 4-Et-5-Me-2-THA], [BH97; 4-Et-5-Et-2-THA], [BH98; 4-Et-5-Pr-2-THA], [BH99; 4-Et-5-i-Pr-2-THA], [BH100; 4-Et-5-CF ₃ -2-THA],

[BH101; 4-Et-5 -CHF 2 -2-THA], [BH102; 4-Et-5-OMe-2-THA], [BH103; 4-Et-5-OEt-2-THA], [ BH104; 4-Et-5- OCF 3 -2-THA], [BH105; 4-Et-5-OCHF 2 -2-THA], [BH106; 4-Et-5-CN-2-THA], [ BH107; 4-Et-5-SMe-2-THA], [BH108; 4-Et-5-SEt-2-THA], [BH109; 4-Et-5-c-Pr-2-THA], [BH109; _{BH110; 4-CF 3 -5-} F-2-THA], [BH111; 4-CF 3 -5-Cl-2-THA], [BH112; 4-CF 3 -5-Br-2-THA], _{[BH113; 4-CF 3 -5} -I-2-THA], [BH114; 4-CF 3 -5-Me-2-THA], [BH115; 4-CF 3 -5-Et-2-THA] _{, [BH116; 4-CF 3} -5-Pr-2-THA], [BH117; 4-CF 3 -5-i-Pr-2-THA], [BH118; 4-CF 3 -5-CF 3 - 2-THA], [BH119; 4-CF 3 -5-CHF 2 -2-THA], [BH120; 4-CF 3 -5-OMe-2-THA], [BH121; 4-CF 3 -5- OEt-2-THA], [ BH122; 4-CF 3 -5-OCF 3 -2-THA], [BH123; 4-CF 3 -5-OCHF 2 -2-THA], [BH124; 4-CF 3 -5-CN-2-THA !, [BH 125; 4-CF ₃ -5-SMe 2-THA], [BH 126; 4-CF ₃ -5-SEt-2-THA], [BH 127; _{3 -5-c-Pr-2} -THA], [BH128; 4-OMe-5-F-2-THA], [BH129; 4-OMe-5-Cl-2-THA], [BH130; 4- OMe-5-Br-2-THA], [BH131; 4-OMe-5-I-2-THA], [BH132; 4-OMe-5-Me-2-THA], [BH133; 4-OMe- 5-Et-2-THA], [BH134; 4-OMe-5-Pr-2-THA], [BH135; 4-OMe-5-i-Pr-2-THA], [BH136; 4-OMe- _{5-CF 3 -2-THA]} , [BH137; 4-OMe-5-CHF 2 -2-THA], [BH138; 4-OMe-5 -OMe-2-THA], [BH139; 4-OMe-5-OEt-2-THA], [BH140; 4-OMe-5-OCF 3 -2-THA], [ BH141; 4-OMe-5- OCHF 2 -2-THA], [BH142; 4-OMe-5-CN-2-THA], [BH143; 4-OMe-5-SMe-2-THA], [BH144 4-OMe-5-SEt-2-THA !, [BH145; 4-OMe-5-c-Pr-2-THA], [BH146; 4-OEt-5-F-2-THA], [BH147; 4-OEt-5-Cl-2-THA !, [BH148; 4-OEt-5-Br-2-THA], [BH149; 4-OEt-5-I-2-THA], [BH150; -OEt-5-Me-2-THA], [BH151; 4-OEt-5-Et-2-THA], [BH152; 4-OEt-5-Pr-2-THA], [BH153; 4-OEt -5-i-Pr-2- THA], [BH154; 4-OEt-5-CF 3 -2-THA], [BH155; 4-OEt-5-CHF 2 -2-THA], [BH156; 4 -OEt-5-OMe-2- THA], [BH157; 4-OEt-5-OEt-2-THA], [BH158; 4-OEt-5-OCF 3 -2-THA], [BH159; 4- _{OEt-5-OCHF 2 -2-} THA], [BH160; 4-OEt-5-CN-2-THA], [BH161; 4-OEt-5-SMe-2-THA], [BH162; 4-OEt -5-SEt-2-THA !, [BH163; 4-OEt-5-c-Pr-2-THA], [BH164; 4-SMe-5-F-2-THA], [BH165; 4-SMe -5-Cl-2-THA], [BH166; 4-SMe-5-Br-2-THA], [BH167; 4-SMe-5-I-2-THA], [BH168; 4-SMe-5 -Me-2-THA], [BH169; 4-SMe-5-Et-2-THA], [BH170; 4-SMe-5-Pr-2-THA], [BH171; 4-SMe-5-i -Pr-2-THA], [ BH172; 4-SMe-5-CF 3 -2-THA], [BH173; 4-SMe-5-CHF 2 -2-THA], [BH174; 4-SMe-5 -OMe-2-THA], [BH175; 4-SMe-5-OEt-2-THA], [BH1 76; 4-SMe-5- OCF 3 -2-THA], [BH177; 4-SMe-5-OCHF 2 -2-THA], [BH178; 4-SMe-5-CN-2-THA], [ BH179; 4-SMe-5-SMe-2-THA], [BH180; 4-SMe-5-SEt-2-THA], [BH181; 4-SMe-5-c-Pr-2-THA], [B. BH182; -4-THA], [BH183; 2-F-4-THA], [BH184; 2-Cl-4-THA], [BH185; 2-Br-4-THA], [BH186; 2-I -4-THA], [BH187; 2-Me-4-THA], [BH188; 2-Et-4-THA], [BH189; 2-Pr-4-THA], [BH190; 2-i-Pr -4-THA], [BH191; 2-CF 3 -4-THA], [BH192; 2-CHF 2 -4-THA], [BH193; 2-OMe-4-THA], [BH194; 2-OEt -4-THA], [BH195; 2-OCF 3 -4-THA], [BH196; 2-OCHF 2 -4-THA], [BH197; 2-CN-4-THA], [BH198; 2-SMe -4-THA], [BH 199; 2-SEt-4-THA], [BH 200; 2-c-Pr-4-THA],

[BH201; 5-F-4-THA], [BH202; 5-Cl-4-THA], [BH203; 5-Br-4-THA], [BH204; 5-I-4-THA], [BH205] 5-Me-4-THA], [BH206; 5-Et-4-THA], [BH207; 5-Pr-4-THA], [BH208; 5-i-Pr-4-THA], [BH209] _{; 5-CF 3 -4-THA} ], [BH210; 5-CHF 2 -4-THA], [BH211; 5-OMe-4-THA], [BH212; 5-OEt-4-THA], [BH213 _{; 5-OCF 3 -4-THA} ], [BH214; 5-OCHF 2 -4-THA], [BH215; 5-CN-4-THA], [BH216; 5-SMe-4-THA], [BH217 5-SEt-4-THA], [BH218; 5-c-Pr-4-THA], [BH219; 2-F-5-F-4-THA], [BH220; 2-F-5-Cl] -4-THA], [BH221; 2-F-5-Br-4-THA], [BH222; 2-F-5-I-4-THA], [BH223; 2-F-5-Me-4 -THA], [BH224; 2-F-5-Et-4-THA], [BH225; 2-F-5-Pr-4-THA], [BH226; 2-F-5-i-Pr-4 -THA], [BH227; 2- F-5-CF 3 -4-THA], [BH228; 2-F-5-CHF 2 -4-THA], [BH229; 2-F-5-OMe-4 -THA], [BH230; 2- F-5-OEt-4-THA], [BH231; 2-F-5-OCF 3 -4-THA], [BH232; 2-F-5-OCHF 2 -4 -THA], [BH233; 2-F-5-CN-4-THA], [BH234; 2-F-5-SMe-4-THA], [BH235; 2-F-5-SEt-4-THA ], [BH236; 2-F-5-c-Pr-4-THA], [BH237; 2-Cl-5-F-4-THA], [BH238; 2-Cl-5-Cl-4-THA ], [BH239; 2-Cl-5-Br-4-THA], [BH240; 2-Cl-5-I-4-THA], [BH241; 2-Cl-5-Me-4-THA], [BH242; 2-Cl-5-Et-4-THA], [BH243; 2-Cl-5-Pr-4-THA], [BH244; 2-Cl-5-i-Pr-4-THA], [BH245; 2 _{-Cl-5-CF 3 -4-} THA], [BH246; 2-Cl-5-CHF 2 -4-THA], [BH247; 2-Cl-5-OMe-4-THA], [BH248; 2 -Cl-5-OEt-4- THA], [BH249; 2-Cl-5-OCF 3 -4-THA], [BH250; 2-Cl-5-OCHF 2 -4-THA], [BH251; 2 -Cl-5-CN-4-THA], [BH252; 2-Cl-5-SMe-4-THA], [BH253; 2-Cl-5-SEt-4-THA], [BH254; 2-Cl -5-c-Pr-4-THA], [BH255; 2-Me-5-F-4-THA], [BH256; 2-Me-5-Cl-4-THA], [BH257; 2-Me -5-Br-4-THA], [BH258; 2-Me-5-I-4-THA], [BH259; 2-Me-5-Me-4-THA], [BH260; 2-Me-5 -Et-4-THA], [BH261; 2-Me-5-Pr-4-THA], [BH262; 2-Me-5-i-Pr-4-THA], [BH263; 2-Me-5 _{-CF 3 -4-THA], [} BH264; 2-Me-5-CHF 2 -4-THA], [BH265; 2-Me-5-OMe-4-THA], [BH266; 2-Me-5 -OEt-4-THA], [ BH267; 2-Me-5-OCF 3 -4-THA], [BH268; 2-Me-5-OCHF 2 -4-THA], [BH269; 2-Me-5 -CN-4-THA], [BH270; 2-Me-5-SMe-4-THA], [BH271; 2-Me-5-SEt-4-THA], [BH272; 2-Me-5-c -Pr-4-THA], [BH273; 2-Et-5-F-4-THA], [BH274; 2-Et-5-Cl-4-THA], [BH275; 2-Et-5-Br -4-THA], [BH 276; 2-Et-5-I-4-THA], [BH 277; 2-Et-5-Me-4-THA], [BH 278; 2-Et-5-Et-4 -THA], [BH279; 2-Et-5-Pr-4-THA], [BH280; 2-Et-5-i-Pr-4-THA], [BH281; 2-Et-5-CF _3- 4-THA], [BH282; 2-Et-5-CHF ₂ -4-THA], [BH 283; 2-Et-5-OMe-4-THA], [BH 284; 2-Et-5-OEt-4 - THA], [BH285; 2- Et-5-OCF 3 -4-THA], [BH286; 2-Et-5-OCHF 2 -4-THA], [BH287; 2-Et-5-CN-4- THA], [BH288; 2-Et-5-SMe-4-THA], [BH 289; 2-Et-5-SEt-4-THA], [BH290; 2-Et-5-c-Pr-4- THA], [BH291; 2- CF 3 -5-F-4-THA], [BH292; 2-CF 3 -5-Cl-4-THA], [BH293; 2-CF 3 -5-Br-4 -THA], [BH294; 2- CF 3 -5-I-4-THA], [BH295; 2-CF 3 -5-Me-4-THA], [BH296; 2-CF 3 -5-Et- 4-THA], [BH297; 2-CF 3 -5-Pr-4-THA], [BH298; 2-CF 3 -5-i-Pr-4-THA], [BH299; 2-CF 3 -5 _{-CF 3 -4-THA], [} BH300; 2-CF 3 -5-CHF 2 -4-THA],

_{[BH301; 2-CF 3 -5} -OMe-4-THA], [BH302; 2-CF 3 -5-OEt-4-THA], [BH303; 2-CF 3 -5-OCF 3 -4-THA ], [BH304; 2-CF 3 -5-OCHF 2 -4-THA], [BH305; 2-CF 3 -5-CN-4-THA], [BH306; 2-CF 3 -5-SMe-4 -THA], [BH307; 2- CF 3 -5-SEt-4-THA], [BH308; 2-CF 3 -5-c-Pr-4-THA], [BH309; 2-OMe-5-F -4-THA], [BH310; 2-OMe-5-Cl-4-THA], [BH311; 2-OMe-5-Br-4-THA], [BH312; 2-OMe-5-I-4 -THA], [BH313; 2-OMe-5-Me-4-THA], [BH314; 2-OMe-5-Et-4-THA], [BH315; 2-OMe-5-Pr-4-THA ], [BH316; 2-OMe -5-i-Pr-4-THA], [BH317; 2-OMe-5-CF 3 -4-THA], [BH318; 2-OMe-5-CHF 2 -4 -THA], [BH319; 2- OMe-5-OMe-4-THA], [BH320; 2-OMe-5-OEt-4-THA], [BH321; 2-OMe-5-OCF 3 -4- THA], [BH322; 2- OMe-5-OCHF 2 -4-THA], [BH323; 2-OMe-5-CN-4-THA], [BH324; 2-OMe-5-SMe-4-THA ], [BH325; 2-OMe-5-SEt-4-THA], [BH326; 2-OMe-5-c-Pr-4-THA], [BH327; 2-OEt-5-F-4-THA] ], [BH328; 2-OEt-5-Cl-4-THA], [BH329; 2-OEt-5-Br-4-THA], [BH330; 2-OEt-5-I-4-THA], [BH331; 2-OEt-5-Me-4-THA], [BH332; 2-OEt-5-Et-4-THA], [BH333; 2-OEt-5-Pr-4-THA], [BH334] ; 2-OEt-5-i -Pr-4-THA], [BH335; 2-OEt-5-CF 3 -4-THA], [BH336; 2-OEt-5-CHF 2 -4-THA], [BH 337; 2-OEt-5-OMe-4-THA], [BH 338; 2-OEt-5 -OEt-4-THA], [ BH339; 2-OEt-5-OCF 3 -4-THA], [BH340; 2-OEt-5-OCHF 2 -4-THA], [BH341; 2-OEt-5 -CN-4-THA], [BH342; 2-OEt-5-SMe-4-THA], [BH343; 2-OEt-5-SEt-4-THA], [BH344; 2-OEt-5-c -Pr-4-THA], [BH345; 2-SMe-5-F-4-THA], [BH346; 2-SMe-5-Cl-4-THA], [BH347; 2-SMe-5-Br -4-THA], [BH348; 2-SMe-5-I-4-THA], [BH349; 2-SMe-5-Me-4-THA], [BH350; 2-SMe-5-Et-4 -THA], [BH 351; 2-SMe-5-Pr-4-THA], [BH 352; 2-SMe-5-i-Pr-4-THA], [BH 353; 2-SMe-5-CF _3- 4-THA], [BH354; 2-SMe-5-CHF ₂ -4-THA], [BH 355; 2-SMe-5-OMe-4-THA], [BH 356; 2-SMe-5-OEt-4 -THA], [BH357; 2- SMe-5-OCF 3 -4-THA], [BH358; 2-SMe-5-OCHF 2 -4-THA], [BH359; 2-SMe-5-CN-4 -THA], [BH360; 2-SMe-5-SMe-4-THA], [BH361; 2-SMe-5-SEt-4-THA], [BH362; 2-SMe-5-c-Pr-4 -THA], [BH363; -5-THA], [BH 364; 2-F-5-THA], [BH365; 2-Cl-5-THA], [BH 366; 2-Br-5-THA], [B. BH367; 2-I-5-THA], [BH 368; 2-Me-5-THA], [BH 369; 2-Et-5-THA], [BH370; 2-Pr-5-THA], [BH 371; 2-i-Pr-5- THA], [BH372; 2-CF 3 -5-THA], [BH373; 2-CHF 2 -5-THA], [BH374; 2-OMe-5-THA], [ BH375; 2-OEt-5- THA], [BH376; 2-OCF 3 -5-THA], [BH377; 2-OCHF 2 -5-THA], [BH378; 2-CN-5-THA], [ BH379; 2-SMe-5-THA], [BH 380; 2-SEt-5- THA], [BH 381; 2-c-Pr-5-THA], [BH 382; 4-F-5-THA], [BH 383; 4-Cl-5-THA], [BH 384; THA], [BH 385; 4-I-5-THA], [BH 386; 4-Me-5-THA], [BH 387; 4-Et-5-THA], [BH 388; 4-Pr-5-THA] , [BH389; 4-i- Pr-5-THA], [BH390; 4-CF 3 -5-THA], [BH391; 4-CHF 2 -5-THA], [BH392; 4-OMe-5- THA], [BH 393; 4-OEt-5-THA], [BH 394; 4-OCF ₃ -5-THA], [BH 395; 4-OCHF ₂ -5-THA], [BH 396; THA], [BH397; 4-SMe-5-THA], [BH 398; 4-SEt-5-THA], [BH 399; 4-c-Pr-5-THA], [BH 400; 2-F-4- 2 F-5-THA],

[BH401; 2-F-4-Cl-5-THA], [BH402; 2-F-4-Br-5-THA], [BH403; 2-F-4-I-5-THA], [BH404] 2-F-4-Me-5-THA], [BH405; 2-F-4-Et-5-THA], [BH406; 2-F-4-Pr-5-THA], [BH407; -F-4-i-Pr- 5-THA], [BH408; 2-F-4-CF 3 -5-THA], [BH409; 2-F-4-CHF 2 -5-THA], [BH410 ; 2-F-4-OMe -5-THA], [BH411; 2-F-4-OEt-5-THA], [BH412; 2-F-4-OCF 3 -5-THA], [BH413; _{2-F-4-OCHF 2} -5-THA], [BH414; 2-F-4-CN-5-THA], [BH415; 2-F-4-SMe-5-THA], [BH416; 2 -F-4-SEt-5-THA], [BH417; 2-F-4-c-Pr-5-THA], [BH418; 2-Cl-4-F-5-THA], [BH419; -Cl-4-Cl-5-THA], [BH420; 2-Cl-4-Br-5-THA], [BH421; 2-Cl-4-I-5-THA], [BH422; 2-Cl -4-Me-5-THA], [BH 423; 2-Cl-4-Et-5-THA], [BH 424; 2-Cl-4-Pr-5-THA], [BH 425; 2-Cl-4 -i-Pr-5-THA] , [BH426; 2-Cl-4-CF 3 -5-THA], [BH427; 2-Cl-4-CHF 2 -5-THA], [BH428; 2-Cl -4-OMe-5-THA] , [BH429; 2-Cl-4-OEt-5-THA], [BH430; 2-Cl-4-OCF 3 -5-THA], [BH431; 2-Cl- _{4-OCHF 2 -5-THA]} , [BH432; 2-Cl-4-CN-5-THA], [BH433; 2-Cl-4-SMe-5-THA], [BH434; 2-Cl-4 -SEt-5-THA], [BH 435; 2-Cl-4-c-Pr-5-THA], [BH 436; 2-Me-4-F-5-THA], [BH 437; 2-Me-4 -Cl-5-THA], [BH 438; 2-Me-4-Br-5-THA], [BH 439; 2-Me-4-I-5-THA], [BH 440; 2-Me-4-Me -5-THA], [BH 441; 2-Me-4- Et-5-THA], [BH 442; 2-Me-4-Pr-5-THA], [BH 443; 2-Me-4-i-Pr-5-THA], [BH 444; _{CF 3 -5-THA], [} BH445; 2-Me-4-CHF 2 -5-THA], [BH446; 2-Me-4-OMe-5-THA], [BH447; 2-Me-4- OEt-5-THA], [ BH448; 2-Me-4-OCF 3 -5-THA], [BH449; 2-Me-4-OCHF 2 -5-THA], [BH450; 2-Me-4- CN-5-THA], [BH 451; 2-Me-4-SMe-5-THA], [BH 452; 2-Me-4-SEt-5-THA], [BH 453; 2-Me-4-c- Pr-5-THA], [BH454; 2-Et-4-F-5-THA], [BH455; 2-Et-4-Cl-5-THA], [BH456; 2-Et-4-Br- 5-THA], [BH457; 2-Et-4-I-5-THA], [BH458; 2-Et-4-Me-5-THA], [BH459; 2-Et-4-Et-5- THA], [BH460; 2- Et-4-Pr-5-THA], [BH461; 2-Et-4-i-Pr-5-THA], [BH462; 2-Et-4-CF 3 -5 -THA], [BH463; 2- Et-4-CHF 2 -5-THA], [BH464; 2-Et-4-OMe-5-THA], [BH465; 2-Et-4-OEt-5- THA], [BH466; 2- Et-4-OCF 3 -5-THA], [BH467; 2-Et-4-OCHF 2 -5-THA], [BH468; 2-Et-4-CN-5- THA], [BH 469; 2-Et-4-SMe-5-THA], [BH 470; 2-Et-4-SEt-5-THA], [BH 471; 2-Et-4-c-Pr-5- THA], [BH 472; 2-CF ₃ -4-F-5-THA], [BH 473; 2-CF ₃ -4-Cl-5-THA], [BH 474; 2-CF ₃ -4-Br-5] -THA], [BH475; 2- CF 3 -4-I-5-THA], [BH476; 2-CF 3 -4-Me-5-THA], [BH477; 2-CF 3 -4-Et- 5-THA], [BH 478; 2-CF ₃ -4-Pr-5-THA], [BH 479; 2-CF ₃ -4-i-Pr-5-THA], [BH 480; _{-CF 3 -4-CF 3 -5-} THA], [BH481; 2-CF 3 -4-CHF 2 -5-THA], [BH482; 2-CF 3 -4-OMe-5-THA], [ _{BH483; 2-CF 3 -4-} OEt-5-THA], [BH484; 2-CF 3 -4-OCF 3 -5-THA], [BH485; 2-CF 3 -4-OCHF 2 -5-THA ], [BH486; 2-CF 3 -4-CN-5-THA], [BH487; 2-CF 3 -4-SMe-5-THA], [BH488; 2-CF 3 -4-SEt-5- THA], [BH 489; 2-CF ₃ -4-c-Pr-5-THA], [BH 490; 2-OMe-4-F-5-THA], [BH 491; 2-OMe-4-Cl-5 -THA], [BH492; 2-OMe-4-Br-5-THA], [BH493; 2-OMe-4-I-5-THA], [BH494; 2-OMe-4-Me-5-THA ], [BH495; 2-OMe-4-Et-5-THA], [BH496; 2-OMe-4-Pr-5-THA], [BH497; 2-OMe-4-i-Pr-5-THA ], [BH498; 2-OMe -4-CF 3 -5-THA], [BH499; 2-OMe-4-CHF 2 -5-THA], [BH500; 2-OMe-4-OMe-5-THA ],

[BH501; 2-OMe-4 -OEt-5-THA], [BH502; 2-OMe-4-OCF 3 -5-THA], [BH503; 2-OMe-4-OCHF 2 -5-THA], [BH504; 2-OMe-4-CN-5-THA], [BH505; 2-OMe-4-SMe-5-THA], [BH506; 2-OMe-4-SEt-5-THA], [BH507] 2-OMe-4-c-Pr-5-THA], [BH508; 2-OEt-4-F-5-THA], [BH509; 2-OEt-4-Cl-5-THA], [BH510] 2-OEt-4-Br-5-THA], [BH511; 2-OEt-4-I-5-THA], [BH512; 2-OEt-4-Me-5-THA], [BH513; -OEt-4-Et-5-THA], [BH514; 2-OEt-4-Pr-5-THA], [BH515; 2-OEt-4-i-Pr-5-THA], [BH516; 2 _{-OEt-4-CF 3 -5-} THA], [BH517; 2-OEt-4-CHF 2 -5-THA], [BH518; 2-OEt-4-OMe-5-THA], [BH519; 2 -OEt-4-OEt-5- THA], [BH520; 2-OEt-4-OCF 3 -5-THA], [BH521; 2-OEt-4-OCHF 2 -5-THA], [BH522; 2 -OEt-4-CN-5-THA], [BH523; 2-OEt-4-SMe-5-THA], [BH524; 2-OEt-4-SEt-5-THA], [BH525; 2-OEt -4-c-Pr-5-THA], [BH 526; 2-SMe-4-F-5-THA], [BH 527; 2-SMe-4-Cl-5-THA], [BH 528; 2-SMe -4-Br-5-THA], [BH 529; 2-SMe-4-I-5-THA], [BH 530; 2-SMe-4-Me-5-THA], [BH 531; 2-SMe-4 -Et-5-THA], [BH532; 2-SMe-4-Pr-5-THA], [BH533; 2-SMe-4-i-Pr-5-THA], [BH534; 2-SMe-4 _{-CF 3 -5-THA], [} BH535; 2-SMe-4-CHF 2 -5-THA], [BH536; 2-SMe-4-OMe-5-THA], [BH537; 2-SMe-4 -OEt-5-THA], [ BH538; 2-SMe-4-OCF 3 -5-THA], [ BH539; 2-SMe-4- OCHF 2 -5-THA], [BH540; 2-SMe-4-CN-5-THA], [BH541; 2-SMe-4-SMe-5-THA], [BH542 2-SMe-4-SEt-5-THA !, [BH543; 2-SMe-4-c-Pr-5-THA], [BH544; 2-OXAA], [BH545; 4-F-2-OXAA] ], [BH546; 4-Cl-2-OXAA], [BH547; 4-Br-2-OXAA], [BH 548; 4-I-2-OXAA], [BH549; 4-Me-2-OXA], [BH550; 4-Et-2-OXA], [BH 551; 4-Pr-2-OXA], [BH 552; 4-i-Pr-2-OXA], [BH 553; 4-CF ₃ -2-OXA] _{, [BH554; 4-CHF 2} -2-OXA], [BH555; 4-OMe-2-OXA], [BH556; 4-OEt-2-OXA], [BH557; 4-OCF 3 -2-OXA] _{, [BH558; 4-OCHF 2} -2-OXA], [BH559; 4-CN-2-OXA], [BH560; 4-SMe-2-OXA], [BH561; 4-SEt-2-OXA], [BH562; 4-c-Pr-2-OXA], [BH563; 5-F-2-OXA], [BH 564; 5-Cl-2-OXA], [BH 565; 5-Br-2-OXA], [BH566; 5-I-2-OXA], [BH 567; 5-Me-2-OXA], [BH 568; 5-Et-2-OXA], [BH569; 5-Pr-2-OXA], [BH570] ; 5-i-Pr-2 -OXA], [BH571; 5-CF 3 -2-OXA], [BH572; 5-CHF 2 -2-OXA], [BH573; 5-OMe-2-OXA], [BH574; 5-OEt-2 -OXA], [BH575; 5-OCF 3 -2-OXA], [BH576; 5-OCHF 2 -2-OXA], [BH577; 5-CN-2-OXA], [BH578; 5-SMe-2-OXA], [BH579; 5-SEt-2-OXA], [BH580; 5-c-Pr-2-OXA], [BH581; 4-F-5-F-2 4-OXA], [BH582; 4-F-5-Cl-2-OXA], [BH583; 4-F-5-Br-2-OXA], [BH584; 4-F-5-I-2-OXA] ], [BH585; 4-F-5-Me-2-OXA], [BH586; 4-F-5-Et-2-OXA], [BH 587; 4-F-5-Pr-2-OXA], [BH 588; 4-F-5-i-Pr-2-OXA], [BH 589; _{4-F-5-CF 3} -2-OXA], [BH590; 4-F-5-CHF 2 -2-OXA], [BH591; 4-F-5-OMe-2-OXA], [BH592; 4-F-5-OEt- 2-OXA], [BH593; 4-F-5-OCF 3 -2-OXA], [BH594; 4-F-5-OCHF 2 -2-OXA], [BH595; 4-F-5-CN-2-OXA], [BH596; 4-F-5-SMe-2-OXA], [BH597; 4-F-5-SEt-2-OXA], [BH598; F-5-c-Pr-2-OXA], [BH599; 4-Cl-5-F-2-OXA], [BH600; 4-Cl-5-Cl-2-OXA],

[BH601; 4-Cl-5-Br-2-OXA], [BH602; 4-Cl-5-I-2-OXA], [BH603; 4-Cl-5-Me-2-OXA], [BH604] 4-Cl-5-Et-2-OXA], [BH605; 4-Cl-5-Pr-2-OXA], [BH606; 4-Cl-5-i-Pr-2-OXA], [BH607] ; 4-Cl-5-CF 3 -2-OXA], [BH608; 4-Cl-5-CHF 2 -2-OXA], [BH609; 4-Cl-5-OMe-2-OXA], [BH610 ; 4-Cl-5-OEt -2-OXA], [BH611; 4-Cl-5-OCF 3 -2-OXA], [BH612; 4-Cl-5-OCHF 2 -2-OXA], [BH613 4-Cl-5-CN-2-OXA], [BH614; 4-Cl-5-SMe-2-OXA], [BH615; 4-Cl-5-SEt-2-OXA], [BH616; -Cl-5-c-Pr-2-OXA], [BH617; 4-Me-5-F-2-OXA], [BH 618; 4-Me-5-Cl-2-OXA], [BH 619; 4 -Me-5-Br-2-OXA], [BH620; 4-Me-5-I-2-OXA], [BH621; 4-Me-5-Me-2-OXA], [BH622; 4-Me -5-Et-2-OXA], [BH623; 4-Me-5-Pr-2-OXA], [BH 624; 4-Me-5-i-Pr-2-OXA], [BH 625; 4-Me -5-CF ₃ -2-OXA !, [BH 626; 4-Me-5-CHF ₂ -2-OXA], [BH 627; 4-Me-5-OMe-2-OXA], [BH 628; 4-Me -5-OEt-2-OXA], [BH 629; 4-Me-5-OCF ₃ -2-OXA], [BH 630; 4-Me-5-OCHF ₂ -2-OXA], [BH 631; 4-Me -5-CN-2-OXA], [BH 632; 4-Me-5-SMe-2-OXA], [BH 633; 4-Me-5-SEt-2-OXA], [BH 634; 4-Me-5 -c-Pr-2-OXA], [BH 635; 4-Et-5-F-2-OXA], [BH 636; 4-Et-5-Cl-2-OXA], [BH 637; 4-Et-5 4-Br-2-OXA], [BH638; 4-Et-5-I-2-OXA], [BH639; 4-Et-5-Me-2-OXA], [BH640; 4-Et-5-Et -2-OX A], [BH641; 4-Et-5-Pr-2-OXA], [BH 642; 4-Et-5-i-Pr-2-OXA], [BH643; 4-Et-5-CF ₃ -2 -OXA], [BH644; 4- Et-5-CHF 2 -2-OXA], [BH645; 4-Et-5-OMe-2-OXA], [BH646; 4-Et-5-OEt-2- OXA], [BH647; 4- Et-5-OCF 3 -2-OXA], [BH648; 4-Et-5-OCHF 2 -2-OXA], [BH649; 4-Et-5-CN-2- OXA], [BH650; 4-Et-5-SMe-2-OXA], [BH651; 4-Et-5-SEt-2-OXA], [BH652; 4-Et-5-c-Pr-2- OXA], [BH653; 4- CF 3 -5-F-2-OXA], [BH654; 4-CF 3 -5-Cl-2-OXA], [BH655; 4-CF 3 -5-Br-2 -OXA], [BH656; 4- CF 3 -5-I-2-OXA], [BH657; 4-CF 3 -5-Me-2-OXA], [BH658; 4-CF 3 -5-Et- 2-OXA], [BH659; 4-CF 3 -5-Pr-2-OXA], [BH660; 4-CF 3 -5-i-Pr-2-OXA], [BH661; 4-CF 3 -5 _{-CF 3 -2-OXA], [} BH662; 4-CF 3 -5-CHF 2 -2-OXA], [BH663; 4-CF 3 -5-OMe-2-OXA], [BH664; 4-CF _{3 -5-OEt-2-OXA} ], [BH665; 4-CF 3 -5-OCF 3 -2-OXA], [BH666; 4-CF 3 -5-OCHF 2 -2-OXA], [BH667; _{4-CF 3 -5-CN-} 2-OXA], [BH668; 4-CF 3 -5-SMe-2-OXA], [BH669; 4-CF 3 -5-SEt-2-OXA], [BH670 _{; 4-CF 3 -5-c} -Pr-2-OXA], [BH671; 4-OMe-5-F-2-OXA], [BH672; 4-OMe-5-Cl-2-OXA], [ BH673; 4-OMe-5-Br-2-OXA], [BH674; 4-OMe-5-I-2-OXA], [BH675; 4-OMe-5-Me-2-OXA], [BH676; 4-OMe-5-Et-2-OXA], [BH 677; 4-OMe-5-Pr-2-OXA], [BH 6 78; 4-OMe-5-i-Pr-2-OXA], [BH 679; 4-OMe-5-CF ₃ -2-OXA], [BH 680; 4-OMe-5-CHF ₂ -2-OXA] 4- [OMe-5-OMe-2-OXA], [BH682; 4-OMe-5-OEt-2-OXA], [BH683; 4-OMe-5-OCF ₃ 2-OXA], [BH684; 4-OMe-5 -OCHF 2 -2-OXA], [BH685; 4-OMe-5-CN-2-OXA], [BH686; 4-OMe-5-SMe-2-OXA], [ BH687; 4-OMe-5-SEt-2-OXA], [BH688; 4-OMe-5-c-Pr-2-OXA], [BH689; 4-OEt-5-F-2-OXA], [BH 687; BH 690; 4-OEt-5-Cl-2-OXA !, [BH691; 4-OEt-5-Br-2-OXA], [BH692; 4-OEt-5-I-2-OXA], [BH693; 4-OEt-5-Me-2-OXA], [BH694; 4-OEt-5-Et-2-OXA], [BH695; 4-OEt-5-Pr-2-OXA], [BH696; 4- OEt-5-i-Pr-2-OXA], [BH 697; 4-OEt-5-CF ₃ -2-OXA], [BH 698; 4-OEt-5-CHF ₂ -2-OXA], [BH 699; 4-OEt-5-OMe-2-OXA], [BH700; 4-OEt-5-OEt-2-OXA],

[BH701; 4-OEt-5 -OCF 3 -2-OXA], [BH702; 4-OEt-5-OCHF 2 -2-OXA], [BH703; 4-OEt-5-CN-2-OXA], [BH704; 4-OEt-5-SMe-2-OXA], [BH705; 4-OEt-5-SEt-2-OXA], [BH706; 4-OEt-5-c-Pr-2-OXA], [BH707; 4-SMe-5-F-2-OXA], [BH708; 4-SMe-5-Cl-2-OXA], [BH709; 4-SMe-5-Br-2-OXA], [BH710] 4-SMe-5-I-2-OXA], [BH711; 4-SMe-5-Me-2-OXA], [BH712; 4-SMe-5-Et-2-OXA], [BH713; 4 -SMe-5-Pr-2-OXA], [BH714; 4-SMe-5-i-Pr-2-OXA], [BH715; 4-SMe-5-CF ₃ -2-OXA], [BH716; _{4-SMe-5-CHF 2} -2-OXA], [BH717; 4-SMe-5-OMe-2-OXA], [BH718; 4-SMe-5-OEt-2-OXA], [BH719; 4 _{-SMe-5-OCF 3 -2-} OXA], [BH720; 4-SMe-5-OCHF 2 -2-OXA], [BH721; 4-SMe-5-CN-2-OXA], [BH722; 4 -SMe-5-SMe-2-OXA], [BH 723; 4-SMe-5-SEt-2-OXA], [BH724; 4-SMe-5-c-Pr-2-OXA], [BH 725; 4-OXA], [BH 726; 2-F-4-OXA], [BH 727; 2-Cl-4-OXA], [BH 728; 2-Br-4-OXA], [BH 729; 2-I-4-] OXA], [BH730; 2-Me-4-OXA], [BH731; 2-Et-4-OXA], [BH732; 2-Pr-4-OXA], [BH733; 2-i-Pr-4- OXA], [BH734; 2- CF 3 -4-OXA], [BH735; 2-CHF 2 -4-OXA], [BH736; 2-OMe-4-OXA], [BH737; 2-OEt-4- OXA], [BH738; 2- OCF 3 -4-OXA], [BH739; 2-OCHF 2 -4-OXA], [BH740; 2-CN-4-OXA], [BH741; 2-SMe-4- OXA], [BH 742; 2-SEt-4-OXA], [BH 743; 2-c-Pr-4-OXA], [BH744; 5-F-4-OXA], [BH745; 5-Cl-4-OXA], [BH746; 5-Br-4-OXA], [BH747; 5-I-4-OXA], [BH 748; 5-Me-4-OXA], [BH 749; 5-Et-4-OXA], [BH 750; 5-Pr-4-OXA], [BH 751; 5-] i-Pr-4-OXA] , [BH752; 5-CF 3 -4-OXA], [BH753; 5-CHF 2 -4-OXA], [BH754; 5-OMe-4-OXA], [BH755; 5-OEt-4-OXA] , [BH756; 5-OCF 3 -4-OXA], [BH757; 5-OCHF 2 -4-OXA], [BH758; 5-CN-4-OXA], [BH759; 5-SMe-4-OXA], [BH760; 5-SEt-4-OXA], [BH761; 5-c-Pr-4-OXA], [BH762; 2-F-5-F-4-OXA] , [BH763; 2-F-5-Cl-4-OXA], [BH764; 2-F-5-Br-4-OXA], [BH765; 2-F-5-I-4-OXA], [BH 763; BH 766; 2-F-5-Me-4-OXA], [BH 767; 2-F-5-Et-4-OXA], [BH 768; 2-F-5-Pr-4-OXA], [BH 769; 2-F-5-i-Pr-4-OXA], [BH 770; 2-F-5-CF ₃ -4-OXA], [BH 771; 2-F-5-CHF ₂ -4-OXA], [B. BH772; 2-F-5- OMe-4-OXA], [BH773; 2-F-5-OEt-4-OXA], [BH774; 2-F-5-OCF 3 -4-OXA], [BH775 2-F-5-OCHF ₂ -4-OXA], [BH 776; 2-F-5-CN-4-OXA], [BH 777; 2-F-5-SMe-4-OXA], [BH 778; 2-F-5-SEt-4-OXA], [BH 779; 2-F-5-c-Pr-4-OXA], [BH780; 2-Cl-5-F-4-OXA], [BH 781; 2-Cl-5-Cl-4-OXA], [BH782; 2-Cl-5-Br-4-OXA], [BH783; 2-Cl-5-I-4-OXA], [BH784; 2- Cl-5-Me-4-OXA], [BH785; 2-Cl-5-Et-4-OXA], [BH 786; 2-Cl-5-Pr-4-OXA], [BH787; 2-Cl- 5-i-Pr-4 -OXA], [BH788; 2- Cl-5-CF 3 -4-OXA], [BH789; 2-Cl-5-CHF 2 -4-OXA], [BH790; 2-Cl-5-OMe-4 -OXA], [BH791; 2- Cl-5-OEt-4-OXA], [BH792; 2-Cl-5-OCF 3 -4-OXA], [BH793; 2-Cl-5-OCHF 2 -4 -OXA], [BH 794; 2-Cl-5-CN-4-OXA], [BH795; 2-Cl-5-SMe-4-OXA], [BH796; 2-Cl-5-SEt-4-OXA ], [BH 797; 2-Cl-5-c-Pr-4-OXA], [BH 798; 2-Me-5-F-4-OXA], [BH 799; 2-Me-5-Cl-4-OXA ], [BH800; 2-Me-5-Br-4-OXA],

[BH801; 2-Me-5-I-4-OXA], [BH802; 2-Me-5-Me-4-OXA], [BH803; 2-Me-5-Et-4-OXA], [BH804 2-Me-5-Pr-4-OXA], [BH 805; 2-Me-5-i-Pr-4-OXA], [BH806; 2-Me-5-CF ₃ -4-OXA], [B. BH 807; 2-Me-5-CHF ₂ -4-OXA], [BH 808; 2-Me-5-OMe-4-OXA], [BH 809; 2-Me-5-OEt-4-OXA], [BH 810] ; 2-Me-5-OCF 3 -4-OXA], [BH811; 2-Me-5-OCHF 2 -4-OXA], [BH812; 2-Me-5-CN-4-OXA], [BH813 2-Me-5-SMe-4-OXA], [BH814; 2-Me-5-SEt-4-OXA], [BH815; 2-Me-5-c-Pr-4-OXA], [BH816; 2-Et-5-F-4-OXA], [BH817; 2-Et-5-Cl-4-OXA], [BH818; 2-Et-5-Br-4-OXA], [BH819; -Et-5-I-4-OXA], [BH820; 2-Et-5-Me-4-OXA], [BH821; 2-Et-5-Et-4-OXA], [BH822; 2-Et -5-Pr-4-OXA] , [BH823; 2-Et-5-i-Pr-4-OXA], [BH824; 2-Et-5-CF 3 -4-OXA], [BH825; 2- Et-5-CHF ₂ -4-OXA], [BH 826; 2-Et-5-OMe-4-OXA], [BH 827; 2-Et-5-OEt-4-OXA], [BH 828; 2-Et -5-OCF ₃ -4-OXA], [BH 829; 2-Et-5-OCHF ₂ -4-OXA], [BH 830; 2-Et-5-CN-4-OXA], [BH 831; 2-Et -5-SMe-4-OXA], [BH 832; 2-Et-5-SEt-4-OXA], [BH 833; 2-Et-5-c-Pr-4-OXA], [BH 834; 2-CF _{3 -5-F-4-OXA} ], [BH835; 2-CF 3 -5-Cl-4-OXA], [BH836; 2-CF 3 -5-Br-4-OXA], [BH837; 2- _{CF 3 -5-I-4-} OXA], [BH838; 2-CF 3 -5-Me-4-OXA], [BH839; 2-CF 3 -5-Et-4-OXA], [BH _{840; 2-CF 3 -5-} Pr-4-OXA], [BH841; 2-CF 3 -5-i-Pr-4-OXA], [BH842; 2-CF 3 -5-CF 3 -4- OXA], [BH843; 2- CF 3 -5-CHF 2 -4-OXA], [BH844; 2-CF 3 -5-OMe-4-OXA], [BH845; 2-CF 3 -5-OEt- 4-OXA], [BH846; 2-CF 3 -5-OCF 3 -4-OXA], [BH847; 2-CF 3 -5-OCHF 2 -4-OXA], [BH848; 2-CF 3 -5 -CN-4-OXA], [ BH849; 2-CF 3 -5-SMe-4-OXA], [BH850; 2-CF 3 -5-SEt-4-OXA], [BH851; 2-CF 3 - 5-c-Pr-4-OXA], [BH 852; 2-OMe-5-F-4-OXA], [BH 853; 2-OMe-5-Cl-4-OXA], [BH 854; 2-OMe- 5-Br-4-OXA], [BH 855; 2-OMe-5-I-4-OXA], [BH 856; 2-OMe-5-Me-4-OXA], [BH 857; 2-OMe-5- Et-4-OXA], [BH 858; 2-OMe-5-Pr-4-OXA], [BH 859; 2-OMe-5-i-Pr-4-OXA], [BH 860; 2-OMe-5- _{CF 3 -4-OXA], [} BH861; 2-OMe-5-CHF 2 -4-OXA], [BH862; 2-OMe-5-OMe-4-OXA], [BH863; 2-OMe-5- OEt-4-OXA], [ BH864; 2-OMe-5-OCF 3 -4-OXA], [BH865; 2-OMe-5-OCHF 2 -4-OXA], [BH866; 2-OMe-5- CN-4-OXA], [BH867; 2-OMe-5-SMe-4-OXA], [BH868; 2-OMe-5-SEt-4-OXA], [BH869; 2-OMe-5-c- Pr-4-OXA], [BH870; 2-OEt-5-F-4-OXA], [BH871; 2-OEt-5-Cl-4-OXA], [BH872; 2-OEt-5-Br- 4-OXA], [BH 873; 2-OEt-5-I-4-OXA], [BH 874; 2-OEt-5-Me-4-OXA], [BH 875; 2-OEt-5-Et-4- OXA], [BH 876; 2-OEt-5-Pr-4-OXA], [BH 877; 2-O Et-5-i-Pr- 4-OXA], [BH878; 2-OEt-5-CF 3 -4-OXA], [BH879; 2-OEt-5-CHF 2 -4-OXA], [BH880; 2-OEt-5-OMe- 4-OXA], [BH881; 2-OEt-5-OEt-4-OXA], [BH882; 2-OEt-5-OCF 3 -4-OXA], [BH883; 2 2-OEt-5-OCHF ₂ -4-OXA !, [BH 884; 2-OEt-5-CN-4-OXA], [BH 885; 2-OEt-5-SMe-4-OXA], [BH 886; OEt-5-SEt-4-OXA], [BH887; 2-OEt-5-c-Pr-4-OXA], [BH888; 2-SMe-5-F-4-OXA], [BH889; SMe-5-Cl-4-OXA], [BH890; 2-SMe-5-Br-4-OXA], [BH891; 2-SMe-5-I-4-OXA], [BH892; 2-SMe- 5-Me-4-OXA], [BH893; 2-SMe-5-Et-4-OXA], [BH894; 2-SMe-5-Pr-4-OXA], [BH895; 2-SMe-5- i-Pr-4-OXA] , [BH896; 2-SMe-5-CF 3 -4-OXA], [BH897; 2-SMe-5-CHF 2 -4-OXA], [BH898; 2-SMe- 5-OMe-4-OXA] , [BH899; 2-SMe-5-OEt-4-OXA], [BH900; 2-SMe-5-OCF 3 -4-OXA],

[BH901; 2-SMe-5-OCHF ₂ -4-OXA], [BH 902; 2-SMe-5-CN-4-OXA], [BH 903; 2-SMe-5-SMe-4-OXA], [BH 901; BH904; 2-SMe-5-SEt-4-OXA], [BH905; 2-SMe-5-c-Pr-4-OXA], [BH906; 5-OXA], [BH 907; 2-F-5 2-OXA], [BH 908; 2-Cl-5-OXA], [BH 909; 2-Br-5-OXA], [BH 910; 2-I-5-OXA], [BH 911; 2-Me-5-OXA ], [BH912; 2-Et -5-OXA], [BH913; 2-Pr-5-OXA], [BH914; 2-i-Pr-5-OXA], [BH915; 2-CF 3 -5- OXA], [BH916; 2- CHF 2 -5-OXA], [BH917; 2-OMe-5-OXA], [BH918; 2-OEt-5-OXA], [BH919; 2-OCF 3 -5- OXA], [BH920; 2-OCHF ₂ -5-OXA], [BH 921; 2-CN-5-OXA], [BH 922; 2-SMe-5-OXA], [BH 923; 2-SEt-5-OXA ], [BH 924; 2-c-Pr-5-OXA], [BH 925; 4-F-5-OXA], [BH 926; 4-Cl-5-OXA], [BH 927; 4-Br-5-OXA] ], [BH 928; 4-I-5-OXA], [BH 929; 4-Me-5- OXA], [BH 930; 4-Et-5- OXA], [BH 931; 4-Pr-5-OXA], [BH932; 4-i-Pr -5-OXA], [BH933; 4-CF 3 -5-OXA], [BH934; 4-CHF 2 -5-OXA], [BH935; 4-OMe-5-OXA ], [BH936; 4-OEt -5-OXA], [BH937; 4-OCF 3 -5-OXA], [BH938; 4-OCHF 2 -5-OXA], [BH939; 4-CN-5-OXA ], [BH 940; 4-SMe-5-OXA], [BH 941; 4-SEt-5-OXA], [BH 942; 4-c-Pr-5-OXA], [BH 943; 2-F-4-F -5-OXA], [BH 944; 2-F-4-Cl-5-OXA], [BH 945; 2-F-4-Br-5-OXA], [BH 946; 2-F-4-I-5 -OXA], [BH947; 2-F-4-Me-5-OXA], [BH948; 2-F -4-Et-5-OXA], [BH949; 2-F-4-Pr-5-OXA], [BH950; 2-F-4-i-Pr-5-OXA], [BH951; 2-F _{-4-CF 3 -5-OXA]} , [BH952; 2-F-4-CHF 2 -5-OXA], [BH953; 2-F-4-OMe-5-OXA], [BH954; 2-F -4-OEt-5-OXA] , [BH955; 2-F-4-OCF 3 -5-OXA], [BH956; 2-F-4-OCHF 2 -5-OXA], [BH957; 2-F -4-CN-5-OXA], [BH958; 2-F-4-SMe-5-OXA], [BH959; 2-F-4-SEt-5-OXA], [BH960; 2-F-4 -c-Pr-5-OXA], [BH961; 2-Cl-4-F-5-OXA], [BH962; 2-Cl-4-Cl-5-OXA], [BH963; 2-Cl-4 -Br-5-OXA], [BH964; 2-Cl-4-I-5-OXA], [BH965; 2-Cl-4-Me-5-OXA], [BH966; 2-Cl-4-Et -5-OXA], [BH967; 2-Cl-4-Pr-5-OXA], [BH968; 2-Cl-4-i-Pr-5-OXA], [BH969; 2-Cl-4-CF _{3 -5-OXA], [BH970} ; 2-Cl-4-CHF 2 -5-OXA], [BH971; 2-Cl-4-OMe-5-OXA], [BH972; 2-Cl-4-OEt -5-OXA], [BH973; 2-Cl-4-OCF 3 -5-OXA], [BH974; 2-Cl-4-OCHF 2 -5-OXA], [BH975; 2-Cl-4-CN -5-OXA], [BH976; 2-Cl-4-SMe-5-OXA], [BH977; 2-Cl-4-SEt-5-OXA], [BH978; 2-Cl-4-c-Pr -5-OXA], [BH979; 2-Me-4-F-5-OXA], [BH 980; 2-Me-4-Cl-5-OXA], [BH981; 2-Me-4-Br-5 2-OXA], [BH982; 2-Me-4-I-5-OXA], [BH983; 2-Me-4-Me-5-OXA], [BH984; 2-Me-4-Et-5-OXA ], [BH985; 2-Me -4-Pr-5-OXA], [BH986; 2-Me-4-i-Pr-5-OXA], [BH987; 2-Me-4-CF 3 -5- OXA], [BH 988; 2-Me-4- _{CHF 2 -5-OXA], [} BH989; 2-Me-4-OMe-5-OXA], [BH990; 2-Me-4-OEt-5-OXA], [BH991; 2-Me-4-OCF _{3 -5-OXA], [BH992} ; 2-Me-4-OCHF 2 -5-OXA], [BH993; 2-Me-4-CN-5-OXA], [BH994; 2-Me-4-SMe -5-OXA], [BH995; 2-Me-4-SEt-5-OXA], [BH996; 2-Me-4-c-Pr-5-OXA], [BH997; 2-Et-4-F -5-OXA], [BH 998; 2-Et-4-Cl-5-OXA], [BH 999; 2-Et-4-Br-5-OXA], [BH 1000; 2-Et-4-I-5 -OXA],

[BH1001; 2-Et-4-Me-5-OXA], [BH1002; 2-Et-4-Et-5-OXA], [BH1003; 2-Et-4-Pr-5-OXA], [BH1004] ; 2-Et-4-i -Pr-5-OXA], [BH1005; 2-Et-4-CF 3 -5-OXA], [BH1006; 2-Et-4-CHF 2 -5-OXA], [BH1007; 2-Et-4 -OMe-5-OXA], [BH1008; 2-Et-4-OEt-5-OXA], [BH1009; 2-Et-4-OCF 3 -5-OXA], [ BH1010; 2-Et-4- OCHF 2 -5-OXA], [BH1011; 2-Et-4-CN-5-OXA], [BH1012; 2-Et-4-SMe-5-OXA], [BH1013 ; 2-Et-4-SEt -5-OXA], [BH1014; 2-Et-4-c-Pr-5-OXA], [BH1015; 2-CF 3 -4-F-5-OXA], [ _{BH1016; 2-CF 3 -4-} Cl-5-OXA], [BH1017; 2-CF 3 -4-Br-5-OXA], [BH1018; 2-CF 3 -4-I-5-OXA], _{[BH1019; 2-CF 3 -4} -Me-5-OXA], [BH1020; 2-CF 3 -4-Et-5-OXA], [BH1021; 2-CF 3 -4-Pr-5-OXA] _{, [BH1022; 2-CF 3} -4-i-Pr-5-OXA], [BH1023; 2-CF 3 -4-CF 3 -5-OXA], [BH1024; 2-CF 3 -4-CHF 2 -5-OXA], [BH1025; 2-CF 3 -4-OMe-5-OXA], [BH1026; 2-CF 3 -4-OEt-5-OXA], [BH1027; 2-CF 3 -4- _{OCF 3 -5-OXA], [} BH1028; 2-CF 3 -4-OCHF 2 -5-OXA], [BH1029; 2-CF 3 -4-CN-5-OXA], [BH1030; 2-CF 3 -4-SMe-5-OXA] , [BH1031; 2-CF 3 -4-SEt-5-OXA], [BH1032; 2-CF 3 -4-c-Pr-5-OXA], [BH1033; 2 -OMe-4-F-5-OXA], [BH1034; 2-OMe-4-Cl-5-OXA], [BH1035; 2-OMe-4-Br-5-OXA], [BH1036; 2-OMe -4-I-5-OXA ], [BH1037; 2-OMe-4-Me-5-OXA], [BH1038; 2-OMe-4-Et-5-OXA], [BH1039; 2-OMe-4-Pr-5-OXA], [BH1040; 2-OMe-4 -i-Pr-5-OXA], [BH1041; 2-OMe-4-CF 3 -5-OXA], [BH1042; 2-OMe-4-CHF 2 -5-OXA ], [BH1043; 2-OMe -4-OMe-5-OXA], [BH1044; 2-OMe-4-OEt-5-OXA], [BH1045; 2-OMe-4-OCF 3 -5-OXA] , [BH1046; 2-OMe- 4-OCHF 2 -5-OXA], [BH1047; 2-OMe-4-CN-5-OXA], [BH1048; 2-OMe-4-SMe-5-OXA], [BH1049; 2-OMe-4-SEt-5-OXA], [BH1050; 2-OMe-4-c-Pr-5-OXA], [BH1051; 2-OEt-4-F-5-OXA], [BH1052; 2-OEt-4-Cl-5-OXA], [BH1053; 2-OEt-4-Br-5-OXA], [BH1054; 2-OEt-4-I-5-OXA], [BH1055] 2-OEt-4-Me-5-OXA], [BH1056; 2-OEt-4-Et-5-OXA], [BH1057; 2-OEt-4-Pr-5-OXA], [BH1058; -OEt-4-i-Pr- 5-OXA], [BH1059; 2-OEt-4-CF 3 -5-OXA], [BH1060; 2-OEt-4-CHF 2 -5-OXA], [BH1061 ; 2-OEt-4-OMe -5-OXA], [BH1062; 2-OEt-4-OEt-5-OXA], [BH1063; 2-OEt-4-OCF 3 -5-OXA], [BH1064; _{2-OEt-4-OCHF 2} -5-OXA], [BH1065; 2-OEt-4-CN-5-OXA], [BH1066; 2-OEt-4-SMe-5-OXA], [BH1067; 2 -OEt-4-SEt-5-OXA], [BH1068; 2-OEt-4-c-Pr-5-OXA], [BH1069; 2-SMe-4-F-5-OXA], [BH1070; -SMe-4-Cl-5-OXA], [BH1071; 2-SMe-4-Br-5-OXA], [BH1072; 2-SMe-4-I-5-OXA], [BH1073; 2-SMe -4-Me -5-OXA], [BH1074; 2-SMe-4-Et-5-OXA], [BH1075; 2-SMe-4-Pr-5-OXA], [BH1076; 2-SMe-4-i-Pr -5-OXA], [BH1077; 2-SMe-4-CF 3 -5-OXA], [BH1078; 2-SMe-4-CHF 2 -5-OXA], [BH1079; 2-SMe-4-OMe -5-OXA], [BH1080; 2-SMe-4-OEt-5-OXA], [BH1081; 2-SMe-4-OCF 3 -5-OXA], [BH1082; 2-SMe-4-OCHF 2 -5-OXA], [BH1083; 2-SMe-4-CN-5-OXA], [BH1084; 2-SMe-4-SMe-5-OXA], [BH1085; 2-SMe-4-SEt-5 -OXA], [BH1086; 2-SMe-4-c-Pr-5-OXA], [BH1087; -2-FURR], [BH1088; 4-F-2-FURR], [BH1089; 4-Cl- 2-FURR], [BH1090; 4-Br-2-FURR], [BH1091; 4-I-2-FURR], [BH1092; 4-Me-2-FURR], [BH1093; 4-Et-2- FURR], [BH1094; 4- Pr-2-FURR], [BH1095; 4-i-Pr-2-FURR], [BH1096; 4-CF 3 -2-FURR], [BH1097; 4-CHF 2 - 2-FURR], [BH1098; 4-OMe-2-FURR], [BH1099; 4-OEt-2-FURR], [BH1100; 4-OCF 3 -2-FURR],

_{[BH1101; 4-OCHF 2 -2} -FURR], [BH1102; 4-CN-2-FUR], [BH1103; 4-SMe-2-FUR], [BH1104; 4-SEt-2-FUR], [ BH1105; 4-c-Pr-2-FUR], [BH1106; 5-F-2-FUR], [BH1107; 5-Cl-2-FUR], [BH1108; 5-Br-2-FUR], [BH 1108; BH1109; 5-I-2-FUR], [BH1 110; 5-Me-2-FUR], [BH 1111; 5-Et-2-FUR], [BH 1112; 5-Pr-2-FUR], [BH 11 13; 5-i-Pr-2- FUR], [BH1114; 5-CF 3 -2-FUR], [BH1115; 5-CHF 2 -2-FUR], [BH1116; 5-OMe-2-FUR], [ BH1 117; 5-OEt-2-FUR !, [BH 1118; 5-OCF ₃ 2-FUR], [BH 1119; 5-OCHF ₂ 2-FUR], [BH 1 120; 5-CN-2-FUR], BH1121; 5-SMe-2-FUR !, [BH1122; 5-SEt-2-FUR], [BH1123; 5-c-Pr-2-FUR], [BH1124; 4-F-5-F-2-] FUR], [BH1125; 4-F-5-Cl-2-FUR], [BH1126; 4-F-5-Br-2-FUR], [BH1127; 4-F-5-I-2-FUR] , [BH1128; 4-F-5-Me-2-FUR], [BH1129; 4-F-5-Et-2-FUR], [BH1130; 4-F-5-Pr-2-FUR], [BH1 130; BH1131; 4-F-5- i-Pr-2-FUR], [BH1132; 4-F-5-CF 3 -2-FUR], [BH1133; 4-F-5-CHF 2 -2-FUR] , [BH1134; 4-F- 5-OMe-2-FUR], [BH1135; 4-F-5-OEt-2-FUR], [BH1136; 4-F-5-OCF 3 -2-FUR], [BH1137; 4-F-5 -OCHF 2 -2-FUR], [BH1138; 4-F-5-CN-2-FUR], [BH1139; 4-F-5-SMe-2-FUR], [ BH1140; 4-F-5-SEt-2-FUR], [BH1141; 4-F-5-c-Pr-2-FUR], [BH1142; 4-Cl-5-F-2-FUR], [BH 1142; BH1143; 4-Cl-5-Cl-2-FUR], [BH11 44; 4-Cl-5-Br-2-FUR !, [BH1145; 4-Cl-5-I-2-FUR], [BH1146; 4-Cl-5-Me-2-FUR], [BH1147; 4-Cl-5-Et-2-FUR], [BH1148; 4-Cl-5-Pr-2-FUR], [BH1149; 4-Cl-5-i-Pr-2-FUR], [BH1150; _{4-Cl-5-CF 3} -2-FUR], [BH1151; 4-Cl-5-CHF 2 -2-FUR], [BH1152; 4-Cl-5-OMe-2-FUR], [BH1153; 4-Cl-5-OEt- 2-FUR], [BH1154; 4-Cl-5-OCF 3 -2-FUR], [BH1155; 4-Cl-5-OCHF 2 -2-FUR], [BH1156; 4-Cl-5-CN-2-FUR !, [BH1157; 4-Cl-5-SMe-2-FUR], [BH1158; 4-Cl-5-SEt-2-FUR], [BH1159; Cl-5-c-Pr-2-FUR], [BH1160; 4-Me-5-F-2-FUR], [BH1161; 4-Me-5-Cl-2-FUR], [BH1162; 4- Me-5-Br-2-FUR !, [BH1163; 4-Me-5-I-2-FUR], [BH1164; 4-Me-5-Me-2-FUR], [BH1165; 4-Me- 5-Et-2-FUR], [BH1166; 4-Me-5-Pr-2-FUR], [BH1167; 4-Me-5-i-Pr-2-FUR], [BH1168; 4-Me- _{5-CF 3 -2-FUR]} , [BH1169; 4-Me-5-CHF 2 -2-FUR], [BH1170; 4-Me-5-OMe-2-FUR], [BH1171; 4-Me- 5-OEt-2-FUR] , [BH1172; 4-Me-5-OCF 3 -2-FUR], [BH1173; 4-Me-5-OCHF 2 -2-FUR], [BH1174; 4-Me- 5-CN-2-FUR !, [BH1175; 4-Me-5-SMe-2-FUR], [BH1176; 4-Me-5-SEt-2-FUR], [BH1177; 4-Me-5-] c-Pr-2-FUR], [BH1178; 4-Et-5-F-2-FUR], [BH1179; 4-Et-5-Cl-2-FUR], [BH 1180; 4-Et-5- Br-2-FUR], [BH1181; 4-Et-5-I-2-FUR], [BH1182; 4-Et -5-Me-2-FUR !, [BH1183; 4-Et-5-Et-2-FUR], [BH 1184; 4-Et-5-Pr-2-FUR], [BH 1185; 4-Et-5 -i-Pr-2-FUR] , [BH1186; 4-Et-5-CF 3 -2-FUR], [BH1187; 4-Et-5-CHF 2 -2-FUR], [BH1188; 4-Et -5-OMe-2-FUR !, [BH1189; 4-Et-5-OEt-2-FUR], [BH 1190; 4-Et-5-OCF ₃ -2-FUR], [BH1191; 4-Et- 5-OCHF ₂ -2-FUR !, [BH1192; 4-Et-5-CN-2-FUR], [BH1193; 4-Et-5-SMe-2-FUR], [BH 1194; 4-Et-5 -SEt-2-FUR], [BH 1195; 4-Et-5-c-Pr-2-FUR], [BH 1196; 4-CF ₃ -5-F-2-FUR], [BH 1197; 4-CF ₃ -5-Cl-2-FUR !, [BH 1198; 4-CF ₃ -5-Br-2-FUR], [BH 1 199; 4-CF ₃ -5-I-2-FUR], [BH 1200; 4-CF ₃ -5-Me-2-FUR],

_{[BH1201; 4-CF 3 -5} -Et-2-FUR], [BH1202; 4-CF 3 -5-Pr-2-FUR], [BH1203; 4-CF 3 -5-i-Pr-2- FUR], [BH1204; 4- CF 3 -5-CF 3 -2-FUR], [BH1205; 4-CF 3 -5-CHF 2 -2-FUR], [BH1206; 4-CF 3 -5-OMe -2-FUR], [BH1207; 4-CF 3 -5-OEt-2-FUR], [BH1208; 4-CF 3 -5-OCF 3 -2-FUR], [BH1209; 4-CF 3 -5 _{-OCHF 2 -2-FUR], [} BH1210; 4-CF 3 -5-CN-2-FUR], [BH1211; 4-CF 3 -5-SMe-2-FUR], [BH1212; 4-CF 3 -4-SEt-2-FUR !, [BH 1213; 4-CF ₃ -5-c-Pr-2-FUR], [BH 1214; 4-OMe-5-F-2-FUR], [BH 1215; OMe-5-Cl-2-FUR], [BH1216; 4-OMe-5-Br-2-FUR], [BH1217; 4-OMe-5-I-2-FUR], [BH1218; 4-OMe- 5-Me-2-FUR !, [BH 1219; 4-OMe-5-Et-2-FUR], [BH 1220; 4-OMe-5-Pr-2-FUR], [BH 1221; 4-OMe-5- i-Pr-2-FUR] , [BH1222; 4-OMe-5-CF 3 -2-FUR], [BH1223; 4-OMe-5-CHF 2 -2-FUR], [BH1224; 4-OMe- 5-OMe-2-FUR] , [BH1225; 4-OMe-5-OEt-2-FUR], [BH1226; 4-OMe-5-OCF 3 -2-FUR], [BH1227; 4-OMe-5 _{-OCHF 2 -2-FUR], [} BH1228; 4-OMe-5-CN-2-FUR], [BH1229; 4-OMe-5-SMe-2-FUR], [BH1230; 4-OMe-5- SEt-2-FUR !, [BH1231; 4-OMe-5-c-Pr-2-FUR], [BH1232; 4-OEt-5-F-2-FUR], [BH1233; 4-OEt-5-] Cl-2-FUR !, [BH1234; 4-OEt-5-Br-2-FUR], [BH1235; 4-OEt-5-I-2-FUR], [BH1236; 4-OEt-5-Me- 2 -FUR], [BH1237; 4-OEt-5-Et-2-FUR], [BH1238; 4-OEt-5-Pr-2-FUR], [BH1239; 4-OEt-5-i-Pr-2 -FUR], [BH1240; 4- OEt-5-CF 3 -2-FUR], [BH1241; 4-OEt-5-CHF 2 -2-FUR], [BH1242; 4-OEt-5-OMe-2 -FUR], [BH1243; 4- OEt-5-OEt-2-FUR], [BH1244; 4-OEt-5-OCF 3 -2-FUR], [BH1245; 4-OEt-5-OCHF 2 -2 -FUR], [BH1246; 4-OEt-5-CN-2-FUR], [BH1247; 4-OEt-5-SMe-2-FUR], [BH1248; 4-OEt-5-SEt-2-FUR] ], [BH1249; 4-OEt-5-c-Pr-2-FUR], [BH1250; 4-SMe-5-F-2-FUR], [BH1251; 4-SMe-5-Cl-2-FUR] ], [BH1252; 4-SMe-5-Br-2-FUR], [BH1253; 4-SMe-5-I-2-FUR], [BH1254; 4-SMe-5-Me-2-FUR], [BH1255; 4-SMe-5-Et-2-FUR], [BH1256; 4-SMe-5-Pr-2-FUR], [BH1257; 4-SMe-5-i-Pr-2-FUR], [BH1258; 4-SMe-5 -CF 3 -2-FUR], [BH1259; 4-SMe-5-CHF 2 -2-FUR], [BH1260; 4-SMe-5-OMe-2-FUR], [BH1261; 4-SMe-5 -OEt-2-FUR], [BH1262; 4-SMe-5-OCF 3 -2-FUR], [BH1263; 4-SMe-5-OCHF 2 -2-FUR], [BH1264; 4-SMe-5-CN-2-FUR], [BH1265; 4-SMe-5-SMe-2-FUR], [BH1266; 4-SMe-5-SEt-2-FUR], [BH1267] 4-SMe-5-c-Pr-2-FUR !, [BH1268; 3-F-2-FUR], [BH1269; 3-Cl-2-FUR], [BH1270; 3-Br-2-FUR] ], [BH1271; 3-I-2-FUR], [BH1272; 3-Me-2-FUR], [BH1273; 3-Et-2-FUR], [BH1274; 3-Pr-2-FUR], [BH1 275; 3-i-Pr- 2-FUR], [BH1276; 3-CF 3 -2-FUR], [BH1277; 3-CHF 2 -2-FUR], [BH1278; 3-OMe-2-FUR] [BH1279; 3-OEt-2-FUR], [BH 1280; 3-OCF ₃ 2-FUR], [BH1281; 3-OCHF ₂ 2-FUR], [BH 1282; 3-F-4-F- 2-FUR], [BH1283; 3-F-4-Cl-2-FUR], [BH1284; 3-F-4-Br-2-FUR], [BH1285; 3-F-4-I-2-] FUR], [BH1286; 3-F-4-Me-2-FUR], [BH1 287; 3-F-4-Et-2-FUR], [BH1288; 3-F-4-Pr-2-FUR] , [BH1289; 3-F- 4-i-Pr-2-FUR], [BH1290; 3-F-4-CF 3 -2-FUR], [BH1291; 3-F-4-CHF 2 -2- FUR], [BH1292; 3-F-4-OMe-2-FUR], [BH1293; 3-F-4-OEt-2-FUR], [BH1294; 3-F-4-OCF ₃ -2-FUR ], [BH1295; 3-F -4-OCHF 2 -2-FUR], [BH1296; 3-F-4-CN-2-FUR], [BH1297; 3-F-4-SMe-2-FUR] , [BH1298; 3-F-4-SEt-2-FUR], [BH1299; 3-F-4-c-Pr-2-FUR], [BH1300; 3-Cl-4-F-2-FUR] ,

[BH1301; 3-Cl-4-Cl-2-FUR], [BH1302; 3-Cl-4-Br-2-FUR], [BH1303; 3-Cl-4-I-2-FUR], [BH1304] 3-Cl-4-Me-2-FUR !, [BH1305; 3-Cl-4-Et-2-FUR], [BH1306; 3-Cl-4-Pr-2-FUR], [BH1307; 3 -Cl-4-i-Pr- 2-FUR], [BH1308; 3-Cl-4-CF 3 -2-FUR], [BH1309; 3-Cl-4-CHF 2 -2-FUR], [BH1310 ; 3-Cl-4-OMe -2-FUR], [BH1311; 3-Cl-4-OEt-2-FUR], [BH1312; 3-Cl-4-OCF 3 -2-FUR], [BH1313; _{3-Cl-4-OCHF 2} -2-FUR], [BH1314; 3-Cl-4-CN-2-FUR], [BH1315; 3-Cl-4-SMe-2-FUR], [BH1316; 3 -Cl-4-SEt-2-FUR !, [BH1317; 3-Cl-4-c-Pr-2-FUR], [BH1318; 3-Me-4-F-2-FUR], [BH1319; 3 -Me-4-Cl-2-FUR !, [BH1320; 3-Me-4-Br-2-FUR], [BH1321; 3-Me-4-I-2-FUR], [BH1322; 3-Me -4-Me-2-FUR !, [BH1323; 3-Me-4-Et-2-FUR], [BH 1324; 3-Me-4-Pr-2-FUR], [BH 1325; 3-Me-4 -i-Pr-2-FUR] , [BH1326; 3-Me-4-CF 3 -2-FUR], [BH1327; 3-Me-4-CHF 2 -2-FUR], [BH1328; 3-Me -4-OMe-2-FUR !, [BH 1329; 3-Me-4-OEt-2-FUR], [BH 1330; 3-Me-4-OCF ₃ 2-FUR], [BH 1331; 3-Me- _{4-OCHF 2 -2-FUR]} , [BH1332; 3-Me-4-CN-2-FUR], [BH1333; 3-Me-4-SMe-2-FUR], [BH1334; 3-Me-4 -SEt-2-FUR !, [BH1335; 3-Me-4-c-Pr-2-FUR], [BH1336; 3-Et-4-F-2-FUR], [BH1337; 3-Et-4 -Cl-2-FUR], [BH1338; 3-Et-4-Br-2-FUR], [BH133] 9; 3-Et-4-I-2-FUR !, [BH1340; 3-Et-4-Me-2-FUR], [BH1341; 3-Et-4-Et-2-FUR], [BH1342; 3-Et-4-Pr- 2-FUR], [BH1343; 3-Et-4-i-Pr-2-FUR], [BH1344; 3-Et-4-CF 3 -2-FUR], [BH1345 ; 3-Et-4-CHF 2 -2-FUR], [BH1346; 3-Et-4-OMe-2-FUR], [BH1347; 3-Et-4-OEt-2-FUR], [BH1348; _{3-Et-4-OCF 3} -2-FUR], [BH1349; 3-Et-4-OCHF 2 -2-FUR], [BH1350; 3-Et-4-CN-2-FUR], [BH1351; 3-Et-4-SMe-2-FUR !, [BH1352; 3-Et-4-SEt-2-FUR], [BH1353; 3-Et-4-c-Pr-2-FUR], [BH1354; _{3-CF 3 -4-F-} 2-FUR], [BH1355; 3-CF 3 -4-Cl-2-FUR], [BH1356; 3-CF 3 -4-Br-2-FUR], [BH1357 _{; 3-CF 3 -4-I} -2-FUR], [BH1358; 3-CF 3 -4-Me-2-FUR], [BH1359; 3-CF 3 -4-Et-2-FUR], [ _{BH1360; 3-CF 3 -4-} Pr-2-FUR], [BH1361; 3-CF 3 -4-i-Pr-2-FUR], [BH1362; 3-CF 3 -4-CF 3 -2- FUR], [BH1363; 3- CF 3 -4-CHF 2 -2-FUR], [BH1364; 3-CF 3 -4-OMe-2-FUR], [BH1365; 3-CF 3 -4-OEt- 2-FUR], [BH1366; 3-CF 3 -4-OCF 3 -2-FUR], [BH1367; 3-CF 3 -4-OCHF 2 -2-FUR], [BH1368; 3-CF 3 -4 -CN-2-FUR], [ BH1369; 3-CF 3 -4-SMe-2-FUR], [BH1370; 3-CF 3 -4-SEt-2-FUR], [BH1371; 3-CF 3 - 4-c-Pr-2-FUR !, [BH1372; 3-OMe-4-F-2-FUR], [BH1373; 3-OMe-4-Cl-2-FUR], [BH1374; 3-OMe- 4-Br-2-FUR], [BH13 75; 3-OMe-4-I-2-FUR !, [BH1376; 3-OMe-4-Me-2-FUR], [BH1377; 3-OMe-4-Et-2-FUR], [BH1378; 3-OMe-4-Pr-2-FUR !, [BH 1379; 3-OMe-4-i-Pr-2-FUR], [BH 1380; 3-OMe-4-CF ₃ -2-FUR], [BH 1381] ; 3-OMe-4-CHF 2 -2-FUR], [BH1382; 3-OMe-4-OMe-2-FUR], [BH1383; 3-OMe-4-OEt-2-FUR], [BH1384; _{3-OMe-4-OCF 3} -2-FUR], [BH1385; 3-OMe-4-OCHF 2 -2-FUR], [BH1386; 3-OMe-4-CN-2-FUR], [BH1387; 3-OMe-4-SMe-2-FUR !, [BH1388; 3-OMe-4-SEt-2-FUR], [BH1389; 3-OMe-4-c-Pr-2-FUR], [BH1390; 3-OEt-4-F-2-FUR !, [BH1391; 3-OEt-4-Cl-2-FUR], [BH1392; 3-OEt-4-Br-2-FUR], [BH1393; OEt-4-I-2-FUR !, [BH1394; 3-OEt-4-Me-2-FUR], [BH 1395; 3-OEt-4-Et-2-FUR], [BH 1396; 3-OEt- 4-Pr-2-FUR !, [BH 1397; 3-OEt-4-i-Pr-2-FUR], [BH 1398; 3-OEt-4-CF ₃ 2-FUR], [BH 1 399; 3-OEt -4-CHF ₂ -2-FUR], [BH1400; 3-OEt-4-OMe-2-FUR],

[BH1401; 3-OEt-4 -OEt-2-FUR], [BH1402; 3-OEt-4-OCF 3 -2-FUR], [BH1403; 3-OEt-4-OCHF 2 -2-FUR], [BH1404; 3-OEt-4-CN-2-FUR], [BH1405; 3-OEt-4-SMe-2-FUR], [BH1406; 3-OEt-4-SEt-2-FUR], [BH1407] 3-OEt-4-c-Pr-2-FUR !, [BH1408; 3-SMe-4-F-2-FUR], [BH1409; 3-SMe-4-Cl-2-FUR], [BH1410] 3-SMe-4-Br-2-FUR !, [BH 1411; 3-SMe-4-I-2-FUR], [BH1412; 3-SMe-4-Me-2-FUR], [BH 1413; -SMe-4-Et-2-FUR !, [BH 1414; 3-SMe-4-Pr-2-FUR], [BH 1415; 3-SMe-4-i-Pr-2-FUR], [BH 1416; _{-SMe-4-CF 3 -2-} FUR], [BH1417; 3-SMe-4-CHF 2 -2-FUR], [BH1418; 3-SMe-4-OMe-2-FUR], [BH1419; 3 -SMe-4-OEt-2- FUR], [BH1420; 3-SMe-4-OCF 3 -2-FUR], [BH1421; 3-SMe-4-OCHF 2 -2-FUR], [BH1422; 3 -SMe-4-CN-2-FUR !, [BH1423; 3-SMe-4-SMe-2-FUR], [BH1424; 3-SMe-4-SEt-2-FUR], [BH1425; 3-SMe -4-c-Pr-2-FUR !, [BH1426; 3-F-5-F-2-FUR], [BH1427; 3-F-5-Cl-2-FUR], [BH1428; 3-F -5-Br-2-FUR !, [BH 1429; 3-F-5-I-2-FUR], [BH 1430; 3-F-5-Me-2-FUR], [BH 1431; 3-F-5 -Et-2-FUR], [BH1432; 3-F-5-Pr-2-FUR], [BH1433; 3-F-5-i-Pr-2-FUR], [BH1434; 3-F-5 _{-CF 3 -2-FUR], [} BH1435; 3-F-5-CHF 2 -2-FUR], [BH1436; 3-F-5-OMe-2-FUR], [BH1437; 3-F-5 -OEt-2-FUR], [BH1438; 3-F-5-OCF _{3 -2-FUR], [BH1439} ; 3-F-5-OCHF 2 -2-FUR], [BH1440; 3-F-5-CN-2-FUR], [BH1441; 3-F-5-SMe -2-FUR !, [BH1442; 3-F-5-SEt-2-FUR], [BH 1443; 3-F-5-c-Pr-2-FUR], [BH 1444; 3-Cl-5-F -2-FUR !, [BH 1445; 3-Cl-5-Cl-2-FUR], [BH 1446; 3-Cl-5-Br-2-FUR], [BH 1447; 3-Cl-5-I-2 -FUR], [BH 1448; 3-Cl-5-Me-2-FUR], [BH 1449; 3-Cl-5-Et-2-FUR], [BH 1450; 3-Cl-5-Pr-2-FUR ], [BH1451; 3-Cl -5-i-Pr-2-FUR], [BH1452; 3-Cl-5-CF 3 -2-FUR], [BH1453; 3-Cl-5-CHF 2 -2 -FUR], [BH1454; 3- Cl-5-OMe-2-FUR], [BH1455; 3-Cl-5-OEt-2-FUR], [BH1456; 3-Cl-5-OCF 3 -2- FUR], [BH1457; 3- Cl-5-OCHF 2 -2-FUR], [BH1458; 3-Cl-5-CN-2-FUR], [BH1459; 3-Cl-5-SMe-2-FUR ], [BH1460; 3-Cl-5-SEt-2-FUR], [BH1461; 3-Cl-5-c-Pr-2-FUR], [BH1462; 3-Me-5-F-2-FUR] ], [BH1463; 3-Me-5-Cl-2-FUR], [BH1464; 3-Me-5-Br-2-FUR], [BH1465; 3-Me-5-I-2-FUR], [BH1466; 3-Me-5-Me-2-FUR], [BH1467; 3-Me-5-Et-2-FUR], [BH1468; 3-Me-5-Pr-2-FUR], [BH1469] ; 3-Me-5-i -Pr-2-FUR], [BH1470; 3-Me-5-CF 3 -2-FUR], [BH1471; 3-Me-5-CHF 2 -2-FUR], [BH1472; 3-Me-5 -OMe-2-FUR], [BH1473; 3-Me-5-OEt-2-FUR], [BH1474; 3-Me-5-OCF 3 -2-FUR], [ BH1475; 3-Me-5-OCHF ₂ -2-FUR], [BH 1476; 3-Me-5-CN-2- FUR], [BH 1477; 3-Me-5-SMe-2-FUR], [BH 1478; 3-Me-5-SEt-2-FUR], [BH 1479; 3-Me-5-c-Pr-2- FUR], [BH1480; 3-Et-5-F-2-FUR], [BH1481; 3-Et-5-Cl-2-FUR], [BH1482; 3-Et-5-Br-2-FUR] , [BH1483; 3-Et-5-I-2-FUR], [BH1484; 3-Et-5-Me-2-FUR], [BH1485; 3-Et-5-Et-2-FUR], [BH BH1486; 3-Et-5-Pr-2-FUR], [BH 1487; 3-Et-5-i-Pr-2-FUR], [BH 1 488; 3-Et-5-CF ₃ -2-FUR], [BH1489; 3-Et-5 -CHF 2 -2-FUR], [BH1490; 3-Et-5-OMe-2-FUR], [BH1491; 3-Et-5-OEt-2-FUR], [ BH1492; 3-Et-5- OCF 3 -2-FUR], [BH1493; 3-Et-5-OCHF 2 -2-FUR], [BH1494; 3-Et-5-CN-2-FUR], [ BH1495; 3-Et-5-SMe-2-FUR], [BH1496; 3-Et-5-SEt-2-FUR], [BH 1497; 3-Et-5-c-Pr-2-FUR], [BH 1495; _{BH1498; 3-CF 3 -5-} F-2-FUR], [BH1499; 3-CF 3 -5-Cl-2-FUR], [BH1500; 3-CF 3 -5-Br-2-FUR],

_{[BH1501; 3-CF 3 -5} -I-2-FUR], [BH1502; 3-CF 3 -5-Me-2-FUR], [BH1503; 3-CF 3 -5-Et-2-FUR] _{, [BH1504; 3-CF 3} -5-Pr-2-FUR], [BH1505; 3-CF 3 -5-i-Pr-2-FUR], [BH1506; 3-CF 3 -5-CF 3 - 2-FUR], [BH1507; 3-CF 3 -5-CHF 2 -2-FUR], [BH1508; 3-CF 3 -5-OMe-2-FUR], [BH1509; 3-CF 3 -5- OEt-2-FUR], [ BH1510; 3-CF 3 -5-OCF 3 -2-FUR], [BH1511; 3-CF 3 -5-OCHF 2 -2-FUR], [BH1512; 3-CF 3 -5-CN-2-FUR !, [BH 1513; 3-CF ₃ -5-SMe-2-FUR], [BH 1514; 3-CF ₃ -5-SEt-2-FUR], [BH 1515; 3-CF _{3 -5-c-Pr-2} -FUR], [BH1516; 3-OMe-5-F-2-FUR], [BH1517; 3-OMe-5-Cl-2-FUR], [BH1518; 3- OMe-5-Br-2-FUR !, [BH 1519; 3-OMe-5-I-2-FUR], [BH 1520; 3-OMe-5-Me-2-FUR], [BH1521; 3-OMe- 5-Et-2-FUR !, [BH1522; 3-OMe-5-Pr-2-FUR], [BH1523; 3-OMe-5-i-Pr-2-FUR], [BH1524; 3-OMe- _{5-CF 3 -2-FUR]} , [BH1525; 3-OMe-5-CHF 2 -2-FUR], [BH1526; 3-OMe-5-OMe-2-FUR], [BH1527; 3-OMe- 5-OEt-2-FUR] , [BH1528; 3-OMe-5-OCF 3 -2-FUR], [BH1529; 3-OMe-5-OCHF 2 -2-FUR], [BH1530; 3-OMe- 5-CN-2-FUR !, [BH1531; 3-OMe-5-SMe-2-FUR], [BH1532; 3-OMe-5-SEt-2-FUR], [BH1533; 3-OMe-5-] c-Pr-2-FUR], [BH1534; 3-OEt-5-F-2-FUR], [BH1535; 3-OEt-5-Cl-2-FUR], [BH1536; 3-OEt-5- Br-2-FUR !, [BH1537; 3-OEt-5-I-2-FUR], [BH1538; 3-OEt-5-Me-2-FUR], [BH1539; 3-OEt-5-Et- 2-FUR], [BH1540; 3-OEt-5-Pr-2-FUR], [BH1541; 3-OEt-5-i-Pr-2-FUR], [BH1542; 3-OEt-5-CF 3 -2-FUR !, [BH 1543; 3-OEt-5-CHF ₂ -2-FUR], [BH 1544; 3-OEt-5-OMe-2-FUR], [BH 1545; 3-OEt-5-OEt- 2-FUR], [BH1546; 3-OEt-5-OCF 3 -2-FUR], [BH1547; 3-OEt-5-OCHF 2 -2-FUR], [BH1548; 3-OEt-5-CN- 2-FUR], [BH1549; 3-OEt-5-SMe-2-FUR], [BH1550; 3-OEt-5-SEt-2-FUR], [BH1551; 3-OEt-5-c-Pr- 2-FUR], [BH1552; 3-SMe-5-F-2-FUR], [BH1553; 3-SMe-5-Cl-2-FUR], [BH1554; 3-SMe-5-Br-2- FUR], [BH1555; 3-SMe-5-I-2-FUR], [BH1556; 3-SMe-5-Me-2-FUR], [BH1557; 3-SMe-5-Et-2-FUR] [BH1558; 3-SMe-5-Pr-2-FUR], [BH1559; 3-SMe-5-i-Pr-2-FUR], [BH1560; 3-SMe-5-CF ₃ -2-FUR ], [BH1561; 3-SMe -5-CHF 2 -2-FUR], [BH1562; 3-SMe-5-OMe-2-FUR], [BH1563; 3-SMe-5-OEt-2-FUR] , [BH1564; 3-SMe- 5-OCF 3 -2-FUR], [BH1565; 3-SMe-5-OCHF 2 -2-FUR], [BH1566; 3-SMe-5-CN-2-FUR] , [BH1567; 3-SMe-5-SMe-2-FUR], [BH1568; 3-SMe-5-SEt-2-FUR], [BH1569; 3-SMe-5-c-Pr-2-FUR] , [BH1570; 3-Me-4-Me-5-F-2-FUR], [BH1571; 3-Me-4-Me-5-Cl-2-FUR], [BH1572; 3-Me-4- Me-5-Br-2-FUR ], [BH1573; 3-Me-4-Me-5-I-2-FUR], [BH1574; 3-Me-4-Me-5-Me-2-FUR], [BH1575; 3-Me-4 -Me-5-Et-2-FUR], [BH1576; 3-Me-4-Me-5-Pr-2-FUR], [BH1577; 3-Me-4-Me-5-i-Pr-2 -FUR], [BH1578; 3- Me-4-Me-5-CF 3 -2-FUR], [BH1579; 3-Me-4-Me-5-CHF 2 -2-FUR], [BH1580; 3 -Me-4-Me-5-OMe-2-FUR !, [BH1581; 3-Me-4-Me-5-OEt-2-FUR], [BH1582; 3-Me-4-Me-5-OCF _{3 -2-FUR], [BH1583} ; 3-Me-4-Me-5-OCHF 2 -2-FUR], [BH1584; 3-Me-4-Me-5-CN-2-FUR], [BH1585 3-Me-4-Me-5-SMe-2-FUR !, [BH1586; 3-Me-4-Me-5-SEt-2-FUR], [BH1587; 3-Me-4-Me-5 -c-Pr-2-FUR], [BH1588; 3-Me-4-F-5-Me-2-FUR], [BH1589; 3-Me-4-Cl-5-Me-2-FUR], [BH1590; 3-Me-4-Br-5-Me-2-FUR], [BH1591; 3-Me-4-I-5-Me-2-FUR], [BH1592; 3-Me-4-Et -5-Me-2-FUR !, [BH1593; 3-Me-4-Pr-5-Me-2-FUR], [BH1594; 3-Me-4-i-Pr-5-Me-2-FUR ], [BH1595; 3-Me -4-CF 3 -5-Me-2-FUR], [BH1596; 3-Me-4-CHF 2 -5-Me-2-FUR], [BH1597; 3-Me -4-OMe-5-Me-2-FUR !, [BH 1598; 3-Me-4-OEt-5-Me-2-FUR], [BH1599; 3-Me-4-OCF ₃ -5-Me- 2-FUR], [BH1600; 3-Me-4-OCHF 2 -5-Me-2-FUR],

[BH1601; 3-Me-4-CN-5-Me-2-FUR], [BH1602; 3-Me-4-SMe-5-Me-2-FUR], [BH1603; 3-Me-4-SEt -5-Me-2-FUR !, [BH1604; 3-Me-4-c-Pr-5-Me-2-FUR], [BH1605; -2-THI], [BH1606; 4-F-2-] THI], [BH1607; 4-Cl-2-THI], [BH1608; 4-Br-2-THI], [BH1609; 4-I-2-THI], [BH1610; 4-Me-2-THI] , [BH 1611; 4-Et-2-THI], [BH 1612; 4-Pr-2-THI], [BH 1613; 4-i-Pr-2-THI], [BH 1614; 4-CF ₃ -2-THI ], [BH1615; 4-CHF 2 -2-THI], [BH1616; 4-OMe-2-THI], [BH1617; 4-OEt-2-THI], [BH1618; 4-OCF 3 -2-THI ], [BH1619; 4-OCHF 2 -2-THI], [BH1620; 4-CN-2-THI], [BH1621; 4-SMe-2-THI], [BH1622; 4-SEt-2-THI] , [BH1623; 4-c-Pr-2-THI], [BH1624; 5-F-2-THI], [BH1625; 5-Cl-2-THI], [BH1626; 5-Br-2-THI] , [BH1627; 5-I-2-THI], [BH1628; 5-Me-2-THI], [BH1629; 5-Et-2-THI], [BH1630; 5-Pr-2-THI], [BH BH1631; 5-i-Pr- 2-THI], [BH1632; 5-CF 3 -2-THI], [BH1633; 5-CHF 2 -2-THI], [BH1634; 5-OMe-2-THI] , [BH1635; 5-OEt- 2-THI], [BH1636; 5-OCF 3 -2-THI], [BH1637; 5-OCHF 2 -2-THI], [BH1638; 5-CN-2-THI] , [BH1639; 5-SMe-2-THI], [BH1640; 5-SEt-2-THI], [BH1641; 5-c-Pr-2-THI], [BH1642; 4-F-5-F- 2-THI], [BH1643; 4-F-5-Cl-2-THI], [BH1644; 4-F-5-Br-2-THI], [BH1645; 4-F-5-I-2-] THI], [B H1646; 4-F-5-Me-2-THI], [BH1647; 4-F-5-Et-2-THI], [BH1648; 4-F-5-Pr-2-THI], [BH1649; 4-F-5-i- Pr-2-THI], [BH1650; 4-F-5-CF 3 -2-THI], [BH1651; 4-F-5-CHF 2 -2-THI], [ BH1652; 4-F-5- OMe-2-THI], [BH1653; 4-F-5-OEt-2-THI], [BH1654; 4-F-5-OCF 3 -2-THI], [BH1655 4-F-5-OCHF ₂ -2-THI !, [BH1656; 4-F-5-CN-2-THI], [BH1657; 4-F-5-SMe-2-THI], [BH1658; 4-F-5-SEt-2-THI, [BH1659; 4-F-5-c-Pr-2-THI], [BH1660; 4-Cl-5-F-2-THI], [BH1661; 4-Cl-5-Cl-2-THI], [BH1662; 4-Cl-5-Br-2-THI], [BH1663; 4-Cl-5-I-2-THI], [BH1664; Cl-5-Me-2-THI], [BH1665; 4-Cl-5-Et-2-THI], [BH1666; 4-Cl-5-Pr-2-THI], [BH1667; 4-Cl- 5-i-Pr-2- THI], [BH1668; 4-Cl-5-CF 3 -2-THI], [BH1669; 4-Cl-5-CHF 2 -2-THI], [BH1670; 4- Cl-5-OMe-2- THI], [BH1671; 4-Cl-5-OEt-2-THI], [BH1672; 4-Cl-5-OCF 3 -2-THI], [BH1673; 4-Cl -5-OCHF ₂ -2-THI], [BH 1 674; 4-Cl-5-CN-2-THI], [BH 1 675; 4-Cl-5-SMe-2-THI], [BH 1 676; 5-SEt-2-THI, [BH1677; 4-Cl-5-c-Pr-2-THI], [BH1678; 4-Me-5-F-2-THI], [BH1679; 4-Me- 5-Cl-2-THI, [BH1680; 4-Me-5-Br-2-THI], [BH1681; 4-Me-5-I-2-THI], [BH1682; 4-Me-5- Me-2-THI, [BH1683; 4-Me-5-Et-2-THI], [BH1684; 4-Me-5-Pr-2-TH I], [BH1685; 4- Me-5-i-Pr-2-THI], [BH1686; 4-Me-5-CF 3 -2-THI], [BH1687; 4-Me-5-CHF 2 - 2-THI], [BH1688; 4-Me-5-OMe-2-THI], [BH1689; 4-Me-5-OEt-2-THI], [BH1690; 4-Me-5-OCF ₃ -2] -THI], [BH1691; 4- Me-5-OCHF 2 -2-THI], [BH1692; 4-Me-5-CN-2-THI], [BH1693; 4-Me-5-SMe-2- THI], [BH1694; 4-Me-5-SEt-2-THI], [BH1695; 4-Me-5-c-Pr-2-THI], [BH1696; 4-Et-5-F-2-] THI], [BH1697; 4-Et-5-Cl-2-THI], [BH1698; 4-Et-5-Br-2-THI], [BH1699; 4-Et-5-I-2-THI] [BH1700; 4-Et-5-Me-2-THI],

[BH1701; 4-Et-5-Et-2-THI], [BH1702; 4-Et-5-Pr-2-THI], [BH1703; 4-Et-5-i-Pr-2-THI], [BH1704; 4-Et-5 -CF 3 -2-THI], [BH1705; 4-Et-5-CHF 2 -2-THI], [BH1706; 4-Et-5-OMe-2-THI], [BH1707; 4-Et-5 -OEt-2-THI], [BH1708; 4-Et-5-OCF 3 -2-THI], [BH1709; 4-Et-5-OCHF 2 -2-THI], [BH1710; 4-Et-5-CN-2-THI], [BH1711; 4-Et-5-SMe-2-THI], [BH1712; 4-Et-5-SEt-2-THI], [BH1713] ; 4-Et-5-c -Pr-2-THI], [BH1714; 4-CF 3 -5-F-2-THI], [BH1715; 4-CF 3 -5-Cl-2-THI], _{[BH1716; 4-CF 3 -5} -Br-2-THI], [BH1717; 4-CF 3 -5-I-2-THI], [BH1718; 4-CF 3 -5-Me-2-THI] _{, [BH1719; 4-CF 3} -5-Et-2-THI], [BH1720; 4-CF 3 -5-Pr-2-THI], [BH1721; 4-CF 3 -5-i-Pr-2 -THI], [BH1722; 4- CF 3 -5-CF 3 -2-THI], [BH1723; 4-CF 3 -5-CHF 2 -2-THI], [BH1724; 4-CF 3 -5- OMe-2-THI], [ BH1725; 4-CF 3 -5-OEt-2-THI], [BH1726; 4-CF 3 -5-OCF 3 -2-THI], [BH1727; 4-CF 3 - _{5-OCHF 2 -2-THI]} , [BH1728; 4-CF 3 -5-CN-2-THI], [BH1729; 4-CF 3 -5-SMe-2-THI], [BH1730; 4-CF _{3 -5-SEt-2-THI} ], [BH1731; 4-CF 3 -5-c-Pr-2-THI], [BH1732; 4-OMe-5-F-2-THI], [BH1733; 4 -OMe-5-Cl-2-THI], [BH1734; 4-OMe-5-Br-2-THI], [BH1735; 4-OMe-5-I-2-THI], [BH1736; 4-OMe -5-Me-2-TH [I], [BH1737; 4-OMe-5-Et-2-THI], [BH1738; 4-OMe-5-Pr-2-THI], [BH1739; 4-OMe-5-i-Pr-2-] THI], [BH1740; 4- OMe-5-CF 3 -2-THI], [BH1741; 4-OMe-5-CHF 2 -2-THI], [BH1742; 4-OMe-5-OMe-2- THI], [BH1743; 4- OMe-5-OEt-2-THI], [BH1744; 4-OMe-5-OCF 3 -2-THI], [BH1745; 4-OMe-5-OCHF 2 -2- THI], [BH1746; 4-OMe-5-CN-2-THI], [BH1747; 4-OMe-5-SMe-2-THI], [BH1748; 4-OMe-5-SEt-2-THI] , [BH1749; 4-OMe-5-c-Pr-2-THI], [BH1750; 4-OEt-5-F-2-THI], [BH1751; 4-OEt-5-Cl-2-THI] , [BH1752; 4-OEt-5-Br-2-THI], [BH1753; 4-OEt-5-I-2-THI], [BH1754; 4-OEt-5-Me-2-THI], [BH1752; BH1755; 4-OEt-5-Et-2-THI], [BH1756; 4-OEt-5-Pr-2-THI], [BH1757; 4-OEt-5-i-Pr-2-THI], [BH1 755; BH1758; 4-OEt-5- CF 3 -2-THI], [BH1759; 4-OEt-5-CHF 2 -2-THI], [BH1760; 4-OEt-5-OMe-2-THI], [ BH1761; 4-OEt-5- OEt-2-THI], [BH1762; 4-OEt-5-OCF 3 -2-THI], [BH1763; 4-OEt-5-OCHF 2 -2-THI], [ BH1764; 4-OEt-5-CN-2-THI], [BH1765; 4-OEt-5-SMe-2-THI], [BH1766; 4-OEt-5-SEt-2-THI], [BH1767; 4-OEt-5-c-Pr-2-THI !, [BH1768; 4-SMe-5-F-2-THI], [BH1769; 4-SMe-5-Cl-2-THI], [BH1770; 4-SMe-5-Br-2-THI, [BH1771; 4-SMe-5-I-2-THI], [BH1772; 4-SMe-5-Me-2-THI], [BH1773; SMe-5-E t-2-THI], [BH1774; 4-SMe-5-Pr-2-THI], [BH1775; 4-SMe-5-i-Pr-2-THI], [BH1776; 4-SMe-5- CF ₃ -2-THI, [BH 1777; 4-SMe-5-CHF ₂ -2-THI], [BH 1778; 4-SMe-5-OMe-2-THI], [BH 1779; 4-SMe-5- OEt-2-THI], [ BH1780; 4-SMe-5-OCF 3 -2-THI], [BH1781; 4-SMe-5-OCHF 2 -2-THI], [BH1782; 4-SMe-5- CN-2-THI, [BH1783; 4-SMe-5-SMe-2-THI], [BH1784; 4-SMe-5-SEt-2-THI], [BH1785; 4-SMe-5-c- Pr-2-THI, [BH1786; 3-F-2-THI], [BH 1787; 3-Cl-2-THI], [BH1788; 3-Br-2-THI], [BH1 789; 3-I- 2-THI], [BH1790; 3-Me-2-THI], [BH1791; 3-Et-2-THI], [BH1792; 3-Pr-2-THI], [BH1793; 3-i-Pr- 2-THI], [BH1794; 3-CF 3 -2-THI], [BH1795; 3-CHF 2 -2-THI], [BH1796; 3-OMe-2-THI], [BH1797; 3-OEt- 2-THI], [BH 1798; 3-OCF ₃ -2-THI], [BH 1799; 3-OCHF ₂ -2-THI], [BH1800; 3-F-4-F-2-THI],

[BH1801; 3-F-4-Cl-2-THI], [BH1802; 3-F-4-Br-2-THI], [BH1803; 3-F-4-I-2-THI], [BH1804] 3-F-4-Me-2-THI], [BH1805; 3-F-4-Et-2-THI], [BH1806; 3-F-4-Pr-2-THI], [BH1807; -F-4-i-Pr- 2-THI], [BH1808; 3-F-4-CF 3 -2-THI], [BH1809; 3-F-4-CHF 2 -2-THI], [BH1810 3-F-4-OMe-2-THI !, [BH1811; 3-F-4-OEt-2-THI], [BH1812; 3-F-4-OCF ₃ -2-THI], [BH1813; _{3-F-4-OCHF 2} -2-THI], [BH1814; 3-F-4-CN-2-THI], [BH1815; 3-F-4-SMe-2-THI], [BH1816; 3 -F-4-SEt-2-THI, [BH1817; 3-F-4-c-Pr-2-THI], [BH1818; 3-Cl-4-F-2-THI], [BH1819; 3 -Cl-4-Cl-2-THI], [BH1820; 3-Cl-4-Br-2-THI], [BH1821; 3-Cl-4-I-2-THI], [BH1822; 3-Cl -4-Me-2-THI], [BH1823; 3-Cl-4-Et-2-THI], [BH1824; 3-Cl-4-Pr-2-THI], [BH1825; 3-Cl-4 -i-Pr-2-THI] , [BH1826; 3-Cl-4-CF 3 -2-THI], [BH1827; 3-Cl-4-CHF 2 -2-THI], [BH1828; 3-Cl -4-OMe-2-THI] , [BH1829; 3-Cl-4-OEt-2-THI], [BH1830; 3-Cl-4-OCF 3 -2-THI], [BH1831; 3-Cl- 4-OCHF ₂ -2-THI, [BH1832; 3-Cl-4-CN-2-THI], [BH1833; 3-Cl-4-SMe-2-THI], [BH1834; 3-Cl-4 -SEt-2-THI, [BH1835; 3-Cl-4-c-Pr-2-THI], [BH1836; 3-Me-4-F-2-THI], [BH1837; 3-Me-4 -Cl-2-THI, [BH1838; 3-Me-4-Br-2-THI], [BH1839; 3-Me-4-I-2-THI] , [BH1840; 3-Me-4-Me-2-THI], [BH1841; 3-Me-4-Et-2-THI], [BH1842; 3-Me-4-Pr-2-THI], [BH1842; BH1843; 3-Me-4- i-Pr-2-THI], [BH1844; 3-Me-4-CF 3 -2-THI], [BH1845; 3-Me-4-CHF 2 -2-THI] , [BH1846; 3-Me- 4-OMe-2-THI], [BH1847; 3-Me-4-OEt-2-THI], [BH1848; 3-Me-4-OCF 3 -2-THI], [BH1849; 3-Me-4 -OCHF 2 -2-THI], [BH1850; 3-Me-4-CN-2-THI], [BH1851; 3-Me-4-SMe-2-THI], [ BH1852; 3-Me-4-SEt-2-THI], [BH1853; 3-Me-4-c-Pr-2-THI], [BH1854; 3-Et-4-F-2-THI], [BH1852; BH1 855; 3-Et-4-Cl-2-THI], [BH1 856; 3-Et-4-Br-2-THI], [BH1 857; 3-Et-4-I-2-THI], [BH1 858; 3-Et-4-Me-2-THI], [BH 1859; 3-Et-4-Et-2-THI], [BH 1860; 3-Et-4-Pr-2-THI], [BH 1861; 3- Et-4-i-Pr-2-THI], [BH1862; 3-Et-4-CF ₃ -2-THI], [BH1863; 3-Et-4-CHF ₂ -2-THI], [BH 1864; 3-Et-4-OMe-2-THI], [BH 1865; 3-Et-4-OEt-2-THI], [BH 1866; 3-Et-4-OCF ₃ -2-THI], [BH 1867; _{-Et-4-OCHF 2 -2-} THI], [BH1868; 3-Et-4-CN-2-THI], [BH1869; 3-Et-4-SMe-2-THI], [BH1870; 3- Et-4-SEt-2- THI], [BH1871; 3-Et-4-c-Pr-2-THI], [BH1872; 3-CF 3 -4-F-2-THI], [BH1873; 3 _{-CF 3 -4-Cl-2-} THI], [BH1874; 3-CF 3 -4-Br-2-THI], [BH1875; 3-CF 3 -4-I-2-THI], [BH1876; 3-CF ₃ -4-Me-2-THI, [BH 1877; 3-CF ₃ -4-Et-2-THI], [BH1 878; 3-CF ₃ -4-Pr-2-THI], [BH 1879; 3-CF ₃ -4-i-Pr-2-THI], [BH 1 880; 3 _{-CF 3 -4-CF 3 -2-} THI], [BH1881; 3-CF 3 -4-CHF 2 -2-THI], [BH1882; 3-CF 3 -4-OMe-2-THI], [ _{BH1883; 3-CF 3 -4-} OEt-2-THI], [BH1884; 3-CF 3 -4-OCF 3 -2-THI], [BH1885; 3-CF 3 -4-OCHF 2 -2-THI ], [BH1886; 3-CF 3 -4-CN-2-THI], [BH1887; 3-CF 3 -4-SMe-2-THI], [BH1888; 3-CF 3 -4-SEt-2- THI], [BH1889; 3- CF 3 -4-c-Pr-2-THI], [BH1890; 3-OMe-4-F-2-THI], [BH1891; 3-OMe-4-Cl-2 -THI], [BH1892; 3-OMe-4-Br-2-THI], [BH1893; 3-OMe-4-I-2-THI], [BH1894; 3-OMe-4-Me-2-THI ], [BH 1895; 3-OMe-4-Et-2-THI], [BH 1896; 3-OMe-4-Pr-2-THI], [BH 1897; 3-OMe-4-i-Pr-2-THI] ], [BH 1898; 3-OMe-4-CF ₃ -2-THI], [BH 1899; 3-OMe-4-CHF ₂ -2-THI], [BH 1900; 3-OMe-4-OMe -2-THI] ],

[BH1901; 3-OMe-4 -OEt-2-THI], [BH1902; 3-OMe-4-OCF 3 -2-THI], [BH1903; 3-OMe-4-OCHF 2 -2-THI], [BH1904; 3-OMe-4-CN-2-THI], [BH1905; 3-OMe-4-SMe-2-THI], [BH1906; 3-OMe-4-SEt-2-THI], [BH1907] 3-OMe-4-c-Pr-2-THI !, [BH1908; 3-OEt-4-F-2-THI], [BH1909; 3-OEt-4-Cl-2-THI], [BH1910] 3-OEt-4-Br-2-THI !, [BH1911; 3-OEt-4-I-2-THI], [BH1912; 3-OEt-4-Me-2-THI], [BH1913; 3 -OEt-4-Et-2-THI], [BH1914; 3-OEt-4-Pr-2-THI], [BH1915; 3-OEt-4-i-Pr-2-THI], [BH1916; 3 _{-OEt-4-CF 3 -2-} THI], [BH1917; 3-OEt-4-CHF 2 -2-THI], [BH1918; 3-OEt-4-OMe-2-THI], [BH1919; 3 -OEt-4-OEt-2- THI], [BH1920; 3-OEt-4-OCF 3 -2-THI], [BH1921; 3-OEt-4-OCHF 2 -2-THI], [BH1922; 3 -OEt-4-CN-2-THI], [BH1923; 3-OEt-4-SMe-2-THI], [BH1924; 3-OEt-4-SEt-2-THI], [BH1925; 3-OEt -4-c-Pr-2-THI, [BH1926; 3-SMe-4-F-2-THI], [BH1 927; 3-SMe-4-Cl-2-THI], [BH1928; 3-SMe -4-Br-2-THI, [BH1 929; 3-SMe-4-I-2-THI], [BH1930; 3-SMe-4-Me-2-THI], [BH1931; 3-SMe-4 -Et-2-THI], [BH1932; 3-SMe-4-Pr-2-THI], [BH1933; 3-SMe-4-i-Pr-2-THI], [BH1934; 3-SMe-4 _{-CF 3 -2-THI], [} BH1935; 3-SMe-4-CHF 2 -2-THI], [BH1936; 3-SMe-4-OMe-2-THI], [BH1937; 3-SMe-4 -OEt- 2-THI], [BH 1938; 3-SMe-4-OCF ₃ -2-THI], [BH 1939; 3-SMe-4-OCHF ₂ 2-THI], [BH 1940; 3-SMe-4-CN- 2-THI], [BH1941; 3-SMe-4-SMe-2-THI], [BH1942; 3-SMe-4-SEt-2-THI], [BH1943; 3-SMe-4-c-Pr- 2-THI], [BH1 944; 3-F-5-F-2-THI], [BH 1945; 3-F-5-Cl-2-THI], [BH 1946; 3-F-5-Br-2- THI], [BH 1947; 3-F-5-I-2-THI], [BH 1948; 3-F-5-Me-2-THI], [BH 1949; 3-F-5-Et-2-THI] , [BH1950; 3-F- 5-Pr-2-THI], [BH1951; 3-F-5-i-Pr-2-THI], [BH1952; 3-F-5-CF 3 -2-THI ], [BH1953; 3-F -5-CHF 2 -2-THI], [BH1954; 3-F-5-OMe-2-THI], [BH1955; 3-F-5-OEt-2-THI] , [BH1956; 3-F- 5-OCF 3 -2-THI], [BH1957; 3-F-5-OCHF 2 -2-THI], [BH1958; 3-F-5-CN-2-THI] [BH1959; 3-F-5-SMe-2-THI], [BH1960; 3-F-5-SEt-2-THI], [BH1961; 3-F-5-c-Pr-2-THI] [BH1962; 3-Cl-5-F-2-THI], [BH1963; 3-Cl-5-Cl-2-THI], [BH1964; 3-Cl-5-Br-2-THI], [BH1962; BH 1 965; 3-Cl-5-I-2-THI], [BH 1966; 3-Cl-5-Me-2-THI], [BH 1967; 3-Cl-5-Et-2-THI], [BH 1968; 3-Cl-5-Pr- 2-THI], [BH1969; 3-Cl-5-i-Pr-2-THI], [BH1970; 3-Cl-5-CF 3 -2-THI], [BH1971 ; 3-Cl-5-CHF 2 -2-THI], [BH1972; 3-Cl-5-OMe-2-THI], [BH1973; 3-Cl-5-OEt-2-THI], [BH1974; _{3-Cl-5-OCF 3} -2-THI], [BH1975; 3-Cl-5-OCHF 2 -2-THI], [B H1976; 3-Cl-5-CN-2-THI], [BH 1977; 3-Cl-5-SMe-2-THI], [BH1978; 3-Cl-5-SEt-2-THI], [BH 1979; 3-Cl-5-c-Pr-2-THI], [BH1980; 3-Me-5-F-2-THI], [BH1981; 3-Me-5-Cl-2-THI], [BH1982; 3-Me-5-Br-2-THI], [BH1983; 3-Me-5-I-2-THI], [BH1984; 3-Me-5-Me-2-THI], [BH1985; 3- Me-5-Et-2-THI], [BH 1986; 3-Me-5-Pr-2-THI], [BH 1987; 3-Me-5-i-Pr-2-THI], [BH 1988; _{Me-5-CF 3 -2-} THI], [BH1989; 3-Me-5-CHF 2 -2-THI], [BH1990; 3-Me-5-OMe-2-THI], [BH1991; 3- Me-5-OEt-2- THI], [BH1992; 3-Me-5-OCF 3 -2-THI], [BH1993; 3-Me-5-OCHF 2 -2-THI], [BH1994; 3- Me-5-CN-2-THI], [BH1995; 3-Me-5-SMe-2-THI], [BH1996; 3-Me-5-SEt-2-THI], [BH1997; 3-Me- 5-c-Pr-2-THI, [BH1998; 3-Et-5-F-2-THI], [BH1999; 3-Et-5-Cl-2-THI], [BH2000; 3-Et- 5-Br-2-THI],

[BH2001; 3-Et-5-I-2-THI], [BH2002; 3-Et-5-Me-2-THI], [BH2003; 3-Et-5-Et-2-THI], [BH2004] 3-Et-5-Pr-2-THI, [BH2005; 3-Et-5-i-Pr-2-THI], [BH2006; 3-Et-5-CF ₃ -2-THI], [B. BH2007; 3-Et-5- CHF 2 -2-THI], [BH2008; 3-Et-5-OMe-2-THI], [BH2009; 3-Et-5-OEt-2-THI], [BH2010 ; 3-Et-5-OCF 3 -2-THI], [BH2011; 3-Et-5-OCHF 2 -2-THI], [BH2012; 3-Et-5-CN-2-THI], [BH2013 3-Et-5-SMe-2-THI], [BH2014; 3-Et-5-SEt-2-THI], [BH2015; 3-Et-5-c-Pr-2-THI], [BH2016] _{; 3-CF 3 -5-F} -2-THI], [BH2017; 3-CF 3 -5-Cl-2-THI], [BH2018; 3-CF 3 -5-Br-2-THI], [ _{BH2019; 3-CF 3 -5-} I-2-THI], [BH2020; 3-CF 3 -5-Me-2-THI], [BH2021; 3-CF 3 -5-Et-2-THI], _{[BH2022; 3-CF 3 -5} -Pr-2-THI], [BH2023; 3-CF 3 -5-i-Pr-2-THI], [BH2024; 3-CF 3 -5-CF 3 -2 -THI], [BH2025; 3- CF 3 -5-CHF 2 -2-THI], [BH2026; 3-CF 3 -5-OMe-2-THI], [BH2027; 3-CF 3 -5-OEt -2-THI], [BH2028; 3-CF 3 -5-OCF 3 -2-THI], [BH2029; 3-CF 3 -5-OCHF 2 -2-THI], [BH2030; 3-CF 3 - 5-CN-2-THI] , [BH2031; 3-CF 3 -5-SMe-2-THI], [BH2032; 3-CF 3 -5-SEt-2-THI], [BH2033; 3-CF 3 -5-c-Pr-2-THI, [BH2034; 3-OMe-5-F-2-THI], [BH2035; 3-OMe-5-Cl-2-THI], [BH2036; 3-OMe -5-Br-2-THI] , [BH2037; 3-OMe-5-I-2-THI], [BH2038; 3-OMe-5-Me-2-THI], [BH2039; 3-OMe-5-Et-2-THI], [BH2039; BH2040; 3-OMe-5- Pr-2-THI], [BH2041; 3-OMe-5-i-Pr-2-THI], [BH2042; 3-OMe-5-CF 3 -2-THI], [BH2043; 3-OMe-5 -CHF 2 -2-THI], [BH2044; 3-OMe-5-OMe-2-THI], [BH2045; 3-OMe-5-OEt-2-THI], [ BH2046; 3-OMe-5- OCF 3 -2-THI], [BH2047; 3-OMe-5-OCHF 2 -2-THI], [BH2048; 3-OMe-5-CN-2-THI], [ BH2049; 3-OMe-5-SMe-2-THI], [BH2050; 3-OMe-5-SEt-2-THI], [BH2051; 3-OMe-5-c-Pr-2-THI], [BH2051; BH2052; 3-OEt-5-F-2-THI], [BH2053; 3-OEt-5-Cl-2-THI], [BH2054; 3-OEt-5-Br-2-THI], [BH2055; 3-OEt-5-I-2-THI, [BH2056; 3-OEt-5-Me-2-THI], [BH2057; 3-OEt-5-Et-2-THI], [BH2058; OEt-5-Pr-2-THI, [BH 2059; 3-OEt-5-i-Pr-2-THI], [BH 2060; 3-OEt-5-CF ₃ -2-THI], [BH 2061; 3 _{-OEt-5-CHF 2 -2-} THI], [BH2062; 3-OEt-5-OMe-2-THI], [BH2063; 3-OEt-5-OEt-2-THI], [BH2064; 3- _{OEt-5-OCF 3 -2-} THI], [BH2065; 3-OEt-5-OCHF 2 -2-THI], [BH2066; 3-OEt-5-CN-2-THI], [BH2067; 3- OEt-5-SMe-2-THI], [BH2068; 3-OEt-5-SEt-2-THI], [BH2069; 3-OEt-5-c-Pr-2-THI], [BH2070; SMe-5-F-2-THI], [BH2071; 3-SMe-5-Cl-2-THI], [BH2072; 3-SMe-5-Br-2-THI], [BH2073; 3-SMe- 5-I-2 -THI], [BH 2074; 3-SMe-5-Me-2-THI], [BH 2075; 3-SMe-5-Et-2-THI], [BH 2076; 3-SMe-5-Pr-2-THI ], [BH2077; 3-SMe -5-i-Pr-2-THI], [BH2078; 3-SMe-5-CF 3 -2-THI], [BH2079; 3-SMe-5-CHF 2 -2 -THI], [BH2080; 3- SMe-5-OMe-2-THI], [BH2081; 3-SMe-5-OEt-2-THI], [BH2082; 3-SMe-5-OCF 3 -2- THI], [BH2083; 3- SMe-5-OCHF 2 -2-THI], [BH2084; 3-SMe-5-CN-2-THI], [BH2085; 3-SMe-5-SMe-2-THI ], [BH 2086; 3-SMe-5-SEt-2-THI], [BH 2087; 3-SMe-5-c-Pr-2-THI], [BH 2088; 3-Me-4-Me-5-F -2-THI, [BH2089; 3-Me-4-Me-5-Cl-2-THI], [BH2090; 3-Me-4-Me-5-Br-2-THI], [BH2091; 3 -Me-4-Me-5-I-2-THI, [BH2092; 3-Me-4-Me-5-Me-2-THI], [BH2093; 3-Me-4-Me-5-Et -2-THI, [BH 2094; 3-Me-4-Me-5-Pr-2-THI], [BH 2095; 3-Me-4-Me-5-i-Pr-2-THI], [BH 2096] ; 3-Me-4-Me -5-CF 3 -2-THI], [BH2097; 3-Me-4-Me-5-CHF 2 -2-THI], [BH2098; 3-Me-4-Me -5-OMe-2-THI, [BH 2099; 3-Me-4-Me-5-OEt-2-THI], [BH 2 100; 3-Me-4-Me-5-OCF ₃ -2-THI] ,

[BH2101; 3-Me-4 -Me-5-OCHF 2 -2-THI], [BH2102; 3-Me-4-Me-5-CN-2-THI], [BH2103; 3-Me-4- Me-5-SMe-2-THI, [BH2104; 3-Me-4-Me-5-SEt-2-THI], [BH2105; 3-Me-4-Me-5-c-Pr-2- THI], [BH2106; 3-Me-4-F-5-Me-2-THI], [BH2107; 3-Me-4-Cl-5-Me-2-THI], [BH2108; 3-Me- 4-Br-5-Me-2-THI, [BH2109; 3-Me-4-I-5-Me-2-THI], [BH2110; 3-Me-4-Et-5-Me-2-] THI], [BH2111; 3-Me-4-Pr-5-Me-2-THI], [BH2112; 3-Me-4-i-Pr-5-Me-2-THI], [BH2113; 3- _{Me-4-CF 3 -5-} Me-2-THI], [BH2114; 3-Me-4-CHF 2 -5-Me-2-THI], [BH2115; 3-Me-4-OMe-5- Me-2-THI], [ BH2116; 3-Me-4-OEt-5-Me-2-THI], [BH2117; 3-Me-4-OCF 3 -5-Me-2-THI], [BH2118 ; 3-Me-4-OCHF 2 -5-Me-2-THI], [BH2119; 3-Me-4-CN-5-Me-2-THI], [BH2120; 3-Me-4-SMe- 5-Me-2-THI, [BH2121; 3-Me-4-SEt-5-Me-2-THI], [BH2122; 3-Me-4-c-Pr-5-Me-2-THI] , [BH2123; -3-FUR], [BH2124; F-3-FUR], [BH2 125; Cl-3-FUR], [BH2126; Br-3-FUR], [BH2127; I-3-FUR], [BH2128; Me-3-FUR ], [BH2129; Et-3-FUR], [BH2130; Pr-3-FUR], [BH2131; i-Pr-3-FUR], [BH2132; CF 3 -3- _{FUR], [BH2133; CHF 2} -3-FUR], [BH2134; OMe-3-FUR], [BH2135; OEt-3-FUR], [BH2136; OCF 3 -3-FUR], [BH2137; OCHF 2 -3-FUR], [BH 2138; CN-3-FUR], [BH 21 39; SMe-3-FUR !, [BH2140; SEt-3-FUR], [BH2141; c-Pr-3-FUR], [BH2142; 5-F-3-FUR], [BH2143; 5-Cl- 3-FUR], [BH2144; 5-Br-3-FUR], [BH 2145; 5-I-3-FUR], [BH 2146; 5-Me-3-FUR], [BH 2147; 5-Et-3- FUR], [BH2148; 5-Pr-3-FUR], [BH 2149; 5-i-Pr-3-FUR], [BH 2150; 5-CF ₃ -3-FUR], [BH 2151; 5-CHF _2- 3-FUR], [BH2152; 5-OMe-3-FUR], [BH2153; 5-OEt-3-FUR], [BH2154; 5-OCF 3 -3-FUR], [BH2155; 5-OCHF 2 - 3-FUR], [BH2156; 5-CN-3-FUR], [BH2157; 5-SMe-3-FUR], [BH2158; 5-SEt-3-FUR], [BH2159; 5-c-Pr- 3-FUR], [BH2160; 2-F-5-F-3-FUR], [BH2161; 2-F-5-Cl-3-FUR], [BH2162; 2-F-5-Br-3- FUR], [BH2163; 2-F-5-I-3-FUR], [BH2164; 2-F-5-Me-3-FUR], [BH2165; 2-F-5-Et-3-FUR] , [BH2166; 2-F- 5-Pr-3-FUR], [BH2167; 2-F-5-i-Pr-3-FUR], [BH2168; 2-F-5-CF 3 -3-FUR ], [BH2169; 2-F -5-CHF 2 -3-FUR], [BH2170; 2-F-5-OMe-3-FUR], [BH2171; 2-F-5-OEt-3-FUR] , [BH2172; 2-F- 5-OCF 3 -3-FUR], [BH2173; 2-F-5-OCHF 2 -3-FUR], [BH2174; 2-F-5-CN-3-FUR] , [BH2175; 2-F-5-SMe-3-FUR], [BH2176; 2-F-5-SEt-3-FUR], [BH2177; 2-F-5-c-Pr-3-FUR] , [BH2178; 2-Cl-5-F-3-FUR], [BH2179; 2-Cl-5-Cl-3-FUR], [BH2180; 2-Cl-5-Br-3-FUR], [BH2 180; BH2181; 2-Cl-5-I-3-FUR], [BH2182; 2-Cl- 5-Me-3-FUR !, [BH 2183; 2-Cl-5-Et-3-FUR], [BH 2184; 2-Cl-5-Pr-3-FUR], [BH 2 185; 2-Cl-5- i-Pr-3-FUR] , [BH2186; 2-Cl-5-CF 3 -3-FUR], [BH2187; 2-Cl-5-CHF 2 -3-FUR], [BH2188; 2-Cl- 5-OMe-3-FUR] , [BH2189; 2-Cl-5-OEt-3-FUR], [BH2190; 2-Cl-5-OCF 3 -3-FUR], [BH2191; 2-Cl-5 _{-OCHF 2 -3-FUR], [} BH2192; 2-Cl-5-CN-3-FUR], [BH2193; 2-Cl-5-SMe-3-FUR], [BH2194; 2-Cl-5- SEt-3-FUR !, [BH2195; 2-Cl-5-c-Pr-3-FUR], [BH2196; 2-Me-5-F-3-FUR], [BH2197; Cl-3-FUR !, [BH 2198; 2-Me-5-Br-3-FUR], [BH 2199; 2-Me-5-I-3-FUR], [BH 2200; 2-Me-5-Me- 3-FUR],

[BH2201; 2-Me-5-Et-3-FUR], [BH2202; 2-Me-5-Pr-3-FUR], [BH2203; 2-Me-5-i-Pr-3-FUR], [BH2204; 2-Me-5 -CF 3 -3-FUR], [BH2205; 2-Me-5-CHF 2 -3-FUR], [BH2206; 2-Me-5-OMe-3-FUR], [BH2207; 2-Me-5 -OEt-3-FUR], [BH2208; 2-Me-5-OCF 3 -3-FUR], [BH2209; 2-Me-5-OCHF 2 -3-FUR], [BH2210; 2-Me-5-CN-3-FUR], [BH2211; 2-Me-5-SMe-3-FUR], [BH2212; 2-Me-5-SEt-3-FUR], [BH2213] 2-Me-5-c-Pr-3-FUR !, [BH2214; 2-Et-5-F-3-FUR], [BH2215; 2-Et-5-Cl-3-FUR], [BH2216] 2-Et-5-Br-3-FUR !, [BH2217; 2-Et-5-I-3-FUR], [BH2218; 2-Et-5-Me-3-FUR], [BH2219; -Et-5-Et-3-FUR], [BH2220; 2-Et-5-Pr-3-FUR], [BH2221; 2-Et-5-i-Pr-3-FUR], [BH2222; 2 _{-Et-5-CF 3 -3-} FUR], [BH2223; 2-Et-5-CHF 2 -3-FUR], [BH2224; 2-Et-5-OMe-3-FUR], [BH2225; 2 -Et-5-OEt-3- FUR], [BH2226; 2-Et-5-OCF 3 -3-FUR], [BH2227; 2-Et-5-OCHF 2 -3-FUR], [BH2228; 2 -Et-5-CN-3-FUR], [BH2229; 2-Et-5-SMe-3-FUR], [BH2230; 2-Et-5-SEt-3-FUR], [BH2231; 2-Et -5-c-Pr-3- FUR], [BH2232; 2-CF 3 -5-F-3-FUR], [BH2233; 2-CF 3 -5-Cl-3-FUR], [BH2234; 2 _{-CF 3 -5-Br-3-} FUR], [BH2235; 2-CF 3 -5-I-3-FUR], [BH2236; 2-CF 3 -5-Me-3-FUR], [BH2237; _{2-CF 3 -5-Et-} 3-FUR], [BH2238; 2-CF _{3 -5-Pr-3-FUR} ], [BH2239; 2-CF 3 -5-i-Pr-3-FUR], [BH2240; 2-CF 3 -5-CF 3 -3-FUR], [BH2241 _{; 2-CF 3 -5-CHF} 2 -3-FUR], [BH2242; 2-CF 3 -5-OMe-3-FUR], [BH2243; 2-CF 3 -5-OEt-3-FUR], _{[BH2244; 2-CF 3 -5} -OCF 3 -3-FUR], [BH2245; 2-CF 3 -5-OCHF 2 -3-FUR], [BH2246; 2-CF 3 -5-CN-3- FUR], [BH2247; 2- CF 3 -5-SMe-3-FUR], [BH2248; 2-CF 3 -5-SEt-3-FUR], [BH2249; 2-CF 3 -5-c-Pr -3-FUR], [BH2250; 2-OMe-5-F-3-FUR], [BH2251; 2-OMe-5-Cl-3-FUR], [BH2252; 2-OMe-5-Br-3 -FUR], [BH2253; 2-OMe-5-I-3-FUR], [BH2254; 2-OMe-5-Me-3-FUR], [BH2255; 2-OMe-5-Et-3-FUR] ], [BH2256; 2-OMe -5-Pr-3-FUR], [BH2257; 2-OMe-5-i-Pr-3-FUR], [BH2258; 2-OMe-5-CF 3 -3- FUR], [BH2259; 2- OMe-5-CHF 2 -3-FUR], [BH2260; 2-OMe-5-OMe-3-FUR], [BH2261; 2-OMe-5-OEt-3-FUR ], [BH2262; 2-OMe -5-OCF 3 -3-FUR], [BH2263; 2-OMe-5-OCHF 2 -3-FUR], [BH2264; 2-OMe-5-CN-3-FUR ], [BH2265; 2-OMe-5-SMe-3-FUR], [BH2266; 2-OMe-5-SEt-3-FUR], [BH2267; 2-OMe-5-c-Pr-3-FUR] ], [BH2268; 2-OEt-5-F-3-FUR], [BH2269; 2-OEt-5-Cl-3-FUR], [BH2270; 2-OEt-5-Br-3-FUR], [BH2271; 2-OEt-5-I-3-FUR], [BH2272; 2-OEt-5-Me-3-FUR], [BH2273; 2-OEt-5-Et-3-FUR], [BH2274] 2 -OEt-5-Pr-3- FUR], [BH2275; 2-OEt-5-i-Pr-3-FUR], [BH2276; 2-OEt-5-CF 3 -3-FUR], [BH2277; _{2-OEt-5-CHF 2} -3-FUR], [BH2278; 2-OEt-5-OMe-3-FUR], [BH2279; 2-OEt-5-OEt-3-FUR], [BH2280; 2 _{-OEt-5-OCF 3 -3-} FUR], [BH2281; 2-OEt-5-OCHF 2 -3-FUR], [BH2282; 2-OEt-5-CN-3-FUR], [BH2283; 2 -OEt-5-SMe-3-FUR !, [BH2284; 2-OEt-5-SEt-3-FUR], [BH2285; 2-OEt-5-c-Pr-3-FUR], [BH2286; -SMe-5-F-3-FUR !, [BH2287; 2-SMe-5-Cl-3-FUR], [BH2288; 2-SMe-5-Br-3-FUR], [BH2289; 2-SMe -5-I-3-FUR !, [BH2290; 2-SMe-5-Me-3-FUR], [BH2291; 2-SMe-5-Et-3-FUR], [BH2292; 2-SMe-5 -Pr-3-FUR], [ BH2293; 2-SMe-5-i-Pr-3-FUR], [BH2294; 2-SMe-5-CF 3 -3-FUR], [BH2295; 2-SMe- _{5-CHF 2 -3-FUR]} , [BH2296; 2-SMe-5-OMe-3-FUR], [BH2297; 2-SMe-5-OEt-3-FUR], [BH2298; 2-SMe-5 _{-OCF 3 -3-FUR], [} BH2299; 2-SMe-5-OCHF 2 -3-FUR], [BH2300; 2-SMe-5-CN-3-FUR],

[BH2301; 2-SMe-5-SMe-3-FUR], [BH2302; 2-SMe-5-SEt-3-FUR], [BH2303; 2-SMe-5-c-Pr-3-FUR], [BH2304; 4-F-3-FUR], [BH2305; 4-Cl-3-FUR], [BH2306; 4-Br-3-FUR], [BH2307; 4-I-3-FUR], [BH2308] 4-Me-3-FUR !, [BH2309; 4-Et-3-FUR], [BH 2310; 4-Pr-3-FUR], [BH2311; 4-i-Pr-3-FUR], [BH2312] _{; 4-CF 3 -3-FUR} ], [BH2313; 4-CHF 2 -3-FUR], [BH2314; 4-OMe-3-FUR], [BH2315; 4-OEt-3-FUR], [BH2316 _{; 4-OCF 3 -3-FUR} ], [BH2317; 4-OCHF 2 -3-FUR], [BH2318; 2-F-4-F-3-FUR], [BH2319; 2-Cl-4-F -3-FUR !, [BH2320; 2-Br-4-F-3-FUR], [BH2321; 2-I-4-F-3-FUR], [BH2322; 2-Me-4-F-3] -FUR], [BH2323; 2-Et-4-F-3-FUR], [BH2324; 2-Pr-4-F-3-FUR], [BH2325; 2-i-Pr-4-F-3 -FUR], [BH2326; 2- CF 3 -4-F-3-FUR], [BH2327; 2-CHF 2 -4-F-3-FUR], [BH2328; 2-OMe-4-F-3 -FUR], [BH2329; 2- OEt-4-F-3-FUR], [BH2330; 2-OCF 3 -4-F-3-FUR], [BH2331; 2-OCHF 2 -4-F-3 -FUR], [BH2332; 2-CN-4-F-3-FUR], [BH2333; 2-SMe-4-F-3-FUR], [BH2334; 2-SEt-4-F-3-FUR] ], [BH2335; 2-c-Pr-4-F-3-FUR], [BH2336; 2-F-4-Cl-3-FUR], [BH2337; 2-Cl-4-Cl-3-FUR] ], [BH2338; 2-Br-4-Cl-3-FUR], [BH2339; 2-I-4-Cl-3-FUR], [BH2340; 2-Me-4-Cl-3-FUR], [BH2341; 2-Et-4-Cl-3-FUR], [BH2342; 2-Pr-4-Cl- 3-FUR], [BH2343; 2-i-Pr-4-Cl-3-FUR], [BH2344; 2-CF 3 -4-Cl-3-FUR], [BH2345; 2-CHF 2 -4- Cl-3-FUR !, [BH2346; 2-OMe-4-Cl-3-FUR], [BH 2347; 2-OEt-4-Cl-3-FUR], [BH 2348; 2-OCF ₃ -4-Cl] -3-FUR !, [BH 2349; 2-OCHF ₂ -4-Cl-3-FUR], [BH 2 350; 2-CN-4-Cl-3-FUR], [BH 2 351; 2-SMe-4-Cl- 3-FUR], [BH2352; 2-SEt-4-Cl-3-FUR], [BH2353; 2-c-Pr-4-Cl-3-FUR], [BH2354; 2-F-4-Me- 3-FUR], [BH2355; 2-Cl-4-Me-3-FUR], [BH2356; 2-Br-4-Me-3-FUR], [BH2357; 2-I-4-Me-3-3. FUR], [BH2358; 2-Me-4-Me-3-FUR], [BH2359; 2-Et-4-Me-3-FUR], [BH2360; 2-Pr-4-Me-3-FUR] , [BH2361; 2-i- Pr-4-Me-3-FUR], [BH2362; 2-CF 3 -4-Me-3-FUR], [BH2363; 2-CHF 2 -4-Me-3- FUR], [BH2364; 2- OMe-4-Me-3-FUR], [BH2365; 2-OEt-4-Me-3-FUR], [BH2366; 2-OCF 3 -4-Me-3-FUR ], [BH2367; 2-OCHF 2 -4-Me-3-FUR], [BH2368; 2-CN-4-Me-3-FUR], [BH2369; 2-SMe-4-Me-3-FUR] , [BH2370; 2-SEt-4-Me-3-FUR], [BH2371; 2-c-Pr-4-Me-3-FUR], [BH2372; 2-F-4-Et-3-FUR] , [BH2373; 2-Cl-4-Et-3-FUR], [BH2374; 2-Br-4-Et-3-FUR], [BH2375; 2-I-4-Et-3-FUR], [BH2 373; BH 2376; 2-Me-4-Et-3-FUR], [BH 2377; 2-Et-4-Et-3-FUR], [BH 2378; 2-Pr-4-Et-3-FUR], [BH 2379; 2-i-Pr-4- Et-3-FUR], [BH2380; 2-CF 3 -4-Et-3 -FUR], [BH2381; 2- CHF 2 -4-Et-3-FUR], [BH2382; 2-OMe-4-Et-3-FUR], [BH2383; 2-OEt-4-Et-3- FUR], [BH2384; 2- OCF 3 -4-Et-3-FUR], [BH2385; 2-OCHF 2 -4-Et-3-FUR], [BH2386; 2-CN-4-Et-3- FUR], [BH2387; 2-SMe-4-Et-3-FUR], [BH2388; 2-SEt-4-Et-3-FUR], [BH2389; 2-c-Pr-4-Et-3- FUR], [BH2390; 2- F-4-CF 3 -3-FUR], [BH2391; 2-Cl-4-CF 3 -3-FUR], [BH2392; 2-Br-4-CF 3 -3 -FUR], [BH2393; 2- I-4-CF 3 -3-FUR], [BH2394; 2-Me-4-CF 3 -3-FUR], [BH2395; 2-Et-4-CF 3 - 3-FUR], [BH2396; 2-Pr-4-CF 3 -3-FUR], [BH2397; 2-i-Pr-4-CF 3 -3-FUR], [BH2398; 2-CF 3 -4 _{-CF 3 -3-FUR], [} BH2399; 2-CHF 2 -4-CF 3 -3-FUR], [BH2400; 2-OMe-4-CF 3 -3-FUR],

[BH2401; 2-OEt-4 -CF 3 -3-FUR], [BH2402; 2-OCF 3 -4-CF 3 -3-FUR], [BH2403; 2-OCHF 2 -4-CF 3 -3- FUR], [BH2404; 2- CN-4-CF 3 -3-FUR], [BH2405; 2-SMe-4-CF 3 -3-FUR], [BH2406; 2-SEt-4-CF 3 -3 -FUR], [BH2407; 2- c-Pr-4-CF 3 -3-FUR], [BH2408; 2-F-4-OMe-3-FUR], [BH2409; 2-Cl-4-OMe- 3-FUR], [BH 2410; 2-Br-4-OMe-3-FUR], [BH 2411; 2-I-4-OMe-3-FUR], [BH 2412; 2-Me-4-OMe-3- FUR], [BH2413; 2-Et-4-OMe-3-FUR], [BH2414; 2-Pr-4-OMe-3-FUR], [BH2415; 2-i-Pr-4-OMe-3- FUR], [BH2416; 2- CF 3 -4-OMe-3-FUR], [BH2417; 2-CHF 2 -4-OMe-3-FUR], [BH2418; 2-OMe-4-OMe-3- FUR], [BH2419; 2- OEt-4-OMe-3-FUR], [BH2420; 2-OCF 3 -4-OMe-3-FUR], [BH2421; 2-OCHF 2 -4-OMe-3- FUR], [BH2422; 2-CN-4-OMe-3-FUR], [BH2423; 2-SMe-4-OMe-3-FUR], [BH2424; 2-SEt-4-OMe-3-FUR] , [BH2425; 2-c-Pr-4-OMe-3-FUR], [BH2426; 2-F-4-OEt-3-FUR], [BH2427; 2-Cl-4-OEt-3-FUR] , [BH2428; 2-Br-4-OEt-3-FUR], [BH2429; 2-I-4-OEt-3-FUR], [BH2430; 2-Me-4-OEt-3-FUR], [BH2428; BH2431; 2-Et-4-OEt-3-FUR], [BH2432; 2-Pr-4-OEt-3-FUR], [BH2433; 2-i-Pr-4-OEt-3-FUR], _{BH2434; 2-CF 3 -4-} OEt-3-FUR], [BH2435; 2-CHF 2 -4-OEt-3-FUR], [BH2436; 2-OMe-4-OEt-3-FUR], [ BH243 7; 2-OEt-4- OEt-3-FUR], [BH2438; 2-OCF 3 -4-OEt-3-FUR], [BH2439; 2-OCHF 2 -4-OEt-3-FUR], [ BH2440; 2-CN-4-OEt-3-FUR !, [BH2441; 2-SMe-4-OEt-3-FUR], [BH2442; 2-SEt-4-OEt-3-FUR], [BH2443; 2-c-Pr-4-OEt-3-FUR !, [BH2444; 2-F-4-SMe-3-FUR], [BH2445; 2-Cl-4-SMe-3-FUR], [BH2446; 2-Br-4-SMe-3-FUR !, [BH2447; 2-I-4-SMe-3-FUR], [BH2448; 2-Me-4-SMe-3-FUR], [BH2449; Et-4-SMe-3-FUR !, [BH2450; 2-Pr-4-SMe-3-FUR], [BH2451; 2-i-Pr-4-SMe-3-FUR], [BH2452; _{CF 3 -4-SMe-3-} FUR], [BH2453; 2-CHF 2 -4-SMe-3-FUR], [BH2454; 2-OMe-4-SMe-3-FUR], [BH2455; 2- OEt-4-SMe-3- FUR], [BH2456; 2-OCF 3 -4-SMe-3-FUR], [BH2457; 2-OCHF 2 -4-SMe-3-FUR], [BH2458; 2- CN-4-SMe-3-FUR !, [BH2459; 2-SMe-4-SMe-3-FUR], [BH2460; 2-SEt-4-SMe-3-FUR], [BH2461; 2-c- Pr-4-SMe-3-FUR !, [BH2462; 4-F-5-F-3-FUR], [BH2463; 4-F-5-Cl-3-FUR], [BH2464; 4-F- 5-Br-3-FUR !, [BH2465; 4-F-5-I-3-FUR], [BH2466; 4-F-5-Me-3-FUR], [BH2467; 4-F-5-4. Et-3-FUR], [BH2468; 4-F-5-Pr-3-FUR], [BH2469; 4-F-5-i-Pr-3-FUR], [BH2470; 4-F-5-] _{CF 3 -3-FUR], [} BH2471; 4-F-5-CHF 2 -3-FUR], [BH2472; 4-F-5-OMe-3-FUR], [BH2473; 4-F-5- OEt-3-FUR], [BH 2474; 4-F-5-OCF ₃ -3- FUR], [BH2475; 4- F-5-OCHF 2 -3-FUR], [BH2476; 4-F-5-CN-3-FUR], [BH2477; 4-F-5-SMe-3-FUR ], [BH2478; 4-F-5-SEt-3-FUR], [BH2479; 4-F-5-c-Pr-3-FUR], [BH2480; 4-Cl-5-F-3-FUR] ], [BH2481; 4-Cl-5-Cl-3-FUR], [BH2482; 4-Cl-5-Br-3-FUR], [BH2483; 4-Cl-5-I-3-FUR], [BH2484; 4-Cl-5-Me-3-FUR], [BH2485; 4-Cl-5-Et-3-FUR], [BH2486; 4-Cl-5-Pr-3-FUR], [BH2487 ; 4-Cl-5-i -Pr-3-FUR], [BH2488; 4-Cl-5-CF 3 -3-FUR], [BH2489; 4-Cl-5-CHF 2 -3-FUR], [BH2490; 4-Cl-5 -OMe-3-FUR], [BH2491; 4-Cl-5-OEt-3-FUR], [BH2492; 4-Cl-5-OCF 3 -3-FUR], [ BH2493; 4-Cl-5- OCHF 2 -3-FUR], [BH2494; 4-Cl-5-CN-3-FUR], [BH2495; 4-Cl-5-SMe-3-FUR], [BH2496 4-Cl-5-SEt-3-FUR !, [BH2497; 4-Cl-5-c-Pr-3-FUR], [BH2498; 4-Me-5-F-3-FUR], [BH2499] 4-Me-5-Cl-3-FUR], [BH2500; 4-Me-5-Br-3-FUR],

[BH2501; 4-Me-5-I-3-FUR], [BH2502; 4-Me-5-Me-3-FUR], [BH2503; 4-Me-5-Et-3-FUR], [BH2504] 4-Me-5-Pr-3-FUR !, [BH2505; 4-Me-5-i-Pr-3-FUR], [BH2506; 4-Me-5-CF ₃ -3-FUR], [B. BH2507; 4-Me-5- CHF 2 -3-FUR], [BH2508; 4-Me-5-OMe-3-FUR], [BH2509; 4-Me-5-OEt-3-FUR], [BH2510 ; 4-Me-5-OCF 3 -3-FUR], [BH2511; 4-Me-5-OCHF 2 -3-FUR], [BH2512; 4-Me-5-CN-3-FUR], [BH2513 4-Me-5-SMe-3-FUR !, [BH 2514; 4-Me-5-SEt-3-FUR], [BH 2515; 4-Me-5-c-Pr-3-FUR], [BH 2516] 4-Et-5-F-3-FUR !, [BH2517; 4-Et-5-Cl-3-FUR], [BH2518; 4-Et-5-Br-3-FUR], [BH2519; -Et-5-I-3-FUR], [BH2520; 4-Et-5-Me-3-FUR], [BH2521; 4-Et-5-Et-3-FUR], [BH2522; 4-Et -5-Pr-3-FUR] , [BH2523; 4-Et-5-i-Pr-3-FUR], [BH2524; 4-Et-5-CF 3 -3-FUR], [BH2525; 4- _{Et-5-CHF 2 -3-} FUR], [BH2526; 4-Et-5-OMe-3-FUR], [BH2527; 4-Et-5-OEt-3-FUR], [BH2528; 4-Et -5-OCF ₃ -3-FUR, [BH 2529; 4-Et-5-OCHF ₂ -3-FUR], [BH 2530; 4-Et-5-CN-3-FUR], [BH 2531; -5-SMe-3-FUR !, [BH2532; 4-Et-5-SEt-3-FUR], [BH2533; 4-Et-5-c-Pr-3-FUR], [BH2534; 4-CF _{3 -5-F-3-FUR} ], [BH2535; 4-CF 3 -5-Cl-3-FUR], [BH2536; 4-CF 3 -5-Br-3-FUR], [BH2537; 4- _{CF 3 -5-I-3-} FUR], [BH2538; 4-CF 3 -5-Me -3-FUR], [BH2539; 4-CF 3 -5-Et-3-FUR], [BH2540; 4-CF 3 -5-Pr-3-FUR], [BH2541; 4-CF 3 -5- i-Pr-3-FUR] , [BH2542; 4-CF 3 -5-CF 3 -3-FUR], [BH2543; 4-CF 3 -5-CHF 2 -3-FUR], [BH2544; 4- _{CF 3 -5-OMe-3-} FUR], [BH2545; 4-CF 3 -5-OEt-3-FUR], [BH2546; 4-CF 3 -5-OCF 3 -3-FUR], [BH2547; _{4-CF 3 -5-OCHF 2} -3-FUR], [BH2548; 4-CF 3 -5-CN-3-FUR], [BH2549; 4-CF 3 -5-SMe-3-FUR], [ _{BH2550; 4-CF 3 -5-} SEt-3-FUR], [BH2551; 4-CF 3 -5-c-Pr-3-FUR], [BH2552; 4-OMe-5-F-3-FUR] , [BH2553; 4-OMe-5-Cl-3-FUR], [BH2554; 4-OMe-5-Br-3-FUR], [BH2555; 4-OMe-5-I-3-FUR], BH2556; 4-OMe-5-Me-3-FUR], [BH2557; 4-OMe-5-Et-3-FUR], [BH2558; 4-OMe-5-Pr-3-FUR], [BH2559; 4-OMe-5-i-Pr-3-FUR !, [BH2560; 4-OMe-5-CF ₃ -3-FUR], [BH2561; 4-OMe-5-CHF ₂ -3-FUR], BH2562; 4-OMe-5- OMe-3-FUR], [BH2563; 4-OMe-5-OEt-3-FUR], [BH2564; 4-OMe-5-OCF 3 -3-FUR], [BH2565 ; 4-OMe-5-OCHF 2 -3-FUR], [BH2566; 4-OMe-5-CN-3-FUR], [BH2567; 4-OMe-5-SMe-3-FUR], [BH2568; 4-OMe-5-SEt-3-FUR !, [BH 2569; 4-OMe-5-c-Pr-3-FUR], [BH 2570; 4-OEt-5-F-3-FUR], [BH2571; 4-OEt-5-Cl-3-FUR !, [BH2572; 4-OEt-5-Br-3-FUR], [BH2573; 4-OEt-5-I-3-FUR], [BH2574; OE t-5-Me-3-FUR !, [BH2575; 4-OEt-5-Et-3-FUR], [BH2576; 4-OEt-5-Pr-3-FUR], [BH 2577; 4-OEt- 5-i-Pr-3- FUR], [BH2578; 4-OEt-5-CF 3 -3-FUR], [BH2579; 4-OEt-5-CHF 2 -3-FUR], [BH2580; 4- OEt-5-OMe-3- FUR], [BH2581; 4-OEt-5-OEt-3-FUR], [BH2582; 4-OEt-5-OCF 3 -3-FUR], [BH2583; 4-OEt -5-OCHF ₂ -3-FUR !, [BH2584; 4-OEt-5-CN-3-FUR], [BH 2585; 4-OEt-5-SMe-3-FUR], [BH 2586; 4-OEt- 5-SEt-3-FUR !, [BH2587; 4-OEt-5-c-Pr-3-FUR], [BH2588; 4-SMe-5-F-3-FUR], [BH2589; 4-SMe- 5-Cl-3-FUR !, [BH2590; 4-SMe-5-Br-3-FUR], [BH2591; 4-SMe-5-I-3-FUR], [BH2592; 4-SMe-5- Me-3-FUR !, [BH 2593; 4-SMe-5-Et-3-FUR], [BH 2594; 4-SMe-5-Pr-3-FUR], [BH 2595; 4-SMe-5-i- Pr-3-FUR], [BH 2596; 4-SMe-5-CF ₃ -3-FUR], [BH 2597; 4-SMe-5-CHF ₂ -3-FUR], [BH 2598; 4-SMe-5- OMe-3-FUR], [ BH2599; 4-SMe-5-OEt-3-FUR], [BH2600; 4-SMe-5-OCF 3 -3-FUR],

[BH2601; 4-SMe-5 -OCHF 2 -3-FUR], [BH2602; 4-SMe-5-CN-3-FUR], [BH2603; 4-SMe-5-SMe-3-FUR], [ BH2604; 4-SMe-5-SEt-3-FUR !, [BH2605; 4-SMe-5-c-Pr-3-FUR], [BH2606; 2-Me-4-Me-5-F-3-3. FUR], [BH2607; 2-Me-4-Me-5-Cl-3-FUR], [BH2608; 2-Me-4-Me-5-Br-3-FUR], [BH2609; 2-Me- 4-Me-5-I-3-FUR !, [BH 2610; 2-Me-4-Me-5-Me-3-FUR], [BH2611; 2-Me-4-Me-5-Et-3- FUR], [BH2612; 2-Me-4-Me-5-Pr-3-FUR], [BH2613; 2-Me-4-Me-5-i-Pr-3-FUR], [BH2614; 2- Me-4-Me-5- CF 3 -3-FUR], [BH2615; 2-Me-4-Me-5-CHF 2 -3-FUR], [BH2616; 2-Me-4-Me-5- OMe-3-FUR], [ BH2617; 2-Me-4-Me-5-OEt-3-FUR], [BH2618; 2-Me-4-Me-5-OCF 3 -3-FUR], [BH2619 ; 2-Me-4-Me -5-OCHF 2 -3-FUR], [BH2620; 2-Me-4-Me-5-CN-3-FUR], [BH2621; 2-Me-4-Me- 5-SMe-3-FUR !, [BH2622; 2-Me-4-Me-5-SEt-3-FUR], [BH2623; 2-Me-4-Me-5-c-Pr-3-FUR] , [BH2624; 2-F-4-Me-5-Me-3-FUR], [BH2625; 2-Cl-4-Me-5-Me-3-FUR], [BH2626; 2-Br-4- Me-5-Me-3-FUR !, [BH2627; 2-I-4-Me-5-Me-3-FUR], [BH2628; 2-Et-4-Me-5-Me-3-FUR] , [BH2629; 2-Pr- 4-Me-5-Me-3-FUR], [BH2630; 2-i-Pr-4-Me-5-Me-3-FUR], [BH2631; 2-CF 3 -4-Me-5-Me-3-FUR !, [BH2632; 2-CHF ₂ -4-Me-5-Me-3-FUR], [BH2633; 2-OMe-4-Me-5-M e-3-FUR], [ BH2634; 2-OEt-4-Me-5-Me-3-FUR], [BH2635; 2-OCF 3 -4-Me-5-Me-3-FUR], [BH2636 _{; 2-OCHF 2 -4-Me} -5-Me-3-FUR], [BH2637; 2-CN-4-Me-5-Me-3-FUR], [BH2638; 2-SMe-4-Me- 5-Me-3-FUR !, [BH2639; 2-SEt-4-Me-5-Me-3-FUR], [BH2640; 2-c-Pr-4-Me-5-Me-3-FUR] , [BH2641; -3-THI], [BH2642; 2-F-3-THI], [BH2643; 2-Cl-3-THI], [BH2644; 2-Br-3-THI], [BH2645; -I-3-THI, [BH2646; 2-Me-3-THI], [BH2647; 2-Et-3-THI], [BH 2648; 2-Pr-3-THI], [BH 2649; 2-i -Pr-3-THI], [ BH2650; 2-CF 3 -3-THI], [BH2651; 2-CHF 2 -3-THI], [BH2652; 2-OMe-3-THI], [BH2653; 2 -OEt-3-THI], [ BH2654; 2-OCF 3 -3-THI], [BH2655; 2-OCHF 2 -3-THI], [BH2656; 2-CN-3-THI], [BH2657; 2 -SMe-3-THI], [BH2658; 2-SEt-3-THI], [BH2659; 2-c-Pr-3-THI], [BH2660; 5-F-3-THI], [BH2661; -Cl-3-THI], [BH2662; 5-Br-3-THI], [BH2663; 5-I-3-THI], [BH2664; 5-Me-3-THI], [BH2665; 5-Et] -3-THI], [BH2666; 5-Pr-3-THI], [BH 2667; 5-i-Pr-3-THI], [BH 2668; 5-CF ₃ -3-THI], [BH 2 669; _{CHF 2 -3-THI], [} BH2670; 5-OMe-3-THI], [BH2671; 5-OEt-3-THI], [BH2672; 5-OCF 3 -3-THI], [BH2673; 5- OCHF ₂ -3-THI], [BH 2674; 5-CN-3-THI], [BH 2 675; 5-SMe-3-THI], [BH 2 676; -c-Pr-3-THI], [BH2678; 2-F-5-F-3-THI], [BH2679; 2-F-5-Cl-3-THI], [BH2680; 2-F-5 -Br-3-THI], [BH2681; 2-F-5-I-3-THI], [BH2682; 2-F-5-Me-3-THI], [BH2683; 2-F-5-Et] -3-THI, [BH2684; 2-F-5-Pr-3-THI], [BH2685; 2-F-5-i-Pr-3-THI], [BH2686; 2-F-5-CF _{3 -3-THI], [BH2687} ; 2-F-5-CHF 2 -3-THI], [BH2688; 2-F-5-OMe-3-THI], [BH2689; 2-F-5-OEt -3-THI], [BH2690; 2-F-5-OCF 3 -3-THI], [BH2691; 2-F-5-OCHF 2 -3-THI], [BH2692; 2-F-5-CN -3-THI, [BH2693; 2-F-5-SMe-3-THI], [BH2694; 2-F-5-SEt-3-THI], [BH2695; 2-F-5-c-Pr -3-THI, [BH2696; 2-Cl-5-F-3-THI], [BH 2697; 2-Cl-5-Cl-3-THI], [BH 2698; 2-Cl-5-Br-3 -THI], [BH2699; 2-Cl-5-I-3-THI], [BH2700; 2-Cl-5-Me-3-THI],

[BH2701; 2-Cl-5-Et-3-THI], [BH2702; 2-Cl-5-Pr-3-THI], [BH2703; 2-Cl-5-i-Pr-3-THI], [BH2704; 2-Cl-5 -CF 3 -3-THI], [BH2705; 2-Cl-5-CHF 2 -3-THI], [BH2706; 2-Cl-5-OMe-3-THI], [BH2707; 2-Cl-5 -OEt-3-THI], [BH2708; 2-Cl-5-OCF 3 -3-THI], [BH2709; 2-Cl-5-OCHF 2 -3-THI], [BH2710; 2-Cl-5-CN-3-THI], [BH2711; 2-Cl-5-SMe-3-THI], [BH2712; 2-Cl-5-SEt-3-THI], [BH2713] 2-Cl-5-c-Pr-3-THI], [BH2714; 2-Me-5-F-3-THI], [BH2715; 2-Me-5-Cl-3-THI], [BH2716; 2-Me-5-Br-3-THI !, [BH2717; 2-Me-5-I-3-THI], [BH2718; 2-Me-5-Me-3-THI], [BH2719; -Me-5-Et-3-THI], [BH2720; 2-Me-5-Pr-3-THI], [BH2721; 2-Me-5-i-Pr-3-THI], [BH2722; 2 _{-Me-5-CF 3 -3-} THI], [BH2723; 2-Me-5-CHF 2 -3-THI], [BH2724; 2-Me-5-OMe-3-THI], [BH2725; 2 -Me-5-OEt-3- THI], [BH2726; 2-Me-5-OCF 3 -3-THI], [BH2727; 2-Me-5-OCHF 2 -3-THI], [BH2728; 2 -Me-5-CN-3-THI], [BH2729; 2-Me-5-SMe-3-THI], [BH2730; 2-Me-5-SEt-3-THI], [BH2731; 2-Me -5-c-Pr-3-THI], [BH2732; 2-Et-5-F-3-THI], [BH2733; 2-Et-5-Cl-3-THI], [BH2734; 2-Et -5-Br-3-THI], [BH2735; 2-Et-5-I-3-THI], [BH2736; 2-Et-5-Me-3-THI], [BH2737; 2-Et-5 -Et-3-THI], [BH2738; 2-Et-5-Pr-3-THI], [BH273] 9; 2-Et-5- i-Pr-3-THI], [BH2740; 2-Et-5-CF 3 -3-THI], [BH2741; 2-Et-5-CHF 2 -3-THI] , [BH2742; 2-Et- 5-OMe-3-THI], [BH2743; 2-Et-5-OEt-3-THI], [BH2744; 2-Et-5-OCF 3 -3-THI], [BH2745; 2-Et-5 -OCHF 2 -3-THI], [BH2746; 2-Et-5-CN-3-THI], [BH2747; 2-Et-5-SMe-3-THI], [ BH2748; 2-Et-5- SEt-3-THI], [BH2749; 2-Et-5-c-Pr-3-THI], [BH2750; 2-CF 3 -5-F-3-THI], _{[BH2751; 2-CF 3 -5} -Cl-3-THI], [BH2752; 2-CF 3 -5-Br-3-THI], [BH2753; 2-CF 3 -5-I-3-THI] _{, [BH2754; 2-CF 3} -5-Me-3-THI], [BH2755; 2-CF 3 -5-Et-3-THI], [BH2756; 2-CF 3 -5-Pr-3-THI ], [BH2757; 2-CF 3 -5-i-Pr-3-THI], [BH2758; 2-CF 3 -5-CF 3 -3-THI], [BH2759; 2-CF 3 -5-CHF _{2 -3-THI], [BH2760} ; 2-CF 3 -5-OMe-3-THI], [BH2761; 2-CF 3 -5-OEt-3-THI], [BH2762; 2-CF 3 -5 _{-OCF 3 -3-THI], [} BH2763; 2-CF 3 -5-OCHF 2 -3-THI], [BH2764; 2-CF 3 -5-CN-3-THI], [BH2765; 2-CF _{3 -5-SMe-3-THI} ], [BH2766; 2-CF 3 -5-SEt-3-THI], [BH2767; 2-CF 3 -5-c-Pr-3-THI], [BH2768; 2-OMe-5-F-3-THI], [BH2769; 2-OMe-5-Cl-3-THI], [BH2770; 2-OMe-5-Br-3-THI], [BH2771; OMe-5-I-3-THI], [BH2772; 2-OMe-5-Me-3-THI], [BH2773; 2-OMe-5-Et-3-THI], [BH2774; 2-OMe- 5-Pr-3-THI], [ BH2775; 2-OMe-5- i-Pr-3-THI], [BH2776; 2-OMe-5-CF 3 -3-THI], [BH2777; 2-OMe-5-CHF 2 -3-THI] , [BH2778; 2-OMe- 5-OMe-3-THI], [BH2779; 2-OMe-5-OEt-3-THI], [BH2780; 2-OMe-5-OCF 3 -3-THI], [BH2781; 2-OMe-5 -OCHF 2 -3-THI], [BH2782; 2-OMe-5-CN-3-THI], [BH2783; 2-OMe-5-SMe-3-THI], [ BH2784; 2-OMe-5-SEt-3-THI], [BH2785; 2-OMe-5-c-Pr-3-THI], [BH2786; 2-OEt-5-F-3-THI], BH 2787; 2-OEt-5-Cl-3-THI], [BH2 788; 2-OEt-5-Br-3-THI], [BH 2 789; 2-OEt-5-I-3-THI], [BH 2 790; 2-OEt-5-Me-3-THI], [BH2791; 2-OEt-5-Et-3-THI], [BH2792; 2-OEt-5-Pr-3-THI], [BH2793; OEt-5-i-Pr- 3-THI], [BH2794; 2-OEt-5-CF 3 -3-THI], [BH2795; 2-OEt-5-CHF 2 -3-THI], [BH2796; 2-OEt-5-OMe- 3-THI], [BH2797; 2-OEt-5-OEt-3-THI], [BH2798; 2-OEt-5-OCF 3 -3-THI], [BH2799; 2 -OEt-5-OCHF ₂ -3-THI], [BH 2800; 2-OEt-5-CN -3-THI],

[BH2801; 2-OEt-5-SMe-3-THI], [BH2802; 2-OEt-5-SEt-3-THI], [BH2803; 2-OEt-5-c-Pr-3-THI], [BH2804; 2-SMe-5-F-3-THI], [BH2805; 2-SMe-5-Cl-3-THI], [BH2806; 2-SMe-5-Br-3-THI], [BH2807] 2-SMe-5-I-3-THI], [BH2808; 2-SMe-5-Me-3-THI], [BH2809; 2-SMe-5-Et-3-THI], [BH 2810; -SMe-5-Pr-3- THI], [BH2811; 2-SMe-5-i-Pr-3-THI], [BH2812; 2-SMe-5-CF 3 -3-THI], [BH2813; _{2-SMe-5-CHF 2} -3-THI], [BH2814; 2-SMe-5-OMe-3-THI], [BH2815; 2-SMe-5-OEt-3-THI], [BH2816; 2 _{-SMe-5-OCF 3 -3-} THI], [BH2817; 2-SMe-5-OCHF 2 -3-THI], [BH2818; 2-SMe-5-CN-3-THI], [BH2819; 2 -SMe-5-SMe-3-THI], [BH2820; 2-SMe-5-SEt-3-THI], [BH2821; 2-SMe-5-c-Pr-3-THI], [BH2822; 4 -F-3-THI, [BH2823; 4-Cl-3-THI], [BH2824; 4-Br-3-THI], [BH2825; 4-I-3-THI], [BH2826; 4-Me -4-THI], [BH2827; 4-Et-3-THI], [BH2828; 4-Pr-3-THI], [BH2829; 4-i-Pr-3-THI], [BH2830; ₃ -3-THI, [BH 2831; 4-CHF ₂ -3-THI], [BH 2832; 4-OMe -3-THI], [BH 2833; 4-OEt -3-THI], [BH 2834; 4-OCF] ₃ -3-THI, [BH2 835; 4-OCHF ₂ -3-THI], [BH 2836; 2-F-4-F-3-THI], [BH 2837; 2-Cl-4-F-3-THI ], [BH2838; 2-Br-4-F-3-THI], [BH2839; 2-I-4-F-3-THI], [BH2840; 2-Me-4-F-3-THI], [BH2841; 2-Et -4-F-3-THI], [BH2842; 2-Pr-4-F-3-THI], [BH2843; 2-i-Pr-4-F-3-THI], [BH2844; 2-CF _{3 -4-F-3-THI} ], [BH2845; 2-CHF 2 -4-F-3-THI], [BH2846; 2-OMe-4-F-3-THI], [BH2847; 2-OEt -4-F-3-THI] , [BH2848; 2-OCF 3 -4-F-3-THI], [BH2849; 2-OCHF 2 -4-F-3-THI], [BH2850; 2-CN -4-F-3-THI], [BH2851; 2-SMe-4-F-3-THI], [BH2852; 2-SEt-4-F-3-THI], [BH2853; 2-c-Pr -4-F-3-THI], [BH2854; 2-F-4-Cl-3-THI], [BH2855; 2-Cl-4-Cl-3-THI], [BH2856; 2-Br-4 -Cl-3-THI], [BH2857; 2-I-4-Cl-3-THI], [BH2858; 2-Me-4-Cl-3-THI], [BH2859; 2-Et-4-Cl -3-THI], [BH2860; 2-Pr-4-Cl-3-THI], [BH2861; 2-i-Pr-4-Cl-3-THI], [BH2862; 2-CF 3 -4- Cl-3-THI], [ BH2863; 2-CHF 2 -4-Cl-3-THI], [BH2864; 2-OMe-4-Cl-3-THI], [BH2865; 2-OEt-4-Cl -3-THI], [BH2866; 2-OCF 3 -4-Cl-3-THI], [BH2867; 2-OCHF 2 -4-Cl-3-THI], [BH2868; 2-CN-4-Cl -3-THI, [BH 2869; 2-SMe-4-Cl-3-THI], [BH 2870; 2-SEt-4-Cl-3-THI], [BH 2 871; 2-c-Pr-4-Cl -3-THI, [BH2872; 2-F-4-Me-3-THI], [BH2873; 2-Cl-4-Me-3-THI], [BH2874; 2-Br-4-Me-3 -THI], [BH2875; 2-I-4-Me-3-THI], [BH2876; 2-Me-4-Me-3-THI], [BH2877; 2-Et-4-Me-3-THI ], [BH2878; 2-Pr-4-Me-3-THI], [BH2879; 2-i-Pr-4-Me-3-THI], [BH2] _{880; 2-CF 3 -4-} Me-3-THI], [BH2881; 2-CHF 2 -4-Me-3-THI], [BH2882; 2-OMe-4-Me-3-THI], [ BH2883; 2-OEt-4- Me-3-THI], [BH2884; 2-OCF 3 -4-Me-3-THI], [BH2885; 2-OCHF 2 -4-Me-3-THI], [ BH2886; 2-CN-4-Me-3-THI], [BH2887; 2-SMe-4-Me-3-THI], [BH2888; 2-SEt-4-Me-3-THI], [BH2889; 2-c-Pr-4-Me-3-THI], [BH2890; 2-F-4-Et-3-THI], [BH2891; 2-Cl-4-Et-3-THI], [BH2892; 2-Br-4-Et-3-THI], [BH2893; 2-I-4-Et-3-THI], [BH2894; 2-Me-4-Et-3-THI], [BH2895; Et-4-Et-3-THI], [BH2896; 2-Pr-4-Et-3-THI], [BH2897; 2-i-Pr-4-Et-3-THI], [BH2898; 2- _{CF 3 -4-Et-3-} THI], [BH2899; 2-CHF 2 -4-Et-3-THI], [BH2900; 2-OMe-4-Et-3-THI],

[BH2901; 2-OEt-4 -Et-3-THI], [BH2902; 2-OCF 3 -4-Et-3-THI], [BH2903; 2-OCHF 2 -4-Et-3-THI], [BH2904; 2-CN-4-Et-3-THI], [BH2905; 2-SMe-4-Et-3-THI], [BH2906; 2-SEt-4-Et-3-THI], [BH2907] ; 2-c-Pr-4 -Et-3-THI], [BH2908; 2-F-4-CF 3 -3-THI], [BH2909; 2-Cl-4-CF 3 -3-THI], [BH2910; 2-Br-4 -CF 3 -3-THI], [BH2911; 2-I-4-CF 3 -3-THI], [BH2912; 2-Me-4-CF 3 -3-THI] , [BH2913; 2-Et- 4-CF 3 -3-THI], [BH2914; 2-Pr-4-CF 3 -3-THI], [BH2915; 2-i-Pr-4-CF 3 -3 -THI], [BH2916; 2- CF 3 -4-CF 3 -3-THI], [BH2917; 2-CHF 2 -4-CF 3 -3-THI], [BH2918; 2-OMe-4-CF _{3 -3-THI], [BH2919} ; 2-OEt-4-CF 3 -3-THI], [BH2920; 2-OCF 3 -4-CF 3 -3-THI], [BH2921; 2-OCHF 2 - _{4-CF 3 -3-THI]} , [BH2922; 2-CN-4-CF 3 -3-THI], [BH2923; 2-SMe-4-CF 3 -3-THI], [BH2924; 2-SEt -4-CF ₃ -3-THI, [BH 2925; 2-c-Pr-4-CF ₃ -3-THI], [BH 2926; 2-F-4-OMe-3-THI], [BH 2 927; -Cl-4-OMe-3-THI], [BH2 928; 2-Br-4-OMe-3-THI], [BH2 929; 2-I-4-OMe-3-THI], [BH2 930; 2-Me -4-OMe-3-THI, [BH2931; 2-Et-4-OMe-3-THI], [BH2932; 2-Pr-4-OMe-3-THI], [BH2933; 2-i-Pr -4-OMe-3-THI] , [BH2934; 2-CF 3 -4-OMe-3-THI], [BH2935; 2-CHF 2 -4-OMe-3-THI], [BH2936; 2-OMe -4-OM e-3-THI], [ BH2937; 2-OEt-4-OMe-3-THI], [BH2938; 2-OCF 3 -4-OMe-3-THI], [BH2939; 2-OCHF 2 -4- OMe-3-THI], [BH2940; 2-CN-4-OMe-3-THI], [BH2941; 2-SMe-4-OMe-3-THI], [BH2942; 2-SEt-4-OMe- 3-THI], [BH2943; 2-c-Pr-4-OMe-3-THI], [BH2944; 2-F-4-OEt-3-THI], [BH2945; 2-Cl-4-OEt- 3-THI], [BH 2946; 2-Br-4-OEt-3-THI], [BH 2947; 2-I-4-OEt-3-THI], [BH 2948; 2-Me-4-OEt-3- THI], [BH 2949; 2-Et-4-OEt-3-THI], [BH 2950; 2-Pr-4-OEt-3-THI], [BH 2951; 2-i-Pr-4-OEt-3- THI], [BH2952; 2- CF 3 -4-OEt-3-THI], [BH2953; 2-CHF 2 -4-OEt-3-THI], [BH2954; 2-OMe-4-OEt-3- THI], [BH2955; 2- OEt-4-OEt-3-THI], [BH2956; 2-OCF 3 -4-OEt-3-THI], [BH2957; 2-OCHF 2 -4-OEt-3- THI], [BH2958; 2-CN-4-OEt-3-THI], [BH2959; 2-SMe-4-OEt-3-THI], [BH2960; 2-SEt-4-OEt-3-THI] , [BH2961; 2-c-Pr-4-OEt-3-THI], [BH2962; 2-F-4-SMe-3-THI], [BH2963; 2-Cl-4-SMe-3-THI] , [BH2964; 2-Br-4-SMe-3-THI], [BH2965; 2-I-4-SMe-3-THI], [BH2966; 2-Me-4-SMe-3-THI], [BH2964; BH2967; 2-Et-4-SMe-3-THI], [BH2968; 2-Pr-4-SMe-3-THI], [BH2969; 2-i-Pr-4-SMe-3-THI], _{BH2970; 2-CF 3 -4-} SMe-3-THI], [BH2971; 2-CHF 2 -4-SMe-3-THI], [BH2972; 2-OMe-4-SMe-3-THI], [ BH 2 973; 2-O Et-4-SMe-3- THI], [BH2974; 2-OCF 3 -4-SMe-3-THI], [BH2975; 2-OCHF 2 -4-SMe-3-THI], [BH2976; 2- CN-4-SMe-3-THI, [BH 2977; 2-SMe-4-SMe-3-THI], [BH 2978; 2-SEt-4-SMe-3-THI], [BH 2979; Pr-4-SMe-3-THI], [BH 2 980; 4-F-5-F-3-THI], [BH 2981; 4-F-5-Cl-3-THI], [BH 2 982; 4-F- 5-Br-3-THI, [BH2983; 4-F-5-I-3-THI], [BH2984; 4-F-5-Me-3-THI], [BH2985; Et-3-THI, [BH2986; 4-F-5-Pr-3-THI], [BH2987; 4-F-5-i-Pr-3-THI], [BH2988; 4-F-5-] CF ₃ -3-THI, [BH 2989; 4-F-5-CHF ₂ -3-THI], [BH ₂ 990; 4-F-5-OMe-3-THI], [BH 299 1; 4-F-5-] OEt-3-THI], [ BH2992; 4-F-5-OCF 3 -3-THI], [BH2993; 4-F-5-OCHF 2 -3-THI], [BH2994; 4-F-5- CN-3-THI, [BH2995; 4-F-5-SMe-3-THI], [BH2996; 4-F-5-SEt-3-THI], [BH2997; 4-F-5-c- Pr-3-THI, [BH 2998; 4-Cl-5-F-3-THI], [BH 2 999; 4-Cl-5-Cl-3-THI], [BH 3000; 4-Cl-5-Br- 3-THI],

[BH3001; 4-Cl-5-I-3-THI], [BH3002; 4-Cl-5-Me-3-THI], [BH3003; 4-Cl-5-Et-3-THI], [BH3004] 4-Cl-5-Pr-3-THI], [BH3005; 4-Cl-5-i-Pr-3-THI], [BH3006; 4-Cl-5-CF ₃ -3-THI], [B. BH3007; 4-Cl-5- CHF 2 -3-THI], [BH3008; 4-Cl-5-OMe-3-THI], [BH3009; 4-Cl-5-OEt-3-THI], [BH3010 ; 4-Cl-5-OCF 3 -3-THI], [BH3011; 4-Cl-5-OCHF 2 -3-THI], [BH3012; 4-Cl-5-CN-3-THI], [BH3013 4-Cl-5-SMe-3-THI !, [BH3014; 4-Cl-5-SEt-3-THI], [BH3015; 4-Cl-5-c-Pr-3-THI], [BH3016] 4-Me-5-F-3-THI !, [BH3017; 4-Me-5-Cl-3-THI], [BH3018; 4-Me-5-Br-3-THI], [BH3019; -Me-5-I-3-THI], [BH3020; 4-Me-5-Me-3-THI], [BH3021; 4-Me-5-Et-3-THI], [BH3022; 4-Me -5-Pr-3-THI] , [BH3023; 4-Me-5-i-Pr-3-THI], [BH3024; 4-Me-5-CF 3 -3-THI], [BH3025; 4- _{Me-5-CHF 2 -3-} THI], [BH3026; 4-Me-5-OMe-3-THI], [BH3027; 4-Me-5-OEt-3-THI], [BH3028; 4-Me _{-5-OCF 3 -3-THI]} , [BH3029; 4-Me-5-OCHF 2 -3-THI], [BH3030; 4-Me-5-CN-3-THI], [BH3031; 4-Me -5-SMe-3-THI, [BH 3032; 4-Me-5-SEt-3-THI], [BH 3033; 4-Me-5-c-Pr-3-THI], [BH 3034; 4-Et -5-F-3-THI], [BH3035; 4-Et-5-Cl-3-THI], [BH3036; 4-Et-5-Br-3-THI], [BH3037; 4-Et-5 -I-3-THI], [BH3038; 4-Et-5-Me-3-THI], [BH3039] 4-Et-5-Et-3-THI], [BH3040; 4-Et-5-Pr-3-THI], [BH3041; 4-Et-5-i-Pr-3-THI], [BH3042] ; 4-Et-5-CF 3 -3-THI], [BH3043; 4-Et-5-CHF 2 -3-THI], [BH3044; 4-Et-5-OMe-3-THI], [BH3045 ; 4-Et-5-OEt -3-THI], [BH3046; 4-Et-5-OCF 3 -3-THI], [BH3047; 4-Et-5-OCHF 2 -3-THI], [BH3048 4-Et-5-CN-3-THI, [BH3049; 4-Et-5-SMe-3-THI], [BH3050; 4-Et-5-SEt-3-THI], [BH3051; -Et-5-c-Pr- 3-THI], [BH3052; 4-CF 3 -5-F-3-THI], [BH3053; 4-CF 3 -5-Cl-3-THI], [BH3054 _{; 4-CF 3 -5-Br} -3-THI], [BH3055; 4-CF 3 -5-I-3-THI], [BH3056; 4-CF 3 -5-Me-3-THI], [ _{BH3057; 4-CF 3 -5-} Et-3-THI], [BH3058; 4-CF 3 -5-Pr-3-THI], [BH3059; 4-CF 3 -5-i-Pr-3-THI ], [BH3060; 4-CF 3 -5-CF 3 -3-THI], [BH3061; 4-CF 3 -5-CHF 2 -3-THI], [BH3062; 4-CF 3 -5-OMe- 3-THI], [BH3063; 4-CF 3 -5-OEt-3-THI], [BH3064; 4-CF 3 -5-OCF 3 -3-THI], [BH3065; 4-CF 3 -5- OFHF ₂ -3-THI, [BH 3066; 4-CF ₃ -5-CN 3-THI], [BH 3067; 4-CF ₃ -5-SMe-3-THI], [BH 3068; 4-CF _3- 5-SEt-3-THI] , [BH3069; 4-CF 3 -5-c-Pr-3-THI], [BH3070; 4-OMe-5-F-3-THI], [BH3071; 4-OMe -5-Cl-3-THI], [BH3072; 4-OMe-5-Br-3-THI], [BH3073; 4-OMe-5-I-3-THI], [BH3074; 4-OMe-5 -Me-3-THI], [BH3 075; 4-OMe-5-Et-3-THI], [BH3076; 4-OMe-5-Pr-3-THI], [BH3077; 4-OMe-5-i-Pr-3-THI], [B. BH3078; 4-OMe-5- CF 3 -3-THI], [BH3079; 4-OMe-5-CHF 2 -3-THI], [BH3080; 4-OMe-5-OMe-3-THI], [ BH3081; 4-OMe-5- OEt-3-THI], [BH3082; 4-OMe-5-OCF 3 -3-THI], [BH3083; 4-OMe-5-OCHF 2 -3-THI], [ BH3084; 4-OMe-5-CN-3-THI], [BH3085; 4-OMe-5-SMe-3-THI], [BH3086; 4-OMe-5-SEt-3-THI], [BH3087; 4-OMe-5-c-Pr-3-THI], [BH3088; 4-OEt-5-F-3-THI], [BH3089; 4-OEt-5-Cl-3-THI], [BH3090; 4-OEt-5-Br-3-THI], [BH3091; 4-OEt-5-I-3-THI], [BH3092; 4-OEt-5-Me-3-THI], [BH3093; OEt-5-Et-3-THI], [BH3094; 4-OEt-5-Pr-3-THI], [BH3095; 4-OEt-5-i-Pr-3-THI], [BH3096; _{OEt-5-CF 3 -3-} THI], [BH3097; 4-OEt-5-CHF 2 -3-THI], [BH3098; 4-OEt-5-OMe-3-THI], [BH3099; 4- OEt-5-OEt-3- THI], [BH3100; 4-OEt-5-OCF 3 -3-THI],

[BH3101; 4-OEt-5 -OCHF 2 -3-THI], [BH3102; 4-OEt-5-CN-3-THI], [BH3103; 4-OEt-5-SMe-3-THI], [ BH3104; 4-OEt-5-SEt-3-THI], [BH3105; 4-OEt-5-c-Pr-3-THI], [BH3106; 4-SMe-5-F-3-THI], [BH3 104; BH3107; 4-SMe-5-Cl-3-THI], [BH3108; 4-SMe-5-Br-3-THI], [BH3109; 4-SMe-5-I-3-THI], [BH3110; 4-SMe-5-Me-3-THI, [BH3111; 4-SMe-5-Et-3-THI], [BH3112; 4-SMe-5-Pr-3-THI], [BH3113; SMe-5-i-Pr- 3-THI], [BH3114; 4-SMe-5-CF 3 -3-THI], [BH3115; 4-SMe-5-CHF 2 -3-THI], [BH3116; 4-SMe-5-OMe- 3-THI], [BH3117; 4-SMe-5-OEt-3-THI], [BH3118; 4-SMe-5-OCF 3 -3-THI], [BH3119; 4 -SMe-5-OCHF ₂ -3-THI], [BH 3120; 4-SMe-5-CN-3-THI], [BH 3121; 4-SMe-5-SMe-3-THI], [BH 3122; 4- SMe-5-SEt-3-THI, [BH3123; 4-SMe-5-c-Pr-3-THI], [BH3124; 2-Me-4-Me-5-F-3-THI], [B. BH3 125; 2-Me-4-Me-5-Cl-3-THI], [BH3126; 2-Me-4-Me-5-Br-3-THI], [BH3127; 2-Me-4-Me- 5-I-3-THI, [BH3128; 2-Me-4-Me-5-Me-3-THI], [BH3129; 2-Me-4-Me-5-Et-3-THI], [B. BH3130; 2-Me-4-Me-5-Pr-3-THI], [BH3131; 2-Me-4-Me-5-i-Pr-3-THI], [BH3132; 2-Me-4- _{Me-5-CF 3 -3-} THI], [BH3133; 2-Me-4-Me-5-CHF 2 -3-THI], [BH3134; 2-Me-4-Me-5-OMe-3- THI], [BH3135; 2-Me-4-Me-5-OEt-3-THI], [B H3136; 2-Me-4- Me-5-OCF 3 -3-THI], [BH3137; 2-Me-4-Me-5-OCHF 2 -3-THI], [BH3138; 2-Me-4- Me-5-CN-3-THI, [BH3139; 2-Me-4-Me-5-SMe-3-THI], [BH3140; 2-Me-4-Me-5-SEt-3-THI] , [BH3141; 2-Me-4-Me-5-c-Pr-3-THI], [BH3142; 2-F-4-Me-5-Me-3-THI], [BH3143; 2-Cl- 4-Me-5-Me-3-THI, [BH3144; 2-Br-4-Me-5-Me-3-THI], [BH3145; 2-I-4-Me-5-Me-3- THI], [BH3146; 2-Et-4-Me-5-Me-3-THI], [BH3147; 2-Pr-4-Me-5-Me-3-THI], [BH3148; 2-i- Pr-4-Me-5- Me-3-THI], [BH3149; 2-CF 3 -4-Me-5-Me-3-THI], [BH3150; 2-CHF 2 -4-Me-5- Me-3-THI], [BH3151; 2-OMe-4-Me-5-Me-3-THI], [BH3152; 2-OEt-4-Me-5-Me-3-THI], [BH3153; _{2-OCF 3 -4-Me-} 5-Me-3-THI], [BH3154; 2-OCHF 2 -4-Me-5-Me-3-THI], [BH3155; 2-CN-4-Me- 5-Me-3-THI], [BH3156; 2-SMe-4-Me-5-Me-3-THI], [BH3157; 2-SEt-4-Me-5-Me-3-THI], [B. BH3158; 2-c-Pr-4-Me-5-Me-3-THI], [BH3159; -2-TRI], [BH3160; 4-F-2-TRI], [BH3161; 4-Cl-2 -TRI], [BH3162; 4-Br-2-TRI], [BH3163; 4-Me-2-TRI], [BH3164; 4-Et-2-TRI], [BH3165; 4-OMe-2-TRI] ], [BH3166; 4-SMe -2-TRI], [BH3167; 4-CF 3 -2-TRI], [BH3168; 4-F-5-F-2-TRI], [BH3169; 4-F- 5-Cl-2-TRI], [BH3170; 4-F-5-Br-2-TRI], [BH3171; 4-F-5-Me-2-TRI], [B H3172; 4-F-5-Et-2-TRI], [BH3173; 4-F-5-OMe-2-TRI], [BH3174; 4-F-5-SMe-2-TRI], [BH3175; _{4-F-5-CF 3} -2-TRI], [BH3176; 4-Me-5-F-2-TRI], [BH3177; 4-Me-5-Cl-2-TRI], [BH3178; 4 -Me-5-Br-2-TRI], [BH3179; 4-Me-5-Me-2-TRI], [BH 3180; 4-Me-5-Et-2-TRI], [BH3181; 4-Me -5-OMe-2-TRI] , [BH3182; 4-Me-5-SMe-2-TRI], [BH3183; 4-Me-5-CF 3 -2-TRI], [BH3184; 4-OMe- 5-F-2-TRI], [BH3185; 4-OMe-5-Cl-2-TRI], [BH3186; 4-OMe-5-Br-2-TRI], [BH3187; 4-OMe-5- Me-2-TRI], [BH3188; 4-OMe-5-Et-2-TRI], [BH3189; 4-OMe-5-OMe-2-TRI], [BH3190; 4-OMe-5-SMe- 2-TRI], [BH3191; 4-OMe-5-CF 3 -2-TRI], [BH3192; 1-TRI], [BH3193; 4-F-1-TRI], [BH3194; 4-Cl-1 -TRI], [BH3195; 4-Br-1-TRI], [BH3196; 4-Me-1-TRI], [BH3197; 4-Et-1-TRI], [BH3198; 4-OMe-1-TRI] ], [BH3199; 4-SMe-1-TRI], [BH3200; 4-CF ₃ -1-TRI],

[BH3201; 5-F-1-TRI], [BH3202; 5-Cl-1-TRI], [BH3203; 5-Br-1-TRI], [BH3204; 5-Me-1-TRI], [BH3205] 5-Et-1-TRI], [BH3206; 5-OMe-1-TRI], [BH3207; 5-SMe-1-TRI], [BH3208; 5-CF ₃ -1-TRI], [BH3209; 4-F-5-F-1-TRI], [BH 3210; 4-F-5-Cl-1-TRI], [BH 3211; 4-F-5-Br-1-TRI], [BH 3212; 4- F-5-Me-1-TRI], [BH3213; 4-F-5-Et-1-TRI], [BH3214; 4-F-5-OMe-1-TRI], [BH3215; 4-F- 5-SMe-1-TRI] , [BH3216; 4-F-5-CF 3 -1-TRI], [BH3217; 4-Me-5-F-1-TRI], [BH3218; 4-Me-5 -Cl-1-TRI], [BH3219; 4-Me-5-Br-1-TRI], [BH3220; 4-Me-5-Me-1-TRI], [BH3221; 4-Me-5-Et] -1-TRI], [BH 3222; 4-Me-5-OMe-1-TRI], [BH 3223; 4-Me-5-SMe-1-TRI], [BH 3224; 4-Me-5-CF _3- 1-TRI], [BH3225; 4-OMe-5-F-1-TRI], [BH3226; 4-OMe-5-Cl-1-TRI], [BH3227; 4-OMe-5-Br-1- TRI], [BH3228; 4-OMe-5-Me-1-TRI], [BH3229; 4-OMe-5-Et-1-TRI], [BH3230; 4-OMe-5-OMe-1-TRI] , [BH3231; 4-OMe- 5-SMe-1-TRI], [BH3232; 4-OMe-5-CF 3 -1-TRI], [BH3233; 2-Oxazolin-4-ly], [BH3234; 2 -Me-2-Oxazolin-4-ly, [BH3235; 4-Me-2-Oxazolin-4-ly], [BH3236; 5-Me-2-Oxazolin-4-ly], [BH3237; 2-Me -4-Me-2-Oxazolin-4-ly], [BH3238; 2-Me-5-Me-2-Oxazolin-4-ly], [BH3239; 4-Me-5-Me-2-Oxazolin-4 -ly], [BH3 240; 5-Me-5-Me-2-Oxazolin-4-ly], [BH3241; 2-Me-4-Me-5-Me-2-Oxazolin-5-ly], [BH3242; 2-Oxazolin- 5-ly, [BH 3243; 2-Me-2-Oxazolin-5-ly], [BH 3244; 5-Me-2-Oxazolin-5-ly], [BH 3245; 4-Me-2-Oxazolin-5- ly], [BH3246; 2-Me-5-Me-2-Oxazolin-5-ly], [BH3247; 2-Me-4-Me-2-Oxazolin-5-ly], [BH 3248; 5-Me- 4-Me-2-Oxazolin-5-ly, [BH3249; 4-Me-4-Me-2-Oxazolin-5-ly], [BH3250; 2-Me-5-Me-4-Me-2- Oxazolin-5-ly, [BH3251; 3-Oxazolin-2-ly], [BH3252; 2-Me-3-Oxazolin-2-ly], [BH3253; 4-Me-3-Oxazolin-2-ly] , [BH3254; 5-Me-3-Oxazolin-2-ly], [BH3255; 2-Me-4-Me-3-Oxazolin-2-ly], [BH3256; 2-Me-5-Me-3-3. Oxazolin-2-ly, [BH3257; 4-Me-5-Me-3-Oxazolin-2-ly], [BH3258; 5-Me-5-Me-3-Oxazolin-2-ly], [BH3259; 2-Me-4-Me-5-Me-3-Oxazolin-2-ly], [BH3260; 3-Oxazolin-4-ly], [BH3261; 2-Me-3-Oxazolin-4-ly], [B. BH3262; 5-Me-3-Oxazolin-4-ly], [BH 3263; 2-Me-2-Me-3-Oxazolin-4-ly], [BH3264; 5-Me-5-Me-3-Oxazolin- 4-ly, [BH3265; 2-Me-5-Me-3-Oxazolin-4-ly], [BH3266; 3-Oxazolin-5-ly], [BH3267; 2-Me-3-Oxazolin-5- ly], [BH3268; 4-Me-3-Oxazolin-5-ly], [BH3269; 5-Me-3-Oxazolin-5-ly], [BH3270; 2-Me-2-Me-3-Oxazolin- 5-ly] , [BH3271; 2-Me-4-Me-3-Oxazolin-5-ly], [BH3272; 2-Me-5-Me-3-Oxazolin-5-ly], [BH3273; 4-Me-5- Me-3-Oxazolin-5-ly, [BH3274; 2-Me-4-Me-5-Me-3-Oxazolin-5-ly], [BH3275; N-Me-4-Oxazolin-2-ly] , [BH3276; 2-Me-N-Me-4-Oxazolin-2-ly], [BH3277; 4-Me-N-Me-4-Oxazolin-2-ly], [BH3278; 5-Me-N- Me-4-Oxazolin-2-ly, [BH3279; 2-Me-5-Me-N-Me-4-Oxazolin-2-ly], [BH3280; 4-Me-5-Me-N-Me- 4-Oxazolin-2-ly, [BH3281; 2-Me-4-Me-5-Me-N-Me-4-Oxazolin-2-ly], [BH3282; 2-Me-4-Me-N- Me-4-Oxazolin-2-ly, [BH3283; N-Me-4-Oxazolin-4-ly], [BH3284; 2-Me-N-Me-4-Oxazolin-4-ly], [BH3285; 5-Me-N-Me-4-Oxazolin-4-ly], [BH3286; 2-Me-5-Me-N-Me-4-Oxazolin-4-ly], [BH3287; 2-Me-2- Me-5-Me-N-Me-4-Oxazolin-4-ly], [BH3288; N-Me-4-Oxazolin-5-ly], [BH3289; 2-Me-N-Me-4-Oxazolin- 5-ly, [BH3290; 5-Me-N-Me-4-Oxazolin-5-ly], [BH3291; 2-Me-5-Me-N-Me-4-Oxazolin-5-ly], [B. BH3292; 2-Me-2-Me-5-Me-N-Me-4-Oxazolin-5-ly], [BH3293; Oxazolidin-2-on-4-ly], [BH3294; 4-Me-Oxazolidin- 2-on-4-ly], [BH3295; 5-Me-Oxazolidin-2-on-4-ly], [BH3296; 4-Me-5-Me-Oxazolidin-2-on-4-ly], [B. BH 3 297; 5-Me-5-Me-Oxazolidin-2-on-4-ly], [BH 3 298; -Oxazolidin-2-on-5-ly], [BH3299; 4-Me-Oxazolidin-2-on-5-ly], [BH3300; 5-Me-Oxazolidin-2-on-5-ly],

[BH3301; 4-Me-5-Me-Oxazolidin-2-on-5-ly], [BH3302; 4-Me-4-Me-Oxazolidin-2-on-5-ly], [BH3303; N-Me -Oxazolidin-4-on-2-ly], [BH3304; 2-Me-N-Me-Oxazolidin-4-on-2-ly], [BH3305; 5-Me-N-Me-Oxazolidin-4-on -2-ly], [BH3306; 2-Me-5-Me-N-Me-Oxazolidin-4-on-2-ly], [BH3307; 2-Me-5-Me-5-Me-N-Me -Oxazolidin-4-on-2-ly], [BH3308; N-Me-Oxazolidin-4-on-5-ly], [BH3309; 2-Me-N-Me-Oxazolidin-4-on-5-ly ], [BH3310; 5-Me-N-Me-Oxazolidin-4-on-5-ly], [BH3311; 2-Me-5-Me-N-Me-O-oxazolidin-4-on-5-ly], [BH3312; 2-Me-2-Me-5-Me-N-Me-Oxazolidin-4-on-5-ly], [BH3313; N-Me-Oxazolidin-5-on-2-ly], [BH3314 2-Me-N-Me-Oxazolidin-5-on-2-ly], [BH3315; 4-Me-N-Me-Oxazolidin-5-on-2-ly], [BH3316; 2-Me-4 -Me-N-Me-Oxazolidin-5-on-2-ly], [BH3317; 2-Me-4-Me-4-Me-N-Me-Oxazolidin-5-on-2-ly], [BH3318 N-Me-Oxazolidin-5-on-4-ly], [BH3319; 2-Me-N-Me-Oxazolidin-5-on-4-ly], [BH3320; 4-Me-N-Me-Oxazolidin [5-on-4-ly], [BH3321; 2-Me-4-Me-N-Me-Oxazolidin-5-on-4-ly], [BH3322; 2-Me-2-Me-4-Me -N-Me-Oxazolidin-5-on-4-ly], [BH3323; 2-Thazolin-4-ly], [BH3324; 2-Me-2-Thazolin-4-ly], [BH3325; 4-Me -2-Thazolin-4 -ly, [BH3326; 5-Me-2-Thazolin-4-ly], [BH3327; 2-Me-4-Me-2-Thazolin-4-ly], [BH3328; 2-Me-5-Me -2-Thazolin-4-ly, [BH3329; 4-Me-5-Me-2-Thazolin-4-ly], [BH3330; 5-Me-5-Me-2-Thazolin-4-ly], [BH3331; 2-Me-4-Me-5-Me-2-Thazolin-5-ly], [BH3332; 2-Thazolin-5-ly], [BH3333; 2-Me-2-Thazolin-5-ly] ], [BH3334; 5-Me-2-Thazolin-5-ly], [BH3335; 4-Me-2-Thazolin-5-ly], [BH3336; 2-Me-5-Me-2-Thazolin-5] -ly, [BH3337; 2-Me-4-Me-2-Thazolin-5-ly], [BH3338; 5-Me-4-Me-2-Thazolin-5-ly], [BH3339; 4-Me -4-Me-2-Thazolin-5-ly], [BH3340; 2-Me-5-Me-4-Me-2-Thazolin-5-ly], [BH3341; 3-Thazolin-2-ly], [BH3342; 2-Me-3-Thazolin-2-ly], [BH3343; 4-Me-3-Thazolin-2-ly], [BH3344; 5-Me-3-Thazolin-2-ly], [BH3345] 2-Me-4-Me-3-Thazolin-2-ly], [BH3346; 2-Me-5-Me-3-Thazolin-2-ly], [BH3347; 4-Me-5-Me-3 -Thazolin-2-ly, [BH3348; 5-Me-5-Me-3-Thazolin-2-ly], [BH3349; 2-Me-4-Me-5-Me-3-Thazolin-2-ly ], [BH3350; 3-Thazolin-4-ly], [BH3351; 2-Me-3-Thazolin-4-ly], [BH3352; 5-Me-3-Thazolin-4-ly], [BH3353; -Me-2-Me-3-Thazolin-4-ly], [BH3354; 5-Me-5-Me-3-Thazolin-4-ly], [BH3355; 2-Me-5-Me-3-Thazolin -4-ly], [BH33 56; 3-Thazolin-5-ly, [BH3357; 2-Me-3-Thazolin-5-ly], [BH3358; 4-Me-3-Thazolin-5-ly], [BH3359; 5-Me- 3-Thazolin-5-ly, [BH3360; 2-Me-2-Me-3-Thazolin-5-ly], [BH3361; 2-Me-4-Me-3-Thazolin-5-ly], [B. BH3362; 2-Me-5-Me-3-Thazolin-5-ly], [BH3363; 4-Me-5-Me-3-Thazolin-5-ly], [BH3364; 2-Me-4-Me- 5-Me-3-Thazolin-5-ly], [BH3365; N-Me-4-Thazolin-2-ly], [BH3366; 2-Me-N-Me-4-Thazolin-2-ly], [B. BH 3367; 4-Me-N-Me-4-Thazolin-2-ly], [BH 3368; 5-Me-N-Me-4-Thazolin-2-ly], [BH 3369; 2-Me-5-Me- N-Me-4-Thazolin-2-ly, [BH3370; 4-Me-5-Me-N-Me-4-Thazolin-2-ly], [BH3371; 2-Py], [BH3372; Me-2-Py !, [BH3373; 4-Me-2-Py], [BH3374; 5-Me-2-Py], [BH3375; 6-Me-2-Py], [BH3376; 3-Me- 4-Me-2-Py, [BH3377; 3-Me-5-Me-2-Py], [BH 3378; 3-Me-6-Me-2-Py], [BH 3379; 4-Me-5- Me-2-Py !, [BH3380; 4-Me-6-Me-2-Py], [BH3381; 5-Me-6-Me-2-Py], [BH3382; 3-Me-4-Me- 5-Me-2-Py !, [BH3383; 3-Me-4-Me-6-Me-2-Py], [BH3384; 3-Me-5-Me-6-Me-2-Py], BH3385; 4-Me-5-Me-6-Me-2-Py], [BH3386; 3-F-4-Me-2-Py], [BH3387; 5-F-4-Me-2-Py] , [BH3388; 6-F-4-Me-2-Py], [BH3389; 3-F-5-Me-2-Py], [BH3390; 4-F-5-Me-2-Py], [BH3 388; BH3391; 6-F-5-Me-2-Py], [BH3392 3-F-6-Me-2-Py !, [BH3393; 4-F-6-Me-2-Py], [BH3394; 5-F-6-Me-2-Py], [BH3395; 3] -F-4-F-6-Me-2-Py], [BH3396; 3-F-5-F-6-Me-2-Py], [BH3397; 4-F-5-F-6-Me -2-Py !, [BH3398; 3-Cl-4-Me-2-Py], [BH3399; 5-Cl-4-Me-2-Py], [BH3400; 6-Cl-4-Me-2 -Py],

[BH3401; 3-Cl-5-Me-2-Py], [BH3402; 4-Cl-5-Me-2-Py], [BH3403; 6-Cl-5-Me-2-Py], [BH3404] 3-Cl-6-Me-2-Py !, [BH3405; 4-Cl-6-Me-2-Py], [BH3406; 5-Cl-6-Me-2-Py], [BH3407; -Cl-4-Cl-6-Me-2-Py], [BH3408; 3-Cl-5-Cl-6-Me-2-Py], [BH3409; 4-Cl-5-Cl-6-Me -2-Py !, [BH 3410; 3-Br-6-Me-2-Py], [BH 3411; 4-Br-6-Me-2-Py], [BH 3412; 5-Br-6-Me-2 -Py], [BH3413; 3-CN-6-Me-2-Py], [BH3414; 4-CN-6-Me-2-Py], [BH3415; 5-CN-6-Me-2-Py ], [BH3416; 3-OMe-6-Me-2-Py], [BH3417; 4-OMe-6-Me-2-Py], [BH3418; 5-OMe-6-Me-2-Py], [BH3419; 3-Et-6-Me-2-Py], [BH3420; 4-Et-6-Me-2-Py], [BH3421; 5-Et-6-Me-2-Py], [BH3422 3-Br-5-Me-2-Py !, [BH3423; 4-Br-5-Me-2-Py], [BH3424; 6-Br-5-Me-2-Py], [BH3425; -CN-5-Me-2-Py], [BH3426; 4-CN-5-Me-2-Py], [BH3427; 6-CN-5-Me-2-Py], [BH3428; 3-OMe -5-Me-2-Py, [BH3429; 4-OMe-5-Me-2-Py], [BH3430; 6-OMe-5-Me-2-Py], [BH3431; 3-Br-4 -Me-2-Py], [BH3432; 5-Br-4-Me-2-Py], [BH3433; 6-Br-4-Me-2-Py], [BH3434; 3-CN-4-Me -2-Py !, [BH3435; 5-CN-4-Me-2-Py], [BH3436; 6-CN-4-Me-2-Py], [BH3437; 3-OMe-4-Me-2 -Py], [BH3438; 5-OMe-4-Me-2-Py], [BH3439; 6-OMe-4-Me-2-Py], [BH3440; 3-Et-4-Me-2-Py ], [BH3441; 5-Et-4-M e-2-Py !, [BH3442; 6-Et-4-Me-2-Py], [BH3443; 3-Et-2-Py], [BH3444; 4-Et-2-Py], [BH3445; 5-Et-2-Py], [BH3446; 6-Et-2-Py], [BH 3447; 3-Et-4-Et-2-Py], [BH 3448; 3-Et-5-Et-2-] Py], [BH3449; 3-Et-6-Et-2-Py], [BH3450; 4-Et-5-Et-2-Py], [BH3451; 4-Et-6-Et-2-Py] , [BH3452; 5-Et-6-Et-2-Py], [BH3453; 3-F-4-Et-2-Py], [BH3454; 5-F-4-Et-2-Py], [BH3452; BH3455; 6-F-4-Et-2-Py], [BH3456; 3-F-5-Et-2-Py], [BH3457; 4-F-5-Et-2-Py], [BH3458; 6-F-5-Et-2-Py], [BH3459; 3-F-6-Et-2-Py], [BH 3460; 4-F-6-Et-2-Py], [BH3461; 5- F-6-Et-2-Py], [BH3462; 3-F-4-F-6-Et-2-Py], [BH3463; 3-F-5-F-6-Et-2-Py] , [BH 3464; 4-F-5-F-6-Et-2-Py], [BH 3465; 3-Cl-4-Et-2-Py], [BH 3466; 5-Cl-4-Et-2- Py], [BH3467; 6-Cl-4-Et-2-Py], [BH3468; 3-Cl-5-Et-2-Py], [BH3469; 4-Cl-5-Et-2-Py] , [BH3470; 6-Cl-5-Et-2-Py], [BH 3471; 3-Cl-6-Et-2-Py], [BH 3472; 4-Cl-6-Et-2-Py], [BH 3470; BH3473; 5-Cl-6-Et-2-Py], [BH3474; 3-Cl-4-Cl-6-Et-2-Py], [BH3475; 3-Cl-5-Cl-6-Et- 2-Py], [BH3476; 4-Cl-5-Cl-6-Et-2-Py], [BH3477; 3-Br-5-Et-2-Py], [BH3478; 4-Br-5- Et-2-Py, [BH3479; 6-Br-5-Et-2-Py], [BH3480; 3-CN-5-Et-2-Py], [BH3481; 4-CN-5-Et- 2-Py], [BH3482; 6-CN-5-Et-2-Py], [BH3483; 3-OMe -5-Et-2-Py], [BH3484; 4-OMe-5-Et-2-Py], [BH3485; 6-OMe-5-Et-2-Py], [BH3486; 3-Et-5 -Et-2-Py], [BH 3487; 4-Et-5-Et-2-Py], [BH 3488; 6-Et-5-Et-2-Py], [BH 3489; 3-Br-6-Et] -2-Py !, [BH3490; 4-Br-6-Et-2-Py], [BH3491; 5-Br-6-Et-2-Py], [BH3492; 3-CN-6-Et-2 -Py], [BH3493; 4-CN-6-Et-2-Py], [BH3494; 5-CN-6-Et-2-Py], [BH3495; 3-OMe-6-Et-2-Py ], [BH3496; 4-OMe-6-Et-2-Py], [BH3497; 5-OMe-6-Et-2-Py], [BH3498; 3-Pr-2-Py], [BH3499; 4] -Pr-2-Py], [BH3500; 5-Pr-2-Py],

[BH3501; 6-Pr-2-Py], [BH3502; 3-i-Pr-2-Py], [BH3503; 4-i-Pr-2-Py], [BH 3504; 5-i-Pr-2 -Py], [BH3505; 6-i-Pr-2-Py], [BH3506; 3-c-Pr-2-Py], [BH3507; 4-c-Pr-2-Py], [BH3508; -c-Pr-2-Py], [BH3509; 6-c-Pr-2-Py], [BH 3510; 3-F-4-c-Pr-2-Py], [BH 3511; 5-F-4 -c-Pr-2-Py], [BH 3512; 6-F-4-c-Pr-2-Py], [BH 3513; 3-F-5-c-Pr-2-Py], [BH 3514; -F-5-c-Pr-2-Py], [BH3515; 6-F-5-c-Pr-2-Py], [BH3516; 3-F-6-c-Pr-2-Py], [BH3517; 4-F-6-c-Pr-2-Py], [BH3518; 5-F-6-c-Pr-2-Py], [BH3519; 3,4-F2-6-c-Pr -2-Py !, [BH3520; 3,5-F2-6-c-Pr-2-Py], [BH3521; 4,5-F2-6-c-Pr-2-Py], [BH3522; 3 -Cl-4-c-Pr-2-Py], [BH3523; 5-Cl-4-c-Pr-2-Py], [BH3524; 6-Cl-4-c-Pr-2-Py], [BH3525; 3-Cl-5-c-Pr-2-Py], [BH3526; 4-Cl-5-c-Pr-2-Py], [BH3527; 6-Cl-5-c-Pr-2 -Py], [BH3528; 3-Cl-6-c-Pr-2-Py], [BH3529; 4-Cl-6-c-Pr-2-Py], [BH3530; 5-Cl-6-c -Pr-2-Py], [BH3531; 3-Cl-4-Cl-6-c-Pr-2-Py], [BH3532; 3-Cl-5-Cl-6-c-Pr-2-Py ], [BH3533; 4-Cl-5-Cl-6-c-Pr-2-Py], [BH3534; 3-F-2-Py], [BH3535; 4-F-2-Py], [BH3536] 5-F-2-Py !, [BH3537; 6-F-2-Py], [BH3538; 3-F-4-F-2-Py], [BH3539; 3-F-5-F-2] -Py], [BH3540; 3-F-6-F-2-Py], [BH3541; 4-F-5-F-2-Py], [BH3542; 4-F -6-F-2-Py !, [BH3543; 5-F-6-F-2-Py], [BH3544; 3-F-4-F-5-F-2-Py], [BH3545; 3] -F-4-F-6-F-2-Py], [BH3546; 3-F-5-F-6-F-2-Py], [BH3547; 4-F-5-F-6-F -2-Py], [BH3548; 3-Cl-2-Py], [BH3549; 4-Cl-2-Py], [BH3550; 5-Cl-2-Py], [BH3551; 6-Cl-2 -Py], [BH3552; 3-F-4-Cl-2-Py], [BH3553; 5-F-4-Cl-2-Py], [BH3554; 6-F-4-Cl-2-Py] ], [BH3555; 3-F-5-Cl-2-Py], [BH3556; 4-F-5-Cl-2-Py], [BH3557; 6-F-5-Cl-2-Py], [BH3558; 3-F-6-Cl-2-Py], [BH3559; 4-F-6-Cl-2-Py], [BH3560; 5-F-6-Cl-2-Py], [BH3561] 3-F-4-F-6-Cl-2-Py !, [BH3562; 3-F-5-F-6-Cl-2-Py], [BH3563; 4-F-5-F-6] -Cl-2-Py], [BH3564; 3-Cl-4-Cl-2-Py], [BH3565; 3-Cl-5-Cl-2-Py], [BH3566; 3-Cl-6-Cl -2-Py], [BH3567; 4-Cl-5-Cl-2-Py], [BH3568; 4-Cl-6-Cl-2-Py], [BH 3569; 5-Cl-6-Cl-2 -Py], [BH3570; 3-Cl-4-Cl-5-Cl-2-Py], [BH3571; 3-Cl-4-Cl-6-Cl-2-Py], [BH3572; 3-Cl -5-Cl-6-Cl-2-Py !, [BH3573; 4-Cl-5-Cl-6-Cl-2-Py], [BH3574; 3-Br-2-Py], [BH3575; 4] -Br-2-Py], [BH3576; 5-Br-2-Py], [BH 3577; 6-Br-2-Py], [BH 3578; 3-CN-2-Py], [BH 3579; 4-CN -2-Py], [BH3 580; 5-CN-2-Py], [BH3581; 6-CN-2-Py], [BH3582; 3-F-4-CN-2-Py], [BH3583; -F-4-CN-2-Py], [BH3584; 6-F-4-CN-2-Py], [BH 3585; 3-F-5-CN-2 -Py], [BH3586; 4-F-5-CN-2-Py], [BH3587; 6-F-5-CN-2-Py], [BH3588; 3-F-6-CN-2-Py ], [BH3589; 4-F-6-CN-2-Py], [BH3590; 5-F-6-CN-2-Py], [BH3591; 3-F-4-F-6-CN-2] -Py], [BH3592; 3-F-5-F-6-CN-2-Py], [BH3593; 4-F-5-F-6-CN-2-Py], [BH3594; 3-Cl] -4-CN-2-Py !, [BH3595; 5-Cl-4-CN-2-Py], [BH3596; 6-Cl-4-CN-2-Py], [BH3597; 3-Cl-5 -CN-2-Py], [BH3598; 4-Cl-5-CN-2-Py], [BH3599; 6-Cl-5-CN-2-Py], [BH3600; 3-Cl-6-CN -2-Py],

[BH3601; 4-Cl-6-CN-2-Py], [BH3602; 5-Cl-6-CN-2-Py], [BH3603; 3-Cl-4-Cl-6-CN-2-Py ], [BH3604; 3-Cl-5-Cl-6-CN-2-Py], [BH3605; 4-Cl-5-Cl-6-CN-2-Py], [BH3606; 3-OMe-2] -Py], [BH3607; 4-OMe-2-Py], [BH3608; 5-OMe-2-Py], [BH3609; 6-OMe-2-Py], [BH3610; 3-OMe-4-OMe -2-Py !, [BH3611; 3-OMe-5-OMe-2-Py], [BH3612; 3-OMe-6-OMe-2-Py], [BH3613; 4-OMe-5-OMe-2 4-Pe], [BH3614; 4-OMe-6-OMe-2-Py], [BH3615; 5-OMe-6-OMe-2-Py], [BH3616; 3-F-4-OMe-2-Py] ], [BH3617; 5-F-4-OMe-2-Py], [BH3618; 6-F-4-OMe-2-Py], [BH3619; 3-F-5-OMe-2-Py], [BH3620; 4-F-5-OMe-2-Py], [BH3621; 6-F-5-OMe-2-Py], [BH3622; 3-F-6-OMe-2-Py], [BH3623] 4-F-6-OMe-2-Py !, [BH3624; 5-F-6-OMe-2-Py], [BH3625; 3,4-F2-6-OMe-2-Py], [BH3626] 3,5-F2-6-OMe-2-Py !, [BH3627; 4,5-F2-6-OMe-2-Py], [BH3628; 3-Cl-4-OMe-2-Py], [BH3629; 5-Cl-4-OMe-2-Py], [BH3630; 6-Cl-4-OMe-2-Py], [BH3631; 3-Cl-5-OMe-2-Py], [BH3632 4-Cl-5-OMe-2-Py !, [BH3633; 6-Cl-5-OMe-2-Py], [BH3634; 3-Cl-6-OMe-2-Py], [BH3635; 4] -Cl-6-OMe-2-Py], [BH3636; 5-Cl-6-OMe-2-Py], [BH3637; 3-Cl-4-Cl-6-OMe-2-Py], [BH3638] 3-Cl-5-Cl-6-OMe-2-Py !, [BH3639; 4-Cl-5-Cl-6-OMe-2-Py], [BH3640; 3-O Et-2-Py], [ BH3641; 4-OEt-2-Py], [BH3642; 5-OEt-2-Py], [BH3643; 6-OEt-2-Py], [BH3644; 3-CF 3 -2-Py], [BH3645; 4-CF 3 -2-Py], [BH3646; 5-CF 3 -2-Py], [BH3647; 6-CF 3 -2-Py], [BH3648; 3- _{F-4-CF 3 -2-} Py], [BH3649; 5-F-4-CF 3 -2-Py], [BH3650; 6-F-4-CF 3 -2-Py], [BH3651; 3 _{-F-5-CF 3 -2-} Py], [BH3652; 4-F-5-CF 3 -2-Py], [BH3653; 6-F-5-CF 3 -2-Py], [BH3654; _{3-F-6-CF 3} -2-Py], [BH3655; 4-F-6-CF 3 -2-Py], [BH3656; 5-F-6-CF 3 -2-Py], [BH3657 ; 3-F-4-F -6-CF 3 -2-Py], [BH3658; 3-F-5-F-6-CF 3 -2-Py], [BH3659; 4-F-5-F -6-CF ₃ -2-Py !, [BH 3660; 3-Cl -4-CF ₃ -2-Py], [BH 366 1; 5-Cl -4-CF ₃ -2-Py], [BH 366 2; _{Cl-4-CF 3 -2-} Py], [BH3663; 3-Cl-5-CF 3 -2-Py], [BH3664; 4-Cl-5-CF 3 -2-Py], [BH3665; 6 _{-Cl-5-CF 3 -2-} Py], [BH3666; 3-Cl-6-CF 3 -2-Py], [BH3667; 4-Cl-6-CF 3 -2-Py], [BH3668; _{5-Cl-6-CF 3} -2-Py], [BH3669; 3-Cl-4-Cl-6-CF 3 -2-Py], [BH3670; 3-Cl-5-Cl-6-CF 3 -2-Py !, [BH 3671; 4-Cl-5-Cl-6-CF ₃ -2-Py], [BH 3672; 3-amino-2-Py], [BH 3673; 4-amino-2-Py] , [BH3674; 5-amino-2-Py], [BH3675; 6-amino-2-Py], [BH3676; 3-N, N-dimethylamino-2-Py], [BH 3677; 4-N, N- dimethylamino-2-Py], [BH3678; 5-N, N-dimethylam ino-2-Py !, [BH3679; 6-N, N-dimethylamino-2-Py], [BH3680; 3-SMe-2-Py], [BH3681; 4-SMe-2-Py], [BH3682; 5-SMe-2-Py, [BH3683; 6-SMe-2-Py], [BH3684; -3-Py], [BH3685; 2-Me-3-Py], [BH3686; 4-Me-3 -Py], [BH3687; 5-Me-3-Py], [BH3688; 6-Me-3-Py], [BH3689; 2-Me-4-Me-3-Py], [BH3690; 2-Me -5-Me-3-Py !, [BH3691; 2-Me-6-Me-3-Py], [BH3692; 4-Me-5-Me-3-Py], [BH3693; 4-Me-6 -Me-3-Py, [BH3694; 5-Me-6-Me-3-Py], [BH3695; 2-Me-4-Me-5-Me-3-Py], [BH3696; 2-Me -4-Me-6-Me-3-Py, [BH 3697; 2-Me-5-Me-6-Me-3-Py], [BH 3698; 4-Me-5-Me-6-Me-3 -Py], [BH3699; 2-F-4-Me-3-Py], [BH3700; 5-F-4-Me-3-Py],

[BH3701; 6-F-4-Me-3-Py], [BH3702; 2-F-5-Me-3-Py], [BH3703; 4-F-5-Me-3-Py], [BH3704] 6-F-5-Me-3-Py !, [BH3705; 2-F-6-Me-3-Py], [BH3706; 4-F-6-Me-3-Py], [BH3707; -F-6-Me-3-Py], [BH3708; 2-F-4-F-6-Me-3-Py], [BH3709; 2-F-5-F-6-Me-3-Py ], [BH3710; 4-F-5-F-6-Me-3-Py], [BH3711; 2-Cl-4-Me-3-Py], [BH3712; 5-Cl-4-Me-3] -Py], [BH3713; 6-Cl-4-Me-3-Py], [BH3714; 2-Cl-5-Me-3-Py], [BH3715; 4-Cl-5-Me-3-Py ], [BH3716; 6-Cl-5-Me-3-Py], [BH3717; 2-Cl-6-Me-3-Py], [BH3718; 4-Cl-6-Me-3-Py], [BH3719; 5-Cl-6-Me-3-Py], [BH3720; 2-Cl-4-Cl-6-Me-3-Py], [BH3721; 2-Cl-5-Cl-6-Me -3-Py !, [BH3722; 4-Cl-5-Cl-6-Me-3-Py], [BH3723; 2-Br-6-Me-3-Py], [BH3724; 4-Br-6 -Me-3-Py, [BH3725; 5-Br-6-Me-3-Py], [BH3726; 2-CN-6-Me-3-Py], [BH3727; 4-CN-6-Me -3-Py !, [BH3728; 5-CN-6-Me-3-Py], [BH3729; 2-OMe-6-Me-3-Py], [BH3730; 4-OMe-6-Me-3 -Py], [BH3731; 5-OMe-6-Me-3-Py], [BH3732; 2-Et-6-Me-3-Py], [BH3733; 4-Et-6-Me-3-Py ], [BH3734; 5-Et-6-Me-3-Py], [BH3735; 3-Br-5-Me-2-Py], [BH3736; 4-Br-5-Me-2-Py], [BH3737; 6-Br-5-Me-2-Py], [BH3738; 3-CN-5-Me-2-Py], [BH3739; 4-CN-5-Me-2-Py], [BH3740] 6-CN-5-Me-2-Py], [BH3741; 3-OMe-5-Me-2 -Py], [BH3742; 4-OMe-5-Me-2-Py], [BH3743; 6-OMe-5-Me-2-Py], [BH3744; 3-Br-4-Me-2-Py ], [BH3745; 5-Br-4-Me-2-Py], [BH3746; 6-Br-4-Me-2-Py], [BH3747; 3-CN-4-Me-2-Py], [BH3748; 5-CN-4-Me-2-Py], [BH3749; 6-CN-4-Me-2-Py], [BH3750; 3-OMe-4-Me-2-Py], [BH3751] 5-OMe-4-Me-2-Py !, [BH3752; 6-OMe-4-Me-2-Py], [BH3753; 3-Et-4-Me-2-Py], [BH3754; -Et-4-Me-2-Py], [BH3755; 6-Et-4-Me-2-Py], [BH3756; 2-Et-3-Py], [BH3757; 4-Et-3-Py ], [BH 3758; 5-Et-3-Py], [BH 3759; 6-Et-3-Py], [BH 3760; 2-Et-4-Et-3-Py], [BH3761; -Et-3-Py], [BH3762; 2-Et-6-Et-3-Py], [BH3763; 4-Et-5-Et-3-Py], [BH3764; 4-Et-6-Et -3-Py, [BH3765; 5-Et-6-Et-3-Py], [BH3766; 2-F-4-Et-3-Py], [BH3767; 5-F-4-Et-3 -Py], [BH3768; 6-F-4-Et-3-Py], [BH3769; 2-F-5-Et-3-Py], [BH3770; 4-F-5-Et-3-Py ], [BH3771; 6-F-5-Et-3-Py], [BH3772; 2-F-6-Et-3-Py], [BH3773; 4-F-6-Et-3-Py], [BH3774; 5-F-6-Et-3-Py], [BH3775; 2-F-4-F-6-Et-3-Py], [BH3776; 2-F-5-F-6-Et] -3-Py, [BH3777; 4-F-5-F-6-Et-3-Py], [BH 3778; 2-Cl-4-Et-3-Py], [BH3779; 5-Cl-4 -Et-3-Py], [BH3780; 6-Cl-4-Et-3-Py], [BH 3781; 2-Cl-5-Et-3-Py], [BH 3782; 4-Cl-5-Et -3-Py, [BH 3783; 6-Cl-5-Et-3-Py], [B H3784; 2-Cl-6-Et-3-Py], [BH3785; 4-Cl-6-Et-3-Py], [BH3786; 5-Cl-6-Et-3-Py], [BH3787; 2-Cl-4-Cl-6-Et-3-Py], [BH3788; 2-Cl-5-Cl-6-Et-3-Py], [BH3789; 4-Cl-5-Cl-6- Et-3-Py, [BH 3790; 2-Br-5-Et-3-Py], [BH 3791; 4-Br-5-Et-3-Py], [BH 3792; 6-Br-5-Et- 3-Py], [BH3793; 2-CN-5-Et-3-Py], [BH3794; 4-CN-5-Et-3-Py], [BH3795; 6-CN-5-Et-3- 3 Py], [BH 3796; 2-OMe-5-Et-3-Py], [BH 3797; 4-OMe-5-Et-3-Py], [BH 3798; 6-OMe-5-Et-3-Py] , [BH3799; 2-Et-5-Et-3-Py], [BH3800; 4-Et-5-Et-3-Py],

[BH3801; 6-Et-5-Et-3-Py], [BH3802; 2-Br-6-Et-3-Py], [BH3803; 4-Br-6-Et-3-Py], [BH3804] 5-Br-6-Et-3-Py !, [BH3805; 2-CN-6-Et-3-Py], [BH3806; 4-CN-6-Et-3-Py], [BH3807; -CN-6-Et-3-Py], [BH3808; 2-OMe-6-Et-3-Py], [BH3809; 4-OMe-6-Et-3-Py], [BH3810; 5-OMe -6-Et-3-Py], [BH3811; 2-Pr-3-Py], [BH3812; 4-Pr-3-Py], [BH3813; 5-Pr-3-Py], [BH3814; -Pr-3-Py], [BH3815; 2-i-Pr-3-Py], [BH3816; 4-i-Pr-3-Py], [BH3817; 5-i-Pr-3-Py], [BH3818; 6-i-Pr-3-Py], [BH3819; 2-c-Pr-3-Py], [BH3820; 4-c-Pr-3-Py], [BH 3821; 5-c-Pr -3-Py, [BH3822; 6-c-Pr-3-Py], [BH3823; 2-F-4-c-Pr-3-Py], [BH3824; 5-F-4-c-Pr -3-Py, [BH3825; 6-F-4-c-Pr-3-Py], [BH3826; 2-F-5-c-Pr-3-Py], [BH3827; 4-F-5 -c-Pr-3-Py], [BH3828; 6-F-5-c-Pr-3-Py], [BH3829; 2-F-6-c-Pr-3-Py], [BH3830; 4 -F-6-c-Pr-3-Py], [BH3831; 5-F-6-c-Pr-3-Py], [BH3832; 2,4-F2-6-c-Pr-3-Py ], [BH3833; 2,5-F2-6-c-Pr-3-Py], [BH3834; 4,5-F2-6-c-Pr-3-Py], [BH3835; 2-Cl-4] -c-Pr-3-Py], [BH3836; 5-Cl-4-c-Pr-3-Py], [BH3837; 6-Cl-4-c-Pr-3-Py], [BH3838; -Cl-5-c-Pr-3-Py], [BH3839; 4-Cl-5-c-Pr-3-Py], [BH3840; 6-Cl-5-c-Pr-3-Py], [BH3841; 2-Cl-6-c-Pr-3-Py], [BH3842; 4-Cl-6-c -Pr-3-Py], [BH3843; 5-Cl-6-c-Pr-3-Py], [BH3844; 2-Cl-4-Cl-6-c-Pr-3-Py], [BH3845] 2-Cl-5-Cl-6-c-Pr-3-Py !, [BH3846; 4-Cl-5-Cl-6-c-Pr-3-Py], [BH3847; 2-F-3 4-Py !, [BH3848; 4-F-3-Py], [BH3849; 5-F-3-Py], [BH3850; 6-F-3-Py], [BH3851; 2-F-4-F -3-Py, [BH3852; 2-F-5-F-3-Py], [BH3853; 2-F-6-F-3-Py], [BH3854; 4-F-5-F-3 -Py], [BH3855; 4-F-6-F-3-Py], [BH3856; 5-F-6-F-3-Py], [BH3857; 2-F-4-F-5-F -3-Py, [BH3858; 2-F-4-F-6-F-3-Py], [BH3859; 2-F-5-F-6-F-3-Py], [BH3860; -F-5-F-6-F-3-Py], [BH3861; 2-Cl-3-Py], [BH3862; 4-Cl-3-Py], [BH3863; 5-Cl-3-Py ], [BH3864; 6-Cl-3-Py], [BH3865; 2-F-4-Cl-3-Py], [BH3866; 5-F-4-Cl-3-Py], [BH3867; 6] -F-4-Cl-3-Py], [BH3868; 2-F-5-Cl-3-Py], [BH3869; 4-F-5-Cl-3-Py], [BH3870; 6-F -5-Cl-3-Py !, [BH 3871; 2-F-6-Cl-3-Py], [BH 3872; 4-F-6-Cl-3-Py], [BH 3873; 5-F-6 -Cl-3-Py], [BH3874; 2-F-4-F-6-Cl-3-Py], [BH3875; 2-F-5-F-6-Cl-3-Py], [BH3876] 4-F-5-F-6-Cl-3-Py !, [BH3877; 2-Cl-4-Cl-3-Py], [BH3878; 2-Cl-5-Cl-3-Py], [BH3879; 2-Cl-6-Cl-3-Py], [BH 3880; 4-Cl-5-Cl-3-Py], [BH3881; 4-Cl-6-Cl-3-Py], [BH3882 5-Cl-6-Cl-3-Py !, [BH 3883; 2-Cl-4-Cl-5-Cl-3-Py], [BH 3884; 2-Cl-4-Cl-6-Cl-3 -P y], [BH3885; 2-Cl-5-Cl-6-Cl-3-Py], [BH 3886; 4-Cl-5-Cl-6-Cl-3-Py], [BH 3887; 2-Br- 3-Py], [BH3888; 4-Br-3-Py], [BH3889; 5-Br-3-Py], [BH 3890; 6-Br-3-Py], [BH3891; 2-CN-3- Py], [BH3892; 4-CN-3-Py], [BH3893; 5-CN-3-Py], [BH3894; 6-CN-3-Py], [BH3895; 2-F-4-CN- 3-Py], [BH3896; 5-F-4-CN-3-Py], [BH3897; 6-F-4-CN-3-Py], [BH3898; 2-F-5-CN-3- Py], [BH3899; 4-F-5-CN-3-Py], [BH3900; 6-F-5-CN-3-Py],

[BH3901; 2-F-6-CN-3-Py], [BH3902; 4-F-6-CN-3-Py], [BH3903; 5-F-6-CN-3-Py], [BH3904] 2-F-4-F-6-CN-3-Py !, [BH3905; 2-F-5-F-6-CN-3-Py], [BH3906; 4-F-5-F-6] -CN-3-Py, [BH3907; 2-Cl-4-CN-3-Py], [BH3908; 5-Cl-4-CN-3-Py], [BH3909; 6-Cl-4-CN -3-Py, [BH3910; 2-Cl-5-CN-3-Py], [BH3911; 4-Cl-5-CN-3-Py], [BH3912; 6-Cl-5-CN-3 -Py], [BH3913; 2-Cl-6-CN-3-Py], [BH3914; 4-Cl-6-CN-3-Py], [BH3915; 5-Cl-6-CN-3-Py ], [BH3916; 2-Cl-4-Cl-6-CN-3-Py], [BH 3917; 2-Cl-5-Cl-6-CN-3-Py], [BH 3918; 4-Cl-5] -Cl-6-CN-3-Py], [BH3919; 2-OMe-3-Py], [BH3920; 4-OMe-3-Py], [BH3921; 5-OMe-3-Py], [BH3922] 6-OMe-3-Py !, [BH3923; 2-OMe-4-OMe-3-Py], [BH3924; 2-OMe-5-OMe-3-Py], [BH3925; 2-OMe-6; 4-OMe-3-Py !, [BH3926; 4-OMe-5-OMe-3-Py], [BH3927; 4-OMe-6-OMe-3-Py], [BH3928; 5-OMe-6-OMe] -3-Py !, [BH3929; 2-F-4-OMe-3-Py], [BH3930; 5-F-4-OMe-3-Py], [BH3931; 6-F-4-OMe-3 -Py], [BH3932; 2-F-5-OMe-3-Py], [BH3933; 4-F-5-OMe-3-Py], [BH3934; 6-F-5-OMe-3-Py ], [BH3935; 2-F-6-OMe-3-Py], [BH3936; 4-F-6-OMe-3-Py], [BH3937; 5-F-6-OMe-3-Py], [BH 3938; 2-F-4-F-6-OMe-3-Py], [BH 3939; 2-F-5-F-6-OMe-3-Py], [BH3940; 4-F-5-F -6-OMe-3-Py], [BH 3941; 2-C l-4-OMe-3-Py !, [BH3942; 5-Cl-4-OMe-3-Py], [BH3943; 6-Cl-4-OMe-3-Py], [BH3944; 2-Cl- 5-OMe-3-Py, [BH3945; 4-Cl-5-OMe-3-Py], [BH3946; 6-Cl-5-OMe-3-Py], [BH3947; 2-Cl-6- OMe-3-Py !, [BH 3948; 4-Cl-6-OMe-3-Py], [BH 3949; 5-Cl-6-OMe-3-Py], [BH 3950; 2-Cl-4-Cl- 6-OMe-3-Py], [BH 3951; 2-Cl-5-Cl-6-OMe-3-Py], [BH 3952; 4-Cl-5-Cl-6-OMe-3-Py], [6 BH3953; 2-OEt-3-Py !, [BH3954; 4-OEt-3-Py], [BH3955; 5-OEt-3-Py], [BH3956; 6-OEt-3-Py], [BH3957; _{2-CF 3 -3-Py]} , [BH3958; 4-CF 3 -3-Py], [BH3959; 5-CF 3 -3-Py], [BH3960; 6-CF 3 -3-Py], [ BH3961; 2-F-4- CF 3 -3-Py], [BH3962; 5-F-4-CF 3 -3-Py], [BH3963; 6-F-4-CF 3 -3-Py], [BH3964; 2-F-5 -CF 3 -3-Py], [BH3965; 4-F-5-CF 3 -3-Py], [BH3966; 6-F-5-CF 3 -3-Py] , [BH3967; 2-F- 6-CF 3 -3-Py], [BH3968; 4-F-6-CF 3 -3-Py], [BH3969; 5-F-6-CF 3 -3-Py ], [BH3970; 2-F -4-F-6-CF 3 -3-Py], [BH3971; 2-F-5-F-6-CF 3 -3-Py], [BH3972; 4-F _{-5-F-6-CF 3} -3-Py], [BH3973; 2-Cl-4-CF 3 -3-Py], [BH3974; 5-Cl-4-CF 3 -3-Py], [ BH3975; 6-Cl-4- CF 3 -3-Py], [BH3976; 2-Cl-5-CF 3 -3-Py], [BH3977; 4-Cl-5-CF 3 -3-Py], [BH3978; 6-Cl-5 -CF 3 -3-Py], [BH3979; 2-Cl-6-CF 3 -3-Py], [BH3980; 4-Cl-6- _{CF 3 -3-Py], [} BH3981; 5-Cl-6-CF 3 -3-Py], [BH3982; 2-Cl-4-Cl-6-CF 3 -3-Py], [BH3983; 2 -Cl-5-Cl-6- CF 3 -3-Py], [BH3984; 4-Cl-5-Cl-6-CF 3 -3-Py], [BH3985; 2-amino-3-Py], [BH3986; 4-amino-3-Py], [BH 3987; 5-amino-3-Py], [BH 3988; 6-amino-3-Py], [BH 3989; 2-N, N-dimethylamino-3-Py ], [BH 3 990; 4-N, N-dimethylamino-3-Py], [BH 399 1; 5-N, N-dimethylamino-3-Py], [BH 399 2; 6-N, N-dimethylamino 3- Py], [BH3993; 2-SMe-3-Py], [BH3994; 4-SMe-3-Py], [BH3995; 5-SMe-3-Py], [BH3996; 6-SMe-3-Py], [BH3997] -2-Pyrimidin !, [BH 3998; 4-Me-2-Pyrimidine], [BH 3 999; 5-Me-2-Pyrimidin], [BH 4000; 4-Me-5-Me-2-Pyrimidine],

[BH4001; 4-Me-6-Me-2-Pyrimidin], [BH4002; 4-Me-5-Me-6-Me-2-Pyrimidin], [BH4003; 5-F-4-Me-2-Pyrimidine] ], [BH4004; 6-F-4-Me-2-pyrimidin], [BH4005; 5-F-6-F-4-Me-2-pyrimidin], [BH4006; 4-F-5-Me-2] -Pyrimidin], [BH 4007; 4-F-6-F-5-Me-2-Pyrimidin], [BH 4008; 6-F-4-Me-5-Me-2-Pyrimidine], [BH 4009; 5-F -4-Me-6-Me-2-Pyrimidin !, [BH 4010; 5-Cl-4-Me-2-Pyrimidin], [BH 4011; 6-Cl-4-Me-2-Pyrimidin], [BH 4012; -Cl-6-Cl-4-Me-2-Pyrimidin], [BH4013; 4-Cl-5-Me-2-Pyrimidin], [BH4014; 4-Cl-6-Cl-5-Me-2-Pyrimidine ], [BH4015; 6-Cl-4-Me-5-Me-2-Pyrimidin], [BH4016; 5-Cl-4-Me-6-Me-2-Pyrimidin], [BH4017; 5-Br-4] -Me-2-Pyrimidin], [BH 4018; 6-Br-4-Me-2-Pyrimidin], [BH 4019; 5-Br-6-Br-4-Me-2-Pyrimidine], [BH 4020; 4-Br -5-Me-2-Pyrimidin], [BH4021; 4-Br-6-Br-5-Me-2-Pyrimidin], [BH4022; 6-Br-4-Me-5-Me-2-Pyrimidine], [BH4023; 5-Br-4-Me-6-Me-2-Pyrimidin], [BH 4024; 4-F-2-Pyrimidin], [BH 4025; 5-F-2-Pyrimidin], [BH 4026; 4-F -5-F-2-Pyrimidin], [BH4027; 4-F-6-F-2-Pyrimidin], [BH4028; 4-F-5-F-6-F-2-Pyrimidine], [BH4029; -Cl-4-F-2-Pyrimidin], [BH4030; 6-Cl-4-F-2-Pyrimidin], [BH4031; 5-Cl-6-Cl-4-F-2-pyrimidin], [BH4032; 4-Cl-5-F-2-pyrimidin], [BH4033; 4-Cl-6-Cl-5-F -2-Pyrimidin !, [BH4034; 6-Cl-4-F-5-F-2-Pyrimidin], [BH4035; 5-Cl-4-F-6-F-2-Pyrimidine], [BH 4036; 4 -Et-2-Pyrimidin], [BH 4037; 5-Et-2-Pyrimidin], [BH 4038; 4-Et-5-Et-2-Pyrimidin], [BH 4039; 4-Et-6-Et-2-Pyrimidine ], [BH4040; 4-Et-5-Et-6-Me-2-Pyrimidin], [BH4041; 5-Cl-4-Et-2-Pyrimidin], [BH4042; 6-Cl-4-Et-2] -Pyrimidin], [BH 4043; 5-Cl-6-Cl-4-Et-2-Pyrimidin], [BH 4044; 4-Cl-5-Et-2-Pyrimidine], [BH 4045; 4-Cl-6-Cl -5-Et-2-Pyrimidin !, [BH 4046; 5-F-4-Et-2-Pyrimidin], [BH 4047; 6-F-4-Et-2-Pyrimidine], [BH 4048; 5-F-6 -F-4-Et-2-Pyrimidin], [BH 4049; 4-F-5-Et-2-Pyrimidin], [BH 4050; 4-OMe-2-pyrimidin !, [BH4052; 5-OMe-2-pyrimidin], [BH4053; 4-OMe-5-OMe-2-pyrimidin], [BH4054; 4-OMe-6-OMe-2 -Pyrimidin], [BH 4055; 5-Cl-4-OMe-2-Pyrimidin], [BH 4056; 6-Cl-4-OMe-2-Pyrimidine], [BH 4057; 5-Cl-6-Cl-4-OMe -2-Pyrimidin !, [BH 4058; 4-Cl-5-OMe-2-Pyrimidin], [BH 4059; 4-Cl-6-Cl-5-OMe-2-Pyrimidine], [BH 4060; 5-F-4 -OMe-2-Pyrimidin], [BH4061; 6-F-4-OMe-2-pyrimidin], [BH4062; 5-F-6-F-4-OMe-2-pyrimidin], [BH4063; 4-F-5-OMe-2-pyrimidin], BH4064; 4-F-6-F-5-OMe-2-pyrimidin], [BH4065; 4-Pr-2-pyrimidin], [BH4066; 5-Pr-2-pyrimidin], [BH4067; 4-SMe- 2-Pyrimidin], [BH4068; 5-SMe-2-Pyrimidin], [BH 4069; Ph], [BH 4070; 2-Me-Ph], [BH4071; 3-Me-Ph], [BH4072; 4-Me- Ph], [BH4073; 2-Me-3-Me-Ph], [BH4074; 2-Me-4-Me-Ph], [BH4075; 2-Me-5-Me-Ph], [BH4076; Me-6-Me-Ph !, [BH4077; 3-Me-4-Me-Ph], [BH4078; 3-Me-5-Me-Ph], [BH4079; 2-Me-3-Me-4- 4 Me-Ph !, [BH4080; 2-Me-3-Me-5-Me-Ph], [BH4081; 2-Me-3-Me-6-Me-Ph], [BH4082; 2-Me-4- Me-5-Me-Ph !, [BH4083; 2-Me-4-Me-6-Me-Ph], [BH4084; 3-Me-4-Me-5-Me-Ph], [BH4085; Me-3-Me-4-Me-5-Me-Ph !, [BH4086; 2-Me-3-Me-4-Me-6-Me-Ph], [BH4087; 2-Me-3-Me- 5-Me-6-Me-Ph !, [BH4088; 2-F-4-Me-Ph], [BH4089; 3-F-4-Me-Ph], [BH4090; 5-F-4-Me- Ph], [BH4091; 2-F-5-Me-Ph], [BH4092; 3-F-5-Me-Ph], [BH4093; 4-F-5-Me-Ph], [BH4094; 6- F-5-Me-Ph !, [BH4095; 2-F-6-Me-Ph], [BH4096; 3-F-6-Me-Ph], [BH4097; 4-F-6-Me-Ph] , [BH4098; 5-F-6-Me-Ph], [BH4099; 2-F-3-F-6-Me-Ph], [BH4100; 2-F-4-F-6-Me-Ph] ,

[BH4101; 2-F-5-F-6-Me-Ph], [BH4102; 3-F-4-F-6-Me-Ph], [BH4103; 3-F-5-F-6-Me -Ph !, [BH4104; 4-F-5-F-6-Me-Ph], [BH4105; 2-Cl-4-Me-Ph], [BH4106; 3-Cl-4-Me-Ph], [BH4107; 5-Cl-4-Me-Ph], [BH4108; 6-Cl-4-Me-Ph], [BH4109; 2-Cl-5-Me-Ph], [BH4110; 3-Cl-5 -Me-Ph], [BH4111; 4-Cl-5-Me-Ph], [BH4112; 6-Cl-5-Me-Ph], [BH4113; 2-Cl-6-Me-Ph], [BH4114] 3-Cl-6-Me-Ph !, [BH4115; 4-Cl-6-Me-Ph], [BH4116; 5-Cl-6-Me-Ph], [BH4117; 2-Cl-3-Cl. -6-Me-Ph !, [BH4118; 2-Cl-4-Cl-6-Me-Ph], [BH4119; 2-Cl-5-Cl-6-Me-Ph], [BH4120; 2-Cl -6-Cl-6-Me-Ph !, [BH4121; 3-Cl-4-Cl-6-Me-Ph], [BH4122; 3-Cl-5-Cl-6-Me-Ph], [BH4123] 4-Cl-5-Cl-6-Me-Ph !, [BH4124; 2-Br-6-Me-Ph], [BH4125; 3-Br-6-Me-Ph], [BH4126; 4-Br. -6-Me-Ph !, [BH4127; 5-Br-6-Me-Ph], [BH4128; 2-CN-6-Me-Ph], [BH4129; 3-CN-6-Me-Ph], [BH4130; 4-CN-6-Me-Ph], [BH4131; 5-CN-6-Me-Ph], [BH4132; 2-OMe-6-Me-Ph], [BH4133; 3-OMe-6 -Me-Ph], [BH4134; 4-OMe-6-Me-Ph], [BH4135; 5-OMe-6-Me-Ph], [BH4136; 2-Et-6-Me-Ph], [BH4137 3-Et-6-Me-Ph !, [BH4138; 4-Et-6-Me-Ph], [BH4139; 5-Et-6-Me-Ph], [BH4140; 2-Br-5-Me -Ph], [BH4141; 3-Br-5-Me-Ph], [BH4142; 4-Br-5-Me-Ph], [BH4143; 6-Br-5-Me-Ph], [BH 4144; 2-CN-5-Me-Ph], [BH4145; 3-CN-5-Me-Ph], [BH4146; 4-CN-5-Me-Ph], [BH4147; 6-CN-5- Me-Ph !, [BH4148; 2-OMe-5-Me-Ph], [BH4149; 3-OMe-5-Me-Ph], [BH4150; 4-OMe-5-Me-Ph], [BH4151; 6-OMe-5-Me-Ph !, [BH4152; 2-Br-4-Me-Ph], [BH4153; 3-Br-4-Me-Ph], [BH4154; 5-Br-4-Me- Ph], [BH4155; 6-Br-4-Me-Ph], [BH4156; 2-CN-4-Me-Ph], [BH4157; 3-CN-4-Me-Ph], [BH4158; CN-4-Me-Ph !, [BH4159; 6-CN-4-Me-Ph], [BH4160; 2-OMe-4-Me-Ph], [BH4161; 3-OMe-4-Me-Ph] , [BH4162; 5-OMe-4-Me-Ph], [BH4163; 6-OMe-4-Me-Ph], [BH4164; 2-Et-4-Me-Ph], [BH4165; 3-Et- 4-Me-Ph !, [BH4166; 5-Et-4-Me-Ph], [BH4167; 6-Et-4-Me-Ph], [BH4168; 2-Et-1-Ph], [BH4169; 3-Et-1-Ph], [BH4170; 4-Et-1-Ph], [BH4171; 5-Et-1-Ph], [BH4172; 6-Et-1-Ph], [BH4173; Et-3-Et-1-Ph], [BH4174; 2-Et-4-Et-1-Ph], [BH4175; 2-Et-5-Et-1-Ph], [BH4176; 2-Et- 6-Et-1-Ph], [BH4177; 3-Et-4-Et-1-Ph], [BH4178; 3-Et-5-Et-1-Ph], [BH4179; 4-Et-6- Et-1-Ph], [BH4 180; 2-F-4-Et-1-Ph], [BH4181; 3-F-4-Et-1-Ph], [BH4182; 5-F-4-Et- 1-Ph !, [BH4183; 6-F-4-Et-1-Ph], [BH4184; 2-F-5-Et-1-Ph], [BH4185; 3-F-5-Et-1-] Ph], [BH4186; 4-F-5-Et-1-Ph], [BH4187; 6-F-5-Et-1-Ph], [BH4188; 2-F-6-Et-1-P h], [BH4189; 3-F-6-Et-1-Ph], [BH4190; 4-F-6-Et-1-Ph], [BH4191; 5-F-6-Et-1-Ph] , [BH4192; 2-F-3-F-6-Et-1-Ph], [BH4193; 2-F-4-F-6-Et-1-Ph], [BH4194; F-6-Et-1-Ph], [BH4195; 3-F-4-F-6-Et-1-Ph], [BH4196; 3-F-5-F-6-Et-1-Ph] , [BH4197; 4-F-5-F-6-Et-1-Ph], [BH 4198; 2-Cl-4-Et-1-Ph], [BH4199; 3-Cl-4-Et-1-. Ph], [BH4200; 5-Cl-4-Et-1-Ph],

[BH4201; 6-Cl-4-Et-1-Ph], [BH4202; 2-Cl-5-Et-1-Ph], [BH4203; 3-Cl-5-Et-1-Ph], [BH4204] 4-Cl-5-Et-1-Ph !, [BH4205; 6-Cl-5-Et-1-Ph], [BH4206; 2-Cl-6-Et-1-Ph], [BH4207; -Cl-6-Et-1-Ph], [BH4208; 4-Cl-6-Et-1-Ph], [BH4209; 5-Cl-6-Et-1-Ph], [BH 4210; 2-Cl -3-Cl-6-Et-1-Ph !, [BH 4211; 2-Cl-4-Cl-6-Et-1-Ph], [BH 4212; 2-Cl-5-Cl-6-Et-1 -Ph], [BH 4213; 3-Cl-4-Cl-6-Et-1-Ph], [BH 4214; 3-Cl-5-Cl-6-Et-1-Ph], [BH 4215; 4-Cl -5-Cl-6-Et-1-Ph !, [BH4216; 2-Br-5-Et-1-Ph], [BH4217; 3-Br-5-Et-1-Ph], [BH4218; -Br-5-Et-1-Ph], [BH4219; 6-Br-5-Et-1-Ph], [BH4220; 2-CN-5-Et-1-Ph], [BH4221; 3-CN -5-Et-1-Ph !, [BH 4222; 4-CN-5-Et-1-Ph], [BH 4223; 6-CN-5-Et-1-Ph], [BH 4224; 2-OMe-5 -Et-1-Ph], [BH4225; 3-OMe-5-Et-1-Ph], [BH4226; 4-OMe-5-Et-1-Ph], [BH4227; 6-OMe-5-Et] -1-Ph], [BH 4228; 2-Et-5-Et-1-Ph], [BH 4229; 3-Et-5-Et-1-Ph], [BH 4230; 4-Et-5-Et-1 -Ph], [BH4231; 6-Et-5-Et-1-Ph], [BH4232; 2-Br-6-Et-1-Ph], [BH4233; 3-Br-6-Et-1-Ph ], [BH4234; 4-Br-6-Et-1-Ph], [BH4235; 5-Br-6-Et-1-Ph], [BH4236; 2-CN-6-Et-1-Ph], [BH4237; 3-CN-6-Et-1-Ph], [BH4238; 4-CN-6-Et-1-Ph], [BH4239; 5-CN-6-Et-1-Ph], [BH4240] 2-OMe-6-Et-1-Ph], [BH42 41; 3-OMe-6-Et-1-Ph !, [BH4242; 4-OMe-6-Et-1-Ph], [BH4243; 5-OMe-6-Et-1-Ph], [BH4244; 2-Pr-1-Ph], [BH4245; 3-Pr-1-Ph], [BH4246; 4-Pr-1-Ph], [BH4247; 5-Pr-1-Ph], [BH4248; 6- Pr-1-Ph], [BH 4249; 2-i-Pr-1-Ph], [BH 4250; 3-i-Pr-1-Ph], [BH 4251; 4-i-Pr-1-Ph], [B. BH 4252; 5-i-Pr-1-Ph], [BH 4253; 6-i-Pr-1-Ph], [BH 4254; 2-c-Pr-1-Ph], [BH 4 255; 3-c-Pr- 1-Ph], [BH4256; 4-c-Pr-1-Ph], [BH4257; 5-c-Pr-1-Ph], [BH4258; 6-c-Pr-1-Ph], [BH4259; 2-F-4-c-Pr-1-Ph !, [BH4260; 3-F-4-c-Pr-1-Ph], [BH4261; 5-F-4-c-Pr-1-Ph] [BH4262; 6-F-4-c-Pr-1-Ph], [BH4263; 2-F-5-c-Pr-1-Ph], [BH4264; 3-F-5-c-Pr- 1-Ph !, [BH4265; 4-F-5-c-Pr-1-Ph], [BH4266; 6-F-5-c-Pr-1-Ph], [BH4267; 2-F-6-6 c-Pr-1-Ph !, [BH4268; 3-F-6-c-Pr-1-Ph], [BH4269; 4-F-6-c-Pr-1-Ph], [BH4270; 5- F-6-c-Pr-1-Ph !, [BH4271; 2-F-3-F-6-c-Pr-1-Ph], [BH4272; 2-F-4-F-6-c- Pr-1-Ph], [BH4273; 2-F-5-F-6-c-Pr-1-Ph], [BH4274; 3-F-4-F-6-c-Pr-1-Ph] , [BH4275; 3-F-5-F-6-c-Pr-l-Ph], [BH4276; 4-F-5-F-6-c-Pr-l-Ph], [BH4277; Cl-4-c-Pr-1-Ph], [BH4278; 3-Cl-4-c-Pr-1-Ph], [BH4279; 5-Cl-4-c-Pr-1-Ph], [B. BH 4280; 6-Cl-4-c-Pr-1-Ph], [BH4281; 2-Cl-5-c-Pr-1-Ph], [BH4282; 3-Cl-5-c-Pr-1 -Ph], [BH4283; 4-Cl-5-c-Pr-1-Ph], [BH4284; 6-Cl-5-c-Pr-1-Ph], [BH4285; 2-Cl-6-c -Pr-1-Ph], [BH4286; 3-Cl-6-c-Pr-1-Ph], [BH4287; 4-Cl-6-c-Pr-1-Ph], [BH4288; 5-Cl -6-c-Pr-1-Ph !, [BH4289; 2-Cl-3-Cl-6-c-Pr-1-Ph], [BH4290; 2-Cl-4-Cl-6-c-Pr -1-Ph], [BH4291; 2-Cl-5-Cl-6-c-Pr-1-Ph], [BH4292; 3-Cl-4-Cl-6-c-Pr-1-Ph], [BH4293; 3-Cl-5-Cl-6-c-Pr-1-Ph], [BH4294; 4-Cl-5-Cl-6-c-Pr-1-Ph], [BH4295; 2-F -1-Ph], [BH 4296; 3-F-1-Ph], [BH 4297; 4-F-1-Ph], [BH 4298; 5-F-1-Ph], [BH 4 299; 6-F-1 -Ph], [BH4300; 2-F-3-F-1-Ph],

[BH4301; 2-F-4-F-1-Ph], [BH4302; 2-F-5-F-1-Ph], [BH4303; 2-F-6-F-1-Ph], [BH4304] 3-F-4-F-1-Ph !, [BH4305; 3-F-5-F-1-Ph], [BH4306; 4-F-5-F-1-Ph], [BH4307; -F-3-F-4-F-1-Ph !, [BH4308; 2-F-3-F-5-F-1-Ph], [BH4309; 2-F-3-F-6-F -1-Ph !, [BH 4310; 2-F-4-F-6-F-1-Ph], [BH4311; 2-F-4-F-5-F-1-Ph], [BH4312; -F-4-F-5-F-1-Ph !, [BH4313; 2-Cl-1-Ph], [BH4314; 3-Cl-1-Ph], [BH4315; 4-Cl-1-Ph ], [BH4316; 5-Cl-1-Ph], [BH4317; 6-Cl-1-Ph], [BH4318; 2-F-4-Cl-1-Ph], [BH4319; 3-F-4] -Cl-1-Ph], [BH4320; 5-F-4-Cl-1-Ph], [BH4321; 6-F-4-Cl-1-Ph], [BH4322; 2-F-5-Cl -1-Ph], [BH 4323; 3-F-5-Cl-1-Ph], [BH 4324; 4-F-5-Cl-1-Ph], [BH 4325; 6-F-5-Cl-1 -Ph], [BH4326; 2-F-6-Cl-1-Ph], [BH4327; 3-F-6-Cl-1-Ph], [BH4328; 4-F-6-Cl-1-Ph ], [BH4329; 5-F-6-Cl-1-Ph], [BH4330; 2-F-3-F-6-Cl-1-Ph], [BH4331; 2-F-4-F-6] -Cl-1-Ph], [BH4332; 2-F-5-F-6-Cl-1-Ph], [BH4333; 3-F-4-F-6-Cl-1-Ph], [BH4334] 3-F-5-F-6-Cl-1-Ph !, [BH4335; 4-F-5-F-6-Cl-1-Ph], [BH4336; 2-Cl-3-Cl-1 -Ph], [BH4 337; 2-Cl-4-Cl-1-Ph], [BH 4338; 2-Cl-5-Cl-1-Ph], [BH 4339; 2-Cl-6-Cl-1-Ph ], [BH4340; 3-Cl-4-Cl-1-Ph], [BH4341; 3-Cl-5-Cl-1-Ph], [BH4342; 4-Cl-5-Cl-1-Ph], [BH4343; 2-C l-3-Cl-4-Cl-1-Ph !, [BH4344; 2-Cl-3-Cl-5-Cl-1-Ph], [BH4345; 2-Cl-3-Cl-6-Cl- 1-Ph !, [BH 4346; 2-Cl-4-Cl-5-Cl-1-Ph], [BH 4347; 2-Cl-4-Cl-6-Cl-1-Ph], [BH 4348; Cl-4-Cl-5-Cl-1-Ph !, [BH4349; 2-Br-1-Ph], [BH4350; 3-Br-1-Ph], [BH4351; 4-Br-1-Ph] , [BH4352; 5-Br-1-Ph], [BH4353; 6-Br-1-Ph], [BH4354; 2-CN-1-Ph], [BH4355; 3-CN-1-Ph], [BH4352; BH4356; 4-CN-1-Ph], [BH4357; 5-CN-1-Ph], [BH4358; 6-CN-1-Ph], [BH4359; 2-F-4-CN-1-Ph] [BH4360; 3-F-4-CN-1-Ph], [BH4361; 5-F-4-CN-1-Ph], [BH4362; 6-F-4-CN-1-Ph], BH4363; 2-F-5-CN-1-Ph !, [BH4364; 3-F-5-CN-1-Ph], [BH4365; 4-F-5-CN-1-Ph], [BH4366; 6-F-5-CN-1-Ph !, [BH 4367; 2-F-6-CN-1-Ph], [BH 4368; 3-F-6-CN-1-Ph], [BH 4369; F-6-CN-1-Ph !, [BH4370; 5-F-6-CN-1-Ph], [BH4371; 2-F-3-F-6-CN-1-Ph], [BH4372; 2-F-4-F-6-CN-1-Ph !, [BH4373; 2-F-5-F-6-CN-1-Ph], [BH4374; 3-F-4-F-6-6 CN-1-Ph !, [BH4375; 3-F-5-F-6-CN-1-Ph], [BH4376; 4-F-5-F-6-CN-1-Ph], [BH4 377; 2-Cl-4-CN-1-Ph !, [BH 4378; 3-Cl-4-CN-1-Ph], [BH 4379; 5-Cl-4-CN-1-Ph], [BH 4380; 6- Cl-4-CN-1-Ph !, [BH4381; 2-Cl-5-CN-1-Ph], [BH4382; 3-Cl-5-CN-1-Ph], [BH4383; 4-Cl- 5-CN-1-Ph !, [BH4384; 6-Cl-5-CN-1-Ph], [BH4385; 2-Cl-6-CN -1-Ph], [BH4386; 3-Cl-6-CN-1-Ph], [BH4387; 4-Cl-6-CN-1-Ph], [BH4388; 5-Cl-6-CN-1 -Ph], [BH4 389; 2-Cl-3-Cl-6-CN-1-Ph], [BH 4390; 2-Cl-4-Cl-6-CN-1-Ph], [BH 4391; 2-Cl -5-Cl-6-CN-1-Ph !, [BH4392; 3-Cl-4-Cl-6-CN-1-Ph], [BH4393; 3-Cl-5-Cl-6-CN-1 4-Ph], [BH 4394; 4-Cl-5-Cl-6-CN-1-Ph], [BH 4395; 2-OMe-Ph], [BH 4396; 3-OMe-Ph], [BH 4397; -Ph], [BH4398; 5-OMe-Ph], [BH4399; 6-OMe-Ph], [BH4400; 2-OMe-3-OMe-Ph],

[BH4401; 2-OMe-4-OMe-Ph], [BH4402; 2-OMe-5-OMe-Ph], [BH4403; 2-OMe-6-OMe-Ph], [BH4404; 3-OMe-4 -OMe-Ph], [BH4405; 3-OMe-5-OMe-Ph], [BH4406; 4-OMe-5-OMe-Ph], [BH4407; 2-F-4-OMe-Ph], [BH4408] 3-F-4-OMe-Ph !, [BH4409; 5-F-4-OMe-Ph], [BH4410; 6-F-4-OMe-Ph], [BH4411; 2-F-5-OMe -Ph], [BH4412; 3-F-5-OMe-Ph], [BH4413; 4-F-5-OMe-Ph], [BH4414; 6-F-5-OMe-Ph], [BH4415; -F-6-OMe-Ph], [BH4416; 3-F-6-OMe-Ph], [BH4417; 4-F-6-OMe-Ph], [BH4418; 5-F-6-OMe-Ph ], [BH4419; 2-F-3-F-6-OMe-Ph], [BH4420; 2-F-4-F-6-OMe-Ph], [BH4421; 2-F-5-F-6] -OMe-Ph], [BH4422; 3-F-4-F-6-OMe-Ph], [BH4423; 3-F-5-F-6-OMe-Ph], [BH4424; 4-F-5 -F-6-OMe-Ph], [BH4425; 2-Cl-4-OMe-Ph], [BH4426; 3-Cl-4-OMe-Ph], [BH4427; 2-Cl-5-OMe-Ph ], [BH4428; 3-Cl-5-OMe-Ph], [BH4429; 4-Cl-5-OMe-Ph], [BH4430; 6-Cl-5-OMe-Ph], [BH4431; -6-OMe-Ph !, [BH4432; 3-Cl-6-OMe-Ph], [BH4433; 4-Cl-6-OMe-Ph], [BH4434; 5-Cl-6-OMe-Ph], [BH4435; 2-Cl-3-Cl-6-OMe-Ph], [BH4436; 2-Cl-4-Cl-6-OMe-Ph], [BH4437; 2-Cl-5-Cl-6-OMe -Ph], [BH4438; 3-Cl-4-Cl-6-OMe-Ph], [BH4439; 3-Cl-5-Cl-6-OMe-Ph], [BH4440; 4-Cl-5-Cl -6-OMe-Ph], [BH4441; 2-OEt-1-Ph], [BH4442; 3-OEt-1-Ph ], [BH4443; 4-OEt-1-Ph], [BH4444; 5-OEt-1-Ph], [BH4445; 6-OEt-1-Ph], [BH4446; 2-CF ₃ -1-Ph] _{, [BH4447; 3-CF 3} -1-Ph], [BH4448; 4-CF 3 -1-Ph], [BH4449; 5-CF 3 -1-Ph], [BH4450; 6-CF 3 -1- Ph], [BH4451; 2- F-4-CF 3 -1-Ph], [BH4452; 3-F-4-CF 3 -1-Ph], [BH4453; 5-F-4-CF 3 -1 -Ph], [BH4454; 6- F-4-CF 3 -1-Ph], [BH4455; 2-F-5-CF 3 -1-Ph], [BH4456; 3-F-5-CF 3 - 1-Ph], [BH4457; 4-F-5-CF 3 -1-Ph], [BH4458; 6-F-5-CF 3 -1-Ph], [BH4459; 2-F-6-CF 3 -1-Ph], [BH4460; 3-F-6-CF 3 -1-Ph], [BH4461; 4-F-6-CF 3 -1-Ph], [BH4462; 5-F-6-CF _{3 -1-Ph], [BH4463} ; 2-F-3-F-6-CF 3 -1-Ph], [BH4464; 2-F-4-F-6-CF 3 -1-Ph], [ BH4465; 2-F-5- F-6-CF 3 -1-Ph], [BH4466; 3-F-4-F-6-CF 3 -1-Ph], [BH4467; 3-F-5- _{F-6-CF 3 -1-} Ph], [BH4468; 4-F-5-F-6-CF 3 -1-Ph], [BH4469; 2-Cl-4-CF 3 -1-Ph], [BH4470; 3-Cl-4 -CF 3 -1-Ph], [BH4471; 5-Cl-4-CF 3 -1-Ph], [BH4472; 6-Cl-4-CF 3 -1-Ph] , [BH4473; 2-Cl- 5-CF 3 -1-Ph], [BH4474; 3-Cl-5-CF 3 -1-Ph], [BH4475; 4-Cl-5-CF 3 -1-Ph ], [BH4476; 6-Cl -5-CF 3 -1-Ph], [BH4477; 2-Cl-6-CF 3 -1-Ph], [BH4478; 3-Cl-6-CF 3 -1- Ph], [BH4479; 4- Cl-6-CF 3 -1-Ph], [BH4480; 5-Cl-6-CF 3 -1-Ph], [BH4481; 2-Cl -3-Cl-6-CF ₃ -1-Ph !, [BH 4482; 2,4-Cl 6-CF ₃ -1-Ph], [BH 4483; 2, 5-Cl 6-CF ₃ -1-] Ph], [BH4484; 3,4- Cl-6-CF 3 -1-Ph], [BH4485; 3,5-Cl-6-CF 3 -1-Ph], [BH4486; 4-Cl-5- _{Cl-6-CF 3 -1-} Ph], [BH4487; 2-amino-1-Ph], [BH4488; 3-amino-1-Ph], [BH4489; 4-amino-1-Ph], [BH4490 5-amino-1-Ph !, [BH4491; 6-amino-1-Ph], [BH4492; 2-N, N-dimethylamino-1-Ph], [BH4493; 3-N, N-dimethylamino-1 -Ph], [BH4494; 4-N, N-dimethylamino-1-Ph], [BH 4495; 5-N, N-dimethylamino-1-Ph], [BH 4496; 6-N, N-dimethylamino-1-Ph ], [BH 4497; 2-SMe-Ph], [BH 4498; 3-SMe-Ph], [BH 4499; 4-SMe-Ph], [BH 4500; 5-SMe-Ph], [BH 4501; 6-SMe-Ph] ].

  In addition, the present compounds AI1-BI1 to AI6096-BI1423 can also be obtained according to the above-mentioned method.

The present compounds AI1-BI1 to AI6096-BI1423 are compounds represented by the following formula (AIBI).

[Wherein, X ^{90 to} X ¹⁰¹ each represent a substituent corresponding to each of substituent numbers (MI1) AI 1 to AI 6096 shown below, wherein E ¹⁰⁹ is a substituent number (MI 2) BI 1 shown below ~ BI 1423. ]
For example, the present compound AI1-BI1 is a compound represented by the formula (AIBI), wherein X ^{90 to} X ¹⁰¹ have a substituent number MI 1 (X ^{90 to} X ⁹³ , X ^{95 to} X ⁹⁷ and X ^{98 a} hydrogen atom, X ⁹⁴ , X ⁹⁹ and X ¹⁰⁰ are oxygen atoms, X ¹⁰¹ is OMe, and E ¹⁰⁹ is a compound in which the substituent number (MI2) is BI1 (pyrazol-1-yl group), and is represented by the following formula.

[Substituent group number ^{(MI1); X 90, X} 91, X 92, X 93, X 94, X 95, X 96, X 97, X 98, X 99, X 100, X 101]: [AI1; H, H, H, H, H, H, H, H, H, H, O, O, OMe], [AI2; H, H, H, H, O, H, H, H, F, O, O, OMe] [AI3; H, H, H, H, H, O, H, H, H, Cl, O, O, OMe], [AI 4; H, H, H, H, O, H, H, H, Br, O, O, OMe], [AI5; H, H, H, H, O, H, H, H, I, O, O, OMe], [AI 6; H, H, H, H, O, H, H, H, Me, O, O, OMe], [AI7; H, H, H, H, H, O, H, H, H, Et, O, O, OMe], [AI 8; H, H, H, H, O, H, H, H, c, Pr, O, O, OMe], [AI 9; H, H, H, H, O, H, H, H, OMe, O, O, OMe], [ AI10; H, H, H, H, H, O, H, H, H, OEt, O, O, OMe], [AI11; H, H, H, H, H, O, H, H, SMe, O, O, OMe], [AI 12; H, H, H, H, O, H, H, H, CF ₃ , O, O, OMe], [AI 13; F, H, H, H, O, H, H , H, H, O, O, OMe], [AI 14; F, H, H, H, O, H, H, H, H, F, O, O, OMe], [AI 15; F, H, H, H , O, H, H, H, H, Cl, O, O, OMe], [AI 16; F, H, H, H, O, H, H, H, Br, O, O, OMe], [AI 17; , H, H, H, O, H, H, H, I, O, O, OMe], [AI 18; F, H, H, H, O, H, H, H, Me, O, O, OMe ], [AI19; F, H, H, H, O, H, H, H, Et, O, O, OMe], [AI 20; F, H, H, H, O, H, H, H, c -Pr, O, O, OMe], [AI 21; F, H, H, H, O, H, H, H, H, OMe, O, O, OMe], [AI 22; F, H, H, H, O , H, H, H, H, OEt, O, O, OMe], [AI23; F, H, H, H, H, O, H, H, S, Me, O, O, OMe], [AI 24; , H, H, O, H , H, H, CF 3, O, O, OMe], [AI25; Cl, H, H, H, O, H, H, H, H, O, O, OMe] , [AI26; Cl, H, H, H, O, H, H, H, H, F, O, O, OMe], [AI 27; Cl, H, H, H, O, H , H, H, Cl, O, O, OMe], [AI 28; Cl, H, H, H, H, O, H, H, H, Br, O, O, OMe], [AI 29; Cl, H, H , H, O, H, H, H, H, I, O, O, OMe], [AI 30; Cl, H, H, H, O, H, H, H, Me, O, O, OMe], [AI 31 Cl, H, H, H, H, O, H, H, H, H, Et, O, O, OMe], [AI 32; Cl, H, H, H, H, O, H, H, H, c-Pr, O , O, OMe], [AI 33; Cl, H, H, H, O, H, H, H, OMe, O, O, OMe], [AI 34; Cl, H, H, H, O, H, H , H, OEt, O, O, OMe], [AI 35; Cl, H, H, H, H, O, H, H, H, SMe, O, O, OMe], [AI 36; Cl, H, H, H , O, H, H, H , CF 3, O, O, OMe], [AI37; Br, H, H, H, O, H, H, H, H, O, O, OMe], [AI38; Br, H, H, H, H, O, H, H, H, H, H, F, O, O, OMe], [AI 39; Br, H, H, H, O, H, H, H, Cl, O, O, O OMe], [AI 40; Br, H, H, H, O, H, H, H, Br, O, O, OMe], [AI 41; Br, H, H, H, O, H, H, H, H, Br, H, H, H, H, O, H, H, H, Me, O, O, OMe], [AI 43; Br, H, H, H, O, I, O, O, OMe], [AI 42; H, H, H, H, Et, O, O, OMe], [AI 44; Br, H, H, H, H, O, H, H, H, c-Pr, O, O, OMe], [AI 45; Br, H, H, H, O, H, H, H, H, OMe, O, O, OMe], [AI 46; Br, H, H, H, O, H, H, H, OEt, O, O, OMe] , [AI47; Br, H, H, H, O, H, H, H, SMe, O, O, OMe], [AI 48; Br, H, H, H, H, O, H, H, H, CF ₃ , O, O, OMe], [AI 49; Me, H, H, H, H, O, H, H, H, H, O, O, OMe], [AI 50; Me, H, H, H, O, H , H, H, F, O, O, OMe], [AI 51; Me, H, H, H, H, O, H, H, H, Cl, O, O, OMe], [AI 52; Me, H, H , H, O, H, H, H, H, Br, O, O, OMe], [AI 53; Me, H, H, H, O, H, H, H, I, O, O, OMe], [AI 54 Me, H, H, H, H, O, H, H, H, H, Me, O, O, OMe], [AI 55; Me, H, H, H, H, O, H, H, H, Et, O, O; , OMe], [AI56; Me, H, H, H, O, H, H, H, c-Pr, O, O, OMe], [AI 57; Me, H, H, H, O, H, H , H, OMe, O, O, OMe], [AI 58; Me, H, H, H, O, H, H, H, H, OE t, O, O, OMe], [AI 59; Me, H, H, H , O, H, H, H, SMe, O, O, OMe], [AI 60; Me, H, H, H, H, O, H, H, H, CF ₃ , O, O, OMe], [AI 61; Et, H, H, H, H, O, H, H, H, H, H, O, O, OMe], [AI 62; Et, H, H, H, H, O, H, H, H, F, O, O, O OMe], [AI 63; Et, H, H, H, O, H, H, H, H, Cl, O, O, OMe], [AI 64; Et, H, H, H, O, H, H, H, H, Br, O, O, OMe], [AI 65; Et, H, H, H, H, O, H, H, H, I, O, O, OMe], [AI 66; Et, H, H, H, O, H, H, H, H, Me, O, O, OMe], [AI 67; Et, H, H, H, H, O, H, H, H, Et, O, O, OMe], [AI 68; Et, H, H, H, O, H, H, H, c, Pr, O, O, OMe], [AI69; Et, H, H, H, O, H, H, H, OMe, O, O, OMe] , [AI70; Et, H, H, H, O, H, H, H, OEt, O, O, OMe], [AI 71; Et, H, H, H, H, O, H, H, H, SMe, O, O, OMe], [ AI72; Et, H, H, H, O, H, H, H, CF 3, O, O, OMe], [AI73; CF 3, H, H, H, O, H, H, H, H, H, O, O, OMe], [AI 74; CF ₃ , H, H, H, O, H, H, H, F, O, O, OMe], [AI 75; CF ₃ , H, H, H, O, H, H, H, Cl, O, O, OMe], [AI76; CF 3, H, H, H, O, H, H, H, Br, O, O, OMe _{], [AI77; CF 3,} H, H, H, O, H, H, H, I, O, O, OMe], [AI78; CF 3, H, H, H, O, H, H, H , Me, O, O, OMe ], [AI79; CF 3, H, H, H, O, H, H, H, Et, O, O, OMe], [AI80; CF 3, H, H, H , O, H, H, H, c, -Pr, O, O, OMe], [AI 81; CF ₃ , H, H, H, O, H, H, H, OMe, O, O, OMe], [ AI 82; CF ₃ , H, H, H, H, O, H, H, H, OE t, O, O, OMe], [AI 83 CF ₃ , H, H, H, H, O, H, H, H, SMe, O, O, OMe], [AI 84; CF ₃ , H, H, H, O, H, H, H, CF ₃ , O, O, OMe], [AI 85; c-Pr, H, H, H, H, O, H, H, H, H, O, O, OMe], [AI 86; c-Pr, H, H, H, O, H, H, H, H, F, O, O, OMe], [AI 87; c-Pr, H, H, H, H, O, H, H, H, Cl, O, O, OMe], [AI 88; c-Pr, H, H, H, H, O, H, H, H, H, Br, O, O, OMe], [AI 89; c-Pr, H, H, H, O, H, H, H, I, I, O, O, OMe], [AI 90; c-Pr, H, H, H, H, O, H, H, H, Me, O, O, OMe], [AI 91; c-Pr, H, H, H, O, H, H, H, H, Et, O, O, OMe], [AI 92; c-Pr, H, H, H, O, H, H, H, c-Pr, O, O, OMe], [[ AI 93; c-Pr, H, H, H, O, H, H, H, OMe, O, O, OMe], [AI 94; c-Pr, H, H, H, O, H, H, H, OEt, O, O, OMe], [AI95; c-Pr, H, H, H, H, O, H, H, H, SMe, O, O, OMe], [AI96; c-Pr, H, H, H, O, H, H, H, CF 3, O, O, OMe], [AI97; H, H, F, H, O, H, H, H, H, O, O, OMe], [AI98 H, H, F, H, O, H, H, H, H, F, O, O, OMe], [AI99; H, H, F, H, O, H, H, H, Cl, O, O , OMe], [AI 100; H, H, F, H, O, H, H, H, Br, O, O, OMe],

[AI 101; H, H, F, H, O, H, H, H, I, O, O, OMe], [AI 102; H, H, F, H, O, H, H, H, Me, O , O, OMe], [AI 103; H, H, F, H, O, H, H, H, Et, O, O, OMe], [AI 104; H, H, F, H, O, H, H , H, c-Pr, O, O, OMe], [AI 105; H, H, F, H, O, H, H, H, OMe, O, O, OMe], [AI 106; H, H, F , H, O, H, H, H, OEt, O, O, OMe], [AI 107; H, H, F, H, O, H, H, H, SMe, O, O, OMe], [AI 108 ; H, H, F, H , O, H, H, H, CF 3, O, O, OMe], [AI109; F, H, F, H, O, H, H, H, H, O, O, OMe], [AI 110; F, H, F, H, O, H, H, H, F, O, O, OMe], [AI 111; F, H, F, H, O, H, H, H, Cl, O, O, OMe], [AI 112; F, H, F, H, O, H, H, H, H, Br, O, O, OMe], [AI 113; F, H, F, H, O, H, H, H, H, I, O, O, OMe], [AI 114; F, H, F, H, O, H, H, H, Me, O, O, OMe], [AI 115; F, H, F, H, O, H, H, H, H, Et, O, O, OMe], [AI 116; F, H, F, H, O, H, H, H, c-Pr, O, O, OMe], [AI117; F, H, F, H, O, H, H, H, OMe, O, O, OMe], [AI 118; F, H, F, H, O, H, H, H, OEt, O, O, OMe], [AI119; F, H, F, H, O, H, H, H, SMe, O, O, OMe], [AI 120; F, H, F, H, O, _{H, H, H, CF 3} , O, O, OMe], [AI121; Cl, H, F, H, O, H, H, H, H, O, O, OMe], [AI122; Cl, H , F, H, O, H, H, H, H, F, O, O, OMe], [AI 123; Cl, H, F, H, O, H, H, H, Cl, O, O, OMe], [AI 124; Cl, H, F, H, O, H, H, H, Br, O, O, OMe], [AI 125; Cl, H, F, H, O, H, H, H, I, O , O, OMe], [AI 126; Cl, H, F, H, O, H, H, H, Me, O, O, OMe], [AI 127; Cl, H, F, H, O, H, H , H, Et, O, O, OMe], [AI 128; Cl, H, F, H, O, H, H, H, c, Pr, O, O, OMe], [, AI129; Cl, H, F, H, O, H, H, OMe, O, O, OMe], [AI 130; Cl, H, F, H, O, H, H, H, OEt, O, O, OMe], [AI 131; Cl, H, F, H, O, H, H, H, SMe, O, O, OMe], [AI 132; Cl, H, F, H, O, H, H, _{H, CF 3, O, O} , OMe], [AI133; Br, H, F, H, O, H, H, H, H, O, O, OMe], [AI134; Br, H, F, H , O, H, H, H, F, O, O, OMe], [AI 135; Br, H, F, H, O, H, H, H, Cl, O, O, OMe], [AI 136; Br , H, F, H, O, H, H, H, H, Br, O, O, OMe], [AI 137; Br, H, F, H, O, H, H, H, I, O, O, OMe , [AI 138; Br, H, F, H, O, H, H, H, Me, O, O, OMe], [AI 139; Br, H, F, H, O, H, H, H, Et, , O, O, OMe], [AI 140; Br, H, F, H, O, H, H, H, c, Pr, O, O, OMe], [AI 141; Br, H, F, H, O , H, H, H, H, OMe, O, O, OMe], [AI 142; Br, H, F, H, O, H, H, H, OEt, O, O, OMe], [AI 143; Br, H , F, H, O, H , H, H, SMe, O, O, OMe], [AI144; Br, H, F, H, O, H, H, H, CF 3, O, O, OMe] , [AI 145; Me, H, F, H, O, H, H, H, H, O, O, OMe], [AI 146; Me, H, F, H, O, H, H, H, F, F, O, O, OMe], [AI 147; Me, H, F, H, O, H, H, H, Cl, O, OMe], [AI 148; Me, H, F, H, O, H, H, H, Br, O, O, OMe], [AI 149; Me, H, F, H, O, H, H, H, I, O, O, OMe], [AI 150; Me, H, F, H, O, H, H, H, H, Me, O, O, OMe], [AI 151; Me, H, F, H, O, H, H, H, Et, O, O, OMe], [AI 152; Me, H, F, H, O, H, H, H, c, Pr, O, O, OMe], [AI 153; Me, H, F, H, O, H, H, H, OMe, O, O, OMe], [AI154; Me, H, F, H, O, H, H, H, OEt, O, O, OMe], [AI 155; Me, H, F, H, O, H, H, H, SMe, O, O, OMe], [AI 156; Me, H, F, H, O, H, H, H, CF 3, O, O, OMe], [AI157; Et, H, F, H, O, H, H, H, H, O, O, OMe], [AI158; Et , H, F, H, O, H, H, H, H, F, O, O, OMe], [AI 159; Et, H, F, H, O, H, H, H, Cl, O, O, OMe ], [AI 160; Et, H, F, H, O, H, H, H, Br, O, O, OMe], [AI 161; Et, H, F, H, O, H, H, H, I , O, O, OMe], [AI 162; Et, H, F, H, O, H, H, H, Me, O, O, OMe], [AI 163; Et, H, F, H, O, H , H, H, Et, O, O, OMe], [AI 164; Et, H, F, H, O, H, H, H, c-Pr, O, O, OMe], [AI 165; Et, H , F, H, O, H, H, H, H, OMe, O, O, OMe], [AI 166; Et, H, F, H, O, H, H, H, OEt, O, O, OMe], [AI 167; Et, H, F, H, O, H, H, H, S Me, O, O, OMe], [AI 168; Et, H, F, H, O, H, H, H, CF ₃ , O, O, OMe], [ AI169; CF 3, H, F, H, O, H, H, H, H, O, O, OMe], [AI170; CF 3, H, F, H, O, H, H, H, F, O, O, OMe], [AI171; CF 3, H, F, H, O, H, H, H, Cl, O, O, OMe], [AI172; CF 3, H, F, H, O, H, H, H, Br, O, O, OMe], [AI173; CF 3, H, F, H, O, H, H, H, I, O, O, OMe _{], [AI174; CF 3,} H, F, H, O, H, H, H, Me, O, O, OMe], [AI175; CF 3, H, F, H, O, H, H, H , Et, O, O, OMe ], [AI176; CF 3, H, F, H, O, H, H, H, c-Pr, O, O, OMe], [AI177; CF 3, H, F , H, O, H, H , H, OMe, O, O, OMe], [AI178; CF 3, H, F, H, O, H, H, H, OEt, O, O, OMe], [ _{AI179; CF 3, H, F} , H, O, H, H, H, SMe, O, O, OMe], [AI180; CF 3, H, F, H, O, H, H, H, CF 3 H, H, Cl, H, O, H, H, H, H, O, O, OMe], [AI 182; H, H, Cl, H, O, H , H, H, F, O, O, OM e, [AI 183; H, H, Cl, H, O, H, H, H, Cl, O, O, OMe], [AI 184; H, H, Cl, H, O, H, H, H, H, Br, O, O, OMe], [AI 185; H, H, Cl, H, O, H, H, H, I, O, O, OMe], [AI 186; H, H, Cl, H, O, H, H, H, Me, O, O, OMe], [AI 187; H, H, Cl, H, O, H, H, H, Et, O, O, OMe], [AI 188; H, H, Cl, H, O, H, H, H, c, Pr, O, O, OMe], [AI 189; H, H, Cl, H, O, H, H, H, OMe, O, O, OMe] , [AI190; H, H, Cl, H, O, H, H, OEt, O, O, OMe], [AI 191; H, H, Cl, H, O, H, H, H, SMe, O, O, OMe], [ AI192; H, H, Cl, H, O, H, H, H, CF 3, O, O, OMe], [AI193; F, H, Cl, H, O, H , H, H, H, H, O, O, OMe], [AI 194; F, H, Cl, H, O, H, H, H, F, O, O, OMe], [AI 195; F, H, Cl , H, O, H, H, H, H, Cl, O, O, OMe], [AI 196; F, H, Cl, H, O, H, H, H, Br, O, O, OMe], [AI 197] F, H, Cl, H, O, H, H, H, H, I, O, O, OMe], [AI 198; F, H, Cl, H, O, H, H, H, Me, O, O; , OMe], [AI 199; F, H, Cl, H, O, H, H, H, Et, O, O, OMe], [AI 200; F, H, Cl, H, O, H, H, H , c-Pr, O, O, OMe],

[AI201; F, H, Cl, H, O, H, H, H, OMe, O, O, OMe], [AI 202; F, H, Cl, H, O, H, H, H, OEt, O , O, OMe], [AI203; F, H, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI 204; F, H, Cl, H, O, H, H _{, H, CF 3, O,} O, OMe], [AI205; Cl, H, Cl, H, O, H, H, H, H, O, O, OMe], [AI206; Cl, H, Cl, H, O, H, H, H, H, F, O, O, OMe], [AI 207; Cl, H, Cl, H, O, H, H, H, Cl, O, O, OMe], [AI 208; Cl, H, Cl, H, O, H, H, H, H, Br, O, O, OMe], [AI 209; Cl, H, Cl, H, O, H, H, H, I, O, O, OMe], [AI 210; Cl, H, Cl, H, O, H, H, H, Me, O, O, OMe], [AI 211; Cl, H, Cl, H, O, H, H, H, H, Et, O, O, OMe], [AI 212; Cl, H, Cl, H, O, H, H, H, c, Pr, O, O, OMe], [AI 213; Cl, H, Cl, H, O, H, H, H, H, OMe, O, O, OMe], [AI 214; Cl, H, Cl, H, O, H, H, H, OEt, O, O, OMe], [AI 215; H, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI216; Cl, H, Cl, H, O, H, H, H, CF 3, O, O, OMe ], [AI 217; Br, H, Cl, H, O, H, H, H, H, H, O, O, OMe], [AI 218; Br, H, Cl, H, O, H, H, H, F] , O, O, OMe], [AI219; Br, H, Cl, H, O, H, H, H, H, Cl, O, OMe], [AI 220; Br, H, Cl, H, O, H , H, H, Br, O, O, OMe], [AI 221; Br, H, Cl, H, O, H, H, H, I, O, O, OMe], [AI 222; Br, H, Cl , H, O, H, H, H, H, Me, O, O, OMe], [AI 223; Br, H, Cl, H, O, H, H, H, Et, O, O, OMe], [AI 224 Br, H, Cl, H, O, H, H, H, c, Pr, O, O, OMe], [AI 225; Br, H, Cl, H, O, H, H, H, OMe, O , O, OMe], [AI 226; Br, H, Cl, H, O, H, H, H, OEt, O, O, OMe], [AI 227; Br, H, Cl, H, O, H, H , H, SMe, O , O, OMe], [AI228 ; Br, H, Cl, H, O, H, H, H, CF 3, O, O, OMe], [AI229; Me, H, Cl, H, O, H, H, H, H, H, O, O, OMe], [AI 230; Me, H, Cl, H, O, H, H, H, F, O, O, OMe], [AI 231; Me, H, Cl, H, O, H, H, H, H, Cl, O, O, OMe], [AI 232; Me, H, Cl, H, O, H, H, H, Br, O, O, OMe], [AI 233; Me, H, Cl, H, O, H, H, H, H, I, O, O, OMe], [AI 234; Me, H, Cl, H, O, H, H, Me, O, O, OMe], [AI235; Me, H, Cl, H, O, H, H, H, Et, O, O, OMe], [AI 236; Me, H, Cl, H, O, H, H, H, H, c-Pr, O, O, OMe], [AI 237; Me, H, Cl, H, O, H, H, H, H, OMe, O, O, OMe], [AI 238; Me, H, Cl, H, O, H, H, H, H, OEt, O, O, OMe], [AI 239; Me, H, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI 240; H, Cl, H, O, H, H, H, CF 3, O, O, OMe], [AI241; Et, H, Cl, H, O, H, H, H, H, O, O, OMe ], [AI 242; Et, H, Cl, H, O, H, H, H, F, O, O, OMe], [AI 243; Et, H, Cl, H, O, H, H, H, Cl, , O, O, OMe], [AI 244; Et, H, Cl, H, O, H, H, H, H, Br, O, O, OMe], [AI 245; Et, H, Cl, H, O, H , H, H, I, O, O, OMe], [AI 246; Et, H, Cl, H, O, H, H, H, Me, O, O, OMe], [AI 247; Et, H, Cl , H, O, H, H, H, H, Et, O, O, OMe], [AI 248; Et, H, Cl, H, O, H, H, H, c-Pr, O, O, OMe], [AI 249; Et, H, Cl, H, O, H, H, H, OMe, O, O, OMe], [AI 250; Et, H, Cl, H, O, H, H, H, OEt, O , O, OMe], [AI 251; Et, H, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI 252; Et, H, Cl, H, O, H, H _{, H, CF 3, O,} O, OMe], [AI253; CF 3, H, Cl, H, O, H, H, H, H, O, O, OMe], [AI254; CF 3, H, Cl, H, O, H, H, H, F, O, O, OMe], [AI255; CF 3, H, Cl, H, O, H, H, H, Cl, O, O, OMe], _{[AI256; CF 3, H,} Cl, H, O, H, H, H, Br, O, O, OMe], [AI257; CF 3, H, Cl, H, O, H, H, H, I , O, O, OMe], [AI258; CF 3, H, Cl, H, O, H, H, H, Me, O, O, OMe], [AI259; CF 3, H, Cl, H, O , H, H, H, Et , O, O, OMe], [AI260; CF 3, H, Cl, H, O, H, H, H, c-Pr, O, O, OMe], [AI261; _{CF 3, H, Cl, H} , O, H, H, H, OMe, O, O, OMe], [AI262; CF 3, H, Cl, H, O, H, H, H, OEt, O, O, OMe], [AI263; CF 3, H, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI264; CF 3, H, Cl, H, O, H, _{H, H, CF 3, O} , O, OMe], [AI265; H, H, Me, H, O, H, H, H, H, O, O, OMe], [AI266; H, H, Me , H, O, H, H, H, H, F, O, O, OMe], [AI 267; H, H, Me, H, O, H, H, H, Cl, O, O, OMe], [AI268] H, H, Me, H, O, H, H, H, H, Br, O, OMe], [AI 269; H, H, Me, H, O, H, H, H, I, O, O , OMe], [AI 270; H, H, Me, H, O, H, H, H, Me, O, O, OMe], [AI 271; H, H, Me, H, O, H, H, H , Et, O, O, OMe], [AI 272; H, H, Me, H, O, H, H, H, c, Pr, O, O, OMe], [AI 273; H, H, Me, H , O, H, H, H, H, OMe, O, O, OMe], [AI 274; H, H, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 275; H , H, Me, H, O , H, H, H, SMe, O, O, OMe], [AI276; H, H, Me, H, O, H, H, H, CF 3, O, O, OMe], [AI 277; F, H, Me, H, O, H, H, H, H, H, O, O, OMe], [AI 278; F, H, Me, H, O, H, H, H, H, F, O, O, OMe], [AI 279; F, H, Me, H, O, H, H, H, H, Cl, O, OMe], [AI 280; F, H, Me, H, O, H, H, H, Br , O, O, OMe], [AI 281; F, H, Me, H, O, H, H, H, I, O, O, OMe], [AI 282; F, H, Me, H, O, H , H, H, Me, O, O, OMe], [AI 283; F, H, Me, H, O, H, H, H, Et, O, O, OMe], [AI 284; F, H, Me , H, O, H, H, H, c, Pr, O, O, OMe], [AI 285; F, H, Me, H, O, H, H, H, OMe, O, O, OMe], [AI286; F, H, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 287; F, H, Me, H, O, H, H, H, SMe, O , O, OMe], [AI288 ; F, H, Me, H, O, H, H, H, CF 3, O, O, OMe], [AI289; Cl, H, Me, H, O, H, H, H, H, H, O, O, OMe], [AI 290; Cl, H, Me, H, O, H, H, H, F, O, O, OMe], [AI 291: Cl, H, Me, H, O, H, H, H, H, Cl, O, O, OMe], [AI 292; Cl, H, Me, H, O, H, H, H, Br, O, O, OMe], [AI 293; Cl, H, Me, H, O, H, H, H, H, I, O, O, OMe], [AI 294; Cl, H, Me, H, O, H, H, H, Me, O, O, O OMe], [AI 295; Cl, H, Me, H, O, H, H, H, Et, O, O, OMe], [AI 296; Cl, H, Me, H, O, H, H, H, H, c-Pr, O, O, OMe], [AI 297; Cl, H, Me, H, O, H, H, H, H, OMe, O, O, OMe], [AI 298; Cl, H, Me, H, O, H, H, H, H, OEt, O, O, OMe], [AI 299; Cl, H, Me, H, O, H, H, H, SMe, O, O, OMe], [AI 300; H, Me, H, O, H, H, H, CF 3, O, O, OMe],

[AI 301; Br, H, Me, H, O, H, H, H, H, O, O, OMe], [AI 302; Br, H, Me, H, O, H, H, H, F, O , O, OMe], [AI303; Br, H, Me, H, O, H, H, H, Cl, O, O, OMe], [AI 304; Br, H, Me, H, O, H, H , H, Br, O, O, OMe], [AI 305; Br, H, Me, H, O, H, H, H, I, O, O, OMe], [AI 306; Br, H, Me, H , O, H, H, H, H, Me, O, O, OMe], [AI 307; Br, H, Me, H, O, H, H, H, Et, O, O, OMe], [AI 308; Br , H, Me, H, O, H, H, H, c, Pr, O, O, OMe], [AI309; Br, H, Me, H, O, H, H, H, OMe, O, O , OMe], [AI 310; Br, H, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 311; Br, H, Me, H, O, H, H, H , SMe, O, O, OMe ], [AI312; Br, H, Me, H, O, H, H, H, CF 3, O, O, OMe], [AI313; Me, H, Me, H, O, H, H, H, H, H, O, O, OMe], [AI 314; Me, H, Me, H, O, H, H, H, F, O, O, OMe], [AI 315; Me, H, Me, H, O, H, H, H, H, Cl, O, O, OMe], [AI 316; Me, H, Me, H, O, H, H, H, Br, O, O, OMe] , [AI 317; Me, H, Me, H, O, H, H, H, I, O, O, OMe], [AI 318; Me, H, Me, H, O, H, H, H, Me, O, O, OMe], [AI 319; Me, H, Me, H, O, H, H, H, Et, O, O, OMe], [AI 320; Me, H, Me, H, O, H, H, H, c-Pr, O, O, OMe], [AI 321; Me, H, Me, H, O, H, H, H, OMe, O, O, OMe], [AI 322; Me, H, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 323; Me, H, Me, H, O, H, H, S, Me, O, O, OMe], [ AI324; Me, H, Me, H, O, H, H, H, CF 3, O, O, OMe], [AI325; Et, H, Me, H, O, H, H, H, H, O , O, OMe], [AI 326; Et, H, Me, H, O, H, H, H, H, F, O, O, OMe], [AI 327; Et, H, Me, H, O, H, H , H, Cl, O, O, OMe], [AI 328; Et, H, Me, H, O, H, H, H, Br, O, O, OMe], [AI 329; Et, H, Me, H, O, H, H, H, I, O, O, OMe], [AI 330; Et, H, Me, H, O, H, H, H, Me, O, O, OMe], [AI 331; Et, H, Me, H, O, H, H, H, H, Et, O, O, OMe], [AI 332; Et, H, Me, H, O, H, H, H, c-Pr, O, O, OMe], [AI 333; Et, H, Me, H, O, H, H, H, H, OMe, O, O, OMe], [AI 334; Et, H, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 335; Et, H, Me, H, O, H, H, H, SMe, O, O, OMe], [AI 336; Et, H, Me, H, O, H, H, H, H, CF ₃ , O, O, OMe], [AI 337; CF ₃ , H, Me, H, O, H, H, H, H, O, O, OMe], [AI 338; CF ₃ , H, Me, H , O, H, H, H , F, O, O, OMe], [AI339; CF 3, H, Me, H, O, H, H, H, Cl, O, O, OMe], [AI340; _{CF 3, H, Me, H} , O, H, H, H, Br, O, O, OMe], [AI341; CF 3, H, Me, H, O, H, H, H, I, O, O, OMe], [AI 342; CF ₃ , H, Me, H, O, H, H, H, Me, O, O, OMe], [AI 343: CF ₃ , H, Me, H, O, H, H, H, Et, O, O, OMe], [AI344; CF 3, H, Me, H, O, H, H, H, c-Pr, O, O, OMe], [AI345; CF 3, H, Me, H, O, H, H, H, OMe, O, O, OMe], [AI346; CF 3, H, Me, H, O, H, H, H, OEt, O, O, OMe _{], [AI347; CF 3,} H, Me, H, O, H, H, H, SMe, O, O, OMe], [AI348; CF 3, H, Me, H, O, H, H, H , CF ₃ , O, O, OMe], [AI 349; H, H, Et, H, O, H, H, H, H, O, O, OMe], [AI 350; H, H, Et, H, O, H, H, H, H, F, O, O, OMe], [AI 351; H, H, Et, H, O, H, H, H, Cl, O, O, OMe], [AI 352; H, H, Et, H, O, H, H, H, H, Br, O, O, OMe], [AI 353; H, H, Et, H, O, H, H, H, I, I, O, O, OMe], [AI 354; H, H, Et, H, O, H, H, H, Me, O, O, OMe], [AI 355; H, H, Et, H, O, H, H, H, Et, O, O, OMe], [AI 356; H, H, Et, H, O, H, H, H, c, Pr, O, O, OMe], [AI 357; H, H, Et, H, O, H, H, H, H, OMe, O, O, OMe], [AI 358; H, H, Et, H, O, H, H, H, OEt, O, O, OMe], [ AI 359; H, H, Et, H, O, H, H, H, SMe, O, O, OMe], [AI 360; H, H, Et, H, O, H, H, H, CF ₃ , O , O, OMe], [AI 361; F, H, Et, H, O, H, H, H, H, O, O, OMe], [AI 362; F, H, Et, H, O, H, H , H, F, O, O, OMe], [AI 363; F, H, Et, H, O, H, H, H, H, Cl, O, O, OMe], [AI 364; F, H, Et, H , O, H, H, H, H, Br, O, O, OMe], [AI 365; F, H, Et, H, O, H, H, H, I, O, O, OMe], [AI 366; F , H, Et, H, O, H, H, H, Me, O, O, OMe], [AI 367; F, H, Et, H, O, H, H, H, Et, O, O, OMe ], [AI 368; F, H, Et, H, O, H, H, H, c, Pr, O, O, OMe], [AI 369; F, H, Et, H, O, H, H, H , OMe, O, O, OMe], [AI 370; F, H, Et, H, O, H, H, H, H, OEt, O, O, OMe], [AI 371; F, H, Et, H, O , H, H, H, SMe , O, O, OMe], [AI372; F, H, Et, H, O, H, H, H, CF 3, O, O, OMe], [AI373; Cl, H, Et, H, O, H, H, H, H, H, O, O, OMe], [AI 374; Cl, H, Et, H, O, H, H, H, F, O, O, OMe] [AI 375; Cl, H, Et, H, O, H, H, H, Cl, O, O, OMe], [AI 376; Cl, H, Et, H, O, H, H, H, Br, O, O, OMe], [AI 377; Cl, H, Et, H, O, H, H, H, I, O, O, OMe], [AI 378; Cl, H, Et, H, O, H, H, H, Me, O, O, OMe], [AI 379; Cl, H, Et, H, O, H, H, H, H, Et, O, O, OMe], [AI 380; Cl, H, Et, H, O, H, H, H, c-Pr, O, O, OMe] , [AI 381; Cl, H, Et, H, O, H, H, OMe, O, O, OMe], [AI 382; Cl, H, Et, H, O, H, H, H, OE t, O, O, OMe], [AI 383; Cl, H, Et, H, O, H, H, H, SMe, O, O, OMe], [AI 384; Cl, H, Et, H, O, H, _{H, H, CF 3, O} , O, OMe], [AI385; Br, H, Et, H, O, H, H, H, H, O, O, OMe], [AI386; Br, H, Et , H, O, H, H, H, H, F, O, O, OMe], [AI 387; Br, H, Et, H, O, H, H, H, Cl, O, O, OMe], [AI 388] Br, H, Et, H, O, H, H, H, H, Br, O, O, OMe], [AI 389; Br, H, Et, H, O, H, H, H, I, O, O; , OMe], [AI390; Br, H, Et, H, O, H, H, H, Me, O, O, OMe], [AI 391; Br, H, Et, H, O, H, H, H , Et, O, O, OMe], [AI 392; Br, H, Et, H, O, H, H, H, c, Pr, O, O, OMe], [AI 393; Br, H, Et, H , O, H, H, H, H, OMe, O, O, OMe], [AI 394; Br, H, Et, H, O, H, H, H, OEt, O, O, OMe], [AI 395; Br , H, Et, H, O , H, H, H, SMe, O, O, OMe], [AI396; Br, H, Et, H, O, H, H, H, CF 3, O, O, OMe], [AI 397; Me, H, Et, H, O, H, H, H, H, H, O, O, OMe], [AI 398; Me, H, Et, H, O, H, H, H, H, F, O, O, OMe], [AI 399; Me, H, Et, H, O, H, H, H, H, Cl, O, O, OMe], [AI 400; Me, H, Et, H, O, H, H, H, Br, O, O, OMe],

[AI 401; Me, H, Et, H, O, H, H, H, I, O, O, OMe], [AI 402; Me, H, Et, H, O, H, H, H, Me, O , O, OMe], [AI 403; Me, H, Et, H, O, H, H, H, Et, O, O, OMe], [AI 404; Me, H, Et, H, O, H, H , H, c-Pr, O, O, OMe], [AI 405; Me, H, Et, H, O, H, H, H, OMe, O, O, OMe], [AI 406; Me, H, Et , H, O, H, H, H, H, OEt, O, O, OMe], [AI 407; Me, H, Et, H, O, H, H, H, SMe, O, O, OMe], [AI 408 ; Me, H, Et, H , O, H, H, H, CF 3, O, O, OMe], [AI409; Et, H, Et, H, O, H, H, H, H, O, O, OMe], [AI 410; Et, H, Et, H, O, H, H, H, H, F, O, O, OMe], [AI 411; Et, H, Et, H, O, H, H, H, H, Cl, O, O, OMe], [AI 412; Et, H, Et, H, O, H, H, H, H, Br, O, O, OMe], [AI 413; Et, H, Et, H, O, H, H, H, H, I, O, O, OMe], [AI 414; Et, H, Et, H, O, H, H, H, Me, O, O, OMe], [AI 415; Et, H, Et, H, O, H, H, H, H, Et, O, O, OMe], [AI 416; Et, H, Et, H, O, H, H, H, c-Pr, O, O, OMe], [AI 417; Et, H, Et, H, O, H, H, H, OMe, O, O, OMe], [AI 418; Et, H, Et, H, O, H, H, H, H, OEt, O, O, OMe], [AI 419; Et, H, Et, H, O, H, H, H, S, Me, O, O, OMe], [AI 420; Et, H, Et, H, O, _{H, H, H, CF 3} , O, O, OMe], [AI421; CF 3, H, Et, H, O, H, H, H, H, O, O, OMe], [AI422; CF 3 , H, Et, H, O , H, H, H, F, O, O, OMe], [AI423; CF 3, H, Et, H, O, H, H, H, Cl, O, O, _{OMe], [AI424; CF 3} , H, Et, H, O, H, H, H, Br, O, O, OMe], [AI425; CF 3, H, Et, H, O, H, H, H, I, O, O, OMe], [AI426; CF 3, H, Et, H, O, H, H, H, Me, O, O, OMe], [AI427; CF 3 , H, Et, H, O , H, H, H, Et, O, O, OMe], [AI428; CF 3, H, Et, H, O, H, H, H, c-Pr, O, O, OMe], [AI429; CF 3, H, Et, H, O, H, H, H, OMe, O, O, OMe], [AI430; CF 3, H, Et, H, O, H, H, H, OEt, O, O, OMe], [AI431; CF 3, H, Et, H, O, H, H, H, SMe, O, O, OMe], [AI432; CF 3, H, Et, H, O, H, H, H, CF 3, O, O, OMe], [AI433; H, H, CF 3, H, O, H, H, H, H, O, O, OMe] , [AI434; H, H, CF 3, H, O, H, H, H, F, O, O, OMe], [AI435; H, H, CF 3, H, O, H, H, H, Cl, O, O, OMe] , [AI436; H, H, CF 3, H, O, H, H, H, Br, O, O, OMe], [AI437; H, H, CF 3, H, O, H, H, H, I, O, O, OMe], [AI438; H, H, CF 3, H, O, H, H, H, Me, O, O, OMe], [AI439; H _{, H, CF 3, H,} O, H, H, H, Et, O, O, OMe], [AI440; H, H, CF 3, H, O, H, H, H, c-Pr, O , O, OMe], [AI441 ; H, H, CF 3, H, O, H, H, H, OMe, O, O, OMe], [AI442; H, H, CF 3, H, O, H , H, H, OEt, O , O, OMe], [AI443; H, H, CF 3, H, O, H, H, H, SMe, O, O, OMe], [AI444; H, H, _{CF 3, H, O, H} , H, H, CF 3, O, O, OMe], [AI445; F, H, CF 3, H, O, H, H, H, H, O, O, OMe ], [AI446; F, H , CF 3, H, O, H, H, H, F, O, O, OMe], [AI447; F, H, CF 3, H, O, H, H, H , Cl, O, O, OMe ], [AI448; F, H, CF 3, H, O, H, H, H, Br, O, O, OMe], [AI449; F, H, CF 3, H , O, H, H, H , I, O, O, OMe], [AI450; F, H, CF 3, H, O, H, H, H, Me, O, O, OMe], [AI451; _{F, H, CF 3, H} , O, H, H, H, Et, O, O, OMe], [AI452; F, H, CF 3, H, O , H, H, H, c -Pr, O, O, OMe], [AI453; F, H, CF 3, H, O, H, H, H, OMe, O, O, OMe], [AI454; _{F, H, CF 3, H} , O, H, H, H, OEt, O, O, OMe], [AI455; F, H, CF 3, H, O, H, H, H, SMe, O, O, OMe], [AI456; F, H, CF 3, H, O, H, H, H, CF 3, O, O, OMe], [AI457; Cl, H, CF 3, H, O, H , H, H, H, O , O, OMe], [AI458; Cl, H, CF 3, H, O, H, H, H, F, O, O, OMe], [AI459; Cl, H, _{CF 3, H, O, H} , H, H, Cl, O, O, OMe], [AI460; Cl, H, CF 3, H, O, H, H, H, Br, O, O, OMe] , [AI461; Cl, H, CF 3, H, O, H, H, H, I, O, O, OMe], [AI462; Cl, H, CF 3, H, O, H, H, H, Me, O, O, OMe] , [AI463; Cl, H, CF 3, H, O, H, H, H, Et, O, O, OMe], [AI464; Cl, H, CF 3, H, O, H, H, H, c-Pr, O, O, OMe], [AI465; Cl, H, CF 3, H, O, H, H, H, OMe, O, O, OMe], [AI466 _{; Cl, H, CF 3,} H, O, H, H, H, OEt, O, O, OMe], [AI467; Cl, H, CF 3, H, O, H, H, H, SMe, O , O, OMe], [AI468 ; Cl, H, CF 3, H, O, H, H, H, CF 3, O, O, OMe], [AI469; Br, H, CF 3, H, O, H, H, H, H, O, O, OMe], [AI470; Br, H, CF 3, H, O, H, H, H, F, O, O, OMe], [AI471; Br, H _{, CF 3, H, O,} H, H, H, Cl, O, O, OMe], [AI472; Br, H, CF 3, H, O, H, H, H, Br, O, O, OMe ], [AI473; Br, H , CF 3, H, O, H, H, H, I, O, O, OMe], [AI474; Br, H, CF 3, H, O, H, H, H , Me, O, O, OMe ], [AI475; Br, H, CF 3, H, O, H, H, H, Et, O, O, OMe], [AI476; Br, H, CF 3, H , O, H, H, H, c, -Pr, O, O, OMe], [AI 477; Br, H, C _{F 3, H, O, H} , H, H, OMe, O, O, OMe], [AI478; Br, H, CF 3, H, O, H, H, H, OEt, O, O, OMe] , [AI479; Br, H, CF 3, H, O, H, H, H, SMe, O, O, OMe], [AI480; Br, H, CF 3, H, O, H, H, H, _{CF 3, O, O, OMe} ], [AI481; Me, H, CF 3, H, O, H, H, H, H, O, O, OMe], [AI482; Me, H, CF 3, H , O, H, H, H , F, O, O, OMe], [AI483; Me, H, CF 3, H, O, H, H, H, Cl, O, O, OMe], [AI484; _{Me, H, CF 3, H} , O, H, H, H, Br, O, O, OMe], [AI485; Me, H, CF 3, H, O, H, H, H, I, O, O, OMe], [AI486; Me, H, CF 3, H, O, H, H, H, Me, O, O, OMe], [AI487; Me, H, CF 3, H, O, H, H, H, Et, O, O, OMe], [AI488; Me, H, CF 3, H, O, H, H, H, c-Pr, O, O, OMe], [AI489; Me, H _{, CF 3, H, O,} H, H, H, OMe, O, O, OMe], [AI490; Me, H, CF 3, H, O, H, H, H, OEt, O, O, OMe ], [AI491; Me, H , CF 3, H, O, H, H, H, SMe, O, O, OMe], [AI492; Me, H, CF 3, H, O, H, H, H , CF ₃ , O, O, OMe], [AI 493; Et, H, CF ₃ , H, CF ₃ , H, O, H, H, H, H, O, O, OMe], [AI 494; Et, H, CF ₃ , H, O, H, H, H, F, O, O, OMe], [AI495; Et, H, CF 3, H, O, H, H, H, Cl, O, O, OMe], [AI496 _{; Et, H, CF 3,} H, O, H, H, H, Br, O, O, OMe], [AI497; Et, H, CF 3, H, O, H, H, H, I, O , O, OMe], [AI498 ; Et, H, CF 3, H, O, H, H, H, Me, O, O, OMe], [AI499; Et, H, CF 3, H, O, H , H, H, Et, O , O, OMe], [AI500; Et, H, CF 3, H, O, H, H, H, c-Pr, O, O, OMe],

[AI501; Et, H, CF 3, H, O, H, H, H, OMe, O, O, OMe], [AI502; Et, H, CF 3, H, O, H, H, H, OEt , O, O, OMe], [AI503; Et, H, CF 3, H, O, H, H, H, SMe, O, O, OMe], [AI504; Et, H, CF 3, H, O , H, H, H, CF 3, O, O, OMe], [AI505; CF 3, H, CF 3, H, O, H, H, H, H, O, O, OMe], [AI506; _{CF 3, H, CF 3,} H, O, H, H, H, F, O, O, OMe], [AI507; CF 3, H, CF 3, H, O, H, H, H, Cl, O, O, OMe], [ AI508; CF 3, H, CF 3, H, O, H, H, H, Br, O, O, OMe], [AI509; CF 3, H, CF 3, H, O, H, H, H, I, O, O, OMe], [AI510; CF 3, H, CF 3, H, O, H, H, H, Me, O, O, OMe], [AI511; _{CF 3, H, CF 3,} H, O, H, H, H, Et, O, O, OMe], [AI512; CF 3, H, CF 3, H, O, H, H, H, c- Pr, O, O, OMe] , [AI513; CF 3, H, CF 3, H, O, H, H, H, OMe, O, O, OMe], [AI514; CF 3, H, CF 3, H, O, H, H, H, OEt, O, O, OMe], [AI515; CF 3, H, CF 3, H, O, H, H, H, SMe, O, O, OMe], [ AI 516; CF ₃ , H, CF ₃ , H, O, H, H, H, CF ₃ , O, O, OMe], [AI 517; H, F, H, H, O, H, H, H, H , O, O, OMe], [AI 518; H, F, H, H, O, H, H, H, H, F, O, O, OMe], [AI 519; H, F, H, H, O, H , H, H, Cl, O, O, OMe], [AI 520; H, F, H, H, O, H, H, H, Br, O, O, OMe], [AI 521; H, F, H , H, O, H, H, H, I, I, O, O, OMe], [AI 522; H, F, H, H, O, H, H, H, Me, O, O, OMe], [AI 523] H, F, H, H, H, O, H, H, H, H, Et, O, O, OMe], [AI 524; H, F, H, H, O, H, H, H, c-Pr, O , O, OMe], [AI 525; H, F, H, H, O, H, H, H, OMe, O, O, OMe ], [AI 526; H, F, H, H, O, H, H, H, OEt, O, O, OMe], [AI 527; H, F, H, H, O, H, H, H, SMe , O, O, OMe], [AI528; H, F, H, H, O, H, H, H, CF 3, O, O, OMe], [AI529; Cl, F, H, H, O, H, H, H, H, H, O, O, OMe], [AI 530; Cl, F, H, H, O, H, H, H, F, O, O, OMe], [AI 531: Cl, F, H, H, O, H, H, H, H, Cl, O, O, OMe], [AI 532; Cl, F, H, H, O, H, H, H, Br, O, O, OMe], [, AI 533; Cl, F, H, H, O, H, H, H, I, O, O, OMe], [AI 534; Cl, F, H, H, O, H, H, H, Me, O, O, OMe], [AI 535; Cl, F, H, H, O, H, H, H, Et, O, O, OMe], [AI 536; Cl, F, H, H, O, H, H, H, c-Pr, O, O, OMe], [AI 537; Cl, F, H, H, O, H, H, H, H, OMe, O, O, OMe], [AI 538; Cl, F, H, H, O, H, H, H, H, OEt, O, O, OMe], [AI 539; Cl, F, H, H, O, H, H, H, SMe, O, O, OMe], [AI 540; Cl, F, H, H, O, H, H, H, CF 3, O, O, OMe], [AI541; Me, F, H, H, O, H, H, H, H, O, O , OMe], [AI 542; Me, F, H, H, O, H, H, H, H, F, O, O, OMe], [AI 543; Me, F, H, H, O, H, H, H , Cl, O, O, OMe], [AI544; Me, F, H, H, O, H, H, H, H, Br, O, O, OMe], [AI 545; Me, F, H, H, O , H, H, H, I, O, O, OMe], [AI 546; Me, F, H, H, O, H, H, H, Me, O, O, OMe], [AI 547; Me, F , H, H, O, H, H, H, Et, O, O, OMe], [AI 548; Me, F, H, H, O, H, H, c, Pr, O, O, OMe Me, F, H, H, O, H, H, H, OMe, O, O, OMe], [AI 550; Me, F, H, H, O, H, H, H, OEt] , O, O, OMe], [AI 551; Me, F, H, H, O, H, H, H, S, S, O, O, OMe], [AI 552: Me, F, H, H, O, H , H, H, CF ₃ , O, O, OMe], [AI 553; Et, F, H, H, O, H, H, H, H, H, H, O, O, OMe], [AI 554; Et, F, H, H, O, H, H, H, F, O, O, OMe], [AI 555; Et, F, H, H, O, H, H, H, H, Cl, O, OMe], [AI 556; Et, F, H, H, O, H, H, H, Br, O, O, OMe], [AI 557; Et, F, H, H, O, H, H, H, I, O, O, OMe], [AI 558; Et, F, H, H, O, H, H, H, H, Me, O, O, OMe], [AI 559; Et, F, H, H, O, H, H, H, H, Et, O, O, OMe], [AI 560; Et, F, H, H, O, H, H, H, H, c-Pr, O, O, OMe], [AI 561; Et, F, H, H, O, H, H, H, OM, O, O, OMe], [AI 562: Et, F, H, H, H, O, H, H, H, H, OEt, O, O, OMe], [AI 563; Et, F, H, H, O, H, H, S, Me, O, O, OMe] , [AI564; Et, F, H, H, O, H, H, H, CF 3, O, O, OMe], [AI565; H, F, F, H, O, H, H, H, H , O, O, OMe], [AI566; H, F, F, H, O, H, H, H, F, O, O, OMe], [AI 567; H, F, F, H, O, H , H, H, Cl, O, O, OMe], [AI 568; H, F, F, H, O, H, H, H, Br, O, O, OMe], [AI 569; H, F, F , H, O, H, H, H, H, I, O, O, OMe], [AI 570; H, F, F, H, O, H, H, H, Me, O, O, OMe], [AI 571] H, F, F, H, O, H, H, H, H, Et, O, O, OMe], [AI 572; H, F, F, H, O, H, H, H, c-Pr, O , O, OMe], [AI 573; H, F, F, H, O, H, H, H, OMe, O, O, OMe], [AI 574; H, F, F, H, O, H, H , H, OEt, O, O, OMe], [AI 575; H, F, F, H, O, H, H, H, SMe, O, O, OMe], [AI 576; H, F, F, H , O, H, H, H , CF 3, O, O, OMe], [AI577; Cl, F, F, H, O, H, H, H, H, O, O, OMe], [AI578; Cl, F, F, H, O, H, H, H, H, F, O, O, OMe], [AI 579; Cl, F, F, H, O, H, H, H, Cl, O, O, O OMe], [AI 580; Cl, F, F, H, O, H, H, H, H, Br, O, O, OMe], [AI 581; Cl, F, F, H, O, H, H, H, I, O, O, OMe], [AI 582; Cl, F, F, H, O, H, H, H, Me, O, O, OMe] [AI 583; Cl, F, F, H, O, H, H, H, Et, O, O, OMe], [AI 584; Cl, F, F, H, O, H, H, H, c- Pr, O, O, OMe], [AI 585; Cl, F, F, H, O, H, H, H, H, OMe, O, O, OMe], [AI 586: Cl, F, F, H, O, H, H, H, H, OEt, O, O, OMe], [AI 587; Cl, F, F, H, O, H, H, H, SMe, O, O, OMe], [AI 588; Cl, F, F, H, O, H, H, H, CF 3, O, O, OMe], [AI589; Me, F, F, H, O, H, H, H, H, O, O, OMe], [AI 590; Me, F, F, H, O, H, H, H, F, O, O, OMe], [AI 591; Me, F, F, H, O, H, H, H, Cl, O , O, OMe], [AI 592; Me, F, F, H, O, H, H, H, H, Br, O, O, OMe], [AI 593; Me, F, F, H, O, H, H , H, I, O, O, OMe], [AI 594; Me, F, F, H, O, H, H, H, Me, O, O, OMe], [AI 595: Me, F, F, H , O, H, H, H, H, Et, O, O, OMe], [AI 596; Me, F, F, H, O, H, H, H, c-Pr, O, O, OMe], [AI 597 Me, F, F, H, O, H, H, H, H, OMe, O, O, OMe], [AI 598; Me, F, F, H, O, H, H, H, OEt, O, O , OMe], [AI599; Me, F, F, H, O, H, H, H, SMe, O, O, OMe], [AI 600; Me, F, F, H, O, H, H, H , CF ₃ , O, O, OMe],

[AI601; Et, F, F, H, O, H, H, H, H, O, O, OMe], [AI 602; Et, F, F, H, O, H, H, H, F, O , O, OMe], [AI 603; Et, F, F, H, O, H, H, H, Cl, O, O, OMe], [AI 604; Et, F, F, H, O, H, H , H, Br, O, O, OMe], [AI 605; Et, F, F, H, O, H, H, H, I, O, O, OMe], [AI 606; Et, F, F, H , O, H, H, H, H, Me, O, O, OMe], [AI 607; Et, F, F, H, O, H, H, H, Et, O, O, OMe], [AI 608; Et , F, F, H, O, H, H, H, c, Pr, O, O, OMe], [AI 609; Et, F, F, H, O, H, H, H, OMe, O, O , OMe], [AI 610; Et, F, F, H, O, H, H, H, OEt, O, O, OMe], [AI 611; Et, F, F, H, O, H, H, H , SMe, O, O, OMe ], [AI612; Et, F, F, H, O, H, H, H, CF 3, O, O, OMe], [AI613; H, F, Cl, H, O, H, H, H, H, H, O, O, OMe], [AI 614; H, F, Cl, H, O, H, H, H, F, O, O, OMe], [AI 615; H, F, Cl, H, O, H, H, H, H, Cl, O, O, OMe], [AI 616; H, F, Cl, H, O, H, H, H, Br, O, O, OMe] [AI 617; H, F, Cl, H, O, H, H, H, I, O, O, OMe], [AI 618; H, F, Cl, H, O, H, H, H, Me, O, O, OMe], [AI 619; H, F, Cl, H, O, H, H, H, Et, O, O, OMe], [AI 620; H, F, Cl, H, O, H, H, H, c-Pr, O, O, OMe], [AI 621; H, F, Cl, H, O, H, H, H, OMe, O, O, OMe], [AI 622; H, F, Cl, H, O, H, H, H, OEt, O, O, OMe], [AI 623; H, F, Cl, H, O, H, H, S, Me, O, O, OMe], [ AI624; H, F, Cl, H, O, H, H, H, CF 3, O, O, OMe], [AI625; Cl, F, Cl, H, O, H, H, H, H, O , O, OMe], [AI 626; Cl, F, Cl, H, O, H, H, H, H, F, O, O, OMe], [AI 627; Cl, F, Cl, H, O, H, H , H, Cl, O, O, OMe], [AI 628; Cl, F, Cl, H, O, H, H, H, H, Br, O, O, OMe], [AI 629; Cl, F, Cl, H, O, H, H, H, I, O, O, OMe], [AI 630; F, Cl, H, O, H, H, H, H, Me, O, O, OMe], [AI 631; Cl, F, Cl, H, O, H, H, H, Et, O, O, OMe] , [AI632; Cl, F, Cl, H, O, H, H, H, c-Pr, O, O, OMe], [AI 633; Cl, F, Cl, H, O, H, H, H, H, OMe, O, O, OMe], [AI 634; Cl, F, Cl, H, O, H, H, H, H, OEt, O, O, OMe], [AI 635; Cl, F, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI636; Cl, F, Cl, H, O, H, H, H, CF 3, O, O, OMe], [AI637; Me, F , Cl, H, O, H, H, H, H, H, O, O, OMe], [AI 638; Me, F, Cl, H, O, H, H, H, F, O, O, OMe], [AI639; Me, F, Cl, H, O, H, H, H, Cl, O, O, OMe], [AI 640; Me, F, Cl, H, O, H, H, H, Br, O , O, OMe], [AI 641; Me, F, Cl, H, O, H, H, H, I, O, O, OMe], [AI 642; Me, F, Cl, H, O, H, H , H, Me, O, O, OMe], [AI643; Me, F, Cl, H, O, H, H, H, Et, O, O, OMe], [AI 644; Me, F, Cl, H , O, H, H, H, c, Pr, O, O, OMe], [AI 645; Me, F, Cl, H, O, H, H, H, OMe, O, O, OMe], [AI 646] Me, F, Cl, H, O, H, H, H, H, OEt, O, O, OMe], [AI 647; Me, F, Cl, H, O, H, H, H, SMe, O, O , OMe], [AI648; Me , F, Cl, H, O, H, H, H, CF 3, O, O, OMe], [AI649; Et, F, Cl, H, O, H, H, H, H, H, O, O, OMe], [AI 650; Et, F, Cl, H, O, H, H, H, H, F, O, O, OMe], [AI 651: Et, F, Cl, H, O, H, H, H, H, Cl, O, O, OMe], [AI 652; Et, F, Cl, H, O, H, H, H, Br, O, O, OMe], [AI 653; Et, F, Cl, H, O, H, H, H, I, O, O, OMe], [AI 654; Et, F, Cl, H, O, H, H, H, Me, O, O, OMe] , [AI 655; Et , F, Cl, H, O, H, H, H, H, Et, O, O, OMe], [AI 656; Et, F, Cl, H, O, H, H, H, c-Pr, O, O , OMe], [AI 657; Et, F, Cl, H, O, H, H, H, OMe, O, O, OMe], [AI 658; Et, F, Cl, H, O, H, H, H , OEt, O, O, OMe], [AI 659; Et, F, Cl, H, O, H, H, H, SMe, O, O, OMe], [AI 660; Et, F, Cl, H, O , H, H, H, CF 3, O, O, OMe], [AI661; H, F, Me, H, O, H, H, H, H, O, O, OMe], [AI662; H, F, Me, H, O, H, H, H, H, F, O, O, OMe], [AI 663; H, F, Me, H, O, H, H, H, Cl, O, O, OMe] [AI664; H, F, Me, H, O, H, H, H, Br, O, O, OMe], [AI 665; H, F, Me, H, O, H, H, H, I, I, O, O, OMe], [AI666; H, F, Me, H, O, H, H, H, Me, O, O, OMe], [AI 667; H, F, Me, H, O, H, H, H, Et, O, O, OMe], [AI 668; H, F, Me, H, O, H, H, H, c-Pr, O, O, OMe], [AI 669; H, F, Me, H, O, H, H, H, H, OMe, O, O, OMe], [AI 670; H, F, Me, H, O, H, H, H, OEt, O, O, OMe], [ AI671; H, F, Me, H, O, H, H, H, SMe, O, O, OMe], [AI 672; H, F, Me, H, O, H, H, H, CF ₃ , O , O, OMe], [AI 673; Cl, F, Me, H, O, H, H, H, H, O, O, OMe], [AI 674; Cl, F, Me, H, O, H, H , H, F, O, O, OMe], [AI 675; Cl, F, Me, H, O, H, H, H, H, Cl, O, O, OMe], [AI 676; Cl, F, Me, H , O, H, H, H, H, Br, O, O, OMe], [AI 677; Cl, F, Me, H, O, H, H, H, I, O, O, OMe], [AI 678; Cl , F, Me, H, O, H, H, H, H, Me, O, O, OMe], [AI 679; Cl, F, Me, H, O, H, H, H, Et, O, O, OMe ], [AI 680; Cl, F, Me, H, O, H, H, H, c-Pr, O, O, OMe], [AI 681; Cl, F, Me, H, O, H, H, H] , OMe, O, O, OMe], [AI 682; Cl , F, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 683; Cl, F, Me, H, O, H, H, H, SMe, O, O, OMe ], [AI684; Cl, F , Me, H, O, H, H, H, CF 3, O, O, OMe], [AI685; Me, F, Me, H, O, H, H, H, H, O, O, OMe], [AI 686; Me, F, Me, H, O, H, H, H, H, F, O, O, OMe], [AI 687; Me, F, Me, H, O, H, H, H, H, Cl, O, O, OMe], [AI 688; Me, F, Me, H, O, H, H, H, Br, O, O, OMe], [AI 689: Me, F, Me, H, O, H, H, H, I, I, O, O, OMe], [AI 690; Me, F, Me, H, O, H, H, Me, O, O, OMe], [ AI 691; Me, F, Me, H, O, H, H, H, Et, O, O, OMe], [AI 692; Me, F, Me, H, O, H, H, H, c-Pr, O, O, OMe], [AI693; Me, F, Me, H, O, H, H, H, H, OMe, O, O, OMe], [AI 694; Me, F, Me, H, O, H, H, H, OEt, O, O, OMe], [AI 695; Me, F, Me, H, O, H, H, H, SMe, O, O, OMe], [AI 696; Me, F, Me, H, O, H, H, H, CF 3, O, O, OMe], [AI697; Et, F, Me, H, O, H, H, H, H, O, O, OMe], [AI698 Et, F, Me, H, O, H, H, H, H, F, O, O, OMe], [AI 699; Et, F, Me, H, O, H, H, H, Cl, O, O , OMe], [AI 700; Et, F, Me, H, O, H, H, H, Br, O, O, OMe],

[AI 701; Et, F, Me, H, O, H, H, H, I, O, O, OMe], [AI 702; Et, F, Me, H, O, H, H, H, Me, O , O, OMe], [AI 703; Et, F, Me, H, O, H, H, H, Et, O, O, OMe], [AI 704; Et, F, Me, H, O, H, H , H, c-Pr, O, O, OMe], [AI 705; Et, F, Me, H, O, H, H, H, OMe, O, O, OMe], [AI 706; Et, F, Me , H, O, H, H, H, H, OEt, O, O, OMe], [AI 707; Et, F, Me, H, O, H, H, H, SMe, O, O, OMe], [AI 708] ; Et, F, Me, H , O, H, H, H, CF 3, O, O, OMe], [AI709; H, F, Et, H, O, H, H, H, H, O, O, OMe], [AI 710; H, F, Et, H, O, H, H, H, F, O, O, OMe], [AI 711; H, F, Et, H, O, H, H, H, Cl, O, O, OMe], [AI 712; H, F, Et, H, O, H, H, H, H, Br, O, O, OMe], [AI 713; H, F, Et, H, O, H, H, H, H, I, O, O, OMe], [AI 714; H, F, Et, H, O, H, H, H, Me, O, O, OMe], [AI 715; H, F, Et, H, O, H, H, H, H, Et, O, O, OMe], [AI 716; H, F, Et, H, O, H, H, H, c-Pr, O, O, OMe], [AI717; H, F, Et, H, O, H, H, H, OMe, O, O, OMe], [AI 718; H, F, Et, H, O, H, H, H, OEt, O, O, OMe], [AI 719; H, F, Et, H, O, H, H, H, SMe, O, O, OMe], [AI 720; H, F, Et, H, O, _{H, H, H, CF 3} , O, O, OMe], [AI721; Cl, F, Et, H, O, H, H, H, H, O, O, OMe], [AI722; Cl, F , Et, H, O, H, H, H, H, F, O, O, OMe], [AI 723; Cl, F, Et, H, O, H, H, H, Cl, O, O, OMe], [AI 724; Cl, F, Et, H, O, H, H, H, Br, O, O, OMe], [AI 725; Cl, F, Et, H, O, H, H, H, I, O , O, OMe], [AI 726; Cl, F, Et, H, O, H, H, H, Me, O, O, OMe], [AI 727; Cl, F, Et, H, O, H, H , H, Et, O, O, OMe], [AI 7 28; Cl, F, Et, H, O, H, H, H, c, Pr, O, O, OMe], [AI 729; Cl, F, Et, H, O, H, H, H, OMe, O, O, OMe], [AI 730; Cl, F, Et, H, O, H, H, H, H, OEt, O, O, OMe], [AI 731; Cl, F, Et, H, O, H, H, H, SMe, O, O, OMe], [AI732; Cl, F, Et, H, O, H, H, H, CF 3, O, O, OMe], [AI733; Me, F, Et , H, O, H, H, H, H, H, O, O, OMe], [AI 734; Me, F, Et, H, O, H, H, H, F, O, O, OMe], [AI 735] Me, F, Et, H, O, H, H, H, H, Cl, O, OMe], [AI 736; Me, F, Et, H, O, H, H, H, Br, O, O , OMe], [AI 737; Me, F, Et, H, O, H, H, H, I, O, O, OMe], [AI 738; Me, F, Et, H, O, H, H, H Me, O, O, OMe], [AI 739; Me, F, Et, H, O, H, H, H, H, Et, O, O, OMe], [AI 740; Me, F, Et, H, O , H, H, H, c-Pr, O, O, OMe], [AI 741; Me, F, Et, H, O, H, H, H, OMe, O, O, OMe], [AI 742; Me , F, Et, H, O, H, H, H, H, OEt, O, O, OMe], [AI 743; Me, F, Et, H, O, H, H, H, SMe, O, O, OMe ], [AI744; Me, F , Et, H, O, H, H, H, CF 3, O, O, OMe], [AI745; Et, F, Et, H, O, H, H, H, H, O, O, OMe], [AI746; Et, F, Et, H, O, H, H, H, H, F, O, O, OMe], [AI 747; Et, F, Et, H, O, H, H, H, H, Cl, O, O, OMe], [AI 748; Et, F, Et, H, O, H, H, H, Br, O, O, OMe], [AI 749; Et, F, Et, H, O, H, H, H, I, O, O, OMe], [AI 750; Et, F, Et, H, O, H, H, Me, O, O, OMe], [AI 750; AI 751: Et, F, Et, H, O, H, H, H, Et, O, O, OMe], [AI 752; Et, F, Et, H, O, H, H, H, c-Pr, O, O, OMe], [AI 753; Et, F, Et, H, O, H, H, H, H, OMe, O, O, OMe], [AI 754; Et, F, Et, H, O, H, H, H, OEt, O, O, OMe], [AI 755; Et, F, Et, H, O, H, H, H, S Me, O, O, OMe], [AI 756; Et, F, Et, H, O, H, _{H, H, CF 3, O} , O, OMe], [AI757; H, H, H, F, O, H, H, H, H, O, O, OMe], [AI758; H, H, H , F, O, H, H, H, F, O, O, OMe], [AI 759; H, H, H, H, F, O, H, H, H, Cl, O, O, OMe], [AI 760] H, H, H, H, F, O, H, H, H, H, Br, O, O, OMe], [AI 761; H, H, H, H, F, O, H, H, H, I, O, O , OMe], [AI762; H, H, H, F, O, H, H, Me, O, O, OMe], [AI 763; H, H, H, F, O, H, H, H , Et, O, O, OMe], [AI764; H, H, H, F, O, H, H, H, c-Pr, O, O, OMe], [AI 765; H, H, H, F , O, H, H, H, H, OMe, O, O, OMe], [AI766; H, H, H, H, F, O, H, H, H, OEt, O, O, OMe], [AI 767; H , H, H, F, O , H, H, H, SMe, O, O, OMe], [AI768; H, H, H, F, O, H, H, H, CF 3, O, O, OMe], [AI 769; Cl, H, H, F, O, H, H, H, H, O, O, OMe], [AI 770; Cl, H, H, F, O, H, H, H, F, O, O, OMe], [AI 771; Cl, H, H, F, O, H, H, H, Cl, O, O, OMe], [AI 772; Cl, H, H, F, O, H, H, H, H, Br, O, O, OMe], [AI 773; Cl, H, H, F, O, H, H, H, I, O, O, OMe], [AI 774; Cl, H, H, F, O, H, H, H, Me, O, O, OMe], [AI 775; Cl, H, H, F, O, H, H, Et, O, O, OMe], [ AI 776; Cl, H, H, F, O, H, H, c, Pr, O, O, OMe], [AI 777; Cl, H, H, F, O, H, H, H, OMe, O, O, OMe], [AI 778; Cl, H, H, F, O, H, H, H, OEt, O, O, OMe], [AI 779; Cl, H, H, F, O, H, H, H, SMe, O, O, OMe], [AI780; Cl, H, H, F, O, H, H, H, CF 3, O, O, OMe], [AI781; Me, H, H , F, O, H, H, H, H, H, O, O, OMe], [AI 782; Me, H, H, F, O, H, H, H, H, F, O, O, OMe], [AI 783; Me, H, H, F, O, H, H, H, Cl, O, O, OMe], [AI 784; H, H, F, O, H, H, H, H, Br, O, O, OMe], [AI 785; Me, H, H, F, O, H, H, I, O, O, OMe] , [AI 786; Me, H, H, F, O, H, H, Me, O, O, OMe], [AI 787; Me, H, H, F, O, H, H, H, Et, O, O, OMe], [AI 788; Me, H, H, F, O, H, H, H, c-Pr, O, O, OMe], [AI 789; Me, H, H, F, O, H, H, H, H, OMe, O, O, OMe], [AI 790; Me, H, H, F, O, H, H, H, OE, O, O, OMe], [AI 791; Me, H, H, F, O, H, H, H, SMe, O, O, OMe], [AI792; Me, H, H, F, O, H, H, H, CF 3, O, O, OMe], [AI793; Et, H, H, F, O, H, H, H, H, O, O, OMe], [AI 794; Et, H, H, F, O, H, H, H, F, O , O, OMe], [AI 795; Et, H, H, F, O, H, H, H, Cl, O, OMe], [AI 796; Et, H, H, F, O, H, H H, Br, O, O, OMe], [AI 797; Et, H, H, H, F, O, H, H, H, I, O, O, OMe], [AI 798; Et, H, H, F , O, H, H, H, H, Me, O, O, OMe], [AI 799; Et, H, H, H, F, O, H, H, H, Et, O, O, OMe], [AI 800; , H, H, F, O, H, H, H, c-Pr, O, O, OMe],

[AI801; Et, H, H, F, O, H, H, OMe, O, O, OMe], [AI 802; Et, H, H, F, O, H, H, H, OEt, O , O, OMe], [AI 803; Et, H, H, F, O, H, H, S, S, O, O, OMe], [AI 804; Et, H, H, F, O, H, H _{, H, CF 3, O,} O, OMe], [AI805; H, H, F, F, O, H, H, H, H, O, O, OMe], [AI806; H, H, F, F, O, H, H, H, F, O, O, OMe], [AI 807; H, H, F, F, O, H, H, H, Cl, O, O, OMe], [AI 808; H, H, F, F, O, H, H, H, H, Br, O, O, OMe], [AI 809; H, H, F, F, O, H, H, I, O, O, OMe], [AI 810; H, H, F, F, O, H, H, Me, O, O, OMe], [AI 811; H, H, F, F, O, H, H, H, Et, O, O, OMe], [AI 812; H, H, F, F, O, H, H, H, c-Pr, O, O, OMe], [AI 813; H, H, F, F, O, H, H, H, H, OMe, O, O, OMe], [AI 814; H, H, F, F, O, H, H, H, OE t, O, O, OMe], [AI 815; H, F, F, O, H, H, H, SMe, O, O, OMe], [AI816; H, H, F, F, O, H, H, H, CF 3, O, O, OMe ], [AI 817; Cl, H, F, F, O, H, H, H, H, O, O, OMe], [AI 818; Cl, H, F, F, O, H, H, H, F] , O, O, OMe], [AI 819; Cl, H, F, F, O, H, H, H, Cl, O, OMe], [AI 820; Cl, H, F, F, O, H , H, H, Br, O, O, OMe], [AI 821; Cl, H, F, F, O, H, H, H, I, O, O, OMe], [AI 822; Cl, H, F , F, O, H, H, H, H, Me, O, O, OMe], [AI 823; Cl, H, F, F, O, H, H, H, Et, O, O, OMe], [AI 824] Cl, H, F, F, O, H, H, H, c, Pr, O, O, OMe], [AI 825; Cl, H, F, F, O, H, H, H, OMe, O , O, OMe], [AI 826; Cl, H, F, F, O, H, H, OEt, O, O, OMe], [AI 827; Cl, H, F, F, O, H, H , H, SMe, O, O, OMe], [AI 828; Cl, H, F, F, O, H, H, H, CF ₃ , O, O, OMe], [AI 829; Me, H, F, F, O, H, H, H, H, O, O, OMe], [AI 830; Me, H, F, F, O, H, H, H, H, F, O, O, OMe], [AI 831; Me, H, F, F, O, H, H, H, Cl, O, OMe], [AI 832: Me, H, F, F, O, H, H, H, H, Br, O, O, OMe], [AI 833; Me, H, F, F, O, H, H, I, O, O, OMe], [, AI 834; Me, H, F, F, O, H, H, Me, O, O, OMe], [AI 835; Me, H, F, F, O, H, H, H, Et, O, O, OMe], [AI 836; Me, H, F, F, O, H, H, c, Pr, O, O, OMe], [AI 837; Me, H, F, F, O, H, H, H, OMe, O, O, OMe], [AI 838; Me, H, F, F, O, H, H, H, OEt, O, O, OMe], [AI 839; Me, H, F, F, O, H, H, H, SMe, O, O, OMe], [AI840; Me, H, F, F, O, H, H, H, CF 3, O, O, OMe], [AI841 Et, H, F, F, O, H, H, H, H, H, O, O, OMe], [AI 842; Et, H, F, F, O, H, H, H, F, O, O; , OMe], [AI 843; Et, H, F, F, O, H, H, H, Cl, O, O, OMe], [AI 844; Et, H, F, F, O, H, H, H , Br, O, O, OMe], [AI 845; Et, H, F, F, O, H, H, H, I, O, O, OMe], [AI 846; Et, H, F, F, O , H, H, H, Me, O, O, OMe], [AI 847; Et, H, F, F, O, H, H, H, Et, O, O, OMe], [AI 848; Et, H , F, F, O, H, H, H, c, Pr, O, O, OMe], [AI 849; Et, H, F, F, O, H, H, H, OMe, O, O, OMe ], [AI 850; Et, H, F, F, O, H, H, H, OEt, O, O, OMe], [AI 851; Et, H, F, F, O, H, H, H, SMe] , O, O, OMe], [AI852; Et, H, F, F, O, H, H, H, CF 3, O, O, OMe], [AI853; H, H, Cl, F, O, H, H, H, H, H, O, O, OMe], [AI 854; H, H, Cl, F, O, H, H, H, F, O, O, OMe], [AI 855; H, H, Cl, F, O, H, H, H, H, Cl, O, O, OMe], [AI 856; H H, Cl, F, O, H, H, H, H, Br, O, O, OMe], [AI 857; H, H, Cl, F, O, H, H, I, O, O, OMe ], [AI 858; H, H, Cl, F, O, H, H, Me, O, O, OMe], [AI 859; H, H, Cl, F, O, H, H, H, Et] , O, O, OMe], [AI 860; H, H, Cl, F, O, H, H, H, c-Pr, O, O, OMe], [AI 861; H, H, Cl, F, O H, H, H, H, OMe, O, O, OMe], [AI 862; H, H, Cl, F, O, H, H, H, OE t, O, O, OMe], [AI 863; H, H , Cl, F, O, H , H, H, SMe, O, O, OMe], [AI864; H, H, Cl, F, O, H, H, H, CF 3, O, O, OMe] , [AI 865; Cl, H, Cl, F, O, H, H, H, H, O, O, OMe], [AI 866; Cl, H, Cl, F, O, H, H, H, F, O, O, OMe], [AI 867; Cl, H, Cl, F, O, H, H, H, Cl, O, OMe], [AI 868; Cl, H, Cl, F, O, H, H, H, Br, O, O, OMe], [AI 869; Cl, H, Cl, F, O, H, H, H, I, O, O, OMe], [AI 870; Cl, H, Cl, F, O, H, H, H, H, Me, O, O, OMe], [AI 871; Cl, H, Cl, F, O, H, H, H, Et, O, O, OMe], [AI 872; Cl, H, Cl, F, O, H, H, H, c, Pr, O, O, OMe], [AI 873; Cl, H, Cl, F, O, H, H, H, OMe, O, O, O, OMe], [AI 874; Cl, H, Cl, F, O, H, H, OEt, O, O, OMe], [AI 875; Cl, H, Cl, F, O, H, H, H, SMe, O, O, OMe], [AI876; Cl, H, Cl, F, O, H, H, H, CF 3, O, O, OMe], [AI877; Me, H, Cl, F , O, H, H, H, H, H, O, O, OMe], [AI 878; Me, H, Cl, F, O, H, H, H, F, O, O, OMe], [AI 879; , H, Cl, F, O, H, H, H, H, Cl, O, O, OMe], [AI 880; Me, H, Cl, F, O, H, H, H, Br, O, O, OMe Me, H, Cl, F, O, H, H, I, O, O, OMe], [AI 882; Me, H, Cl, F, O, H, H, H, Me] , O, O, OMe], [AI 883; Me , H, Cl, F, O, H, H, H, Et, O, O, OMe], [AI 884; Me, H, Cl, F, O, H, H, H, c-Pr, O, O , OMe], [AI885; Me, H, Cl, F, O, H, H, OMe, O, O, OMe], [AI 886; Me, H, Cl, F, O, H, H, H , OEt, O, O, OMe], [AI 887; Me, H, Cl, F, O, H, H, H, SMe, O, O, OMe], [AI 888; Me, H, Cl, F, O , H, H, H, CF 3, O, O, OMe], [AI889; Et, H, Cl, F, O, H, H, H, H, O, O, OMe], [AI890; Et, H, Cl, F, O, H, H, H, H, F, O, O, OMe], [AI891; Et, H, Cl, F, O, H, H, H, Cl, O, O, OMe] [AI 892; Et, H, Cl, F, O, H, H, H, Br, O, O, OMe], [AI 893; Et, H, Cl, F, O, H, H, H, I, O, O, OMe], [AI 894; Et, H, Cl, F, O, H, H, Me, O, O, OMe], [AI 895; Et, H, Cl, F, O, H, H, H, Et, O, O, OMe], [AI 896; Et, H, Cl, F, O, H, H, H, c-Pr, O, O, OMe], [AI 897; Et, H, Cl, F, O, H, H, H, H, OMe, O, O, OMe], [AI 898; Et, H, Cl, F, O, H, H, H, OEt, O, O, OMe], [ AI 899; Et, H, Cl, F, O, H, H, H, S Me, O, O, OMe], [AI 900; Et, H, Cl, F, O, H, H, H, CF ₃ , O , O, OMe],

[AI 901; H, H, Me, F, O, H, H, H, O, O, OMe], [AI 902; H, H, Me, F, O, H, H, H, F, O , O, OMe], [AI 903; H, H, Me, F, O, H, H, Cl, O, OMe], [AI 904; H, H, Me, F, O, H, H , H, Br, O, O, OMe], [AI 905; H, H, Me, F, O, H, H, H, I, O, O, OMe], [AI 906; H, H, Me, F , O, H, H, H, Me, O, O, OMe], [AI 907; H, H, Me, F, O, H, H, H, Et, O, O, OMe], [AI 908; H , H, Me, F, O, H, H, H, c, Pr, O, O, OMe], [AI 909; H, H, Me, F, O, H, H, H, OMe, O, O , OMe], [AI 910; H, H, Me, F, O, H, H, H, OEt, O, O, OMe], [AI 911; H, H, Me, F, O, H, H, H , SMe, O, O, OMe ], [AI912; H, H, Me, F, O, H, H, H, CF 3, O, O, OMe], [AI913; Cl, H, Me, F, O, H, H, H, H, H, O, O, OMe], [AI 914; Cl, H, Me, F, O, H, H, H, F, O, O, OMe], [AI 915; Cl, H, Me, F, O, H, H, H, H, Cl, O, O, OMe], [AI 916; Cl, H, Me, F, O, H, H, H, Br, O, O, OMe] , [AI 917; Cl, H, Me, F, O, H, H, I, O, O, OMe], [AI 918; Cl, H, Me, F, O, H, H, H, Me, O, O, OMe], [AI 919; Cl, H, Me, F, O, H, H, Et, O, O, OMe], [AI 920; Cl, H, Me, F, O, H, H, H, c-Pr, O, O, OMe], [AI 921; Cl, H, Me, F, O, H, H, H, OMe, O, O, OMe], [AI 922; Cl, H, Me, F, O, H, H, H, OEt, O, O, OMe], [AI 923; Cl, H, Me, F, O, H, H, S, Me, O, O, OMe], [ AI924; Cl, H, Me, F, O, H, H, H, CF 3, O, O, OMe], [AI925; Me, H, Me, F, O, H, H, H, H, O , O, OMe], [AI 926; Me, H, Me, F, O, H, H, H, F, O, O, OMe], [AI 927; Me, H, Me, F, O, H, H , H, Cl, O, O, OMe], [AI 92 8; Me, H, Me, F, O, H, H, H, H, Br, O, O, OMe], [AI 929; Me, H, Me, F, O, H, H, H, I, O, O, OMe], [AI 930; Me, H, Me, F, O, H, H, Me, O, O, OMe], [AI 931; Me, H, Me, F, O, H, H, H, Et, O, O, OMe], [AI 932; Me, H, Me, F, O, H, H, H, c-Pr, O, O, OMe], [AI 933; Me, H, Me, F, O, H, H, H, H, OMe, O, O, OMe], [AI 934; Me, H, Me, F, O, H, H, H, OEt, O, O, OMe], [AI 935; Me, H, Me, F, O, H, H, H, SMe, O, O, OMe], [AI 936; Me, H, Me, F, O, H, H, H, CF ₃ , O, O , OMe], [AI 937; Et, H, Me, F, O, H, H, H, H, O, O, OMe], [AI 938; Et, H, Me, F, O, H, H, H , F, O, O, OMe], [AI 939; Et, H, Me, F, O, H, H, H, Cl, O, O, OMe], [AI 940; Et, H, Me, F, O , H, H, H, H, Br, O, O, OMe], [AI 941; Et, H, Me, F, O, H, H, H, I, O, O, OMe], [AI 942; Et, H , Me, F, O, H, H, H, Me, O, O, OMe], [AI 943; Et, H, Me, F, O, H, H, H, Et, O, O, OMe], [AI 944; Et, H, Me, F, O, H, H, H, c-Pr, O, O, OMe], [AI 945; Et, H, Me, F, O, H, H, H, OMe , O, O, OMe], [AI 946; Et, H, Me, F, O, H, H, H, OEt, O, O, OMe], [AI 947; Et, H, Me, F, O, H , H, H, SMe, O , O, OMe], [AI948; Et, H, Me, F, O, H, H, H, CF 3, O, O, OMe], [AI949; H, H, Et, F, O, H, H, H, H, H, O, O, OMe], [AI 950; H, H, Et, F, O, H, H, F, O, O, OMe], [AI 950; AI 951; H, H, Et, F, O, H, H, H, Cl, O, OMe], [AI 952; H, H, Et, F, O, H, H, H, Br, O, H, H, Et, F, O, H, H, H, I, O, O, OMe], [AI 954; H, H, Et, F, O, H, H, O, OMe], [AI953; H, Me, O, O, OMe], [AI 955; H, H, Et, F, O, H, H, H, Et, O, O, OMe], [AI956; H, H, Et, F, O, H, H, H, c-Pr, O, O, OMe], [AI957; H, H, Et, F, O, H, H, OMe, O, O, OMe], [AI 958; H, H, Et, F, O, H, H, H, OEt, O, O, OMe], [AI 959; H, H, Et, F, O, H, H, S, O, O, OMe], [AI 960; H, H, Et, F, O, H, H, H, CF 3, O, O, OMe], [AI961; Cl, H, Et, F, O, H, H, H, H, O, O, OMe], [AI962 Cl, H, Et, F, O, H, H, H, H, F, O, O, OMe], [AI963; Cl, H, Et, F, O, H, H, H, Cl, O, O , OMe], [AI964; Cl, H, Et, F, O, H, H, H, Br, O, O, OMe], [AI 965; Cl, H, Et, F, O, H, H, H , I, O, O, OMe], [AI966; Cl, H, Et, F, O, H, H, H, Me, O, O, OMe], [AI 967; Cl, H, Et, F, O , H, H, H, H, Et, O, O, OMe], [AI 968; Cl, H, Et, F, O, H, H, H, c-Pr, O, O, OMe], [AI 969; Cl , H, Et, F, O, H, H, H, OMe, O, O, OMe], [AI 970; Cl, H, Et, F, O, H, H, H, OEt, O, O, OMe ], [AI971; Cl, H, Et, F, O, H, H, SMe, O, O, OMe], [AI 972; Cl, H, Et, F, O, H, H, H, CF] ₃ , O, O, OMe], [AI 973; Me, H, Et, F, O, H, H, H, H, O, O, OMe], [AI 974; Me, H, Et, F, O, H, H, H, H, F, O, O, OMe], [AI 975; Me, H, Et, F, O, H, H, H, Cl, O, O, OMe], [AI 976; Me, H, Et, F, O, H, H, H, H, Br, O, O, OMe], [AI 977; Me, H, Et, F, O, H, H, H, I, O, O, OMe], [ AI 978; Me, H, Et, F, O, H, H, H, Me, O, O, OMe], [AI 979; Me, H, Et, F, O, H, H, H, Et, O, O, OMe], [AI 980; Me, H, Et, F, O, H, H, c, Pr, O, O, OMe], [AI 981; Me, H, Et, F, O, H, H, H, OMe, O, O, OM e], [AI 982, Me, H, Et, F, O, H, H, H, OEt, O, O, OMe], [AI 983; Me, H, Et, F, O, H, H, H, SMe, O, O, OMe] , [AI984; Me, H, Et, F, O, H, H, H, CF 3, O, O, OMe], [AI985; Et, H, Et, F, O , H, H, H, H, H, O, O, OMe], [AI986; Et, H, Et, F, O, H, H, H, F, O, O, OMe], [AI 987; Et, H , Et, F, O, H, H, H, H, Cl, O, O, Oe], [AI 988; Et, H, Et, F, O, H, H, H, Br, O, O, OMe], [AI 989; Et, H, Et, F, O, H, H, H, I, O, O, OMe], [AI 990; Et, H, Et, F, O, H, H, H, Me, O , O, OMe], [AI991; Et, H, Et, F, O, H, H, H, Et, O, O, OMe], [AI992; Et, H, Et, F, O, H, H , H, c-Pr, O, O, OMe], [AI993; Et, H, Et, F, O, H, H, H, OMe, O, O, OMe], [AI994; Et, H, Et , F, O, H, H, H, H, OEt, O, O, OMe], [AI 995; Et, H, Et, F, O, H, H, S Me, O, O, OMe], [AI 996 ; Et, H, Et, F , O, H, H, H, CF 3, O, O, OMe], [AI997; H, H, H, H, O, F, H, H, H, O, O, OMe], [AI 998; H, H, H, H, O, F, H, H, F, O, O, OMe], [AI 999; H, H, H, H, O, F, H, H, Cl, O, O, OMe], [AI 1000; H, H, H, H, H, O, F, H, H, Br, O, O, OMe],

[AI1001; H, H, H, H, H, O, F, H, I, O, O, OMe], [AI 1002; H, H, H, H, O, F, H, H, Me, O , O, OMe], [AI 1003; H, H, H, H, H, O, F, H, Et, O, O, OMe], [AI 1004; H, H, H, H, O, F, H , H, c-Pr, O, O, OMe], [AI 1005; H, H, H, H, H, O, F, H, OMe, O, O, OMe], [AI 1006; H, H, H , H, O, F, H, H, OEt, O, O, OMe], [AI 1007; H, H, H, H, O, F, H, S Me, O, O, OMe], [AI 1008 ; H, H, H, H , O, F, H, H, CF 3, O, O, OMe], [AI1009; Cl, H, H, H, O, F, H, H, H, O, O, OMe], [AI1010; Cl, H, H, H, O, F, H, H, F, O, O, OMe], [AI 1011; Cl, H, H, H, O, F, H, H, Cl, O, O, OMe], [AI1012; Cl, H, H, H, H, O, F, H, H, Br, O, O, OMe], [AI1013; Cl, H, H, H, O, F, H, H, I, O, O, OMe], [AI 1014; Cl, H, H, H, H, O, F, H, Me, O, O, OMe], [AI 1015; Cl, H, H, H, H, O, F, H, H, Et, O, O, OMe], [AI 1016; Cl, H, H, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1017; Cl, H, H, H, O, F, H, H, OMe, O, O, OMe], [AI 1018; Cl, H, H, H, O, F, H, H, H, OEt, O, O, OMe], [AI 1019; Cl, H, H, H, H, O, F, H, SMe, O, O, OMe], [AI 1020; Cl, H, H, H, O, _{F, H, H, CF 3} , O, O, OMe], [AI1021; Me, H, H, H, O, F, H, H, H, O, O, OMe], [AI1022; Me, H , H, H, O, F, H, H, F, O, O, OMe], [AI1023; Me, H, H, H, O, F, H, H, Cl, O, O, OMe], [AI 1024; Me, H, H, H, H, O, F, H, H, Br, O, O, OMe], [AI 1025; Me, H, H, H, O, F, H, H, I, O , O, OMe], [AI 1026; Me, H, H, H, H, O, F, H, Me, O, O, OMe], [AI 1027; Me, H, H, H, O, F, H H, Et, O, O, OMe], [AI 10 28; Me, H, H, H, H, O, F, H, c, Pr, O, O, OMe], [AI 1029; Me, H, H, H, O, F, H, H, OMe , O, O, OMe], [AI 1030; Me, H, H, H, O, F, H, H, OEt, O, O, OMe], [AI 1031; Me, H, H, H, O, F , H, H, SMe, O , O, OMe], [AI1032; Me, H, H, H, O, F, H, H, CF 3, O, O, OMe], [AI1033; Et, H, H, H, O, F, H, H, H, O, O, OMe], [AI 1034; Et, H, H, H, O, F, H, F, O, O, OMe], [A AI 1035; Et, H, H, H, H, O, F, H, H, Cl, O, OMe], [AI 1036; Et, H, H, H, H, O, F, H, H, Br, O, O, OMe], [AI 1037; Et, H, H, H, H, O, F, H, I, O, O, OMe], [AI 1038; Et, H, H, H, O, F, H, H, Me, O, O, OMe], [AI 1039; Et, H, H, H, H, O, F, H, Et, O, O, OMe], [AI 1040; Et, H, H, H, O, F, H, H, c, Pr, O, O, OMe], [AI1041; Et, H, H, H, H, O, F, H, OMe, O, O, OMe], [AI 1042; Et, H, H, H, H, O, F, H, H, OEt, O, O, OMe], [AI1043; Et, H, H, H, H, O, F, H, SMe, O, O, OMe], [AI1044; Et, H, H, H, O, F, H, H, CF 3, O, O, OMe], [AI1045; H, H, F, H, O, F, H, H , H, O, O, OMe], [AI 1046; H, H, F, H, O, F, H, F, O, O, OMe], [AI 1047; H, H, F, H, O , F, H, H, Cl, O, O, OMe], [AI 1048; H, H, F, H, O, F, H, H, Br, O, O, OMe], [AI 1049; H, H , F, H, O, F, H, H, I, O, O, OMe], [AI 1050; H, H, F, H, O, F, H, Me, O, O, OMe], [AI1051; H, H, F, H, O, F, H, H, Et, O, O, OMe], [AI 1052; H, H, F, H, O, F, H, H, c-Pr , O, O, OMe], [AI1053; H, H, F, H, O, F, H, H, OMe, O, O, OMe], [AI 1054; H, H, F, H, O, F , H, H, OEt, O, O, OM e], [AI 1055; H, H, F, H, O, F, H, S Me, O, O, OMe], [AI 1056; H, H, F, H, O, F, H, H, CF ₃ , O, O, OMe], [AI 1057; Cl, H, F, H, O, F, H, H, H, O, O, OMe], [AI 1058; Cl, H, F, H, O , F, H, H, F, O, O, OMe], [AI 1059; Cl, H, F, H, O, F, H, H, Cl, O, O, OMe], [AI 1060; Cl, H , F, H, O, F, H, H, Br, O, O, OMe], [AI 1061; Cl, H, F, H, O, F, H, I, O, O, OMe], [AI1062; Cl, H, F, H, O, F, H, Me, O, O, OMe], [AI 1063; Cl, H, F, H, O, F, H, H, Et, O , O, OMe], [AI1064; Cl, H, F, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1065; Cl, H, F, H, O, F , H, H, OMe, O, O, OMe], [AI 1066; Cl, H, F, H, O, F, H, H, OEt, O, O, OMe], [AI 1067; Cl, H, F , H, O, F, H, H, SMe, O, O, OMe], [AI 1068; Cl, H, F, H, O, F, H, H, CF ₃ , O, O, OMe], [ AI 1069; Me, H, F, H, O, F, H, H, H, O, O, OMe], [AI 1070; Me, H, F, H, O, F, H, H, F, O, O, OMe], [AI 1071; Me, H, F, H, O, F, H, H, Cl, O, OMe], [AI 1072; Me, H, F, H, O, F, H, H, Br, O, O, OMe], [AI1073; Me, H, F, H, O, F, H, I, O, O, OMe], [AI 1074; Me, H, F, H, O, F, H, H, Me, O, O, OMe], [AI 1075; Me, H, F, H, O, F, H, Et, O, O, OMe], [AI 1076; Me, H, F, H, O, F, H, H, c, Pr, O, O, OMe], [AI 1077; Me, H, F, H, O, F, H, OMe, O, O, OMe], [AI1078; Me, H, F, H, O, F, H, H, OEt, O, O, OMe], [AI 1079; Me, H, F, H, O, F, H, H, H, SMe, O, O, OMe] , [AI1080; Me, H, F, H, O, F, H, H, CF 3, O, O, OMe], [AI1081; Et, H, F, H, O , F, H, H, H, O, O, OMe], [AI 1082; Et, H, F, H, O, F, H, F, O, O, OMe], [AI 1083; Et, H, F, H, O, F, H, H, Cl, O, O, OMe], [AI 1084; Et, H, F, H, O, F, H, H, Br, O, O, OMe], [AI 1085; Et, H, F, H, O, F, H, H, I, O, O, OMe], [AI 1086; Et, H, F, H, O, F, H, H, Me, O, O, OMe] , [AI 1087; Et, H, F, H, O, F, H, H, Et, O, O, OMe], [AI 1088; Et, H, F, H, O, F, H, H, c- Pr, O, O, OMe], [AI 1089; Et, H, F, H, O, F, H, H, OMe, O, O, OMe], [AI 1090; Et, H, F, H, O, F, H, H, H, OEt, O, O, OMe], [AI1091; Et, H, F, H, O, F, H, S, Me, O, O, OMe], [AI1092; Et, H, F, H, O, F, H, H, CF 3, O, O, OMe], [AI1093; H, H, Cl, H, O, F, H, H, H, O, O, OMe], [AI 1094; H, H, Cl, H, O, F, H, H, F, O, O, OMe], [AI 1095; H, H, Cl, H, O, F, H, H, Cl, O , O, OMe], [AI 1096; H, H, Cl, H, O, F, H, H, Br, O, O, OMe], [AI 1097; H, H, Cl, H, O, F, H H, I, O, O, OMe], [AI 1098; H, H, Cl, H, O, F, H, Me, O, O, OMe], [AI 1099; H, H, Cl, H , O, F, H, H, Et, O, O, OMe], [AI 1100; H, H, Cl, H, O, F, H, H, c-Pr, O, O, OMe],

[AI 1101; H, H, Cl, H, O, F, H, OMe, O, O, OMe], [AI 1102; H, H, Cl, H, O, F, H, H, OE t, O , O, OMe], [AI1103; H, H, Cl, H, O, F, H, SMe, O, O, OMe], [AI 1104; H, H, Cl, H, O, F, H _{, H, CF 3, O,} O, OMe], [AI1105; Cl, H, Cl, H, O, F, H, H, H, O, O, OMe], [AI1106; Cl, H, Cl, H, O, F, H, H, F, O, O, OMe], [AI 1107; Cl, H, Cl, H, O, F, H, Cl, O, O, OMe], [AI 1108; Cl, H, Cl, H, O, F, H, H, Br, O, O, OMe], [AI 1109; Cl, H, Cl, H, O, F, H, I, O, O, OMe], [AI 1110; Cl, H, Cl, H, O, F, H, Me, O, O, OMe], [AI 1111; Cl, H, Cl, H, O, F, H, H, Et, O, O, OMe], [AI 1112; Cl, H, Cl, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1113; Cl, H, Cl, H, O, F, H, H, OMe, O, O, OMe], [AI 1114; Cl, H, Cl, H, O, F, H, OEt, O, O, OMe], [AI 1115; Cl, H, Cl, H, O, F, H, H, SMe, O, O, OMe], [AI1116; Cl, H, Cl, H, O, F, H, H, CF 3, O, O, OMe Me, H, Cl, H, O, F, H, H, H, O, O, OMe], [AI 1118; Me, H, Cl, H, O, F, H, H, F] , O, O, OMe], [AI 1119; Me, H, Cl, H, O, F, H, H, Cl, O, O, OMe], [AI 1 120; Me, H, Cl, H, O, F , H, H, Br, O, O, OMe], [AI 1121; Me, H, Cl, H, O, F, H, I, O, O, OMe], [AI 1122; Me, H, Cl , H, O, F, H, H, Me, O, O, OMe], [AI 1123; Me, H, Cl, H, O, F, H, Et, O, O, OMe], [AI 1 124 Me, H, Cl, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1 125; Me, H, Cl, H, O, F, H, H, OMe, O , O, OMe], [AI 1 126; Me, H, Cl, H, O, F, H, H, OEt, O, O, OMe], [AI 1 127; Me, H, Cl, H, O, F, H, H, SMe, O, O, OMe], [AI 1128; Me, H, Cl, H, O, F, H, H, CF ₃ , O , O, OMe], [AI 1129; Et, H, Cl, H, O, F, H, H, H, O, O, OMe], [AI 1130; Et, H, Cl, H, O, F, H , H, F, O, O, OMe], [AI 1131; Et, H, Cl, H, O, F, H, Cl, O, O, OMe], [AI 1132; Et, H, Cl, H , O, F, H, H, Br, O, O, OMe], [AI 1133; Et, H, Cl, H, O, F, H, I, O, O, OMe], [AI 1 134; Et , H, Cl, H, O, F, H, H, Me, O, O, OMe], [AI 1 135; Et, H, Cl, H, O, F, H, H, Et, O, O, OMe ], [AI 1136; Et, H, Cl, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1 137; Et, H, Cl, H, O, F, H, H] , OMe, O, O, OMe], [AI 1138; Et, H, Cl, H, O, F, H, OE, O, O, OMe], [AI 1139; Et, H, Cl, H, O , F, H, H, SMe , O, O, OMe], [AI1140; Et, H, Cl, H, O, F, H, H, CF 3, O, O, OMe], [AI1141; H, H, Me, H, O, F, H, H, H, O, O, OMe], [AI 1142; H, H, Me, H, O, F, H, F, O, O, OMe] , [AI1143; H, H, Me, H, O, F, H, H, Cl, O, O, OMe], [AI 1144; H, H, Me, H, O, F, H, H, Br, O, O, OMe], [AI 1145; H, H, Me, H, O, F, H, I, O, O, OMe], [AI 1146; H, H, Me, H, O, F, H, H, Me, O, O, OMe], [AI 1147; H, H, Me, H, O, F, H, Et, O, O, OMe], [AI 1148; H, H, Me, H, O, F, H, H, c, Pr, O, O, OMe], [AI 1149; H, H, Me, H, O, F, H, OMe, O, O, OMe], [ AI 1150; H, H, Me, H, O, F, H, OEt, O, O, OMe], [AI 1151; H, H, Me, H, O, F, H, S, M, O, O, OMe], [AI1152; H, H, Me, H, O, F, H, H, CF 3, O, O, OMe], [AI1153; Cl, H, M e, H, O, F, H, H, H, O, O, OMe], [AI 1154; Cl, H, Me, H, O, F, H, F, O, O, OMe], [ AI 1 155; Cl, H, Me, H, O, F, H, H, Cl, O, OMe], [AI 1156; Cl, H, Me, H, O, F, H, H, Br, O, O, OMe], [AI 1 157; Cl, H, Me, H, O, F, H, I, O, O, OMe], [AI 1158; Cl, H, Me, H, O, F, H, H, Me, O, O, OMe], [AI 1159; Cl, H, Me, H, O, F, H, H, Et, O, O, OMe], [AI 1 160; Cl, H, Me, H, O, F, H, H, c, -Pr, O, O, OMe], [AI1161; Cl, H, Me, H, O, F, H, OMe, O, O, OMe], [AI1162; Cl, H, Me, H, O, F, H, H, OEt, O, O, OMe], [AI1163; Cl, H, Me, H, O, F, H, SMe, O, O, OMe], [AI1164; Cl, H, Me, H, O, F, H, H, CF 3, O, O, OMe], [AI1165; Me, H, Me, H, O, F, H, H , H, O, O, OMe], [AI 1166; Me, H, Me, H, O, F, H, F, O, O, OMe], [AI 1 167; Me, H, Me, H, O , F, H, H, Cl, O, O, OMe], [AI 1168; Me, H, Me, H, O, F, H, H, Br, O, O, OMe], [AI 1169; Me, H , Me, H, O, F, H, H, I, O, O, OMe], [AI 1170; Me, H, Me, H, O, F, H, Me, O, O, OMe], [AI1171; Me, H, Me, H, O, F, H, H, Et, O, O, OMe], [AI1172; Me, H, Me, H, O, F, H, H, c-Pr , O, O, OMe], [AI1173; Me, H, Me, H, O, F, H, H, OMe, O, O, OMe], [AI 1174; Me, H, Me, H, O, F , H, H, OEt, O, O, OMe], [AI 1175; Me, H, Me, H, O, F, H, S, S, O, O, OMe], [AI 1176; Me, H, Me , H, O, F, H , H, CF 3, O, O, OMe], [AI1177; Et, H, Me, H, O, F, H, H, H, O, O, OMe], [ AI1178; Et, H, Me, H, O, F, H, H, F, O, O, OMe], [AI1179; Et, H, Me, H, O, F, H, H, Cl, O, O, OMe], [AI 1180; Et, H, Me, H, O, F, H, Br, O, O, OMe], [AI 1181; Et, H, Me, H, O, F, H, H, I, O, O, OMe], [AI 1182; Et, H, Me, H, O, F, H, Me, O, O, OMe] , [AI1183; Et, H, Me, H, O, F, H, H, Et, O, O, OMe], [AI 1184; Et, H, Me, H, O, F, H, H, c- Pr, O, O, OMe], [AI 1185; Et, H, Me, H, O, F, H, H, OMe, O, O, OMe], [AI 1186; Et, H, Me, H, O, F, H, H, H, OEt, O, O, OMe], [AI 1187; Et, H, Me, H, O, F, H, S, Me, O, O, OMe], [AI 1188; Et, H, Me, H, O, F, H, H, CF 3, O, O, OMe], [AI1189; H, H, Et, H, O, F, H, H, H, O, O, OMe], [AI 1190; H, H, Et, H, O, F, H, H, F, O, O, OMe], [AI1191; H, H, Et, H, O, F, H, H, Cl, O , O, OMe], [AI1192; H, H, Et, H, O, F, H, H, Br, O, O, OMe], [AI1193; H, H, Et, H, O, F, H , H, I, O, O, OMe], [AI 1194; H, H, Et, H, O, F, H, Me, O, O, OMe], [AI 1195; H, H, Et, H , O, F, H, H, Et, O, O, OMe], [AI 1196; H, H, Et, H, O, F, H, c, Pr, O, O, OMe], [AI 1197 H, H, Et, H, O, F, H, H, OMe, O, O, OMe], [AI 1198; H, H, Et, H, O, F, H, OEt, O, O , OMe], [AI 1199; H, H, Et, H, O, F, H, SMe, O, O, OMe], [AI 1200; H, H, Et, H, O, F, H, H , CF ₃ , O, O, OMe],

[AI 1201; Cl, H, Et, H, O, F, H, H, H, O, O, OMe], [AI 1202; Cl, H, Et, H, O, F, H, H, F, O , O, OMe], [AI 1203; Cl, H, Et, H, O, F, H, H, Cl, O, OMe], [AI 1204; Cl, H, Et, H, O, F, H , H, Br, O, O, OMe], [AI 1205; Cl, H, Et, H, O, F, H, I, O, O, OMe], [AI 1206; Cl, H, Et, H , O, F, H, H, Me, O, O, OMe], [AI1207; Cl, H, Et, H, O, F, H, Et, O, O, OMe], [AI 1208; Cl , H, Et, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1209; Cl, H, Et, H, O, F, H, OMe, O, O , OMe], [AI 1210; Cl, H, Et, H, O, F, H, H, OEt, O, O, OMe], [AI 1211; Cl, H, Et, H, O, F, H, H , SMe, O, O, OMe ], [AI1212; Cl, H, Et, H, O, F, H, H, CF 3, O, O, OMe], [AI1213; Me, H, Et, H, O, F, H, H, H, H, O, O, OMe], [AI 1214; Me, H, Et, H, O, F, H, F, O, O, OMe], [AI 1215; Me, H, Et, H, O, F, H, H, Cl, O, O, OMe], [AI 1216; Me, H, Et, H, O, F, H, H, Br, O, O, OMe] , [AI1217; Me, H, Et, H, O, F, H, H, I, O, O, OMe], [AI 1218; Me, H, Et, H, O, F, H, H, Me, O, O, OMe], [AI 1219; Me, H, Et, H, O, F, H, H, Et, O, O, OMe], [AI 1220; Me, H, Et, H, O, F, H, H, c-Pr, O, O, OMe], [AI 1221; Me, H, Et, H, O, F, H, H, OMe, O, O, OMe], [AI 1222; Me, H, Et, H, O, F, H, H, OEt, O, O, OMe], [AI1223; Me, H, Et, H, O, F, H, S, Me, O, O, OMe], [ AI1224; Me, H, Et, H, O, F, H, H, CF 3, O, O, OMe], [AI1225; Et, H, Et, H, O, F, H, H, H, O , O, OMe], [AI 1226; Et, H, Et, H, O, F, H, F, O, O, OMe], [AI 1 227; Et, H, Et, H, O, F, H, H, Cl, O, O, OMe], [AI1228; Et, H, Et, H, O, F, H, H, Br, O, O, OMe], [AI 1229; Et, H, Et, H, O, F, H, I, O, O, OMe], [AI 1230; Et, H, Et, H, O, F, H, H, Me, O, O, OMe], [AI 1231; Et, H, Et, H, O, F, H, Et, O, O, OMe], [AI 1232; Et, H, Et, H, O, F, H, H, c, Pr, O, O, OMe], [AI 1233; Et, H, Et, H, O, F, H, OM, O, O, OMe], [AI 1234; Et, H, Et, H, O, F, H, H, OEt, O, O, OMe], [AI 1235; Et, H, Et, H, O, F, H, SMe, O, O, OMe], [AI1236; Et, H, Et, H, O, F, H, H, CF 3, O, O, OMe], [AI1237; H, H, H, H, O, H, F, H H, H, H, H, H, H, O, H, H, F, H, F, O, O, OMe], [AI 1239; H, H, H, H, H, O , H, F, H, Cl, O, O, OMe], [AI 1240; H, H, H, H, H, O, H, F, H, Br, O, O, OMe], [AI 1241; H, H , H, H, O, H, F, H, I, O, O, OMe], [AI 1242; H, H, H, H, O, H, F, H, Me, O, O, OMe], [AI 1243; H, H, H, H, H, O, H, F, H, Et, O, O, OMe], [AI 1244; H, H, H, H, O, H, F, H, c-Pr , O, O, OMe], [AI 1245; H, H, H, H, O, H, H, F, H, OMe, O, O, OMe], [AI 1246; H, H, H, H, O, H , F, H, OEt, O, O, OMe], [AI 1247; H, H, H, H, H, O, H, F, H, SMe, O, O, OMe], [AI 1248; H, H, H , H, O, H, F , H, CF 3, O, O, OMe], [AI1249; Cl, H, H, H, O, H, F, H, H, O, O, OMe], [ AI 1 250; Cl, H, H, H, H, O, H, F, H, F, O, O, OMe], [AI 1251; Cl, H, H, H, H, O, H, F, H, Cl, O, O, OMe], [AI 1252; Cl, H, H, H, O, H, F, H, H, Br, O, O, OMe], [AI 1253; Cl, H, H, H, O, H, F, H, I, O, O, OMe ], [AI 1254; Cl, H, H, H, O, H, F, H, Me, O, O, OMe], [AI 1 255; Cl, H, H, H, O, H, F, H, Et, , O, O, OMe], [AI 1 256; Cl, H, H, H, H, O, H, H, F, H, c-Pr, O, O, OMe], [AI 1 257; Cl, H, H, H, O , H, F, H, OMe, O, O, OMe], [AI 1258; Cl, H, H, H, H, O, H, F, H, OEt, O, O, OMe], [AI 1259; Cl, H , H, H, O, H , F, H, SMe, O, O, OMe], [AI1260; Cl, H, H, H, O, H, F, H, CF 3, O, O, OMe] [AI 1261; Me, H, H, H, H, O, H, F, H, H, O, O, OMe], [AI 1262; Me, H, H, H, O, H, F, H, F, F, O, O, OMe], [AI 1263; Me, H, H, H, H, O, H, F, H, Cl, O, OMe], [AI 1264; Me, H, H, H, O, H, F, H, Br, O, O, OMe], [AI 1 265; Me, H, H, H, H, O, H, F, H, I, O, O, OMe], [AI 1 266; Me, H, H, H, O, H, F, H, Me, O, O, OMe], [AI1267; Me, H, H, H, H, O, H, F, H, Et, O, O, OMe], [AI1268; Me, H, H, H, H, O, H, F, H, c-Pr, O, O, OMe], [AI 1269; Me, H, H, H, O, H, F, H, OMe, O, O, OMe], [AI1270; Me, H, H, H, O, H, F, H, OEt, O, O, OMe], [AI 1271; Me, H, H, H, O, H, F, H, SMe, O, O, OMe], [AI1272; Me, H, H, H, O, H, F, H, CF 3, O, O, OMe], [AI1273; Et, H, H, H , O, H, F, H, H, O, O, OMe], [AI 1274; Et, H, H, H, H, O, H, F, H, F, O, O, OMe], [AI 1275; Et , H, H, H, O, H, F, H, Cl, O, O, OMe], [AI 1276; Et, H, H, H, H, O, H, F, H, Br, O, O, OMe ], [AI1277; Et, H, H, H, H, O, H, F, H, I, O, O, OMe], [AI 1278; Et, H, H, H, O, H, F, H, Me , O, O, OMe], [AI 1279; Et, H, H, H, H, O, H, F, H, Et, O, O, OMe], [AI 1280; Et, H, H, H, O, H , F, H, c -Pr, O, O, OMe], [AI 1281; Et, H, H, H, H, O, H, F, H, O, O, O, OMe], [AI 1282; Et, H, H, H, O , H, F, H, OEt, O, O, OMe], [AI1283; Et, H, H, H, H, O, H, F, H, SMe, O, O, OMe], [AI 1284; Et, H , H, H, O, H , F, H, CF 3, O, O, OMe], [AI1285; H, H, F, H, O, H, F, H, H, O, O, OMe] [AI 1286; H, H, F, H, O, H, F, H, F, O, O, OMe], [AI 1287; H, H, F, H, O, H, F, H, Cl, O, O, OMe], [AI 1 288; H, H, F, H, O, H, F, H, Br, O, O, OMe], [AI 1 289; H, H, F, H, O, H, F, H, I, O, O, OMe], [AI 1290; H, H, F, H, O, H, F, H, Me, O, O, OMe], [AI 1291; H, H, F, H, O, H, F, H, Et, O, O, OMe], [AI1292; H, H, F, H, O, H, F, H, c-Pr, O, O, OMe], [ AI 1293; H, H, F, H, O, H, F, H, OMe, O, O, OMe], [AI 1294; H, H, F, H, O, H, F, H, OEt, O, O, OMe], [AI 1295; H, H, F, H, O, H, F, H, SMe, O, O, OMe], [AI 1296; H, H, F, H, O, H, F, _{H, CF 3, O, O} , OMe], [AI1297; Cl, H, F, H, O, H, F, H, H, O, O, OMe], [AI1298; Cl, H, F, H , O, H, F, H, F, O, O, OMe], [AI 1299; Cl, H, F, H, O, H, F, H, Cl, O, O, OMe], [AI 1300; , H, F, H, O, H, F, H, Br, O, O, OMe],

[AI 1301; Cl, H, F, H, O, H, F, H, I, O, O, OMe], [AI 1302; Cl, H, F, H, O, H, F, H, Me, O , O, OMe], [AI 1303; Cl, H, F, H, O, H, F, H, Et, O, O, OMe], [AI 1304, Cl, H, F, H, O, H, F , H, c-Pr, O, O, OMe], [AI 1305; Cl, H, F, H, O, H, F, H, OMe, O, O, OMe], [AI 1306; Cl, H, F , H, O, H, F, H, OEt, O, O, OMe], [AI 1307; Cl, H, F, H, O, H, F, H, SMe, O, O, OMe], [AI 1308 ; Cl, H, F, H , O, H, F, H, CF 3, O, O, OMe], [AI1309; Me, H, F, H, O, H, F, H, H, O, O, OMe], [AI 1310; Me, H, F, H, O, H, F, H, F, O, O, OMe], [AI 1311; Me, H, F, H, O, H, F, H, Cl, O, O, OMe], [AI 1312; Me, H, F, H, O, H, F, H, Br, O, O, OMe], [AI 1313; Me, H, F, H, O, H, F, H, I, O, O, OMe], [AI 1314; Me, H, F, H, O, H, F, H, Me, O, O, OMe], [AI 1315; H, F, H, O, H, F, H, Et, O, O, OMe], [AI 1316; Me, H, F, H, O, H, F, H, c-Pr, O, O, OMe], [AI 1317; Me, H, F, H, O, H, F, H, OMe, O, O, OMe], [AI 1318; Me, H, F, H, O, H, F, H, OEt, O, O, OMe], [AI 1319; Me, H, F, H, O, H, F, H, S Me, O, O, OMe], [AI 1320; Me, H, F, H, O, _{H, F, H, CF 3} , O, O, OMe], [AI1321; Et, H, F, H, O, H, F, H, H, O, O, OMe], [AI1322; Et, H , F, H, O, H, F, H, F, O, O, OMe], [AI 1323; Et, H, F, H, O, H, F, H, Cl, O, O, OMe], [AI1324; Et, H, F, H, O, H, F, H, Br, O, O, OMe], [AI 1325; Et, H, F, H, O, H, F, H, I, O , O, OMe], [AI 1326; Et, H, F, H, O, H, F, H, Me, O, O, OMe], [AI 1327; Et, H, F, H, O, H, F , H, Et, O , O, OMe], [AI 1328; Et, H, F, H, O, H, F, H, c-Pr, O, O, OMe], [AI 1329; Et, H, F, H, O, H , F, H, OMe, O, O, OMe], [AI 1330; Et, H, F, H, O, H, F, H, OE t, O, O, OMe], [AI 1331; Et, H, F , H, O, H, F , H, SMe, O, O, OMe], [AI1332; Et, H, F, H, O, H, F, H, CF 3, O, O, OMe], [ AI1333; H, H, Cl, H, O, H, F, H, H, O, O, OMe], [AI 1334; H, H, Cl, H, O, H, F, H, F, O, O, OMe], [AI 1335; H, H, Cl, H, O, H, F, H, Cl, O, O, OMe], [AI 1336; H, H, Cl, H, O, H, F, H, Br, O, O, OMe], [AI 1337; H, H, Cl, H, O, H, F, H, I, O, O, OMe], [AI 1 338; H, H, Cl, H, O, H, F, H, Me, O, O, OMe], [AI 1339; H, H, Cl, H, O, H, F, H, Et, O, O, OMe], [AI 1340; H, H, Cl, H, O, H, F, H, c-Pr, O, O, OMe], [AI 1341; H, H, Cl, H, O, H, F, H, OMe, O, O, OMe], [AI1342; H, H, Cl, H, O, H, F, H, OEt, O, O, OMe], [AI1343; H, H, Cl, H, O, H, F, H, H, SMe, O, O, OMe] , [AI1344; H, H, Cl, H, O, H, F, H, CF 3, O, O, OMe], [AI1345; Cl, H, Cl, H, O , H, F, H, H, H, O, O, OMe], [AI 1346; Cl, H, Cl, H, O, H, F, H, F, O, O, OMe], [AI 1347; Cl, H , Cl, H, O, H, F, H, Cl, O, O, OMe], [AI 1348; Cl, H, Cl, H, O, H, F, H, Br, O, O, OMe], [AI1349; Cl, H, Cl, H, O, H, F, H, I, O, O, OMe], [AI 1 350; Cl, H, Cl, H, O, H, F, H, Me, O , O, OMe], [AI 1351; Cl, H, Cl, H, O, H, F, H, Et, O, O, OMe], [AI 1352; Cl, H, Cl, H, O, H, F , H, c-Pr, O, O, OMe], [AI1353; Cl, H, Cl, H, O, H, F, H, OMe, O, O, OMe], [AI 1354; Cl, H, Cl, H, O, H, F, H, OEt, O, O, OMe], [AI 1355; Cl, H, Cl, H, O, H, F, H, SMe, O, O, OMe], [AI1356; Cl, H, Cl, H, O, H, F, H, CF 3, O, O, OMe], [AI1357; Me, H, Cl, H, O, H, F, H , H, O, O, OMe], [AI 1358; Me, H, Cl, H, O, H, F, H, F, O, O, OMe], [AI 1359; Me, H, Cl, H, O , H, F, H, Cl, O, O, OMe], [AI 1 360; Me, H, Cl, H, O, H, F, H, Br, O, O, OMe], [AI 1361; Me, H , Cl, H, O, H, F, H, I, O, O, OMe], [AI 1362; Me, H, Cl, H, O, H, F, H, Me, O, O, OMe], [AI1363; Me, H, Cl, H, O, H, F, H, Et, O, O, OMe], [AI 1364; Me, H, Cl, H, O, H, F, H, c-Pr , O, O, OMe], [AI 1365; Me, H, Cl, H, O, H, F, H, OMe, O, O, OMe], [AI 1 366; Me, H, Cl, H, O, H , F, H, OEt, O, O, OMe], [AI 1367; Me, H, Cl, H, O, H, F, H, SMe, O, O, OMe], [AI 1 368; Me, H, Cl , H, O, H, F , H, CF 3, O, O, OMe], [AI1369; Et, H, Cl, H, O, H, F, H, H, O, O, OMe], [ AI 1370; Et, H, Cl, H, O, H, F, H, F, O, O, OMe], [AI1371; Et, H, Cl, H, O, H, F, H, Cl, O, O, OMe], [AI1372; Et, H, Cl, H, O, H, F, H, Br, O, O, OMe], [AI 1373; Et, H, Cl, H, O, H, F, H, I, O, O, OMe], [AI 1374; Et, H, Cl, H, O, H, F, H, Me, O, O, OMe], [AI 1 375; Et, H, Cl, H, O, H, F, H, Et, O, O, OMe], [AI 1376; Et, H, Cl, H, O, H, F, H, c-Pr, O, O, OMe], [AI 1377; Et, H, Cl, H, O, H, F, H, OMe, O, O, OMe], [AI 1378; Et, H, Cl, H, O, H, F, H, OEt, O, O, OMe], [AI 1379; Et, H, Cl, H, O, H, F, H, SMe, O, O, OMe], [AI 1380; Et, H, Cl, H, O, H, F, H, CF 3, O, O, OMe], [AI1381; H, H, Me, H, O, H, F, H, H, O, O , OMe], [AI1382; H, H, Me, H, O, H, F, H, F, O, O, OMe], [AI1383; H, H, Me, H, O, H, F, H , Cl, O, O, OMe], [AI 1384; H, H, Me, H, O, H, F, H, Br, O, O, OMe], [AI 1385; H, H, Me, H, O , H, F, H, I, O, O, OMe], [AI 1386; H, H, Me, H, O, H, F, H, Me, O, O, OMe], [AI 1387; H, H , Me, H, O, H, F, H, Et, O, O, OMe], [AI 1388; H, H, Me, H, O, H, F, H, c-Pr, O, O, OMe H, H, Me, H, O, H, F, H, OMe, O, O, OMe], [AI 1390; H, H, Me, H, O, H, F, H, OEt] , O, O, OMe], [AI1391; H, H, Me, H, O, H, F, H, SMe, O, O, OMe], [AI1392; H, H, Me, H, O, H _{, F, H, CF 3,} O, O, OMe], [AI1393; Cl, H, Me, H, O, H, F, H, H, O, O, OMe], [AI1394; Cl, H, Me, H, O, H, F, H, F, O, O, OMe], [AI 1395; Cl, H, Me, H, O, H, F, H, Cl, O, O, OMe], [ AI 1396; Cl, H, Me, H, O, H, F, H, Br, O, O, OMe], [AI 1397; Cl, H, Me, H, O, H, F, H, I, O, O, OMe], [AI 1398; Cl, H, Me, H, O, H, F, H, Me, O, O, OMe], [AI 1399; Cl, H, Me, H, O, H, F, H, Et, O, O, OMe], [AI 1400; Cl, H, Me, H, O, H, F, H, c-Pr, O, O, OMe],

[AI 1401; Cl, H, Me, H, O, H, F, H, OMe, O, O, OMe], [AI 1402; Cl, H, Me, H, O, H, F, H, OE t, O , O, OMe], [AI 1403; Cl, H, Me, H, O, H, F, H, S Me, O, O, OMe], [AI 1404; Cl, H, Me, H, O, H, F _{, H, CF 3, O,} O, OMe], [AI1405; Me, H, Me, H, O, H, F, H, H, O, O, OMe], [AI1406; Me, H, Me, H, O, H, F, H, F, O, O, OMe], [AI 1407; Me, H, Me, H, O, H, F, H, Cl, O, O, OMe], [AI 1408; Me, H, Me, H, O, H, F, H, Br, O, O, OMe], [AI 1409; Me, H, Me, H, O, H, F, H, I, O, O, OMe], [AI 1410; Me, H, Me, H, O, H, F, H, Me, O, O, OMe], [AI 1411; Me, H, Me, H, O, H, F, H, Et, O, O, OMe], [AI 1412; Me, H, Me, H, O, H, F, H, c, Pr, O, O, OMe], [AI 1413; Me, H, Me, H, O, H, F, H, OMe, O, O, OMe], [AI 1414; Me, H, Me, H, O, H, F, H, OE t, O, O, OMe], [AI 1415; Me, H, Me, H, O, H, F, H, SMe, O, O, OMe], [AI1416; Me, H, Me, H, O, H, F, H, CF 3, O, O, OMe ], [AI1417; Et, H, Me, H, O, H, F, H, H, O, O, OMe], [AI 1418; Et, H, Me, H, O, H, F, H, F] , O, O, OMe], [AI 1419; Et, H, Me, H, O, H, F, H, Cl, O, O, OMe], [AI 1420; Et, H, Me, H, O, H , F, H, Br, O, O, OMe], [AI 1421; Et, H, Me, H, O, H, F, H, I, O, O, OMe], [AI 1422; Et, H, Me , H, O, H, F, H, Me, O, O, OMe], [AI 1423; Et, H, Me, H, O, H, F, H, Et, O, O, OMe], [AI 1424 Et, H, Me, H, O, H, F, H, c-Pr, O, O, OMe], [AI 1425; Et, H, Me, H, O, H, F, H, OMe, O , O, OMe], [AI 1426; Et, H, Me, H, O, H, F, H, OEt, O, O, OMe], [AI1427; Et, H, Me, H, O, H, F, H, SMe, O, O, OMe], [AI 1428; Et, H, Me, H, O, H, F, H, CF ₃ , O, O, OMe], [AI1429; H, H, Et, H, O, H, F, H, H, O, O, OMe], [AI 1430; H, H, Et, H, O, H, F, H, F, O, O, OMe], [AI 1431; H, H, Et, H, O, H, F, H, Cl, O, OMe], [AI 1432; H, H, Et, H, O, H, F, H, Br, O, O, OMe], [AI 1433; H, H, Et, H, O, H, F, H, I, O, O, OMe], [AI 1434; H, H, Et, H, O, H, F, H, Me, O, O, OMe], [AI 1435; H, H, Et, H, O, H, F, H, Et, O, O, OMe], [AI 1436; H, H, Et, H, O, H, F, H, c, Pr, O, O, OMe], [AI 1437; H, H, Et, H, O, H, F, H, OMe, O, O, OMe], [AI 1438; H, H, Et, H, O, H, F, H, OE, O, O, OMe], [AI 1439; H, H, Et, H, O, H, F, H, SMe, O, O, OMe], [AI1440; H, H, Et, H, O, H, F, H, CF 3, O, O, OMe], [AI1441; Cl , H, Et, H, O, H, F, H, H, O, O, OMe], [AI1442; Cl, H, Et, H, O, H, F, H, F, O, O, OMe ], [AI 1443; Cl, H, Et, H, O, H, F, H, Cl, O, O, OMe], [AI 1444; Cl, H, Et, H, O, H, F, H, Br] , O, O, OMe], [AI 1445; Cl, H, Et, H, O, H, F, H, I, O, O, OMe], [AI 1446; Cl, H, Et, H, O, H , F, H, Me, O, O, OMe], [AI1447; Cl, H, Et, H, O, H, F, H, Et, O, O, OMe], [AI 1448; Cl, H, Et , H, O, H, F, H, c-Pr, O, O, OMe], [AI1449; Cl, H, Et, H, O, H, F, H, OMe, O, O, OMe], [AI 1450; Cl, H, Et, H, O, H, F, H, OEt, O, O, OMe], [AI 1451; Cl, H, Et, H, O, H, F, H, SMe, O , O, OMe], [AI1452 ; Cl, H, Et, H, O, H, F, H, CF 3, O, O, OMe], [AI1453; Me , H, Et, H, O, H, F, H, H, O, O, OMe], [AI 1454; Me, H, Et, H, O, H, F, H, F, O, O, OMe Me, H, Et, H, O, H, F, H, Cl, O, O, OMe], [AI 1456; Me, H, Et, H, O, H, F, H, Br] , O, O, OMe], [AI 1457; Me, H, Et, H, O, H, F, H, I, O, O, OMe], [AI 1458; Me, H, Et, H, O, H , F, H, Me, O, O, OMe], [AI 1459; Me, H, Et, H, O, H, F, H, Et, O, O, OMe], [AI 1460; Me, H, Et , H, O, H, F, H, c-Pr, O, O, OMe], [AI 1461; Me, H, Et, H, O, H, F, H, OMe, O, O, OMe], [AI1462; Me, H, Et, H, O, H, F, H, OEt, O, O, OMe], [AI 1463; Me, H, Et, H, O, H, F, H, SMe, O , O, OMe], [AI 1464; Me, H, Et, H, O, H, F, H, CF ₃ , O, O, OMe], [AI 1465; Et, H, Et, H, O, H, F, H, H, H, O, O, OMe], [AI 1466; Et, H, Et, H, O, H, F, H, F, O, O, OMe], [AI 1467; Et, H, Et, H, O, H, F, H, Cl, O, O, OMe], [AI 1468; Et, H, Et, H, O, H, F, H, Br, O, O, OMe], [AI 1469; Et, H, Et, H, O, H, F, H, I, O, O, OMe], [AI 1470; Et, H, Et, H, O, H, F, H, Me, O, O, OMe], [AI1471; Et, H, Et, H, O, H, F, H, H, Et, O, O, OMe], [AI1472; Et, H, Et, H, O, H, F, H, c-Pr, O, O, OMe], [AI1473; Et, H, Et, H, O, H, F, H, OMe, O, O, OMe], [AI1474; Et, H, Et, H, O, H, F, H, OEt, O, O, OMe], [AI1475; Et, H, Et, H, O, H, F, H, SMe, O, O, OMe], [AI 1476; Et, H, Et, H, O, H, F, H, CF 3, O, O, OMe], [AI1477; H, H, H, H, O, H, H, F, H, O, O, OMe ], [AI 1478; H, H, H, H, H, O, H, H, F, F, O, O, OMe], [AI 1479; H, H, H, H, O, H, H, F, Cl, O, O, OMe], [AI 1480; H, H, H, H, H, O, H, H, F, Br, O, O, OMe], [AI 1481; H, H, H, H, O, H, H, F, I, O, O, OMe], [AI 1482; H, H, H, H, O, H, F, Me, O, O, OMe], [ AI 1483; H, H, H, H, H, O, H, H, F, Et, O, O, OMe], [AI 1484; H, H, H, H, H, O, H, F, c-Pr, H, H, H, H, H, O, H, H, H, F, OMe, O, O, OMe], [AI 1486; H, H, H, H, O, H, O, O, OMe], [AI 1485; H, F, OEt, O, O, O, OMe], [AI 1487; H, H, H, H, H, O, H, H, F, SMe, O, O, OMe], [AI 1 488; H, H, H, H, O, H, H, F, CF 3, O, O, OMe], [AI1489; Cl, H, H, H, O, H, H, F, H, O, O, OMe], [AI1490 Cl, H, H, H, H, O, H, H, H, F, F, O, O, OMe], [AI1491; Cl, H, H, H, H, O, H, F, Cl, O, O , OMe], [AI1492; Cl, H, H, H, O, H, H, F, Br, O, O, OMe], [AI 1493; Cl, H, H, H, O, H, H, F Cl, H, H, H, H, O, H, H, F, Me, O, O, OMe], [AI 1495; Cl, H, H, H, H, O , H, H, F, Et, O, O, OMe], [AI1496; Cl, H, H, H, H, O, H, H, F, c-Pr, O, O, OMe], [AI 1497; Cl , H, H, H, O, H, H, F, OMe, O, O, OMe], [AI 1498; Cl, H, H, H, O, H, H, F, OEt, O, O, OMe ], [AI1499; Cl, H, H, H, O, H, H, F, SMe, O, O, OMe], [AI 1500; Cl, H, H, H, O, H, H, F, CF] ₃ , O, O, OMe],

[AI 1501; Me, H, H, H, H, O, H, H, F, H, O, O, OMe], [AI 1502; Me, H, H, H, O, H, H, F, F, O , O, OMe], [AI 1503; Me, H, H, H, H, O, H, H, F, Cl, O, OMe], [AI 1504; Me, H, H, H, O, H, H , F, Br, O, O, OMe], [AI 1505; Me, H, H, H, H, O, H, H, F, I, O, O, OMe], [AI 1506; Me, H, H, H , O, H, H, F, Me, O, O, OMe], [AI1507; Me, H, H, H, H, O, H, H, F, Et, O, O, OMe], [AI1508; Me , H, H, H, O, H, H, F, c, Pr, O, O, OMe], [AI 1509; Me, H, H, H, O, H, H, F, OMe, O, O , OMe], [AI 1510; Me, H, H, H, O, H, H, F, OEt, O, O, OMe], [AI 1511; Me, H, H, H, O, H, H, F , SMe, O, O, OMe ], [AI1512; Me, H, H, H, O, H, H, F, CF 3, O, O, OMe], [AI1513; Et, H, H, H, O, H, H, H, F, H, O, O, OMe], [AI 1514; Et, H, H, H, H, O, H, H, F, F, O, O, OMe], [AI 1515; Et, H, H, H, H, O, H, H, F, Cl, O, O, OMe], [AI 1516; Et, H, H, H, H, O, H, F, Br, O, O, OMe] [AI 1517; Et, H, H, H, H, O, H, H, F, I, O, O, OMe], [AI 1518; Et, H, H, H, O, H, H, F, Me, O, O, OMe], [AI 1519; Et, H, H, H, H, O, H, H, F, Et, O, O, OMe], [AI 1520; Et, H, H, H, O, H, H, F, c-Pr, O, O, OMe], [AI1521; Et, H, H, H, H, O, H, H, F, OMe, O, O, OMe], [AI1522; Et, H, H, H, O, H, H, F, OEt, O, O, OMe], [AI1523; Et, H, H, H, H, O, H, F, SMe, O, O, OMe], [ AI1524; Et, H, H, H, O, H, H, F, CF 3, O, O, OMe], [AI1525; H, H, F, H, O, H, H, F, H, O , O, OMe], [AI1526; H, H, F, H, O, H, H, F, F, O, O, OMe], [AI 1527; H, H, F, H, O, H, H , F, Cl, O, O, O Me, [AI 1528; H, H, F, H, O, H, H, F, Br, O, O, OMe], [AI 1529; H, H, F, H, O, H, H, F, I, O, O, OMe], [AI 1530; H, H, F, H, O, H, H, F, Me, O, O, OMe], [AI 1531; H, H, F, H, O, H, H, F, Et, O, O, OMe], [AI 1532; H, H, F, H, O, H, H, F, c-Pr, O, O, OMe], [AI 1533; H, H, F, H, O, H, H, F, OMe, O, O, OMe], [AI1534; H, H, F, H, O, H, H, F, OEt, O, O, OMe] , [AI1535; H, H, F, H, O, H, H, F, SMe, O, O, OMe], [AI 1536; H, H, F, H, O, H, H, F, CF ₃ , O, O, OMe], [AI1537; Cl, H, F, H, O, H, H, F, H, O, O, OMe], [AI 1538; Cl, H, F, H, O, H , H, F, F, O, O, OMe], [AI1539; Cl, H, F, H, O, H, H, F, Cl, O, OMe], [AI 1540; Cl, H, F , H, O, H, H, F, Br, O, O, OMe], [AI1541; Cl, H, F, H, O, H, F, I, O, O, OMe], [AI 1542 Cl, H, F, H, O, H, H, F, Me, O, O, OMe], [AI 1543; Cl, H, F, H, O, H, H, F, Et, O, O , OMe], [AI 1544; Cl, H, F, H, O, H, H, F, c, Pr, O, O, OMe], [AI 1545; Cl, H, F, H, O, H, H , F, OMe, O, O, OMe], [AI 1546; Cl, H, F, H, O, H, H, F, OEt, O, O, OMe], [AI 1547; Cl, H, F, H , O, H, H, F, SMe, O, O, OMe], [AI 1548; Cl, H, F, H, O, H, H, F, CF ₃ , O, O, OMe], [AI 1 549; Me, H, F, H, O, H, H, F, H, O, O, OMe], [AI 1550; Me, H, F, H, O, H, F, F, O, O, O OMe], [AI 1551; Me, H, F, H, O, H, H, F, Cl, O, O, OMe], [AI 1552; Me, H, F, H, O, H, H, F, Br, O, O, OMe], [AI 1553; Me, H, F, H, O, H, H, F, I, O, O, OMe], [AI 1554; Me, H, F, H, O, H, H, F, Me, O, O, OM e], [AI 1 555; Me, H, F, H, O, H, H, F, Et, O, O, OMe], [AI 1 556; Me, H, F, H, O, H, H, F, c-Pr, O, O, OMe], [AI 1557; Me, H, F, H, O, H, H, F, OMe, O, O, OMe], [AI 1 558; Me, H, F, H, O, H, H, F, OEt, O, O, OMe], [AI 1559; Me, H, F, H, O, H, H, F, SMe, O, O, OMe], [AI 1560; Me, H, F, H, O, H, H, F, CF 3, O, O, OMe], [AI1561; Et, H, F, H, O, H, H, F, H, O, O, OMe ], [AI1562; Et, H, F, H, O, H, H, F, F, O, O, OMe], [AI 1563; Et, H, F, H, O, H, H, F, Cl] , O, O, OMe], [AI1564; Et, H, F, H, O, H, H, F, Br, O, O, OMe], [AI 1 565; Et, H, F, H, O, H , H, F, I, O, O, OMe], [AI 1 566; Et, H, F, H, O, H, H, F, Me, O, O, OMe], [AI 1567; Et, H, F , H, O, H, H, F, Et, O, O, OMe], [AI1568; Et, H, F, H, O, H, H, F, c-Pr, O, O, OMe], [AI 1569; Et, H, F, H, O, H, H, F, OMe, O, O, OMe], [AI 1570; Et, H, F, H, O, H, H, F, OEt, O , O, OMe], [AI 1571; Et, H, F, H, O, H, H, F, S Me, O, O, OMe], [AI 1572; Et, H, F, H, O, H, H _{, F, CF 3, O,} O, OMe], [AI1573; H, H, Cl, H, O, H, H, F, H, O, O, OMe], [AI1574; H, H, Cl, H, O, H, H, F, F, F, O, O, OMe], [AI 1575; H, H, Cl, H, O, H, F, Cl, O, O, OMe], [AI 1576; H, H, Cl, H, O, H, H, F, Br, O, OMe], [AI 1577; H, H, Cl, H, O, H, H, F, I, O, O, OMe], [AI 1578; H, H, Cl, H, O, H, H, F, Me, O, O, OMe], [AI 1579; H, H, Cl, H, O, H, H, F, Et, O, O, OMe], [AI 1580; H, H, Cl, H, O, H, H, F, c-Pr, O, O, OMe], [AI 1581; H, H, Cl, H, O, H, H, F, OMe, O, O, OMe], [AI 1582; H, H, Cl, H, O, H, H, F, OE t, O, O, OMe], [AI 1583; H, H, Cl, H, O, H, H, F, SMe, O, O, OMe], [AI1584; H, H, Cl, H, O, H, H, F, CF 3, O, O, OMe], [AI1585; Cl , H, Cl, H, O, H, H, F, H, O, O, OMe], [AI 1586; Cl, H, Cl, H, O, H, H, F, F, O, O, OMe ], [AI1587; Cl, H, Cl, H, O, H, H, F, Cl, O, O, OMe], [AI 1588; Cl, H, Cl, H, O, H, H, F, Br] , O, O, OMe], [AI1589; Cl, H, Cl, H, O, H, H, F, I, O, O, OMe], [AI 1590; Cl, H, Cl, H, O, H , H, F, Me, O, O, OMe], [AI1591; Cl, H, Cl, H, O, H, H, F, Et, O, O, OMe], [AI1592; Cl, H, Cl , H, O, H, H, F, c, Pr, O, O, OMe], [AI 1593; Cl, H, Cl, H, O, H, F, OM, O, O, OMe], [AI1594; Cl, H, Cl, H, O, H, H, F, OEt, O, O, OMe], [AI 1595; Cl, H, Cl, H, O, H, H, F, SMe, O , O, OMe], [AI 1596; Cl, H, Cl, H, O, H, H, F, CF ₃ , O, O, OMe], [AI 1597; Me, H, Cl, H, O, H, H, F, H, O, O, O, OMe], [AI 1598; Me, H, Cl, H, O, H, H, F, F, O, O, OMe], [AI 1 599; Me, H, Cl, H, O, H, H, F, Cl, O, O, OMe], [AI1600; Me, H, Cl, H, O, H, H, F, Br, O, O, OMe],

[AI 1601; Me, H, Cl, H, O, H, H, F, I, O, O, OMe], [AI 1602; Me, H, Cl, H, O, H, H, F, Me, O , O, OMe], [AI1603; Me, H, Cl, H, O, H, H, F, Et, O, O, OMe], [AI 1604, Me, H, Cl, H, O, H, H , F, c-Pr, O, O, OMe], [AI 1605; Me, H, Cl, H, O, H, H, F, OMe, O, O, OMe], [AI 1606; Me, H, Cl , H, O, H, H, F, OEt, O, O, OMe], [AI 1607; Me, H, Cl, H, O, H, F, S Me, O, O, OMe], [AI 1608 ; Me, H, Cl, H , O, H, H, F, CF 3, O, O, OMe], [AI1609; Et, H, Cl, H, O, H, H, F, H, O, O, OMe], [AI 1610; Et, H, Cl, H, O, H, H, F, F, O, O, OMe], [AI 1611; Et, H, Cl, H, O, H, H, F, Cl, O, O, OMe], [AI 1612; Et, H, Cl, H, O, H, H, H, F, Br, O, O, OMe], [AI 1613; Et, H, Cl, H, O, H, H, F, I, O, O, OMe], [AI 1614; Et, H, Cl, H, O, H, H, F, Me, O, O, OMe], [AI 1615; Et, H, Cl, H, O, H, H, F, Et, O, O, OMe], [AI 1616; Et, H, Cl, H, O, H, F, c, Pr, O, O, OMe], [AI1617; Et, H, Cl, H, O, H, H, F, OMe, O, O, OMe], [AI 1618; Et, H, Cl, H, O, H, H, F, OEt, O, O, OMe], [AI 1619; Et, H, Cl, H, O, H, H, F, SMe, O, O, OMe], [AI 1620; Et, H, Cl, H, O, _{H, H, F, CF 3} , O, O, OMe], [AI1621; H, H, Me, H, O, H, H, F, H, O, O, OMe], [AI1622; H, H , Me, H, O, H, H, F, F, O, O, OMe], [AI1623; H, H, Me, H, O, H, H, F, Cl, O, O, OMe], [AI1624; H, H, Me, H, O, H, H, F, Br, O, O, OMe], [AI 1625; H, H, Me, H, O, H, H, F, I, O , O, OMe], [AI1626; H, H, Me, H, O, H, H, F, Me, O, O, OMe], [AI 1627; H , H, Me, H, O, H, H, F, Et, O, O, OMe], [AI 1628; H, H, Me, H, O, H, H, F, c-Pr, O, O , OMe], [AI1629; H, H, Me, H, O, H, H, F, OMe, O, O, OMe], [AI 1630; H, H, Me, H, O, H, H, F , OEt, O, O, OMe], [AI1631; H, H, Me, H, O, H, H, F, SMe, O, O, OMe], [AI1632; H, H, Me, H, O , H, H, F, CF 3, O, O, OMe], [AI1633; Cl, H, Me, H, O, H, H, F, H, O, O, OMe], [AI1634; Cl, H, Me, H, O, H, H, F, F, O, O, OMe], [AI 1635; Cl, H, Me, H, O, H, H, F, Cl, O, O, OMe] , [AI1636; Cl, H, Me, H, O, H, H, F, Br, O, O, OMe], [AI 1637; Cl, H, Me, H, O, H, H, F, I, O, O, OMe], [AI1638; Cl, H, Me, H, O, H, H, F, Me, O, O, OMe], [AI 1639; Cl, H, Me, H, O, H, H, F, Et, O, O, OMe], [AI 1640; Cl, H, Me, H, O, H, H, F, c, Pr, O, O, OMe], [AI 1641; Cl, H, Me, H, O, H, H, F, OMe, O, O, OMe], [AI 1642; Cl, H, Me, H, O, H, H, F, OEt, O, O, OMe], [ AI 1643; Cl, H, Me, H, O, H, H, F, SMe, O, O, OMe], [AI 1644; Cl, H, Me, H, O, H, H, F, CF ₃ , O , O, OMe], [AI 1645; Me, H, Me, H, O, H, H, H, F, H, O, O, OMe], [AI 1 646; Me, H, Me, H, O, H, H , F, F, O, O, OMe], [AI 1647; Me, H, Me, H, O, H, H, F, Cl, O, OMe], [AI 1648; Me, H, Me, H , O, H, H, F, Br, O, O, OMe], [AI 1649; Me, H, Me, H, O, H, H, F, I, O, O, OMe], [AI 1650; Me , H, Me, H, O, H, H, F, Me, O, O, OMe], [AI 1651; Me, H, Me, H, O, H, H, F, Et, O, O, OMe ], [AI1652; Me, H, Me, H, O, H, H, F, c-Pr, O, O, OMe], [AI1653; Me, H, Me , H, O, H, H, F, OMe, O, O, OMe], [AI1654; Me, H, Me, H, O, H, H, F, OEt, O, O, OMe], [AI 1655] Me, H, Me, H, O, H, H, F, SMe, O, O, OMe], [AI 1656; Me, H, Me, H, O, H, H, F, CF ₃ , O, O, OMe], [AI1657; Et, H, Me, H, O, H, H, F, H, O, O, OMe], [AI 1658; Et, H, Me, H, O, H, H, F, F, O, O, OMe], [AI 1659; Et, H, Me, H, O, H, H, F, Cl, O, O, OMe], [AI 1660; Et, H, Me, H, O, H, H, F, Br, O, O, OMe], [AI1661; Et, H, Me, H, O, H, H, F, I, O, O, OMe], [AI1662; Et, H, Me, H, O, H, H, F, Me, O, O, OMe], [AI1663; Et, H, Me, H, O, H, H, F, Et, O, O, OMe] , [AI1664; Et, H, Me, H, O, H, H, F, c-Pr, O, O, OMe], [AI 1 665; Et, H, Me, H, O, H, H, F, OMe, O, O, OMe], [AI1666; Et, H, Me, H, O, H, H, F, OEt, O, O, OMe], [AI 1 667; Et, H, Me, H, O, H, H, F, SMe, O, O, OMe], [AI1668; Et, H, Me, H, O, H, H, F, CF 3, O, O, OMe], [AI1669; H, H , Et, H, O, H, H, F, H, O, O, OMe], [AI 1670; H, H, Et, H, O, H, F, F, O, O, OMe], [AI1671; H, H, Et, H, O, H, H, F, Cl, O, OMe], [AI1672; H, H, Et, H, O, H, H, F, Br, O , O, OMe], [AI1673; H, H, Et, H, O, H, H, F, I, O, O, OMe], [AI 1674; H, H, Et, H, O, H, H H, H, Et, H, Et, H, O, H, H, F, Et, O, O, OMe], [AI 1 676; H, H, Et, H. , O, H, H, F, c-Pr, O, O, OMe], [AI 1677; H, H, Et, H, O, H, F, OMe, O, O, OMe], [AI 1678 H, H, Et, H, O, H, H, F, OEt, O, O, OMe], [AI 1679; H, H, Et, H, O, H, H, F, SMe, O, O, OMe] , [AI1680; H, H, Et, H, O, H, H, F, CF 3, O, O, OMe], [AI1681; Cl, H, Et, H, O , H, H, F, H, O, O, OMe], [AI1682; Cl, H, Et, H, O, H, H, F, F, O, O, OMe], [AI 1683; Cl, H , Et, H, O, H, H, F, Cl, O, O, Oe], [AI 1684; Cl, H, Et, H, O, H, H, F, Br, O, O, OMe], [AI 1 685; Cl, H, Et, H, O, H, H, F, I, O, O, OMe], [AI 1686; Cl, H, Et, H, O, H, H, F, Me, O , O, OMe], [AI 1687; Cl, H, Et, H, O, H, H, F, Et, O, O, OMe], [AI 1688; Cl, H, Et, H, O, H, H , F, c-Pr, O, O, OMe], [AI 1689; Cl, H, Et, H, O, H, H, F, OMe, O, O, OMe], [AI 1690; Cl, H, Et , H, O, H, H, F, OEt, O, O, OMe], [AI1691; Cl, H, Et, H, O, H, F, SMe, O, O, OMe], [AI1692 ; Cl, H, Et, H , O, H, H, F, CF 3, O, O, OMe], [AI1693; Me, H, Et, H, O, H, H, F, H, O, O, OMe], [AI 1694; Me, H, Et, H, O, H, H, F, F, O, O, OMe], [AI 1695; Me, H, Et, H, O, H, H, F, Cl, O, O, OMe], [AI1696; Me, H, Et, H, O, H, H, F, Br, O, O, OMe], [AI 1697; Me, H, Et, H, O, H, H, F, I, O, O, OMe], [AI 1698; Me, H, Et, H, O, H, H, F, Me, O, O, OMe], [AI 1699; H, Et, H, O, H, H, F, Et, O, O, OMe], [AI1700; Me, H, Et, H, O, H, H, F, c-Pr, O, O, OMe],

[AI 1701; Me, H, Et, H, O, H, H, F, OMe, O, O, OMe], [AI 1702; Me, H, Et, H, O, H, H, F, OE t, O , O, OMe], [AI1703; Me, H, Et, H, O, H, H, F, SMe, O, O, OMe], [AI 1704; Me, H, Et, H, O, H, H _{, F, CF 3, O,} O, OMe], [AI1705; Et, H, Et, H, O, H, H, F, H, O, O, OMe], [AI1706; Et, H, Et, H, O, H, H, F, F, F, O, O, OMe], [AI 1707; Et, H, Et, H, O, H, H, F, Cl, O, O, OMe], [AI 1708; Et, H, Et, H, O, H, H, H, F, Br, O, O, OMe], [AI 1709; Et, H, Et, H, O, H, H, F, I, O, O, OMe], [AI 1710; Et, H, Et, H, O, H, H, F, Me, O, O, OMe], [AI 1711; Et, H, Et, H, O, H, H, F, Et, O, O, OMe], [AI 1712; Et, H, Et, H, O, H, H, F, c, Pr, O, O, OMe], [AI 1713; Et, H, Et, H, O, H, H, F, OMe, O, O, OMe], [AI1714; Et, H, Et, H, O, H, H, F, OEt, O, O, OMe], [AI 1715; Et, H, Et, H, O, H, H, F, SMe, O, O, OMe], [AI1716; Et, H, Et, H, O, H, H, F, CF 3, O, O, OMe H, H, H, H, O, H, H, H, H, O, S, OMe], [AI 1718; H, H, H, H, O, H, H, H, F] H, H, H, H, H, O, H, H, H, Cl, O, S, OMe], [AI 1720; H, H, H, H, O, H , H, H, Br, O, S, OMe], [AI1721; H, H, H, H, H, O, H, H, H, I, O, S, OMe], [AI 1722; H, H, H , H, O, H, H, H, H, Me, O, S, OMe], [AI1723; H, H, H, H, H, O, H, H, Et, O, S, OMe], [AI 1724 H, H, H, H, H, O, H, H, H, c, Pr, O, S, OMe], [AI1725; H, H, H, H, O, H, H, H, OMe, O , S, OMe], [AI1726; H, H, H, H, O, H, H, H, OEt, O, S, OMe], [AI 1727; H, H, H, H, O, H, H, H, SMe, O, S, OMe], [AI1728; H, H, H, H, O, H, H, H, CF 3, O, S, OMe], [AI1729; Cl, H, H , H, O, H, H, H, H, H, O, S, OMe], [AI 1730; Cl, H, H, H, O, H, H, H, F, O, S, OMe], [AI1731 Cl, H, H, H, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1732; Cl, H, H, H, H, O, H, H, H, Br, O, S , OMe], [AI1733; Cl, H, H, H, O, H, H, H, I, O, S, OMe], [AI 1734; Cl, H, H, H, O, H, H, H , Me, O, S, OMe], [AI 1735; Cl, H, H, H, H, O, H, H, H, Et, O, S, OMe], [AI 1 736; Cl, H, H, H, H, O , H, H, H, c-Pr, O, S, OMe], [AI 1 737; Cl, H, H, H, H, O, H, H, H, OMe, O, S, OMe], [AI 1 738; Cl , H, H, H, O, H, H, H, OEt, O, S, OMe], [AI 1739; Cl, H, H, H, O, H, H, S, O, S, OMe ], [AI1740; Cl, H , H, H, O, H, H, H, CF 3, O, S, OMe], [AI1741; Me, H, H, H, O, H, H, H, H, O, S, OMe], [AI 1742; Me, H, H, H, O, H, H, H, H, F, O, S, OMe], [AI 1743; Me, H, H, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1 744; Me, H, H, H, H, O, H, H, H, Br, O, S, OMe], [AI 1 745: Me, H, H, H, O, H, H, H, I, I, O, S, OMe], [AI 1746; Me, H, H, H, O, H, H, Me, O, S, OMe], [ AI 1 747; Me, H, H, H, H, O, H, H, H, Et, O, S, OMe], [AI 1 748; Me, H, H, H, H, O, H, H, H, c-Pr, O, S, OMe], [AI 1749; Me, H, H, H, O, H, H, H, H, OMe, O, S, OMe], [AI 1 750; Me, H, H, H, O, H, H, H, OEt, O, S, OMe], [AI1751; Me, H, H, H, H, O, H, H, S, O, S, OMe], [AI1752; Me, H, H, H, O, H, H, H, CF 3, O, S, OMe], [AI1753; Et, H, H, H, O, H, H, H, H, O, S, OMe], [AI1754 ; Et , H, H, H, O, H, H, H, H, F, O, S, OMe], [AI 1755; Et, H, H, H, O, H, H, H, Cl, O, S, OMe ], [AI 1756; Et, H, H, H, H, O, H, H, H, Br, O, S, OMe], [AI 1757; Et, H, H, H, O, H, H, H, I , O, S, OMe], [AI 1758; Et, H, H, H, H, O, H, H, H, Me, O, S, OMe], [AI 1759; Et, H, H, H, O, H , H, H, Et, O, S, OMe], [AI 1760; Et, H, H, H, H, O, H, H, c, Pr, O, S, OMe], [AI 1761; Et, H , H, H, O, H, H, H, H, OMe, O, S, OMe], [AI 1762; Et, H, H, H, H, O, H, H, H, OEt, O, S, OMe], [AI1763; Et, H, H, H, H, O, H, H, SMe, O, S, OMe], [AI 1764; Et, H, H, H, H, O, H, H, H, CF ₃ , O, S, OMe], [AI 1765; H, H, F, H, O, H, H, H, H, O, S, OMe], [AI 1766; H, H, F, H, O, H, H, H, F, O, S, OMe], [AI 1767; H, H, F, H, O, H, H, H, Cl, O, S, OMe], [AI 1768; H, H, F, H, O, H, H, H, H, Br, O, S, OMe], [AI 1769; H, H, F, H, O, H, H, H, I, O, S, OMe], [AI 1 770; H, H, F, H, O, H, H, H, Me, O, S, OMe], [AI 1771; H, H, F, H, O, H, H, H, Et, O, S, OMe], [AI1772; H, H, F, H, O, H, H, H, c-Pr, O, S, OMe], [AI1773; H, H, F, H, O, H, H, H, OMe, O, S, OMe], [AI 1774; H, H, F, H, O, H, H, H, OEt, O, S, OMe], [AI 1 775; H, H, F, H, O, H, H, H, SMe, O, S, OMe], [AI1776; H, H, F, H, O, H, H, H, CF 3, O, S, OMe], [AI1777; Cl , H, F, H, O, H, H, H, H, H, O, S, OMe], [AI 1778; Cl, H, F, H, O, H, H, F, O, S, OMe ], [AI 1779; Cl, H, F, H, O, H, H, H, Cl, O, S, OMe], [AI 1 780; Cl, H, F, H, O, H, H, H, Br] , O, S, OMe], [AI 1781; Cl, H, F , H, O, H, H, H, H, I, O, S, OMe], [AI 1782; Cl, H, F, H, O, H, H, Me, O, S, OMe], [AI 1783 Cl, H, F, H, O, H, H, H, H, Et, O, S, OMe], [AI 1784; Cl, H, F, H, O, H, H, H, c-Pr, O , S, OMe], [AI 1785; Cl, H, F, H, O, H, H, H, OMe, O, S, OMe], [AI 1786; Cl, H, F, H, O, H, H , H, OEt, O, S, OMe], [AI 1787; Cl, H, F, H, O, H, H, H, SMe, O, S, OMe], [AI 1 788; Cl, H, F, H , O, H, H, H , CF 3, O, S, OMe], [AI1789; Me, H, F, H, O, H, H, H, H, O, S, OMe], [AI1790; Me, H, F, H, O, H, H, H, H, F, O, S, OMe], [AI1791; Me, H, F, H, O, H, H, H, Cl, O, S, OMe], [AI1792; Me, H, F, H, O, H, H, H, Br, O, S, OMe], [AI 1793; Me, H, F, H, O, H, H, H, I, O, S, OMe], [AI 1794; Me, H, F, H, O, H, H, H, Me, O, S, OMe], [AI 1795: Me, H, F, H, O, H, H, H, H, Et, O, S, OMe], [AI 1796; Me, H, F, H, O, H, H, H, c-Pr, O, S, OMe], [AI 1 797; H, F, H, O, H, H, H, H, OMe, O, S, OMe], [AI 1798; Me, H, F, H, O, H, H, H, OEt, O, S, OMe] , [AI1799; Me, H, F, H, O, H, H, SMe, O, S, OMe], [AI1800; Me, H, F, H, O, H, H, H, CF ₃ , O, S, OMe],

[AI 1801; Et, H, F, H, O, H, H, H, H, O, S, OMe], [AI 1802; Et, H, F, H, O, H, H, H, F, O , S, OMe], [AI 1803; Et, H, F, H, O, H, H, H, Cl, O, S, OMe], [AI 1804, Et, H, F, H, O, H, H , H, Br, O, S, OMe], [AI 1805; Et, H, F, H, O, H, H, H, I, O, S, OMe], [AI 1 806; Et, H, F, H , O, H, H, H, H, Me, O, S, OMe], [AI 1807; Et, H, F, H, O, H, H, H, Et, O, S, OMe], [AI 1 808; , H, F, H, O, H, H, H, c, Pr, O, S, OMe], [AI 1809; Et, H, F, H, O, H, H, H, OMe, O, S , OMe], [AI 1810; Et, H, F, H, O, H, H, H, OEt, O, S, OMe], [AI 1811; Et, H, F, H, O, H, H, H , SMe, O, S, OMe ], [AI1812; Et, H, F, H, O, H, H, H, CF 3, O, S, OMe], [AI1813; H, H, Cl, H, O, H, H, H, H, H, O, S, OMe], [AI 1814; H, H, Cl, H, O, H, H, F, O, S, OMe], [AI 1815; H, H, Cl, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1816; H, H, Cl, H, O, H, H, H, Br, O, S, OMe] , [AI1817; H, H, Cl, H, O, H, H, I, O, S, OMe], [AI 1818; H, H, Cl, H, O, H, H, H, Me, O, S, OMe], [AI 1819; H, H, Cl, H, O, H, H, H, Et, O, S, OMe], [AI 1820; H, H, Cl, H, O, H, H, H, c-Pr, O, S, OMe], [AI 1821; H, H, Cl, H, O, H, H, H, OMe, O, S, OMe], [AI 1 822; H, H, Cl, H, O, H, H, H, OEt, O, S, OMe], [AI 1823; H, H, Cl, H, O, H, H, SMe, O, S, OMe], [ AI1824; H, H, Cl, H, O, H, H, H, CF 3, O, S, OMe], [AI1825; Cl, H, Cl, H, O, H, H, H, H, O , S, OMe], [AI 1826; Cl, H, Cl, H, O, H, H, H, H, F, O, S, OMe], [AI 1827; Cl, H, Cl, H, O, H, H , H, Cl Cl, H, Cl, H, O, H, H, H, H, Br, O, S, OMe], [AI 1829; Cl, H, Cl, H, O, H , H, H, I, O, S, OMe], [AI 1830; Cl, H, Cl, H, O, H, H, H, Me, O, S, OMe], [AI 1831; Cl, H, Cl , H, O, H, H, H, H, Et, O, S, OMe], [AI 1832; Cl, H, Cl, H, O, H, H, c, Pr, O, S, OMe], [AI1833; Cl, H, Cl, H, O, H, H, OMe, O, S, OMe], [AI 1834; Cl, H, Cl, H, O, H, H, H, OEt, O , S, OMe], [AI 1835; Cl, H, Cl, H, O, H, H, H, SMe, O, S, OMe], [AI 1836; Cl, H, Cl, H, O, H, H _{, H, CF 3, O,} S, OMe], [AI1837; Me, H, Cl, H, O, H, H, H, H, O, S, OMe], [AI1838; Me, H, Cl, H, O, H, H, H, H, F, O, S, OMe], [AI 1839; Me, H, Cl, H, O, H, H, H, Cl, O, S, OMe], [AI 1840; Me, H, Cl, H, O, H, H, H, H, Br, O, S, OMe], [AI 1841; Me, H, Cl, H, O, H, H, H, I, O, S, OMe], [AI1842; Me, H, Cl, H, O, H, H, H, Me, O, S, OMe], [AI1843; Me, H, Cl, H, O, H, H, H, Et, O, S, OMe], [AI 1844; Me, H, Cl, H, O, H, H, H, c, Pr, O, S, OMe], [AI 1845; Me, H, Cl, H, O, H, H, H, H, OMe, O, S, OMe], [AI 1846; Me, H, Cl, H, O, H, H, H, OEt, O, S, OMe], [AI 1 847; Me, H, Cl, H, O, H, H, H, SMe, O, S, OMe], [AI1848; Me, H, Cl, H, O, H, H, H, CF 3, O, S, OMe ], [AI 1849; Et, H, Cl, H, O, H, H, H, H, H, O, S, OMe], [AI 1850; Et, H, Cl, H, O, H, H, H, F, , O, S, OMe], [AI 1851; Et, H, Cl, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1852; Et, H, Cl, H, O, H H, H, Br, O, S, OMe], [AI 1853; Et, H, Cl, H, O, H, H, H, I, O, S, OMe], [AI 1 854; Et, H, Cl, H, O, H, H, H, Me, O, S, OMe], [AI 1 855; Et, H, Cl, H, O, H, H, H, Et, O, S, OMe], [AI 1856; Et, H, Cl, H, O, H, H, H, c, Pr, O, S, OMe], [AI 1 857; Et, H, Cl, H, O, H, H, H, H, OMe, O, S, OMe], [AI 1858; Et, H, Cl, H, O, H, H, H, OEt, O, S, OMe], [AI 1859; Et, H, Cl, H, O, H, H, H, SMe, O, S, OMe], [AI1860; Et, H, Cl, H, O, H, H, H, CF 3, O, S , OMe], [AI 1861; H, H, Me, H, O, H, H, H, H, O, S, OMe], [AI 1862; H, H, Me, H, O, H, H, H , F, O, S, OMe], [AI 1863; H, H, Me, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1864; H, H, Me, H, O , H, H, H, Br, O, S, OMe], [AI 1865; H, H, Me, H, O, H, H, H, I, O, S, OMe], [AI 1 866; H, H , Me, H, O, H, H, H, Me, O, S, OMe], [AI 1867; H, H, Me, H, O, H, H, H, Et, O, S, OMe], [AI1868; H, H, Me, H, O, H, H, c, Pr, O, S, OMe], [AI 1869; H, H, Me, H, O, H, H, H, H, OMe , O, S, OMe], [AI 1 870; H, H, Me, H, O, H, H, H, H, OEt, O, S, OMe], [AI 1871; H, H, Me, H, O, H , H, H, SMe, O , S, OMe], [AI1872; H, H, Me, H, O, H, H, H, CF 3, O, S, OMe], [AI1873; Cl, H, Me, H, O, H, H, H, H, H, O, S, OMe], [AI 1874; Cl, H, Me, H, O, H, H, F, O, S, OMe], [ AI 1875; Cl, H, Me, H, O, H, H, H, Cl, O, S, OMe], [AI 1876; Cl, H, Me, H, O, H, H, H, Br, O, S, OMe], [AI 1877; Cl, H, Me, H, O, H, H, H, I, O, S, OMe], [AI 1878; Cl, H, Me, H, O, H, H, H, Me, O, S, OMe], [AI 1879; Cl, H, Me, H, O, H, H, H, Et, O, S, OMe], [AI 1 880] Cl, H, Me, H, O, H, H, H, c, Pr, O, S, OMe], [AI 1881; Cl, H, Me, H, O, H, H, H, OMe, O , S, OMe], [AI1882; Cl, H, Me, H, O, H, H, H, OEt, O, S, OMe], [AI 1883; Cl, H, Me, H, O, H, H , H, SMe, O, S, OMe], [AI 1884; Cl, H, Me, H, O, H, H, H, CF ₃ , O, S, OMe], [AI 1885; Me, H, Me, H, O, H, H, H, H, H, O, S, OMe], [AI 1886; Me, H, Me, H, O, H, H, H, F, O, S, OMe], [AI 1887; Me, H, Me, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1888; Me, H, Me, H, O, H, H, H, Br, O, S, OMe], [AI 1889; Me, H, Me, H, O, H, H, H, I, O, S, OMe], [AI 1890; Me, H, Me, H, O, H, H, H, Me, O, S, OMe], [AI1891; Me, H, Me, H, O, H, H, H, H, Et, O, S, OMe], [AI1892; Me, H, Me, H, O, H, H, H, c-Pr, O, S, OMe], [AI 1893; Me, H, Me, H, O, H, H, H, OMe, O, S, OMe], [AI 1894; Me, H, Me, H, O, H, H, H, H, OEt, O, S, OMe], [AI 1895; Me, H, Me, H, O, H, H, S, Me, O, S, OMe] , [AI1896; Me, H, Me, H, O, H, H, H, CF 3, O, S, OMe], [AI1897; Et, H, Me, H, O, H, H, H, H , O, S, OMe], [AI 1898; Et, H, Me, H, O, H, H, H, H, F, O, S, OMe], [AI 1899; Et, H, Me, H, O, H , H, H, Cl, O, S, OMe], [AI 1900; Et, H, Me, H, O, H, H, H, Br, O, S, OMe],

[AI1901; Et, H, Me, H, O, H, H, I, O, S, OMe], [AI1902; Et, H, Me, H, O, H, H, H, Me, O , S, OMe], [AI 1903; Et, H, Me, H, O, H, H, H, Et, O, S, OMe], [AI 1904; Et, H, Me, H, O, H, H , H, c-Pr, O, S, OMe], [AI 1905; Et, H, Me, H, O, H, H, H, OMe, O, S, OMe], [AI 1906; Et, H, Me , H, O, H, H, H, H, OEt, O, S, OMe], [AI 1 907; Et, H, Me, H, O, H, H, S Me, O, S, OMe], [AI 1908 ; Et, H, Me, H , O, H, H, H, CF 3, O, S, OMe], [AI1909; H, H, Et, H, O, H, H, H, H, O, S, OMe], [AI 1910; H, H, Et, H, O, H, H, H, H, F, O, S, OMe], [AI 1911; H, H, Et, H, O, H, H, H, Cl, O, S, OMe], [AI1912; H, H, Et, H, O, H, H, H, H, Br, O, S, OMe], [AI1913; H, H, Et, H, O, H, H, H, H, I, O, S, OMe], [AI1914; H, H, Et, H, O, H, H, H, Me, O, S, OMe], [AI 1915; H, H, Et, H, O, H, H, H, H, Et, O, S, OMe], [AI1916; H, H, Et, H, O, H, H, H, c-Pr, O, S, OMe], [AI1917; H, H, Et, H, O, H, H, H, OMe, O, S, OMe], [AI 1918; H, H, Et, H, O, H, H, H, H, OEt, O, S, OMe], [AI 1919; H, H, Et, H, O, H, H, H, SMe, O, S, OMe], [AI 1920; H, H, Et, H, O, _{H, H, H, CF 3} , O, S, OMe], [AI1921; Cl, H, Et, H, O, H, H, H, H, O, S, OMe], [AI1922; Cl, H , Et, H, O, H, H, H, H, F, O, S, OMe], [AI1923; Cl, H, Et, H, O, H, H, H, Cl, O, S, OMe], [AI1924; Cl, H, Et, H, O, H, H, H, Br, O, S, OMe], [AI 1 925; Cl, H, Et, H, O, H, H, H, I, O , S, OMe], [AI 1926; Cl, H, Et, H, O, H, H, H, Me, O, S, OMe], [AI 1 927; Cl, H, Et , H, O, H, H, H, H, Et, O, S, OMe], [AI 1928; Cl, H, Et, H, O, H, H, c, Pr, O, S, OMe], [AI 1 929; Cl, H, Et, H, O, H, H, OMe, O, S, OMe], [AI 1930; Cl, H, Et, H, O, H, H, H, OEt, O , S, OMe], [AI1931; Cl, H, Et, H, O, H, H, H, SMe, O, S, OMe], [AI 1932; Cl, H, Et, H, O, H, H , H, CF ₃ , O, S, OMe], [AI 1933; Me, H, Et, H, O, H, H, H, H, O, S, OMe], [AI 1 934; Me, H, Et, H, O, H, H, H, H, F, O, S, OMe], [AI 1935; Me, H, Et, H, O, H, H, H, Cl, O, S, OMe], [AI 1936; Me, H, Et, H, O, H, H, H, H, Br, O, S, OMe], [AI 1937; Me, H, Et, H, O, H, H, H, I, O, S, OMe], [AI 1938; Me, H, Et, H, O, H, H, H, Me, O, S, OMe], [AI 1939; Me, H, Et, H, O, H, H, H, Et, O, S, OMe], [AI1940; Me, H, Et, H, O, H, H, H, c, Pr, O, S, OMe], [AI1941; Me, H, Et, H, O, H, H, H, H, OMe, O, S, OMe], [AI1942; Me, H, Et, H, O, H, H, H, OEt, O, S, OMe], [AI1943; Me, H, Et, H, O, H, H, H, SMe, O, S, OMe], [AI1944; Me, H, Et, H, O, H, H, H, CF 3, O, S, OMe ], [AI 1945; Et, H, Et, H, O, H, H, H, H, H, O, S, OMe], [AI 1946; Et, H, Et, H, O, H, H, H, F , O, S, OMe], [AI1947; Et, H, Et, H, O, H, H, H, H, Cl, O, S, OMe], [AI 1948; Et, H, Et, H, O, H , H, H, Br, O, S, OMe], [AI 1 949; Et, H, Et, H, O, H, H, H, I, O, S, OMe], [AI 1950; Et, H, Et , H, O, H, H, H, H, Me, O, S, OMe], [AI1951; Et, H, Et, H, O, H, H, H, Et, O, S, OMe], [AI1952 Et, H, Et, H, O, H, H, H, c, Pr, O, S, OMe], [AI1953; Et, H, Et , H, O, H, H, H, H, OMe, O, S, OMe], [AI1954; Et, H, Et, H, O, H, H, H, OEt, O, S, OMe], [AI 1 955] ; Et, H, Et, H , O, H, H, H, SMe, O, S, OMe], [AI1956; Et, H, Et, H, O, H, H, H, CF 3, O, S, OMe], [AI 1957; H, H, H, H, H, O, H, H, H, H, NH, O, OMe], [AI 1958; H, H, H, H, O, H, H, H, F, NH, O, OMe], [AI1959; H, H, H, H, H, O, H, H, H, H, Cl, NH, O, OMe], [AI1960; H, H, H, H, O, H, H, H, H, Br, NH, O, OMe], [AI 1961; H, H, H, H, H, O, H, H, H, I, NH, O, OMe], [AI 1962; H, H, H, H, H, O, H, H, H, Me, NH, O, OMe], [AI1963; H, H, H, H, H, O, H, H, Et, NH, O, OMe] [AI 1964; H, H, H, H, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 1 965; H, H, H, H, O, H, H, H, H, OMe, NH, O, OMe], [AI1966; H, H, H, H, O, H, H, H, H, OEt, NH, O, OMe], [AI 1967; H, H, H, H, O, H, H, H, SMe, NH, O, OMe], [AI1968; H, H, H, H, O, H, H, H, CF 3, NH, O, OMe], [AI1969; F, H , H, H, O, H, H, H, H, NH, O, OMe], [AI1970; F, H, H, H, O, H, H, H, F, NH, O, OMe], [AI 1971; F, H, H, H, H, O, H, H, H, Cl, NH, O, OMe], [AI 1972; F, H, H, H, O, H, H, H, Br, NH , O, OMe], [AI 1973; F, H, H, H, O, H, H, H, I, NH, O, OMe], [AI 1974; F, H, H, H, O, H, H , H, Me, NH, O, OMe], [AI1975; F, H, H, H, H, O, H, H, H, Et, NH, O, OMe], [AI1976; F, H, H, H , O, H, H, H, c, Pr, NH, O, OMe], [AI 1977; F, H, H, H, H, O, H, H, H, OM, NH, O, OMe], [AI1978 F, H, H, H, H, O, H, H, H, OEt, NH, O, OMe], [AI 1979; F, H, H, H, H, O, H, H, SMe, NH, O , OMe] , [AI1980; F, H, H, H, O, H, H, H, CF 3, NH, O, OMe], [AI1981; Cl, H, H, H, O, H, H, H, H , NH, O, OMe], [AI 1982; Cl, H, H, H, H, O, H, H, H, F, NH, O, OMe], [AI 1983; Cl, H, H, H, O, H , H, H, Cl, NH, O, OMe], [AI1984; Cl, H, H, H, H, O, H, H, H, Br, NH, O, OMe], [AI1985; Cl, H, H , H, O, H, H, H, H, I, NH, O, OMe], [AI 1986; Cl, H, H, H, H, O, H, H, Me, NH, O, OMe], [AI 1987] Cl, H, H, H, H, O, H, H, H, H, Et, NH, O, OMe], [AI1988; Cl, H, H, H, H, O, H, H, H, c-Pr, NH , O, OMe], [AI1989; Cl, H, H, H, H, O, H, H, H, OMe, NH, O, OMe], [AI 1990; Cl, H, H, H, O, H, H , H, OEt, NH, O, OMe], [AI 1991; Cl, H, H, H, H, O, H, H, H, SMe, NH, O, OMe], [AI 1992; Cl, H, H, H , O, H, H, H , CF 3, NH, O, OMe], [AI1993; Br, H, H, H, O, H, H, H, H, NH, O, OMe], [AI1994; Br, H, H, H, O, H, H, H, H, F, NH, O, OMe], [AI1995; Br, H, H, H, H, O, H, H, H, Cl, NH, O, OMe], [AI1996; Br, H, H, H, O, H, H, H, Br, NH, O, OMe], [AI 1997; Br, H, H, H, O, H, H, H, H, I, NH, O, OMe], [AI1998; Br, H, H, H, H, O, H, H, H, Me, NH, O, OMe], [AI1999; Br, H, H, H, O, H, H, H, H, Et, NH, O, OMe], [AI 2000; Br, H, H, H, O, H, H, H, c-Pr, NH, O, OMe],

[AI 2001; Br, H, H, H, O, H, H, OMe, NH, O, OMe], [AI 2002; Br, H, H, H, H, O, H, H, H, OEt, NH , O, OMe], [AI2003; Br, H, H, H, O, H, H, H, SMe, NH, O, OMe], [AI 2004; Br, H, H, H, O, H, H _{, H, CF 3, NH,} O, OMe], [AI2005; Me, H, H, H, O, H, H, H, H, NH, O, OMe], [AI2006; Me, H, H, H, O, H, H, H, H, F, NH, O, OMe], [AI2007; Me, H, H, H, H, O, H, H, H, Cl, NH, O, OMe], [AI 2008; Me, H, H, H, H, O, H, H, H, H, Br, NH, O, OMe], [AI2009; Me, H, H, H, O, H, H, H, I, NH, O, OMe], [AI2010; Me, H, H, H, O, H, H, H, Me, NH, O, OMe], [AI 2011; Me, H, H, H, O, H, H, H, H, Et, NH, O, OMe], [AI2012; Me, H, H, H, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2013; Me, H, H, H, O, H, H, H, H, OMe, NH, O, OMe], [AI2014; Me, H, H, H, H, O, H, H, H, OEt, NH, O, OMe], [AI2015; H, H, H, O, H, H, H, SMe, NH, O, OMe], [AI2016; Me, H, H, H, O, H, H, H, CF 3, NH, O, OMe ], [AI 2017; Et, H, H, H, H, O, H, H, H, H, NH, O, OMe], [AI 2018; Et, H, H, H, O, H, H, H, F, , NH, O, OMe], [AI 2019; Et, H, H, H, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2020; Et, H, H, H, O, H , H, H, Br, NH, O, OMe], [AI 2021; Et, H, H, H, H, O, H, H, H, I, NH, O, OMe], [AI 2022; Et, H, H , H, O, H, H, H, Me, NH, O, OMe], [AI2023; Et, H, H, H, H, O, H, H, H, Et, NH, O, OMe], [AI 2024 Et, H, H, H, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2025; Et, H, H, H, H, O, H, H, H, OMe, NH , O, OMe], [AI 2026; Et, H, H, H, H, O, H, H, H, OEt, NH, O, OMe], [AI2027; Et, H, H, H, H, O, H, H, SMe, NH, O, OMe], [AI 2028; Et, H, H, H, H, O, H, H, H, CF ₃ , NH, O, OMe], [ AI2029; CF 3, H, H, H, O, H, H, H, H, NH, O, OMe], [AI2030; CF 3, H, H, H, O, H, H, H, F, NH, O, OMe], [AI2031; CF 3, H, H, H, O, H, H, H, Cl, NH, O, OMe], [AI2032; CF 3, H, H, H, O, H, H, H, Br, NH, O, OMe], [AI2033; CF 3, H, H, H, O, H, H, H, I, NH, O, OMe _{], [AI2034; CF 3,} H, H, H, O, H, H, H, Me, NH, O, OMe], [AI2035; CF 3, H, H, H, O, H, H, H , Et, NH, O, OMe ], [AI2036; CF 3, H, H, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2037; CF 3, H, H , H, O, H, H , H, OMe, NH, O, OMe], [AI2038; CF 3, H, H, H, O, H, H, H, OEt, NH, O, OMe], [ AI 2039; CF ₃ , H, H, H, O, H, H, S Me, NH, O, OMe], [AI 2040; CF ₃ , H, H, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI 2041; c-Pr, H, H, H, H, O, H, H, H, H, NH, O, OMe], [AI 2042; c-Pr, H, H, H , O, H, H, H, H, F, NH, O, OMe], [AI 2043; c-Pr, H, H, H, H, O, H, H, H, Cl, NH, O, OMe], [AI 2044 c-Pr, H, H, H, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2045; c-Pr, H, H, H, O, H, H, H, I , NH, O, OMe], [AI 2046; c-Pr, H, H, H, H, O, H, H, H, Me, NH, O, OMe], [AI 2047; c-Pr, H, H, H , O, H, H, H, Et, NH, O, OMe], [AI 2048; c-Pr, H, H, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2049; c-Pr, H, H, H, O, H, H, H, OMe, NH, O, OMe], [AI 2050; c-Pr, H, H, H, O, H, H, H , OEt, NH, O, OMe], [AI 2051; c-Pr, H, H, H, O, H , H, H, SMe, NH , O, OMe], [AI2052; c-Pr, H, H, H, O, H, H, H, CF 3, NH, O, OMe], [AI2053; H, H, F, H, O, H, H, H, H, H, NH, O, OMe], [AI 2054; H, H, F, H, O, H, H, F, NH, O, OMe] , [AI 2055; H, H, F, H, O, H, H, H, Cl, NH, O, OMe], [AI 2056; H, H, F, H, O, H, H, H, Br, NH, O, OMe], [AI 2057; H, H, F, H, O, H, H, H, I, NH, O, OMe], [AI 2058; H, H, F, H, O, H, H, H, Me, NH, O, OMe], [AI 2059; H, H, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2060; H, H, F, H, O, H, H, H, c, Pr, NH, O, OMe], [AI2061; H, H, F, H, O, H, H, H, OMe, NH, O, OMe], [ AI2062; H, H, F, H, O, H, H, OEt, NH, O, OMe], [AI 2063; H, H, F, H, O, H, H, H, SMe, NH, O, OMe], [AI 2064; H, H, F, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI 2065; F, H, F, H, O, H, H , H, H, NH, O, OMe], [AI 2066; F, H, F, H, O, H, H, H, F, NH, O, OMe], [AI 2067; F, H, F, H , O, H, H, H, Cl, NH, O, OMe], [AI 2068; F, H, F, H, O, H, H, H, Br, NH, O, OMe], [AI 2069; F , H, F, H, O, H, H, H, I, NH, O, OMe], [AI 2070; F, H, F, H, O, H, H, H, Me, NH, O, OMe ], [AI 2071; F, H, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2072; F, H, F, H, O, H, H, H, c -Pr, NH, O, OMe], [AI 2073; F, H, F, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2074; F, H, F, H, O , H, H, H, OEt, NH, O, OMe], [AI 2075; F, H, F, H, O, H, H, H, SMe, NH, O, OMe], [AI 2076; F, H , F, H, O, H , H, H, CF 3, NH, O, OMe], [AI2077; Cl, H, F, H, O, H, H, H, H, NH, O, OMe] , [AI 2078; Cl, H, F, H, O, H, H, H, F, NH, O, OMe], [AI 2079; Cl, H, F, H, O, H, H, H, Cl, NH, O, OMe], [AI 2080; Cl, H, F, H, O, H, H, H, Br, NH, O, OMe], [AI 2081; Cl, H, F, H, O, H, H, H, I, NH, O, OMe], [AI2082; Cl, H, F, H, O, H, H, H, Me, NH, O, OMe], [AI 2083; Cl, H, F, H, O, H, H, H, H, Et, NH, O, OMe], [AI 2084; Cl, H, F, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2085; Cl, H, F, H, O, H, H, H, OMe, NH, O, OMe], [AI 2086; Cl, H, F, H, O, H, H, H, OEt, NH, O, OMe], [AI 2087; Cl, H, F, H, O, H, H, S, NH, O, OMe], [AI 2088; Cl, H, F, H, O, H, H, H, H, _{CF 3, NH, O, OMe} ], [AI2089; Br, H, F, H, O, H, H, H, H, NH, O, OMe], [AI2090; Br, H, F, H, O , H, H, H, F, NH, O, OMe], [AI2091; Br, H, F, H, O, H, H, H, Cl, NH, O, OMe], [AI2092; Br, H , F, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2093; Br, H, F, H, O, H, H, H, I, NH, O, OMe], [AI 2094; Br, H, F, H, O, H, H, Me, NH, O, OMe], [AI 2095; Br, H, F, H, O, H, H, H, Et, NH , O, OMe], [AI 2096; Br, H, F, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2097; Br, H, F, H, O, H , H, H, OMe, NH, O, OMe], [AI 2098; Br, H, F, H, O, H, H, H, OEt, NH, O, OMe], [AI 2099; Br, H, F , H, O, H, H , H, SMe, NH, O, OMe], [AI2100; Br, H, F, H, O, H, H, H, CF 3, NH, O, OMe],

[AI2101; Me, H, F, H, O, H, H, H, H, NH, O, OMe], [AI 2102; Me, H, F, H, O, H, H, H, F, NH , O, OMe], [AI 2103; Me, H, F, H, O, H, H, H, Cl, NH, O, OMe], [AI 2104; Me, H, F, H, O, H, H , H, Br, NH, O, OMe], [AI 2 105; Me, H, F, H, O, H, H, H, I, NH, O, OMe], [AI 2106; Me, H, F, H , O, H, H, H, Me, NH, O, OMe], [AI 2 107; Me, H, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2 108; Me , H, F, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2109; Me, H, F, H, O, H, H, H, OMe, NH, O , OMe], [AI 2110; Me, H, F, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 111; Me, H, F, H, O, H, H, H , SMe, NH, O, OMe ], [AI2112; Me, H, F, H, O, H, H, H, CF 3, NH, O, OMe], [AI2113; Et, H, F, H, O, H, H, H, H, H, NH, O, OMe], [AI 2114; Et, H, F, H, O, H, H, H, F, NH, O, OMe], [AI 2 115; Et, H, F, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2116; Et, H, F, H, O, H, H, H, Br, NH, O, OMe] [AI 2 117; Et, H, F, H, O, H, H, I, NH, O, OMe], [AI 2 118; Et, H, F, H, O, H, H, H, Me, NH, O, OMe], [AI 2 119; Et, H, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2 120; Et, H, F, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2121; Et, H, F, H, O, H, H, H, OMe, NH, O, OMe], [AI 2122; Et, H, F, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 123; Et, H, F, H, O, H, H, S Me, NH, O, OMe], [ AI2124; Et, H, F, H, O, H, H, H, CF 3, NH, O, OMe], [AI2125; CF 3, H, F, H, O, H, H, H, H, NH, O, OMe], [ AI2126; CF 3, H, F, H, O, H, H, H, F, NH, O, OMe _{], [AI2127; CF 3,} H, F, H, O, H, H, H, Cl, NH, O, OMe], [AI2128; CF 3, H, F, H, O, H, H, H , Br, NH, O, OMe ], [AI2129; CF 3, H, F, H, O, H, H, H, I, NH, O, OMe], [AI2130; CF 3, H, F, H , O, H, H, H, Me, NH, O, OMe], [AI 2 131; CF ₃ , H, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2 132; _{CF 3, H, F, H} , O, H, H, H, c-Pr, NH, O, OMe], [AI2133; CF 3, H, F, H, O, H, H, H, OMe, NH, O, OMe], [ AI2134; CF 3, H, F, H, O, H, H, H, OEt, NH, O, OMe], [AI2135; CF 3, H, F, H, O, H, H, H, SMe, NH, O, OMe], [AI2136; CF 3, H, F, H, O, H, H, H, CF 3, NH, O, OMe], [AI2137; H, H, Cl, H, O, H, H, H, H, H, NH, O, OMe], [AI 2138; H, H, Cl, H, O, H, H, F, NH, O, OMe] , [AI 2 139; H, H, Cl, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 140; H, H, Cl, H, O, H, H, H, Br, NH, O, OMe], [AI 2141; H, H, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2142; H, H, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI 2143; H, H, Cl, H, O, H, H, H, Et, NH, O, OMe], [AI 2 144; H, H, Cl, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2145; H, H, Cl, H, O, H, H, H, OMe, NH, O, OMe], [ AI 2146; H, H, Cl, H, O, H, H, OEt, NH, O, OMe], [AI 2147; H, H, Cl, H, O, H, H, H, SMe, NH, O, OMe], [AI 2 148; H, H, Cl, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI 2 149; F, H, Cl, H, O, H, H , H, H, NH, O, OMe], [AI 2150; F, H, Cl, H, O, H, H, H, H, F, NH, O, OMe], [AI 2151; F, H, Cl, H , O, H, H, H, H, Cl, NH, O, OMe], [AI2152; F, H, Cl, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2 153; F, H, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2154; F, H, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI 2 155; F, H, Cl, H, O, H, H, H, Et, NH, O, OMe], [AI 2156; F, H, Cl, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2 157; F, H, Cl, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2158; F, H, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 159; F, H, Cl, H, O, H, H, H, SMe, NH, O, OMe], [AI2160; F, H, Cl, H, O, H, H, H, CF 3, NH, O, OMe Cl, H, Cl, H, O, H, H, H, H, NH, O, OMe], [AI 2162; Cl, H, Cl, H, O, H, H, H, F] , NH, O, OMe], [AI 2 163; Cl, H, Cl, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2 164; Cl, H, Cl, H, O, H , H, H, Br, NH, O, OMe], [AI 2 165; Cl, H, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2 166; Cl, H, Cl , H, O, H, H, H, Me, NH, O, OMe], [AI 2 167; Cl, H, Cl, H, O, H, H, H, Et, NH, O, OMe], [AI 2 168] Cl, H, Cl, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2169; Cl, H, Cl, H, O, H, H, H, OMe, NH , O, OMe], [AI2170; Cl, H, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2171; Cl, H, Cl, H, O, H, H , H, SMe, NH, O , OMe], [AI2172; Cl, H, Cl, H, O, H, H, H, CF 3, NH, O, OMe], [AI2173; Br, H, Cl, H, O, H, H, H, H, H, NH, O, OMe], [AI 2 174; Br, H, Cl, H, O, H, H, F, NH, O, OMe], [AI 2 175; Br, H, Cl, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2176; Br, H, Cl, H, O, H, H, H, Br, NH, O, OMe], [AI2177; Br, H, Cl, H, O, H, H, H, I, NH, O , OMe], [AI2178; Br, H, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI 2179; Br, H, Cl, H, O, H, H, H , Et, NH, O, OMe], [AI 2180; Br, H, Cl, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2181; Br, H, Cl, H , O, H, H, H, H, OMe, NH, O, OMe], [AI 2182; Br, H, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2183; Br , H, Cl, H, O , H, H, H, SMe, NH, O, OMe], [AI2184; Br, H, Cl, H, O, H, H, H, CF 3, NH, O, OMe], [AI 2 185; Me, H, Cl, H, O, H, H, H, H, NH, O, OMe], [AI 2186; Me, H, Cl, H, O, H, H, H, F, NH, O, OMe], [AI 2187; Me, H, Cl, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2188; Me, H, Cl, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2189; Me, H, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2 190; Me, H, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI2191; Me, H, Cl, H, O, H, H, H, Et, NH, O, OMe], [ AI 2 192; Me, H, Cl, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2193; Me, H, Cl, H, O, H, H, H, OMe, NH, O, OMe], [AI 2194; Me, H, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2195; Me, H, Cl, H, O, H, H, H, SMe, NH, O, OMe], [AI2196; Me, H, Cl, H, O, H, H, H, CF 3, NH, O, OMe], [AI2197; Et, H, Cl , H, O, H, H, H, H, H, NH, O, OMe], [AI 2198; Et, H, Cl, H, O, H, H, H, F, NH, O, OMe], [AI 2199 Et, H, Cl, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2200; Et, H, Cl, H, O, H, H, H, Br, NH, O , OMe],

[AI 2201; Et, H, Cl, H, O, H, H, I, NH, O, OMe], [AI 2202; Et, H, Cl, H, O, H, H, H, Me, NH , O, OMe], [AI 2203; Et, H, Cl, H, O, H, H, H, Et, NH, O, OMe], [AI 2 204; Et, H, Cl, H, O, H, H , H, c-Pr, NH, O, OMe], [AI 2205; Et, H, Cl, H, O, H, H, H, OMe, NH, O, OMe], [AI 2206; Et, H, Cl , H, O, H, H, H, OEt, NH, O, OMe], [AI 2207; Et, H, Cl, H, O, H, H, S Me, NH, O, OMe], [AI 2208 ; Et, H, Cl, H , O, H, H, H, CF 3, NH, O, OMe], [AI2209; CF 3, H, Cl, H, O, H, H, H, H, NH , O, OMe], [AI2210 ; CF 3, H, Cl, H, O, H, H, H, F, NH, O, OMe], [AI2211; CF 3, H, Cl, H, O, H , H, H, Cl, NH , O, OMe], [AI2212; CF 3, H, Cl, H, O, H, H, H, Br, NH, O, OMe], [AI2213; CF 3, H , Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2214; CF ₃ , H, Cl, H, O, H, H, H, Me, NH, O, OMe] _{, [AI2215; CF 3, H} , Cl, H, O, H, H, H, Et, NH, O, OMe], [AI2216; CF 3, H, Cl, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2217; CF 3, H, Cl, H, O, H, H, H, OMe, NH, O, OMe], [AI2218; CF 3, H, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI2219; CF 3, H, Cl, H, O, H, H, H, SMe, NH, O, OMe], [AI2220 CF ₃ , H, Cl, H, O, H, H, H, H, CF ₃ , NH, O, OMe], [AI 2221; H, H, Me, H, O, H, H, H, H, NH , O, OMe], [AI2222; H, H, Me, H, O, H, H, H, F, NH, O, OMe], [AI 2223; H, H, Me, H, O, H, H , H, Cl, NH, O, OMe], [AI 2224; H, H, Me, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2225; H, H, Me, H , O, H, H , H, I, NH, O, OMe], [AI 2226; H, H, Me, H, O, H, H, H, Me, NH, O, OMe], [AI 2 227; H, H, Me, H , O, H, H, H, Et, NH, O, OMe], [AI 2228; H, H, Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2 229] H, H, Me, H, O, H, H, H, OMe, NH, O, OMe], [AI 2 230; H, H, Me, H, O, H, H, H, OEt, NH, O H, H, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI 2232; H, H, Me, H, O, H, H, H _{, CF 3, NH, O,} OMe], [AI2233; F, H, Me, H, O, H, H, H, H, NH, O, OMe], [AI2234; F, H, Me, H, O, H, H, H, H, F, NH, O, OMe], [AI 2 235; F, H, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 236; F, H, Me, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2 237; F, H, Me, H, O, H, H, H, I, NH, O, OMe] , [AI2238; F, H, Me, H, O, H, H, Me, NH, O, OMe], [AI 2239; F, H, Me, H, O, H, H, H, Et, NH, O, OMe], [AI 2 240; F, H, Me, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2241; F, H, Me, H, O, H, H, H, H, OMe, NH, O, OMe], [AI2242; F, H, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI 2243; F, H, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI2244; F, H, Me, H, O, H, H, H, CF 3, NH, O, OMe], [AI2245; Cl, H, Me, H, O, H, H, H, H, NH, O, OMe], [AI 2246; Cl, H, Me, H, O, H, H, H, F, NH , O, OMe], [AI2247; Cl, H, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI 2248; Cl, H, Me, H, O, H, H , H, Br, NH, O, OMe], [AI 2249; Cl, H, Me, H, O, H, H, H, I, NH, O, OMe], [AI 2 250; Cl, H, Me, H , O, H, H, H, Me, NH, O, OMe], [AI 2251; Cl, H, Me, H, O , H, H, H, Et, NH, O, OMe], [AI 2252; Cl, H, Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2 253; Cl , H, Me, H, O, H, H, H, OMe, NH, O, OMe], [AI 2254; Cl, H, Me, H, O, H, H, H, OEt, NH, O, OMe ], [AI2255; Cl, H, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI 2 256; Cl, H, Me, H, O, H, H, H, CF] ₃ , NH, O, OMe], [AI 2 257; Br, H, Me, H, O, H, H, H, H, H, NH, O, OMe], [AI 2 258; Br, H, Me, H, O, H, H, H, H, F, NH, O, OMe], [AI 2259; Br, H, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 260; Br, H, Me, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2261; Br, H, Me, H, O, H, H, H, I, NH, O, OMe], [ AI 2262; Br, H, Me, H, O, H, H, Me, NH, O, OMe], [AI 2263; Br, H, Me, H, O, H, H, H, Et, NH, O, OMe], [AI 2 264; Br, H, Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2 265; Br, H, Me, H, O, H, H, H, OMe, NH, O, OMe], [AI 2 266; Br, H, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 267; Br, H, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI2268; Br, H, Me, H, O, H, H, H, CF 3, NH, O, OMe], [AI2269 Me, H, Me, H, O, H, H, H, H, NH, O, OMe], [AI 2 270; Me, H, Me, H, O, H, H, H, F, NH, O , OMe], [AI2271; Me, H, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI 2272; Me, H, Me, H, O, H, H, H , Br, NH, O, OMe], [AI 2273; Me, H, Me, H, O, H, H, H, I, NH, O, OMe], [AI 2 274; Me, H, Me, H, O , H, H, H, Me, NH, O, OMe], [AI 2275; Me, H, Me, H, O, H, H, H, Et, NH, O, OMe], [AI 2276; Me, H , Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2 277; Me, H, Me, H, O, H, H, H, OMe, NH, O, OMe], [AI 2 278; Me, H, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI2279; Me, H, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI 2280; Me, H, Me, H, O, H, H, H, CF 3, NH, O, OMe], [AI2281; Et, H, Me, H, O, H, H, H, H, NH, O, OMe], [AI2282; Et , H, Me, H, O, H, H, H, F, NH, O, OMe], [AI 2283; Et, H, Me, H, O, H, H, H, Cl, NH, O, OMe ], [AI2284; Et, H, Me, H, O, H, H, H, Br, NH, O, OMe], [AI 2285; Et, H, Me, H, O, H, H, H, I , NH, O, OMe], [AI 2286; Et, H, Me, H, O, H, H, H, H, Me, NH, O, OMe], [AI 2 287; Et, H, Me, H, O, H , H, H, Et, NH, O, OMe], [AI 2 288; Et, H, Me, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2 289; Et, H , Me, H, O, H, H, H, OMe, NH, O, OMe], [AI 2290; Et, H, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI2291; Et, H, Me, H, O, H, H, SMe, NH, O, OMe], [AI 2 229; Et, H, Me, H, O, H, H, H, CF ₃ , NH, O, OMe], [ AI2293; CF 3, H, Me, H, O, H, H, H, H, NH, O, OMe], [AI2294; CF 3, H, Me, H, O, H, H, H, F, NH, O, OMe], [AI2295; CF 3, H, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI2296; CF 3, H, Me, H, O, H, H, H, Br, NH, O, OMe], [AI2297; CF 3, H, Me, H, O, H, H, H, I, NH, O, OMe _{], [AI2298; CF 3,} H, Me, H, O, H, H, H, Me, NH, O, OMe], [AI2299; CF 3, H, Me, H, O, H, H, H , Et, NH, O, OMe], [AI 2300; CF ₃ , H, Me, H, O, H, H, H, c, Pr, NH, O, OMe],

_{[AI2301; CF 3, H,} Me, H, O, H, H, H, OMe, NH, O, OMe], [AI2302; CF 3, H, Me, H, O, H, H, H, OEt , NH, O, OMe], [AI2303; CF 3, H, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI2304; CF 3, H, Me, H, O , H, H, H, CF 3, NH, O, OMe], [AI2305; H, H, Et, H, O, H, H, H, H, NH, O, OMe], [AI2306; H, H, Et, H, O, H, H, H, H, F, NH, O, OMe], [AI 2307; H, H, Et, H, O, H, H, H, Cl, NH, O, OMe] , [AI 2 308; H, H, Et, H, O, H, H, H, Br, NH, O, OMe], [AI 2 309; H, H, Et, H, O, H, H, H, I, NH, O, OMe], [AI 2310; H, H, Et, H, O, H, H, H, Me, NH, O, OMe], [AI 2311; H, H, Et, H, O, H, H, H, Et, NH, O, OMe], [AI2312; H, H, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI2313; H, H, Et, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2314; H, H, Et, H, O, H, H, H, OEt, NH, O, OMe], [ AI 2315; H, H, Et, H, O, H, H, SMe, NH, O, OMe], [AI 2316; H, H, Et, H, O, H, H, H, CF ₃ , NH , O, OMe], [AI 2317; F, H, Et, H, O, H, H, H, H, NH, O, OMe], [AI 2318; F, H, Et, H, O, H, H , H, F, NH, O, OMe], [AI 2319; F, H, Et, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 320; F, H, Et, H , O, H, H, H, H, Br, NH, O, OMe], [AI2321; F, H, Et, H, O, H, H, H, I, NH, O, OMe], [AI2322; F , H, Et, H, O, H, H, H, Me, NH, O, OMe], [AI 2323; F, H, Et, H, O, H, H, H, Et, NH, O, OMe ], [AI 2324; F, H, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2325; F, H, Et, H, O, H, H, H , OMe, NH, O, OMe], [AI 2326; F, H, Et, H, O, H, H, H, OEt, NH, O, OMe], [AI 2327; F, H, Et, H, O, H, H, H, S Me, NH, O, OMe], [AI 2 328; F, H, Et, H, O, H, H, H, CF 3, NH, O, OMe], [AI2329; Cl, H, Et, H, O, H, H, H, H, NH, O, OMe], [AI2330; Cl , H, Et, H, O, H, H, H, F, NH, O, OMe], [AI 2331; Cl, H, Et, H, O, H, H, H, Cl, NH, O, OMe ], [AI2332; Cl, H, Et, H, O, H, H, H, Br, NH, O, OMe], [AI 2333; Cl, H, Et, H, O, H, H, H, I , NH, O, OMe], [AI 2334; Cl, H, Et, H, O, H, H, H, Me, NH, O, OMe], [AI 2 335; Cl, H, Et, H, O, H , H, H, Et, NH, O, OMe], [AI 2336; Cl, H, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2 337; Cl, H , Et, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2338; Cl, H, Et, H, O, H, H, H, OEt, NH, O, OMe], [AI2339; Cl, H, Et, H, O, H, H, SMe, NH, O, OMe], [AI 2340; Cl, H, Et, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI2341; Br, H, Et, H, O, H, H, H, H, NH, O, OMe], [AI 2342; Br, H, Et, H, O, H, H, H, F, NH, O, OMe], [AI 2343; Br, H, Et, H, O, H, H, H, Cl, NH, O, OMe], [AI 2344; Br, H, Et, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2345; Br, H, Et, H, O, H, H, H, I, NH, O, OMe], [AI 2346; Br, H, Et, H, O, H, H, H, Me, NH, O, OMe], [AI 2347; Br, H, Et, H, O, H, H, H, Et, NH, O, OMe], [AI2348; Br, H, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2349; Br, H, Et, H, O, H, H, H, OMe, NH, O, OMe], [AI 2 350; Br, H, Et, H, O, H, H, H, H, OEt, NH, O, OMe], [AI 2351; Br, H, Et, H, O, H, H, H, SMe, NH, O, OMe], [AI2352; Br, H, Et , H, O, H, H, H, CF 3, NH, O, OMe], [AI2353; Me, H, Et, H, O, H, H, H, H, NH, O, OMe], [AI 2354; Me, H, Et, H, O, H, H, H, H, F, NH, O, OMe], [AI 2 355; Me, H, Et, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 356; Me, H, Et, H, O, H, H, H, Br, NH, O, OMe], [AI 2 357; Me, H, Et, H, O, H, H, H, I, NH, O, OMe], [AI 2358; Me, H, Et, H, O, H, H, Me, NH, O, OMe], [AI 2359; Me, H, Et, H, O, H, H, H, H, Et, NH, O, OMe], [AI 2 360; Me, H, Et, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2361; Me, H, Et, H, O, H, H, H, OMe, NH, O, OMe], [AI2362; Me, H, Et, H, O, H, H, H, OEt, NH, O, OMe], [AI2363; Me, H, Et, H, O, H, H, H, SMe, NH, O, OMe], [AI 2364; Me, H, Et, H, O, H, H, H, CF 3, NH, O, OMe], [AI2365; Et, H, Et, H, O, H, H, H, H, NH, O, OMe], [AI2366; Et , H, Et, H, O, H, H, H, F, NH, O, OMe], [AI 2367; Et, H, Et, H, O, H, H, H, Cl, NH, O, OMe ], [AI 2 368; Et, H, Et, H, O, H, H, H, Br, NH, O, OMe], [AI 2369; Et, H, Et, H, O, H, H, H, I , NH, O, OMe], [AI 2370; Et, H, Et, H, O, H, H, H, H, Me, NH, O, OMe], [AI 2371; Et, H, Et, H, O, H , H, H, Et, NH, O, OMe], [AI 2372; Et, H, Et, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2 373; Et, H Et, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2374; Et, H, Et, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 375; Et, H, Et, H, O, H, H, S Me, NH, O, OMe], [AI 2 376; Et, H, Et, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI 2377; CF ₃ , H, Et, H, O , H, H, H, H, NH, O, OMe], [AI2378; CF 3, H, Et, H, O, H, H, H, F, NH, O, OMe], [AI 2379; CF ₃ , H, Et, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 380; CF ₃ , H, Et, H, O, H, H, H, Br, NH, O, OMe], [AI2381; CF 3, H, Et, H, O, H, H, H, I, NH, O, OMe], [AI2382; CF 3, H, Et, H, O, H, H, H, Me, NH, O, OMe], [AI2383; CF 3, H, Et, H, O, H, H, H, Et, NH, O, OMe], [AI2384 CF ₃ , H, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2385; CF ₃ , H, Et, H, O, H, H, H, H, OMe , NH, O, OMe], [AI 2 386; CF ₃ , H, Et, H, O, H, H, H, H, Oe, NH, O, OMe], [AI 2387; CF ₃ , H, Et, H, O , H, H, H, SMe , NH, O, OMe], [AI2388; CF 3, H, Et, H, O, H, H, H, CF 3, NH, O, OMe], [AI2389; H _{, H, CF 3, H,} O, H, H, H, H, NH, O, OMe], [AI2390; H, H, CF 3, H, O, H, H, H, F, NH, O , OMe], [AI2391; H , H, CF 3, H, O, H, H, H, Cl, NH, O, OMe], [AI2392; H, H, CF 3, H, O, H, H , H, Br, NH, O , OMe], [AI2393; H, H, CF 3, H, O, H, H, H, I, NH, O, OMe], [AI2394; H, H, CF 3 , H, O, H, H , H, Me, NH, O, OMe], [AI2395; H, H, CF 3, H, O, H, H, H, Et, NH, O, OMe], [ _{AI2396; H, H, CF 3} , H, O, H, H, H, c-Pr, NH, O, OMe], [AI2397; H, H, CF 3, H, O, H, H, H, OMe, NH, O, OMe] , [AI2398; H, H, CF 3, H, O, H, H, H, OEt, NH, O, OMe], [AI2399; H, H, CF 3, H, O, H, H, H, SMe, NH, O, OMe], [AI2400; H, H, CF 3, H, O, H, H, H, CF 3, NH, O, OMe],

[AI2401; F, H, CF 3, H, O, H, H, H, H, NH, O, OMe], [AI2402; F, H, CF 3, H, O, H, H, H, F , NH, O, OMe], [AI2403; F, H, CF 3, H, O, H, H, H, Cl, NH, O, OMe], [AI2404; F, H, CF 3, H, O , H, H, H, Br, NH, O, OMe], [AI 2 405; F, H, CF ₃ , H, O, H, H, H, I, NH, O, OMe], [AI 2406; _{H, CF 3, H, O} , H, H, H, Me, NH, O, OMe], [AI2407; F, H, CF 3, H, O, H, H, H, Et, NH, O, OMe], [AI2408; F, H, CF 3, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2409; F, H, CF 3, H, O, H, H, H, OMe, NH, O, OMe], [AI2410; F, H, CF 3, H, O, H, H, H, OEt, NH, O, OMe], [AI2411; F, H, CF _{3, H, O, H,} H, H, SMe, NH, O, OMe], [AI2412; F, H, CF 3, H, O, H, H, H, CF 3, NH, O, OMe] , [AI2413; Cl, H, CF 3, H, O, H, H, H, H, NH, O, OMe], [AI2414; Cl, H, CF 3, H, O, H, H, H, F, NH, O, OMe] , [AI2415; Cl, H, CF 3, H, O, H, H, H, Cl, NH, O, OMe], [AI2416; Cl, H, CF 3, H, O, H, H, H, Br, NH, O, OMe], [AI2417; Cl, H, CF 3, H, O, H, H, H, I, NH, O, OMe], [AI2418; Cl _{, H, CF 3, H,} O, H, H, H, Me, NH, O, OMe], [AI2419; Cl, H, CF 3, H, O, H, H, H, Et, NH, O , OMe], [AI2420; Cl , H, CF 3, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2421; Cl, H, CF 3, H, O, H , H, H, OMe, NH , O, OMe], [AI2422; Cl, H, CF 3, H, O, H, H, H, OEt, NH, O, OMe], [AI2423; Cl, H, _{CF 3, H, O, H} , H, H, SMe, NH, O, OMe], [AI2424; Cl, H, CF 3, H, O, H, H, H, CF 3, NH, O , OMe], [AI2425; Br , H, CF 3, H, O, H, H, H, H, NH, O, OMe], [AI2426; Br, H, CF 3, H, O, H, H , H, F, NH, O , OMe], [AI2427; Br, H, CF 3, H, O, H, H, H, Cl, NH, O, OMe], [AI2428; Br, H, CF 3 , H, O, H, H , H, Br, NH, O, OMe], [AI2429; Br, H, CF 3, H, O, H, H, H, I, NH, O, OMe], [ _{AI2430; Br, H, CF 3} , H, O, H, H, H, Me, NH, O, OMe], [AI2431; Br, H, CF 3, H, O, H, H, H, Et, NH, O, OMe], [ AI2432; Br, H, CF 3, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2433; Br, H, CF 3, H, O, H, H, H, OMe, NH, O, OMe], [AI2434; Br, H, CF 3, H, O, H, H, H, OEt, NH, O, OMe], [AI2435; Br _{, H, CF 3, H,} O, H, H, H, SMe, NH, O, OMe], [AI2436; Br, H, CF 3, H, O, H, H, H, CF 3, NH, O, OMe], [AI2437; Me, H, CF 3, H, O, H, H, H, H, NH, O, OMe], [AI2438; Me, H, CF 3, H, O, H, H, H, F, NH, O, OMe], [AI2439; Me, H, CF 3, H, O, H, H, H, Cl, NH, O, OMe], [AI2440; Me, H, CF _{3, H, O, H,} H, H, Br, NH, O, OMe], [AI2441; Me, H, CF 3, H, O, H, H, H, I, NH, O, OMe], [AI2442; Me, H, CF 3, H, O, H, H, H, Me, NH, O, OMe], [AI2443; Me, H, CF 3, H, O, H, H, H, Et , NH, O, OMe], [AI2444; Me, H, CF 3, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2445; Me, H, CF 3, H , O, H, H, H , OMe, NH, O, OMe], [AI2446; Me, H, CF 3, H, O, H, H, H, OEt, NH, O, OMe], [AI2447; _{Me, H, CF 3, H} , O, H, H, H, SMe, NH, O, OMe], [AI2448; Me, H, CF 3, H, O, H, H, H, CF 3, NH, O, OMe], [AI2449; Et, H, CF 3, H, O, H, H, H, H, NH, O, OMe], [AI2450; _{Et, H, CF 3, H} , O, H, H, H, F, NH, O, OMe], [AI2451; Et, H, CF 3, H, O, H, H, H, Cl, NH, O, OMe], [AI2452; Et, H, CF 3, H, O, H, H, H, Br, NH, O, OMe], [AI2453; Et, H, CF 3, H, O, H, H, H, I, NH, O, OMe], [AI2454; Et, H, CF 3, H, O, H, H, H, Me, NH, O, OMe], [AI2455; Et, H, CF _{3, H, O, H,} H, H, Et, NH, O, OMe], [AI2456; Et, H, CF 3, H, O, H, H, H, c-Pr, NH, O, OMe ], [AI2457; Et, H , CF 3, H, O, H, H, H, OMe, NH, O, OMe], [AI2458; Et, H, CF 3, H, O, H, H, H , OEt, NH, O, OMe ], [AI2459; Et, H, CF 3, H, O, H, H, H, SMe, NH, O, OMe], [AI2460; Et, H, CF 3, H , O, H, H, H , CF 3, NH, O, OMe], [AI2461; CF 3, H, CF 3, H, O, H, H, H, H, NH, O, OMe], [ AI 2462; CF ₃ , H, CF ₃ , H, O, H, H, F, NH, O, OMe], [AI 2463; CF ₃ , H, CF ₃ , H, O, H, H, H, Cl, NH, O, OMe] , [AI2464; CF 3, H, CF 3, H, O, H, H, H, Br, NH, O, OMe], [AI2465; CF 3, H, CF 3, H, O, H, H, H, I, NH, O, OMe], [AI 2466; CF ₃ , H, CF ₃ , H, O, H, H, Me, NH, O, OMe], [ _{AI2467; CF 3, H, CF} 3, H, O, H, H, H, Et, NH, O, OMe], [AI2468; CF 3, H, CF 3, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2469; CF 3, H, CF 3, H, O, H, H, H, OMe, NH, O, OMe], [AI2470; CF 3, H, CF _{3, H, O, H,} H, H, OEt, NH, O, OMe], [AI2471; CF 3, H, _{CF 3, H, O, H} , H, H, SMe, NH, O, OMe], [AI2472; CF 3, H, CF 3, H, O, H, H, H, CF 3, NH, O, OMe], [AI2473; H, F, H, H, O, H, H, H, H, NH, O, OMe], [AI 2474; H, F, H, H, O, H, H, H, F, NH, O, OMe], [AI 2475; H, F, H, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2476; H, F, H, H, O, H, H, H, H, Br, NH, O, OMe], [AI2477; H, F, H, H, O, H, H, H, I, NH, O, OMe], [AI2478; H, F, H, H, O, H, H, H, Me, NH, O, OMe], [AI 2479; H, F, H, H, O, H, H, H, Et, NH, O, OMe], [ AI 2 480; H, F, H, H, O, H, H, c, Pr, NH, O, OMe], [AI2481; H, F, H, H, O, H, H, H, OMe, NH, O, OMe], [AI2482; H, F, H, H, O, H, H, H, OEt, NH, O, OMe], [AI2483; H, F, H, H, O, H, H, H, SMe, NH, O, OMe], [AI2484; H, F, H, H, O, H, H, H, CF 3, NH, O, OMe], [AI2485; Cl, F, H , H, O, H, H, H, H, H, NH, O, OMe], [AI 2486; Cl, F, H, H, O, H, H, F, NH, O, OMe], [AI 2487 Cl, F, H, H, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2488; Cl, F, H, H, O, H, H, H, Br, NH, O , OMe], [AI2489; Cl, F, H, H, O, H, H, H, I, NH, O, OMe], [AI 2490; Cl, F, H, H, O, H, H, H , Me, NH, O, OMe], [AI2491; Cl, F, H, H, O, H, H, H, H, Et, NH, O, OMe], [AI2492; Cl, F, H, H, O , H, H, H, c-Pr, NH, O, OMe], [AI2493; Cl, F, H, H, O, H, H, H, OMe, NH, O, OMe], [AI2494; , F, H, H, O, H, H, H, OEt, NH, O, OMe], [AI 2495; Cl, F, H, H, O, H, H, S, NH, O, OMe ], [AI2496; Cl, F , H, H, O, H, H, H, CF 3, NH, O, OMe], [AI2497; Me, F , H, H, O, H, H, H, H, NH, O, OMe], [AI 2498; Me, F, H, H, O, H, H, H, F, NH, O, OMe], [AI2499; Me, F, H, H, O, H, H, H, Cl, NH, O, OMe], [AI2500; Me, F, H, H, O, H, H, H, Br, NH , O, OMe],

[AI 2501; Me, F, H, H, O, H, H, I, NH, O, OMe], [AI 2502; Me, F, H, H, O, H, H, H, Me, NH , O, OMe], [AI 2503; Me, F, H, H, O, H, H, H, Et, NH, O, OMe], [AI 2504; Me, F, H, H, O, H, H , H, c-Pr, NH, O, OMe], [AI 2505; Me, F, H, H, O, H, H, H, OMe, NH, O, OMe], [AI 2506; Me, F, H , H, O, H, H, H, OEt, NH, O, OMe], [AI 2507; Me, F, H, H, O, H, H, S Me, NH, O, OMe], [AI 2508 ; Me, F, H, H , O, H, H, H, CF 3, NH, O, OMe], [AI2509; Et, F, H, H, O, H, H, H, H, NH, O, OMe], [AI 2510; Et, F, H, H, O, H, H, H, H, F, NH, O, OMe], [AI 2511; Et, F, H, H, O, H, H, H, Cl, NH, O, OMe], [AI 2512; Et, F, H, H, O, H, H, H, H, H, Br, NH, O, OMe], [AI 2513; Et, F, H, H, O, H, H, H, I, NH, O, OMe], [AI 2514; Et, F, H, H, H, O, H, H, H, Me, NH, O, OMe], [AI 2515; Et, F, H, H, H, O, H, H, H, H, Et, NH, O, OMe], [AI 2516; Et, F, H, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2517; Et, F, H, H, O, H, H, H, OMe, NH, O, OMe], [AI 2518; Et, F, H, H, O, H, H, H, H, OEt, NH, O, OMe], [AI2519; Et, F, H, H, H, O, H, H, H, SMe, NH, O, OMe], [AI 2520; Et, F, H, H, O, _{H, H, H, CF 3} , NH, O, OMe], [AI2521; H, F, F, H, O, H, H, H, H, NH, O, OMe], [AI2522; H, F , F, H, O, H, H, H, F, NH, O, OMe], [AI 2523; H, F, F, H, O, H, H, H, Cl, NH, O, OMe], [AI2524; H, F, F, H, O, H, H, H, Br, NH, O, OMe], [AI 2525; H, F, F, H, O, H, H, H, I, NH , O, OMe], [AI 2526; H, F, F, H, O, H, H, H, Me, NH, O, OMe], [AI 2527; H , F, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2528; H, F, F, H, O, H, H, H, c-Pr, NH, O , OMe], [AI 2529; H, F, F, H, O, H, H, H, OMe, NH, O, OMe], [AI 2530; H, F, F, H, O, H, H, H , OEt, NH, O, OMe], [AI2531; H, F, F, H, O, H, H, H, SMe, NH, O, OMe], [AI 2532; H, F, F, H, O , H, H, H, CF 3, NH, O, OMe], [AI2533; Cl, F, F, H, O, H, H, H, H, NH, O, OMe], [AI2534; Cl, F, F, H, O, H, H, H, F, NH, O, OMe], [AI 2535; Cl, F, F, H, O, H, H, H, Cl, NH, O, OMe] , [AI 2536; Cl, F, F, H, O, H, H, H, Br, NH, O, OMe], [AI 2537; Cl, F, F, H, O, H, H, H, I, NH, O, OMe], [AI 2538; Cl, F, F, H, O, H, H, H, Me, NH, O, OMe], [AI 2539; Cl, F, F, H, O, H, H, H, Et, NH, O, OMe], [AI2540; Cl, F, F, H, O, H, H, H, c, Pr, NH, O, OMe], [AI2541; Cl, F, F, H, O, H, H, H, OMe, NH, O, OMe], [AI 2542; Cl, F, F, H, O, H, H, H, OEt, NH, O, OMe], [ AI 2543; Cl, F, F, H, O, H, H, SMe, NH, O, OMe], [AI 2544; Cl, F, F, H, O, H, H, H, CF ₃ , NH , O, OMe], [AI 2545; Me, F, F, H, O, H, H, H, H, H, NH, O, OMe], [AI 2546; Me, F, F, H, O, H, H , H, F, NH, O, OMe], [AI 2547; Me, F, F, H, O, H, H, H, Cl, NH, O, OMe], [AI 2548; Me, F, F, H , O, H, H, H, H, Br, NH, O, OMe], [AI 2549; Me, F, F, H, O, H, H, H, I, NH, O, OMe], [AI 2550; , F, F, H, O, H, H, H, Me, NH, O, OMe], [AI2551; Me, F, F, H, O, H, H, H, Et, NH, O, OMe ], [AI2552; Me, F, F, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2553; Me, F, F, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2554; Me, F, F, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 555; Me, F, F, H, O, H, H, H, SMe, NH, O, OMe], [AI 2556; Me, F, F, H, O, H, H, H, CF ₃ , NH, O , OMe], [AI 2557; Et, F, F, H, O, H, H, H, H, NH, O, OMe], [AI 2 558; Et, F, F, H, O, H, H, H , F, NH, O, OMe], [AI 2559; Et, F, F, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2560; Et, F, F, H, O , H, H, H, Br, NH, O, OMe], [AI2561; Et, F, F, H, O, H, H, H, I, NH, O, OMe], [AI 2562, Et, F , F, H, O, H, H, H, Me, NH, O, OMe], [AI2563; Et, F, F, H, O, H, H, H, Et, NH, O, OMe], [AI 2564; Et, F, F, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2565; Et, F, F, H, O, H, H, H, H, OMe , NH, O, OMe], [AI 2566; Et, F, F, H, O, H, H, H, H, OEt, NH, O, OMe], [AI 2 567; Et, F, F, H, O, H , H, H, SMe, NH , O, OMe], [AI2568; Et, F, F, H, O, H, H, H, CF 3, NH, O, OMe], [AI2569; H, F, Cl, H, O, H, H, H, H, H, NH, O, OMe], [AI 2570; H, F, Cl, H, O, H, H, F, NH, O, OMe], [ AI 2571; H, F, Cl, H, O, H, H, H, Cl, NH, O, OMe], [AI2572; H, F, Cl, H, O, H, H, H, Br, NH, O, OMe], [AI 2573; H, F, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2574; H, F, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI2575; H, F, Cl, H, O, H, H, H, H, Et, NH, O, OMe], [AI2576; H, F, Cl, H, O, H, H, H, c, Pr-NH, O, OMe], [AI 2577; H, F, Cl, H, O, H, H, H, OMe, NH, O, OMe], [AI 2578; H, F, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2579; H, F, Cl, H, O, H, H, H, SMe, NH, O, OMe], [AI2580; H, F, Cl, H, O, H, H, H, CF 3, NH, O, OMe], [AI2581 Cl, F, Cl, H, O, H, H, H, H, H, NH, O, OMe], [AI 2582; Cl, F, Cl, H, O, H, H, H, F, NH, O , OMe], [AI 2583; Cl, F, Cl, H, O, H, H, H, Cl, NH, O, OMe], [AI 2584; Cl, F, Cl, H, O, H, H, H , Br, NH, O, OMe], [AI 2585; Cl, F, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2586; Cl, F, Cl, H, O , H, H, H, Me, NH, O, OMe], [AI 2587; Cl, F, Cl, H, O, H, H, H, Et, NH, O, OMe], [AI 2588; Cl, F , Cl, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2589; Cl, F, Cl, H, O, H, H, H, OMe, NH, O, OMe ], [AI 2590; Cl, F, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2591; Cl, F, Cl, H, O, H, H, H, SMe , NH, O, OMe], [AI2592; Cl, F, Cl, H, O, H, H, H, CF 3, NH, O, OMe], [AI2593; Me, F, Cl, H, O, H, H, H, H, H, NH, O, OMe], [AI2594; Me, F, Cl, H, O, H, H, H, F, NH, O, OMe], [AI2595; Me, F, Cl, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2596; Me, F, Cl, H, O, H, H, H, Br, NH, O, OMe], [ AI 2597; Me, F, Cl, H, O, H, H, I, NH, O, OMe], [AI 2598; Me, F, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI 2599; Me, F, Cl, H, O, H, H, H, Et, NH, O, OMe], [AI 2600; Me, F, Cl, H, O, H, H, H, c-Pr, NH, O, OMe],

[AI 2601; Me, F, Cl, H, O, H, H, OMe, NH, O, OMe], [AI 2602; Me, F, Cl, H, O, H, H, H, OE t, NH , O, OMe], [AI 2603; Me, F, Cl, H, O, H, H, H, S Me, NH, O, OMe], [AI 2604; Me, F, Cl, H, O, H, H _{, H, CF 3, NH,} O, OMe], [AI2605; Et, F, Cl, H, O, H, H, H, H, NH, O, OMe], [AI2606; Et, F, Cl, H, O, H, H, H, H, F, NH, O, OMe], [AI 2607; Et, F, Cl, H, O, H, H, H, Cl, NH, O, OMe], [AI 2608; Et, F, Cl, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2609; Et, F, Cl, H, O, H, H, H, I, NH, O, OMe], [AI 2610; Et, F, Cl, H, O, H, H, H, Me, NH, O, OMe], [AI 2611; Et, F, Cl, H, O, H, H, H, H, Et, NH, O, OMe], [AI2612; Et, F, Cl, H, O, H, H, H, H, c-Pr, NH, O, OMe], [AI 2613; Et, F, Cl, H, O, H, H, H, H, OMe, NH, O, OMe], [AI 2614; Et, F, Cl, H, O, H, H, H, OEt, NH, O, OMe], [AI 2615; Et, F, Cl, H, O, H, H, H, SMe, NH, O, OMe], [AI2616; Et, F, Cl, H, O, H, H, H, CF 3, NH, O, OMe H, F, Me, H, O, H, H, H, H, NH, O, OMe], [AI 2618; H, F, Me, H, O, H, H, H, F] , NH, O, OMe], [AI 2619; H, F, Me, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2620; H, F, Me, H, O, H , H, H, Br, NH, O, OMe], [AI2621; H, F, Me, H, O, H, H, H, I, NH, O, OMe], [AI 2622; H, F, Me , H, O, H, H, H, H, Me, NH, O, OMe], [AI 2623; H, F, Me, H, O, H, H, H, Et, NH, O, OMe], [AI 2624 H, F, Me, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2625; H, F, Me, H, O, H, H, H, OMe, NH , O, OMe], [AI2626; H, F, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI2627; H, F, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI2628; H, F, Me, H, O, H, H, H, CF 3, NH, O, OMe], [AI2629; Cl, F, Me, H, O, H, H, H, H, NH, O, OMe], [AI2630; Cl , F, Me, H, O, H, H, H, F, NH, O, OMe], [AI2631; Cl, F, Me, H, O, H, H, H, Cl, NH, O, OMe ], [AI2632; Cl, F, Me, H, O, H, H, H, Br, NH, O, OMe], [AI 2633; Cl, F, Me, H, O, H, H, H, I , NH, O, OMe], [AI 2634; Cl, F, Me, H, O, H, H, H, H, Me, NH, O, OMe], [AI 2635; Cl, F, Me, H, O, H , H, H, Et, NH, O, OMe], [AI2636; Cl, F, Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2637; Cl, F , Me, H, O, H, H, H, OMe, NH, O, OMe], [AI 2638; Cl, F, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI2639; Cl, F, Me, H, O, H, H, SMe, NH, O, OMe], [AI 2640; Cl, F, Me, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI2641; Me, F, Me, H, O, H, H, H, H, H, NH, O, OMe], [AI2642; Me, F, Me, H, O, H, H, H, F, NH, O, OMe], [AI 2643; Me, F, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 644; Me, F, Me, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2645; Me, F, Me, H, O, H, H, H, I, NH, O, OMe], [AI 2 646; Me, F, Me, H, O, H, H, H, Me, NH, O, OMe], [AI 2647; Me, F, Me, H, O, H, H, H, Et, NH, O, OMe], [AI 2648; Me, F, Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2649; Me, F, Me, H, O, H, H, H, OMe, NH, O, OMe], [AI2650; Me, F, Me, H, O, H, H, H, H, OEt, NH, O, OMe], [AI2651; Me, F, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI2652; Me, F, Me , H, O, H, H, H, CF 3, NH, O, OMe], [AI2653; Et, F, Me, H, O, H, H, H, H, NH, O, OMe], [AI2654; Et, F, Me, H, O, H, H, H, H, F, NH, O, OMe], [AI 2655; Et, F, Me, H, O, H, H, H, Cl, NH, O, OMe], [AI 2 656; Et, F, Me, H, O, H, H, H, Br, NH, O, OMe], [AI 2657; Et, F, Me, H, O, H, H, H, H, I, NH, O, OMe], [AI 2658; Et, F, Me, H, O, H, H, Me, NH, O, OMe], [AI 2659; Et, F, Me, H, O, H, H, H, H, Et, NH, O, OMe], [AI 2660; Et, F, Me, H, O, H, H, H, c-Pr, NH, O, OMe], [AI2661; Et, F, Me, H, O, H, H, H, OMe, NH, O, OMe], [AI2662; Et, F, Me, H, O, H, H, H, OEt, NH, O, OMe], [AI2663; Et, F, Me, H, O, H, H, H, SMe, NH, O, OMe], [AI2664; Et, F, Me, H, O, H, H, H, CF 3, NH, O, OMe], [AI2665; H, F, Et, H, O, H, H, H, H, NH, O, OMe], [AI2666; H , F, Et, H, O, H, H, H, F, NH, O, OMe], [AI 2667; H, F, Et, H, O, H, H, H, Cl, NH, O, OMe H, F, Et, H, O, H, H, H, Br, NH, O, OMe], [AI 2669; H, F, Et, H, O, H, H, H, I] , NH, O, OMe], [AI 2 670; H, F, Et, H, O, H, H, H, Me, NH, O, OMe], [AI 2671; H, F, Et, H, O, H , H, H, Et, NH, O, OMe], [AI 2672; H, F, Et, H, O, H, H, H, c-Pr, NH, O, OMe], [AI 2673; H, F , Et, H, O, H, H, H, OMe, NH, O, OMe], [AI 2674; H, F, Et, H, O, H, H, H, OEt, NH, O, OMe], [AI 2 675; H, F, Et, H, O, H, H, S Me, NH, O, OMe], [AI 2 676; H, F, Et, H, O, H, H, H, CF ₃ , NH, O, OMe], [AI 2677; Cl, F, Et, H, O, H, H, H, H, NH, O, OMe], [AI2678; Cl, F, Et, H, O, H, H, H, H, F, NH, O, OMe], [AI2679; Cl, F, Et, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2 680; Cl, F, Et, H, O, H, H, H, Br, NH, O, OMe], [AI2681; F, Et, H, O, H, H, H, I, NH, O, OMe], [AI2682; Cl, F, Et, H, O, H, H, H, Me, NH, O, OMe] , [AI2683; Cl, F, Et, H, O, H, H, H, Et, NH, O, OMe], [AI 2684; Cl, F, Et, H, O, H, H, H, c- Pr, NH, O, OMe], [AI2685; Cl, F, Et, H, O, H, H, H, H, OMe, NH, O, OMe], [AI2686; Cl, F, Et, H, O, H, H, H, H, OEt, NH, O, OMe], [AI2687; Cl, F, Et, H, O, H, H, H, SMe, NH, O, OMe], [AI2688; Cl, F, Et, H, O, H, H, H, CF 3, NH, O, OMe], [AI2689; Me, F, Et, H, O, H, H, H, H, NH, O, OMe], [AI2690; Me, F, Et, H, O, H, H, H, F, NH, O, OMe], [AI 2691; Me, F, Et, H, O, H, H, H, Cl, NH , O, OMe], [AI2692; Me, F, Et, H, O, H, H, H, H, Br, NH, O, OMe], [AI 2693; Me, F, Et, H, O, H, H , H, I, NH, O, OMe], [AI 2694; Me, F, Et, H, O, H, H, H, Me, NH, O, OMe], [AI 2 695; Me, F, Et, H , O, H, H, H, H, Et, NH, O, OMe], [AI 2 696; Me, F, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2697 Me, F, Et, H, O, H, H, H, OMe, NH, O, OMe], [AI 2698; Me, F, Et, H, O, H, H, H, OEt, NH, O , OMe], [AI 2699; Me, F, Et, H, O, H, H, H, SMe, NH, O, OMe], [AI 2700; Me, F, Et, H, O, H, H, H , CF ₃ , NH, O, OMe],

[AI 2701; Et, F, Et, H, O, H, H, H, H, NH, O, OMe], [AI 2702; Et, F, Et, H, O, H, H, H, F, NH , O, OMe], [AI 2703; Et, F, Et, H, O, H, H, H, H, Cl, NH, O, OMe], [AI 2704; Et, F, Et, H, O, H, H , H, Br, NH, O, OMe], [AI 2705; Et, F, Et, H, O, H, H, H, I, NH, O, OMe], [AI 2706; Et, F, Et, H , O, H, H, H, Me, NH, O, OMe], [AI 2 707; Et, F, Et, H, O, H, H, H, Et, NH, O, OMe], [AI 2 708; , F, Et, H, O, H, H, H, c, Pr, NH, O, OMe], [AI 2709; Et, F, Et, H, O, H, H, H, OMe, NH, O , OMe], [AI 2710; Et, F, Et, H, O, H, H, H, OEt, NH, O, OMe], [AI 2711; Et, F, Et, H, O, H, H, H , SMe, NH, O, OMe ], [AI2712; Et, F, Et, H, O, H, H, H, CF 3, NH, O, OMe], [AI2713; H, H, H, F, O, H, H, H, H, H, NH, O, OMe], [AI 2714; H, H, H, H, F, O, H, H, H, F, NH, O, OMe], [AI 2715; H, H, H, F, O, H, H, H, H, Cl, NH, O, OMe], [AI 2716; H, H, H, F, O, H, H, H, Br, NH, O, OMe] [AI 2717; H, H, H, F, O, H, H, I, NH, O, OMe], [AI 2718; H, H, H, F, O, H, H, H, Me, NH, O, OMe], [AI 2719; H, H, H, F, O, H, H, H, Et, NH, O, OMe], [AI 2720; H, H, H, F, O, H, H, H, c-Pr, NH, O, OMe], [AI 2272; H, H, H, H, F, O, H, H, H, OMe, NH, O, OMe], [AI 2722; H, H, H, F, O, H, H, H, OEt, NH, O, OMe], [AI 2723; H, H, H, F, O, H, H, S Me, NH, O, OMe], [ AI2724; H, H, H, F, O, H, H, H, CF 3, NH, O, OMe], [AI2725; Cl, H, H, F, O, H, H, H, H, NH , O, OMe], [AI 2726; Cl, H, H, F, O, H, H, H, F, NH, O, OMe], [AI 2 727; Cl, H, H, F, O, H, H, H, Cl, NH, O, OMe], [AI 2 728; Cl, H, H, F, O, H, H, H, Br, NH, O, OMe], [AI 2729; Cl, H, H, F, O, H, H, I, NH, O, OMe], [AI 2730; Cl, H, H, F, O, H, H, H, Me, NH, O, OMe], [AI 2731; Cl, H, H, F, O, H, H, H, H, Et, NH, O, OMe], [AI 2732; Cl, H, H, F, O, H, H, H, c, Pr, NH, O, OMe], [AI 2733; Cl, H, H, H, F, O, H, H, H, OMe, NH, O, OMe], [AI 2734; Cl, H, H, F, O, H, H, H, OEt, NH, O, OMe], [AI 2735; Cl, H, H, F, O, H, H, S, NH, O, OMe], [AI2736; Cl, H, H, F, O, H, H, H, CF 3, NH, O, OMe], [AI2737; Me, H, H, F, O, H, H, H , H, NH, O, OMe], [AI 2738; Me, H, H, F, O, H, H, H, F, NH, O, OMe], [AI 2739; Me, H, H, F, O , H, H, H, Cl, NH, O, OMe], [AI 2740; Me, H, H, F, O, H, H, H, Br, NH, O, OMe], [AI 2741; Me, H , H, F, O, H, H, H, I, NH, O, OMe], [AI2742; Me, H, H, F, O, H, H, Me, NH, O, OMe], [AI2743; Me, H, H, F, O, H, H, Et, NH, O, OMe], [AI 2 744; Me, H, H, F, O, H, H, H, c-Pr , NH, O, OMe], [AI 2 745; Me, H, H, F, O, H, H, H, OMe, NH, O, OMe], [AI 2 746; Me, H, H, F, O, H , H, H, OEt, NH, O, OMe], [AI 2 747; Me, H, H, F, O, H, H, S, NH, O, OMe], [AI 2 748; Me, H, H , F, O, H, H , H, CF 3, NH, O, OMe], [AI2749; Et, H, H, F, O, H, H, H, H, NH, O, OMe], [ AI 2 750; Et, H, H, F, O, H, H, H, F, NH, O, OMe], [AI 2751; Et, H, H, F, O, H, H, H, Cl, NH, O, OMe], [AI 2752; Et, H, H, F, O, H, H, H, Br, NH, O, OMe], [AI 275 3; Et, H, H, F, O, H, H, H, I, NH, O, OMe], [AI 2754; Et, H, H, F, O, H, H, H, Me, NH, O, OMe], [AI 2755; Et, H, H, F, O, H, H, H, Et, NH, O, OMe], [AI 2756; Et, H, H, F, O, H, H, H, c-Pr, NH, O, OMe], [AI 2757; Et, H, H, F, O, H, H, H, H, OMe, NH, O, OMe], [AI 2758; Et, H, H, F, O, H, H, H, H, OEt, NH, O, OMe], [AI 2759; Et, H, H, F, O, H, H, S Me, NH, O, OMe], [AI 2760; Et, H, H, F, O, H, H, H, CF 3, NH, O, OMe], [AI2761; H, H, F, F, O, H, H, H, H, NH, O , OMe], [AI2762; H, H, F, F, O, H, H, H, F, NH, O, OMe], [AI2763; H, H, F, F, O, H, H, H , Cl, NH, O, OMe], [AI 2764; H, H, F, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2 765; H, H, F, F, O , H, H, H, H, I, NH, O, OMe], [AI 2766; H, H, F, F, O, H, H, H, Me, NH, O, OMe], [AI 2 767; H, H , F, F, O, H, H, H, H, Et, NH, O, OMe], [AI 2768; H, H, F, F, O, H, H, c, Pr, NH, O, OMe H, H, F, F, O, H, H, OMe, NH, O, OMe], [AI 2 770; H, H, F, F, O, H, H, H, OEt] , NH, O, OMe], [AI2771; H, H, F, F, O, H, H, S, NH, O, OMe], [AI 2772; H, H, F, F, O, H _{, H, H, CF 3,} NH, O, OMe], [AI2773; Cl, H, F, F, O, H, H, H, H, NH, O, OMe], [AI2774; Cl, H, F, F, O, H, H, H, F, NH, O, OMe], [AI 2775; Cl, H, F, F, O, H, H, Cl, NH, O, OMe], [A AI 2776; Cl, H, F, F, O, H, H, H, Br, NH, O, OMe], [AI 2777; Cl, H, F, F, O, H, H, H, I, NH, O, OMe], [AI 2778; Cl, H, F, F, O, H, H, Me, NH, O, OMe], [AI 2779; Cl, H, F, F, O, H, H, H, Et, NH, O, OMe], [AI 2 780; Cl, H, F, F, O, H, H, c, Pr, NH, O, OMe], [AI 2781; Cl, H, F, F, O, H, H, H, H, OMe, NH, O, OMe], [AI 2782; Cl, H, F, F, O, H, H, H, OEt, NH, O, OMe], [ AI 2783; Cl, H, F, F, O, H, H, SMe, NH, O, OMe], [AI 2784; Cl, H, F, F, O, H, H, H, CF ₃ , NH , O, OMe], [AI 2 785; Me, H, F, F, O, H, H, H, H, NH, O, OMe], [AI 2 786; Me, H, F, F, O, H, H , H, F, NH, O, OMe], [AI 2787; Me, H, F, F, O, H, H, H, Cl, NH, O, OMe], [AI 2 788; Me, H, F, F , O, H, H, H, H, Br, NH, O, OMe], [AI 2 789; Me, H, F, F, O, H, H, H, I, NH, O, OMe], [AI 2 790; , H, F, F, O, H, H, H, Me, NH, O, OMe], [AI 2791; Me, H, F, F, O, H, H, Et, NH, O, OMe Me, H, F, F, O, H, H, H, c-Pr, NH, O, OMe], [AI 2793; Me, H, F, F, O, H, H, H] , OMe, NH, O, OMe], [AI 2794; Me, H, F, F, O, H, H, H, H, OEt, NH, O, OMe], [AI 2795; Me, H, F, F, O , H, H, H, SMe , NH, O, OMe], [AI2796; Me, H, F, F, O, H, H, H, CF 3, NH, O, OMe], [AI2797; Et, H, F, F, O, H, H, H, H, H, NH, O, OMe], [AI 2798; Et, H, F, F, O, H, H, F, NH, O, OMe] , [AI2799; Et, H, F, F, O, H, H, H, Cl, NH, O, OMe], [AI 2800; Et, H, F, F, O, H, H, H, Br, NH, O, OMe],

[AI2801; Et, H, F, F, O, H, H, I, NH, O, OMe], [AI 2802; Et, H, F, F, O, H, H, H, Me, NH , O, OMe], [AI 2803; Et, H, F, F, O, H, H, H, Et, NH, O, OMe], [AI 2804; Et, H, F, F, O, H, H , H, c-Pr, NH, O, OMe], [AI 2 805; Et, H, F, F, O, H, H, H, OMe, NH, O, OMe], [AI 2 806; Et, H, F , F, O, H, H, H, OEt, NH, O, OMe], [AI 2 807; Et, H, F, F, O, H, H, S Me, NH, O, OMe], [AI 2 808] ; Et, H, F, F , O, H, H, H, CF 3, NH, O, OMe], [AI2809; H, H, Cl, F, O, H, H, H, H, NH, O, OMe], [AI 2810; H, H, Cl, F, O, H, H, H, F, NH, O, OMe], [AI 2811; H, H, Cl, F, O, H, H, H, Cl, NH, O, OMe], [AI 2812; H, H, Cl, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2813; H, H, Cl, F, O, H, H, H, H, I, NH, O, OMe], [AI 2814; H, H, Cl, F, O, H, H, Me, NH, O, OMe], [AI 2815; H, H, Cl, F, O, H, H, H, H, Et, NH, O, OMe], [AI 2816; H, H, Cl, F, O, H, H, c, Pr, NH, O, OMe], [AI 2817; H, H, Cl, F, O, H, H, OMe, NH, O, OMe], [AI 2818; H, H, Cl, F, O, H, H, H, H, OEt, NH, O, OMe], [AI2819; H, H, Cl, F, O, H, H, H, SMe, NH, O, OMe], [AI2820; H, H, Cl, F, O, _{H, H, H, CF 3} , NH, O, OMe], [AI2821; Cl, H, Cl, F, O, H, H, H, H, NH, O, OMe], [AI2822; Cl, H , Cl, F, O, H, H, H, F, NH, O, OMe], [AI 2823; Cl, H, Cl, F, O, H, H, H, Cl, NH, O, OMe], [AI 2824; Cl, H, Cl, F, O, H, H, H, Br, NH, O, OMe], [AI 2825; Cl, H, Cl, F, O, H, H, H, I, NH , O, OMe], [AI 2826; Cl, H, Cl, F, O, H, H, H, Me, NH, O, OM e, [AI 2827; Cl, H, Cl, F, O, H, H, H, Et, NH, O, OMe], [AI 2828; Cl, H, Cl, F, O, H, H, H, c-Pr, NH, O, OMe], [AI 2829; Cl, H, Cl, F, O, H, H, H, H, OMe, NH, O, OMe], [AI 2830; Cl, H, Cl, F, O, H, H, H, H, OEt, NH, O, OMe], [AI 2831; Cl, H, Cl, F, O, H, H, S, NH, O, OMe], [AI 2832; Cl, H, Cl, F, O, H, H, H, CF 3, NH, O, OMe], [AI2833; Me, H, Cl, F, O, H, H, H, H, NH, O, OMe Me, H, Cl, F, O, H, H, H, F, NH, O, OMe], [AI 2 835; Me, H, Cl, F, O, H, H, H, Cl, , NH, O, OMe], [AI 2836; Me, H, Cl, F, O, H, H, H, Br, NH, O, OMe], [AI 2837; Me, H, Cl, F, O, H , H, H, I, NH, O, OMe], [AI 2 838; Me, H, Cl, F, O, H, H, H, Me, NH, O, OMe], [AI 2839; Me, H, Cl , F, O, H, H, H, H, Et, NH, O, OMe], [AI 2840; Me, H, Cl, F, O, H, H, c, Pr, NH, O, OMe], [AI2841; Me, H, Cl, F, O, H, H, OMe, NH, O, OMe], [AI 2842; Me, H, Cl, F, O, H, H, H, OEt, NH , O, OMe], [AI 2843; Me, H, Cl, F, O, H, H, S Me, NH, O, OMe], [AI 2844; Me, H, Cl, F, O, H, H _{, H, CF 3, NH,} O, OMe], [AI2845; Et, H, Cl, F, O, H, H, H, H, NH, O, OMe], [AI2846; Et, H, Cl, F, O, H, H, H, H, F, NH, O, OMe], [AI 2 847; Et, H, Cl, F, O, H, H, H, Cl, NH, O, OMe], [AI 2848; Et, H, Cl, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2849; Et, H, Cl, F, O, H, H, H, I, NH, O, OMe], [AI2850; Et, H, Cl, F, O, H, H, Me, NH, O, OMe], [AI 2851; Et, H, Cl, F, O, H, H, H, Et, NH, O, OMe], [AI 2852; Et, H , Cl, F, O, H, H, H, c, Pr, NH, O, OMe], [AI 2853; Et, H, Cl, F, O, H, H, H, OMe, NH, O, OMe ], [AI2854; Et, H, Cl, F, O, H, H, H, OEt, NH, O, OMe], [AI 2 855; Et, H, Cl, F, O, H, H, H, SMe , NH, O, OMe], [AI2856; Et, H, Cl, F, O, H, H, H, CF 3, NH, O, OMe], [AI2857; H, H, Me, F, O, H, H, H, H, H, NH, O, OMe], [AI 2858; H, H, Me, F, O, H, H, H, F, NH, O, OMe], [AI 2859; H, H, Me, F, O, H, H, H, H, Cl, NH, O, OMe], [AI 2860; H, H, Me, F, O, H, H, Br, NH, O, OMe], [ AI 2861; H, H, Me, F, O, H, H, I, NH, O, OMe], [AI 2862; H, H, Me, F, O, H, H, Me, NH, H, H, Me, F, O, H, H, Et, NH, O, OMe], [AI 2864; H, H, Me, F, O, H, H, O, OMe], [AI 2863; H, c-Pr, NH, O, OMe], [AI 2865; H, H, Me, F, O, H, H, H, OMe, NH, O, OMe], [AI 2866; H, H, Me, F, O, H, H, H, H, OEt, NH, O, OMe], [AI 2867; H, H, Me, F, O, H, H, S Me, NH, O, OMe], [AI 2868; H, H, Me, F, O, H, H, H, CF 3, NH, O, OMe], [AI2869; Cl, H, Me, F, O, H, H, H, H, NH, O , OMe], [AI 2870; Cl, H, Me, F, O, H, H, H, F, NH, O, OMe], [AI 2 871; Cl, H, Me, F, O, H, H, H , Cl, NH, O, OMe], [AI2872; Cl, H, Me, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2873; Cl, H, Me, F, O , H, H, H, I, NH, O, OMe], [AI 2 874; Cl, H, Me, F, O, H, H, H, Me, NH, O, OMe], [AI 2 875; Cl, H , Me, F, O, H, H, H, H, Et, NH, O, OMe], [AI 2876; Cl, H, Me, F, O, H, H, c, Pr, NH, O, OMe ], [AI 2877; Cl, H, Me, F, O, H, H, H, OMe, NH, O, OM e], [AI2878; Cl, H, Me, F, O, H, H, H, OEt, NH, O, OMe], [AI 2879; Cl, H, Me, F, O, H, H, H, SMe, NH, O, OMe] , [AI2880; Cl, H, Me, F, O, H, H, H, CF 3, NH, O, OMe], [AI2881; Me, H, Me, F, O , H, H, H, H, H, NH, O, OMe], [AI2882; Me, H, Me, F, O, H, H, H, F, NH, O, OMe], [AI2883; Me, H , Me, F, O, H, H, H, H, Cl, NH, O, OMe], [AI 2884; Me, H, Me, F, O, H, H, H, Br, NH, O, OMe], [AI 2885; Me, H, Me, F, O, H, H, I, NH, O, OMe], [AI 2886; Me, H, Me, F, O, H, H, H, Me, NH , O, OMe], [AI 2887; Me, H, Me, F, O, H, H, Et, NH, O, OMe], [AI 2 888; Me, H, Me, F, O, H, H , H, c-Pr, NH, O, OMe], [AI 2889; Me, H, Me, F, O, H, H, H, OMe, NH, O, OMe], [AI 2 890: Me, H, Me , F, O, H, H, H, H, OEt, NH, O, OMe], [AI2891; Me, H, Me, F, O, H, H, SMe, NH, O, OMe], [AI2892 ; Me, H, Me, F , O, H, H, H, CF 3, NH, O, OMe], [AI2893; Et, H, Me, F, O, H, H, H, H, NH, O, OMe], [AI2894; Et, H, Me, F, O, H, H, H, F, NH, O, OMe], [AI 2895; Et, H, Me, F, O, H, H, H, Cl, NH, O, OMe], [AI2896; Et, H, Me, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2897; Et, H, Me, F, O, H, H, H, I, NH, O, OMe], [AI 2898; Et, H, Me, F, O, H, H, Me, NH, O, OMe], [AI 2899; Et, H, Me, F, O, H, H, H, H, Et, NH, O, OMe], [AI 2900; Et, H, Me, F, O, H, H, H, c-Pr, NH, O, OMe],

[AI 2901; Et, H, Me, F, O, H, H, OMe, NH, O, OMe], [AI 2902; Et, H, Me, F, O, H, H, H, OE t, NH , O, OMe], [AI 2 903; Et, H, Me, F, O, H, H, S Me, NH, O, OMe], [AI 2904; Et, H, Me, F, O, H, H _{, H, CF 3, NH,} O, OMe], [AI2905; H, H, Et, F, O, H, H, H, H, NH, O, OMe], [AI2906; H, H, Et, F, O, H, H, H, H, F, NH, O, OMe], [AI 2907; H, H, Et, F, O, H, H, H, Cl, NH, O, OMe], [AI 2 908; H, H, Et, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2 909; H, H, Et, F, O, H, H, H, I, NH, O, OMe], [AI 2910; H, H, Et, F, O, H, H, Me, NH, O, OMe], [AI 2911; H, H, Et, F, O, H, H, H, Et, NH, O, OMe], [AI 2912; H, H, Et, F, O, H, H, H, c, Pr, NH, O, OMe], [AI 2913; H, H, Et, F, O, H, H, H, H, OMe, NH, O, OMe], [AI 2914; H, H, Et, F, O, H, H, H, OEt, NH, O, OMe], [AI 2915; H, H, Et, F, O, H, H, H, SMe, NH, O, OMe], [AI2916; H, H, Et, F, O, H, H, H, CF 3, NH, O, OMe ], [AI2917; Cl, H, Et, F, O, H, H, H, H, NH, O, OMe], [AI 2918; Cl, H, Et, F, O, H, H, H, F] , NH, O, OMe], [AI 2919; Cl, H, Et, F, O, H, H, H, Cl, NH, O, OMe], [AI 2920; Cl, H, Et, F, O, H , H, H, Br, NH, O, OMe], [AI 2921; Cl, H, Et, F, O, H, H, I, NH, O, OMe], [AI 2 922; Cl, H, Et , F, O, H, H, H, H, Me, NH, O, OMe], [AI 2923; Cl, H, Et, F, O, H, H, H, Et, NH, O, OMe], [AI 2 924] Cl, H, Et, F, O, H, H, H, c, Pr, NH, O, OMe], [AI 2925; Cl, H, Et, F, O, H, H, H, OMe, NH , O, OMe], [AI2926; Cl, H, Et, F, O, H, H, H, OEt, NH, O, OMe], [AI 2 927; Cl, H, Et, F, O, H, H, H, SMe, NH, O, OMe], [AI 2 928; Cl, H, Et, F, O, _{H, H, H, CF 3} , NH, O, OMe], [AI2929; Me, H, Et, F, O, H, H, H, H, NH, O, OMe], [AI2930; Me, H , Et, F, O, H, H, H, H, F, NH, O, OMe], [AI2931; Me, H, Et, F, O, H, H, H, Cl, NH, O, OMe], [AI2932; Me, H, Et, F, O, H, H, H, Br, NH, O, OMe], [AI 2933; Me, H, Et, F, O, H, H, H, I, NH , O, OMe], [AI 2 934; Me, H, Et, F, O, H, H, H, Me, NH, O, OMe], [AI 2935; Me, H, Et, F, O, H, H , H, Et, NH, O, OMe], [AI 2 936; Me, H, Et, F, O, H, H, H, c, Pr, NH, O, OMe], [AI 2 937; Me, H, Et , F, O, H, H, H, H, OMe, NH, O, OMe], [AI 2938; Me, H, Et, F, O, H, H, H, OEt, NH, O, OMe], [AI 2939 Me, H, Et, F, O, H, H, H, SMe, NH, O, OMe], [AI 2 940; Me, H, Et, F, O, H, H, H, CF ₃ , NH, O, OMe], [AI2941; Et, H, Et, F, O, H, H, H, H, NH, O, OMe], [AI2942; Et, H, Et, F, O, H, H, H, F, NH, O, OMe], [AI2943; Et, H, Et, F, O, H, H, H, H, Cl, NH, O, OMe], [AI 2944; Et, H, Et, F, O, H, H, H, H, Br, NH, O, OMe], [AI 2 945; Et, H, Et, Et, F, O, H, H, H, I, NH, O, OMe], [AI 2 946; Et, H, Et, F, O, H, H, H, Me, NH, O, OMe], [AI2947; Et, H, Et, F, O, H, H, H, Et, NH, O, OMe] , [AI 2948; Et, H, Et, F, O, H, H, H, c-Pr, NH, O, OMe], [AI 2949; Et, H, Et, F, O, H, H, H, H, OMe, NH, O, OMe], [AI 2 950; Et, H, Et, F, O, H, H, H, H, OEt, NH, O, OMe], [AI 2951; Et, H, Et, F, O, H, H, H, SMe, NH, O, OMe], [AI 2952; Et, H, Et, F, O, H, H, H, CF ₃ , NH, O, OMe], [AI 2953; H, H, H, H, O, F, H, H, H, NH, O, OMe], [AI 2 954; H, H, H, H, H, O, F, H, H, F, NH, O, OMe], [AI 2 955; H, H, H, H, O, F, H, H, Cl, NH, O, OMe], [AI 2956; H, H, H, H, H, O, F, H, Br, NH, O, OMe], [AI 2 957; H, H, H, H, O, F, H, H, I, NH, O, OMe], [AI 2958; H, H, H, H, H, O, F, H, Me, NH, O, OMe], [AI 2959; H, H, H, H, H, O, F, H, H, Et, NH, O, OMe], [AI 2960; H, H, H, H, H, O, F, H, c, Pr, NH, O, OMe], [AI 2961; H, H, H, H, H, O, F, H, OMe, NH, O, OMe], [AI 296 2; H, H, H, H, O, F, H, H, OEt, NH, O, OMe], [AI 2963; H, H, H, H, H, O, F, H, S Me, NH, O, OMe], [AI 2964; H, H, H, H, O, F, H, H, CF 3, NH, O, OMe], [AI2965; Cl, H, H, H, O, F, H, H, H, NH, O, OMe], [AI2966; Cl , H, H, H, O, F, H, H, F, NH, O, OMe], [AI 2967; Cl, H, H, H, H, O, F, H, Cl, NH, O, OMe ], [AI2968; Cl, H, H, H, O, F, H, H, Br, NH, O, OMe], [AI2969; Cl, H, H, H, O, F, H, H, I , NH, O, OMe], [AI 2 970; Cl, H, H, H, H, O, F, H, H, Me, NH, O, OMe], [AI 2971; Cl, H, H, H, O, F , H, H, Et, NH, O, OMe], [AI 2972; Cl, H, H, H, H, O, F, H, c, Pr, NH, O, OMe], [AI 2 973; Cl, H , H, H, O, F, H, H, OMe, NH, O, OMe], [AI 2974; Cl, H, H, H, H, O, F, H, OEt, NH, O, OMe], [AI 2 975; Cl, H, H, H, H, O, F, H, S Me, NH, O, OMe], [AI 2976; Cl, H, H, H, H, O, F, H, H, CF ₃ , NH, O, OMe], [AI2977; Me, H, H, H, H, O, F, H, H, H, NH, O, OMe], [AI 2978; Me, H, H, H, H, O, F, H, H, F, NH, O, OMe], [AI 2979; Me, H, H, H, H, O, F, H, Cl, NH, O, OMe] [AI 2 980; Me, H, H, H, H, O, F, H, H, Br, NH, O, OMe], [AI 2981; Me, H, H, H, O, F, H, H, I, NH, O, OMe], [AI2982; Me, H, H, H, H, O, F, H, Me, NH, O, OMe], [AI 2983; Me, H, H, H, O, F, H, H, Et, NH, O, OMe], [AI 2984; Me, H, H, H, H, O, F, H, c, Pr, NH, O, OMe], [AI 2985; Me, H, H, H, O, F, H, H, OMe, NH, O, OMe], [AI2986; Me, H, H, H, O, F, H, OEt, NH, O, OMe], [ AI 2 987; Me, H, H, H, H, O, F, H, S Me, NH, O, OMe], [AI 2988; Me, H, H, H, H, O, F, H, H ₃ , CF ₃ , NH , O, OMe], [AI2989; Et, H, H, H, H, O, F, H, H, H, NH, O, OMe], [AI 2 990; Et, H, H, H, O, F, H , H, F, NH, O, OMe], [AI 2991; Et, H, H, H, H, O, F, H, Cl, NH, O, OMe], [AI 299; Et, H, H, H , O, F, H, H, Br, NH, O, OMe], [AI2993; Et, H, H, H, H, O, F, H, I, NH, O, OMe], [AI 2994; Et , H, H, H, O, F, H, H, Me, NH, O, OMe], [AI 2995; Et, H, H, H, H, O, F, H, Et, NH, O, OMe ], [AI2996; Et, H, H, H, H, O, F, H, H, c-Pr, NH, O, OMe], [AI 2 997; Et, H, H, H, O, F, H, H , OMe, NH, O, OMe], [AI 2998; Et, H, H, H, H, O, F, H, OEt, NH, O, OMe], [AI 2 999; Et, H, H, H, O , F, H, H, SMe , NH, O, OMe], [AI3000; Et, H, H, H, O, F, H, H, CF 3, NH, O, OMe],

[AI 3001; H, H, F, H, O, F, H, H, H, NH, O, OMe], [AI 3002; H, H, F, H, O, F, H, H, F, NH , O, OMe], [AI 3003; H, H, F, H, O, F, H, H, Cl, NH, O, OMe], [AI 3004; H, H, F, H, O, F, H , H, Br, NH, O, OMe], [AI 3005; H, H, F, H, O, F, H, I, NH, O, OMe], [AI 3006; H, H, F, H , O, F, H, H, Me, NH, O, OMe], [AI 3007; H, H, F, H, O, F, H, Et, NH, O, OMe], [AI 3008; H , H, F, H, O, F, H, H, c, Pr, NH, O, OMe], [AI 3009; H, H, F, H, O, F, H, OMe, NH, O , OMe], [AI 3010; H, H, F, H, O, F, H, OEt, NH, O, OMe], [AI 3011; H, H, F, H, O, F, H, H , SMe, NH, O, OMe ], [AI3012; H, H, F, H, O, F, H, H, CF 3, NH, O, OMe], [AI3013; Cl, H, F, H, O, F, H, H, H, H, NH, O, OMe], [AI 3014; Cl, H, F, H, O, F, H, F, H, F, NH, O, OMe], [AI 3015; Cl, H, F, H, O, F, H, H, Cl, NH, O, OMe], [AI 3016; Cl, H, F, H, O, F, H, H, Br, NH, O, OMe] [AI 3017; Cl, H, F, H, O, F, H, I, NH, O, OMe], [AI 3018; Cl, H, F, H, O, F, H, H, Me, NH, O, OMe], [AI 3019; Cl, H, F, H, O, F, H, H, Et, NH, O, OMe], [AI 3020; Cl, H, F, H, O, F, H, H, c-Pr, NH, O, OMe], [AI 3021; Cl, H, F, H, O, F, H, H, OMe, NH, O, OMe], [AI 3022; Cl, H, F, H, O, F, H, H, OEt, NH, O, OMe], [AI3023; Cl, H, F, H, O, F, H, SMe, NH, O, OMe], [ AI 3024, Cl, H, F, H, O, F, H, H, CF ₃ , NH, O, OMe], [AI 3025; Me, H, F, H, O, F, H, H, H, NH , O, OMe], [AI 3026; Me, H, F, H, O, F, H, F, NH, O, OMe], [AI 3027; Me, H, F, H , O, F, H, H, Cl, NH, O, OMe], [AI3028; Me, H, F, H, O, F, H, Br, NH, O, OMe], [AI3029; Me , H, F, H, O, F, H, H, I, NH, O, OMe], [AI3030; Me, H, F, H, O, F, H, Me, NH, O, OMe Me, H, F, H, O, F, H, H, Et, NH, O, OMe], [AI 3032; Me, H, F, H, O, F, H, H, c] -Pr, NH, O, OMe], [AI 3033; Me, H, F, H, O, F, H, H, OMe, NH, O, OMe], [AI 3034; Me, H, F, H, O , F, H, H, OEt, NH, O, OMe], [AI 3035; Me, H, F, H, O, F, H, S Me, NH, O, OMe], [AI 3036; Me, H , F, H, O, F , H, H, CF 3, NH, O, OMe], [AI3037; Et, H, F, H, O, F, H, H, H, NH, O, OMe] , [AI3038; Et, H, F, H, O, F, H, H, F, NH, O, OMe], [AI 3039; Et, H, F, H, O, F, H, H, Cl, NH, O, OMe], [AI 3040; Et, H, F, H, O, F, H, H, Br, NH, O, OMe], [AI 3041; Et, H, F, H, O, F, H, H, I, NH, O, OMe], [AI3042; Et, H, F, H, O, F, H, Me, NH, O, OMe], [AI 3043; Et, H, F, H, O, F, H, H, Et, NH, O, OMe], [AI 3044; Et, H, F, H, O, F, H, c, Pr, NH, O, OMe], [ AI 3045; Et, H, F, H, O, F, H, OMe, NH, O, OMe], [AI 3046; Et, H, F, H, O, F, H, H, OEt, NH, O, OMe], [AI 3047; Et, H, F, H, O, F, H, S Me, NH, O, OMe], [AI 3048; Et, H, F, H, O, F, H, _{H, CF 3, NH, O} , OMe], [AI3049; H, H, Cl, H, O, F, H, H, H, NH, O, OMe], [AI3050; H, H, Cl, H , O, F, H, H, F, NH, O, OMe], [AI 3051; H, H, Cl, H, O, F, H, Cl, NH, O, OMe], [AI 3052; H , H, Cl, H, O, F, H, H, Br, NH, O, OMe], [AI 3053; H, H, Cl, H, O , F, H, H, I, NH, O, OMe], [AI 3054; H, H, Cl, H, O, F, H, Me, NH, O, OMe], [AI 3055; H, H , Cl, H, O, F, H, H, Et, NH, O, OMe], [AI 3056; H, H, Cl, H, O, F, H, c, Pr, NH, O, OMe ], [AI 3057; H, H, Cl, H, O, F, H, H, OMe, NH, O, OMe], [AI 3058; H, H, Cl, H, O, F, H, H, OEt , NH, O, OMe], [AI 3059; H, H, Cl, H, O, F, H, H, SMe, NH, O, OMe], [AI 3060; H, H, Cl, H, O, F _{, H, H, CF 3,} NH, O, OMe], [AI3061; Cl, H, Cl, H, O, F, H, H, H, NH, O, OMe], [AI3062; Cl, H, Cl, H, O, F, H, H, F, NH, O, OMe], [AI 3063; Cl, H, Cl, H, O, F, H, Cl, NH, O, OMe], [ AI 3064; Cl, H, Cl, H, O, F, H, H, Br, NH, O, OMe], [AI 3065; Cl, H, Cl, H, O, F, H, H, I, NH, O, OMe], [AI 3066; Cl, H, Cl, H, O, F, H, Me, NH, O, OMe], [AI 3067; Cl, H, Cl, H, O, F, H, H, Et, NH, O, OMe], [AI 3068; Cl, H, Cl, H, O, F, H, c, Pr, NH, O, OMe], [AI 3069; Cl, H, Cl, H, O, F, H, H, OMe, NH, O, OMe], [AI3070; Cl, H, Cl, H, O, F, H, OEt, NH, O, OMe], [AI 3071; Cl, H, Cl, H, O, F, H, H, SMe, NH, O, OMe], [AI3072; Cl, H, Cl, H, O, F, H, H, CF 3, NH, O , OMe], [AI 3073; Me, H, Cl, H, O, F, H, H, NH, O, OMe], [AI 3074; Me, H, Cl, H, O, F, H, H , F, NH, O, OMe], [AI 3075; Me, H, Cl, H, O, F, H, H, Cl, NH, O, OMe], [AI 3076; Me, H, Cl, H, O , F, H, H, Br, NH, O, OMe], [AI 3077; Me, H, Cl, H, O, F, H, I, NH, O, OMe], [AI 3078; Me, H , Cl, H, O, F, H, H, Me, NH, O, OMe], [AI 3079; Me, H, Cl, H, O, F, H, H, Et, NH, O, OMe], [AI 3080; Me, H, Cl, H, O, F, H, H, c-Pr, NH, O, OMe], [AI3081; Me, H, Cl, H, O, F, H, H, OMe, NH, O, OMe], [AI3082; Me, H, Cl, H, O, F, H, H, OEt, NH, O, OMe], [AI 3083; Me, H, Cl, H, O, F, H, S Me, NH, O, OMe], [AI 3084; Me, H, Cl, H, O, F, H, H, CF 3, NH, O, OMe], [AI3085; Et, H, Cl, H, O, F, H, H, H, NH, O, OMe], [AI3086 Et, H, Cl, H, O, F, H, H, F, NH, O, OMe], [AI 3087; Et, H, Cl, H, O, F, H, Cl, NH, O , OMe], [AI 3088; Et, H, Cl, H, O, F, H, H, Br, NH, O, OMe], [AI 3089; Et, H, Cl, H, O, F, H, H , I, NH, O, OMe], [AI 3090; Et, H, Cl, H, O, F, H, Me, NH, O, OMe], [AI 3091; Et, H, Cl, H, O , F, H, H, Et, NH, O, OMe], [AI3092; Et, H, Cl, H, O, F, H, c, Pr, NH, O, OMe], [AI 3093; Et , H, Cl, H, O, F, H, H, OMe, NH, O, OMe], [AI 3094; Et, H, Cl, H, O, F, H, OEt, NH, O, OMe ], [AI 3095; Et, H, Cl, H, O, F, H, S Me, NH, O, OMe], [AI 3096; Et, H, Cl, H, O, F, H, H, CF] ₃ , NH, O, OMe], [AI 3097; H, H, Me, H, O, F, H, H, H, NH, O, OMe], [AI 3098; H, H, Me, H, O, F, H, H, F, NH, O, OMe], [AI 3099; H, H, Me, H, O, F, H, H, Cl, NH, O, OMe], [AI 3 100; H, H, Me, H, O, F, H, H, Br, NH, O, OMe],

[AI3101; H, H, Me, H, O, F, H, I, NH, O, OMe], [AI 3102; H, H, Me, H, O, F, H, H, Me, NH , O, OMe], [AI 3103; H, H, Me, H, O, F, H, Et, NH, O, OMe], [AI 3104; H, H, Me, H, O, F, H , H, c-Pr, NH, O, OMe], [AI 3105; H, H, Me, H, O, F, H, OMe, NH, O, OMe], [AI 3106; H, H, Me , H, O, F, H, H, OEt, NH, O, OMe], [AI 3107; H, H, Me, H, O, F, H, S Me, NH, O, OMe], [AI 3108 ; H, H, Me, H , O, F, H, H, CF 3, NH, O, OMe], [AI3109; Cl, H, Me, H, O, F, H, H, H, NH, O, OMe], [AI 3110; Cl, H, Me, H, O, F, H, H, F, NH, O, OMe], [AI 3 111; Cl, H, Me, H, O, F, H, H, Cl, NH, O, OMe], [AI 3 112; Cl, H, Me, H, O, F, H, H, Br, NH, O, OMe], [AI 3 113; Cl, H, Me, H, O, F, H, H, I, NH, O, OMe], [AI 3114; Cl, H, Me, H, O, F, H, Me, NH, O, OMe], [AI 3 115; Cl, H, Me, H, O, F, H, H, Et, NH, O, OMe], [AI 3116; Cl, H, Me, H, O, F, H, H, c-Pr, NH, O, OMe], [AI3117; Cl, H, Me, H, O, F, H, H, OMe, NH, O, OMe], [AI 3118; Cl, H, Me, H, O, F, H, H, H, OEt, NH, O, OMe], [AI3119; Cl, H, Me, H, O, F, H, SMe, NH, O, OMe], [AI 3 120; Cl, H, Me, H, O, _{F, H, H, CF 3} , NH, O, OMe], [AI3121; Me, H, Me, H, O, F, H, H, H, NH, O, OMe], [AI3122; Me, H , Me, H, O, F, H, H, F, NH, O, OMe], [AI 3123; Me, H, Me, H, O, F, H, Cl, NH, O, OMe], [AI 3 124; Me, H, Me, H, O, F, H, H, Br, NH, O, OMe], [AI 3 125; Me, H, Me, H, O, F, H, H, I, NH , O, OMe], [AI 3 126; Me, H, Me, H, O, F, H, H, Me, NH, O, OMe], [AI 3 127; Me, H, Me, H, O, F, H, H, Et, NH, O, OMe], [AI 3 128; Me, H, Me, H, O, F, H, H, c-Pr, NH, O, OMe], [AI 3129; Me, H, Me, H, O, F, H, OMe, NH, O, OMe], [AI 3130; Me, H, Me, H, O, F, H, H, OEt, NH, O, OMe], [AI 3131; Me, H, Me, H, O, F, H, SMe, NH, O, OMe], [AI3132; Me, H, Me, H, O, F, H, H, CF 3, NH, O, OMe], [AI3133; Et, H, Me, H, O, F, H, H H, NH, O, OMe], [AI 3 134; Et, H, Me, H, O, F, H, F, H, F, NH, O, OMe], [AI 3 135; Et, H, Me, H, O , F, H, H, Cl, NH, O, OMe], [AI 3136; Et, H, Me, H, O, F, H, H, Br, NH, O, OMe], [AI 3 137; Et, H , Me, H, O, F, H, H, I, NH, O, OMe], [AI 3138; Et, H, Me, H, O, F, H, Me, NH, O, OMe], [AI3139; Et, H, Me, H, O, F, H, H, Et, NH, O, OMe], [AI 3140; Et, H, Me, H, O, F, H, H, c-Pr , NH, O, OMe], [AI 3141; Et, H, Me, H, O, F, H, H, OMe, NH, O, OMe], [AI 3142; Et, H, Me, H, O, F , H, H, OEt, NH, O, OMe], [AI3143; Et, H, Me, H, O, F, H, SMe, NH, O, OMe], [AI 3144; Et, H, Me , H, O, F, H , H, CF 3, NH, O, OMe], [AI3145; H, H, Et, H, O, F, H, H, H, NH, O, OMe], [ AI 3146; H, H, Et, H, O, F, H, H, F, NH, O, OMe], [AI 3147; H, H, Et, H, O, F, H, H, Cl, NH, O, OMe], [AI3148; H, H, Et, H, O, F, H, H, Br, NH, O, OMe], [AI 3149; H, H, Et, H, O, F, H, H, I, NH, O, OMe], [AI 3150; H, H, Et, H, O, F, H, Me, NH, O, OMe], [AI 3151; H, H, Et, H, O, F, H, H, Et, NH, O, OMe], [AI 3152 H, H, Et, H, O, F, H, H, c-Pr, NH, O, OMe], [AI 3153; H, H, Et, H, O, F, H, H, OMe, NH , O, OMe], [AI 3 154; H, H, Et, H, O, F, H, OEt, NH, O, OMe], [AI 3 155; H, H, Et, H, O, F, H , H, SMe, NH, O, OMe], [AI 3156; H, H, Et, H, O, F, H, CF ₃ , NH, O, OMe], [AI ₃ 157; Cl, H, Et, H, O, F, H, H, H, H, NH, O, OMe], [AI 3158; Cl, H, Et, H, O, F, H, F, NH, O, OMe], [AI 3 159; Cl, H, Et, H, O, F, H, H, Cl, NH, O, OMe], [AI 3 160; Cl, H, Et, H, O, F, H, H, Br, NH, O, OMe], [AI3161; Cl, H, Et, H, O, F, H, I, NH, O, OMe], [AI3162; Cl, H, Et, H, O, F, H, H, Me, NH, O, OMe], [AI 3163; Cl, H, Et, H, O, F, H, H, Et, NH, O, OMe], [AI 3 164; Cl, H, Et, H, O, F, H, H, c-Pr, NH, O, OMe], [AI 3165; Cl, H, Et, H, O, F, H, H, OMe, NH, O, OMe], [AI 3166; H, Et, H, O, F, H, H, OEt, NH, O, OMe], [AI 3 167; Cl, H, Et, H, O, F, H, S Me, NH, O, OMe] , [AI3168; Cl, H, Et, H, O, F, H, H, CF 3, NH, O, OMe], [AI3169; Me, H, Et, H, O, F, H, H, H , NH, O, OMe], [AI 3170; Me, H, Et, H, O, F, H, H, F, NH, O, OMe], [AI 3171; Me, H, Et, H, O, F , H, H, Cl, NH, O, OMe], [AI 3172; Me, H, Et, H, O, F, H, H, Br, NH, O, OMe], [AI 3173; Me, H, Et , H, O, F, H, H, I, NH, O, OMe], [AI 3174; Me, H, Et, H, O, F, H, Me, NH, O, OMe], [AI 3 175 Me, H, Et, H, O, F, H, H, Et, NH, O, OMe], [AI 3176; Me, H, Et, H, O, F, H, H, c-Pr, NH , O, OMe], [AI3177; Me, H, Et, H, O, F, H, H , OMe, NH, O, OMe], [AI3178; Me, H, Et, H, O, F, H, OEt, NH, O, OMe], [AI 3179; Me, H, Et, H, O , F, H, H, SMe , NH, O, OMe], [AI3180; Me, H, Et, H, O, F, H, H, CF 3, NH, O, OMe], [AI3181; Et, H, Et, H, O, F, H, H, H, H, NH, O, OMe], [AI 3182; Et, H, Et, H, O, F, H, F, H, F, NH, O, OMe] [AI 3183; Et, H, Et, H, O, F, H, H, Cl, NH, O, OMe], [AI 3184; Et, H, Et, H, O, F, H, H, Br, NH, O, OMe], [AI 3 185; Et, H, Et, H, O, F, H, H, I, NH, O, OMe], [AI 3186; Et, H, Et, H, O, F, H, H, Me, NH, O, OMe], [AI3187; Et, H, Et, H, O, F, H, Et, NH, O, OMe], [AI 3188; Et, H, Et, H, O, F, H, H, c-Pr, NH, O, OMe], [AI 3189; Et, H, Et, H, O, F, H, OMe, NH, O, OMe], [ AI 3190; Et, H, Et, H, O, F, H, H, OEt, NH, O, OMe], [AI 3191; Et, H, Et, H, O, F, H, H, SMe, NH, O, OMe], [AI3192; Et, H, Et, H, O, F, H, H, CF 3, NH, O, OMe], [AI3193; H, H, H, H, O, H, F , H, H, NH, O, OMe], [AI 3194; H, H, H, H, H, O, H, F, H, F, NH, O, OMe], [AI 3 195; H, H, H, H , O, H, F, H, Cl, NH, O, OMe], [AI 3 196; H, H, H, H, H, O, H, F, H, Br, NH, O, OMe], [AI 3 197; H , H, H, H, O, H, F, H, I, NH, O, OMe], [AI 3198; H, H, H, H, O, H, F, H, Me, NH, O, OMe ], [AI 3199; H, H, H, H, O, H, F, H, Et, NH, O, OMe], [AI 3200; H, H, H, H, O, H, F, H, c -Pr, NH, O, OMe],

[AI3201; H, H, H, H, H, O, H, F, H, OMe, NH, O, OMe], [AI 3202; H, H, H, H, H, O, H, F, H, OEt, NH H, H, H, H, H, O, H, F, H, SMe, NH, O, OMe], [AI 3 204; H, H, H, H, O, H, F _{, H, CF 3, NH,} O, OMe], [AI3205; Cl, H, H, H, O, H, F, H, H, NH, O, OMe], [AI3206; Cl, H, H, H, O, H, F, H, F, NH, O, OMe], [AI 3207; Cl, H, H, H, H, O, H, F, H, Cl, NH, O, OMe], [AI 3 208; Cl, H, H, H, H, O, H, F, H, Br, NH, O, OMe], [AI 3209; Cl, H, H, H, H, O, H, F, H, I, NH, O, OMe], [AI 3210; Cl, H, H, H, O, H, F, H, Me, NH, O, OMe], [AI 3211; Cl, H, H, H, O, H, F, H, Et, NH, O, OMe], [AI 3212; Cl, H, H, H, H, O, H, F, H, c, Pr, NH, O, OMe], [AI 3213; Cl, H, H, H, O, H, F, H, OMe, NH, O, OMe], [AI 3214; Cl, H, H, H, H, O, H, F, H, OE t, NH, O, OMe], [AI 3215; Cl, H, H, H, O, H, F, H, SMe, NH, O, OMe], [AI3216; Cl, H, H, H, O, H, F, H, CF 3, NH, O, OMe Me, H, H, H, H, O, H, F, H, H, NH, O, OMe], [AI 3218; Me, H, H, H, O, H, F, H, F] , NH, O, OMe], [AI 3219; Me, H, H, H, H, O, H, H, F, H, Cl, NH, O, OMe], [AI 3220; Me, H, H, H, O, H , F, H, Br, NH, O, OMe], [AI3221; Me, H, H, H, H, O, H, F, H, I, NH, O, OMe], [AI 3222; Me, H, H , H, O, H, F, H, Me, NH, O, OMe], [AI 3223; Me, H, H, H, H, O, H, F, H, Et, NH, O, OMe], [AI 3224 Me, H, H, H, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3225; Me, H, H, H, H, O, H, F, H, OMe, NH , O, OMe], [AI 3226; Me, H, H, H, O, H, F, H, OEt, NH, O, OMe], [AI 3 227; Me, H, H, H, H, O, H, F, H, SMe, NH, O, OMe], [AI 3228; Me, H, H, H, H, O, H, F, H, CF ₃ , NH , O, OMe], [AI 3229; Et, H, H, H, H, O, H, F, H, H, NH, O, OMe], [AI 3230; Et, H, H, H, O, H, F , H, F, NH, O, OMe], [AI3231; Et, H, H, H, H, O, H, F, H, Cl, NH, O, OMe], [AI3232; Et, H, H, H , O, H, F, H, Br, NH, O, OMe], [AI3233; Et, H, H, H, H, O, H, F, H, I, NH, O, OMe], [AI 3234; Et , H, H, H, O, H, F, H, Me, NH, O, OMe], [AI 3235; Et, H, H, H, H, O, H, F, H, Et, NH, O, OMe ], [AI 3236; Et, H, H, H, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3237; Et, H, H, H, O, H, F, H , OMe, NH, O, OMe], [AI 3238; Et, H, H, H, H, O, H, F, H, OEt, NH, O, OMe], [AI 3239; Et, H, H, H, O , H, F, H, SMe , NH, O, OMe], [AI3240; Et, H, H, H, O, H, F, H, CF 3, NH, O, OMe], [AI3241; H, H, F, H, O, H, F, H, H, NH, O, OMe], [AI 3242; H, H, F, H, O, H, F, H, F, NH, O, OMe] [AI 3243; H, H, F, H, O, H, F, H, Cl, NH, O, OMe], [AI 3244; H, H, F, H, O, H, F, H, Br, NH, O, OMe], [AI 3245; H, H, F, H, O, H, F, H, I, NH, O, OMe], [AI 3246; H, H, F, H, O, H, F, H, Me, NH, O, OMe], [AI3247; H, H, F, H, O, H, F, H, Et, NH, O, OMe], [AI 3248; H, H, F, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3249; H, H, F, H, O, H, F, H, OMe, NH, O, OMe], [ AI 3250; H, H, F, H, O, H, F, H, OEt, NH, O, OMe], [AI 3251; H, H, F, H, O, H, F, H, SMe, NH, O, OMe], [AI 3252; H, H, F, H, O, H, F, H, CF ₃ , NH, O, OMe], [AI 3253; Cl, H, F , H, O, H, F, H, H, NH, O, OMe], [AI 3 254; Cl, H, F, H, O, H, F, H, F, NH, O, OMe], [AI 3 255 Cl, H, F, H, O, H, F, H, Cl, NH, O, OMe], [AI 3256; Cl, H, F, H, O, H, F, H, Br, NH, O , OMe], [AI 3 257; Cl, H, F, H, O, H, F, H, I, NH, O, OMe], [AI 3 258; Cl, H, F, H, O, H, F, H , Me, NH, O, OMe], [AI 3259; Cl, H, F, H, O, H, F, H, Et, NH, O, OMe], [AI 3 260; Cl, H, F, H, O , H, F, H, c-Pr, NH, O, OMe], [AI3261; Cl, H, F, H, O, H, F, H, OMe, NH, O, OMe], [AI 3262; Cl , H, F, H, O, H, F, H, OEt, NH, O, OMe], [AI 3263; Cl, H, F, H, O, H, F, H, SMe, NH, O, OMe ], [AI3264; Cl, H, F, H, O, H, F, H, CF3, NH, O, OMe], [AI ₃ 265; Me, H, F, H, O, H, F, H, H, NH, O, OMe], [AI 3 266; Me, H, F, H, O, H, F, H, F, NH, O, OMe], [AI 3 267: Me, H, F, H, O, H, F, H, Cl, NH, O, OMe], [AI 3268; Me, H, F, H, O, H, F, H, Br, NH, O, OMe], [AI 3269; Me, H, F, H, O, H, F, H, I, NH, O, OMe], [AI 3270; Me, H, F, H, O, H, F, H, Me, NH, O, OMe], [ AI3271; Me, H, F, H, O, H, F, H, Et, NH, O, OMe], [AI3272; Me, H, F, H, O, H, F, H, c-Pr, NH, O, OMe], [AI3273; Me, H, F, H, O, H, F, H, OMe, NH, O, OMe], [AI 3274; Me, H, F, H, O, H, F, H, OEt, NH, O, OMe], [AI3275; Me, H, F, H, O, H, F, H, SMe, NH, O, OMe], [AI 3276; Me, H, F, H, O, H, F, H, CF 3, NH, O, OMe], [AI3277; Et, H, F, H, O, H, F, H, H, NH, O, OMe], [AI3278 Et, H, F, H, O, H, F, H, F, NH, O, OMe], [AI 3279; Et, H, F, H, O , H, F, H, Cl, NH, O, OMe], [AI 3280; Et, H, F, H, O, H, F, H, Br, NH, O, OMe], [AI 3281; Et, H , F, H, O, H, F, H, I, NH, O, OMe], [AI3282; Et, H, F, H, O, H, F, H, Me, NH, O, OMe], [AI 3283; Et, H, F, H, O, H, F, H, Et, NH, O, OMe], [AI 3284; Et, H, F, H, O, H, F, H, c-Pr , NH, O, OMe], [AI 3285; Et, H, F, H, O, H, F, H, OMe, NH, O, OMe], [AI 3 286; Et, H, F, H, O, H , F, H, OEt, NH, O, OMe], [AI 3 287; Et, H, F, H, O, H, F, H, SMe, NH, O, OMe], [AI 3 288; Et, H, F , H, O, H, F , H, CF 3, NH, O, OMe], [AI3289; H, H, Cl, H, O, H, F, H, H, NH, O, OMe], [ AI 3290; H, H, Cl, H, O, H, F, H, F, NH, O, OMe], [AI 3291; H, H, Cl, H, O, H, F, H, Cl, NH, O, OMe], [AI3292; H, H, Cl, H, O, H, F, H, Br, NH, O, OMe], [AI 3293; H, H, Cl, H, O, H, F, H, I, NH, O, OMe], [AI3294; H, H, Cl, H, O, H, F, H, Me, NH, O, OMe], [AI 3295; H, H, Cl, H, O, H, F, H, Et, NH, O, OMe], [AI 3 296; H, H, Cl, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3 297; H, H, Cl, H, O, H, F, H, OMe, NH, O, OMe], [AI 3298; H, H, Cl, H, O, H, F, H, OEt, NH, O, OMe], [AI3299; H, H, Cl, H, O, H, F, H, SMe, NH, O, OMe], [AI 3300; H, H, Cl, H, O, H, F, H, _{CF 3, NH, O, OMe} ],

[AI 3301; Cl, H, Cl, H, O, H, F, H, H, NH, O, OMe], [AI 3302; Cl, H, Cl, H, O, H, F, H, F, NH , O, OMe], [AI 3303; Cl, H, Cl, H, O, H, F, H, Cl, NH, O, OMe], [AI 3304; Cl, H, Cl, H, O, H, F , H, Br, NH, O, OMe], [AI 3305; Cl, H, Cl, H, O, H, F, H, I, NH, O, OMe], [AI 3306; Cl, H, Cl, H , O, H, F, H, Me, NH, O, OMe], [AI 3307; Cl, H, Cl, H, O, H, F, H, Et, NH, O, OMe], [AI 3308; Cl , H, Cl, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3309; Cl, H, Cl, H, O, H, F, H, OMe, NH, O , OMe], [AI 3310; Cl, H, Cl, H, O, H, F, H, OEt, NH, O, OMe], [AI 3311; Cl, H, Cl, H, O, H, F, H , SMe, NH, O, OMe ], [AI3312; Cl, H, Cl, H, O, H, F, H, CF 3, NH, O, OMe], [AI3313; Me, H, Cl, H, O, H, F, H, H, NH, O, OMe], [AI 3314; Me, H, Cl, H, O, H, F, H, F, NH, O, OMe], [AI 3315; H, Cl, H, O, H, F, H, Cl, NH, O, OMe], [AI3316; Me, H, Cl, H, O, H, F, H, Br, NH, O, OMe] , [AI3317; Me, H, Cl, H, O, H, F, H, I, NH, O, OMe], [AI 3318; Me, H, Cl, H, O, H, F, H, Me, NH, O, OMe], [AI 3319; Me, H, Cl, H, O, H, F, H, Et, NH, O, OMe], [AI 3320; Me, H, Cl, H, O, H, F, H, c-Pr, NH, O, OMe], [AI3321; Me, H, Cl, H, O, H, F, H, OMe, NH, O, OMe], [AI3322; Me, H, Cl, H, O, H, F, H, OEt, NH, O, OMe], [AI3323; Me, H, Cl, H, O, H, F, H, SMe, NH, O, OMe], [ AI3324; Me, H, Cl, H, O, H, F, H, CF 3, NH, O, OMe], [AI3325; Et, H, Cl, H, O, H, F, H, H, NH , O, OMe], [AI 3326; Et, H, Cl, H, O, H, F, H, F, NH, O, OMe], [AI 3327; Et, H, Cl, H, O, H, F, H, Cl, NH, O, OMe], [AI 3328; Et, H, Cl, H, O, H, F, H, Br, NH, O, OMe], [AI 3329; Et, H, Cl, H, O, H, F, H, I, NH, O, OMe], [AI3330; Et, H, Cl, H, O, H, F, H, Me, NH, O, OMe], [AI3331; Et, H, Cl, H, O, H, F, H, Et, NH, O, OMe], [AI3332; Et, H, Cl, H, O, H, H, F, H, c-Pr, NH, O, OMe], [AI3333; Et, H, Cl, H, O, H, F, H, OMe, NH, O, OMe], [AI 3334; Et, H, Cl, H, O, H, F, H, OE t, NH, O, OMe], [AI 3 335; Et, H, Cl, H, O, H, F, H, SMe, NH, O, OMe], [AI3336; Et, H, Cl, H, O, H, F, H, CF 3, NH, O, OMe H, H, Me, H, O, H, F, H, H, NH, O, OMe], [AI 3338; H, H, Me, H, O, H, F, H, F] , NH, O, OMe], [AI3339; H, H, Me, H, O, H, F, H, Cl, NH, O, OMe], [AI 3340; H, H, Me, H, O, H , F, H, Br, NH, O, OMe], [AI3341; H, H, Me, H, O, H, F, H, I, NH, O, OMe], [AI3342; H, H, Me , H, O, H, F, H, Me, NH, O, OMe], [AI 3343; H, H, Me, H, O, H, F, H, Et, NH, O, OMe], [AI 3344 H, H, Me, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3345; H, H, Me, H, O, H, F, H, OMe, NH , O, OMe], [AI 3346; H, H, Me, H, O, H, F, H, OEt, NH, O, OMe], [AI 3347; H, H, Me, H, O, H, F , H, SMe, NH, O , OMe], [AI3348; H, H, Me, H, O, H, F, H, CF 3, NH, O, OMe], [AI3349; Cl, H, Me, H, O, H, F, H, H, NH, O, OMe], [AI 3 350; Cl, H, Me, H, O, H, F, H, F, NH, O, OMe], [AI 3351; Cl, H, Me, H, O, H, F, H, Cl, NH, O, OMe], [AI 33 52; Cl, H, Me, H, O, H, F, H, Br, NH, O, OMe], [AI 3353; Cl, H, Me, H, O, H, F, H, I, NH, O, OMe], [AI 3354; Cl, H, Me, H, O, H, F, H, Me, NH, O, OMe], [AI 3355; Cl, H, Me, H, O, H, F, H, Et, NH, O, OMe], [AI 3356; Cl, H, Me, H, O, H, F, H, c, Pr, NH, O, OMe], [AI 3357; Cl, H, Me, H, O, H, F, H, OMe, NH, O, OMe], [AI 3358; Cl, H, Me, H, O, H, F, H, OEt, NH, O, OMe], [AI 3359; Cl, H, Me, H, O, H, F, H, SMe, NH, O, OMe], [AI 3360; Cl, H, Me, H, O, H, F, H, CF ₃ , NH, O , OMe], [AI3361; Me, H, Me, H, O, H, F, H, H, NH, O, OMe], [AI3362; Me, H, Me, H, O, H, F, H , F, NH, O, OMe], [AI3363; Me, H, Me, H, O, H, H, F, H, Cl, NH, O, OMe], [AI 3364; Me, H, Me, H, O , H, F, H, Br, NH, O, OMe], [AI 3365; Me, H, Me, H, O, H, F, H, I, NH, O, OMe], [AI 3 366; Me, H , Me, H, O, H, F, H, Me, NH, O, OMe], [AI 3367; Me, H, Me, H, O, H, F, H, Et, NH, O, OMe], [AI3368; Me, H, Me, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3369; Me, H, Me, H, O, H, F, H, OMe , NH, O, OMe], [AI3370; Me, H, Me, H, O, H, F, H, OEt, NH, O, OMe], [AI3371; Me, H, Me, H, O, H , F, H, SMe, NH , O, OMe], [AI3372; Me, H, Me, H, O, H, F, H, CF 3, NH, O, OMe], [AI3373; Et, H, Me, H, O, H, F, H, H, NH, O, OMe], [AI 3374; Et, H, Me, H, O, H, F, H, F, NH, O, OMe], [ AI 3375; Et, H, Me, H, O, H, F, H, Cl, NH, O, OMe], [AI 3376; Et, H, Me, H, O, H, F, H, Br, NH, O, OMe], [AI 3377; Et, H, Me, H, O, H, F, H, I, NH, O, OMe], [AI 3378; Et, H, Me, H, O, H, F, H, Me, NH, O, OMe], [AI 3379; Et, H, Me, H, O, H, F, H, Et, NH, O, OMe], [AI 3380; Et, H, Me, H, O, H, F, H, c-Pr, NH, O, OMe] [AI3381; Et, H, Me, H, O, H, F, H, OMe, NH, O, OMe], [AI3382; Et, H, Me, H, O, H, F, H, OEt, NH, O, OMe], [AI 3383; Et, H, Me, H, O, H, F, H, S Me, NH, O, OMe], [AI 3384; Et, H, Me, H, O, H, _{F, H, CF 3, NH} , O, OMe], [AI3385; H, H, Et, H, O, H, F, H, H, NH, O, OMe], [AI3386; H, H, Et , H, O, H, F, H, F, NH, O, OMe], [AI 3387; H, H, Et, H, O, H, F, H, Cl, NH, O, OMe], [AI 3388] H, H, Et, H, O, H, F, H, Br, NH, O, OMe], [AI 3389; H, H, Et, H, O, H, F, H, I, NH, O , OMe], [AI 3390; H, H, Et, H, O, H, F, H, Me, NH, O, OMe], [AI3391; H, H, Et, H, O, H, F, H , Et, NH, O, OMe], [AI3392; H, H, Et, H, O, H, F, H, c, Pr, NH, O, OMe], [AI3393; H, H, Et, H , O, H, F, H, OMe, NH, O, OMe], [AI 3394; H, H, Et, H, O, H, F, H, OEt, NH, O, OMe], [AI 3395; H , H, Et, H, O, H, F, H, SMe, NH, O, OMe], [AI 3396; H, H, Et, H, O, H, F, H, CF ₃ , NH, O, OMe], [AI 3397; Cl, H, Et, H, O, H, F, H, H, NH, O, OMe], [AI 3398; Cl, H, Et, H, O, H, F, H, F, NH, O, OMe], [AI 3399; Cl, H, Et, H, O, H, F, H, Cl, NH, O, OMe], [AI 3400; Cl, H, Et, H, O, H, F, H, Br, NH, O, OMe],

[AI 3401; Cl, H, Et, H, O, H, F, H, I, NH, O, OMe], [AI 3402; Cl, H, Et, H, O, H, F, H, Me, NH , O, OMe], [AI 3403; Cl, H, Et, H, O, H, F, H, Et, NH, O, OMe], [AI 3404; Cl, H, Et, H, O, H, F , H, c-Pr, NH, O, OMe], [AI 3405; Cl, H, Et, H, O, H, F, H, OMe, NH, O, OMe], [AI 3406; Cl, H, Et , H, O, H, F, H, OEt, NH, O, OMe], [AI 3407; Cl, H, Et, H, O, H, F, H, SMe, NH, O, OMe], [AI 3408 ; Cl, H, Et, H , O, H, F, H, CF 3, NH, O, OMe], [AI3409; Me, H, Et, H, O, H, F, H, H, NH, O, OMe], [AI 3410; Me, H, Et, H, O, H, F, H, F, NH, O, OMe], [AI 3411; Me, H, Et, H, O, H, F, H, Cl, NH, O, OMe], [AI 3412; Me, H, Et, H, O, H, F, H, H, Br, NH, O, OMe], [AI 3413; Me, H, Et, H, O, H, F, H, I, NH, O, OMe], [AI 3414; Me, H, Et, H, O, H, F, H, Me, NH, O, OMe], [AI 3415; H, Et, H, O, H, F, H, Et, NH, O, OMe], [AI 3416; Me, H, Et, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3417; Me, H, Et, H, O, H, F, H, OMe, NH, O, OMe], [AI 3418; Me, H, Et, H, O, H, F, H, OEt, NH, O, OMe], [AI3419; Me, H, Et, H, O, H, H, F, H, SMe, NH, O, OMe], [AI 3420; Me, H, Et, H, O, _{H, F, H, CF 3} , NH, O, OMe], [AI3421; Et, H, Et, H, O, H, F, H, H, NH, O, OMe], [AI3422; Et, H , Et, H, O, H, F, H, F, NH, O, OMe], [AI 3423; Et, H, Et, H, O, H, F, H, Cl, NH, O, OMe], [AI 3424; Et, H, Et, H, O, H, F, H, Br, NH, O, OMe], [AI 3425; Et, H, Et, H, O, H, F, H, I, NH , O, OMe], [AI 3426; Et, H, Et, H, O, H, F, H, Me, NH, O, OMe], [AI 3427; Et, H, Et, H, O, H, F, H, Et, NH, O, OMe], [AI 3428; Et, H, Et, H, O, H, F, H, c-Pr, NH, O, OMe], [AI 3429; Et, H, Et, H, O, H, F, H, OMe, NH, O, OMe], [AI 3430; Et, H, Et, H, O, H, F, H, OEt, NH, O, OMe], [AI 3431; Et, H, Et, H, O, H, F, H, SMe, NH, O, OMe], [AI 3432; Et, H, Et, H, O, H, F, H, CF ₃ , NH, O, OMe], [AI 3433; H, H, H, H , O, H, H, F, H, NH, O, OMe], [AI 3434; H, H, H, H, H, O, H, F, F, NH, O, OMe], [AI 3435; H , H, H, H, O, H, H, F, Cl, NH, O, OMe], [AI 3436; H, H, H, H, O, H, H, F, Br, NH, O, OMe H, H, H, H, H, O, H, H, F, I, NH, O, OMe], [AI 3438; H, H, H, H, O, H, H, F, Me] , NH, O, OMe], [AI 3439; H, H, H, H, H, O, H, H, F, Et, NH, O, OMe], [AI 3440; H, H, H, H, O, H , H, F, c-Pr, NH, O, OMe], [AI3441; H, H, H, H, H, O, H, F, OMe, NH, O, OMe], [AI3442; H, H , H, H, O, H, H, F, OEt, NH, O, OMe], [AI 3443; H, H, H, H, H, O, H, F, SMe, NH, O, OMe], [AI3444; H, H, H , H, O, H, H, F, CF 3, NH, O, OMe], [AI3445; Cl, H, H, H, O, H, H, F, H, NH, O, OMe], [AI3446; Cl, H, H, H, H, O, H, H, H, F, F, NH, O, OMe], [AI 3447; Cl, H, H, H, O, H, H, F, Cl, NH, O, OMe], [AI 3448; Cl, H, H, H, H, O, H, H, F, Br, NH, O, OMe], [AI 3449; Cl, H, H, H, O, H, H, F, I, NH, O, OMe], [AI 3450; Cl, H, H, H, H, O, H, F, Me, NH, O, OMe], [AI 3451; Cl, H, H, H, H, O, H, H, F, Et, NH, O, OMe], [AI3452; Cl, H, H, H, O, H, H, H, H F, c-Pr, NH, O, OMe], [AI 3453; Cl, H, H, H, H, O, H, H, F, OMe, NH, O, OMe], [AI 3454; Cl, H, H, H, O, H, H, F, OEt, NH, O, OMe], [AI 3455; Cl, H, H, H, H, O, H, F, SMe, NH, O, OMe], [AI 3456; Cl, H, H, H, O, H, H, F, CF 3, NH, O, OMe], [AI3457; Me, H, H, H, O, H, H, F, H, NH, O , OMe], [AI 3458; Me, H, H, H, O, H, H, F, F, NH, O, OMe], [AI 3459; Me, H, H, H, O, H, H, F , Cl, NH, O, OMe], [AI 3460; Me, H, H, H, H, O, H, H, F, Br, NH, O, OMe], [AI3461; Me, H, H, H, O , H, H, F, I, NH, O, OMe], [AI3462; Me, H, H, H, H, O, H, H, F, Me, NH, O, OMe], [AI3463; , H, H, O, H, H, F, Et, NH, O, OMe], [AI 3464; Me, H, H, H, O, H, F, c, Pr, NH, O, OMe Me, H, H, H, H, O, H, H, F, OMe, NH, O, OMe], [AI 3466; Me, H, H, H, O, H, H, F, OEt] , NH, O, OMe], [AI 3467; Me, H, H, H, H, O, H, H, F, SMe, NH, O, OMe], [AI 3468; Me, H, H, H, O, H _{, H, F, CF 3,} NH, O, OMe], [AI3469; Et, H, H, H, O, H, H, F, H, NH, O, OMe], [AI3470; Et, H, H, H, O, H, H, F, F, F, NH, O, OMe], [AI 3471; Et, H, H, H, O, H, F, Cl, NH, O, OMe], [ AI 3472; Et, H, H, H, H, O, H, H, F, Br, NH, O, OMe], [AI 3473; Et, H, H, H, H, O, H, H, F, I, NH, O, OMe], [AI3474; Et, H, H, H, H, O, H, H, F, Me, NH, O, OMe], [AI 3475; Et, H, H, H, O, H, H, F, Et, NH, O, OMe], [AI 3476; Et, H, H, H, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3477; Et, H, H, H, O, H, H, F, OMe, NH, O, OMe], [AI 3478; Et, H, H, H, O, H, H , F, OEt, NH, O, OMe], [AI 3479; Et, H, H, H, H, O, H, H, F, SMe, NH, O, OMe], [AI 3 480; Et, H, H, H , O, H, H, F , CF 3, NH, O, OMe], [AI3481; H, H, F, H, O, H, H, F, H, NH, O, OMe], [AI3482; H, H, F, H, O, H, H, F, F, NH, O, OMe], [AI3483; H, H, F, H, O, H, H, F, Cl, NH, O, OMe], [AI3484; H, H, F, H, O, H, H, F, Br, NH, O, OMe], [AI 3485; H, H, F, H, O, H, H, F, H, H, F, H, O, H, H, F, Me, NH, O, OMe], [AI 3487; H, H, F, H, O, I, NH, O, OMe], [AI 3486; H, H, F, Et, NH, O, OMe], [AI 3488; H, H, F, H, O, H, F, c, Pr, NH, O, OMe], [AI 3489; H, H, F, H, O, H, H, F, OMe, NH, O, OMe], [AI 3490; H, H, F, H, O, H, H, F, OE t, NH, O, OMe] , [AI3491; H, H, F, H, O, H, H, F, SMe, NH, O, OMe], [AI3492; H, H, F, H, O, H, H, F, CF ₃ , NH, O, OMe], [AI3493; Cl, H, F, H, O, H, H, F, H, NH, O, OMe], [AI 3494; Cl, H, F, H, O, H , H, F, F, NH, O, OMe], [AI 3495; Cl, H, F, H, O, H, H, F, Cl, NH, O, OMe], [AI 3 496; Cl, H, F , H, O, H, H, F, Br, NH, O, OMe], [AI 3497; Cl, H, F, H, O, H, H, F, I, NH, O, OMe], [AI 3498 Cl, H, F, H, O, H, H, F, Me, NH, O, OMe], [AI 3499; Cl, H, F, H, O, H, H, F, Et, NH, O , OMe], [AI3500; Cl, H, F, H, O, H, H, F, c-Pr, NH, O, OMe],

[AI 3501; Cl, H, F, H, O, H, H, F, OMe, NH, O, OMe], [AI 3502; Cl, H, F, H, O, H, H, F, OEt, NH , O, OMe], [AI3503; Cl, H, F, H, O, H, H, F, SMe, NH, O, OMe], [AI 3504; Cl, H, F, H, O, H, H _{, F, CF 3, NH,} O, OMe], [AI3505; Me, H, F, H, O, H, H, F, H, NH, O, OMe], [AI3506; Me, H, F, H, O, H, H, F, F, F, NH, O, OMe], [AI 3507; Me, H, F, H, O, H, F, Cl, NH, O, OMe], [AI 3508; Me, H, F, H, O, H, H, F, Br, NH, O, OMe], [AI 3509; Me, H, F, H, O, H, H, F, I, NH, O, OMe], [AI 3510; Me, H, F, H, O, H, H, F, Me, NH, O, OMe], [AI 3511; Me, H, F, H, O, H, H, F, Et, NH, O, OMe], [AI 3512; Me, H, F, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3513; Me, H, F, H, O, H, H, F, OMe, NH, O, OMe], [AI 3514; Me, H, F, H, O, H, H, F, OEt, NH, O, OMe], [AI 3515; Me, H, F, H, O, H, H, F, SMe, NH, O, OMe], [AI3516; Me, H, F, H, O, H, H, F, CF 3, NH, O, OMe ], [AI 3517; Et, H, F, H, O, H, H, F, H, NH, O, OMe], [AI 3518; Et, H, F, H, O, H, H, F, F] , NH, O, OMe], [AI 3519; Et, H, F, H, O, H, H, H, F, Cl, NH, O, OMe], [AI 3520; Et, H, F, H, O, H , H, F, Br, NH, O, OMe], [AI 3521; Et, H, F, H, O, H, H, F, I, NH, O, OMe], [AI 3522; Et, H, F , H, O, H, H, F, Me, NH, O, OMe], [AI 3523; Et, H, F, H, O, H, F, Et, NH, O, OMe], [AI 3524] Et, H, F, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3525; Et, H, F, H, O, H, H, F, OMe, NH , O, OMe], [AI 3526; Et, H, F, H, O, H, H, F, OEt, NH, O, OMe], [AI 3527; Et, H, F, H, O, H, H, F, SMe, NH, O, OMe], [AI 3528; Et, H, F, H, O, H, H, F, CF ₃ , NH, O, OMe], [AI 3529; H, H, Cl, H, O, H, H, F, H, NH, O, OMe], [AI 3530; H, H, Cl, H, O, H, H, F, F, NH, O, OMe], [AI3531; H, H, Cl, H, O, H, H, F, Cl, NH, O, OMe], [AI 3532; H, H, Cl, H, O, H, H, F, Br, NH, O, OMe], [AI 3533; H, H, Cl, H, O, H, F, I, NH, O, OMe], [AI 3534; H, H, Cl, H, O, H, H, F, Me, NH, O, OMe], [AI 3535; H, H, Cl, H, O, H, H, F, Et, NH, O, OMe], [AI 3536; H, H, Cl, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3537; H, H, Cl, H, O, H, H, F, OMe, NH, O, OMe], [AI 3538; H, H, Cl, H, O, H, H, F, OEt, NH, O, OMe], [AI 3539; H, H, Cl, H, O, H, H, F, SMe, NH, O, OMe], [AI3540; H, H, Cl, H, O, H, H, F, CF 3, NH, O, OMe], [AI3541; Cl , H, Cl, H, O, H, H, F, H, NH, O, OMe], [AI 3542; Cl, H, Cl, H, O, H, H, F, F, NH, O, OMe ], [AI 3543; Cl, H, Cl, H, O, H, H, F, Cl, NH, O, OMe], [AI 3544; Cl, H, Cl, H, O, H, H, F, Br] , NH, O, OMe], [AI 3545; Cl, H, Cl, H, O, H, H, F, I, NH, O, OMe], [AI 3546; Cl, H, Cl, H, O, H , H, F, Me, NH, O, OMe], [AI 3547; Cl, H, Cl, H, O, H, H, F, Et, NH, O, OMe], [AI 3548; Cl, H, Cl , H, O, H, H, F, c, Pr, NH, O, OMe], [AI 3549; Cl, H, Cl, H, O, H, F, OM, NH, O, OMe], [AI 3550; Cl, H, Cl, H, O, H, H, F, OEt, NH, O, OMe], [AI 3551; Cl, H, Cl, H, O, H, H, F, SMe, NH , O, OMe], [AI 3552; Cl, H, Cl, H, O, H, H, F, CF ₃ , NH, O, OMe], [AI 3553; Me, H, Cl, H, O, H, H, F, H, NH, O, OMe], [AI 3554; Me, H, Cl, H, O, H, H, F, F, NH, O, OMe], [AI 3 555; Me, H, Cl, H, O, H, H, F, Cl, NH, O, OMe], [AI 3 556; Me, H, Cl, H, O, H, H, F, Br, NH, O, OMe], [AI 3557; Me, H, Cl, H, O, H, F, I, NH, O, OMe], [ AI 3 558; Me, H, Cl, H, O, H, H, F, Me, NH, O, OMe], [AI 3559; Me, H, Cl, H, O, H, H, F, Et, NH, O, OMe], [AI 3560; Me, H, Cl, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3561; Me, H, Cl, H, O, H, H, F, OMe, NH, O, OMe], [AI3562; Me, H, Cl, H, O, H, H, F, OEt, NH, O, OMe], [AI 3563; Me, H, Cl, H, O, H, H, F, SMe, NH, O, OMe], [AI 3564; Me, H, Cl, H, O, H, H, F, CF3, NH, O, OMe], [AI ₃ 565] Et, H, Cl, H, O, H, H, F, H, NH, O, OMe], [AI3566; Et, H, Cl, H, O, H, H, F, F, NH, O , OMe], [AI3567; Et, H, Cl, H, O, H, H, F, Cl, NH, O, OMe], [AI 3568; Et, H, Cl, H, O, H, H, F , Br, NH, O, OMe], [AI 3569; Et, H, Cl, H, O, H, H, F, I, NH, O, OMe], [AI 3 570; Et, H, Cl, H, O , H, H, F, Me, NH, O, OMe], [AI3571; Et, H, Cl, H, O, H, H, F, Et, NH, O, OMe], [AI3572; Et, H , Cl, H, O, H, H, F, c, Pr, NH, O, OMe], [AI 3573; Et, H, Cl, H, O, H, H, F, OMe, NH, O, OMe ], [AI 3574; Et, H, Cl, H, O, H, H, F, OEt, NH, O, OMe], [AI 3575; Et, H, Cl, H, O, H, H, F, SMe , NH, O, OMe], [AI3576; Et, H, Cl, H, O, H, H, F, CF 3, NH, O, OMe], [AI3577; H, H, Me, H, O, H, H, F, H, NH, O, OMe], [AI H, H, Me, H, O, H, H, F, F, NH, O, OMe], [AI 3579; H, H, Me, H, O, H, H, F, Cl, NH, O, OMe], [AI 3 580; H, H, Me, H, O, H, H, F, Br, NH, O, OMe], [AI 3581; H, H, Me, H, O, H, H, F, I, NH, O, OMe], [AI3582; H, H, Me, H, O, H, H, F, Me, NH, O, OMe], [AI 3583; H, H, Me, H, O, H, H, H, F, Et, NH, O, OMe], [AI 3584; H, H, Me, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3585; H, H, Me, H, O, H, H, F, OMe, NH, O, OMe], [AI 3586; H, H, Me, H, O, H, H, F, OEt, NH, O, OMe], [AI 3587; H, H, Me, H, O, H, H, F, SMe, NH, O, OMe], [AI 3588; H, H, Me, H, O, H, H, F, _{CF 3, NH, O, OMe} ], [AI3589; Cl, H, Me, H, O, H, H, F, H, NH, O, OMe], [AI3590; Cl, H, Me, H, O , H, H, F, F, NH, O, OMe], [AI3591; Cl, H, Me, H, O, H, H, F, Cl, NH, O, OMe], [AI3592; Cl, H , Me, H, O, H, H, F, Br, NH, O, OMe], [AI 3593; Cl, H, Me, H, O, H, H, F, I, NH, O, OMe], [AI3594; Cl, H, Me, H, O, H, H, F, Me, NH, O, OMe], [AI 3595; Cl, H, Me, H, O, H, H, F, Et, NH , O, OMe], [AI 3596; Cl, H, Me, H, O, H, H, F, c, Pr, NH, O, OMe], [AI 3597; Cl, H, Me, H, O, H , H, F, OMe, NH, O, OMe], [AI 3598; Cl, H, Me, H, O, H, H, F, OEt, NH, O, OMe], [AI 3599; Cl, H, Me , H, O, H, H , F, SMe, NH, O, OMe], [AI3600; Cl, H, Me, H, O, H, H, F, CF 3, NH, O, OMe],

[AI 3601; Me, H, Me, H, O, H, H, F, H, NH, O, OMe], [AI 3602; Me, H, Me, H, O, H, H, F, F, NH , O, OMe], [AI 3603; Me, H, Me, H, O, H, H, F, Cl, NH, O, OMe], [AI 3604; Me, H, Me, H, O, H, H , F, Br, NH, O, OMe], [AI 3605; Me, H, Me, H, O, H, H, F, I, NH, O, OMe], [AI 3606; Me, H, Me, H , O, H, H, F, Me, NH, O, OMe], [AI 3607; Me, H, Me, H, O, H, H, F, Et, NH, O, OMe], [AI 3608; Me , H, Me, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3609; Me, H, Me, H, O, H, H, F, OMe, NH, O , OMe], [AI 3610; Me, H, Me, H, O, H, H, F, OEt, NH, O, OMe], [AI 3611; Me, H, Me, H, O, H, H, F , SMe, NH, O, OMe], [AI 3612; Me, H, Me, H, O, H, H, F, CF ₃ , NH, O, OMe], [AI 3613; Et, H, Me, H, O, H, H, F, H, NH, O, OMe], [AI 3614; Et, H, Me, H, O, H, H, F, F, NH, O, OMe], [AI 3615; Et, H, Me, H, O, H, H, F, Cl, NH, O, OMe], [AI 3616; Et, H, Me, H, O, H, H, F, Br, NH, O, OMe] [AI 3617; Et, H, Me, H, O, H, H, F, I, NH, O, OMe], [AI 3618; Et, H, Me, H, O, H, H, F, Me, NH, O, OMe], [AI 3619; Et, H, Me, H, O, H, H, F, Et, NH, O, OMe], [AI 3620; Et, H, Me, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3621; Et, H, Me, H, O, H, H, F, OMe, NH, O, OMe], [AI 3622; Et, H, Me, H, O, H, H, F, OEt, NH, O, OMe], [AI 3623; Et, H, Me, H, O, H, F, S Me, NH, O, OMe], [ AI3624; Et, H, Me, H, O, H, H, F, CF 3, NH, O, OMe], [AI3625; H, H, Et, H, O, H, H, F, H, NH , O, OMe], [AI 3626; H, H, Et, H, O, H, H, F, F, NH, O, OMe], [AI 3627; H, H, Et, H, O, H, H, F, Cl, NH, O, OMe], [AI 3628; H, H, Et, H, O, H, H, F, Br, NH, O, OMe], [AI 3629; H, H, Et, H, O, H, H, F, I, NH, O, OMe] , [AI 3630; H, H, Et, H, O, H, H, F, Me, NH, O, OMe], [AI 3631; H, H, Et, H, O, H, H, F, Et, NH, O, OMe], [AI 3632; H, H, Et, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3633; H, H, Et, H, O, H, H, F, OMe, NH, O, OMe], [AI3634; H, H, Et, H, O, H, H, F, OEt, NH, O, OMe], [AI 3635; H, H, Et, H, O, H, H, F, SMe, NH, O, OMe], [AI3636; H, H, Et, H, O, H, H, F, CF 3, NH, O, OMe], [AI 3637; Cl, H, Et, H, O, H, H, F, H, NH, O, OMe], [AI 3638; Cl, H, Et, H, O, H, H, F, F, NH , O, OMe], [AI 3639; Cl, H, Et, H, O, H, H, F, Cl, NH, O, OMe], [AI 3640; Cl, H, Et, H, O, H, H , F, Br, NH, O, OMe], [AI3641; Cl, H, Et, H, O, H, H, F, I, NH, O, OMe], [AI3642; Cl, H, Et, H , O, H, H, F, Me, NH, O, OMe], [AI 3643; Cl, H, Et, H, O, H, H, F, Et, NH, O, OMe], [AI 3644; , H, Et, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3645; Cl, H, Et, H, O, H, H, F, OMe, NH, O , OMe], [AI3646; Cl, H, Et, H, O, H, H, F, OEt, NH, O, OMe], [AI 3647; Cl, H, Et, H, O, H, H, F , SMe, NH, O, OMe], [AI 3648; Cl, H, Et, H, O, H, H, F, CF ₃ , NH, O, OMe], [AI 3649; Me, H, Et, H, O, H, H, H, F, H, NH, O, OMe], [AI3650; Me, H, Et, H, O, H, H, F, F, NH, O, OMe], [AI3651; H, Et, H, O, H, H, F, Cl, NH, O, OMe], [AI 36 52; Me, H, Et, H, O, H, H, H, F, Br, NH, O, OMe], [AI3653; Me, H, Et, H, O, H, H, F, I, NH, O, OMe], [AI3654; Me, H, Et, H, O, H, H, F, Me, NH, O, OMe], [AI 3655; Me, H, Et, H, O, H, H, F, Et, NH, O, OMe], [AI 3656; Me, H, Et, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3657; Me, H, Et, H, O, H, H, F, OMe, NH, O, OMe], [AI 3658; Me, H, Et, H, O, H, F, OEt, NH, O, OMe], [AI 3659; Me, H, Et, H, O, H, H, F, SMe, NH, O, OMe], [AI 3660; Me, H, Et, H, O, H, H, F, CF ₃ , NH, O , OMe], [AI3661; Et, H, Et, H, O, H, H, F, H, NH, O, OMe], [AI3662; Et, H, Et, H, O, H, H, F , F, NH, O, OMe], [AI3663; Et, H, Et, H, O, H, H, H, F, Cl, NH, O, OMe], [AI3664; Et, H, Et, H, O , H, H, F, Br, NH, O, OMe], [AI 3 665; Et, H, Et, H, O, H, H, F, I, NH, O, OMe], [AI 3 666; Et, H , Et, H, O, H, H, F, Me, NH, O, OMe], [AI3667; Et, H, Et, H, O, H, H, F, Et, NH, O, OMe], [AI3668; Et, H, Et, H, O, H, H, F, c-Pr, NH, O, OMe], [AI 3669; Et, H, Et, H, O, H, H, F, OMe , NH, O, OMe], [AI3670; Et, H, Et, H, O, H, H, F, OEt, NH, O, OMe], [AI 3671; Et, H, Et, H, O, H , H, F, SMe, NH , O, OMe], [AI3672; Et, H, Et, H, O, H, H, F, CF 3, NH, O, OMe], [AI3673; H, H, H, H, O, H, H, H, H, H, NH, S, OMe], [AI 3674; H, H, H, H, O, H, H, F, NH, S, OMe], [ AI 3 675; H, H, H, H, H, O, H, H, H, Cl, NH, S, OMe], [AI 3 676; S, OMe], [AI 3677; H, H, H, H, O, H, H, H, I, NH , S, OMe], [AI3678; H, H, H, H, O, H, H, H, Me, NH, S, OMe], [AI 3679; H, H, H, H, O, H, H , H, Et, NH, S, OMe], [AI 3 680; H, H, H, H, H, O, H, H, c, Pr, NH, S, OMe], [AI 3681; H, H, H , H, O, H, H, H, H, OMe, NH, S, OMe], [AI 3682; H, H, H, H, H, O, H, H, OEt, NH, S, OMe], [AI 3683 H, H, H, H, H, O, H, H, H, SMe, NH, S, OMe], [AI 3684; H, H, H, H, H, O, H, H, H, CF ₃ , NH, S, OMe], [AI3685; Cl, H, H, H, O, H, H, H, H, NH, S, OMe], [AI 3686; Cl, H, H, H, O, H, H, H, F, NH, S, OMe], [AI 3687; Cl, H, H, H, H, O, H, H, H, H, Cl, NH, S, OMe], [AI 3688; Cl, H, H, H, O, H, H, H, H, Br, NH, S, OMe], [AI 3689; Cl, H, H, H, H, O, H, H, H, I, NH, S, OMe], [AI 3 690; H, H, H, H, O, H, H, H, Me, NH, S, OMe], [AI 3691; Cl, H, H, H, H, O, H, H, Et, NH, S, OMe] [AI 3692; Cl, H, H, H, H, O, H, H, H, c-Pr, NH, S, OMe], [AI 3693; Cl, H, H, H, O, H, H, H, H, OMe, NH, S, OMe], [AI 3694; Cl, H, H, H, H, O, H, H, H, H, OEt, NH, S, OMe], [AI 3 695; Cl, H, H, H, O, H, H, H, SMe, NH, S, OMe], [AI3696; Cl, H, H, H, O, H, H, H, CF 3, NH, S, OMe], [AI3697; Me, H , H, H, O, H, H, H, H, NH, S, OMe], [AI 3698; Me, H, H, H, O, H, H, F, NH, S, OMe], [AI 3699; Me, H, H, H, H, O, H, H, H, Cl, NH, S, OMe], [AI 3700; Me, H, H, H, O, H, H, H, Br, NH , S, OMe],

[AI 3701; Me, H, H, H, H, O, H, H, I, NH, S, OMe], [AI 3702; Me, H, H, H, O, H, H, H, Me, NH , S, OMe], [AI 3703; Me, H, H, H, H, O, H, H, H, Et, NH, S, OMe], [AI 3704; Me, H, H, H, O, H, H , H, c-Pr, NH, S, OMe], [AI 3705; Me, H, H, H, H, O, H, H, H, OMe, NH, S, OMe], [AI 3706; Me, H, H , H, O, H, H, H, OEt, NH, S, OMe], [AI3707; Me, H, H, H, O, H, H, SMe, NH, S, OMe], [AI 3708 ; Me, H, H, H , O, H, H, H, CF 3, NH, S, OMe], [AI3709; Et, H, H, H, O, H, H, H, H, NH, S, OMe], [AI 3710; Et, H, H, H, O, H, H, H, H, F, NH, S, OMe], [AI 3711; Et, H, H, H, O, H, H, H, Cl, NH, S, OMe], [AI 3712; Et, H, H, H, H, O, H, H, H, H, Br, NH, S, OMe], [AI 3713; Et, H, H, H, O, H, H, H, I, NH, S, OMe], [AI 3714; Et, H, H, H, H, O, H, H, Me, NH, S, OMe], [AI 3715; Et, H, H, H, H, O, H, H, H, Et, NH, S, OMe], [AI 3716; Et, H, H, H, H, O, H, H, c, Pr, NH, S, OMe], [AI3717; Et, H, H, H, O, H, H, H, OMe, NH, S, OMe], [AI 3718; Et, H, H, H, O, H, H, H, H, OEt, NH, S, OMe], [AI 3719; Et, H, H, H, H, O, H, H, H, SMe, NH, S, OMe], [AI 3720; Et, H, H, H, O, _{H, H, H, CF 3} , NH, S, OMe], [AI3721; H, H, F, H, O, H, H, H, H, NH, S, OMe], [AI3722; H, H , F, H, O, H, H, H, F, NH, S, OMe], [AI 3723; H, H, F, H, O, H, H, H, Cl, NH, S, OMe], [AI 3724; H, H, F, H, O, H, H, H, Br, NH, S, OMe], [AI 3725; H, H, F, H, O, H, H, H, I, NH , S, OMe], [AI3726; H, H, F, H, O, H, H, H, Me, NH, S, OMe], [AI 3727; H , H, F, H, O, H, H, H, Et, NH, S, OMe], [AI 3728; H, H, F, H, O, H, H, H, c-Pr, NH, S , OMe], [AI3729; H, H, F, H, O, H, H, H, OMe, NH, S, OMe], [AI 3730; H, H, F, H, O, H, H, H , OEt, NH, S, OMe], [AI3731; H, H, F, H, O, H, H, H, SMe, NH, S, OMe], [AI 3732; H, H, F, H, O , H, H, H, CF 3, NH, S, OMe], [AI3733; Cl, H, F, H, O, H, H, H, H, NH, S, OMe], [AI3734; Cl, H, F, H, O, H, H, H, F, NH, S, OMe], [AI 3735; Cl, H, F, H, O, H, H, H, Cl, NH, S, OMe] [AI 3 736; Cl, H, F, H, O, H, H, H, Br, NH, S, OMe], [AI 3 737; Cl, H, F, H, O, H, H, H, I, NH, S, OMe], [AI3738; Cl, H, F, H, O, H, H, H, Me, NH, S, OMe], [AI 3739; Cl, H, F, H, O, H, H, H, Et, NH, S, OMe], [AI 3740; Cl, H, F, H, O, H, H, H, c-Pr, NH, S, OMe], [AI 3741; Cl, H, F, H, O, H, H, H, OMe, NH, S, OMe], [AI 3742; Cl, H, F, H, O, H, H, H, OEt, NH, S, OMe], [ AI 3743; Cl, H, F, H, O, H, H, S Me, NH, S, OMe], [AI 3 744; Cl, H, F, H, O, H, H, H, CF ₃ , NH , S, OMe], [AI 3745; Me, H, F, H, O, H, H, H, H, NH, S, OMe], [AI 3746; Me, H, F, H, O, H, H , H, F, NH, S, OMe], [AI 3747; Me, H, F, H, O, H, H, H, Cl, NH, S, OMe], [AI 3 748; Me, H, F, H , O, H, H, H, Br, NH, S, OMe], [AI 3749; Me, H, F, H, O, H, H, H, I, NH, S, OMe], [AI 3 750; Me , H, F, H, O, H, H, H, Me, NH, S, OMe], [AI 3751; Me, H, F, H, O, H, H, Et, NH, S, OMe ], [AI3752; Me, H, F, H, O, H, H, H, c-Pr, NH, S, OMe], [AI3753; Me, H, F, H, O, H, H, H, H, OMe, NH, S, OMe], [AI 3754; Me, H, F, H, O, H, H, H, OEt, NH, S, OMe], [AI 3755; Me, H, F, H, O, H, H, H, SMe, NH, S, OMe], [AI3756; Me, H, F, H, O, H, H, H, CF 3, NH, S , OMe], [AI 3757; Et, H, F, H, O, H, H, H, H, NH, S, OMe], [AI 3758; Et, H, F, H, O, H, H, H , F, NH, S, OMe], [AI 3759; Et, H, F, H, O, H, H, H, H, Cl, NH, S, OMe], [AI 3760; Et, H, F, H, O , H, H, H, Br, NH, S, OMe], [AI3761; Et, H, F, H, O, H, H, H, I, NH, S, OMe], [AI3762; Et, H , F, H, O, H, H, H, Me, NH, S, OMe], [AI3763; Et, H, F, H, O, H, H, Et, NH, S, OMe], [AI 3764; Et, H, F, H, O, H, H, H, c-Pr, NH, S, OMe], [AI 3765; Et, H, F, H, O, H, H, H, H, OMe , NH, S, OMe], [AI3766; Et, H, F, H, O, H, H, H, H, OEt, NH, S, OMe], [AI 3767; Et, H, F, H, O, H , H, H, SMe, NH , S, OMe], [AI3768; Et, H, F, H, O, H, H, H, CF 3, NH, S, OMe], [AI3769; H, H, Cl, H, O, H, H, H, H, H, NH, S, OMe], [AI 3 770; H, H, Cl, H, O, H, H, F, NH, S, OMe], [ AI 3772; H, H, Cl, H, O, H, H, H, Cl, NH, S, OMe], [AI 3772; H, H, Cl, H, O, H, H, H, Br, NH, S, OMe], [AI3773; H, H, Cl, H, O, H, H, H, I, NH, S, OMe], [AI 3774; H, H, Cl, H, O, H, H, H, Me, NH, S, OMe], [AI 3775; H, H, Cl, H, O, H, H, H, H, Et, NH, S, OMe], [AI 3776; H, H, Cl, H, O, H, H, H, H, c-Pr, NH, S, OMe], [AI 3777; H, H, Cl, H, O, H, H, H, OMe, NH, S, OMe], [AI 3778; H, H, Cl, H, O, H, H, H, OEt, NH, S, OMe], [AI 3779; H, H, Cl, H, O, H, H, H, SMe, NH, S, OMe], [AI3780; H, H, Cl, H, O, H, H, H, CF 3, NH, S, OMe], [AI3781 Cl, H, Cl, H, O, H, H, H, H, H, NH, S, OMe], [AI 3782; Cl, H, Cl, H, O, H, H, H, F, NH, S , OMe], [AI 3783; Cl, H, Cl, H, O, H, H, H, Cl, NH, S, OMe], [AI 3784; Cl, H, Cl, H, O, H, H, H , Br, NH, S, OMe], [AI3785; Cl, H, Cl, H, O, H, H, H, I, NH, S, OMe], [AI 3786; Cl, H, Cl, H, O , H, H, H, Me, NH, S, OMe], [AI 3787; Cl, H, Cl, H, O, H, H, H, Et, NH, S, OMe], [AI 3788; Cl, H , Cl, H, O, H, H, H, c, Pr, NH, S, OMe], [AI 3789; Cl, H, Cl, H, O, H, H, H, OMe, NH, S, OMe ], [AI 3790; Cl, H, Cl, H, O, H, H, H, OEt, NH, S, OMe], [AI 3791; Cl, H, Cl, H, O, H, H, H, SMe , NH, S, OMe], [AI3792; Cl, H, Cl, H, O, H, H, H, CF 3, NH, S, OMe], [AI3793; Me, H, Cl, H, O, H, H, H, H, H, NH, S, OMe], [AI 3794; Me, H, Cl, H, O, H, H, H, F, NH, S, OMe], [AI 3795; Me, H, Cl, H, O, H, H, H, H, Cl, NH, S, OMe], [AI 3796; Me, H, Cl, H, O, H, H, Br, NH, S, OMe], [ AI 3 797; Me, H, Cl, H, O, H, H, I, NH, S, OMe], [AI 3798; Me, H, Cl, H, O, H, H, H, Me, NH, S, OMe], [AI3799; Me, H, Cl, H, O, H, H, H, Et, NH, S, OMe], [AI 3800; Me, H, Cl, H, O, H, H, H, c-Pr, NH, S, OMe],

[AI3801; Me, H, Cl, H, O, H, H, OMe, NH, S, OMe], [AI 3802; Me, H, Cl, H, O, H, H, H, OEt, NH , S, OMe], [AI 3803; Me, H, Cl, H, O, H, H, H, S Me, NH, S, OMe], [AI 3804; Me, H, Cl, H, O, H, H , H, CF3, NH, S, OMe], [AI ₃ 805; Et, H, Cl, H, O, H, H, H, H, NH, S, OMe], [AI 3 806; Et, H, Cl, H, O, H, H, H, H, F, NH, S, OMe], [AI 3807; Et, H, Cl, H, O, H, H, Cl, NH, S, OMe], [AI 3 808; Et, H, Cl, H, O, H, H, H, H, Br, NH, S, OMe], [AI 3809; Et, H, Cl, H, O, H, H, H, I, NH, S, OMe], [AI 3810; Et, H, Cl, H, O, H, H, H, Me, NH, S, OMe], [AI 3811; Et, H, Cl, H, O, H, H, H, H, Et, NH, S, OMe], [AI 3812; Et, H, Cl, H, O, H, H, H, c, Pr, NH, S, OMe], [AI 3813; Et, H, Cl, H, O, H, H, H, H, OMe, NH, S, OMe], [AI 3814; Et, H, Cl, H, O, H, H, H, OEt, NH, S, OMe], [AI 3815; Et, H, Cl, H, O, H, H, H, SMe, NH, S, OMe], [AI3816; Et, H, Cl, H, O, H, H, H, CF 3, NH, S, OMe H, H, Me, H, O, H, H, H, H, NH, S, OMe], [AI 3818; H, H, Me, H, O, H, H, H, F] , NH, S, OMe], [AI 3819; H, H, Me, H, O, H, H, H, Cl, NH, S, OMe], [AI 3820; H, H, Me, H, O, H , H, H, Br, NH, S, OMe], [AI 3821; H, H, Me, H, O, H, H, I, NH, S, OMe], [AI 3822; H, H, Me , H, O, H, H, H, Me, NH, S, OMe], [AI 3823; H, H, Me, H, O, H, H, Et, NH, S, OMe], [AI 3824 H, H, Me, H, O, H, H, H, c, Pr, NH, S, OMe], [AI 3825; H, H, Me, H, O, H, H, H, OMe, NH , S, OMe], [AI 3826; H, H, Me, H, O, H, H, H, OEt, NH, S, OMe], [AI3827; H, H, Me, H, O, H, H, H, SMe, NH, S, OMe], [AI3828; H, H, Me, H, O, H, H, H, CF 3, NH, S, OMe], [AI3829; Cl, H, Me, H, O, H, H, H, H, NH, S, OMe], [AI3830; Cl , H, Me, H, O, H, H, H, F, NH, S, OMe], [AI3831; Cl, H, Me, H, O, H, H, H, Cl, NH, S, OMe Cl, H, Me, H, O, H, H, H, Br, NH, S, OMe], [AI 3833; Cl, H, Me, H, O, H, H, H, I] , NH, S, OMe], [AI 3834; Cl, H, Me, H, O, H, H, H, Me, NH, S, OMe], [AI 3835; Cl, H, Me, H, O, H , H, H, Et, NH, S, OMe], [AI 3836; Cl, H, Me, H, O, H, H, c, Pr, NH, S, OMe], [AI 3837; Cl, H , Me, H, O, H, H, H, OMe, NH, S, OMe], [AI 3838; Cl, H, Me, H, O, H, H, H, OEt, NH, S, OMe], [AI 3839; Cl, H, Me, H, O, H, H, S Me, NH, S, OMe], [AI 3840; Cl, H, Me, H, O, H, H, H, CF ₃ , NH, S, OMe], [AI3841; Me, H, Me, H, O, H, H, H, H, NH, S, OMe], [AI3842; Me, H, Me, H, O, H, H, H, F, NH, S, OMe], [AI3843; Me, H, Me, H, O, H, H, H, Cl, NH, S, OMe], [AI 3484; Me, H, Me, H, O, H, H, H, H, Br, NH, S, OMe], [AI 3845; Me, H, Me, H, O, H, H, H, I, NH, S, OMe], [AI 3846; Me, H, Me, H, O, H, H, H, Me, NH, S, OMe], [AI 3847; Me, H, Me, H, O, H, H, H, Et, NH, S, OMe], [AI3848; Me, H, Me, H, O, H, H, H, c-Pr, NH, S, OMe], [AI 3849; Me, H, Me, H, O, H, H, H, OMe, NH, S, OMe], [AI 3850; Me, H, Me, H, O, H, H, H, OEt, NH, S, OMe], [AI 3851; Me, H, Me, H, O, H, H, H, SMe, NH, S, OMe], [AI3852; Me, H, Me , H, O, H, H, H, CF 3, NH, S, OMe], [AI3853; Et, H, Me, H, O, H, H, H, H, NH, S, OMe], [AI 3854; Et, H, Me, H, O, H, H, H, F, NH, S, OMe], [AI 3855; Et, H, Me, H, O, H, H, H, Cl, NH, S, OMe], [AI3856; Et, H, Me, H, O, H, H, H, Br, NH, S, OMe], [AI 3857; Et, H, Me, H, O, H, H, H, I, I, NH, S, OMe], [AI 3858; Et, H, Me, H, O, H, H, Me, NH, S, OMe], [AI 3859; Et, H, Me, H, O, H, H, H, H, Et, NH, S, OMe], [AI 3860; Et, H, Me, H, O, H, H, H, c-Pr, NH, S, OMe], [AI3861; Et, H, Me, H, O, H, H, H, OMe, NH, S, OMe], [AI3862; Et, H, Me, H, O, H, H, H, H, OEt, NH, S, OMe], [AI3863; Et, H, Me, H, O, H, H, H, SMe, NH, S, OMe], [AI3864; Et, H, Me, H, O, H, H, H, CF 3, NH, S, OMe], [AI3865; H, H, Et, H, O, H, H, H, H, NH, S, OMe], [AI3866; H , H, Et, H, O, H, H, H, F, NH, S, OMe], [AI3867; H, H, Et, H, O, H, H, H, Cl, NH, S, OMe H, H, Et, H, O, H, H, H, Br, NH, S, OMe], [AI 3869; H, H, Et, H, O, H, H, H, I] , NH, S, OMe], [AI3870; H, H, Et, H, O, H, H, H, Me, NH, S, OMe], [AI 3871; H, H, Et, H, O, H , H, H, Et, NH, S, OMe], [AI 3872; H, H, Et, H, O, H, H, c, Pr, NH, S, OMe], [AI 3873; H, H , Et, H, O, H, H, H, OMe, NH, S, OMe], [AI 3874; H, H, Et, H, O, H, H, H, OEt, NH, S, OMe], [AI3875; H, H, Et, H, O, H, H, SMe, NH, S, OMe], [AI 3876; H, H, Et, H, O, H, H, H, CF ₃ , NH, S, OMe], [AI 3877; Cl, H, Et, H, O, H, H, H, H, NH, S, OMe], [AI3878; Cl, H, Et, H, O, H, H, H, H, F, NH, S, OMe], [AI 3879; Cl, H, Et, H, O, H, H, H, H, Cl, NH, S, OMe], [AI 3 880; Cl, H, Et, H, O, H, H, H, Br, NH, S, OMe], [AI 3881; Cl, H, Et, H, O, H, H, H, I, NH, S, OMe], [AI3882; Cl, H, Et, H, O, H, H, Me, NH, S, OMe] [AI 3883; Cl, H, Et, H, O, H, H, H, Et, NH, S, OMe], [AI 3884; Cl, H, Et, H, O, H, H, H, c- Pr, NH, S, OMe], [AI 3885; Cl, H, Et, H, O, H, H, H, H, OMe, NH, S, OMe], [AI 3886; Cl, H, Et, H, O, H, H, H, H, OEt, NH, S, OMe], [AI 3887; Cl, H, Et, H, O, H, H, H, SMe, NH, S, OMe], [AI 3 888; Cl, H, Et, H, O, H, H, H, CF 3, NH, S, OMe], [AI3889; Me, H, Et, H, O, H, H, H, H, NH, S, OMe], [AI 3 890; Me, H, Et, H, O, H, H, H, F, NH, S, OMe], [AI 3891; Me, H, Et, H, O, H, H, H, Cl, NH S, OMe], [AI3892; Me, H, Et, H, O, H, H, H, Br, NH, S, OMe], [AI 3893; Me, H, Et, H, O, H, H , H, I, NH, S, OMe], [AI 3894; Me, H, Et, H, O, H, H, H, Me, NH, S, OMe], [AI 3895; Me, H, Et, H , O, H, H, H, H, Et, NH, S, OMe], [AI 3896; Me, H, Et, H, O, H, H, H, c-Pr, NH, S, OMe], [AI 3897 Me, H, Et, H, O, H, H, H, OMe, NH, S, OMe], [AI 3898; Me, H, Et, H, O, H, H, H, OEt, NH, S , OMe], [AI3899; Me, H, Et, H, O, H, H, H, SMe, NH, S, OMe], [AI 3900; Me, H, Et, H, O, H, H, H , CF ₃ , NH, S, OMe],

[AI3901; Et, H, Et, H, O, H, H, H, H, NH, S, OMe], [AI3902; Et, H, Et, H, O, H, H, H, F, NH , S, OMe], [AI 3903; Et, H, Et, H, O, H, H, H, Cl, NH, S, OMe], [AI 3904; Et, H, Et, H, O, H, H , H, Br, NH, S, OMe], [AI 3905; Et, H, Et, H, O, H, H, H, I, NH, S, OMe], [AI 3906; Et, H, Et, H , O, H, H, H, Me, NH, S, OMe], [AI3907; Et, H, Et, H, O, H, H, H, Et, NH, S, OMe], [AI 3908; Et , H, Et, H, O, H, H, H, c, Pr, NH, S, OMe], [AI 3909; Et, H, Et, H, O, H, H, H, OMe, NH, S , OMe], [AI3910; Et, H, Et, H, O, H, H, H, OEt, NH, S, OMe], [AI3911; Et, H, Et, H, O, H, H, H , SMe, NH, S, OMe ], [AI3912; Et, H, Et, H, O, H, H, H, CF 3, NH, S, OMe], [AI3913; H, H, H, H, O, H, H, H, H, H, O, O, NHMe], [AI3914; H, H, H, H, H, O, H, H, H, F, O, O, NHMe], [AI 3915; H, H, H, H, H, O, H, H, H, H, Cl, O, O, NHMe], [AI3916; H, H, H, H, H, O, H, H, Br, O, O, NHMe] [AI 3917; H, H, H, H, H, O, H, H, I, O, O, NHMe], [AI 3918; H, H, H, H, O, H, H, H, Me, O, O, NHMe], [AI3919; H, H, H, H, H, O, H, H, H, Et, O, O, NHMe], [AI3920; H, H, H, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 3921; H, H, H, H, H, O, H, H, H, OMe, O, O, NHMe], [AI 3922; H, H, H, H, O, H, H, H, OEt, O, O, NHMe], [AI 3923; H, H, H, H, H, O, H, H, SMe, O, O, NHMe], [ AI3924; H, H, H, H, O, H, H, H, CF 3, O, O, NHMe], [AI3925; F, H, H, H, O, H, H, H, H, O , O, NHMe], [AI 3926; F, H, H, H, O, H, H, H, F, O, O, NHMe], [AI 392 7; F, H, H, H, H, O, H, H, H, H, Cl, O, NHMe], [AI 3928; F, H, H, H, O, H, H, H, Br, O, O, NHMe], [AI3 929; F, H, H, H, O, H, H, H, I, O, O, NHMe], [AI 3930; F, H, H, H, O, H, H, H, Me, O, O, NHMe], [AI3931; F, H, H, H, H, O, H, H, H, H, Et, O, O, NHMe], [AI3932; F, H, H, H, O, H, H, H, H, c-Pr, O, O, NHMe], [AI 3933; F, H, H, H, H, O, H, H, H, OMe, O, O, NHMe], [AI 3934; F, H, H, H, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 3935; F, H, H, H, O, H, H, S, O, O, NHMe], [AI3936; F, H, H, H, O, H, H, H, CF 3, O, O, NHMe], [AI3937; Cl, H, H, H, O, H, H, H , H, O, O, NHMe], [AI 3938; Cl, H, H, H, H, O, H, H, H, F, O, O, NH Me], [AI 3939; Cl, H, H, H, O , H, H, H, Cl, O, O, NHMe], [AI 3940; Cl, H, H, H, H, O, H, H, H, Br, O, O, NHMe], [AI 3941; Cl, H , H, H, O, H, H, H, H, I, O, O, NHMe], [AI3942; Cl, H, H, H, O, H, H, H, Me, O, O, NHMe], [AI3943; Cl, H, H, H, H, O, H, H, H, Et, O, O, NHMe], [AI 3944; Cl, H, H, H, H, O, H, H, H, c-Pr , O, O, NHMe], [AI3945; Cl, H, H, H, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 3946; Cl, H, H, H, O, H , H, H, OEt, O, O, NHMe], [AI 3947; Cl, H, H, H, H, O, H, H, H, SMe, O, O, NHMe], [AI 3948; Cl, H, H , H, O, H, H , H, CF 3, O, O, NHMe], [AI3949; Br, H, H, H, O, H, H, H, H, O, O, NHMe], [ AI 3950; Br, H, H, H, H, O, H, H, H, F, O, O, NHMe], [AI 3951; Br, H, H, H, H, O, H, H, H, Cl, O, O, NHMe], [AI3952; Br, H, H, H, H, O, H, H, H, Br, O, O, NHMe], [AI 3953; Br, H, H, H, O , H, H, H, I, I, O, O, NHMe], [AI 3954; Br, H, H, H, H, O, H, H, H, Me, O, O, NHMe], [AI 3 955; Br, H , H, H, O, H, H, H, H, Et, O, O, NHMe], [AI 3956; Br, H, H, H, O, H, H, H, c-Pr, O, O, NHMe Br, H, H, H, H, O, H, H, H, OMe, O, O, NHMe], [AI 3958; Br, H, H, H, O, H, H, H, OEt] , O, O, NHMe], [AI3959; Br, H, H, H, H, O, H, H, H, SMe, O, O, NHMe], [AI 3 960; Br, H, H, H, O, H _{, H, H, CF 3,} O, O, NHMe], [AI3961; Me, H, H, H, O, H, H, H, H, O, O, NHMe], [AI3962; Me, H, H, H, O, H, H, H, H, F, O, O, NHMe], [AI3963; Me, H, H, H, O, H, H, H, Cl, O, O, NHMe], [ AI 3964; Me, H, H, H, H, O, H, H, H, Br, O, NH, NHMe], [AI 3 965; O, NHMe], [AI 3966; Me, H, H, H, O, H, H, H, Me, O, O, NHMe], [AI 3967; Me, H, H, H, O, H, H, H, Et, O, O, NHMe], [AI 3968; Me, H, H, H, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 3969; Me, H, H, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 3970; Me, H, H, H, H, O, H, H, H, OEt, O, O, NHMe], [AI 3971; Me, H, H, H, O, H, H, H, SMe, O, O, NHMe], [AI3972; Me, H, H, H, O, H, H, H, CF 3, O, O , NHMe], [AI 3 973; Et, H, H, H, H, O, H, H, H, H, O, O, NH Me], [AI 3 974; Et, H, H, H, O, H, H, H , F, O, O, NHMe], [AI3 975; Et, H, H, H, H, O, H, H, H, H, Cl, O, O, NHMe], [AI3976; Et, H, H, H, H, O , H, H, H, Br, O, O, NHMe], [AI 3977; Et, H, H, H, H, O, H, H, H, I, O, O, NHMe], [AI 3978; Et, H , H, H, O, H, H, H, Me, O, O, NHMe], [AI 3979; Et, H, H, H, O, H, H, H, Et, O, O, NH, Me: [AI 3 980; Et, H, H, H, H, O, H, H, H, c-Pr, O, O, NH Me], [AI 3981; Et, H, H, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 3982; Et, H, H, H, H, O, H, H, H, OEt, O, O, NHMe], [ AI 3983; Et, H, H, H, H, O, H, H, S Me, O, O, NH Me], [AI 3984; Et, H, H, H, H, O, H, H, H, CF ₃ , O , O, NHMe], [AI 3985; CF ₃ , H, H, H, H, O, H, H, H, H, O, O, NH Me], [AI 3986; CF ₃ , H, H, H, O, H , H, H, F, O , O, NHMe], [AI3987; CF 3, H, H, H, O, H, H, H, Cl, O, O, NHMe], [AI3988; CF 3, H , H, H, O, H , H, H, Br, O, O, NHMe], [AI3989; CF 3, H, H, H, O, H, H, H, I, O, O, NHMe] _{, [AI3990; CF 3, H} , H, H, O, H, H, H, Me, O, O, NHMe], [AI3991; CF 3, H, H, H, O, H, H, H, Et, O, O, NHMe] , [AI3992; CF 3, H, H, H, O, H, H, H, c-Pr, O, O, NHMe], [AI3993; CF 3, H, H, H, O, H, H, H, OMe, O, O, NHMe], [AI3994; CF 3, H, H, H, O, H, H, H, OEt, O, O, NHMe], [AI3995 CF ₃ , H, H, H, H, O, H, H, H, SMe, O, O, NHMe], [AI 3996; CF ₃ , H, H, H, O, H, H, H, CF ₃ , O, O, NHMe], [AI 3 997; H, H, F, H, O, H, H, H, H, O, O, NH Me], [AI 3998; H, H, F, H, O, H, H, H, F, O, O, NHMe], [AI 3 999; H, H, F, H, O, H, H, H, Cl, O, NH, Me], [AI 4000; H, H, F, H, O, H, H, H, H, Br, O, O, NHMe],

[AI 4001; H, H, F, H, O, H, H, I, O, O, NHMe], [AI 4002; H, H, F, H, O, H, H, H, Me, O H, H, F, H, O, H, H, H, Et, O, O, NHMe], [AI 4004; H, H, F, H, O, H, H , H, c-Pr, O, O, NHMe], [AI 4005; H, H, F, H, O, H, H, H, OMe, O, O, NHMe], [AI 4006; H, H, F , H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4007; H, H, F, H, O, H, H, H, SMe, O, O, NHMe], [AI 4008 ; H, H, F, H , O, H, H, H, CF 3, O, O, NHMe], [AI4009; F, H, F, H, O, H, H, H, H, O, O, NHMe], [AI 4010; F, H, F, H, O, H, H, H, F, O, O, NH Me], [AI 4011; F, H, F, H, O, H, H, H, Cl, O, O, NHMe], [AI 4012; F, H, F, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4013; F, H, F, H, O, H, H, H, H, I, O, O, NHMe], [AI 4014; F, H, F, H, O, H, H, H, Me, O, O, NHMe], [AI 4015; F, H, F, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4016; F, H, F, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4017; F, H, F, H, O, H, H, H, OMe, O, O, NH Me], [AI 4018; F, H, F, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4019; F, H, F, H, O, H, H, H, S Me, O, O, NHMe], [AI 4020; F, H, F, H, O, _{H, H, H, CF 3} , O, O, NHMe], [AI4021; Cl, H, F, H, O, H, H, H, H, O, O, NHMe], [AI4022; Cl, H , F, H, O, H, H, H, H, F, O, O, NHMe], [AI 4023; Cl, H, F, H, O, H, H, H, Cl, O, O, NHMe], [AI4024; Cl, H, F, H, O, H, H, H, Br, O, O, NHMe], [AI 4025; Cl, H, F, H, O, H, H, H, I, O , O, NHMe], [AI 4026; Cl, H, F, H, O, H, H, H, Me, O, O, NH Me], [AI 4027; Cl, H, F, H, O, H, H , H, Et, O, O, NHMe], [AI 4028; Cl, H, F, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4029; Cl, H, F, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4030; Cl, H, F, H, O, H, H, H, OEt, O, O, NHMe], [AI 4031; Cl, H, F, H, O, H, H, H, SMe, O, O, NHMe], [AI4032; Cl, H, F, H, O, H, H, H, CF 3, O, O , NHMe], [AI 4033; Br, H, F, H, O, H, H, H, H, O, O, NH Me], [AI 4034; Br, H, F, H, O, H, H, H , F, O, O, NHMe], [AI 4035; Br, H, F, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4036; Br, H, F, H, O , H, H, H, H, Br, O, O, NHMe], [AI 4037; Br, H, F, H, O, H, H, H, I, O, O, NHMe], [AI 4038; Br, H , F, H, O, H, H, H, Me, O, O, NHMe], [AI 4039; Br, H, F, H, O, H, H, H, Et, O, O, NHMe], [AI 4040; Br, H, F, H, O, H, H, c, Pr, O, O, NHMe], [AI 4041; Br, H, F, H, O, H, H, H, H, OMe , O, O, NHMe], [AI4042; Br, H, F, H, O, H, H, H, H, OEt, O, O, NHMe], [AI4043; Br, H, F, H, O, H , H, H, SMe, O , O, NHMe], [AI4044; Br, H, F, H, O, H, H, H, CF 3, O, O, NHMe], [AI4045; Me, H, F, H, O, H, H, H, H, H, O, O, NHMe], [AI 4046; Me, H, F, H, O, H, H, F, O, O, NHMe], [ AI 4047; Me, H, F, H, O, H, H, H, Cl, O, NHMe], [AI 4048; Me, H, F, H, O, H, H, H, Br, O, O, NHMe], [AI 4049; Me, H, F, H, O, H, H, H, I, O, O, NH Me], [AI 4050; Me, H, F, H, O, H, H, H, Me, O, O, NHMe], [AI4051; Me, H, F, H, O, H, H, H, H, Et, O, O, NHMe], [AI4052; Me, H, F, H, O, H, H, H, c, -Pr, O, O, NHMe], [AI 4053; Me, H, F, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4054; Me, H, F, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4055; Me, H, F, H, O, H, H, H, SMe, O, O, NHMe], [AI4056; Me, H, F, H, O, H, H, H, CF 3, O, O, NHMe], [AI4057; Et , H, F, H, O, H, H, H, H, H, O, O, NHMe], [AI 4058; Et, H, F, H, O, H, H, H, F, O, O, NHMe ], [AI 4059; Et, H, F, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4060; Et, H, F, H, O, H, H, H, Br] , O, O, NHMe], [AI4061; Et, H, F, H, O, H, H, H, I, O, O, NHMe], [AI4062; Et, H, F, H, O, H , H, H, Me, O, O, NHMe], [AI4063; Et, H, F, H, O, H, H, H, Et, O, O, NHMe], [AI 4064; Et, H, F , H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4065; Et, H, F, H, O, H, H, H, OMe, O, O, NHMe], [AI 4066; Et, H, F, H, O, H, H, OEt, O, O, NHMe], [AI 4067; Et, H, F, H, O, H, H, H, SMe, O , O, NHMe], [AI4068 ; Et, H, F, H, O, H, H, H, CF 3, O, O, NHMe], [AI4069; CF 3, H, F, H, O, H , H, H, H, O , O, NHMe], [AI4070; CF 3, H, F, H, O, H, H, H, F, O, O, NHMe], [AI4071; CF 3, H , F, H, O, H , H, H, Cl, O, O, NHMe], [AI4072; CF 3, H, F, H, O, H, H, H, Br, O, O, NHMe] _{, [AI4073; CF 3, H} , F, H, O, H, H, H, I, O, O, NHMe], [AI4074; CF 3, H, F, H, O, H, H, H, Me, O, O, NHMe] , [AI4075; CF 3, H, F, H, O, H, H, H, Et, O, O, NHMe], [AI4076; CF 3, H, F, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4077; CF 3, H, F, H, O, H, H, H, OMe, O, O, NHMe], [AI4078 CF ₃ , H, F, H, O, H, H, H, OEt, O, O , NHMe], [AI4079; CF 3, H, F, H, O, H, H, H, SMe, O, O, NHMe], [AI4080; CF 3, H, F, H, O, H, H _{, H, CF 3, O,} O, NHMe], [AI4081; H, H, Cl, H, O, H, H, H, H, O, O, NHMe], [AI4082; H, H, Cl, H, O, H, H, H, H, F, O, O, NHMe], [AI4083; H, H, Cl, H, O, H, H, H, Cl, O, O, NHMe], [AI4084; H, H, Cl, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4085; H, H, Cl, H, O, H, H, H, I, O, O, NHMe], [AI 4086; H, H, Cl, H, O, H, H, Me, O, O, NH Me], [AI 4087; H, H, Cl, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4088; H, H, Cl, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4089; H, H, Cl, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4090; H, H, Cl, H, O, H, H, H, OEt, O, O, NHMe], [AI4091; H, H, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI4092; H, H, Cl, H, O, H, H, H, CF 3, O, O, NHMe F, H, Cl, H, O, H, H, H, H, O, O, NHMe], [AI 4094; F, H, Cl, H, O, H, H, H, F] , O, O, NHMe], [AI 4095; F, H, Cl, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4096; F, H, Cl, H, O, H , H, H, Br, O, O, NHMe], [AI 4097; F, H, Cl, H, O, H, H, H, I, O, O, NHMe], [AI 4098; F, H, Cl , H, O, H, H, H, H, Me, O, O, NHMe], [AI 4099; F, H, Cl, H, O, H, H, H, Et, O, O, NHMe], [AI 4100 F, H, Cl, H, O, H, H, H, c-Pr, O, O, NHMe],

[AI 4101; F, H, Cl, H, O, H, H, OMe, O, O, NHMe], [AI 4102; F, H, Cl, H, O, H, H, H, OEt, O , O, NHMe], [AI 4103; F, H, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI 4104; F, H, Cl, H, O, H, H _{, H, CF 3, O,} O, NHMe], [AI4105; Cl, H, Cl, H, O, H, H, H, H, O, O, NHMe], [AI4106; Cl, H, Cl, H, O, H, H, H, H, F, O, O, NHMe], [AI 4107; Cl, H, Cl, H, O, H, H, H, Cl, O, O, NHMe], [AI 4108; Cl, H, Cl, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4109; Cl, H, Cl, H, O, H, H, H, I, O, O, NHMe], [AI 4110; Cl, H, Cl, H, O, H, H, H, Me, O, O, NHMe], [AI 4111; Cl, H, Cl, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4112; Cl, H, Cl, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4113; Cl, H, Cl, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4114; Cl, H, Cl, H, O, H, H, H, OEt, O, O, NHMe], [AI 4 115; Cl, H, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI4116; Cl, H, Cl, H, O, H, H, H, CF 3, O, O, NHMe ], [AI 4117; Br, H, Cl, H, O, H, H, H, H, H, O, O, NHMe], [AI 4118; Br, H, Cl, H, O, H, H, H, F] , O, O, NHMe], [AI 4119; Br, H, Cl, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4120; Br, H, Cl, H, O, H , H, H, Br, O, O, NHMe], [AI 4121; Br, H, Cl, H, O, H, H, H, I, O, O, NHMe], [AI 4122; Br, H, Cl , H, O, H, H, H, H, Me, O, O, NHMe], [AI 4123; Br, H, Cl, H, O, H, H, H, Et, O, O, NHMe], [AI 4124 Br, H, Cl, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4125; Br, H, Cl, H, O, H, H, H, OMe, O , O, NHMe], [AI 4126; Br, H, Cl, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4127; Br, H, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI 4128; Br, H, Cl, H, O, H, H, H, CF 3, O, O, NHMe], [AI4129; Me, H, Cl, H, O, H, H, H, H, O, O, NHMe Me, H, Cl, H, O, H, H, H, F, O, O, NHMe], [AI 4131; Me, H, Cl, H, O, H, H, H, Cl, , O, O, NHMe], [AI 4132; Me, H, Cl, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4133; Me, H, Cl, H, O, H , H, H, I, O, O, NHMe], [AI 4 134; Me, H, Cl, H, O, H, H, H, Me, O, O, NHMe], [AI 4 135; Me, H, Cl , H, O, H, H, H, H, Et, O, O, NHMe], [AI 4136; Me, H, Cl, H, O, H, H, c, Pr, O, O, NHMe], [AI 4 137; Me, H, Cl, H, O, H, H, OMe, O, O, NHMe], [AI 4138; Me, H, Cl, H, O, H, H, H, OEt, O , O, NHMe], [AI 4139; Me, H, Cl, H, O, H, H, H, SMe, O, O, NH Me], [AI 4140; Me, H, Cl, H, O, H, H _{, H, CF 3, O,} O, NHMe], [AI4141; Et, H, Cl, H, O, H, H, H, H, O, O, NHMe], [AI4142; Et, H, Cl, H, O, H, H, H, H, F, O, O, NHMe], [AI 4143; Et, H, Cl, H, O, H, H, H, Cl, O, O, NHMe], [AI 4144; Et, H, Cl, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4145; Et, H, Cl, H, O, H, H, H, I, O, O, NHMe], [AI 4146; Et, H, Cl, H, O, H, H, H, Me, O, O, NHMe], [AI 4147; Et, H, Cl, H, O, H, H, H, H, Et, O, O, NHMe], [AI4148; Et, H, Cl, H, O, H, H, H, H, c-Pr, O, O, NHMe], [AI 4149; Et, H, Cl, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4150; Et, H, Cl, H, O, H, H, H, OEt, O, O, NHMe], [AI 4151; Et, H, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI4152; Et, H, Cl, H, O, H, H, H, CF 3, O, O, NHMe], [AI4153; CF 3, H, Cl, H, O, H, H, H, H, O, O, NHMe], [AI4154; CF 3, H, Cl, H, O, H, H, H, F, O, O, NHMe], [AI4155; CF 3, H, Cl, H, O, H, H, H, Cl, O, O, NHMe], [AI4156; CF 3, H, Cl, H, O, H, H, H, Br, O, O, NHMe], _{[AI4157; CF 3, H,} Cl, H, O, H, H, H, I, O, O, NHMe], [AI4158; CF 3, H, Cl, H, O, H, H, H, Me , O, O, NHMe], [AI4159; CF 3, H, Cl, H, O, H, H, H, Et, O, O, NHMe], [AI4160; CF 3, H, Cl, H, O , H, H, H, c -Pr, O, O, NHMe], [AI4161; CF 3, H, Cl, H, O, H, H, H, OMe, O, O, NHMe], [AI4162; _{CF 3, H, Cl, H} , O, H, H, H, OEt, O, O, NHMe], [AI4163; CF 3, H, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI4164; CF 3, H, Cl, H, O, H, H, H, CF 3, O, O, NHMe], [AI4165; H, H, Me, H, O, H, H, H, H, H, O, O, NHMe], [AI 4166; H, H, Me, H, O, H, H, H, F, O, O, NHMe], [AI 4 167; H, H, Me, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4168; H, H, Me, H, O, H, H, H, Br, O, O, NHMe], [AI 4169; H, H, Me, H, O, H, H, H, H, I, O, O, NHMe], [AI 4170; H, H, Me, H, O, H, H, Me, O, O, NHMe], [AI4171; H, H, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4172; H, H, Me, H, O, H, H, H, H, c-Pr, O, O, NHMe], [AI 4173; H, H, Me, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4174; H, H, Me, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4175; H, H, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI 4176; H, H, Me, H, O, H, _{H, H, CF 3, O} , O, NHMe], [AI4177; F, H, Me, H, O, H, H, H, H, O, O, NHMe], [AI4178; F, H, Me , H, O, H, H, H, H, F, O, O, NHMe], [AI 4179; F, H, Me, H, O, H, H, H, Cl, O, O, NHMe], [AI 4 180 F, H, Me, H, O, H, H, H, H, Br, O, O, NHMe], [AI4181; F, H, Me, H, O, H, H, H, I, O, O NH Me], [AI4182; F, H, Me, H, O, H, H, H, Me, O, O, NH Me], [AI 4183; F, H, Me, H, O, H, H, H , Et, O, O, NHMe], [AI 4184; F, H, Me, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4 185; F, H, Me, H , O, H, H, H, H, OMe, O, O, NHMe], [AI 4186; F, H, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI 4187; F , H, Me, H, O , H, H, H, SMe, O, O, NHMe], [AI4188; F, H, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI 4189; Cl, H, Me, H, O, H, H, H, H, H, O, O, NHMe], [AI 4190; Cl, H, Me, H, O, H, H, H, H, F, O, O, NHMe], [AI4191; Cl, H, Me, H, O, H, H, H, H, Cl, O, O, NHMe], [AI4192; Cl, H, Me, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4193; Cl, H, Me, H, O, H, H, H, I, O, O, NHMe], [AI 4194; Cl, H, Me, H, O, H, H, H, Me, O, O, NHMe], [AI 4195; Cl, H, Me, H, O, H, H, H, Et, O, O, NHMe], [ AI 4196; Cl, H, Me, H, O, H, H, c, Pr, O, O, NHMe], [AI 4197; Cl, H, Me, H, O, H, H, H, OMe, O, O, NHMe], [AI 4198; Cl, H, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI 4199; Cl, H, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI4200; Cl, H, Me, H, O, H, H, H, CF 3, O, O, NHMe],

[AI4201; Br, H, Me, H, O, H, H, H, H, O, O, NHMe], [AI 4202; Br, H, Me, H, O, H, H, H, F, O , O, NHMe], [AI 4203; Br, H, Me, H, O, H, H, H, H, Cl, O, NH, Me], [AI 4204; Br, H, Me, H, O, H, H , H, Br, O, O, NHMe], [AI 4205; Br, H, Me, H, O, H, H, H, I, O, O, NHMe], [AI 4206; Br, H, Me, H , O, H, H, H, H, Me, O, O, NHMe], [AI 4207; Br, H, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4208; Br , H, Me, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4209; Br, H, Me, H, O, H, H, H, OMe, O, O , NHMe], [AI 4210; Br, H, Me, H, O, H, H, H, OEt, O, O, NH Me], [AI 4211; Br, H, Me, H, O, H, H, H , SMe, O, O, NHMe ], [AI4212; Br, H, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI4213; Me, H, Me, H, O, H, H, H, H, H, O, O, NHMe], [AI 4214; Me, H, Me, H, O, H, H, H, F, O, O, NHMe], [AI 4215; Me, H, Me, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4216; Me, H, Me, H, O, H, H, H, Br, O, O, NHMe] [AI 4217; Me, H, Me, H, O, H, H, I, O, O, NHMe], [AI 4218; Me, H, Me, H, O, H, H, H, Me, O, O, NHMe], [AI 4219; Me, H, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4220; Me, H, Me, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4221; Me, H, Me, H, O, H, H, H, OMe, O, O, NHMe], [AI4222; Me, H, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI 4223; Me, H, Me, H, O, H, H, H, SMe, O, O, NHMe], [ AI4224; Me, H, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI4225; Et, H, Me, H, O, H, H, H, H, O , O, NHMe], [AI 4226; Et, H, Me, H, O, H, H, H, H, F, O, O, NHMe], [AI 4227; Et, H, Me, H, O, H, H, H, Cl, O, O, NHMe], [AI 4228; Et, H, Me, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4229; Et, H, Me, H, O, H, H, H, I, O, O, NHMe], [AI 4230; Et, H, Me, H, O, H, H, H, Me, O, O, NHMe], [AI 421; Et, H, Me, H, O, H, H, H, H, Et, O, O, NHMe], [AI4232; Et, H, Me, H, O, H, H, H, c, Pr, O, O, NHMe], [AI4233; Et, H, Me, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4234; Et, H, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI 4235; Et, H, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI4236; Et, H, Me, H, O, H, H, H, CF 3, O, O, NHMe _{], [AI4237; CF 3,} H, Me, H, O, H, H, H, H, O, O, NHMe], [AI4238; CF 3, H, Me, H, O, H, H, H , F, O, O, NHMe ], [AI4239; CF 3, H, Me, H, O, H, H, H, Cl, O, O, NHMe], [AI4240; CF 3, H, Me, H , O, H, H, H , Br, O, O, NHMe], [AI4241; CF 3, H, Me, H, O, H, H, H, I, O, O, NHMe], [AI4242; _{CF 3, H, Me, H} , O, H, H, H, Me, O, O, NHMe], [AI4243; CF 3, H, Me, H, O, H, H, H, Et, O, O, NHMe], [AI4244; CF 3, H, Me, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4245; CF 3, H, Me, H, O, H, H, H, OMe, O, O, NHMe], [AI4246; CF 3, H, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI4247; CF 3, H, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI4248; CF 3, H, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI 4249; H, H, Et, H, O, H, H, H, H, H, O, O, NHMe], [AI 4250; H, H, Et, H, O, H, H, H, H, F, O, O, NHMe ], [AI4251; H, H, Et, H, O, H, H, H, Cl, O, O, NHMe], [AI 4252; H, H, Et, H, O, H, H, H, Br] , O, O, NHMe], [AI4253; H, H, Et, H, O, H, H, H, I, O, O, NHMe], [AI 4254; H, H, Et, H, O, H , H, H, Me, O, O, NHMe], [AI 4 255; H, H, Et, H, O, H, H, H, Et, O, O, NHMe], [AI 4 256; H, H, Et , H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4 257; H, H, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI4258; H, H, Et, H, O, H, H, OEt, O, O, NHMe], [AI 4259; H, H, Et, H, O, H, H, H, SMe, O , O, NHMe], [AI4260 ; H, H, Et, H, O, H, H, H, CF 3, O, O, NHMe], [AI4261; F, H, Et, H, O, H, H, H, H, H, O, O, NHMe], [AI4262; F, H, Et, H, O, H, H, H, F, O, O, NHMe], [AI 4263; F, H, Et, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4264; F, H, Et, H, O, H, H, H, Br, O, O, NHMe], [AI 4265; F, H, Et, H, O, H, H, H, H, I, O, O, NHMe], [AI 4266; F, H, Et, H, O, H, H, H, Me, O, O, NHMe], [AI4267; F, H, Et, H, O, H, H, H, Et, O, O, NHMe], [AI 4268; F, H, Et, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4269; F, H, Et, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4270; F, H, Et, H, O, H, H, H, H, OEt, O, O, NHMe], [AI4271; F, H, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI4272; F, H, Et, H, O, H, H, H, CF 3, O, O, NHMe], [AI4273; Cl, H, Et, H, O, H, H, H, H, O, O, NHMe ], [AI 4274; Cl, H, Et, H, O, H, H, H, H, F, O, O, NHMe], [AI 4275; Cl, H, Et, H, O, H, H, H, Cl, , O, O, NHMe], [AI 4276; Cl, H, Et, H, O, H, H, H, Br, O, O, NH Me, [AI 4277; Cl, H, Et, H, O, H, H, H, I, O, O, NHMe], [AI 4 278; Cl, H, Et, H, O, H, H, H, Me, O, O, NHMe], [AI 4279; Cl, H, Et, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4280; Cl, H, Et, H, O, H, H, H, H, c-Pr, O, O, NHMe], [AI4281; Cl, H, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI4282; H, Et, H, O, H, H, H, H, OEt, O, O, NHMe], [AI4283; Cl, H, Et, H, O, H, H, H, SMe, O, O, NHMe] , [AI4284; Cl, H, Et, H, O, H, H, H, CF 3, O, O, NHMe], [AI4285; Br, H, Et, H, O, H, H, H, H , O, O, NHMe], [AI4286; Br, H, Et, H, O, H, H, H, H, F, O, O, NHMe], [AI 4287; Br, H, Et, H, O, H , H, H, Cl, O, O, NHMe], [AI 4288; Br, H, Et, H, O, H, H, H, Br, O, O, NHMe], [AI 4289; Br, H, Et , H, O, H, H, H, H, I, I, O, O, NHMe], [AI 4290; Br, H, Et, H, O, H, H, H, Me, O, O, NHMe], [AI4291 Br, H, Et, H, O, H, H, H, H, Et, O, O, NHMe], [AI4292; Br, H, Et, H, O, H, H, H, c-Pr, O , O, NHMe], [AI 4293; Br, H, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI 4294; Br, H, Et, H, O, H, H , H, OEt, O, O, NHMe], [AI 4295; Br, H, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI 4296; Br, H, Et, H , O, H, H, H , CF 3, O, O, NHMe], [AI4297; Me, H, Et, H, O, H, H, H, H, O, O, NHMe], [AI4298; Me, H, Et, H, O, H, H, H, H, F, O, O, NHMe], [AI 4299; Me, H, Et, H, O, H, H, H, Cl, O, O, NHMe], [AI 4300; Me, H, Et, H, O, H, H, H, Br, O, O, NHMe],

[AI 4301; Me, H, Et, H, O, H, H, H, I, O, O, NHMe], [AI 4302; Me, H, Et, H, O, H, H, H, Me, O , O, NHMe], [AI4303; Me, H, Et, H, O, H, H, H, Et, O, O, NHMe], [AI 4304; Me, H, Et, H, O, H, H , H, c-Pr, O, O, NHMe], [AI 4305; Me, H, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI 4306; Me, H, Et , H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4307; Me, H, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI 4308 ; Me, H, Et, H , O, H, H, H, CF 3, O, O, NHMe], [AI4309; Et, H, Et, H, O, H, H, H, H, O, O, NHMe], [AI 4310; Et, H, Et, H, O, H, H, H, H, F, O, O, NH Me], [AI 4311; Et, H, Et, H, O, H, H, H, Cl, O, O, NHMe], [AI 4312; Et, H, Et, H, O, H, H, H, H, H, Br, O, O, NH Me], [AI 4313; Et, H, Et, H, O, H, H, H, H, I, O, O, NHMe], [AI 4314; Et, H, Et, H, O, H, H, H, Me, O, O, NHMe], [AI 4315; Et, H, Et, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4316; Et, H, Et, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4317; Et, H, Et, H, O, H, H, H, OMe, O, O, NH Me], [AI 4318; Et, H, Et, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4319; Et, H, Et, H, O, H, H, H, H, SMe, O, O, NHMe], [AI 4320; Et, H, Et, H, O, _{H, H, H, CF 3} , O, O, NHMe], [AI4321; CF 3, H, Et, H, O, H, H, H, H, O, O, NHMe], [AI4322; CF 3 , H, Et, H, O , H, H, H, F, O, O, NHMe], [AI4323; CF 3, H, Et, H, O, H, H, H, Cl, O, O, _{NHMe], [AI4324; CF 3} , H, Et, H, O, H, H, H, Br, O, O, NHMe], [AI4325; CF 3, H, Et, H, O, H, H, H, I, O, O, NHMe], [ AI 4326; CF ₃ , H, Et, H, O, H, H, H, Me, O, O, NH Me], [AI 4327; CF ₃ , H, Et, H, O, H, H, H, Et, O, O, NHMe], [ AI4328; CF 3, H, Et, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4329; CF 3, H, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI4330; CF 3, H, Et, H, O, H, H, H, OEt, O, O, NHMe], [AI4331; CF _{3, H, Et, H,} O, H, H, H, SMe, O, O, NHMe], [AI4332; CF 3, H, Et, H, O, H, H, H, CF 3, O, O, NHMe], [AI4333; H, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4334; H, H, CF 3, H, O, H, H, H, F, O, O, NHMe], [AI4335; H, H, CF 3, H, O, H, H, H, Cl, O, O, NHMe], [AI4336; H, H, CF _{3, H, O, H,} H, H, Br, O, O, NHMe], [AI4337; H, H, CF 3, H, O, H, H, H, I, O, O, NHMe], [AI4338; H, H, CF 3, H, O, H, H, H, Me, O, O, NHMe], [AI4339; H, H, CF 3, H, O, H, H, H, Et , O, O, NHMe], [AI4340; H, H, CF 3, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4341; H, H, CF 3, H , O, H, H, H , OMe, O, O, NHMe], [AI4342; H, H, CF 3, H, O, H, H, H, OEt, O, O, NHMe], [AI4343; _{H, H, CF 3, H} , O, H, H, H, SMe, O, O, NHMe], [AI4344; H, H, CF 3, H, O, H, H, H, CF 3, O , O, NHMe], [AI4345 ; F, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4346; F, H, CF 3, H, O, H , H, H, F, O , O, NHMe], [AI4347; F, H, CF 3, H, O, H, H, H, Cl, O, O, NHMe], [AI4348; F, H, _{CF 3, H, O, H} , H, H, Br, O, O, NHMe], [AI4349; F, H, CF 3, H, O, H, H, H, I, O, O, NHMe] , [AI4350; F, H, CF 3, H, O, H, H, H, Me, O, O, NHMe], [AI4351; F, H, CF 3, H, O, H, H, H, Et , O, O, NHMe], [AI4352; F, H, CF 3, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4353; F, H, CF 3, H , O, H, H, H , OMe, O, O, NHMe], [AI4354; F, H, CF 3, H, O, H, H, H, OEt, O, O, NHMe], [AI4355; _{F, H, CF 3, H} , O, H, H, H, SMe, O, O, NHMe], [AI4356; F, H, CF 3, H, O, H, H, H, CF 3, O , O, NHMe], [AI4357 ; Cl, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4358; Cl, H, CF 3, H, O, H , H, H, F, O , O, NHMe], [AI4359; Cl, H, CF 3, H, O, H, H, H, Cl, O, O, NHMe], [AI4360; Cl, H, _{CF 3, H, O, H} , H, H, Br, O, O, NHMe], [AI4361; Cl, H, CF 3, H, O, H, H, H, I, O, O, NHMe] , [AI4362; Cl, H, CF 3, H, O, H, H, H, Me, O, O, NHMe], [AI4363; Cl, H, CF 3, H, O, H, H, H, Et, O, O, NHMe] , [AI4364; Cl, H, CF 3, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4365; Cl, H, CF 3, H, O, H, H, H, OMe, O, O, NHMe], [AI4366; Cl, H, CF 3, H, O, H, H, H, OEt, O, O, NHMe], [AI4367 _{; Cl, H, CF 3,} H, O, H, H, H, SMe, O, O, NHMe], [AI4368; Cl, H, CF 3, H, O, H, H, H, CF 3, O, O, NHMe], [ AI4369; Br, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4370; Br, H, CF 3, H, O, H, H, H, F, O, O, NHMe], [AI4371; Br, H, CF 3, H, O, H, H, H, Cl, O, O, NHMe], [AI4372; Br, H _{, CF 3, H, O,} H, H, H, Br, O, O, NHMe], [AI4373; Br, H, CF 3, H, O, H, H, H, I , O, O, NHMe], [AI4374; Br, H, CF 3, H, O, H, H, H, Me, O, O, NHMe], [AI4375; Br, H, CF 3, H, O , H, H, H, Et , O, O, NHMe], [AI4376; Br, H, CF 3, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4377; _{Br, H, CF 3, H} , O, H, H, H, OMe, O, O, NHMe], [AI4378; Br, H, CF 3, H, O, H, H, H, OEt, O, O, NHMe], [AI4379; Br, H, CF 3, H, O, H, H, H, SMe, O, O, NHMe], [AI4380; Br, H, CF 3, H, O, H, _{H, H, CF 3, O} , O, NHMe], [AI4381; Me, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4382; Me, H, _{CF 3, H, O, H} , H, H, F, O, O, NHMe], [AI4383; Me, H, CF 3, H, O, H, H, H, Cl, O, O, NHMe] , [AI4384; Me, H, CF 3, H, O, H, H, H, Br, O, O, NHMe], [AI4385; Me, H, CF 3, H, O, H, H, H, I, O, O, NHMe] , [AI4386; Me, H, CF 3, H, O, H, H, H, Me, O, O, NHMe], [AI4387; Me, H, CF 3, H, O, H, H, H, Et, O, O, NHMe], [AI4388; Me, H, CF 3, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4389 _{; Me, H, CF 3,} H, O, H, H, H, OMe, O, O, NHMe], [AI4390; Me, H, CF 3, H, O, H, H, H, OEt, O , O, NHMe], [AI 4391; Me, H, CF ₃ , H, O, H, H, H, S Me, O, O, NH Me], [AI 4392; Me, H, CF ₃ , H, O, H _{, H, H, CF 3,} O, O, NHMe], [AI4393; Et, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4394; Et, H , CF ₃ , H, O, H, H, H, H, F, O, NH, NH Me], [AI 4395; Et, H, CF ₃ , H, O, H, H, H, Cl, O, O, NH Me ], [AI4396; Et, H , CF 3, H, O, H, H, H, Br, O, O, NHMe], [AI4397; Et, H _{, CF 3, H, O,} H, H, H, I, O, O, NHMe], [AI4398; Et, H, CF 3, H, O, H, H, H, Me, O, O, NHMe ], [AI4399; Et, H , CF 3, H, O, H, H, H, Et, O, O, NHMe], [AI4400; Et, H, CF 3, H, O, H, H, H , c-Pr, O, O, NHMe],

[AI4401; Et, H, CF 3, H, O, H, H, H, OMe, O, O, NHMe], [AI4402; Et, H, CF 3, H, O, H, H, H, OEt , O, O, NHMe], [AI4403; Et, H, CF 3, H, O, H, H, H, SMe, O, O, NHMe], [AI4404; Et, H, CF 3, H, O , H, H, H, CF 3, O, O, NHMe], [AI4405; CF 3, H, CF 3, H, O, H, H, H, H, O, O, NHMe], [AI4406; _{CF 3, H, CF 3,} H, O, H, H, H, F, O, O, NHMe], [AI4407; CF 3, H, CF 3, H, O, H, H, H, Cl, O, O, NHMe], [ AI4408; CF 3, H, CF 3, H, O, H, H, H, Br, O, O, NHMe], [AI4409; CF 3, H, CF 3, H, O, H, H, H, I, O, O, NHMe], [AI4410; CF 3, H, CF 3, H, O, H, H, H, Me, O, O, NHMe], [AI4411; _{CF 3, H, CF 3,} H, O, H, H, H, Et, O, O, NHMe], [AI4412; CF 3, H, CF 3, H, O, H, H, H, c- Pr, O, O, NHMe] , [AI4413; CF 3, H, CF 3, H, O, H, H, H, OMe, O, O, NHMe], [AI4414; CF 3, H, CF 3, H, O, H, H, H, OEt, O, O, NHMe], [AI4415; CF 3, H, CF 3, H, O, H, H, H, SMe, O, O, NHMe], [ _{AI4416; CF 3, H, CF} 3, H, O, H, H, H, CF 3, O, O, NHMe], [AI4417; H, F, H, H, O, H, H, H, H , O, O, NHMe], [AI4418; H, F, H, H, O, H, H, H, H, F, O, O, NHMe], [AI 4419; H, F, H, H, O, H , H, H, Cl, O, O, NHMe], [AI 4420; H, F, H, H, O, H, H, H, Br, O, NH, Me], [AI 4421; H, F, H , H, O, H, H, H, H, I, I, O, O, NHMe], [AI4422; H, F, H, H, O, H, H, Me, O, O, NHMe], [AI 4423] H, F, H, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4424; H, F, H, H, O, H, H, H, c -Pr, O, O, NHMe], [AI 4425; H, F, H, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4426; H, F, H, H, O , H, H, H, OEt, O, O, NHMe], [AI 4427; H, F, H, H, O, H, H, H, SMe, O, O, NHMe], [AI 4428; H, F , H, H, O, H , H, H, CF 3, O, O, NHMe], [AI4429; Cl, F, H, H, O, H, H, H, H, O, O, NHMe] , [AI4430; Cl, F, H, H, O, H, H, H, F, O, O, NHMe], [AI 443 1; Cl, F, H, H, O, H, H, H, Cl, O, O, NHMe], [AI4432; Cl, F, H, H, O, H, H, H, H, Br, O, O, NHMe], [AI4433; Cl, F, H, H, O, H, H, H, I, O, O, NHMe], [AI 4434; Cl, F, H, H, O, H, H, H, Me, O, O, NHMe], [AI 4435; Cl, F, H, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4436; Cl, F, H, H, O, H, H, H, c-Pr, O, O, NHMe], [ AI 4437; Cl, F, H, H, O, H, H, H, OMe, O, O, NHMe], [AI 4438; Cl, F, H, H, O, H, H, H, OEt, O, O, NHMe], [AI4439; Cl, F, H, H, O, H, H, H, SMe, O, O, NHMe], [AI 4440; Cl, F, H, H, O, H, H, _{H, CF 3, O, O} , NHMe], [AI4441; Me, F, H, H, O, H, H, H, H, O, O, NHMe], [AI4442; Me, F, H, H , O, H, H, H, H, F, O, O, NHMe], [AI4443; Me, F, H, H, O, H, H, H, Cl, O, O, NHMe], [AI4444; , F, H, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4445; Me, F, H, H, O, H, H, H, I, O, O, NHMe ], [AI 4446; Me, F, H, H, O, H, H, H, Me, O, O, NH, Me], [AI 4 447; Me, F, H, H, O, H, H, H, Et, , O, O, NHMe], [AI4448; Me, F, H, H, O, H, H, H, H, c-Pr, O, O, NHMe], [AI 4449; Me, F, H, H, O , H, H, H, OMe, O, O, NHMe], [AI 4450; Me, F, H, H, O, H, H, H, OEt, O, O, NHMe], [AI4451; Me, F, H, H, O, H, H, H, SMe, O, O, NHMe], [AI4452; Me, F, H, H, O, H, _{H, H, CF 3, O} , O, NHMe], [AI4453; Et, F, H, H, O, H, H, H, H, O, O, NHMe], [AI4454; Et, F, H , H, O, H, H, H, H, F, O, O, NHMe], [AI 4455; Et, F, H, H, O, H, H, H, Cl, O, O, NHMe], [AI 4456 Et, F, H, H, H, O, H, H, H, H, Br, O, NH, NHMe], [AI 4457; Et, F, H, H, O, H, H, H, I, O, O , NHMe], [AI 4458; Et, F, H, H, O, H, H, H, Me, O, O, NHMe], [AI 4459; Et, F, H, H, O, H, H, H Et, O, O, NHMe], [AI 4460; Et, F, H, H, O, H, H, H, c, Pr, O, O, NHMe], [AI4461; Et, F, H, H , O, H, H, H, H, OMe, O, O, NHMe], [AI4462; Et, F, H, H, O, H, H, H, OEt, O, O, NHMe], [AI4463; Et , F, H, H, O , H, H, H, SMe, O, O, NHMe], [AI4464; Et, F, H, H, O, H, H, H, CF 3, O, O, NHMe], [AI 4465; H, F, F, H, O, H, H, H, H, H, O, O, NHMe], [AI 4466; H, F, F, H, O, H, H, H, F, O, O, NHMe], [AI4467; H, F, F, H, O, H, H, H, H, Cl, O, NH, Me], [AI 4468; H, F, F, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4469; H, F, F, H, O, H, H, H, I, O, NH, Me], [AI 4470; H, F, F, H, O, H, H, H, Me, O, O, NHMe], [AI4471; H, F, F, H, O, H, H, H, Et, O, O, NHMe], [ AI 4472; H, F, F, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4473; H, F, F, H, O, H, H, H, OMe, O, O, NHMe], [AI 4474; H, F, F, H, O, H, H, H, OEt, O, O, NHMe], [AI 4475; H, F, F, H, O, H, H, H, SMe, O, O, NHMe], [AI4476; H, F, F, H, O, H, H, H, CF 3, O, O, NHMe], [AI 4477; Cl, F, F, H, O, H, H, H, H, O, O, NHMe], [AI 4478; Cl, F, F, H, O, H, H, H, F, O , O, NHMe], [AI 4479; Cl, F, F, H, O, H, H, H, H, Cl, O, NH Me], [AI 4480; Cl, F, F, H, O, H, H , H, Br, O, O, NHMe], [AI 4481; Cl, F, F, H, O, H, H, H, I, O, O, NHMe], [AI 4482; Cl, F, F, H , O, H, H, H, H, Me, O, O, NHMe], [AI 4483; Cl, F, F, H, O, H, H, H, Et, O, O, NHMe], [AI 4484; Cl , F, F, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4485; Cl, F, F, H, O, H, H, H, OMe, O, O , NHMe], [AI 4486; Cl, F, F, H, O, H, H, H, OEt, O, O, NHMe], [AI 4487; Cl, F, F, H, O, H, H, H , SMe, O, O, NHMe ], [AI4488; Cl, F, F, H, O, H, H, H, CF 3, O, O, NHMe], [AI4489; Me, F, F, H, O, H, H, H, H, H, O, O, NHMe], [AI 4490; Me, F, F, H, O, H, H, H, F, O, O, NHMe], [AI4491; F, F, H, O, H, H, H, H, H, Cl, O, O, NHMe], [AI4492; Me, F, F, H, O, H, H, H, Br, O, O, NHMe] [AI4493; Me, F, F, H, O, H, H, H, I, O, O, NHMe], [AI4494; Me, F, F, H, O, H, H, H, Me, O, O, NHMe], [AI4495; Me, F, F, H, O, H, H, H, Et, O, O, NHMe], [AI 4496; Me, F, F, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4497; Me, F, F, H, O, H, H, H, OMe, O, O, NHMe], [AI 4498; Me, F, F, H, O, H, H, H, OEt, O, O, NHMe], [AI 4499; Me, F, F, H, O, H, H, S, S, O, O, NHMe], [ AI 4500; Me, F, F, H, O, H, H, H, CF ₃ , O, O, NHMe],

[AI4501; Et, F, F, H, O, H, H, H, H, O, O, NHMe], [AI 4502; Et, F, F, H, O, H, H, H, F, O , O, NHMe], [AI4503; Et, F, F, H, O, H, H, H, H, Cl, O, NHMe], [AI 4504; Et, F, F, H, O, H, H , H, Br, O, O, NHMe], [AI 4505; Et, F, F, H, O, H, H, H, I, O, O, NHMe], [AI 4506; Et, F, F, H , O, H, H, H, H, Me, O, O, NHMe], [AI 4507; Et, F, F, H, O, H, H, H, Et, O, O, NHMe], [AI 4508; Et , F, F, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4509; Et, F, F, H, O, H, H, H, OMe, O, O , NHMe], [AI 4510; Et, F, F, H, O, H, H, H, OEt, O, O, NH Me], [AI 4511; Et, F, F, H, O, H, H, H , SMe, O, O, NHMe ], [AI4512; Et, F, F, H, O, H, H, H, CF 3, O, O, NHMe], [AI4513; H, F, Cl, H, O, H, H, H, H, H, O, O, NHme !, [AI 4514; H, F, Cl, H, O, H, H, H, F, O, O, NHMe], [AI 4515; H, F, Cl, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4516; H, F, Cl, H, O, H, H, H, Br, O, O, NHMe] [AI 4517; H, F, Cl, H, O, H, H, I, O, O, NHMe], [AI 4518; H, F, Cl, H, O, H, H, H, Me, O, O, NHMe], [AI 4519; H, F, Cl, H, O, H, H, H, Et, O, O, NH Me], [AI 4520; H, F, Cl, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4521; H, F, Cl, H, O, H, H, H, OMe, O, O, NHMe], [AI 4522; H, F, Cl, H, O, H, H, H, OEt, O, O, NHMe], [AI 4523; H, F, Cl, H, O, H, H, S, S, O, O, NHMe], [ AI4524; H, F, Cl, H, O, H, H, H, CF 3, O, O, NHMe], [AI4525; Cl, F, Cl, H, O, H, H, H, H, O , O, NHMe], [AI 4526; Cl, F, Cl, H, O, H, H, H, F, O, O, NHMe], [A Cl, F, Cl, H, O, H, H, H, Cl, O, NHMe], [AI 4528; Cl, F, Cl, H, O, H, H, H, Br, O, O, NHMe], [AI 4529; Cl, F, Cl, H, O, H, H, H, I, O, O, NH Me], [AI 4530; Cl, F, Cl, H, O, H, H, H, Me, O, O, NHMe], [AI4531; Cl, F, Cl, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4532; Cl, F, Cl, H, O, H, H, H, H, c-Pr, O, O, NHMe], [AI4533; Cl, F, Cl, H, O, H, H, H, OMe, O, O, NHMe], [AI4534; Cl, F, Cl, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4535; Cl, F, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI4536; Cl, F, Cl, H, O, H, H, H, CF 3, O, O, NHMe], [AI4537; Me, F, Cl, H, O, H, H, H , H, O, O, NHMe], [AI 4538; Me, F, Cl, H, O, H, H, H, H, F, O, O, NHMe], [AI 4539; Me, F, Cl, H, O , H, H, H, H, Cl, O, O, NHMe], [AI 4540; Me, F, Cl, H, O, H, H, H, Br, O, O, NHMe], [AI 451; , Cl, H, O, H, H, H, H, I, O, O, NHMe], [AI4542; Me, F, Cl, H, O, H, H, H, Me, O, O, NHMe], [AI4543; Me, F, Cl, H, O, H, H, H, Et, O, O, NHMe], [AI4544; Me, F, Cl, H, O, H, H, H, c-Pr , O, O, NHMe], [AI 4545; Me, F, Cl, H, O, H, H, H, H, OMe, O, O, NHMe], [AI 4546; Me, F, Cl, H, O, H , H, H, OEt, O, O, NHMe], [AI 4547; Me, F, Cl, H, O, H, H, H, SMe, O, O, NHMe], [AI 4548; Me, F, Cl , H, O, H, H , H, CF 3, O, O, NHMe], [AI4549; Et, F, Cl, H, O, H, H, H, H, O, O, NHMe], [ AI 4550; Et, F, Cl, H, O, H, H, H, F, O, O, NHMe], [AI 4551; Et, F, Cl, H, O, H, H, H, Cl, O, O, NHMe], [AI4552; Et, F, Cl, H , O, H, H, H, H, Br, O, O, NHMe], [AI 4553; Et, F, Cl, H, O, H, H, H, I, O, O, NHMe], [AI 4554; Et , F, Cl, H, O, H, H, H, H, Me, O, O, NHMe], [AI 4555; Et, F, Cl, H, O, H, H, H, Et, O, O, NHMe ], [AI 4556; Et, F, Cl, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4557; Et, F, Cl, H, O, H, H, H , OMe, O, O, NHMe], [AI 4558; Et, F, Cl, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4559; Et, F, Cl, H, O , H, H, H, SMe , O, O, NHMe], [AI4560; Et, F, Cl, H, O, H, H, H, CF 3, O, O, NHMe], [AI4561; H, F, Me, H, O, H, H, H, H, H, O, O, NHMe], [AI4562; H, F, Me, H, O, H, H, H, F, O, O, NHMe] , [AI4563; H, F, Me, H, O, H, H, H, Cl, O, NHMe], [AI 4564; H, F, Me, H, O, H, H, H, Br, O, O, NHMe], [AI 4565; H, F, Me, H, O, H, H, H, I, O, O, NHMe], [AI 4 566; H, F, Me, H, O, H, H, H, Me, O, O, NHMe], [AI 4567; H, F, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4568; H, F, Me, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4569; H, F, Me, H, O, H, H, H, OMe, O, O, NHMe], [ AI 4570; H, F, Me, H, O, H, H, OEt, O, O, NHMe], [AI 4571; H, F, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI4572; H, F, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI4573; Cl, F, Me, H, O, H, H , H, H, O, O, NHMe], [AI 4574; Cl, F, Me, H, O, H, H, H, F, O, O, NHMe], [AI 4575; Cl, F, Me, H , O, H, H, H, H, Cl, O, O, NHMe], [AI 4576; Cl, F, Me, H, O, H, H, H, Br, O, O, NHMe], [AI 4577; Cl , F, Me, H, O, H, H, H, I, O, O, NHMe], [AI 457] 8; Cl, F, Me, H, O, H, H, H, Me, O, O, NHMe], [AI 4579; Cl, F, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4580; Cl, F, Me, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 451; Cl, F, Me, H, O, H, H, H, OMe, O, O, NH, NHMe], [AI4582; Cl, F, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI 4583; Cl, F, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI4584; Cl, F, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI4585 Me, F, Me, H, O, H, H, H, H, H, O, O, NHMe], [AI 4586; Me, F, Me, H, O, H, H, H, F, O, O , NHMe], [AI 4587; Me, F, Me, H, O, H, H, H, Cl, O, NH, Me], [AI 4588; Me, F, Me, H, O, H, H, H , Br, O, O, NHMe], [AI 4589; Me, F, Me, H, O, H, H, H, I, O, O, NHMe], [AI 4590; Me, F, Me, H, O H, H, H, H, Me, O, O, O, NHMe], [AI 4591; Me, F, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4592; Me, F , Me, H, O, H, H, H, c, Pr, O, O, NHMe], [AI 4593; Me, F, Me, H, O, H, H, H, OMe, O, O, NHMe Me, F, Me, H, O, H, H, H, OEt, O, O, NHMe], [AI 4595; Me, F, Me, H, O, H, H, H, SMe] , O, O, NHMe], [AI4596; Me, F, Me, H, O, H, H, H, CF 3, O, O, NHMe], [AI4597; Et, F, Me, H, O, H, H, H, H, H, O, O, NHMe], [AI 4598; Et, F, Me, H, O, H, H, H, F, O, O, NHMe], [AI 4599; Et, F, Me, H, O, H, H, H, H, Cl, O, O, NHMe], [AI 4600; Et, F, Me, H, O, H, H, H, Br, O, O, NHMe],

[AI4601; Et, F, Me, H, O, H, H, H, I, O, O, NHMe], [AI 4602; Et, F, Me, H, O, H, H, H, Me, O , O, NHMe], [AI4603; Et, F, Me, H, O, H, H, H, Et, O, O, NHMe], [AI 4604; Et, F, Me, H, O, H, H , H, c-Pr, O, O, NHMe], [AI 4605; Et, F, Me, H, O, H, H, H, OMe, O, O, NHMe], [AI 4606; Et, F, Me , H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4607; Et, F, Me, H, O, H, H, H, SMe, O, O, NHMe], [AI 4608 ; Et, F, Me, H , O, H, H, H, CF 3, O, O, NHMe], [AI4609; H, F, Et, H, O, H, H, H, H, O, O, NHMe], [AI 4610; H, F, Et, H, O, H, H, H, H, F, O, NH, Me], [AI 4611; H, F, Et, H, O, H, H, H, Cl, O, O, NHMe], [AI 4612; H, F, Et, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4613; H, F, Et, H, O, H, H, H, H, I, O, O, NHMe], [AI 4614; H, F, Et, H, O, H, H, H, Me, O, O, NHMe], [AI 4615; H, F, Et, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4616; H, F, Et, H, O, H, H, H, c-Pr, O, O, NHMe], [AI 4617; H, F, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI 4618; H, F, Et, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4619; H, F, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI 4620; H, F, Et, H, O, _{H, H, H, CF 3} , O, O, NHMe], [AI4621; Cl, F, Et, H, O, H, H, H, H, O, O, NHMe], [AI4622; Cl, F , Et, H, O, H, H, H, H, F, O, O, NHMe], [AI 4623; Cl, F, Et, H, O, H, H, H, Cl, O, O, NHMe], [AI 4624; Cl, F, Et, H, O, H, H, H, Br, O, O, NHMe], [AI 4625; Cl, F, Et, H, O, H, H, H, I, O , O, NHMe], [AI 4626; Cl, F, Et, H, O, H, H, H, Me , O, O, NHMe], [AI4627; Cl, F, Et, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4628; Cl, F, Et, H, O, H , H, H, c-Pr, O, O, NHMe], [AI 4629; Cl, F, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI 4630; Cl, F , Et, H, O, H, H, H, OEt, O, O, NHMe], [AI 4631; Cl, F, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI4632; Cl, F, Et , H, O, H, H, H, CF 3, O, O, NHMe], [AI4633; Me, F, Et, H, O, H, H, H, H, O, O, NHMe], [AI4634; Me, F, Et, H, O, H, H, H, H, F, O, NH, Me], [AI 4635; Me, F, Et, H, O, H, H, H, Cl, O, O, NHMe], [AI 4636; Me, F, Et, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4637; Me, F, Et, H, O, H, H, H, H, I, I, O, O, NHMe], [AI 4638; Me, F, Et, H, O, H, H, H, Me, O, O, NHMe], [AI 4639; Me, F, Et, H, O, H, H, H, H, Et, O, O, NHMe], [AI 4640; Me, F, Et, H, O, H, H, H, c-Pr, O, O, NHMe], [AI4641; Me, F, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI4642; Me, F, Et, H, O, H, H, H, OEt, O, O, NHMe], [AI4643; Me, F, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI 4644; Me, F, Et, H, O, H, H, H, CF 3, O, O, NHMe], [AI4645; Et, F, Et, H, O, H, H, H, H, O, O, NHMe], [AI4646; Et , F, Et, H, O, H, H, H, H, F, O, O, NHMe], [AI 4647; Et, F, Et, H, O, H, H, H, Cl, O, O, NHMe ], [AI 4648; Et, F, Et, H, O, H, H, H, H, Br, O, O, NHMe], [AI 4649; Et, F, Et, H, O, H, H, H, I , O, O, NHMe], [AI4650; Et, F, Et, H, O, H, H, H, H, Me, O, O, NHMe], [AI4651; Et, F, Et, H, O, H , H, H, Et, O, O, NHMe], [AI 4 652; Et, F, Et, H, O, H, H, H, c, Pr, O, O, NHMe], [AI4653; Et, F, Et, H, O, H, H, H, OMe, O, O, NHMe], [AI4654; Et, F, Et, H, O, H, H, H, H, OEt, O, O, NHMe], [AI 4655; Et, F, Et, H, O, H, H, H, SMe, O, O, NHMe], [AI4656; Et, F, Et, H, O, H, H, H, CF 3, O, O, NHMe], [AI4657; H, H, H , F, O, H, H, H, H, H, H, O, O, NHMe], [AI 4658; H, H, H, H, F, O, H, H, F, O, O, NHMe], [AI 4659 H, H, H, H, F, O, H, H, H, H, Cl, O, NHMe], [AI 4660; H, H, H, H, F, O, H, H, H, Br, O, O , NHMe], [AI4661; H, H, H, F, O, H, H, I, O, O, NHMe], [AI4662; H, H, H, F, O, H, H, H , Me, O, O, NHMe], [AI4663; H, H, H, F, O, H, H, H, Et, O, O, NHMe], [AI4664; H, H, H, F, O , H, H, H, c-Pr, O, O, NHMe], [AI 4665; H, H, H, H, F, O, H, H, H, OMe, O, O, NHMe], [AI 4666; H , H, H, F, O, H, H, H, OEt, O, O, NHMe], [AI 4667; H, H, H, H, F, O, H, H, SMe, O, O, NHMe ], [AI4668; H, H , H, F, O, H, H, H, CF 3, O, O, NHMe], [AI4669; Cl, H, H, F, O, H, H, H, H, O, O, NHMe], [AI 4670; Cl, H, H, F, O, H, H, H, F, O, O, NHMe], [AI 4671; Cl, H, H, F, O, H, H, H, H, Cl, O, O, NHMe], [AI 4672; Cl, H, H, F, O, H, H, H, Br, O, O, NHMe], [AI 4673; Cl, H, H, F, O, H, H, H, I, I, O, NH, NH Me], [AI 4674; Cl, H, H, F, O, H, H, Me, O, O, NH Me], [ AI 4 675; Cl, H, H, F, O, H, H, H, Et, O, O, NHMe], [AI 4676; Cl, H, H, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4677; Cl, H, H, F, O, H, H, H, OMe, O, O, NHMe], [AI 4678; Cl , H, H, F, O, H, H, H, OEt, O, O, NHMe], [AI 4679; Cl, H, H, F, O, H, H, S, O, O, NHMe ], [AI4680; Cl, H , H, F, O, H, H, H, CF 3, O, O, NHMe], [AI4681; Me, H, H, F, O, H, H, H, H, O, O, NHMe], [AI4682; Me, H, H, F, O, H, H, H, F, O, O, NHMe], [AI4683; Me, H, H, F, O, H, H, H, H, Cl, O, O, NHMe], [AI 4684; Me, H, H, F, O, H, H, H, Br, O, NH, Me], [AI 4 685; H, F, O, H, H, H, I, I, O, O, NHMe], [AI 4686; Me, H, H, F, O, H, H, Me, O, O, NHMe], [ AI 4687; Me, H, H, F, O, H, H, H, Et, O, O, NHMe], [AI 4688; Me, H, H, F, O, H, H, H, c-Pr, O, O, NHMe], [AI4689; Me, H, H, F, O, H, H, H, OMe, O, O, NHMe], [AI 4690; Me, H, H, F, O, H, H, H, OEt, O, O, NHMe], [AI4691; Me, H, H, F, O, H, H, S, O, O, NHMe], [AI4692; Me, H, H, F, O, H, H, H, CF 3, O, O, NHMe], [AI4693; Et, H, H, F, O, H, H, H, H, O, O, NHMe], [AI4694 Et, H, H, F, O, H, H, H, H, F, O, O, NHMe], [AI 4695; Et, H, H, F, O, H, H, H, Cl, O, O , NHMe], [AI4696; Et, H, H, F, O, H, H, H, Br, O, O, NHMe], [AI 4697; Et, H, H, F, O, H, H, H , I, O, O, NHMe], [AI 4698; Et, H, H, H, F, O, H, H, H, Me, O, O, NH Me], [AI 4699; Et, H, H, F, O , H, H, H, H, Et, O, O, NHMe], [AI 4700; Et, H, H, H, F, O, H, H, H, c-Pr, O, O, NHMe],

[AI4701; Et, H, H, F, O, H, H, OMe, O, O, NHMe], [AI 4702; Et, H, H, F, O, H, H, H, OEt, O , O, NHMe], [AI4703; Et, H, H, F, O, H, H, SMe, O, O, NHMe], [AI 4704; Et, H, H, F, O, H, H _{, H, CF 3, O,} O, NHMe], [AI4705; H, H, F, F, O, H, H, H, H, O, O, NHMe], [AI4706; H, H, F, F, O, H, H, H, H, F, O, O, NHMe], [AI 4707; H, H, F, F, O, H, H, H, Cl, O, O, NHMe], [AI 4708; H, H, F, F, O, H, H, H, H, Br, O, O, NHMe], [AI 4709; H, H, F, F, O, H, H, H, I, O, O, NHMe], [AI 4710; H, H, F, F, O, H, H, Me, O, O, NH Me], [AI 4711; H, H, F, F, O, H, H, H, Et, O, O, NHMe], [AI 4712; H, H, F, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4713; H, H, F, F, O, H, H, H, H, OMe, O, O, NHMe], [AI 4714; H, H, F, F, O, H, H, H, OEt, O, O, NHMe], [AI 4715; H, H, F, F, O, H, H, H, SMe, O, O, NHMe], [AI4716; H, H, F, F, O, H, H, H, CF 3, O, O, NHMe Cl, H, F, F, O, H, H, H, H, O, O, NHMe], [AI 4718; Cl, H, F, F, O, H, H, H, F] , O, O, NHMe], [AI 4719; Cl, H, F, F, O, H, H, H, H, Cl, O, NH, Me], [AI 4720; Cl, H, F, F, O, H , H, H, Br, O, O, NHMe], [AI4721; Cl, H, F, F, O, H, H, I, O, O, NHMe], [AI4722; Cl, H, F , F, O, H, H, H, H, Me, O, O, NHMe], [AI 4723; Cl, H, F, F, O, H, H, H, Et, O, O, NHMe], [AI 4724 Cl, H, F, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4725; Cl, H, F, F, O, H, H, H, OMe, O , O, NHMe], [AI 4726; Cl, H, F, F, O, H, H, H, OEt, O, O, NHMe], [AI 4727; Cl, H , F, F, O, H , H, H, SMe, O, O, NHMe], [AI4728; Cl, H, F, F, O, H, H, H, CF 3, O, O, NHMe] [AI 4729; Me, H, F, F, O, H, H, H, H, O, O, NHMe], [AI 4730; Me, H, F, F, O, H, H, H, F, O, O, NHMe], [AI 4731; Me, H, F, F, O, H, H, H, Cl, O, NH Me], [AI 4732; Me, H, F, F, O, H, H, H, Br, O, O, NHMe], [AI4733; Me, H, F, F, O, H, H, H, I, O, O, NHMe], [AI 4734; Me, H, F, F, O, H, H, H, H, Me, O, O, NHMe], [AI 4735; Me, H, F, F, O, H, H, H, Et, O, O, NHMe], [AI 4736; Me, H, F, F, O, H, H, H, c, Pr, O, O, NHMe], [AI 4737; Me, H, F, F, O, H, H, H, OMe, O, O, NHMe], [AI 4738; Me, H, F, F, O, H, H, OEt, O, O, NHMe], [AI 4739; Me, H, F, F, O, H, H, H, SMe, O, O, NHMe], [AI4740; Me, H, F, F, O, H, H, H, CF 3, O, O, NHMe], [AI4741; Et, H, F, F , O, H, H, H, H, H, O, O, NHMe], [AI4742; Et, H, F, F, O, H, H, H, F, O, O, NHMe], [AI4743; Et , H, F, F, O, H, H, H, H, Cl, O, O, NHMe], [AI 4744; Et, H, F, F, O, H, H, H, Br, O, O, NHMe ], [AI 4745; Et, H, F, F, O, H, H, H, I, O, O, NHMe], [AI 4746; Et, H, F, F, O, H, H, H, Me , O, O, NHMe], [AI 4747; Et, H, F, F, O, H, H, H, Et, O, O, NH Me], [AI 4748; Et, H, F, F, O, H , H, H, c-Pr, O, O, NHMe], [AI 4749; Et, H, F, F, O, H, H, H, OMe, O, O, NHMe], [AI 4 750; Et, H , F, F, O, H, H, H, H, OEt, O, O, NHMe], [AI 4751; Et, H, F, F, O, H, H, SMe, O, O, NHMe], [AI4752; Et, H, F , F, O, H, H, H, CF 3, O, O, NHMe], [AI4753; H, H, Cl, F, O, H, H, H, H, H, O, O, NHMe], [AI 4754; H, H, Cl, F, O, H, H, F, O, O, NHMe] H, H, Cl, F, O, H, H, H, Cl, O, NHMe], [AI 4756; H, H, Cl, F, O, H, H, H, Br, O, O, NHMe], [AI4757; H, H, Cl, F, O, H, H, I, O, O, NHMe], [AI4758; H, H, Cl, F, O, H, H, H, Me, O, O, NHMe], [AI4759; H, H, Cl, F, O, H, H, H, Et, O, O, NHMe], [AI 4760; H, H, Cl, F, O, H, H, H, H, c-Pr, O, O, NHMe], [AI4761; H, H, Cl, F, O, H, H, H, OMe, O, O, NHMe], [ AI4762; H, H, Cl, F, O, H, H, OEt, O, O, NHMe], [AI4763; H, H, Cl, F, O, H, H, H, SMe, O, O, NHMe], [AI4764; H, H, Cl, F, O, H, H, H, CF 3, O, O, NHMe], [AI4765; Cl, H, Cl, F, O, H, H , H, H, O, O, NHMe], [AI 4766; Cl, H, Cl, F, O, H, H, H, F, O, O, NHMe], [AI 4767; Cl, H, Cl, F , O, H, H, H, H, Cl, O, O, NHMe], [AI 4768; Cl, H, Cl, F, O, H, H, H, Br, O, O, NHMe], [AI 4769; Cl , H, Cl, F, O, H, H, H, I, O, O, NHMe], [AI 4770; Cl, H, Cl, F, O, H, H, Me, O, O, NHMe ], [AI 4771; Cl, H, Cl, F, O, H, H, H, Et, O, O, NH Me], [AI 4772; Cl, H, Cl, F, O, H, H, H, c -Pr, O, O, NHMe], [AI 4773; Cl, H, Cl, F, O, H, H, H, H, OMe, O, O, NHMe], [AI 4774; Cl, H, Cl, F, O H, H, H, H, OEt, O, O, NHMe], [AI 4775; Cl, H, Cl, F, O, H, H, H, SMe, O, O, NHMe], [AI 4776; Cl, H , Cl, F, O, H , H, H, CF 3, O, O, NHMe], [AI4777; Me, H, Cl, F, O, H, H, H, H, O, O, NHMe] , [AI 4778; Me, H, Cl, F, O, H, H, H, F, O, O, NHMe], [AI 4779; Me, H, Cl, F, O, H, H, H, Cl, O, NH, NHMe], [AI 4780; Me, H, Cl, F, O, H, H, H, Br, O Me, H, Cl, F, O, H, H, I, O, O, NH Me], [AI 4782; Me, H, Cl, F, O, H, H , H, Me, O, O, NHMe], [AI 4783; Me, H, Cl, F, O, H, H, H, Et, O, O, NHMe], [AI 4784; Me, H, Cl, F , O, H, H, H, c, -Pr, O, O, NHMe], [AI 4 785; Me, H, Cl, F, O, H, H, H, O, O, O, NH Me], [AI 4786 Me, H, Cl, F, O, H, H, H, H, OEt, O, O, NHMe], [AI4787; Me, H, Cl, F, O, H, H, H, SMe, O, O , NHMe], [AI4788; Me , H, Cl, F, O, H, H, H, CF 3, O, O, NHMe], [AI4789; Et, H, Cl, F, O, H, H, H, H, O, O, NHMe], [AI 4790; Et, H, Cl, F, O, H, H, H, H, F, O, O, NHMe], [AI4791; Et, H, Cl, F, O, H, H, H, H, Cl, O, O, NHMe], [AI4792; Et, H, Cl, F, O, H, H, H, Br, O, O, NHMe], [AI4793; Et, H, Cl, F, O, H, H, H, H, I, O, O, NHMe], [AI 4794; Et, H, Cl, F, O, H, H, Me, O, O, NHMe] [AI4795; Et, H, Cl, F, O, H, H, H, Et, O, O, NHMe], [AI4796; Et, H, Cl, F, O, H, H, H, c- Pr, O, O, NHMe], [AI 4797; Et, H, Cl, F, O, H, H, H, H, OMe, O, O, NHMe], [AI 4798; Et, H, Cl, F, O, H, H, H, H, OEt, O, O, NHMe], [AI 4799; Et, H, Cl, F, O, H, H, H, SMe, O, O, NHMe], [AI 4800; Et, H, Cl, F, O, H, H, H, CF 3, O, O, NHMe],

[AI4801; H, H, Me, F, O, H, H, H, H, O, O, NHMe], [AI 4802; H, H, Me, F, O, H, H, H, F, O , O, NHMe], [AI4803; H, H, Me, F, O, H, H, H, Cl, O, NHMe], [AI 4804; H, H, Me, F, O, H, H , H, Br, O, O, NHMe], [AI 4805; H, H, Me, F, O, H, H, I, O, O, NHMe], [AI 4806; H, H, Me, F , O, H, H, H, H, Me, O, O, NHMe], [AI 4807; H, H, Me, F, O, H, H, H, Et, O, O, NHMe], [AI 4808; H , H, Me, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4809; H, H, Me, F, O, H, H, H, OMe, O, O , NHMe], [AI 4810; H, H, Me, F, O, H, H, OEt, O, O, NH Me], [AI 4811; H, H, Me, F, O, H, H, H , SMe, O, O, NHMe ], [AI4812; H, H, Me, F, O, H, H, H, CF 3, O, O, NHMe], [AI4813; Cl, H, Me, F, O, H, H, H, H, H, O, O, NHMe], [AI 4814; Cl, H, Me, F, O, H, H, H, F, O, O, NHMe], [AI 4815; Cl, H, Me, F, O, H, H, H, H, Cl, O, NH, NH Me], [AI 4816; Cl, H, Me, F, O, H, H, H, Br, O, O, NH Me] [AI 4817; Cl, H, Me, F, O, H, H, I, O, O, NHMe], [AI 4818; Cl, H, Me, F, O, H, H, H, Me, O, O, NHMe], [AI 4819; Cl, H, Me, F, O, H, H, H, Et, O, O, NH Me], [AI 4820; Cl, H, Me, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4821; Cl, H, Me, F, O, H, H, H, OMe, O, O, NHMe], [AI 4822; Cl, H, Me, F, O, H, H, H, OEt, O, O, NHMe], [AI 4823; Cl, H, Me, F, O, H, H, S, S, O, O, NHMe], [ AI4824; Cl, H, Me, F, O, H, H, H, CF 3, O, O, NHMe], [AI4825; Me, H, Me, F, O, H, H, H, H, O , O, NHMe], [AI 4826; Me, H, Me, F, O, H, H, H, F, O, O, NHMe], [AI 4827; Me, H, Me, F, O, H, H, H, Cl, O, NH Me], [AI 4828; Me, H, Me, F, O, H, H, H, Br, O, O, NHMe], [AI4829; Me, H, Me, F, O, H, H, I, O, O, NHMe], [AI 4830; Me, H, Me, F, O, H, H, H, H, Me, O, O, NHMe], [AI 4831; Me, H, Me, F, O, H, H, H, Et, O, O, NHMe], [AI 4832; Me, H, Me, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4833; Me, H, Me, F, O, H, H, H, OMe, O, O, NHMe], [AI 4834; Me, H, Me, F, O, H, H, OEt, O, O, NHMe], [AI 4835; Me, H, Me, F, O, H, H, H, SMe, O, O, NHMe], [AI4836; Me, H, Me, F, O, H, H, H, CF 3, O, O, NHMe], [AI4837; Et, H, Me, F , O, H, H, H, H, H, O, O, NHMe], [AI 4838; Et, H, Me, F, O, H, H, H, F, O, O, NHMe], [AI 4839; Et , H, Me, F, O, H, H, H, H, Cl, O, O, NHMe], [AI 4840; Et, H, Me, F, O, H, H, H, Br, O, O, NHMe ], [AI4841; Et, H, Me, F, O, H, H, H, I, O, O, NHMe], [AI4842; Et, H, Me, F, O, H, H, H, Me , O, O, NHMe], [AI4843; Et, H, Me, F, O, H, H, H, Et, O, O, NHMe], [AI 4844; Et, H, Me, F, O, H , H, H, c-Pr, O, O, NHMe], [AI 4845; Et, H, Me, F, O, H, H, H, OMe, O, O, NHMe], [AI 4846; Et, H , Me, F, O, H, H, H, H, OEt, O, O, NHMe], [AI 4847; Et, H, Me, F, O, H, H, H, SMe, O, O, NHMe], [AI4848; Et, H, Me , F, O, H, H, H, CF 3, O, O, NHMe], [AI4849; H, H, Et, F, O, H, H, H, H, O, O, NHMe], [AI4850; H, H, Et, F, O, H, H, H, F, O, NH, Me], [AI4851; H, H, Et, F, O, H, H, H, Cl, O, O, NHMe], [AI4852; H, H, Et, F, O, H, H, H, H, Br, O, O, NHMe], [AI 4853; H, H, Et, F, O, H, H, H, I, O, O, NHMe], [AI4854; H, H, Et, F, O, H, H, Me, O, O, NHMe], [AI 4855; H, H, Et, F, O, H, H, H, H, Et, O, O, NHMe], [AI 4856; H, H, Et, F, O, H, H, H, c-Pr, O, O, NHMe], [AI 4857; H, H, Et, F, O, H, H, H, H, OMe, O, O, NHMe], [AI 4858; H, H, Et, F, O, H, H, H, OEt, O, O, NHMe], [AI 4859; H, H, Et, F, O, H, H, H, SMe, O, O, NHMe], [AI4860; H, H, Et, F, O, H, H, H, CF 3, O, O, NHMe ], [AI4861; Cl, H, Et, F, O, H, H, H, H, O, O, NHMe], [AI4862; Cl, H, Et, F, O, H, H, H, F] , O, O, NHMe], [AI4863; Cl, H, Et, F, O, H, H, H, H, Cl, O, NH, Me], [AI 4864; Cl, H, Et, F, O, H , H, H, Br, O, O, NHMe], [AI4865; Cl, H, Et, F, O, H, H, H, I, O, O, NHMe], [AI 4866; Cl, H, Et , F, O, H, H, H, H, Me, O, O, NHMe], [AI 4867; Cl, H, Et, F, O, H, H, H, Et, O, O, NHMe], [AI 4868 Cl, H, Et, F, O, H, H, H, c, Pr, O, O, NHMe], [AI 4869; Cl, H, Et, F, O, H, H, H, OMe, O , O, NHMe], [AI4870; Cl, H, Et, F, O, H, H, H, OEt, O, O, NHMe], [AI 4871; Cl, H, Et, F, O, H, H , H, SMe, O, O , NHMe], [AI4872; Cl, H, Et, F, O, H, H, H, CF 3, O, O, NHMe], [AI4873; Me, H, Et, F, O, H, H, H, H, H, H, O, O, NHMe], [AI 4874; Me, H, Et, F, O, H, H, H, F, O, O, NHMe], [AI 4875; Me, H, Et, F, O, H, H, H, H, Cl, O, NHMe], [AI 4876; Me, H, Et, F, O, H, H, H, Br, O, O, NHMe], [AI 4877; Me, H, Et, F, O, H, H, H, I, O, O, NHMe], [AI4878; Me, H, Et, F, O, H, H, H, Me, O, O, NHMe], [AI 4879; Me, H, Et, F, O, H, H, H, Et, O, O, NHMe], [AI 4880; Me, H, Et, F, O, H, H, H, c-Pr, O, O, NHMe], [AI4881; Me, H, Et, F, O, H, H, H, H, OMe, O, O, NHMe], [AI4882; Me, H, Et, F, O, H, H, H, OEt, O, O, NHMe], [AI4883; Me, H, Et, F, O, H, H, H, SMe, O, O, NHMe], [AI4884; Me, H, Et, F, O, H, H, H, CF 3, O, O, NHMe ], [AI 4885; Et, H, Et, F, O, H, H, H, H, O, O, NH Me], [AI 4886; Et, H, Et, F, O, H, H, H, F] , O, O, NHMe], [AI4887; Et, H, Et, F, O, H, H, H, Cl, O, NH, Me], [AI 4888; Et, H, Et, F, O, H , H, H, Br, O, O, NHMe], [AI 4889; Et, H, Et, F, O, H, H, H, I, O, O, NHMe], [AI 4890; Et, H, Et , F, O, H, H, H, H, Me, O, O, NHMe], [AI4891; Et, H, Et, F, O, H, H, H, Et, O, O, NHMe], [AI4892 Et, H, Et, F, O, H, H, H, c, Pr, O, O, NHMe], [AI4893; Et, H, Et, F, O, H, H, H, OMe, O , O, NHMe], [AI 4894; Et, H, Et, F, O, H, H, H, OEt, O, O, NH Me], [AI 4895; Et, H, Et, F, O, H, H , H, SMe, O, O , NHMe], [AI4896; Et, H, Et, F, O, H, H, H, CF 3, O, O, NHMe], [AI4897; H, H, H, H, O, F, H, H, H, H, O, O, NHMe], [AI 4898; H, H, H, H, H, O, F, H, F, O, O, NHMe], [AI 4899; H, H, H, H, H, O, F, H, H, Cl, O, NH, NHMe], [AI 4900; H, H, H, H, H, O, F, H, Br, O, O, NHMe],

[AI4901; H, H, H, H, H, O, F, H, I, O, O, NHMe], [AI4902; H, H, H, H, O, F, H, H, Me, O H, H, H, H, H, H, O, F, H, Et, O, O, NHMe], [AI 4904; H, H, H, H, O, F, H , H, c-Pr, O, O, NHMe], [AI 4905; H, H, H, H, H, O, F, H, OMe, O, O, NHMe], [AI 4906; H, H, H , H, O, F, H, H, OEt, O, O, NHMe], [AI 4907; H, H, H, H, H, O, F, H, SMe, O, O, NHMe], [AI 4908 ; H, H, H, H , O, F, H, H, CF 3, O, O, NHMe], [AI4909; Cl, H, H, H, O, F, H, H, H, O, O, NHMe], [AI 4910; Cl, H, H, H, H, O, F, H, H, F, O, O, NH Me], [AI 4911; Cl, H, H, H, O, F, H, H, Cl, O, O, NHMe], [AI4912; Cl, H, H, H, H, O, F, H, H, Br, O, O, NHMe], [AI4913; Cl, H, H, H, O, F, H, H, I, O, O, NHMe], [AI 4914; Cl, H, H, H, H, O, F, H, Me, O, O, NHMe], [AI 4915; H, H, H, H, O, F, H, H, Et, O, O, NHMe], [AI 4916; Cl, H, H, H, H, O, F, H, c, Pr, O, O, NHMe], [AI 4917; Cl, H, H, H, O, F, H, H, OMe, O, O, NHMe], [AI 4918; Cl, H, H, H, O, F, H, H, H, OEt, O, O, NHMe], [AI4919; Cl, H, H, H, H, O, F, H, SMe, O, O, NHMe], [AI4920; Cl, H, H, H, O, _{F, H, H, CF 3} , O, O, NHMe], [AI4921; Me, H, H, H, O, F, H, H, H, O, O, NHMe], [AI4922; Me, H , H, H, O, F, H, H, F, O, O, NHMe], [AI 4923; Me, H, H, H, O, F, H, H, Cl, O, O, NHMe], [AI4924; Me, H, H, H, H, O, F, H, H, Br, O, O, NHMe], [AI 4925; Me, H, H, H, O, F, H, H, I, O , O, NHMe], [AI 4926; Me, H, H, H, O, F, H, H, Me, O, O, NHMe], [AI 4 927; Me, H, H, H, H, O, F, H, H, Et, O, O, NHMe], [AI 4928; Me, H, H, H, O, F, H, H, c-Pr, O, O, NHMe], [AI 4929; Me, H, H, H, O, F, H, OMe, O, O, NHMe], [AI 4930; Me, H, H, H, O, F, H, H, OEt, O, O, NHMe], [AI4931; Me, H, H, H, H, O, F, H, SMe, O, O, NHMe], [AI4932; Me, H, H, H, O, _{F, H, H, CF 3} , O, O, NHMe], [AI4933; Et, H, H, H, O, F, H, H, H, O, O, NHMe], [AI4934; Et, H , H, H, O, F, H, H, F, O, O, NHMe], [AI 4935; Et, H, H, H, O, F, H, H, Cl, O, O, NHMe], [AI4936; Et, H, H, H, H, O, F, H, H, Br, O, O, NHMe], [AI 4937; Et, H, H, H, H, O, F, H, H, I, O , O, NHMe], [AI 4938; Et, H, H, H, H, O, F, H, Me, O, O, NH Me], [AI 4939; Et, H, H, H, O, F, H , H, Et, O, O, NHMe], [AI 4940; Et, H, H, H, H, O, F, H, c, Pr, O, O, NHMe], [AI4941; Et, H, H , H, O, F, H, H, OMe, O, O, NHMe], [AI4942; Et, H, H, H, H, O, F, H, OEt, O, O, NHMe], [AI4943 Et, H, H, H, H, O, F, H, H, S Me, O, O, NH Me], [AI 4944; Et, H, H, H, H, O, F, H, CF ₃ , O, O, NHMe], [AI 4945; H, H, F, H, O, F, H, H, H, O, O, NHMe], [AI 4946; H, H, F, H, O, F, H, H, F, O, O, NHMe], [AI 4947; H, H, F, H, O, F, H, H, Cl, O, O, NHMe], [AI 4948; H, H, F, H, O, F, H, H, Br, O, O, NHMe], [AI 4949; H, H, F, H, O, F, H, I, O, O, NHMe], [AI 4950; H, H, F, H, O, F, H, H, Me, O, O, NHMe], [AI 4951; H, H, F, H, O, F, H, H, Et, O, O, NHMe] [AI4952; H, H, F, H, O, F, H, c, Pr, O, O, NHMe], [AI 4953; H, H, F, H, O, F , H, H, OMe, O, O, NHMe], [AI 4954; H, H, F, H, O, F, H, H, OEt, O, O, NHMe], [AI 4 955; H, H, F , H, O, F, H , H, SMe, O, O, NHMe], [AI4956; H, H, F, H, O, F, H, H, CF 3, O, O, NHMe], [ AI 4957; Cl, H, F, H, O, F, H, H, H, O, O, NHMe], [AI 4958; Cl, H, F, H, O, F, H, H, F, O, O, NHMe], [AI 4959; Cl, H, F, H, O, F, H, H, Cl, O, NH, Me], [AI 4960; Cl, H, F, H, O, F, H, H, Br, O, O, NHMe], [AI4961; Cl, H, F, H, O, F, H, I, O, O, NHMe], [AI4962; Cl, H, F, H, O, F, H, H, Me, O, O, NHme !, [AI 4963; Cl, H, F, H, O, F, H, H, Et, O, O, NHMe], [AI 4964; Cl, H, F, H, O, F, H, H, c, Pr, O, O, NHMe], [AI 4965; Cl, H, F, H, O, F, H, OMe, O, O, NHMe], [AI4966; Cl, H, F, H, O, F, H, H, OEt, O, O, NHMe], [AI 4967; Cl, H, F, H, O, F, H, H, H, SMe, O, O, NHMe] , [AI4968; Cl, H, F, H, O, F, H, H, CF 3, O, O, NHMe], [AI4969; Me, H, F, H, O , F, H, H, H, H, O, O, O, NHMe], [AI 4970; Me, H, F, H, O, F, H, H, F, O, O, NHMe], [AI 4971; Me, H , F, H, O, F, H, H, H, Cl, O, O, NHMe], [AI 4972; Me, H, F, H, O, F, H, H, Br, O, O, NHMe], [AI 4973; Me, H, F, H, O, F, H, I, O, O, NHMe], [AI 4974; Me, H, F, H, O, F, H, H, Me, O , O, NHMe], [AI 4 975; Me, H, F, H, O, F, H, H, Et, O, O, NH Me], [AI 4976; Me, H, F, H, O, F, H , H, c-Pr, O, O, NHMe], [AI 4977; Me, H, F, H, O, F, H, OMe, O, O, NHMe], [AI 4978; Me, H, F , H, O, F, H, H, OEt, O, O, NHMe], [AI 4979; Me, H, F, H, O, F, H, H, SMe, O, O, NHMe], [AI4980; Me, H, F, H, O, F, H, H, CF 3, O, O, NHMe], [AI4981; Et, H, F, H , O, F, H, H, H, H, O, O, NHMe], [AI4982; Et, H, F, H, O, F, H, F, O, O, NHMe], [AI4983; Et , H, F, H, O, F, H, H, H, Cl, O, O, NHMe], [AI4984; Et, H, F, H, O, F, H, H, Br, O, O, NHMe ], [AI4985; Et, H, F, H, O, F, H, I, O, O, NHMe], [AI 4986; Et, H, F, H, O, F, H, H, Me , O, O, NHMe], [AI 4987; Et, H, F, H, O, F, H, H, Et, O, O, NH Me], [AI 4988; Et, H, F, H, O, F , H, H, c-Pr, O, O, NHMe], [AI 4989; Et, H, F, H, O, F, H, H, OMe, O, O, NHMe], [AI 4 990; Et, H , F, H, O, F, H, H, OEt, O, O, NHMe], [AI4991; Et, H, F, H, O, F, H, H, SMe, O, O, NHMe], [AI4992; Et, H, F , H, O, F, H, H, CF 3, O, O, NHMe], [AI4993; H, H, Cl, H, O, F, H, H, H, O, O, NHMe], [AI4994; H, H, Cl, H, O, F, H, H, F, O, O, NHMe], [AI 4995; H, H, Cl, H, O, F, H, H, Cl, O, O, NHMe], [AI 4996; H, H, Cl, H, O, F, H, H, Br, O, O, NHMe], [AI 4 997; H, H, Cl, H, O, F, H, H, I, I, O, O, NHMe], [AI 4998; H, H, Cl, H, O, F, H, Me, O, O, NHMe], [AI 4999; H, H, Cl, H, O, F, H, H, Et, O, O, NHMe], [AI 5000; H, H, Cl, H, O, F, H, H, c-Pr, O, O, NHMe],

[AI 5001; H, H, Cl, H, O, F, H, OMe, O, O, NHMe], [AI 5002; H, H, Cl, H, O, F, H, H, OE t, O , O, NHMe], [AI 5003; H, H, Cl, H, O, F, H, S Me, O, O, NH Me], [AI 5004; H, H, Cl, H, O, F, H _{, H, CF 3, O,} O, NHMe], [AI5005; Cl, H, Cl, H, O, F, H, H, H, O, O, NHMe], [AI5006; Cl, H, Cl, H, O, F, H, H, F, O, O, NHMe], [AI 5007; Cl, H, Cl, H, O, F, H, Cl, O, O, NHMe], [AI 5008; Cl, H, Cl, H, O, F, H, H, Br, O, O, NHMe], [AI 5009; Cl, H, Cl, H, O, F, H, I, O, O, NHMe], [AI 5010; Cl, H, Cl, H, O, F, H, Me, O, O, NH Me], [AI 5011; Cl, H, Cl, H, O, F, H, H, Et, O, O, NHMe], [AI 5012; Cl, H, Cl, H, O, F, H, c, Pr, O, O, NHMe], [AI 5013; Cl, H, Cl, H, O, F, H, H, OMe, O, O, NHMe], [AI 5014; Cl, H, Cl, H, O, F, H, OEt, O, O, NHMe], [AI 5015; Cl, H, Cl, H, O, F, H, H, SMe, O, O, NHMe], [AI5016; Cl, H, Cl, H, O, F, H, H, CF 3, O, O, NHMe Me, H, Cl, H, O, F, H, H, H, O, O, NHMe], [AI 5018; Me, H, Cl, H, O, F, H, H, F] , O, O, NHMe], [AI 5019; Me, H, Cl, H, O, F, H, H, Cl, O, O, NH Me], [AI 5020; Me, H, Cl, H, O, F , H, H, Br, O, O, NHMe], [AI 5021; Me, H, Cl, H, O, F, H, I, O, O, NHMe], [AI 5022; Me, H, Cl , H, O, F, H, H, Me, O, O, NHMe], [AI 5023; Me, H, Cl, H, O, F, H, Et, O, O, NHMe], [AI 5024 Me, H, Cl, H, O, F, H, H, c-Pr, O, O, NHMe], [AI 5025; Me, H, Cl, H, O, F, H, H, OMe, O , O, NHMe], [AI 5026; Me, H, Cl, H, O, F, H, H, OEt, O, O, NHMe], [AI 5027; Me, H, Cl, H, O, F, H, SMe, O, O, NHMe], [AI 5028; Me, H, Cl, H, O, F, H, H, CF 3, O, O, NHMe], [AI5029; Et, H, Cl, H, O, F, H, H, H, O, O, NHMe ], [AI 5030; Et, H, Cl, H, O, F, H, H, F, O, O, NHMe], [AI 5031; Et, H, Cl, H, O, F, H, H, Cl, , O, O, NHMe], [AI 5032; Et, H, Cl, H, O, F, H, H, Br, O, O, NH Me], [AI 5033; Et, H, Cl, H, O, F , H, H, I, O, O, NHMe], [AI 5034; Et, H, Cl, H, O, F, H, Me, O, O, NHMe], [AI 5035; Et, H, Cl , H, O, F, H, H, Et, O, O, NHMe], [AI 5036; Et, H, Cl, H, O, F, H, c, Pr, O, O, NHMe], [AI5037; Et, H, Cl, H, O, F, H, OMe, O, O, NHMe], [AI 5038; Et, H, Cl, H, O, F, H, H, OEt, O , O, NHMe], [AI5039; Et, H, Cl, H, O, F, H, SMe, O, O, NHMe], [AI 5040; Et, H, Cl, H, O, F, H _{, H, CF 3, O,} O, NHMe], [AI5041; H, H, Me, H, O, F, H, H, H, O, O, NHMe], [AI5042; H, H, Me, H, O, F, H, H, F, O, O, NHMe], [AI 5043; H, H, Me, H, O, F, H, Cl, O, O, NHMe], [AI 5044; H, H, Me, H, O, F, H, H, Br, O, O, NHMe], [AI 5045; H, H, Me, H, O, F, H, I, O, O, NHMe], [AI 5046; H, H, Me, H, O, F, H, H, Me, O, O, NHMe], [AI 5047; H, H, Me, H, O, F, H, H, Et, O, O, NHMe], [AI 5048; H, H, Me, H, O, F, H, c, Pr, O, O, NHMe], [AI 5049; H, H, Me, H, O, F, H, H, OMe, O, O, NHMe], [AI 5050; H, H, Me, H, O, F, H, OEt, O, O, NHMe], [AI 5051; H, H, Me, H, O, F, H, H, SMe, O, O, NHMe], [AI 5052; H, H, Me, H, O, F, H, H, CF 3, O, O, NHMe], [AI5053; Cl, H, Me, H, O, F, H, H, H, O , O, NHMe], [AI 5054; Cl, H, Me, H, O, F, H, H, F, O, O, NH Me], [AI 5055; Cl, H, Me, H, O, F, H , H, Cl, O, O, NHMe], [AI 5056; Cl, H, Me, H, O, F, H, H, Br, O, O, NHMe], [AI 5057; Cl, H, Me, H , O, F, H, H, I, I, O, O, NHMe], [AI 5058; Cl, H, Me, H, O, F, H, Me, O, O, NHMe], [AI 5059; Cl , H, Me, H, O, F, H, H, Et, O, O, NHMe], [AI 5060; Cl, H, Me, H, O, F, H, H, c-Pr, O, O , NHMe], [AI5061; Cl, H, Me, H, O, F, H, OMe, O, O, NHMe], [AI5062; Cl, H, Me, H, O, F, H, H , OEt, O, O, NHMe], [AI 5063; Cl, H, Me, H, O, F, H, S, S, O, O, NHMe], [AI 5064; Cl, H, Me, H, O , F, H, H, CF 3, O, O, NHMe], [AI5065; Me, H, Me, H, O, F, H, H, H, O, O, NHMe], [AI5066; Me, H, Me, H, O, F, H, H, F, O, O, NHMe], [AI 5067; Me, H, Me, H, O, F, H, H, Cl, O, O, NHMe] , [AI 50 68; Me, H, Me, H, O, F, H, H, Br, O, O, NHMe], [AI 5069; Me, H, Me, H, O, F, H, H, I, O, O, NHMe], [AI 5070; Me, H, Me, H, O, F, H, H, Me, O, O, NHMe], [AI 5071; Me, H, Me, H, O, F, H, H, Et, O, O, NHMe], [AI5072; Me, H, Me, H, O, F, H, c, Pr, O, O, NHMe], [AI 5073; Me, H, Me, H, O, F, H, H, OMe, O, O, NHMe], [AI 5074; Me, H, Me, H, O, F, H, H, OEt, O, O, NHMe], [ AI 50 75; Me, H, Me, H, O, F, H, S, S, O, O, NH Me], [AI 5076; Me, H, Me, H, O, F, H, H, CF ₃ , O , O, NHMe], [AI 5077; Et, H, Me, H, O, F, H, H, H, H, O, O, NHMe], [AI 5078; Et, H, Me, H, O, F, H, F, O, O, NHMe], [AI 5079; Et, H, Me, H, O, F, H, H, Cl, O, NHme !, [AI 5080; Et, H, Me, H, O, F, H, Br, O, O, NHMe], [AI5081; Et, H, Me, H, O, F, H, I, O, O, NHMe], [AI5082; Et, H, Me, H, O, F, H, H, H, Me, O, O, NHMe], [AI 5083; Et, H, Me, H, O, F, H, H, Et, O, O, NH Me], [AI 5084; Et, H, Me, H, O, F, H, H, H, c-Pr, O, O, NHMe], [AI5085; Et, H, Me, H, O, F, H, H, OMe, O, O, NHMe], [AI 5086; Et, H, Me, H, O, F, H, H, OEt, O, O, NHMe], [AI 5087; Et, H, Me, H, O, F, H, H, SMe, O, O, NHMe] , [AI5088; Et, H, Me, H, O, F, H, H, CF 3, O, O, NHMe], [AI5089; H, H, Et, H, O, F, H, H, H , O, O, NHMe], [AI5090; H, H, Et, H, O, F, H, H, F, O, O, NHMe], [AI5091; H, H, Et, H, O, F , H, H, Cl, O, O, NHMe], [AI5092; H, H, Et, H, O, F, H, H, Br, O, NHMe], [AI 5093; H, H, Et , H, O, F, H, H, I, I, O, O, NHMe], [AI 5094; H, H, Et, H, O, F, H, Me, O, O, NHMe], [AI 5095 H, H, Et, H, O, F, H, H, Et, O, O, NHMe], [AI 5096; H, H, Et, H, O, F, H, H, c-Pr, O , O, NHMe], [AI 5097; H, H, Et, H, O, F, H, OMe, O, O, NH Me], [AI 5098; H, H, Et, H, O, F, H , H, OEt, O, O, NHMe], [AI 5099; H, H, Et, H, O, F, H, S, S, O, O, NHMe], [AI 5100; H, H, Et, H , O, F, H, H, CF ₃ , O, O, NHMe],

[AI5101; Cl, H, Et, H, O, F, H, H, H, O, O, NHMe], [AI 5102; Cl, H, Et, H, O, F, H, H, F, O , O, NHMe], [AI 5103; Cl, H, Et, H, O, F, H, H, Cl, O, NH Me], [AI 5104; Cl, H, Et, H, O, F, H , H, Br, O, O, NHMe], [AI 5105; Cl, H, Et, H, O, F, H, I, O, O, NHMe], [AI 5106; Cl, H, Et, H , O, F, H, H, Me, O, O, NHMe], [AI 5107; Cl, H, Et, H, O, F, H, Et, O, O, NHMe], [AI 5108; Cl , H, Et, H, O, F, H, H, c-Pr, O, O, NHMe], [AI 5109; Cl, H, Et, H, O, F, H, OMe, O, O , NHMe], [AI5110; Cl, H, Et, H, O, F, H, OEt, O, O, NHMe], [AI 5111; Cl, H, Et, H, O, F, H, H , SMe, O, O, NHMe ], [AI5112; Cl, H, Et, H, O, F, H, H, CF 3, O, O, NHMe], [AI5113; Me, H, Et, H, O, F, H, H, H, H, O, O, NHMe], [AI 5114; Me, H, Et, H, O, F, H, F, O, O, NHMe], [AI 5115; Me, H, Et, H, O, F, H, H, H, Cl, O, O, NHMe], [AI 5116; Me, H, Et, H, O, F, H, H, Br, O, O, NHMe] , [AI5117; Me, H, Et, H, O, F, H, I, O, O, NHMe], [AI 5118; Me, H, Et, H, O, F, H, H, Me, O, O, NHMe], [AI5119; Me, H, Et, H, O, F, H, H, Et, O, O, NHMe], [AI 5120; Me, H, Et, H, O, F, H, H, c-Pr, O, O, NHMe], [AI5121; Me, H, Et, H, O, F, H, H, OMe, O, O, NHMe], [AI5122; Me, H, Et, H, O, F, H, H, OEt, O, O, NHMe], [AI 5123; Me, H, Et, H, O, F, H, H, SMe, O, O, NHMe], [ AI5124; Me, H, Et, H, O, F, H, H, CF 3, O, O, NHMe], [AI5125; Et, H, Et, H, O, F, H, H, H, O , O, NHMe], [AI 5126; Et, H, Et, H, O, F, H, H, F, O, O, NHMe], [AI 5127; Et, H, Et, H, O, F, H, Cl, O, O, NHMe], [AI 5128; Et, H, Et, H, O, F, H, H, Br, O, O, NHMe], [AI 5129; Et, H, Et, H, O, F, H, I, O, O, NH Me], [AI 5130; Et, H, Et, H, O, F, H, Me, O, O, NH Me], [AI 5131; Et, H, Et, H, O, F, H, H, Et, O, O, NHMe], [AI 5132; Et, H, Et, H, O, F, H, c, Pr, O, O, NHMe], [AI 5133; Et, H, Et, H, O, F, H, H, OMe, O, O, NHMe], [AI 5134; Et, H, Et, H, O, F, H, OE, O, O, NHMe], [AI 5 135; Et, H, Et, H, O, F, H, H, SMe, O, O, NHMe], [AI5136; Et, H, Et, H, O, F, H, H, CF 3, O, O, NHMe ], [AI 5137; H, H, H, H, H, O, H, F, H, H, O, O, NHMe], [AI 5138; H, H, H, H, O, H, F, H, F] , O, O, NHMe], [AI 5139; H, H, H, H, H, O, H, H, F, H, Cl, O, O, NH Me], [AI 5140; H, H, H, H, O, H , F, H, Br, O, O, NHMe], [AI5141; H, H, H, H, H, O, H, F, H, I, O, O, NHMe], [AI5142; H, H, H , H, O, H, F, H, Me, O, O, NHMe], [AI 5143; H, H, H, H, H, O, H, F, H, Et, O, O, NHMe], [AI 5144 H, H, H, H, H, O, H, F, H, c-Pr, O, O, NHMe], [AI 5145; H, H, H, H, O, H, F, H, OMe, O H, H, H, H, H, O, H, F, H, OEt, O, O, NHMe], [AI 5147; H, H, H, H, O, H, F , H, SMe, O, O , NHMe], [AI5148; H, H, H, H, O, H, F, H, CF 3, O, O, NHMe], [AI5149; Cl, H, H, H, O, H, F, H, H, H, O, O, NHMe], [AI 5150; Cl, H, H, H, H, O, H, F, H, F, O, O, NHMe], [AI 5151; Cl, H, H, H, H, O, H, F, H, Cl, O, O, NHMe], [AI 5152; Cl, H, H, H, H, O, H , F, H, Br, O, O, NHMe], [AI 5153; Cl, H, H, H, H, O, H, F, H, I, O, O, NHMe], [AI 5154; Cl, H, H , H, O, H, F, H, Me, O, O, NHMe], [AI 5 155; Cl, H, H, H, H, O, H, F, H, Et, O, O, NHMe], [AI 5156 Cl, H, H, H, H, O, H, F, H, c-Pr, O, O, NHMe], [AI 5157; Cl, H, H, H, H, O, H, F, H, OMe, O , O, NHMe], [AI5158; Cl, H, H, H, H, O, H, F, H, OEt, O, O, NHMe], [AI 5159; Cl, H, H, H, O, H, F , H, SMe, O, O , NHMe], [AI5160; Cl, H, H, H, O, H, F, H, CF 3, O, O, NHMe], [AI5161; Me, H, H, H, O, H, F, H, H, H, O, O, NHMe], [AI5162; Me, H, H, H, H, O, H, F, H, F, O, O, NHMe], [AI5163; Me, H, H, H, H, O, H, F, H, Cl, O, NH, NHMe], [AI 5164; Me, H, H, H, H, O, H, F, H, Br, O, O, NHMe], [AI5165; Me, H, H, H, O, H, F, H, I, O, O, NHMe], [AI 5166; Me, H, H, H, O, H, F, H, Me, O, O, NHMe], [AI5167; Me, H, H, H, H, O, H, F, H, Et, O, O, NHMe], [AI 5168; Me, H, H, H, O, H, F, H, c-Pr, O, O, NHMe], [AI 5169; Me, H, H, H, H, O, H, F, H, OMe, O, O, NHMe], [AI 5170; H, H, H, H, O, H, F, H, OEt, O, O, NHMe], [AI 5171; Me, H, H, H, O, H, F, H, SMe, O, O, NHMe] , [AI5172; Me, H, H, H, O, H, F, H, CF 3, O, O, NHMe], [AI5173; Et, H, H, H, O, H, F, H, H , O, O, NHMe], [AI 5174; Et, H, H, H, H, O, H, F, H, F, F, O, O, NH Me], [AI 5175; Et, H, H, H, O, H , F, H, Cl, O, O, NHMe], [AI 5176; Et, H, H, H, H, O, H, F, H, Br, O, O, NHMe], [AI 5177; Et, H, H , H, O, H, F, H, I, O, O, NHMe], [AI 5178; Et, H, H, H, O, H, F, H, Me, O, O, NHMe], [AI 5179; Et, H, H, H, H, O, H, F, H, Et, O, O, NHMe], [AI 5 180; Et, H, H, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5181; Et, H, H, H, H, O, H, F, H, OMe, O, O, NHMe], [AI5182; Et, H, H, H, H, O, H, F, H, OEt, O, O, NHMe], [AI 5183; Et, H, H, H, O, H, F, H, SMe, O, O, NHMe], [AI5184; Et, H, H, H, O, H, F, H, CF 3, O, O, NHMe], [AI5185; H, H, F, H, O, H, F, H , H, O, O, NHMe], [AI 5186; H, H, F, H, O, H, F, H, F, O, O, NHMe], [AI 5187; H, H, F, H, O , H, F, H, Cl, O, O, NHMe], [AI 5188; H, H, F, H, O, H, F, H, Br, O, O, NHMe], [AI 5189; H, H , F, H, O, H, F, H, I, O, O, NHMe], [AI 5190; H, H, F, H, O, H, F, H, Me, O, O, NHMe], [AI5191; H, H, F, H, O, H, F, H, Et, O, O, NHMe], [AI5192; H, H, F, H, O, H, F, H, c-Pr , O, O, NHMe], [AI5193; H, H, F, H, O, H, F, H, OMe, O, O, NHMe], [AI 5194; H, H, F, H, O, H , F, H, OEt, O, O, NHMe], [AI 5195; H, H, F, H, O, H, F, H, SMe, O, O, NHMe], [AI 5196; H, H, F , H, O, H, F , H, CF 3, O, O, NHMe], [AI5197; Cl, H, F, H, O, H, F, H, H, O, O, NHMe], [ AI 5198; Cl, H, F, H, O, H, F, H, F, O, O, NHMe], [AI 5199; Cl, H, F, H, O, H, F, H, Cl, O, O, NHMe], [AI 5200; Cl, H, F, H, O, H, F, H, Br, O, O, NHMe],

[AI5201; Cl, H, F, H, O, H, F, H, I, O, O, NHMe], [AI 5202; Cl, H, F, H, O, H, F, H, Me, O , O, NHMe], [AI 5203; Cl, H, F, H, O, H, F, H, Et, O, O, NHMe], [AI 5204; Cl, H, F, H, O, H, F , H, c-Pr, O, O, NHMe], [AI 5205; Cl, H, F, H, O, H, F, H, OMe, O, O, NHMe], [AI 5206; Cl, H, F , H, O, H, F, H, OEt, O, O, NHMe], [AI 5207; Cl, H, F, H, O, H, F, H, SMe, O, O, NHMe], [AI 5208 ; Cl, H, F, H , O, H, F, H, CF 3, O, O, NHMe], [AI5209; Me, H, F, H, O, H, F, H, H, O, O, NHMe], [AI 5210; Me, H, F, H, O, H, F, H, F, O, O, NH Me], [AI 5211; Me, H, F, H, O, H, F, H, Cl, O, O, NHMe], [AI 5212; Me, H, F, H, O, H, F, H, H, Br, O, O, NHMe], [AI 5213; Me, H, F, H, O, H, F, H, I, O, O, NHMe], [AI 5214; Me, H, F, H, O, H, F, H, Me, O, O, NHMe], [AI 5215; H, F, H, O, H, F, H, Et, O, O, NHMe], [AI 5216; Me, H, F, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5217; Me, H, F, H, O, H, F, H, OMe, O, O, NHMe], [AI 5218; Me, H, F, H, O, H, F, H, OEt, O, O, NHMe], [AI5219; Me, H, F, H, O, H, F, H, S, SMe, O, O, NHMe], [AI 5220; Me, H, F, H, O, _{H, F, H, CF 3} , O, O, NHMe], [AI5221; Et, H, F, H, O, H, F, H, H, O, O, NHMe], [AI5222; Et, H , F, H, O, H, F, H, F, O, O, NHMe], [AI 5223; Et, H, F, H, O, H, F, H, Cl, O, O, NHMe], [AI 5224; Et, H, F, H, O, H, F, H, Br, O, O, NHMe], [AI 5225; Et, H, F, H, O, H, F, H, I, O , O, NHMe], [AI5226; Et, H, F, H, O, H, F, H, Me, O, O, NHMe], [AI 5227; Et, H, F, H, O, H, F, H, Et, O, O, NHMe], [AI 5228; Et, H, F, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5229; Et, H, F, H, O, H, F, H, OMe, O, O, NHMe], [AI 5230; Et, H, F, H, O, H, F, H, OEt, O, O, NHMe], [AI5231; Et, H, F, H, O, H, F, H, SMe, O, O, NHMe], [AI5232; Et, H, F, H, O, H, F, H, CF 3, O, O, NHMe], [AI5233; H, H, Cl, H, O, H, F, H, H, O, O, NHMe], [AI5234 H, H, Cl, H, O, H, F, H, F, F, O, O, NHMe], [AI 5235; H, H, Cl, H, O, H, F, H, Cl, O, O , NHMe], [AI5236; H, H, Cl, H, O, H, F, H, Br, O, O, NHMe], [AI 5237; H, H, Cl, H, O, H, F, H H, H, Cl, H, O, H, H, F, H, Me, O, O, NHMe], [AI 5239; H, H, Cl, H, O, I, O, O, NHMe], [AI 5238; , H, F, H, Et, O, O, NHMe], [AI5240; H, H, Cl, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5241; H , H, Cl, H, O, H, F, H, OMe, O, O, NHMe], [AI5242; H, H, Cl, H, O, H, F, H, OEt, O, O, NHMe H, H, Cl, H, O, H, F, H, SMe, O, O, NHMe], [AI 5244; H, H, Cl, H, O, H, F, H, CF] ₃ , O, O, NHMe], [AI 5245; Cl, H, Cl, H, O, H, F, H, H, O, O, NHMe], [AI 5246; Cl, H, Cl, H, O, H, F, H, F, O, O, NHMe], [AI 5247; Cl, H, Cl, H, O, H, F, H, Cl, O, O, NHMe], [AI 5248; Cl, H, Cl, H, O, H, F, H, Br, O, O, NHMe], [AI 5249; Cl, H, Cl, H, O, H, F, H, I, O, O, NHMe], [ AI 5250; Cl, H, Cl, H, O, H, F, H, Me, O, O, NHMe], [AI 5251; Cl, H, Cl, H, O, H, F, H, Et, O, O, NHMe], [AI 5252; Cl, H, Cl, H, O, H, F, H, c-Pr, O, O, N HMe], [AI 5253; Cl, H, Cl, H, O, H, F, H, OMe, O, O, NHMe], [AI 5254; Cl, H, Cl, H, O, H, F, H, OEt, O, O, NHMe], [AI 5255; Cl, H, Cl, H, O, H, H, F, H, SMe, O, O, NHMe], [AI 5 256; Cl, H, Cl, H, O, _{H, F, H, CF 3} , O, O, NHMe], [AI5257; Me, H, Cl, H, O, H, F, H, H, O, O, NHMe], [AI5258; Me, H , Cl, H, O, H, F, H, F, O, O, NHMe], [AI 5259; Me, H, Cl, H, O, H, F, H, Cl, O, O, NHMe], [AI5260; Me, H, Cl, H, O, H, F, H, Br, O, O, NHMe], [AI5261; Me, H, Cl, H, O, H, F, H, I, O , O, NHMe], [AI5262; Me, H, Cl, H, O, H, F, H, Me, O, O, NHMe], [AI 5263; Me, H, Cl, H, O, H, F , H, Et, O, O, NHMe], [AI5264; Me, H, Cl, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5265; Me, H, Cl , H, O, H, F, H, OMe, O, O, NHMe], [AI5266; Me, H, Cl, H, O, H, F, H, OEt, O, O, NHMe], [AI5267 ; Me, H, Cl, H , O, H, F, H, SMe, O, O, NHMe], [AI5268; Me, H, Cl, H, O, H, F, H, CF 3, O, O, NHMe], [AI5269; Et, H, Cl, H, O, H, F, H, H, O, O, NHMe], [AI 5270; Et, H, Cl, H, O, H, F, H, F, O, O, NHMe], [AI5271; Et, H, Cl, H, O, H, F, H, H, Cl, O, O, NHMe], [AI5272; Et, H, Cl, H, O, H, F, H, Br, O, O, NHMe], [AI 5273; Et, H, Cl, H, O, H, F, H, I, O, O, NHMe], [AI 5274; Et, H, Cl, H, O, H, F, H, Me, O, O, NHMe], [AI 5275; Et, H, Cl, H, O, H, F, H, Et, O, O, NHMe] , [AI5276; Et, H, Cl, H, O, H, F, H, c-Pr, O, O, NHMe], [AI 5277; Et, H, Cl, H, O, H, F, H, OMe, O, O, NHMe], [AI5278; E t, H, Cl, H, O, H, F, H, OEt, O, O, NHMe], [AI 5279; Et, H, Cl, H, O, H, F, H, SMe, O, O, NHMe], [AI5280; Et, H, Cl, H, O, H, F, H, CF 3, O, O, NHMe], [AI5281; H, H, Me, H, O, H, F, H , H, O, O, NHMe], [AI5282; H, H, Me, H, O, H, F, H, F, O, O, NHMe], [AI 5283; H, H, Me, H, O , H, F, H, Cl, O, O, NHMe], [AI 5284; H, H, Me, H, O, H, F, H, Br, O, O, NHMe], [AI 5285; H, H , Me, H, O, H, F, H, I, O, O, NHMe], [AI 5286; H, H, Me, H, O, H, F, H, Me, O, O, NHMe], [AI5287; H, H, Me, H, O, H, F, H, Et, O, O, NHMe], [AI 5288; H, H, Me, H, O, H, F, H, c-Pr , O, O, NHMe], [AI5289; H, H, Me, H, O, H, F, H, OMe, O, O, NHMe], [AI 5290; H, H, Me, H, O, H , F, H, OEt, O, O, NHMe], [AI 5291; H, H, Me, H, O, H, F, H, SMe, O, O, NHMe], [AI 5292; H, H, Me , H, O, H, F , H, CF 3, O, O, NHMe], [AI5293; Cl, H, Me, H, O, H, F, H, H, O, O, NHMe], [ AI 5294; Cl, H, Me, H, O, H, F, H, F, O, O, NHMe], [AI 5295; Cl, H, Me, H, O, H, F, H, Cl, O, O, NHMe], [AI5296; Cl, H, Me, H, O, H, F, H, H, Br, O, O, NHMe], [AI 5297; Cl, H, Me, H, O, H, F, H, I, O, O, NHMe], [AI5298; Cl, H, Me, H, O, H, F, H, Me, O, O, NHMe], [AI5299; Cl, H, Me, H, O, H, F, H, Et, O, O, NHMe], [AI 5300; Cl, H, Me, H, O, H, F, H, c-Pr, O, O, NHMe],

[AI 5301; Cl, H, Me, H, O, H, F, H, OMe, O, O, NH Me], [AI 5302; Cl, H, Me, H, O, H, F, H, OE t, O , O, NHMe], [AI 5303; Cl, H, Me, H, O, H, F, H, SMe, O, O, NHMe], [AI 5304; Cl, H, Me, H, O, H, F _{, H, CF 3, O,} O, NHMe], [AI5305; Me, H, Me, H, O, H, F, H, H, O, O, NHMe], [AI5306; Me, H, Me, H, O, H, F, H, F, F, O, O, NHMe], [AI 5307; Me, H, Me, H, O, H, F, H, Cl, O, O, NHMe], [AI 5308; Me, H, Me, H, O, H, F, H, Br, O, O, NHMe], [AI 5309; Me, H, Me, H, O, H, F, H, I, O, O, NHMe], [AI 5310; Me, H, Me, H, O, H, F, H, Me, O, O, NH Me], [AI 5311; Me, H, Me, H, O, H, F, H, Et, O, O, NHMe], [AI5312; Me, H, Me, H, O, H, F, H, c, Pr, O, O, NHMe], [AI5313; Me, H, Me, H, O, H, F, H, OMe, O, O, NHMe], [AI5314; Me, H, Me, H, O, H, F, H, OEt, O, O, NHMe], [AI 5315; Me, H, Me, H, O, H, F, H, SMe, O, O, NHMe], [AI5316; Me, H, Me, H, O, H, F, H, CF 3, O, O, NHMe ], [AI 5317; Et, H, Me, H, O, H, F, H, H, O, O, NH Me], [AI 5318; Et, H, Me, H, O, H, F, H, F , O, O, NHMe], [AI 5319; Et, H, Me, H, O, H, H, F, H, Cl, O, NH, Me], [AI 5320; Et, H, Me, H, O, H , F, H, Br, O, O, NHMe], [AI5321; Et, H, Me, H, O, H, F, H, I, O, O, NHMe], [AI5322; Et, H, Me , H, O, H, F, H, Me, O, O, NHMe], [AI 5323; Et, H, Me, H, O, H, F, H, Et, O, O, NHMe], [AI 5324 Et, H, Me, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5325; Et, H, Me, H, O, H, F, H, OMe, O , O, NHMe], [AI 5326; Et, H, M e, H, O, H, F, H, OEt, O, O, NHMe], [AI 5327; Et, H, Me, H, O, H, F, H, SMe, O, O, NHMe], [ AI5328; Et, H, Me, H, O, H, F, H, CF 3, O, O, NHMe], [AI5329; H, H, Et, H, O, H, F, H, H, O , O, NHMe], [AI 5330; H, H, Et, H, O, H, F, H, F, O, O, NH Me], [AI 5331; H, H, Et, H, O, H, F H, Cl, O, O, NHMe], [AI5332; H, H, Et, H, O, H, F, H, Br, O, O, NHMe], [AI 5333; H, H, Et, H , O, H, F, H, I, O, O, NHMe], [AI 5334; H, H, Et, H, O, H, F, H, Me, O, O, NHMe], [AI 5335; H , H, Et, H, O, H, F, H, Et, O, O, NHMe], [AI 5336; H, H, Et, H, O, H, F, H, c-Pr, O, O , NHMe], [AI 5337; H, H, Et, H, O, H, F, H, OMe, O, O, NH Me], [AI 5338; H, H, Et, H, O, H, F, H , OEt, O, O, NHMe], [AI5339; H, H, Et, H, O, H, F, H, SMe, O, O, NHMe], [AI5340; H, H, Et, H, O , H, F, H, CF 3, O, O, NHMe], [AI5341; Cl, H, Et, H, O, H, F, H, H, O, O, NHMe], [AI5342; Cl, H, Et, H, O, H, F, H, F, F, O, O, NHMe], [AI 5343; Cl, H, Et, H, O, H, F, H, Cl, O, O, NHMe] , [AI 5344; Cl, H, Et, H, O, H, F, H, Br, O, O, NHMe], [AI 5345; Cl, H, Et, H, O, H, F, H, I, O, O, NHMe], [AI5346; Cl, H, Et, H, O, H, F, H, Me, O, O, NHMe], [AI 5347; Cl, H, Et, H, O, H, F, H, Et, O, O, NH, Me: [AI 5348; Cl, H, Et, H, O, H, F, H, c, Pr, O, O, NHMe], [AI 5349; Cl, H, Et, H, O, H, F, H, OMe, O, O, NHMe], [AI 5350; Cl, H, Et, H, O, H, F, H, OEt, O, O, NHMe], [ AI 5351; Cl, H, Et, H, O, H, F, H, SMe, O, O, NHMe], [AI5352; Cl, H, Et , H, O, H, F, H, CF 3, O, O, NHMe], [AI5353; Me, H, Et, H, O, H, F, H, H, O, O, NHMe], [AI 5354; Me, H, Et, H, O, H, F, H, F, O, O, NH Me], [AI 5 355; Me, H, Et, H, O, H, F, H, Cl, O, O, NHMe], [AI 5356; Me, H, Et, H, O, H, F, H, Br, O, O, NHMe], [AI 5357; Me, H, Et, H, O, H, F, H, I, I, O, O, NHMe], [AI 5358; Me, H, Et, H, O, H, F, H, Me, O, O, NHMe], [AI 5359; Me, H, Et, H, O, H, F, H, Et, O, O, NHMe], [AI 5360; Me, H, Et, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5361; Me, H, Et, H, O, H, F, H, OMe, O, O, NHMe], [AI5362; Me, H, Et, H, O, H, F, H, OEt, O, O, NHMe], [AI5363; Me, H, Et, H, O, H, F, H, SMe, O, O, NHMe], [AI5364; Me, H, Et, H, O, H, F, H, CF 3, O, O, NHMe], [AI5365; Et, H, Et, H, O, H, F, H, H, O, O, NHMe], [AI5366; Et , H, Et, H, O, H, F, H, F, O, O, NHMe], [AI 5367; Et, H, Et, H, O, H, F, H, Cl, O, O, NHMe ], [AI5368; Et, H, Et, H, O, H, F, H, Br, O, O, NHMe], [AI5369; Et, H, Et, H, O, H, F, H, I , O, O, NHMe], [AI5370; Et, H, Et, H, O, H, H, F, H, Me, O, O, NHMe], [AI5371; Et, H, Et, H, O, H , F, H, Et, O, O, NHMe], [AI5372; Et, H, Et, H, O, H, F, H, c-Pr, O, O, NHMe], [AI5373, Et, H , Et, H, O, H, F, H, OMe, O, O, NHMe], [AI 5374; Et, H, Et, H, O, H, F, H, OEt, O, O, NHMe], [AI 5375; Et, H, Et, H, O, H, F, H, SMe, O, O, NH, Me], [AI 5376; Et, H, Et, H, O, H, F, H, CF ₃ , O, O, NHMe], [AI5377; H, H, H, H, O, H, H, F, H, O, O, NHMe], [AI 5378; H, H, H, H, O, H, F, F, O, O, NHMe], [ AI 5379; H, H, H, H, H, O, H, H, F, Cl, O, NHMe], [AI 5380; H, H, H, H, H, O, H, F, Br, O, O, NHMe], [AI5381; H, H, H, H, O, H, H, F, I, O, O, NHMe], [AI5382; H, H, H, H, O, H, H, F, Me, O, O, NHMe], [AI5383; H, H, H, H, H, O, H, H, F, Et, O, O, NHMe], [AI 5384; H, H, H, H, O, H, H, F, c-Pr, O, O, NHMe], [AI5385; H, H, H, H, H, O, H, H, F, OMe, O, O, NHMe], [AI5386; H, H, H, H, H, O, H, H, F, OEt, O, O, NHMe], [AI 5387; H, H, H, H, O, H, H, F, SMe, O, O, NHMe], [AI5388; H, H, H, H, O, H, H, F, CF 3, O, O, NHMe], [AI5389; Cl, H, H, H, O, H, H, F , H, O, O, NHMe], [AI5390; Cl, H, H, H, H, O, H, H, F, F, O, O, NHMe], [AI5391; Cl, H, H, H, O , H, H, F, Cl, O, O, NHMe], [AI5392; Cl, H, H, H, H, O, H, H, F, Br, O, O, NHMe], [AI5393; Cl, H , H, H, O, H, H, F, I, O, O, NHMe], [AI5394; Cl, H, H, H, O, H, F, Me, O, O, NHMe], [AI5395; Cl, H, H, H, H, O, H, H, F, Et, O, O, NHMe], [AI 5396; Cl, H, H, H, O, H, H, F, c-Pr , O, O, NHMe], [AI5397; Cl, H, H, H, H, O, H, H, F, OMe, O, O, NHMe], [AI5398; Cl, H, H, H, O, H , H, F, OEt, O, O, NHMe], [AI5399; Cl, H, H, H, H, O, H, F, SMe, O, O, NHMe], [AI 5400; Cl, H, H , H, O, H, H, F, CF ₃ , O, O, NHMe],

[AI5401; Me, H, H, H, H, O, H, H, F, H, O, O, NHMe], [AI 5402; Me, H, H, H, O, H, H, F, F, O , O, NHMe], [AI5403; Me, H, H, H, H, O, H, H, F, Cl, O, NH, Me], [AI 5404; Me, H, H, H, O, H, H , F, Br, O, O, NHMe], [AI 5405; Me, H, H, H, H, O, H, H, F, I, O, O, NHMe], [AI 5406; Me, H, H, H , O, H, H, F, Me, O, O, NHMe], [AI 5407; Me, H, H, H, H, O, H, H, F, Et, O, O, NHMe], [AI 5408; Me , H, H, H, O, H, H, F, c-Pr, O, O, NHMe], [AI 5409; Me, H, H, H, O, H, F, O, O, O , NHMe], [AI 5410; Me, H, H, H, O, H, H, F, OEt, O, O, NH Me], [AI 5411; Me, H, H, H, O, H, H, F , SMe, O, O, NHMe ], [AI5412; Me, H, H, H, O, H, H, F, CF 3, O, O, NHMe], [AI5413; Et, H, H, H, O, H, H, H, F, H, O, O, NHMe], [AI 5414; Et, H, H, H, H, O, H, H, F, F, O, O, NHMe], [AI 5415; Et, H, H, H, H, O, H, H, F, F, Cl, O, O, NHMe], [AI 5416; Et, H, H, H, H, O, H, F, Br, O, O, NHMe] [AI 5417; Et, H, H, H, H, O, H, H, F, I, O, O, NHMe], [AI 5418; Et, H, H, H, O, H, H, F, Me, O, O, NHMe], [AI 5419; Et, H, H, H, H, O, H, H, H, F, Et, O, O, NH Me], [AI 5420; Et, H, H, H, O, H, H, F, c-Pr, O, O, NHMe], [AI 5421; Et, H, H, H, H, O, H, H, F, OMe, O, O, NHMe], [AI 542; Et, H, H, H, O, H, H, F, OEt, O, O, NHMe], [AI 5423; Et, H, H, H, H, O, H, F, SMe, O, O, NHMe], [ AI5424; Et, H, H, H, O, H, H, F, CF 3, O, O, NHMe], [AI5425; H, H, F, H, O, H, H, F, H, O , O, NHMe], [AI5426; H, H, F, H, O, H, H, F, F, O, O, NHMe], [AI 542 7; H, H, F, H, O, H, H, F, Cl, O, NHMe], [AI5428; H, H, F, H, O, H, H, F, Br, O, O, NHMe], [AI5429; H, H, F, H, O, H, H, F, I, O, O, NHMe], [AI 5430; H, H, F, H, O, H, H, F, Me, O, O, NHMe], [AI5431; H, H, F, H, O, H, H, F, Et, O, O, NHMe], [AI5432; H, H, F, H, O, H, H, F, c-Pr, O, O, NHMe], [AI5433; H, H, F, H, O, H, H, F, OMe, O, O, NHMe], [AI 5434; H, H, F, H, O, H, H, F, OEt, O, O, NHMe], [AI 5435; H, H, F, H, O, H, H, F, SMe, O, O, NHMe], [AI5436; H, H, F, H, O, H, H, F, CF 3, O, O, NHMe], [AI5437; Cl, H, F, H, O, H, H, F , H, O, O, NHMe], [AI5438; Cl, H, F, H, O, H, H, F, F, O, O, NHMe], [AI5439; Cl, H, F, H, O , H, H, F, Cl, O, O, NHMe], [AI 5440; Cl, H, F, H, O, H, H, F, Br, O, O, NHMe], [AI5441; Cl, H , F, H, O, H, H, F, I, O, O, NHMe], [AI5442; Cl, H, F, H, O, H, F, Me, O, O, NHMe], [AI5443; Cl, H, F, H, O, H, H, F, Et, O, O, NHMe], [AI5444; Cl, H, F, H, O, H, H, F, c-Pr , O, O, NHMe], [AI5445; Cl, H, F, H, O, H, H, F, OMe, O, O, NHMe], [AI5446; Cl, H, F, H, O, H , H, F, OEt, O, O, NHMe], [AI5447; Cl, H, F, H, O, H, H, F, SMe, O, O, NHMe], [AI 5448; Cl, H, F , H, O, H, H , F, CF 3, O, O, NHMe], [AI5449; Me, H, F, H, O, H, H, F, H, O, O, NHMe], [ AI5450; Me, H, F, H, O, H, H, F, F, O, NH, NHMe], [AI5451; Me, H, F, H, O, H, H, F, Cl, O, O, NHMe], [AI5452; Me, H, F, H, O, H, H, F, Br, O, O, NHMe], [AI5453; Me, H, F, H, O , H, H, F, I, O, O, NHMe], [AI 5454; Me, H, F, H, O, H, H, F, Me, O, O, NHMe], [AI 5455; Me, H , F, H, O, H, H, F, Et, O, O, NHMe], [AI 5456; Me, H, F, H, O, H, F, c, Pr, O, O, NHMe Me, H, F, H, O, H, H, F, OMe, O, O, NHMe], [AI 5458; Me, H, F, H, O, H, H, F, OEt] , O, O, NHMe], [AI5459; Me, H, F, H, O, H, H, F, SMe, O, O, NHMe], [AI 5460; Me, H, F, H, O, H _{, H, F, CF 3,} O, O, NHMe], [AI5461; Et, H, F, H, O, H, H, F, H, O, O, NHMe], [AI5462; Et, H, F, H, O, H, H, F, F, O, O, NHMe], [AI5463; Et, H, F, H, O, H, F, Cl, O, O, NHMe], [ AI 5464; Et, H, F, H, O, H, H, F, Br, O, NH, NHMe], [AI 5465; Et, H, F, H, O, H, H, F, I, O, O, NHMe], [AI5466; Et, H, F, H, O, H, H, F, Me, O, O, NHMe], [AI 5467; Et, H, F, H, O, H, H, F, Et, O, O, NHMe], [AI5468; Et, H, F, H, O, H, H, F, c-Pr, O, O, NHMe], [AI 5469; Et, H, F, H, O, H, H, F, OMe, O, O, NHMe], [AI5470; Et, H, F, H, O, H, H, F, OEt, O, O, NHMe], [AI5471; Et, H, F, H, O, H, H, F, SMe, O, O, NHMe], [AI5472; Et, H, F, H, O, H, H, F, CF 3, O, O , NHMe], [AI5473; H, H, Cl, H, O, H, H, F, H, O, O, NHMe], [AI 5474; H, H, Cl, H, O, H, H, F , F, O, O, NHMe], [AI 5475; H, H, Cl, H, O, H, H, F, Cl, O, O, NHMe], [AI 5476; H, H, Cl, H, O , H, H, F, Br, O, O, NHMe], [AI5477; H, H, Cl, H, O, H, H, F, I, O, O, NHMe], [AI5478; H, H , Cl, H, O, H, H, F, Me, O, O, NHMe], [AI5479; H, H, Cl, H, O, H, H, F, Et, O, O, NHMe], [AI5480; H, H, Cl, H, O, H, H, F, c-Pr, O, O, NHMe], [AI5481; H, H, Cl, H, O, H, H, F, OMe, O, O, NHMe], [AI 5482; H, H, Cl, H, O, H, H, F, OEt, O, O, NHMe], [ AI 5483; H, H, Cl, H, O, H, H, F, SMe, O, O, NHMe], [AI 5484; H, H, Cl, H, O, H, H, F, CF ₃ , O , O, NHMe], [AI 5485; Cl, H, Cl, H, O, H, H, F, H, O, O, NHMe], [AI 5486; Cl, H, Cl, H, O, H, H , F, F, O, O, NHMe], [AI 5487; Cl, H, Cl, H, O, H, H, F, Cl, O, NH, Me], [AI 5488; Cl, H, Cl, H , O, H, H, F, Br, O, O, NHMe], [AI5489; Cl, H, Cl, H, O, H, H, F, I, O, O, NHMe], [AI5490; Cl , H, Cl, H, O, H, H, F, Me, O, O, NHMe], [AI5491; Cl, H, Cl, H, O, H, H, F, Et, O, O, NHMe ], [AI5492; Cl, H, Cl, H, O, H, H, F, c, Pr, O, O, NHMe], [AI5493; Cl, H, Cl, H, O, H, H, F , OMe, O, O, NHMe], [AI5494; Cl, H, Cl, H, O, H, H, F, OEt, O, O, NHMe], [AI5495; Cl, H, Cl, H, O , H, H, F, SMe , O, O, NHMe], [AI5496; Cl, H, Cl, H, O, H, H, F, CF 3, O, O, NHMe], [AI5497; Me, H, Cl, H, O, H, H, F, H, O, O, NHMe], [AI 5498; Me, H, Cl, H, O, H, H, F, F, O, O, NHMe] , [AI5499; Me, H, Cl, H, O, H, H, F, Cl, O, NH, Me], [AI 5500; Me, H, Cl, H, O, H, H, F, Br, O, O, NHMe],

[AI 5501; Me, H, Cl, H, O, H, H, F, I, O, NH, Me], [AI 5502; Me, H, Cl, H, O, H, H, F, Me, O , O, NHMe], [AI5503; Me, H, Cl, H, O, H, H, F, Et, O, O, NHMe], [AI 5504; Me, H, Cl, H, O, H, H , F, c-Pr, O, O, NHMe], [AI 5505; Me, H, Cl, H, O, H, H, F, OMe, O, O, NHMe], [AI 5506; Me, H, Cl , H, O, H, H, F, OEt, O, O, NHMe], [AI 5507; Me, H, Cl, H, O, H, F, SMe, O, O, NHMe], [AI 5508 ; Me, H, Cl, H , O, H, H, F, CF 3, O, O, NHMe], [AI5509; Et, H, Cl, H, O, H, H, F, H, O, O, NHMe], [AI 5510; Et, H, Cl, H, O, H, H, F, F, O, O, NH Me], [AI 5511; Et, H, Cl, H, O, H, H, F, Cl, O, O, NHMe], [AI 5512; Et, H, Cl, H, O, H, H, H, F, Br, O, O, NHMe], [AI 5513; Et, H, Cl, H, O, H, H, H, F, I, O, O, NHMe], [AI 5514; Et, H, Cl, H, O, H, H, F, Me, O, O, NHMe], [AI 5515; Et, H, Cl, H, O, H, H, F, Et, O, O, NHMe], [AI 5516; Et, H, Cl, H, O, H, H, F, c-Pr, O, O, NHMe], [AI 5517; Et, H, Cl, H, O, H, H, F, OMe, O, O, NH Me], [AI 5518; Et, H, Cl, H, O, H, H, F, OEt, O, O, NHMe], [AI 5519; Et, H, Cl, H, O, H, H, F, SMe, O, O, NHMe], [AI 5520; Et, H, Cl, H, O, _{H, H, F, CF 3} , O, O, NHMe], [AI5521; H, H, Me, H, O, H, H, F, H, O, O, NHMe], [AI5522; H, H , Me, H, O, H, H, F, F, F, O, O, NHMe], [AI5523; H, H, Me, H, O, H, F, Cl, O, O, NHMe], [AI 5524; H, H, Me, H, O, H, H, F, Br, O, NH, NHMe], [AI 5525; H, H, Me, H, O, H, H, F, I, O , O, NHMe], [AI5526; H, H, Me, H, O, H, H, F, Me, O, O, NHMe], [AI5527; H, H, Me, H, O, H, H, F, Et, O, O, NHMe], [AI5528; H, H, Me, H, O, H, H, F, c, Pr, O, O, NHMe], [AI 5529; H, H, Me, H, O, H, H, F, OMe, O, O, NHMe], [ AI 5530; H, H, Me, H, O, H, H, F, OEt, O, O, NHMe], [AI5531; H, H, Me, H, O, H, H, F, SMe, O, O, NHMe], [AI5532; H, H, Me, H, O, H, H, F, CF 3, O, O, NHMe], [AI5533; Cl, H, Me, H, O, H, H , F, H, O, O, NHMe], [AI 5534; Cl, H, Me, H, O, H, H, F, F, O, NH, Me], [AI 5535; Cl, H, Me, H , O, H, H, F, Cl, O, O, NHMe], [AI 5536; Cl, H, Me, H, O, H, H, F, Br, O, O, NHMe], [AI 5537; Cl , H, Me, H, O, H, H, F, I, O, NHMe], [AI 5538; Cl, H, Me, H, O, H, H, F, Me, O, O, NHMe ], [AI 5539; Cl, H, Me, H, O, H, H, F, Et, O, O, NH Me], [AI 5540; Cl, H, Me, H, O, H, H, F, c -Pr, O, O, NHMe], [AI5541; Cl, H, Me, H, O, H, H, F, OMe, O, O, NHMe], [AI5542; Cl, H, Me, H, O , H, H, F, OEt, O, O, NHMe], [AI5543; Cl, H, Me, H, O, H, H, F, SMe, O, O, NHMe], [AI5544; Cl, H , Me, H, O, H , H, F, CF 3, O, O, NHMe], [AI5545; Me, H, Me, H, O, H, H, F, H, O, O, NHMe] , [AI5546; Me, H, Me, H, O, H, H, F, F, O, O, NHMe], [AI 5547; Me, H, Me, H, O, H, H, F, Cl, O, O, NHMe], [AI5548; Me, H, Me, H, O, H, H, F, Br, O, O, NHMe], [AI5549; Me, H, Me, H, O, H, H, F, I, O, O, NHMe], [AI 5550; Me, H, Me, H, O, H, H, F, Me, O, O, NHMe], [AI5551; Me, H, Me, H, O, H, H, F, Et, O, O, NHMe], [AI5 552; Me, H, Me, H, O, H, H, F, c-Pr, O, O, NHMe], [AI5553; Me, H, Me, H, O, H, H, F, OMe, O, O, NHMe], [AI5554; Me, H, Me, H, O, H, H, F, OEt, O, O, NHMe], [AI5555; Me, H, Me, H, O, H, H, F, SMe, O, O, NHMe], [AI5556; Me, H, Me, H, O, H, H, F, CF 3, O, O, NHMe], [AI5557; Et, H, Me , H, O, H, H, F, H, H, O, O, NHMe], [AI 5558; Et, H, Me, H, O, H, H, F, F, O, NH, Me], [AI 5559] Et, H, Me, H, O, H, H, F, Cl, O, NHMe], [AI 5560; Et, H, Me, H, O, H, H, F, Br, O, O , NHMe], [AI5561; Et, H, Me, H, O, H, H, F, I, O, O, NHMe], [AI5562; Et, H, Me, H, O, H, H, F , Me, O, O, NHMe], [AI5563; Et, H, Me, H, O, H, H, F, Et, O, O, NHMe], [AI 5564; Et, H, Me, H, O , H, H, F, c-Pr, O, O, NHMe], [AI5565; Et, H, Me, H, O, H, H, F, OMe, O, O, NHMe], [AI5566; Et , H, Me, H, O, H, H, F, OEt, O, O, NHMe], [AI 5567; Et, H, Me, H, O, H, H, F, SMe, O, O, NHMe ], [AI5568; Et, H , Me, H, O, H, H, F, CF 3, O, O, NHMe], [AI5569; H, H, Et, H, O, H, H, F, H, O, O, NHMe], [AI 5570; H, H, Et, H, O, H, H, F, F, O, O, NHMe], [AI 5571; H, H, Et, H, O, H, H, F, Cl, O, O, NHMe], [AI5572; H, H, Et, H, O, H, H, F, Br, O, NHMe], [AI5573; H, H, Et, H, O, H, H, F, I, O, NHMe], [AI 5574; H, H, Et, H, O, H, F, Me, O, O, NHMe], [ AI 5575; H, H, Et, H, O, H, H, F, Et, O, O, NHMe], [AI 5576; H, H, Et, H, O, H, H, F, c-Pr, O, O, NHMe], [AI 5577; H, H, Et, H, O, H, H, F, OMe, O, O, NHMe], [AI 5578; H, H, Et, H, O, H, H, F, OEt, O, O, NHMe], [AI 5579; H, H, Et, H, O, H, H, F, SMe, O, O, NHMe], [AI5580; H, H, Et, H, O, H, H, F, CF 3, O, O, NHMe], [AI5581; Cl, H , Et, H, O, H, H, F, H, O, O, NHMe], [AI5582; Cl, H, Et, H, O, H, H, F, F, O, O, NHMe], [AI 5583; Cl, H, Et, H, O, H, H, F, Cl, O, NHMe], [AI 5584; Cl, H, Et, H, O, H, H, F, Br, O , O, NHMe], [AI 5585; Cl, H, Et, H, O, H, H, H, F, I, O, O, NH Me], [AI 5586; Cl, H, Et, H, O, H, H , F, Me, O, O, NHMe], [AI 5587; Cl, H, Et, H, O, H, H, F, Et, O, O, NHMe], [AI 5588; Cl, H, Et, H , O, H, H, F, c-Pr, O, O, NHMe], [AI 5589; Cl, H, Et, H, O, H, F, OMe, O, O, NHMe], [AI 5590 Cl, H, Et, H, O, H, H, F, OEt, O, O, NHMe], [AI5591; Cl, H, Et, H, O, H, H, F, SMe, O, O , NHMe], [AI5592; Cl , H, Et, H, O, H, H, F, CF 3, O, O, NHMe], [AI5593; Me, H, Et, H, O, H, H, F, H, O, O, NHMe], [AI 5594; Me, H, Et, H, O, H, H, F, F, O, O, NHMe], [AI 5595; Me, H, Et, H, O, H, H, F, Cl, O, O, NHMe], [AI 5596; Me, H, Et, H, O, H, H, F, Br, O, O, NHMe], [AI 5597; Me, H, Et, H, O, H, H, F, I, O, NHMe], [AI 5598; Me, H, Et, H, O, H, H, F, Me, O, O, NHMe] , [AI5599; Me, H, Et, H, O, H, H, F, Et, O, O, NHMe], [AI 5600; Me, H, Et, H, O, H, H, F, c- Pr, O, O, NHMe],

[AI 5601; Me, H, Et, H, O, H, H, F, OMe, O, O, NHMe], [AI 5602; Me, H, Et, H, O, H, H, F, OEt, O , O, NHMe], [AI 5603; Me, H, Et, H, O, H, H, F, SMe, O, O, NHMe], [AI 5604; Me, H, Et, H, O, H, H _{, F, CF 3, O,} O, NHMe], [AI5605; Et, H, Et, H, O, H, H, F, H, O, O, NHMe], [AI5606; Et, H, Et, H, O, H, H, F, F, F, O, O, NHMe], [AI 5607; Et, H, Et, H, O, H, H, F, Cl, O, O, NHMe], [AI 5608; Et, H, Et, H, O, H, H, H, F, Br, O, NH, NHMe], [AI5609; Et, H, Et, H, O, H, H, F, I, O, O, NHMe], [AI 5610; Et, H, Et, H, O, H, H, F, Me, O, O, NH Me], [AI 5611; Et, H, Et, H, O, H, H, F, Et, O, O, NHMe], [AI 5612; Et, H, Et, H, O, H, H, F, c, Pr, O, O, NH Me], [AI 5613; Et, H, Et, H, O, H, H, F, OMe, O, O, NHMe], [AI 5614; Et, H, Et, H, O, H, H, F, OEt, O, O, NH Me], [AI 5615; Et, H, Et, H, O, H, H, F, SMe, O, O, NHMe], [AI5616; Et, H, Et, H, O, H, H, F, CF 3, O, O, NHMe H, H, H, H, O, H, H, H, H, S, O, NHMe], [AI 5618; H, H, H, H, O, H, H, H, F] , S, O, NHMe], [AI 5619; H, H, H, H, H, O, H, H, H, H, Cl, S, O, NH Me], [AI 5620; H, H, H, H, O, H , H, H, Br, S, O, NHMe], [AI5621; H, H, H, H, H, O, H, H, H, I, S, O, NHMe], [AI5622; H, H, H , H, O, H, H, H, H, Me, S, O, NHMe], [AI 5623; H, H, H, H, H, O, H, H, H, Et, S, O, NHMe], [AI 5624 H, H, H, H, H, O, H, H, H, c, Pr, S, O, NHMe], [AI 5625; H, H, H, H, O, H, H, H, OMe, S , O, NHMe], [AI 5626; H, H, H, H, O, H, H, H, OEt, S, O, NHMe], [AI5627; H, H, H, H, O, H, H, H, SMe, S, O, NHMe], [AI 5628; H, H, H, H, O, H, H, H, H, _{CF 3, S, O, NHMe} ], [AI5629; Cl, H, H, H, O, H, H, H, H, S, O, NHMe], [AI5630; Cl, H, H, H, O , H, H, H, H, F, S, O, NHMe], [AI5631; Cl, H, H, H, H, O, H, H, H, Cl, S, O, NHMe], [AI5632; Cl, H , H, H, O, H, H, H, H, Br, S, O, NHMe], [AI5633; Cl, H, H, H, O, H, H, H, I, S, O, NHMe], [AI 5634; Cl, H, H, H, H, O, H, H, Me, S, O, NHMe], [AI 5635; Cl, H, H, H, H, O, H, H, H, Et, S , O, NHMe], [AI 5636; Cl, H, H, H, H, O, H, H, H, c-Pr, S, O, NHMe], [AI 5637; Cl, H, H, H, O, H , H, H, OMe, S, O, NHMe], [AI5638; Cl, H, H, H, H, O, H, H, H, OEt, S, O, NHMe], [AI 5639; Cl, H, H , H, O, H, H , H, SMe, S, O, NHMe], [AI5640; Cl, H, H, H, O, H, H, H, CF 3, S, O, NHMe], [ AI 564 1; Me, H, H, H, H, O, H, H, H, S, O, NHMe], [AI 5642; Me, H, H, H, O, H, H, H, F, S, O, NHMe], [AI5643; Me, H, H, H, H, O, H, H, H, Cl, S, O, NHMe], [AI 5644; Me, H, H, H, O, H, H, H, Br, S, O, NHMe], [AI5645; Me, H, H, H, H, O, H, H, H, I, S, O, NHMe], [AI 5646; Me, H, H, H, O, H, H, H, H, Me, S, O, NHMe], [AI 5647; Me, H, H, H, H, O, H, H, H, Et, S, O, NHMe], [AI 5648; Me, H, H, H, H, O, H, H, H, c, Pr, S, O, NHMe], [AI 5649; Me, H, H, H, O, H, H, H, OMe, S, O, NHMe], [AI5650; Me, H, H, H, O, H, H, H, OEt, S, O, NHMe], [AI 5651; Me, H, H, H, O, H, H, H, H, SMe, S, O, NHMe] , [AI5652; Me, H, H, H, O, H, H, H, CF 3, S, O, NHMe], [AI5653; Et, H, H, H, H, O, H, H, H, H, S, O, NHMe], [AI5654; Et, H, H, H, O, H, H, H, H, F, S, O, NHMe], [AI5655; Et, H, H, H, H, O, H, H, H, H, Cl, S, O, NHMe], [AI 5656; Et, H, H, H, O, H, H, H, H, Br, S, O, NHMe], [AI5657; Et, H, H, H, H, O, H, H, H, I, S, O, NHMe], [AI5658; Et, H, H, H, O, H, H, H, Me, S, O, NHMe], [AI 5659; Et, H, H, H, O, H, H, H, Et, S, O, NHMe], [ AI 5660; Et, H, H, H, H, O, H, H, H, c-Pr, S, O, NHMe], [AI5661; Et, H, H, H, O, H, H, H, OMe, S, O, NHMe], [AI5662; Et, H, H, H, H, O, H, H, H, OEt, S, O, NHMe], [AI5663; Et, H, H, H, O, H, H, H, SMe, S, O, NHMe], [AI5664; Et, H, H, H, O, H, H, H, CF 3, S, O, NHMe], [AI5665; H, H, F , H, O, H, H, H, H, H, S, O, NHMe], [AI5666; H, H, F, H, O, H, H, H, F, S, O, NHMe], [AI5667 H, H, F, H, O, H, H, H, H, Cl, S, O, NHMe], [AI5668; H, H, F, H, O, H, H, H, Br, S, O , NHMe], [AI5669; H, H, F, H, O, H, H, I, S, O, NHMe], [AI 5670; H, H, F, H, O, H, H, H , Me, S, O, NHMe], [AI5671; H, H, F, H, O, H, H, H, Et, S, O, NHMe], [AI5672; H, H, F, H, O , H, H, H, c-Pr, S, O, NHMe], [AI5673; H, H, F, H, O, H, H, H, OMe, S, O, NHMe], [AI 5674; H , H, F, H, O, H, H, H, OEt, S, O, NHMe], [AI 5675; H, H, F, H, O, H, H, S, S, O, NHMe ], [AI5676; H, H , F, H, O, H, H, H, CF 3, S, O, NHMe], [AI5677; Cl, H, F, H, O, H, H, H, H, S, O, NHMe], [AI 5678; Cl, H, F, H, O, H, H, H, F, S, O, NHMe], [AI 5679; Cl , H, F, H, O, H, H, H, H, Cl, S, O, NHMe], [AI 5680; Cl, H, F, H, O, H, H, H, Br, S, O, NHMe ], [AI5681; Cl, H, F, H, O, H, H, H, I, S, O, NHMe], [AI5682; Cl, H, F, H, O, H, H, H, Me , S, O, NHMe], [AI5683; Cl, H, F, H, O, H, H, H, Et, S, O, NHMe], [AI5684; Cl, H, F, H, O, H , H, H, c-Pr, S, O, NHMe], [AI5685; Cl, H, F, H, O, H, H, H, OMe, S, O, NHMe], [AI 5686; Cl, H , F, H, O, H, H, H, OEt, S, O, NHMe], [AI5687; Cl, H, F, H, O, H, H, S, S, O, NHMe], [AI5688; Cl, H, F , H, O, H, H, H, CF 3, S, O, NHMe], [AI5689; Me, H, F, H, O, H, H, H, H, S, O, NHMe], [AI5690; Me, H, F, H, O, H, H, H, H, F, S, O, NHMe], [AI 5691; Me, H, F, H, O, H, H, H, Cl, S, O, NHMe], [AI 5692; Me, H, F, H, O, H, H, H, Br, S, O, NHMe], [AI 5693; Me, H, F, H, O, H, H, H, H, I, S, O, NHMe], [AI5694; Me, H, F, H, O, H, H, H, Me, S, O, NHMe], [AI5695; Me, H, F, H, O, H, H, H, H, Et, S, O, NHMe], [AI5696; Me, H, F, H, O, H, H, H, c-Pr, S, O, NHMe], [AI5697; Me, H, F, H, O, H, H, H, OMe, S, O, NHMe], [AI 5698; Me, H, F, H, O, H, H, H, OEt, S, O, NHMe], [AI5699; Me, H, F, H, O, H, H, H, SMe, S, O, NHMe], [AI 5700; Me, H, F, H, O, H, H, H, CF 3, S, O, NHMe],

[AI5701; Et, H, F, H, O, H, H, H, S, O, NHMe], [AI 5702; Et, H, F, H, O, H, H, H, F, S , O, NHMe], [AI5703; Et, H, F, H, O, H, H, H, Cl, S, O, NHMe], [AI 5704; Et, H, F, H, O, H, H , H, Br, S, O, NHMe], [AI 5705; Et, H, F, H, O, H, H, H, I, S, O, NHMe], [AI 5706; Et, H, F, H , O, H, H, H, H, Me, S, O, NHMe], [AI 5707; Et, H, F, H, O, H, H, H, Et, S, O, NHMe], [AI 5708; Et , H, F, H, O, H, H, H, c, Pr, S, O, NHMe], [AI 5709; Et, H, F, H, O, H, H, H, OMe, S, O , NHMe], [AI5710; Et, H, F, H, O, H, H, H, OEt, S, O, NHMe], [AI5711; Et, H, F, H, O, H, H, H , SMe, S, O, NHMe ], [AI5712; Et, H, F, H, O, H, H, H, CF 3, S, O, NHMe], [AI5713; H, H, Cl, H, O, H, H, H, H, H, S, O, NHMe], [AI 5714; H, H, Cl, H, O, H, H, H, F, S, O, NHMe], [AI 5715; H, H, Cl, H, O, H, H, H, H, Cl, S, O, NHMe], [AI 5716; H, H, Cl, H, O, H, H, H, Br, S, O, NHMe] [AI 5717; H, H, Cl, H, O, H, H, I, S, O, NHMe], [AI 5718; H, H, Cl, H, O, H, H, H, Me, H, H, Cl, H, O, H, H, H, Et, S, O, NH Me], [AI 5720; H, H, Cl, H, O, H, S, O, NHMe], [AI 5719; H, H, c-Pr, S, O, NHMe], [AI5721; H, H, Cl, H, O, H, H, H, OMe, S, O, NHMe], [AI5722; H, H, Cl, H, O, H, H, H, OEt, S, O, NHMe], [AI 5723; H, H, Cl, H, O, H, H, S, S, O, NHMe], [ AI5724; H, H, Cl, H, O, H, H, H, CF 3, S, O, NHMe], [AI5725; Cl, H, Cl, H, O, H, H, H, H, S , O, NHMe], [AI5726; Cl, H, Cl, H, O, H, H, H, F, S, O, NHMe], [A Cl, H, Cl, H, O, H, H, H, Cl, S, O, NHMe], [AI5728; Cl, H, Cl, H, O, H, H, H, Br, S, O, NHMe], [AI 5729; Cl, H, Cl, H, O, H, H, H, I, S, O, NHMe], [AI 5730; Cl, H, Cl, H, O, H, H, H, Me, S, O, NHMe], [AI5731; Cl, H, Cl, H, O, H, H, H, H, Et, S, O, NHMe], [AI5732; Cl, H, Cl, H, O, H, H, H, H, c-Pr, S, O, NHMe], [AI5733; Cl, H, Cl, H, O, H, H, H, OMe, S, O, NHMe], [AI 5734; Cl, H, Cl, H, O, H, H, H, H, OEt, S, O, NHMe], [AI 5735; Cl, H, Cl, H, O, H, H, S, S, O, NHMe], [AI5736; Cl, H, Cl, H, O, H, H, H, CF 3, S, O, NHMe], [AI5737; Me, H, Cl, H, O, H, H, H , H, S, O, NHMe], [AI 5738; Me, H, Cl, H, O, H, H, H, H, F, S, O, NHMe], [AI 5739; Me, H, Cl, H, O , H, H, H, H, Cl, S, O, NHMe], [AI5740; Me, H, Cl, H, O, H, H, H, Br, S, O, NHMe], [AI5741; Me, H , Cl, H, O, H, H, H, I, S, O, NHMe], [AI5742; Me, H, Cl, H, O, H, H, H, Me, S, O, NHMe], [AI5743; Me, H, Cl, H, O, H, H, H, Et, S, O, NHMe], [AI 5744; Me, H, Cl, H, O, H, H, H, c-Pr , S, O, NHMe], [AI 5745; Me, H, Cl, H, O, H, H, H, OMe, S, O, NHMe], [AI 5746; Me, H, Cl, H, O, H , H, H, OEt, S, O, NHMe], [AI5747; Me, H, Cl, H, O, H, H, H, SMe, S, O, NHMe], [AI 5748; Me, H, Cl , H, O, H, H , H, CF 3, S, O, NHMe], [AI5749; Et, H, Cl, H, O, H, H, H, H, S, O, NHMe], [ AI 5750; Et, H, Cl, H, O, H, H, H, F, S, O, NHMe], [AI 5751; Et, H, Cl, H, O, H, H, H, Cl, S, O, NHMe], [AI 5752; Et, H, Cl, H , O, H, H, H, H, Br, S, O, NHMe], [AI5753; Et, H, Cl, H, O, H, H, H, I, S, O, NHMe], [AI 5754; Et , H, Cl, H, O, H, H, H, Me, S, O, NHMe], [AI 5755; Et, H, Cl, H, O, H, H, H, Et, S, O, NHMe ], [AI 5756; Et, H, Cl, H, O, H, H, H, c, Pr, S, O, NHMe], [AI 5757; Et, H, Cl, H, O, H, H, H , OMe, S, O, NHMe], [AI 5758; Et, H, Cl, H, O, H, H, H, H, OEt, S, O, NHMe], [AI 5759; Et, H, Cl, H, O , H, H, H, SMe , S, O, NHMe], [AI5760; Et, H, Cl, H, O, H, H, H, CF 3, S, O, NHMe], [AI5761; H, H, Me, H, O, H, H, H, H, H, S, O, NHMe], [AI5762; H, H, Me, H, O, H, H, H, F, S, O, NHMe] [AI5763; H, H, Me, H, O, H, H, H, Cl, S, O, NHMe], [AI 5764; H, H, Me, H, O, H, H, H, Br, S, O, NHMe], [AI 5765; H, H, Me, H, O, H, H, H, I, S, O, NHMe], [AI 5766; H, H, Me, H, O, H, H, H, Me, S, O, NHMe], [AI 5767; H, H, Me, H, O, H, H, H, Et, S, O, NHMe], [AI 5768; H, H, Me, H, O, H, H, H, c, Pr, S, O, NHMe], [AI5769; H, H, Me, H, O, H, H, H, OMe, S, O, NHMe], [ AI 5 770; H, H, Me, H, O, H, H, H, OEt, S, O, NHMe], [AI5771; H, H, Me, H, O, H, H, H, SMe, S, O, NHMe], [AI5772; H, H, Me, H, O, H, H, H, CF 3, S, O, NHMe], [AI5773; Cl, H, Me, H, O, H, H , H, H, S, O, NHMe], [AI5774; Cl, H, Me, H, O, H, H, H, F, S, O, NHMe], [AI 5775; Cl, H, Me, H , O, H, H, H, H, Cl, S, O, NHMe], [AI 5776; Cl, H, Me, H, O, H, H, H, Br, S, O, NHMe], [AI 5777; Cl , H, Me, H, O, H, H, H, I, S, O, NHMe], [AI577 8; Cl, H, Me, H, O, H, H, H, Me, S, O, NHMe], [AI 5779; Cl, H, Me, H, O, H, H, H, Et, S, S O, NHMe], [AI 5780; Cl, H, Me, H, O, H, H, H, c-Pr, S, O, NHMe], [AI 5781; Cl, H, Me, H, O, H, H, H, OMe, S, O, NHMe], [AI5782; Cl, H, Me, H, O, H, H, H, OEt, S, O, NHMe], [AI5783; Cl, H, Me, H, O, H, H, H, SMe, S, O, NHMe], [AI5784; Cl, H, Me, H, O, H, H, H, CF 3, S, O, NHMe], [AI5785 Me, H, Me, H, O, H, H, H, H, S, O, NHMe], [AI 5786; Me, H, Me, H, O, H, H, H, F, S, O , NHMe], [AI5787; Me, H, Me, H, O, H, H, H, Cl, S, O, NHMe], [AI 5788; Me, H, Me, H, O, H, H, H , Br, S, O, NHMe], [AI5789; Me, H, Me, H, O, H, H, H, I, S, O, NHMe], [AI5790; Me, H, Me, H, O , H, H, H, Me, S, O, NHMe], [AI5791; Me, H, Me, H, O, H, H, H, Et, S, O, NHMe], [AI5792; Me, H , Me, H, O, H, H, H, c, Pr, S, O, NHMe], [AI5793; Me, H, Me, H, O, H, H, H, OMe, S, O, NHMe Me, H, Me, H, O, H, H, H, OEt, S, O, NHMe], [AI5795; Me, H, Me, H, O, H, H, H, SMe] , S, O, NHMe], [AI5796; Me, H, Me, H, O, H, H, H, CF 3, S, O, NHMe], [AI5797; Et, H, Me, H, O, H, H, H, H, H, S, O, NHMe], [AI5798; Et, H, Me, H, O, H, H, H, F, S, O, NHMe], [AI5799; Et, H, Me, H, O, H, H, H, H, Cl, S, O, NHMe], [AI 5800; Et, H, Me, H, O, H, H, H, Br, S, O, NHMe],

[AI5801; Et, H, Me, H, O, H, H, I, S, O, NHMe], [AI 5802; Et, H, Me, H, O, H, H, H, Me, S , O, NHMe], [AI5803; Et, H, Me, H, O, H, H, H, Et, S, O, NHMe], [AI 5804; Et, H, Me, H, O, H, H , H, c-Pr, S, O, NHMe], [AI 5 805; Et, H, Me, H, O, H, H, H, OMe, S, O, NHMe], [AI 5806; Et, H, Me , H, O, H, H, H, H, OEt, S, O, NHMe], [AI 5807; Et, H, Me, H, O, H, H, H, SMe, S, O, NHMe], [AI 5808 ; Et, H, Me, H , O, H, H, H, CF 3, S, O, NHMe], [AI5809; H, H, Et, H, O, H, H, H, H, S, H, H, Et, H, O, H, H, H, H, F, S, O, NHMe], [AI 5811; H, H, Et, H, O, H, H, O, NHMe], [AI 5810; H, Cl, S, O, NHMe], [AI5812; H, H, Et, H, O, H, H, H, H, Br, S, O, NHMe], [AI5813; H, H, Et, H, O, H, H, H, H, I, S, O, NHMe], [AI 5814; H, H, Et, H, O, H, H, H, Me, S, O, NHMe], [AI 5815; H, H, Et, H, O, H, H, H, H, Et, S, O, NHMe], [AI 5816; H, H, Et, H, O, H, H, H, c-Pr, S, O, NHMe], [AI 5817; H, H, Et, H, O, H, H, H, OMe, S, O, NHMe], [AI 5818; H, H, Et, H, O, H, H, H, H, OEt, S, O, NHMe], [AI 5819; H, H, Et, H, O, H, H, H, SMe, S, O, NHMe], [AI 5820; H, H, Et, H, O, _{H, H, H, CF 3} , S, O, NHMe], [AI5821; Cl, H, Et, H, O, H, H, H, H, S, O, NHMe], [AI5822; Cl, H , Et, H, O, H, H, H, H, F, S, O, NHMe], [AI 5823; Cl, H, Et, H, O, H, H, H, Cl, S, O, NHMe], [AI 5824; Cl, H, Et, H, O, H, H, H, Br, S, O, NHMe], [AI 5825; Cl, H, Et, H, O, H, H, H, I, S , O, NHMe], [AI 5826; Cl, H, Et, H, O, H, H, H, Me , S, O, NHMe], [AI5827; Cl, H, Et, H, O, H, H, H, H, Et, S, O, NHMe], [AI5828; Cl, H, Et, H, O, H , H, H, c-Pr, S, O, NHMe], [AI 5829; Cl, H, Et, H, O, H, H, H, OMe, S, O, NHMe], [AI 5830; Cl, H , Et, H, O, H, H, H, OEt, S, O, NHMe], [AI 5831; Cl, H, Et, H, O, H, H, H, SMe, S, O, NHMe], [AI5832; Cl, H, Et , H, O, H, H, H, CF 3, S, O, NHMe], [AI5833; Me, H, Et, H, O, H, H, H, H, S, O, NHMe], [AI 5834; Me, H, Et, H, O, H, H, H, H, F, S, O, NH Me], [AI 5835; Me, H, Et, H, O, H, H, H, Cl, S, O, NHMe], [AI5836; Me, H, Et, H, O, H, H, H, Br, S, O, NHMe], [AI 5837; Me, H, Et, H, O, H, H, H, H, I, S, O, NHMe], [AI 5838; Me, H, Et, H, O, H, H, H, Me, S, O, NHMe], [AI 5839; Me, H, Et, H, O, H, H, H, H, Et, S, O, NHMe], [AI 5840; Me, H, Et, H, O, H, H, H, c-Pr, S, O, NHMe], [AI5841; Me, H, Et, H, O, H, H, H, OMe, S, O, NHMe], [AI5842; Me, H, Et, H, O, H, H, H, OEt, S, O, NHMe], [AI5843; Me, H, Et, H, O, H, H, H, SMe, S, O, NHMe], [AI5844; Me, H, Et, H, O, H, H, H, CF 3, S, O, NHMe], [AI5845; Et, H, Et, H, O, H, H, H, H, S, O, NHMe], [AI5846; Et , H, Et, H, O, H, H, H, H, F, S, O, NHMe], [AI 5847; Et, H, Et, H, O, H, H, H, Cl, S, O, NHMe ], [AI 5848; Et, H, Et, H, O, H, H, H, H, Br, S, O, NHMe], [AI 5849; Et, H, Et, H, O, H, H, H, I , S, O, NHMe], [AI 5850; Et, H, Et, H, O, H, H, H, H, Me, S, O, NHMe], [AI 5851; Et, H, Et, H, O, H , H, H, Et, S, O, NHMe], [AI 5 852; Et, H, Et, H, O, H, H, H, c-Pr, S, O, NHMe], [AI 5853; Et, H, Et, H, O, H, H, H, OMe, S, O, NHMe], [AI5854; Et, H, Et, H, O, H, H, H, H, OEt, S, O, NHMe], [AI 5855; Et, H, Et, H, O, H, H, H, SMe, S, O, NHMe], [AI5856; Et, H, Et, H, O, H, H, H, CF 3, S, O, NHMe], [AI5857; H, H, H , H, O, H, H, H, H, H, O, S, NHMe], [AI 5858; H, H, H, H, H, O, H, H, F, O, S, NH Me], [AI 5859 H, H, H, H, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 5860; H, H, H, H, H, O, H, H, H, Br, O, S , NHMe], [AI5861; H, H, H, H, O, H, H, H, I, O, S, NHMe], [AI5862; H, H, H, H, O, H, H, H , Me, O, S, NHMe], [AI5863; H, H, H, H, H, O, H, H, H, Et, O, S, NHMe], [AI5864; H, H, H, H, O , H, H, H, c-Pr, O, S, NHMe], [AI5865; H, H, H, H, H, O, H, H, H, OMe, O, S, NHMe], [AI5866; H , H, H, H, O, H, H, H, OEt, O, S, NHMe], [AI5867; H, H, H, H, H, O, H, H, SMe, O, S, NHMe ], [AI5868; H, H , H, H, O, H, H, H, CF 3, O, S, NHMe], [AI5869; Cl, H, H, H, O, H, H, H, H, O, S, NHMe], [AI5870; Cl, H, H, H, O, H, H, H, H, F, O, S, NHMe], [AI 5871; Cl, H, H, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 5872; Cl, H, H, H, H, O, H, H, H, Br, O, S, NHMe], [AI 5873; Cl, H, H, H, O, H, H, H, I, I, O, S, NHMe], [AI 5874; Cl, H, H, H, O, H, H, Me, O, S, NHMe], [ AI 5875; Cl, H, H, H, H, O, H, H, H, Et, O, S, NHMe], [AI 5876; Cl, H, H, H, H, O, H, H, H, c-Pr, O, S, NHMe], [AI 5877; Cl, H, H, H, O, H, H, H, H, OMe, O, S, NH Me], [AI 5878; Cl , H, H, H, O, H, H, H, OEt, O, S, NHMe], [AI 5879; Cl, H, H, H, H, O, H, H, SMe, O, S, NHMe ], [AI5880; Cl, H , H, H, O, H, H, H, CF 3, O, S, NHMe], [AI5881; Me, H, H, H, O, H, H, H, H, O, S, NHMe], [AI 5882; Me, H, H, H, O, H, H, H, H, F, O, S, NH Me], [AI 5883; Me, H, H, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 5884; Me, H, H, H, H, O, H, H, H, Br, O, S, NHMe], [AI 5885; H, H, O, H, H, H, I, I, O, S, NHMe], [AI 5886; Me, H, H, H, O, H, H, Me, O, S, NHMe], [ AI 5887; Me, H, H, H, H, O, H, H, H, Et, O, S, NHMe], [AI 5888; Me, H, H, H, O, H, H, H, c-Pr, O, S, NHMe], [AI 5889; Me, H, H, H, O, H, H, H, OMe, O, S, NHMe], [AI 5890; Me, H, H, H, O, H, H, H, OEt, O, S, NHMe], [AI5891; Me, H, H, H, H, O, H, H, S, S, O, S, NHMe], [AI5892; Me, H, H, H, O, H, H, H, CF 3, O, S, NHMe], [AI5893; Et, H, H, H, O, H, H, H, H, O, S, NHMe], [AI5894 Et, H, H, H, H, O, H, H, H, H, F, O, S, NHMe], [AI 5895; Et, H, H, H, H, O, H, H, H, Cl, O, S , NHMe], [AI5896; Et, H, H, H, H, O, H, H, H, Br, O, S, NHMe], [AI5897; Et, H, H, H, O, H, H, H , I, O, S, NHMe], [AI 5898; Et, H, H, H, H, O, H, H, H, Me, O, S, NHMe], [AI 5899; Et, H, H, H, O , H, H, H, H, Et, O, S, NHMe], [AI 5900; Et, H, H, H, H, O, H, H, H, c-Pr, O, S, NHMe],

[AI5901; Et, H, H, H, H, O, H, H, OMe, O, S, NHMe], [AI5902; Et, H, H, H, H, O, H, H, H, OEt, O , S, NHMe], [AI5903; Et, H, H, H, H, O, H, H, H, SMe, O, S, NHMe], [AI 5904; Et, H, H, H, O, H, H , H, CF ₃ , O, S, NHMe], [AI 5905; H, H, F, H, O, H, H, H, H, O, S, NHMe], [AI 5906; H, H, F, H, O, H, H, H, H, F, O, S, NHMe], [AI 5907; H, H, F, H, O, H, H, H, Cl, O, S, NHMe], [AI 5908; H, H, F, H, O, H, H, H, H, Br, O, S, NHMe], [AI 5909; H, H, F, H, O, H, H, H, I, O, S, NHMe], [AI5910; H, H, F, H, O, H, H, H, Me, O, S, NHMe], [AI5911; H, H, F, H, O, H, H, H, Et, O, S, NHMe], [AI5912; H, H, F, H, O, H, H, H, c, Pr, O, S, NHMe], [AI5913; H, H, F, H, O, H, H, H, H, OMe, O, S, NHMe], [AI5914; H, H, F, H, O, H, H, H, OEt, O, S, NHMe], [AI5915; H, H, F, H, O, H, H, H, SMe, O, S, NHMe], [AI5916; H, H, F, H, O, H, H, H, CF 3, O, S, NHMe Cl, H, F, H, O, H, H, H, H, O, S, NHMe], [AI 5918; Cl, H, F, H, O, H, H, H, F] , O, S, NHMe], [AI5919; Cl, H, F, H, O, H, H, H, H, Cl, O, S, NHMe], [AI5920; Cl, H, F, H, O, H , H, H, Br, O, S, NHMe], [AI 5921; Cl, H, F, H, O, H, H, H, I, O, S, NH Me], [AI 5922; Cl, H, F , H, O, H, H, H, H, Me, O, S, NHMe], [AI 5923; Cl, H, F, H, O, H, H, H, Et, O, S, NHMe], [AI 5924 Cl, H, F, H, O, H, H, H, c, Pr, O, S, NHMe], [AI5925; Cl, H, F, H, O, H, H, H, OMe, O , S, NHMe], [AI 5926; Cl, H, F, H, O, H, H, H, OEt, O, S, NHMe], [AI 5927; Cl, H , F, H, O, H , H, H, SMe, O, S, NHMe], [AI5928; Cl, H, F, H, O, H, H, H, CF 3, O, S, NHMe] [AI5929; Me, H, F, H, O, H, H, H, H, O, S, NHMe], [AI 5930; Me, H, F, H, O, H, H, H, F, O, S, NHMe], [AI5931; Me, H, F, H, O, H, H, H, Cl, O, S, NHMe], [AI5932; Me, H, F, H, O, H, H, H, Br, O, S, NHMe], [AI5933; Me, H, F, H, O, H, H, H, I, O, S, NHMe], [AI5934; Me, H, F, H, O, H, H, H, H, Me, O, S, NHMe], [AI5935; Me, H, F, H, O, H, H, H, Et, O, S, NHMe], [AI5936; Me, H, F, H, O, H, H, H, c, Pr, O, S, NHMe], [AI 5937; Me, H, F, H, O, H, H, H, OMe, O, S, NHMe], [AI5938; Me, H, F, H, O, H, H, H, OEt, O, S, NHMe], [AI5939; Me, H, F, H, O, H, H, H, SMe, O, S, NHMe], [AI5940; Me, H, F, H, O, H, H, H, CF 3, O, S, NHMe], [AI5941; Et, H, F, H , O, H, H, H, H, H, O, S, NHMe], [AI5942; Et, H, F, H, O, H, H, H, F, O, S, NHMe], [AI5943; Et , H, F, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 5944; Et, H, F, H, O, H, H, H, Br, O, S, NHMe ], [AI5945; Et, H, F, H, O, H, H, H, I, O, S, NHMe], [AI 5946; Et, H, F, H, O, H, H, H, Me , O, S, NHMe], [AI5947; Et, H, F, H, O, H, H, H, Et, O, S, NHMe], [AI5948; Et, H, F, H, O, H , H, H, c-Pr, O, S, NHMe], [AI 5949; Et, H, F, H, O, H, H, H, OMe, O, S, NHMe], [AI 5950; Et, H , F, H, O, H, H, H, OEt, O, S, NHMe], [AI 5951; Et, H, F, H, O, H, H, H, SMe, O, S, NHMe], [AI 595 2; Et, H, F, H, O, H, H, H, CF ₃ , O, S, NH Me], [AI 5953; H, H, Cl, H, O, H, H, H, H, H, O, S, NHMe], [AI 5954; H, H, Cl, H, O, H, H, F, O, S, NHMe] [AI 5 955; H, H, Cl, H, O, H, H, H, Cl, O, S, NHMe], [AI 5956; H, H, Cl, H, O, H, H, H, Br, O, S, NHMe], [AI 5957; H, H, Cl, H, O, H, H, H, I, O, S, NHMe], [AI5958; H, H, Cl, H, O, H, H, H, Me, O, S, NHMe], [AI5959; H, H, Cl, H, O, H, H, H, Et, O, S, NHMe], [AI 5960; H, H, Cl, H, O, H, H, H, c, Pr, O, S, NHMe], [AI5961; H, H, Cl, H, O, H, H, H, OMe, O, S, NHMe], [ AI5962; H, H, Cl, H, O, H, H, OEt, O, S, NHMe], [AI5963; H, H, Cl, H, O, H, H, H, SMe, O, S, NHMe], [AI5964; H, H, Cl, H, O, H, H, H, CF 3, O, S, NHMe], [AI5965; Cl, H, Cl, H, O, H, H , H, H, O, S, NHMe], [AI 5966; Cl, H, Cl, H, O, H, H, H, H, F, O, S, NHMe], [AI 5967; Cl, H, Cl, H , O, H, H, H, H, Cl, O, S, NHMe], [AI5968; Cl, H, Cl, H, O, H, H, H, Br, O, S, NHMe], [AI5969; Cl , H, Cl, H, O, H, H, H, I, O, S, NHMe], [AI 5970; Cl, H, Cl, H, O, H, H, Me, O, S, NHMe , [AI5971; Cl, H, Cl, H, O, H, H, H, Et, O, S, NHMe], [AI 5972; Cl, H, Cl, H, O, H, H, H, c -Pr, O, S, NHMe], [AI 5973; Cl, H, Cl, H, O, H, H, H, H, OMe, O, S, NHMe], [AI 5974; Cl, H, Cl, H, O , H, H, H, H, OEt, O, S, NHMe], [AI5975; Cl, H, Cl, H, O, H, H, H, SMe, O, S, NHMe], [AI5976; Cl, H , Cl, H, O, H , H, H, CF 3, O, S, NHMe], [AI5977; Me, H, Cl, H, O, H, H, H, H, O, S, NHMe] , [AI5978; Me, H, Cl, H, O, H, H, H, F, O, S, NHMe], [AI5979; Me, H, Cl, H, O, H, H, H, Cl, O, S, NHMe], [AI 5980; Me, H, Cl, H, O, H, H, H, Br, O , S, NHMe], [AI5981; Me, H, Cl, H, O, H, H, H, I, O, S, NHMe], [AI 5982; Me, H, Cl, H, O, H, H , H, Me, O, S, NHMe], [AI 5983; Me, H, Cl, H, O, H, H, H, H, Et, O, S, NH Me], [AI 5984; Me, H, Cl, H , O, H, H, H, c, -Pr, O, S, NHMe], [AI5985; Me, H, Cl, H, O, H, H, H, OMe, O, S, NHMe], [AI5986 Me, H, Cl, H, O, H, H, H, OEt, O, S, NHMe], [AI5987; Me, H, Cl, H, O, H, H, H, SMe, O, S , NHMe], [AI5988; Me , H, Cl, H, O, H, H, H, CF 3, O, S, NHMe], [AI5989; Et, H, Cl, H, O, H, H, H, H, O, S, NHMe], [AI5990; Et, H, Cl, H, O, H, H, H, H, F, O, S, NHMe], [AI5991; Et, H, Cl, H, O, H, H, H, H, Cl, O, S, NHMe], [AI5992; Et, H, Cl, H, O, H, H, H, Br, O, S, NHMe], [AI5993; Et, H, Cl, H, O, H, H, H, H, I, O, S, NHMe], [AI 5994; Et, H, Cl, H, O, H, H, H, Me, O, S, NHMe] [AI5995; Et, H, Cl, H, O, H, H, H, Et, O, S, NHMe], [AI5996; Et, H, Cl, H, O, H, H, H, c- Pr, O, S, NHMe], [AI5997; Et, H, Cl, H, O, H, H, H, H, OMe, O, S, NHMe], [AI5998; Et, H, Cl, H, O, H, H, H, H, OEt, O, S, NHMe], [AI5999; Et, H, Cl, H, O, H, H, H, SMe, O, S, NHMe], [AI6000; Et, H, Cl, H, O, H, H, H, CF 3, O, S, NHMe],

[AI 6001; H, H, Me, H, O, H, H, H, H, O, S, NHMe], [AI 6002; H, H, Me, H, O, H, H, H, F, O , S, NHMe], [AI 6003; H, H, Me, H, O, H, H, H, Cl, O, S, NH Me], [AI 6004; H, H, Me, H, O, H, H , H, Br, O, S, NHMe], [AI 6005; H, H, Me, H, O, H, H, H, I, O, S, NH Me], [AI 6006; H, H, Me, H , O, H, H, H, H, Me, O, S, NHMe], [AI 6007; H, H, Me, H, O, H, H, H, Et, O, S, NH Me], [AI 6008; H , H, Me, H, O, H, H, H, c-Pr, O, S, NHMe], [AI 6009; H, H, Me, H, O, H, H, H, OMe, O, S H, H, Me, H, O, H, H, H, OEt, O, S, NHMe], [AI 6011; H, H, Me, H, O, H, H, H , SMe, O, S, NHMe ], [AI6012; H, H, Me, H, O, H, H, H, CF 3, O, S, NHMe], [AI6013; Cl, H, Me, H, O, H, H, H, H, H, O, S, NHMe], [AI 6014; Cl, H, Me, H, O, H, H, H, F, O, S, NHMe], [AI 6015; Cl, H, Me, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 6016; Cl, H, Me, H, O, H, H, H, Br, O, S, NHMe] , [AI 6017; Cl, H, Me, H, O, H, H, I, O, S, NHMe], [AI 6018; Cl, H, Me, H, O, H, H, H, Me, O, S, NHMe], [AI 6019; Cl, H, Me, H, O, H, H, H, Et, O, S, NH Me], [AI 6020; Cl, H, Me, H, O, H, H, H, c-Pr, O, S, NHMe], [AI6021; Cl, H, Me, H, O, H, H, H, OMe, O, S, NHMe], [AI6022; Cl, H, Me, H, O, H, H, H, OEt, O, S, NHMe], [AI6023; Cl, H, Me, H, O, H, H, H, SMe, O, S, NHMe], [ AI6024; Cl, H, Me, H, O, H, H, H, CF 3, O, S, NHMe], [AI6025; Me, H, Me, H, O, H, H, H, H, O , S, NHMe], [AI 6026; Me, H, Me, H, O, H, H, H, F, O, S, NHMe], [AI 6027; Me, H, Me, H, O, H, H, H, H, Cl, O, S, NH Me], [AI 6028; Me, H, Me, H, O, H, H, H, Br, O, S, NHMe], [AI 6029; Me, H, Me, H, O, H, H, H, I, O, S, NHMe], [AI 6030; Me, H, Me, H, O, H, H, H, H, Me, O, S, NHMe], [AI6031; Me, H, Me, H, O, H, H, H, Et, O, S, NHMe], [AI6032; Me, H, Me, H, O, H, H, H, c, Pr, O, S, NHMe], [AI6033; Me, H, Me, H, O, H, H, H, OMe, O, S, NHMe], [AI6034; Me, H, Me, H, O, H, H, H, OEt, O, S, NHMe], [AI 6035; Me, H, Me, H, O, H, H, H, SMe, O, S, NHMe], [AI6036; Me, H, Me, H, O, H, H, H, CF 3, O, S, NHMe], [AI6037; Et, H, Me, H , O, H, H, H, H, H, O, S, NHMe], [AI 6038; Et, H, Me, H, O, H, H, H, F, O, S, NHMe], [AI 6039; Et , H, Me, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 6040; Et, H, Me, H, O, H, H, H, Br, O, S, NHMe ], [AI6041; Et, H, Me, H, O, H, H, H, I, O, S, NHMe], [AI6042; Et, H, Me, H, O, H, H, H, Me , O, S, NHMe], [AI6043; Et, H, Me, H, O, H, H, H, H, Et, O, S, NHMe], [AI6044; Et, H, Me, H, O, H , H, H, c-Pr, O, S, NHMe], [AI 6045; Et, H, Me, H, O, H, H, H, OMe, O, S, NHMe], [AI 6046; Et, H , Me, H, O, H, H, H, OEt, O, S, NHMe], [AI 6047; Et, H, Me, H, O, H, H, H, SMe, O, S, NHMe], [AI6048; Et, H, Me , H, O, H, H, H, CF 3, O, S, NHMe], [AI6049; H, H, Et, H, O, H, H, H, H, O, S, NHMe], [AI 6050; H, H, Et, H, O, H, H, H, H, F, O, S, NHMe], [AI 6051; H, H, Et, H, O, H, H, H, Cl, O, S, NHMe], [AI6052; H, H, Et, H, O, H, H, H, H, Br, O, S, NHMe], [AI 6053; H, H, Et, H, O, H, H, H, I, O, S, NHMe], [AI6054; H, H, Et, H, O, H, H, H, Me, O, S, NHMe], [AI 6055; H, H, Et, H, O, H, H, H, H, Et, O, S, NHMe], [AI6056; H, H, Et, H, O, H, H, H, c, Pr, O, S, NHMe], [AI 6057; H, H, Et, H, O, H, H, H, H, OMe, O, S, NHMe], [AI 6058; H, H, Et, H, O, H, H, H, OEt, O, S, NHMe], [AI 6059; H, H, Et, H, O, H, H, H, SMe, O, S, NHMe], [AI6060; H, H, Et, H, O, H, H, H, CF 3, O, S, NHMe ], [AI6061; Cl, H, Et, H, O, H, H, H, H, H, O, S, NHMe], [AI6062; Cl, H, Et, H, O, H, H, H, F] , O, S, NHMe], [AI6063; Cl, H, Et, H, O, H, H, H, H, Cl, O, S, NHMe], [AI6064; Cl, H, Et, H, O, H , H, H, Br, O, S, NHMe], [AI 6065; Cl, H, Et, H, O, H, H, H, I, O, S, NHMe], [AI 6066; Cl, H, Et , H, O, H, H, H, H, Me, O, S, NHMe], [AI 6067; Cl, H, Et, H, O, H, H, H, Et, O, S, NH Me], [AI 6068 Cl, H, Et, H, O, H, H, H, c, Pr, O, S, NHMe], [AI 6069; Cl, H, Et, H, O, H, H, H, OMe, O , S, NHMe], [AI 6070; Cl, H, Et, H, O, H, H, H, OEt, O, S, NHMe], [AI 6071; Cl, H, Et, H, O, H, H , H, SMe, O, S , NHMe], [AI6072; Cl, H, Et, H, O, H, H, H, CF 3, O, S, NHMe], [AI6073; Me, H, Et, H, O, H, H, H, H, H, O, S, NHMe], [AI 6074; Me, H, Et, H, O, H, H, H, F, O, S, NHMe], [AI 6075; Me, H, Et, H, O, H, H, H, H, Cl, O, S, NHMe], [AI 6076; Me, H, Et, H, O, H, H, H, Br, O, S, NHMe], [AI 6077; Me, H, Et, H, O, H, H, H, I, O, S, NHMe], [AI 6078; Me, H, Et, H, O, H, H, H, Me, O, S, NH Me], [AI 6079; Me, H, Et, H, O, H, H, H, Et, O, S, NHMe], [AI6080; Me, H, Et, H, O, H, H, H, c, Pr, O, S, NHMe], [AI6081; Me, H, Et, H, O, H, H, H, H, OMe, O, S, NHMe], [AI6082; Me, H, Et, H, O, H, H, H, OEt, O, S, NHMe], [AI 6083; H, Et, H, O, H, H, H, SMe, O, S, NHMe], [AI6084; Me, H, Et, H, O, H, H, H, CF 3, O, S, NHMe ], [AI 6085; Et, H, Et, H, O, H, H, H, H, H, O, S, NHMe], [AI 6086; Et, H, Et, H, O, H, H, H, F , O, S, NHMe], [AI 6087; Et, H, Et, H, O, H, H, H, H, Cl, O, S, NH Me], [AI 6088; Et, H, Et, H, O, H , H, H, Br, O, S, NHMe], [AI 6089; Et, H, Et, H, O, H, H, H, I, O, S, NHMe], [AI 6090; Et, H, Et , H, O, H, H, H, H, Me, O, S, NHMe], [AI6091; Et, H, Et, H, O, H, H, H, Et, O, S, NHMe], [AI6092 Et, H, Et, H, O, H, H, H, c, Pr, O, S, NHMe], [AI 6093; Et, H, Et, H, O, H, H, H, OMe, O , S, NHMe], [AI 6094; Et, H, Et, H, O, H, H, H, OEt, O, S, NH Me], [AI 6095; Et, H, Et, H, O, H, H , H, SMe, O, S , NHMe], [AI6096; Et, H, Et, H, O, H, H, H, CF 3, O, S, NHMe].

[Substituent number (MI2); E ¹⁰⁹ ]: [BI1; 1-PYR], [BI2; 3-Me-1-PYR], [BI3; 3-Me-4-F-1-PYR], [BI4 3-Me-4-Cl-1-PYR], [BI5; 3-Me-4-Br-1-PYR], [BI6; 3-Me-4-Me-1-PYR], [BI7; 3 -Me-4-Et-1-PYR], [BI8; 3-Me-4-OMe-1-PYR], [BI9; 3-Me-4-OEt-1-PYR], [BI10; 3-Me -4-CN-1-PYR] , [BI11; 3-Me-4-c-Pr-1-PYR], [BI12; 3-Me-4-CHF 2 -1-PYR], [BI13; 3- _{Me-4-CF 3 -1-} PYR], [BI14; 3-Me-5-F-1-PYR], [BI15; 3-Me-4-F-5-F-1-PYR], [BI16 3-Me-4-Cl-5-F-1-PYR !, [BI17; 3-Me-4-Br-5-F-1-PYR], [BI18; 3-Me-4-Me-5 -F-1-PYR], [BI19; 3-Me-4-Et-5-F-1-PYR], [BI20; 3-Me-4-OMe-5-F-1-PYR], [BI21 3-Me-4-OEt-5-F-1-PYR !, [BI22; 3-Me-4-CN-5-F-1-PYR], [BI23; 3-Me-4-c-Pr -5-F-1-PYR], [BI 24; 3-Me-4-CHF ₂ -5-F-1-PYR], [BI 25; 3-Me-4-CF ₃ -5-F-1-PYR ], [BI 26; 3-Me-5-Cl-1-PYR], [BI 27; 3-Me-4-F-5-Cl-1-PYR], [BI 28; 3-Me-4-Cl-5] -Cl-1-PYR], [BI29; 3-Me-4-Br-5-Cl-1-PYR], [BI30; 3-Me-4-Me-5-Cl-1-PYR], [BI31 3-Me-4-Et-5-Cl-1-PYR], [BI 32; 3-Me-4-OMe-5-Cl-1-PYR], [BI 33; 3-Me-4-OEt-5 -Cl-1-PYR], [BI34; 3-Me-4-CN-5-Cl-1-PYR], [BI35; 3-Me-4-c-Pr-5-Cl-1-PYR], [BI36; 3-Me-4 -CHF 2 -5-Cl-1-PYR], [BI37; 3-Me-4-CF 3 -5-Cl-1-PYR], [BI38; 3-Me -5-Br-1-PYR], [BI 39; 3-Me-4-F-5-Br-1-PYR], [BI 40; 3-Me-4-Cl-5-Br-1-PYR], [BI 41; 3-Me-4-Br-5-Br-1-PYR], [BI 42; 3-Me-4-Me-5-Br-1-PYR], [BI 43; 3-Me-4-Et -5-Br-1-PYR], [BI 44; 3-Me-4-OMe-5-Br-1-PYR], [BI 45; 3-Me-4-OEt-5-Br-1-PYR], [BI 46; 3-Me-4-CN-5-Br-1-PYR], [BI 47; 3-Me-4-c-Pr-5-Br-1-PYR], [BI 48; 3-Me-4 _{-CHF 2 -5-Br-1-} PYR], [BI49; 3-Me-4-CF 3 -5-Br-1-PYR], [BI50; 3-Me-5-Me-1-PYR], [BI 51; 3-Me-4-F-5-Me-1-PYR], [BI 52; 3-Me-4-Cl-5-Me-1-PYR], [BI 53; 3-Me-4-Br -5-Me-1-PYR], [BI 54; 3-Me-4-Me-5-Me-1-PYR], [BI 55; 3-Me-4-Et-5-Me-1-PYR], [BI 56; 3-Me-4-OMe-5-Me-1-PYR], [BI 57; 3-Me-4-OEt-5-Me-1-PYR], [BI 58; 3-Me-4-CN -5-Me-1-PYR], [BI 59; 3-Me-4-c-Pr-5-Me-1-PYR], [BI 60; 3-Me-4-CHF ₂ -5-Me-1- 1 PYR], [BI61; 3- Me-4-CF 3 -5-Me-1-PYR], [BI62; 3-Me-5-Et-1-PYR], [BI63; 3-Me-4-F -5-Et-1-PYR], [BI 64; 3-Me-4-Cl-5-Et-1-PYR], [BI 65; 3-Me-4-Br-5-Et-1-PYR], [BI 66; 3-Me-4-Me-5-Et-1-PYR], [BI 67; 3-Me-4-Et-5-Et-1-PYR], [BI 68; 3-Me-4-OMe -5-Et-1-PYR], [BI69; 3-Me-4-OEt-5-Et-1-PYR], [BI70; 3-Me-4-CN-5-Et-1-PYR], [BI71; 3-Me-4 -c-Pr-5-Et-1-PYR], [BI72; 3-Me-4-CHF 2 -5-Et-1-PYR], [BI73; 3-Me- 4-CF ₃ -5-Et-1-PYR], [BI 74; 3-Me-5-OMe-1-PYR], [BI 75; 3-Me-4-F-5-OMe-1-PYR], [BI 76; -Me-4-Cl-5-OMe-1-PYR], [BI 77; 3-Me-4-Br-5-OMe-1-PYR], [BI 78; 3-Me-4-Me-5-OMe -1-PYR !, [BI 79; 3-Me-4-Et-5-OMe-1-PYR], [BI 80; 3-Me-4-OMe-5-OMe-1-PYR], [BI 81; -Me-4-OEt-5-OMe-1-PYR], [BI 82; 3-Me-4-CN-5-OMe-1-PYR], [BI 83; 3-Me-4-c-Pr-5 -OMe-1-PYR], [BI 84; 3-Me-4-CHF ₂ -5-OMe-1-PYR], [BI 85; 3-Me-4-CF ₃ -5-OMe-1-PYR], [BI 86; 3-Me-5-OEt-1-PYR], [BI 87; 3-Me-4-F-5-OEt-1-PYR], [BI 88; 3-Me-4-Cl-5-OEt -1-PYR !, [BI 89; 3-Me-4-Br-5-OEt-1-PYR], [BI 90; 3-Me-4-Me-5-OEt-1-PYR], [BI 91; -Me-4-Et-5-OEt-1-PYR], [BI 92; 3-Me-4-OMe-5-OEt-1-PYR], [BI 93; 3-Me-4-OEt-5-OEt -1-PYR !, [BI 94; 3-Me-4-CN-5-OEt-1-PYR], [BI 95; 3-Me-4-c-Pr-5-OEt-1-PYR], [BI 96] ; 3-Me-4-CHF 2 -5-OEt-1-PYR], [BI97; 3-Me-4-CF 3 -5-OEt-1-PYR], [BI98; 3-Me-5-CN -1-PYR], [BI99; 3-Me-4-F-5-CN-1-PYR], [BI100; 3-Me-4-Cl-5-CN-1-PYR],

[BI101; 3-Me-4-Br-5-CN-1-PYR], [BI102; 3-Me-4-Me-5-CN-1-PYR], [BI103; 3-Me-4-Et -5-CN-1-PYR], [BI104; 3-Me-4-OMe-5-CN-1-PYR], [BI105; 3-Me-4-OEt-5-CN-1-PYR], [BI106; 3-Me-4-CN-5-CN-1-PYR], [BI107; 3-Me-4-c-Pr-5-CN-1-PYR], [BI108; 3-Me-4 _{-CHF 2 -5-CN-1-} PYR], [BI109; 3-Me-4-CF 3 -5-CN-1-PYR], [BI110; 3-Me-5-c-Pr-1-PYR ], [BI 111; 3-Me-4-F-5-c-Pr-1-PYR], [BI 112; 3-Me-4-Cl-5-c-Pr-1-PYR], [BI 113; -Me-4-Br-5-c-Pr-1-PYR], [BI 114; 3-Me-4-Me-5-c-Pr-1-PYR], [BI 115; 3-Me-4-Et -5-c-Pr-1-PYR], [BI116; 3-Me-4-OMe-5-c-Pr-1-PYR], [BI117; 3-Me-4-OEt-5-c-Pr -1-PYR !, [BI 118; 3-Me-4-CN-5-c-Pr-1-PYR], [BI119; 3-Me-4-c-Pr-5-c-Pr-1-PYR ], [BI120; 3-Me -4-CHF 2 -5-c-Pr-1-PYR], [BI121; 3-Me-4-CF 3 -5-c-Pr-1-PYR], [BI122 3-Me-5-CHF ₂ -1-PYR !, [BI 123; 3-Me-4-F-5-CHF ₂ -1-PYR], [BI 124; 3-Me-4-Cl-5-CHF _{2 -1-PYR], [BI125} ; 3-Me-4-Br-5-CHF 2 -1-PYR], [BI126; 3-Me-4-Me-5-CHF 2 -1-PYR], [ BI127; 3-Me-4- Et-5-CHF 2 -1-PYR], [BI128; 3-Me-4-OMe-5-CHF 2 -1-PYR], [BI129; 3-Me-4- OEt-5-CHF ₂ -1-PYR !, [BI 130; 3-Me-4-CN-5-CHF ₂ -1-PYR], [BI 131; 3-Me-4-c-Pr-5-CHF ₂ -1-PYR], [BI 132; 3-Me-4-CHF ₂ -5- CHF ₂ -1-PYR], [BI 133; 3-Me-4-CF ₃ -5-CHF ₂ -1-PYR], [BI 134; 3-Me-5-CF ₃ -1-PYR], [BI 135; 3-Me-4-F- 5-CF 3 -1-PYR], [BI136; 3-Me-4-Cl-5-CF 3 -1-PYR], [BI137; 3-Me-4-Br- 5-CF ₃ -1-PYR], [BI 138; 3-Me-4-Me-5-CF ₃ -1-PYR], [BI 139; 3-Me-4-Et-5-CF ₃ -1-PYR ], [BI140; 3-Me -4-OMe-5-CF 3 -1-PYR], [BI141; 3-Me-4-OEt-5-CF 3 -1-PYR], [BI142; 3-Me -4-CN-5-CF ₃ -1-PYR !, [BI 143; 3-Me-4-c-Pr-5-CF ₃ -1-PYR], [BI 144; 3-Me-4-CHF _2- 5-CF ₃ -1-PYR], [BI 145; 3-Me-4-CF ₃ -5-CF ₃ -1-PYR], [BI 146; 3-Et-1-PYR], [BI 147; 3-Et] -4-F-1-PYR], [BI 148; 3-Et-4-Cl-1-PYR], [BI 149; 3-Et-4-Br-1-PYR], [BI 150; 3-Et-4 -Me-1-PYR], [BI 151; 3-Et-4-Et-1-PYR], [BI 152; 3-Et-4-OMe-1-PYR], [BI 153; 3-Et-4-OEt -1-PYR !, [BI 154; 3-Et-4-CN-1-PYR], [BI 155; 3-Et-4-c-Pr-1-PYR], [BI 156; 3-Et-4-CHF _{2 -1-PYR], [BI157} ; 3-Et-4-CF 3 -1-PYR], [BI158; 3-Et-5-F-1-PYR], [BI159; 3-Et-4-F -5-F-1-PYR], [BI 160; 3-Et-4-Cl-5-F-1-PYR], [BI 161; 3-Et-4-Br-5-F-1-PYR], [BI162; 3-Et-4-Me-5-F-1-PYR], [BI163; 3-Et-4-Et-5-F-1-PYR], [BI164; 3-Et-4-OMe -5-F-1-PYR], [BI 165; 3-Et-4-OEt-5-F-1-PYR], [BI 166; 3-Et-4-CN-5-F-1-PYR], [BI 167; 3-Et-4-c-Pr-5 -F-1-PYR], [ BI168; 3-Et-4-CHF 2 -5-F-1-PYR], [BI169; 3-Et-4-CF 3 -5-F-1-PYR], [BI 170; 3-Et-5-Cl-1-PYR], [BI 171; 3-Et-4-F-5-Cl-1-PYR], [BI 172; 3-Et-4-Cl-5-Cl -1-PYR !, [BI 173; 3-Et-4-Br-5-Cl-1-PYR], [BI 174; 3-Et-4-Me-5-Cl-1-PYR], [BI 175; -Et-4-Et-5-Cl-1-PYR], [BI 176; 3-Et-4-OMe-5-Cl-1-PYR], [BI 177; 3-Et-4-OEt-5-Cl -1-PYR !, [BI 178; 3-Et-4-CN-5-Cl-1-PYR], [BI 179; 3-Et-4-c-Pr-5-Cl-1-PYR], [BI 180] ; 3-Et-4-CHF 2 -5-Cl-1-PYR], [BI181; 3-Et-4-CF 3 -5-Cl-1-PYR], [BI182; 3-Et-5-Br -1-PYR !, [BI 183; 3-Et-4-F-5-Br-1-PYR], [BI 184; 3-Et-4-Cl-5-Br-1-PYR], [BI 185; -Et-4-Br-5-Br-1-PYR], [BI 186; 3-Et-4-Me-5-Br-1-PYR], [BI 187; 3-Et-4-Et-5-Br -1-PYR !, [BI 188; 3-Et-4-OMe-5-Br-1-PYR], [BI 189; 3-Et-4-OEt-5-Br-1-PYR], [BI 190; -Et-4-CN-5-Br-1-PYR], [BI 191; 3-Et-4-c-Pr-5-Br-1-PYR], [BI 192; 3-Et-4-CHF _2- 5-Br-1-PYR] , [BI193; 3-Et-4-CF 3 -5-Br-1-PYR], [BI194; 3-Et-5-Me-1-PYR], [BI195; 3 -Et-4-F-5-Me-1-PYR], [BI 196; 3-Et-4-Cl-5-Me-1-PYR], [BI 197; 3-Et-4-Br-5-Me -1-PYR !, [BI 198; 3-Et-4-Me-5-Me-1-PYR], [BI 199; 3-Et-4-Et-5-Me-1-PYR], [BI 200; -Et-4-OMe-5-Me-1-PYR],

[BI 201; 3-Et-4-OEt-5-Me-1-PYR], [BI 202; 3-Et-4-CN-5-Me-1-PYR], [BI 203; 3-Et-4-c -Pr-5-Me-1-PYR], [BI 204; 3-Et-4-CHF ₂ -5-Me-1-PYR], [BI 205; 3-Et-4-CF ₃ -5-Me-1 -PYR], [BI 206; 3-Et-5-Et-1-PYR], [BI 207; 3-Et-4-F-5-Et-1-PYR], [BI 208; 3-Et-4-Cl -5-Et-1-PYR], [BI 209; 3-Et-4-Br-5-Et-1-PYR], [BI 210; 3-Et-4-Me-5-Et-1-PYR], [BI 211; 3-Et-4-Et-5-Et-1-PYR], [BI 212; 3-Et-4-OMe-5-Et-1-PYR], [BI 213; 3-Et-4-OEt -5-Et-1-PYR], [BI 214; 3-Et-4-CN-5-Et-1-PYR], [BI 215; 3-Et-4-c-Pr-5-Et-1-PYR ], [BI 216; 3-Et-4-CHF ₂ -5-Et-1-PYR], [BI 217; 3-Et-4-CF ₃ -5-Et-1-PYR], [BI 218; -5-OMe-1-PYR], [BI 219; 3-Et-4-F-5-OMe-1-PYR], [BI 220; 3-Et-4-Cl-5-OMe-1-PYR], [BI 221; 3-Et-4-Br-5-OMe-1-PYR], [BI 222; 3-Et-4-Me-5-OMe-1-PYR], [BI 223; 3-Et-4-Et -5-OMe-1-PYR], [BI 224; 3-Et-4-OMe-5-OMe-1-PYR], [BI 225; 3-Et-4-OEt-5-OMe-1-PYR], [BI 226; 3-Et-4-CN-5-OMe-1-PYR], [BI 227; 3-Et-4-c-Pr-5-OMe-1-PYR], [BI 228; 3-Et-4 _{-CHF 2 -5-OMe-1-} PYR], [BI229; 3-Et-4-CF 3 -5-OMe-1-PYR], [BI230; 3-Et-5-OEt-1-PYR], [BI 231; 3-Et-4-F-5-OEt-1-PYR], [BI 232; 3-Et-4-Cl-5-OEt-1-PYR], [BI 233; 3-Et-4-Br -5-OEt-1-PYR], [BI 234; 3-Et-4 -Me-5-OEt-1-PYR], [BI235; 3-Et-4-Et-5-OEt-1-PYR], [BI236; 3-Et-4-OMe-5-OEt-1-PYR ], [BI 237; 3-Et-4-OEt-5-OEt-1-PYR], [BI 238; 3-Et-4-CN-5-OEt-1-PYR], [BI 239; 3-Et-4] -c-Pr-5-OEt- 1-PYR], [BI240; 3-Et-4-CHF 2 -5-OEt-1-PYR], [BI241; 3-Et-4-CF 3 -5-OEt -1-PYR !, [BI 242; 3-Et-5-CN-1-PYR], [BI 243; 3-Et-4-F-5-CN-1-PYR], [BI 244; 3-Et-4 -Cl-5-CN-1-PYR], [BI 245; 3-Et-4-Br-5-CN-1-PYR], [BI 246; 3-Et-4-Me-5-CN-1-PYR ], [BI 247; 3-Et-4-Et-5-CN-1-PYR], [BI 248; 3-Et-4-OMe-5-CN-1-PYR], [BI 249; 3-Et-4] -OEt-5-CN-1-PYR], [BI 250; 3-Et-4-CN-5-CN-1-PYR], [BI 251; 3-Et-4-c-Pr-5-CN-1 -PYR], [BI252; 3- Et-4-CHF 2 -5-CN-1-PYR], [BI253; 3-Et-4-CF 3 -5-CN-1-PYR], [BI254; 3 -Et-5-c-Pr-1-PYR], [BI 255; 3-Et-4-F-5-c-Pr-1-PYR], [BI 256; 3-Et-4-Cl-5-c -Pr-1-PYR], [BI 257; 3-Et-4-Br-5-c-Pr-1-PYR], [BI 258; 3-Et-4-Me-5-c-Pr-1-PYR ], [BI 259; 3-Et-4-Et-5-c-Pr-1-PYR], [BI 260; 3-Et-4-OMe-5-c-Pr-1-PYR], [BI 261; -Et-4-OEt-5-c-Pr-1-PYR], [BI 262; 3-Et-4-CN-5-c-Pr-1-PYR], [BI 263; 3-Et-4-c -Pr-5-c-Pr- 1-PYR], [BI264; 3-Et-4-CHF 2 -5-c-Pr-1-PYR], [BI265; 3-Et-4-CF 3 -5 -c-Pr-1-PYR], [BI 266; 3-Et-5-CHF ₂ -1-PYR], [BI ₂ 67; 3-Et-4-F-5-CHF ₂ -1-PYR], [BI 268; 3-Et-4-Cl-5-CHF ₂ -1-PYR], [BI 269; 3-Et-4- Br-5-CHF ₂ -1-PYR !, [BI 270; 3-Et-4-Me-5-CHF ₂ -1-PYR], [BI 271; 3-Et-4-Et-5-CHF ₂ -1 -PYR], [BI 272; 3-Et-4-OMe-5-CHF ₂ -1-PYR], [BI 273; 3-Et-4-OEt-5-CHF ₂ -1-PYR], [BI 274; -Et-4-CN-5-CHF ₂ -1-PYR], [BI 275; 3-Et-4-c-Pr-5-CHF ₂ -1-PYR], [BI 276; 3-Et-4-CHF ₂ -5-CHF ₂ -1-PYR], [BI 277; 3-Et-4-CF ₃ -5-CHF ₂ -1-PYR], [BI 278; 3-Et-5-CF ₃ -1-PYR] , [BI 279; 3-Et-4-F-5-CF ₃ -1-PYR], [BI 280; 3-Et-4-Cl-5-CF ₃ -1-PYR], [BI 281; 3-Et- 4-Br-5-CF ₃ -1-PYR !, [BI 282; 3-Et-4-Me-5-CF ₃ -1-PYR], [BI 283; 3-Et-4-Et-5-CF ₃ -1-PYR !, [BI 284; 3-Et-4-OMe-5-CF ₃ -1-PYR], [BI 285; 3-Et-4-OEt-5-CF ₃ -1-PYR], [BI 286] 3-Et-4-CN-5-CF ₃ -1-PYR !, [BI 287; 3-Et-4-c-Pr-5-CF ₃ -1-PYR], [BI 288; 3-Et-4 -CHF ₂ -5-CF ₃ -1-PYR], [BI 289; 3-Et-4-CF ₃ -5-CF ₃ -1-PYR], [BI 290; 5-Me 1-PYR], [BI 291 3-F-5-Me-1-PYR], [BI292; 3-Cl-5-Me-1-PYR], [BI293; 3-Br-5-Me-1-PYR], [BI 294; 3 -OMe-5-Me-1-PYR], [BI 295; 3-OEt-5-Me-1-PYR], [BI 296; 3-CN-5-Me-1-PYR], [BI 297; 3-c -Pr-5-Me-1-PYR], [BI 298; 3-CHF ₂ -5-Me-1-PYR], [BI 299; 3-CF ₃ -5-Me-1-PY R], [BI 300; 4-F-5-Me-1-PYR],

[BI301; 3-F-4-F-5-Me-1-PYR], [BI302; 3-Cl-4-F-5-Me-1-PYR], [BI303; 3-Br-4-F -5-Me-1-PYR], [BI 304; 3-OMe-4-F-5-Me-1-PYR], [BI 305; 3-OEt-4-F-5-Me-1-PYR], [BI306; 3-CN-4-F-5-Me-1-PYR], [BI307; 3-c-Pr-4-F-5-Me-1-PYR], [BI308; 3-CHF _2- 4-F-5-Me- 1-PYR], [BI309; 3-CF 3 -4-F-5-Me-1-PYR], [BI310; 4-Cl-5-Me-1-PYR], [BI 311; 3-F-4-Cl-5-Me-1-PYR], [BI 312; 3-Cl-4-Cl-5-Me-1-PYR], [BI 313; 3-Br-4-Cl -5-Me-1-PYR], [BI 314; 3-OMe-4-Cl-5-Me-1-PYR], [BI 315; 3-OEt-4-Cl-5-Me-1-PYR], [BI 316; 3-CN-4-Cl-5-Me-1-PYR], [BI 317; 3-c-Pr-4-Cl-5-Me-1-PYR], [BI 318; 3-CHF _2- 4-Cl-5-Me-1-PYR], [BI 319; 3-CF ₃ -4-Cl-5-Me-1-PYR], [BI 320; 4-Br-5-Me-1-PYR], [BI 321; 3-F-4-Br-5-Me-1-PYR], [BI 322; 3-Cl-4-Br-5-Me-1-PYR], [BI 323; 3-Br-4-Br -5-Me-1-PYR], [BI 324; 3-OMe-4-Br-5-Me-1-PYR], [BI 325; 3-OEt-4-Br-5-Me-1-PYR], [BI 326; 3-CN-4-Br-5-Me-1-PYR], [BI 327; 3-c-Pr-4-Br-5-Me-1-PYR], [BI 328; 3-CHF _2- 4-Br-5-Me- 1-PYR], [BI329; 3-CF 3 -4-Br-5-Me-1-PYR], [BI330; 4-Me-5-Me-1-PYR], [BI 331; 3-F-4-Me-5-Me-1-PYR], [BI 332; 3-Cl-4-Me-5-Me-1-PYR], [BI 333; 3-Br-4-Me -5-Me-1-PYR], [BI 334; 3-OMe-4-Me-5-Me-1-PYR], [BI 335; 3 -OEt-4-Me-5-Me-1-PYR], [BI 336; 3-CN-4-Me-5-Me-1-PYR], [BI 337; 3-c-Pr-4-Me-5 -Me-1-PYR], [BI 338; 3-CHF ₂ -4-Me-5-Me-1-PYR], [BI 339; 3-CF ₃ -4-Me-5-Me-1-PYR], [BI 340; 4-Et-5-Me-1-PYR], [BI 341; 3-F-4-Et-5-Me-1-PYR], [BI 342; 3-Cl-4-Et-5-Me -1-PYR !, [BI 343; 3-Br-4-Et-5-Me-1-PYR], [BI 344; 3-OMe-4-Et-5-Me-1-PYR], [BI 345; -OEt-4-Et-5-Me-1-PYR], [BI 346; 3-CN-4-Et-5-Me-1-PYR], [BI 347; 3-c-Pr-4-Et-5 -Me-1-PYR], [BI 348; 3-CHF ₂ 4-Et-5-Me-1-PYR], [BI 349; 3-CF ₃ 4-Et-5-Me-1-PYR], [BI 350; 4-OMe-5-Me-1-PYR], [BI 351; 3-F-4-OMe-5-Me-1-PYR], [BI 352; 3-Cl-4-OMe-5-Me -1-PYR !, [BI 353; 3-Br-4-OMe-5-Me-1-PYR], [BI 354; 3-OMe-4-OMe-5-Me-1-PYR], [BI 355; 3] -OEt-4-OMe-5-Me-1-PYR], [BI 356; 3-CN-4-OMe-5-Me-1-PYR], [BI 357; 3-c-Pr-4-OMe-5 -Me-1-PYR], [BI 358; 3-CHF ₂ -4-OMe-5-Me-1-PYR], [BI 359; 3-CF ₃ -4-OMe-5-Me-1-PYR], [BI 360; 4-OEt-5-Me-1-PYR], [BI 361; 3-F-4-OEt-5-Me-1-PYR], [BI 362; 3-Cl-4-OEt-5-Me -1-PYR !, [BI 363; 3-Br-4-OEt-5-Me-1-PYR], [BI 364; 3-OMe-4-OEt-5-Me-1-PYR], [BI 365; -OEt-4-OEt-5-Me-1-PYR], [BI 366; 3-CN-4-OEt-5-Me-1-PYR], [BI 367; 3-c-Pr-4-OEt-5 -Me-1-PYR], [BI 368; 3-CHF ₂ -4-OEt-5-Me-1-PYR], [BI 369; 3-CF ₃ -4-OEt-5-Me-1-PYR], [BI 370; 4-CN-5-Me-1-PYR] , [BI 371; 3-F-4-CN-5-Me-1-PYR], [BI 372; 3-Cl-4-CN-5-Me-1-PYR], [BI 373; CN-5-Me-1-PYR], [BI 374; 3-OMe-4-CN-5-Me-1-PYR], [BI 375; 3-OEt-4-CN-5-Me-1-PYR] [BI 376; 3-CN-4-CN-5-Me-1-PYR], [BI 377; 3-c-Pr-4-CN-5-Me-1-PYR], [BI 378; 3-CHF ₂ -4-CN-5-Me-1-PYR], [BI 379; 3-CF ₃ -4-CN-5-Me-1-PYR], [BI 380; 4-c-Pr-5-Me-1- 1 PYR], [BI 381; 3-F-4-c-Pr-5-Me-1-PYR], [BI 382; 3-Cl-4-c-Pr-5-Me-1-PYR], [BI 383; 3-Br-4-c-Pr-5-Me-1-PYR], [BI 384; 3-OMe-4-c-Pr-5-Me-1-PYR], [BI 385; 3-OEt-4- 4 c-Pr-5-Me-1-PYR], [BI 386; 3-CN-4-c-Pr-5-Me-1-PYR], [BI 387; 3-c-Pr-4-c-Pr- 5-Me-1-PYR], [BI 388; 3-CHF ₂ -4-c-Pr-5-Me-1-PYR], [BI 389; 3-CF ₃ -4-c-Pr-5-Me- 1-PYR], [BI390; 4-CHF 2 -5-Me-1-PYR], [BI391; 3-F-4-CHF 2 -5-Me-1-PYR], [BI392; 3-Cl- _{4-CHF 2 -5-Me-} 1-PYR], [BI393; 3-Br-4-CHF 2 -5-Me-1-PYR], [BI394; 3-OMe-4-CHF 2 -5-Me -1-PYR !, [BI 395; 3-OEt-4-CHF ₂ -5-Me-1-PYR], [BI 396; 3-CN-4-CHF ₂ -5-Me-1-PYR], [BI 397] ; 3-c-Pr-4 -CHF 2 -5-Me-1-PYR], [BI398; 3-CHF 2 -4-CHF 2 -5-Me-1-PYR], [BI399; 3-CF 3 -4-CHF ₂ -5-Me-1-PYR], [BI 400; 4-CF ₃ -5-Me-1-PYR],

[BI401; 3-F-4 -CF 3 -5-Me-1-PYR], [BI402; 3-Cl-4-CF 3 -5-Me-1-PYR], [BI403; 3-Br-4 _{-CF 3 -5-Me-1-} PYR], [BI404; 3-OMe-4-CF 3 -5-Me-1-PYR], [BI405; 3-OEt-4-CF 3 -5-Me- 1-PYR], [BI406; 3-CN-4-CF 3 -5-Me-1-PYR], [BI407; 3-c-Pr-4-CF 3 -5-Me-1-PYR], [ _{BI408; 3-CHF 2 -4-} CF 3 -5-Me-1-PYR], [BI409; 3-CF 3 -4-CF 3 -5-Me-1-PYR], [BI410; 5-Et- 1-PYR], [BI 411; 3-F-5-Et-1-PYR], [BI 412; 3-Cl-5-Et-1-PYR], [BI 413; 3-Br-5-Et-1-] PYR], [BI 414; 3-OMe-5-Et-1-PYR], [BI 415; 3-OEt-5-Et-1-PYR], [BI 416; 3-CN-5-Et-1-PYR] , [BI417; 3-c- Pr-5-Et-1-PYR], [BI418; 3-CHF 2 -5-Et-1-PYR], [BI419; 3-CF 3 -5-Et-1- PYR], [BI 420; 4-F-5-Et-1-PYR], [BI 421; 3-F-4-F-5-Et-1-PYR], [BI 422; 3-Cl-4-F- 5-Et-1-PYR], [BI 423; 3-Br-4-F-5-Et-1-PYR], [BI 424; 3-OMe-4-F-5-Et-1-PYR], [BI BI 425; 3-OEt-4-F-5-Et-1-PYR], [BI 426; 3-CN-4-F-5-Et-1-PYR], [BI 427; 3-c-Pr-4- F-5-Et-1-PYR], [BI 428; 3-CHF ₂ -4-F-5-Et-1-PYR], [BI 429; 3-CF ₃ -4-F-5-Et -1-] PYR], [BI 430; 4-Cl-5-Et-1-PYR], [BI 431; 3-F-4-Cl-5-Et-1-PYR], [BI 432; 3-Cl-4-Cl- 5-Et-1-PYR], [BI 433; 3-Br-4-Cl-5-Et-1-PYR], [BI 434; 3-OMe-4-Cl-5-Et-1-PYR], [BI BI 435; 3-OEt-4-Cl-5-Et-1-PYR], [B I 436; 3-CN-4-Cl-5-Et-1-PYR], [BI 437; 3-c-Pr-4-Cl-5-Et-1-PYR], [BI 438; 3-CHF _2-4 -Cl-5-Et-1-PYR], [BI 439; 3-CF ₃ -4-Cl-5-Et-1-PYR], [BI 440; 4-Br-5-Et-1-PYR], [BI BI 441; 3-F-4-Br-5-Et-1-PYR], [BI 442; 3-Cl-4-Br-5-Et-1-PYR], [BI 443; 3-Br-4-Br- 5-Et-1-PYR], [BI 444; 3-OMe-4-Br-5-Et-1-PYR], [BI 445; 3-OEt-4-Br-5-Et-1-PYR], [BI BI446; 3-CN-4-Br-5-Et-1-PYR], [BI 447; 3-c-Pr-4-Br-5-Et-1-PYR], [BI 448; 3-CHF ₂ -4 -Br-5-Et-1- PYR], [BI449; 3-CF 3 -4-Br-5-Et-1-PYR], [BI450; 4-Me-5-Et-1-PYR], [ BI 451; 3-F-4-Me-5-Et-1-PYR], [BI 452; 3-Cl-4-Me-5-Et-1-PYR], [BI 453; 3-Br-4-Me- 5-Et-1-PYR], [BI 454; 3-OMe-4-Me-5-Et-1-PYR], [BI 455; 3-OEt-4-Me-5-Et-1-PYR], [BI BI 456; 3-CN-4-Me-5-Et-1-PYR], [BI 457; 3-c-Pr-4-Me-5-Et-1-PYR], [BI 458; 3-CHF ₂ -4 -Me-5-Et-1-PYR], [BI 459; 3-CF ₃ -4-Me-5-Et-1-PYR], [BI 460; 4-Et-5-Et-1-PYR], [BI BI 461; 3-F-4-Et-5-Et-1-PYR], [BI 462; 3-Cl-4-Et-5-Et-1-PYR], [BI 463; 3-Br-4-Et- 5-Et-1-PYR], [BI 464; 3-OMe-4-Et-5-Et-1-PYR], [BI 465; 3-OEt-4-Et-5-Et-1-PYR], [BI BI 466; 3-CN-4-Et-5-Et-1-PYR], [BI 467; 3-c-Pr-4-Et-5-Et-1-PYR], [BI 468; 3-CHF _2-4 -Et-5-Et-1-PYR], [BI 469; 3-CF _3- 4-Et-5-Et -1-PYR], [BI 470; 4-OMe-5-Et-1-PYR], [BI 471; 3-F-4-OMe-5-Et-1-PYR], [BI 472; 3-Cl-4 -OMe-5-Et-1-PYR], [BI 473; 3-Br-4-OMe-5-Et-1-PYR], [BI 474; 3-OMe-4-OMe-5-Et-1-PYR ], [BI 475; 3-OEt-4-OMe-5-Et-1-PYR], [BI 476; 3-CN-4-OMe-5-Et-1-PYR], [BI 477; 3-c-Pr -4-OMe-5-Et-1-PYR], [BI 478; 3-CHF ₂ -4-OMe-5-Et-1-PYR], [BI 479; 3-CF ₃ -4-OMe-5-Et -1-PYR !, [BI 480; 4-OEt-5-Et-1-PYR], [BI 481; 3-F-4-OEt-5-Et-1-PYR], [BI 482; 3-Cl-4 -OEt-5-Et-1-PYR], [BI 483; 3-Br-4-OEt-5-Et-1-PYR], [BI 484; 3-OMe-4-OEt-5-Et-1-PYR ], [BI 485; 3-OEt-4-OEt-5-Et-1-PYR], [BI 486; 3-CN-4-OEt-5-Et-1-PYR], [BI 487; 3-c-Pr -4-OEt-5-Et-1-PYR], [BI 488; 3-CHF ₂ -4-OEt-5-Et-1-PYR], [BI 489; 3-CF ₃ -4-OEt-5-Et -1-PYR !, [BI 490; 4-CN-5-Et-1-PYR], [BI 491; 3-F-4-CN-5-Et-1-PYR], [BI 492; 3-Cl-4 -CN-5-Et-1-PYR], [BI 493; 3-Br-4-CN-5-Et-1-PYR], [BI 494; 3-OMe-4-CN-5-Et-1-PYR ], [BI 495; 3-OEt-4-CN-5-Et-1-PYR], [BI 496; 3-CN-4-CN-5-Et-1-PYR], [BI 497; 3-c-Pr] -4-CN-5-Et-1-PYR], [BI 498; 3-CHF ₂ -4-CN-5-Et-1-PYR], [BI 499; 3-CF ₃ -4-CN-5-Et -1-PYR], [BI 500; 4-c-Pr-5-Et-1-PYR],

[BI 501; 3-F-4-c-Pr-5-Et-1-PYR], [BI 502; 3-Cl-4-c-Pr-5-Et-1-PYR], [BI 503; 3-Br -4-c-Pr-5-Et-1-PYR], [BI 504; 3-OMe-4-c-Pr-5-Et-1-PYR], [BI 505; 3-OEt-4-c-Pr -5-Et-1-PYR], [BI 506; 3-CN-4-c-Pr-5-Et-1-PYR], [BI 507; 3-c-Pr-4-c-Pr-5-Et -1-PYR !, [BI 508; 3-CHF ₂ -4-c-Pr-5-Et-1-PYR], [BI 509; 3-CF ₃ -4-c-Pr-5-Et-1-PYR ], [BI510; 4-CHF 2 -5-Et-1-PYR], [BI511; 3-F-4-CHF 2 -5-Et-1-PYR], [BI512; 3-Cl-4-CHF _{2 -5-Et-1-PYR} ], [BI513; 3-Br-4-CHF 2 -5-Et-1-PYR], [BI514; 3-OMe-4-CHF 2 -5-Et-1- PYR], [BI515; 3- OEt-4-CHF 2 -5-Et-1-PYR], [BI516; 3-CN-4-CHF 2 -5-Et-1-PYR], [BI517; 3- c-Pr-4-CHF ₂ -5-Et-1-PYR], [BI 518; 3-CHF ₂ -4-CHF ₂ -5-Et-1-PYR], [BI 519; 3-CF ₃ -4- _{CHF 2 -5-Et-1-} PYR], [BI520; 4-CF 3 -5-Et-1-PYR], [BI521; 3-F-4-CF 3 -5-Et-1-PYR], [BI522; 3-Cl-4 -CF 3 -5-Et-1-PYR], [BI523; 3-Br-4-CF 3 -5-Et-1-PYR], [BI524; 3-OMe-4 _{-CF 3 -5-Et-1-} PYR], [BI525; 3-OEt-4-CF 3 -5-Et-1-PYR], [BI526; 3-CN-4-CF 3 -5-Et- 1-PYR], [BI527; 3-c-Pr-4-CF 3 -5-Et-1-PYR], [BI528; 3-CHF 2 -4-CF3-5-Et-1-PYR], [ BI 529; 3-CF ₃ -4-CF ₃ -5-Et-1-PYR], [BI 530; 1-Me-3-PYR], [BI 531; 1-Me-4-F-3-PYR], [BI 53 2; BI 532; 1-Me -4-Cl-3-PYR !, [BI 533; 1-Me-4-Br-3-PYR], [BI 534; 1-Me-4-Me-3-PYR], [BI 535; 1-Me-4 -Et-3-PYR], [BI 536; 1-Me-4-OMe-3-PYR], [BI 537; 1-Me-4-OEt-3-PYR], [BI 538; 1-Me-4-CN -3-PYR !, [BI 539; 1-Me-4-c-Pr-3-PYR], [BI 540; 1-Me-4-CHF ₂ -3-PYR], [BI 541; 1-Me-4- 4 CF ₃ -3-PYR !, [BI 542; 1-Me-5-F-3-PYR], [BI 543; 1-Me-4-F-5-F-3-PYR], [BI 544; 1-Me -4-Cl-5-F-3-PYR !, [BI 545; 1-Me-4-Br-5-F-3-PYR], [BI 546; 1-Me-4-Me-5-F-3 -PYR], [BI 547; 1-Me-4-Et-5-F-3-PYR], [BI 548; 1-Me-4-OMe-5-F-3-PYR], [BI 549; 1-Me -4-OEt-5-F-3-PYR !, [BI 550; 1-Me-4-CN-5-F-3-PYR], [BI 551; 1-Me-4-c-Pr-5-F -3-PYR !, [BI 552; 1-Me-4-CHF ₂ -5-F-3-PYR], [BI 553; 1-Me-4-CF ₃ -5-F-3-PYR], [BI 554] 1-Me-5-Cl-3-PYR !, [BI 555; 1-Me-4-F-5-Cl-3-PYR], [BI 556; 1-Me-4-Cl-5-Cl-3 -PYR], [BI 557; 1-Me-4-Br-5-Cl-3-PYR], [BI 558; 1-Me-4-Me-5-Cl-3-PYR], [BI 559; 1-Me -4-Et-5-Cl-3-PYR], [BI 560; 1-Me-4-OMe-5-Cl-3-PYR], [BI 561; 1-Me-4-OEt-5-Cl-3 -PYR], [BI 562; 1-Me-4-CN-5-Cl-3-PYR], [BI 563; 1-Me-4-c-Pr-5-Cl-3-PYR], [BI 564; 1 _{-Me-4-CHF 2 -6-} Cl-3-PYR], [BI565; 1-Me-4-CF 3 -7-Cl-3-PYR], [BI566; 1-Me-5-Br-3 -PYR], [BI 567; 1-Me-4-F-5-Br-3-PYR], [BI 568; 1-Me-4- Cl-5-Br-3-PYR], [BI 569; 1-Me-4-Br-5-Br-3-PYR], [BI 570; 1-Me-4-Me-5-Br-3-PYR] , [BI 571; 1-Me-4-Et-5-Br-3-PYR], [BI 572; 1-Me-4-OMe-5-Br-3-PYR], [BI 573; OEt-5-Br-3-PYR], [BI 574; 1-Me-4-CN-5-Br-3-PYR], [BI 575; 1-Me-4-c-Pr-5-Br-3- PYR], [BI576; 1- Me-4-CHF 2 -5-Br-3-PYR], [BI577; 1-Me-4-CF 3 -5-Br-3-PYR], [BI578; 1- Me-5-Me-3-PYR], [BI 579; 1-Me-4-F-5-Me-3-PYR], [BI 580; 1-Me-4-Cl-5-Me-3-PYR] , [BI 581; 1-Me-4-Br-5-Me-3-PYR], [BI 582; 1-Me-4-Me-5-Me-3-PYR], [BI 583; 1-Me-4- 4 Et-5-Me-3-PYR], [BI 584; 1-Me-4-OMe-5-Me-3-PYR], [BI 585; 1-Me-4-OEt-5-Me-3-PYR] [BI 586; 1-Me-4-CN-5-Me-3-PYR], [BI 587; 1-Me-4-c-Pr-5-Me-3-PYR], [BI 588; 1-Me- _{4-CHF 2 -5-Me-} 3-PYR], [BI589; 1-Me-4-CF 3 -5-Me-3-PYR], [BI590; 1-Me-5-Et-3-PYR] , [BI 591; 1-Me-4-F-5-Et-3-PYR], [BI 592; 1-Me-4-Cl-5-Et-3-PYR], [BI 593; 1-Me-4- 4 Br-5-Et-3-PYR], [BI 594; 1-Me-4-Me-5-Et-3-PYR], [BI 595; 1-Me-4-Et-5-Et-3-PYR] , [BI 596; 1-Me-4-OMe-5-Et-3-PYR], [BI 597; 1-Me-4-OEt-5-Et-3-PYR], [BI 598; 1-Me-4- 4 CN-5-Et-3-PYR], [BI 599; 1-Me-4-c-Pr-5-Et-3-PYR], [BI600; 1-Me-4-CHF ₂ -5-Et-3 -PYR],

[BI601; 1-Me-4 -CF 3 -5-Et-3-PYR], [BI602; 1-Me-5-OMe-3-PYR], [BI603; 1-Me-4-F-5- OMe-3-PYR], [BI 604; 1-Me-4-Cl-5-OMe-3-PYR], [BI 605; 1-Me-4-Br-5-OMe-3-PYR], [BI 606; 1-Me-4-Me-5-OMe-3-PYR], [BI 607; 1-Me-4-Et-5-OMe-3-PYR], [BI 608; 1-Me-4-OMe-5-) OMe-3-PYR], [BI 609; 1-Me-4-OEt-5-OMe-3-PYR], [BI 610; 1-Me-4-CN-5-OMe-3-PYR], [BI 611; 1-Me-4-c-Pr-5-OMe-3-PYR], [BI 612; 1-Me-4-CHF ₂ -5-OMe-3-PYR], [BI 613; 1-Me-4-CF _{3 -5-OMe-3-PYR} ], [BI614; 1-Me-5-OEt-3-PYR], [BI615; 1-Me-4-F-5-OEt-3-PYR], [BI616; 1-Me-4-Cl-5-OEt-3-PYR], [BI 617; 1-Me-4-Br-5-OEt-3-PYR], [BI 618; 1-Me-4-Me-5-5 OEt-3-PYR], [BI619; 1-Me-4-Et-5-OEt-3-PYR], [BI620; 1-Me-4-OMe-5-OEt-3-PYR], [BI 621; 1-Me-4-OEt-5-OEt-3-PYR], [BI 622; 1-Me-4-CN-5-OEt-3-PYR], [BI 623; 1-Me-4-c-Pr- 5-OEt-3-PYR] , [BI624; 1-Me-4-CHF 2 -5-OEt-3-PYR], [BI625; 1-Me-4-CF 3 -5-OEt-3-PYR] , [BI 626; 1-Me-5-CN-3-PYR], [BI 627; 1-Me-4-F-5-CN-3-PYR], [BI 628; 1-Me-4-Cl-5-. CN-3-PYR !, [BI 629; 1-Me-4-Br-5-CN-3-PYR], [BI 630; 1-Me-4-Me-5-CN-3-PYR], [BI 631; 1-Me-4-Et-5-CN-3-PYR], [BI 632; 1-Me-4-OMe-5-CN-3-PYR], [BI 633; 1-Me-4-OEt-5-] CN-3-PYR], [BI 634; 1-M e-4-CN-5- CN-3-PYR], [BI635; 1-Me-4-c-Pr-5-CN-3-PYR], [BI636; 1-Me-4-CHF 2 -5 -CN-3-PYR], [ BI637; 1-Me-4-CF 3 -5-CN-3-PYR], [BI638; 1-Me-5-c-Pr-3-PYR], [BI639; 1-Me-4-F-5-c-Pr-3-PYR], [BI 640; 1-Me-4-Cl-5-c-Pr-3-PYR], [BI 641; 1-Me-4- 4 Br-5-c-Pr-3-PYR], [BI 642; 1-Me-4-Me-5-c-Pr-3-PYR], [BI 643; 1-Me-4-Et-5-c- Pr-3-PYR], [BI 644; 1-Me-4-OMe-5-c-Pr-3-PYR], [BI 645; 1-Me-4-OEt-5-c-Pr-3-PYR] , [BI 646; 1-Me-4-CN-5-c-Pr-3-PYR], [BI 647; 1-Me-4-c-Pr-5-c-Pr-3-PYR], [BI 648; _{1-Me-4-CHF 2} -5-c-Pr-3-PYR], [BI649; 1-Me-4-CF 3 -5-c-Pr-3-PYR], [BI650; 1-Me- _{5-CHF 2 -3-PYR]} , [BI651; 1-Me-4-F-5-CHF 2 -3-PYR], [BI652; 1-Me-4-Cl-5-CHF 2 -3-PYR ], [BI 653; 1-Me-4-Br-5-CHF ₂ -3-PYR], [BI 654; 1-Me-4-Me-5-CHF ₂ -3-PYR], [BI 655; 1-Me -4-Et-5-CHF ₂ -3-PYR !, [BI 656; 1-Me -4-OMe -5-CHF ₂ -3-PYR], [BI 657; 1-Me -4-OEt -5-CHF ₂ -3-PYR !, [BI 658; 1-Me-4-CN-5-CHF ₂ -3-PYR], [BI 659; 1-Me-4-c-Pr-5-CHF ₂ -3-PYR] , [BI 660; 1-Me-4-CHF ₂ -5-CHF ₂ -3-PYR], [BI 661; 1-Me-4-CF ₃ -5-CHF ₂ -3-PYR], [BI 662; _{Me-5-CF 3 -3-} PYR], [BI663; 1-Me-4-F-5-CF 3 -3-PYR], [BI664; 1-Me-4-Cl-5-CF 3 -3 -PYR], [BI 665; 1-Me-4-Br- _{5-CF 3 -3-PYR]} , [BI666; 1-Me-4-Me-5-CF 3 -3-PYR], [BI667; 1-Me-4-Et-5-CF 3 -3-PYR ], [BI668; 1-Me -4-OMe-5-CF3-3-PYR], [BI669; 1-Me-4-OEt-5-CF 3 -3-PYR], [BI670; 1-Me- _{4-CN-5-CF 3} -3-PYR], [BI671; 1-Me-4-c-Pr-5-CF 3 -3-PYR], [BI672; 1-Me-4-CHF 2 -5 -CF3-3-PYR], [BI673; 1-Me-4-CF 3 -5-CF3-3-PYR], [BI674; 1-Me-5-OPr-3-PYR], [BI675; 1- Me-4-F-5-OPr-3-PYR], [BI 676; 1-Me-4-Cl-5-OPr-3-PYR], [BI 677; 1-Me-4-Br-5-OPr- 3-PYR], [BI 678; 1-Me-4-Me-5-OPr-3-PYR], [BI 679; 1-Me-4-Et-5-OPr-3-PYR], [BI 680; Me-4-OMe-5-OPr-3-PYR], [BI 681; 1-Me-4-OEt-5-OPr-3-PYR], [BI 682; 1-Me-4-CN-5-OPr- 3-PYR], [BI683; 1-Me-4-c-Pr-5-OPr-3-PYR], [BI684; 1-Me-4-CHF 2 -5-OPr-3-PYR], [BI685 ; 1-Me-4-CF 3 -5-OPr-3-PYR], [BI686; 1-Me-5-OCH 2 CH = CH 2 -3-PYR], [BI687; 1-Me-4-F -5-OCH ₂ CH = CH ₂ -3-PYR], [BI 688; 1-Me-4-Cl-5-OCH ₂ CH = CH ₂ -3-PYR], [BI 689; 1-Me-4-Br -5-OCH ₂ CH = CH ₂ -3-PYR], [BI 690; 1-Me-4-Me-5-OCH ₂ CH = CH ₂ -3-PYR], [BI 691; 1-Me-4-Et] _{-5-OCH 2 CH = CH 2} -3-PYR], [BI692; 1-Me-4-OMe-5-OCH 2 CH = CH 2 -3-PYR], [BI693; 1-Me-4-OEt -5-OCH ₂ CH = CH ₂ -3-PYR], [BI 694; 1-Me-4-CN-5-OCH ₂ CH = CH ₂ -3 -PYR], [BI695; 1- Me-4-c-Pr-5-OCH 2 CH = CH 2 -3-PYR], [BI696; 1-Me-4-CHF 2 -5-OCH 2 CH = CH ₂ -3-PYR !, [BI 697; 1-Me-4-CF ₃ -5-OCH ₂ CH = CH ₂ -3-PYR], [BI 698; 1-Me-5-OCH ₂ CH = CCl ₂ -3 -PYR], [BI699; 1- Me-4-F-5-OCH 2 CH = CCl 2 -3-PYR], [BI700; 1-Me-4-Cl-5-OCH 2 CH = CCl 2 -3 -PYR],

[BI701; 1-Me-4 -Br-5-OCH 2 CH = CCl 2 -3-PYR], [BI702; 1-Me-4-Me-5-OCH 2 CH = CCl 2 -3-PYR], [BI703; 1-Me-4 -Et-5-OCH 2 CH = CCl 2 -3-PYR], [BI704; 1-Me-4-OMe-5-OCH 2 CH = CCl 2 -3-PYR], [BI705; 1-Me-4 -OEt-5-OCH 2 CH = CCl 2 -3-PYR], [BI706; 1-Me-4-CN-5-OCH 2 CH = CCl 2 -3-PYR], [BI 707; 1-Me-4-c-Pr-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 708; 1-Me-4-CHF ₂ -5-OCH ₂ CH = CCl ₂ -3- PYR], [BI709; 1- Me-4-CF 3 -5-OCH 2 CH = CCl 2 -3-PYR], [BI710; 1-Me-5-OCH 2 C≡CH-3-PYR], [ BI 711; 1-Me-4-F-5-OCH ₂ C≡CH-3-PYR], [BI 712; 1-Me-4-Cl-5-OCH ₂ C≡CH-3-PYR], [BI 713; 1-Me-4-Br-5-OCH ₂ C≡CH-3-PYR], [BI 714; 1-Me-4-Me-5-OCH ₂ C≡CH-3-PYR], [BI 715; 1- Me-4-Et-5-OCH ₂ C≡CH-3-PYR], [BI 716; 1-Me-4-OMe-5-OCH ₂ C≡CH-3-PYR], [BI 717; 1-Me- 4-OEt-5-OCH ₂ C≡CH-3-PYR], [BI 718; 1-Me-4-CN-5-OCH ₂ C≡CH-3-PYR], [BI 719; 1-Me-4- c-Pr-5-OCH ₂ C≡CH-3-PYR], [BI 720; 1-Me-4-CHF ₂ -5-OCH ₂ C≡CH-3-PYR], [BI 721; 1-Me-4 _{-CF 3 -5-OCH 2 C≡CH-} 3-PYR], [BI722; 1-Me-5-OCH 2 CF 3 -3-PYR], [BI723; 1-Me-4-F-5-OCH ₂ CF ₃ -3-PYR !, [BI 724; 1-Me-4-Cl-5-OCH ₂ CF ₃ -3-PYR], [BI 725; 1-Me-4-Br-5-OCH ₂ CF ₃ -3-PYR], [BI726; 1-Me-4-Me-5-OCH 2 CF 3 -3-PYR], [BI727; 1-Me-4-Et-5-OCH 2 CF 3 -3-PYR ], [BI728; 1-Me -4-OMe-5-OCH 2 CF 3 -3-PYR], [BI729; 1-Me-4-OEt-5-OCH 2 CF 3 -3-PYR], [BI730 ; 1-Me-4-CN -5-OCH 2 CF 3 -3-PYR], [BI731; 1-Me-4-c-Pr-5-OCH 2 CF 3 -3-PYR], [BI732; 1 _{-Me-4-CHF 2 -5-} OCH 2 CF 3 -3-PYR], [BI733; 1-Me-4-CF 3 -5-OCH 2 CF 3 -3-PYR], [BI734; 1-Me -5-CH ₂ OCH ₃ -3-PYR !, [BI 735; 1-Me-4-F-5-CH ₂ OCH ₃ -3-PYR], [BI 736; 1-Me-4-Cl-5-CH ₂ OCH ₃ -3-PYR !, [BI 737; 1-Me-4-Br-5-CH ₂ OCH ₃ -3-PYR], [BI 738; 1-Me-4-Me-5-CH ₂ OCH _3- 3-PYR], [BI739; 1-Me-4-Et-5-CH 2 OCH 3 -3-PYR], [BI740; 1-Me-4-OMe-5-CH 2 OCH 3 -3-PYR] [BI 741; 1-Me-4-OEt-5-CH ₂ OCH ₃ -3-PYR], [BI 742; 1-Me-4-CN-5-CH ₂ OCH ₃ -3-PYR], [BI 743; 1-Me-4-c- Pr-5-CH 2 OCH 3 -3-PYR], [BI744; 1-Me-4-CHF 2 -5-CH 2 OCH 3 -3-PYR], [BI745; 1 _{-Me-4-CF 3 -5-} CH 2 OCH 3 -3-PYR], [BI746; 1-Et-3-PYR], [BI747; 1-Et-4-F-3-PYR], [BI748 1-Et-4-Cl-3-PYR], [BI 749; 1-Et-4-Br-3-PYR], [BI 750; 1-Et-4-Me-3-PYR], [BI 751; -Et-4-Et-3-PYR], [BI 752; 1-Et-4-OMe-3-PYR], [BI 753; 1-Et-4-OEt-3-PYR], [BI 754; 1-Et -4-CN-3-PYR], [BI7 55; 1-Et-4- c-Pr-3-PYR], [BI756; 1-Et-4-CHF 2 -3-PYR], [BI757; 1-Et-4-CF 3 -3-PYR] , [BI 758; 1-Et-5-F-3-PYR], [BI 759; 1-Et-4-F-5-F-3-PYR], [BI 760; 1-Et-4-Cl-5-. F-3-PYR], [BI 761; 1-Et-4-Br-5-F-3-PYR], [BI 762; 1-Et-4-Me-5-F-3-PYR], [BI 763; 1-Et-4-Et-5-F-3-PYR], [BI 764; 1-Et-4-OMe-5-F-3-PYR], [BI 765; 1-Et-4-OEt-5-] F-3-PYR], [BI 766; 1-Et-4-CN-5-F-3-PYR], [BI 767; 1-Et-4-c-Pr-5-F-3-PYR], [BI 767; BI768; 1-Et-4- CHF 2 -5-F-3-PYR], [BI769; 1-Et-4-CF 3 -5-F-3-PYR], [BI770; 1-Et-5- Cl-3-PYR !, [BI 771; 1-Et-4-F-5-Cl-3-PYR], [BI 772; 1-Et-4-Cl-5-Cl-3-PYR], [BI 773; 1-Et-4-Br-5-Cl-3-PYR], [BI 774; 1-Et-4-Me-5-Cl-3-PYR], [BI 775; 1-Et-4-Et-5-] Cl-3-PYR], [BI 776; 1-Et-4-OMe-5-Cl-3-PYR], [BI 777; 1-Et-4-OEt-5-Cl-3-PYR], [BI 778; 1-Et-4-CN-5-Cl-3-PYR], [BI 779; 1-Et-4-c-Pr-5-Cl-3-PYR], [BI 780; 1-Et-4-CHF ₂ -5-Cl-3-PYR !, [BI 781; 1-Et-4-CF ₃ -5-Cl-3-PYR], [BI 782; 1-Et-5-Br-3-PYR], [BI 783; 1-Et-4-F-5-Br-3-PYR], [BI 784; 1-Et-4-Cl-5-Br-3-PYR], [BI 785; 1-Et-4-Br-5- Br-3-PYR], [BI 786; 1-Et-4-Me-5-Br-3-PYR], [BI 787; 1-Et-4-Et-5-Br-3-PYR], [BI 788; 1-Et-4-OMe-5-Br-3-PYR], [BI 789; 1-Et-4-OEt-5-Br-3-PYR], [BI BI 790; 1-Et-4-CN-5-Br-3-PYR], [BI 791; 1-Et-4-c-Pr-5-Br-3-PYR], [BI 792; 1-Et-4- _{CHF 2 -5-Br-3-} PYR], [BI793; 1-Et-4-CF 3 -5-Br-3-PYR], [BI794; 1-Et-5-Me-3-PYR], [ BI795; 1-Et-4-F-5-Me-3-PYR], [BI 796; 1-Et-4-Cl-5-Me-3-PYR], [BI 797; 1-Et-4-Br- 5-Me-3-PYR, [BI 798; 1-Et-4-Me-5-Me-3-PYR], [BI 799; 1-Et-4-Et-5-Me-3-PYR], [BI BI 800; 1-Et-4-OMe-5-Me-3-PYR],

[BI 801; 1-Et-4-OEt-5-Me-3-PYR], [BI 802; 1-Et-4-CN-5-Me-3-PYR], [BI 803; 1-Et-4-c] -Pr-5-Me-3- PYR], [BI804; 1-Et-4-CHF 2 -5-Me-3-PYR], [BI805; 1-Et-4-CF 3 -5-Me-3 -PYR], [BI 806; 1-Et-5-Et-3-PYR], [BI 807; 1-Et-4-F-5-Et-3-PYR], [BI 808; 1-Et-4-Cl] -5-Et-3-PYR], [BI 809; 1-Et-4-Br-5-Et-3-PYR], [BI 810; 1-Et-4-Me-5-Et-3-PYR], [BI 811; 1-Et-4-Et-5-Et-3-PYR], [BI 812; 1-Et-4-OMe-5-Et-3-PYR], [BI 813; 1-Et-4-OEt] -5-Et-3-PYR], [BI 814; 1-Et-4-CN-5-Et-3-PYR], [BI 815; 1-Et-4-c-Pr-5-Et-3-PYR ], [BI 816; 1-Et-4-CHF ₂ -5-Et-3-PYR], [BI 817; 1-Et-4-CF ₃ -5-Et-3-PYR], [BI 818; 1-Et] -5-OMe-3-PYR], [BI 819; 1-Et-4-F-5-OMe-3-PYR], [BI 820; 1-Et-4-Cl-5-OMe-3-PYR], [BI 821; 1-Et-4-Br-5-OMe-3-PYR], [BI 822; 1-Et-4-Me-5-OMe-3-PYR], [BI 823; 1-Et-4-Et] -5-OMe-3-PYR], [BI 824; 1-Et-4-OMe-5-OMe-3-PYR], [BI 825; 1-Et-4-OEt-5-OMe-3-PYR], [BI 826; 1-Et-4-CN-5-OMe-3-PYR], [BI 827; 1-Et-4-c-Pr-5-OMe-3-PYR], [BI 828; 1-Et-4 _{-CHF 2 -5-OMe-3-} PYR], [BI829; 1-Et-4-CF 3 -5-OMe-3-PYR], [BI830; 1-Et-5-OEt-3-PYR], [BI 831; 1-Et-4-F-5-OEt-3-PYR], [BI 832; 1-Et-4-Cl-5-OEt-3-PYR], [BI 833; 1-Et-4-Br -5-OEt-3-PYR], [BI 834; 1-Et-4 -Me-5-OEt-3-PYR], [BI 835; 1-Et-4-Et-5-OEt-3-PYR], [BI 836; 1-Et-4-OMe-5-OEt-3-PYR ], [BI 837; 1-Et-4-OEt-5-OEt-3-PYR], [BI 838; 1-Et-4-CN-5-OEt-3-PYR], [BI 839; 1-Et-4] -c-Pr-5-OEt- 3-PYR], [BI840; 1-Et-4-CHF 2 -5-OEt-3-PYR], [BI841; 1-Et-4-CF 3 -5-OEt -3-PYR !, [BI 842; 1-Et-5-CN-3-PYR], [BI 843; 1-Et-4-F-5-CN-3-PYR], [BI 844; 1-Et-4 -Cl-5-CN-3-PYR], [BI 845; 1-Et-4-Br-5-CN-3-PYR], [BI 846; 1-Et-4-Me-5-CN-3-PYR ], [BI 847; 1-Et-4-Et-5-CN-3-PYR], [BI 848; 1-Et-4-OMe-5-CN-3-PYR], [BI 849; 1-Et-4] -OEt-5-CN-3-PYR], [BI 850; 1-Et-4-CN-5-CN-3-PYR], [BI 851; 1-Et-4-c-Pr-5-CN-3 -PYR], [BI 852; 1-Et-4-CHF ₂ -5-CN-3-PYR], [BI 853; 1-Et-4-CF ₃ -5-CN-3-PYR], [BI 854; 1 -Et-5-c-Pr-3-PYR], [BI 855; 1-Et-4-F-5-c-Pr-3-PYR], [BI 856; 1-Et-4-Cl-5-c -Pr-3-PYR], [BI 857; 1-Et-4-Br-5-c-Pr-3-PYR], [BI 858; 1-Et-4-Me-5-c-Pr-3-PYR ], [BI 859; 1-Et-4-Et-5-c-Pr-3-PYR], [BI 860; 1-Et-4-OMe-5-c-Pr-3-PYR], [BI 861; 1] -Et-4-OEt-5-c-Pr-3-PYR], [BI 862; 1-Et-4-CN-5-c-Pr-3-PYR], [BI 863; 1-Et-4-c -Pr-5-c-Pr- 3-PYR], [BI864; 1-Et-4-CHF 2 -5-c-Pr-3-PYR], [BI865; 1-Et-4-CF 3 -5 -c-Pr-3-PYR], [BI 866; 1-Et-5-CHF ₂ -3-PYR], [BI 8 67; 1-Et-4- F-5-CHF 2 -3-PYR], [BI868; 1-Et-4-Cl-5-CHF 2 -3-PYR], [BI869; 1-Et-4- _{br-5-CHF 2 -3-} PYR], [BI870; 1-Et-4-Me-5-CHF 2 -3-PYR], [BI871; 1-Et-4-Et-5-CHF 2 -3 -PYR], [BI 872; 1-Et-4-OMe-5-CHF ₂ -3-PYR], [BI 873; 1-Et-4-OEt-5-CHF ₂ -3-PYR], [BI 874; -Et-4-CN-5- CHF 2 -3-PYR], [BI875; 1-Et-4-c-Pr-5-CHF 2 -3-PYR], [BI876; 1-Et-4-CHF ₂ -5-CHF ₂ -3-PYR !, [BI 877; 1-Et-4-CF ₃ -5-CHF ₂ -3-PYR], [BI 878; 1-Et-5-CF ₃ -3-PYR] , [BI 879; 1-Et-4-F-5-CF ₃ -3-PYR], [BI 880; 1-Et-4-Cl-5-CF ₃ -3-PYR], [BI 881; 1-Et- _{4-Br-5-CF 3} -3-PYR], [BI882; 1-Et-4-Me-5-CF 3 -3-PYR], [BI883; 1-Et-4-Et-5-CF 3 -3-PYR], [BI884; 1-Et-4-OMe-5-CF 3 -3-PYR], [BI885; 1-Et-4-OEt-5-CF 3 -3-PYR], [BI886 ; 1-Et-4-CN -5-CF 3 -3-PYR], [BI887; 1-Et-4-c-Pr-5-CF 3 -3-PYR], [BI888; 1-Et-4 _{-CHF 2 -5-CF3-3-PYR]} , [BI889; 1-Et-4-CF 3 -5-CF 3 -3-PYR], [BI890; 1-Et-5-OPr-3-PYR] , [BI 891; 1-Et-4-F-5-OPr-3-PYR], [BI 892; 1-Et-4-Cl-5-OPr-3-PYR], [BI 893; 1-Et-4- Br-5-OPr-3-PYR], [BI 894; 1-Et-4-Me-5-OPr-3-PYR], [BI 895; 1-Et-4-Et-5-OPr-3-PYR] , [BI 896; 1-Et-4-OMe-5-OPr-3-PYR], [BI 897; 1-Et-4-OEt-5-OPr-3-PYR], [BI 898; 1 -Et-4-CN-5-OPr-3-PYR], [BI 899; 1-Et-4-c-Pr-5-OPr-3-PYR], [BI 900; 1-Et-4-CHF _2- 5-OPr-3-PYR],

[BI901; 1-Et-4 -CF 3 -5-OPr-3-PYR], [BI902; 1-Et-5-OCH 2 CH = CH 2 -3-PYR], [BI903; 1-Et-4 _{-F-5-OCH 2 CH =} CH 2 -3-PYR], [BI904; 1-Et-4-Cl-5-OCH 2 CH = CH 2 -3-PYR], [BI905; 1-Et-4 _{-Br-5-OCH 2 CH =} CH 2 -3-PYR], [BI906; 1-Et-4-Me-5-OCH 2 CH = CH 2 -3-PYR], [BI907; 1-Et-4 _{-Et-5-OCH 2 CH =} CH 2 -3-PYR], [BI908; 1-Et-4-OMe-5-OCH 2 CH = CH 2 -3-PYR], [BI909; 1-Et-4 _{-OEt-5-OCH 2 CH =} CH 2 -3-PYR], [BI910; 1-Et-4-CN-5-OCH 2 CH = CH 2 -3-PYR], [BI911; 1-Et-4 _{-c-Pr-5-OCH 2} CH = CH 2 -3-PYR], [BI912; 1-Et-4-CHF 2 -5-OCH 2 CH = CH 2 -3-PYR], [BI913; 1- _{Et-4-CF 3 -5-} OCH 2 CH = CH 2 -3-PYR], [BI914; 1-Et-5-OCH 2 CH = CCl 2 -3-PYR], [BI915; 1-Et-4 -F-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 916; 1-Et-4-Cl-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 917; 1-Et-4 —Br-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 918; 1-Et-4-Me-5-OCH ₂ CHCCCl ₂ -3-PYR], [BI 919; 1-Et-4 -Et-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 920; 1-Et-4-OMe-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 921; 1-Et-4 -OEt-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 922; 1-Et-4-CN-5-OCH ₂ CH = CCl ₂ -3-PYR], [BI 923; 1-Et-4 _{-c-Pr-5-OCH 2} CH = CCl 2 -3-PYR], [BI924; 1-Et-4-CHF 2 -5-OCH 2 CH = CCl 2 -3-PYR], [BI925 ; 1-Et-4-CF 3 -5-OCH 2 CH = CCl 2 -3-PYR], [BI926; 1-Et-5-OCH 2 C≡CH-3-PYR], [BI927; 1-Et -4-F-5-OCH ₂ C≡CH-3-PYR], [BI 928; 1-Et-4-Cl-5-OCH ₂ C≡CH-3-PYR], [BI 929; 1-Et-4 -Br-5-OCH ₂ C≡CH-3-PYR], [BI 930; 1-Et-4-Me-5-OCH ₂ C≡CH-3-PYR], [BI 931; 1-Et-4-Et -5-OCH ₂ C≡CH-3-PYR], [BI 932; 1-Et-4-OMe-5-OCH ₂ C≡CH-3-PYR], [BI 933; 1-Et-4-OEt-5 -OCH ₂ C≡CH-3-PYR], [BI 934; 1-Et-4-CN-5-OCH ₂ C≡CH-3-PYR], [BI 935; 1-Et-4-c-Pr-5 _{-OCH 2 C≡CH-3-PYR]} , [BI936; 1-Et-4-CHF 2 -5-OCH 2 C≡CH-3-PYR], [BI937; 1-Et-4-CF 3 -5 _{-OCH 2 C≡CH-3-PYR]} , [BI938; 1-Et-5-OCH 2 CF 3 -3-PYR], [BI939; 1-Et-4-F-5-OCH 2 CF 3 -3 -PYR], [BI940; 1- Et-4-Cl-5-OCH 2 CF 3 -3-PYR], [BI941; 1-Et-4-Br-5-OCH 2 CF 3 -3-PYR], [BI942; 1-Et-4 -Me-5-OCH 2 CF 3 -3-PYR], [BI943; 1-Et-4-Et-5-OCH 2 CF 3 -3-PYR], [BI944; 1 -Et-4-OMe-5- OCH 2 CF 3 -3-PYR], [BI945; 1-Et-4-OEt-5-OCH 2 CF 3 -3-PYR], [BI946; 1-Et-4 _{-CN-5-OCH 2 CF 3} -3-PYR], [BI947; 1-Et-4-c-Pr-5-OCH 2 CF 3 -3-PYR], [BI948; 1-Et-4-CHF ₂ -5-OCH ₂ CF ₃ -3-PYR !, [BI 949; 1-Et-4-CF ₃ -5-OCH ₂ CF ₃ -3-PYR], [BI 950; 1-Et-5-CH ₂ OCH ₃ -3 -PYR], [BI 951; 1-Et-4-F-5-CH ₂ OCH ₃ -3-PYR], [BI 952; 1-Et-4-Cl-5-CH ₂ OCH ₃ -3-PYR], [BI 953; 1-Et-4-Br-5-CH ₂ OCH ₃ -3-PYR], [BI 954; 1-Et-4-Me-5-CH ₂ OCH ₃ -3-PYR], [BI 955; 1 -Et-4-Et-5-CH ₂ OCH ₃ -3-PYR], [BI 956; 1-Et-4-OMe-5-CH ₂ OCH ₃ -3-PYR], [BI 957; 1-Et-4 -OEt-5-CH ₂ OCH ₃ -3-PYR], [BI 958; 1-Et-4-CN-5-CH ₂ OCH ₃ -3-PYR], [BI 959; 1-Et-4-c-Pr _{-5-CH 2 OCH 3 -3-} PYR], [BI960; 1-Et-4-CHF 2 -5-CH 2 OCH 3 -3-PYR], [BI961; 1-Et-4-CF 3 -5 -CH ₂ OCH ₃ -3-PYR], [BI 962; 3-Me-2-Py], [BI 963; 3-Et-2-Py], [BI 964; 3-Pr-2-Py], [BI 965; 3-i-Pr-2-Py, [BI 966; 4-Me-2-Py], [BI 967; 4-Et-2-Py], [BI 968; 4-Pr-2-Py], [BI 969; 4-i-Pr-2-Py !, [BI 970; 5-Me-2-Py], [BI 971; 5-Et-2-Py], [BI 972; 5-Pr-2-Py], [BI 973; 5-i-Pr-2-Py !, [BI 974; 6-Me-2-Py], [BI 975; 6-Et-2-Py], [BI 976; 6-Pr-2-Py], [BI 977; 6-i-Pr-2-Py !, [BI 978; 3-Me-4-Me-2-Py], [BI 979; 3-Me-4-Et-2-Py], [BI 980; 3-Me- 4-Pr-2-Py, [BI 981; 3-Me-4-i-Pr-2-Py], [BI 982; 3-Me-5-Me-2-Py], [BI 983; 5-Et-2-Py !, [BI 984; 3-Me-5-Pr-2-Py], [BI 985; 3-Me-5-i-Pr-2-Py], [BI 986; 3-Me- 6-Me-2-Py, [BI 987; 3-Me-6-Et-2-Py], [BI 988; 3-Me-6-Pr-2-Py], [BI 989; 3-Me-6 -i-Pr-2-Py], [BI 990; 3-Et-4-Me-2-Py], [BI 991; 3-Et-4-Et-2-Py], [BI 992; 3-Et-4 -Pr-2-Py], [BI993; 3-Et-4-i-Pr-2-Py], [BI994; 3-Et-5-Me-2-Py], [BI995; 3-Et-5 -Et-2-Py, [BI 996; 3-Et-5-Pr-2-Py], [BI 997; 3-Et-5-i-Pr-2-Py], [BI 998; 3-Et-6 -Me-2-Py], [BI 999; 3-Et-6-Et-2-Py], [BI 1000; 3-Et-6-Pr-2-Py],

[BI1001; 3-Et-6-i-Pr-2-Py], [BI1002; 3-Pr-4-Me-2-Py], [BI1003; 3-Pr-4-Et-2-Py], [BI 1004; 3-Pr-4-Pr-2-Py], [BI 1005; 3-Pr-4-i-Pr-2-Py], [BI 1006; 3-Pr-5-Me-2-Py], [BI 1007; 3-Pr-5-Et-2-Py], [BI 1008; 3-Pr-5-Pr-2-Py], [BI 1009; 3-Pr-5-i-Pr-2-Py], [BI1010; 3-Pr-6-Me-2-Py], [BI1011; 3-Pr-6-Et-2-Py], [BI1012; 3-Pr-6-Pr-2-Py], [BI1013] 3-Pr-6-i-Pr-2-Py !, [BI 1014; 4-Me-5-Me-2-Py], [BI 1015; 4-Me-5-Et-2-Py], [BI 1016; 4-Me-5-Pr-2-Py !, [BI 1017; 4-Me-5-i-Pr-2-Py], [BI 1018; 4-Me-6-Me-2-Py], [BI 10 19] 4-Me-6-Et-2-Py !, [BI 1020; 4-Me-6-Pr-2-Py], [BI 1021; 4-Et-5-Me-2-Py], [BI 1022; -Et-5-Et-2-Py], [BI 1023; 4-Et-5-Pr-2-Py], [BI 1024; 4-Et-5-i-Pr-2-Py], [BI 1025; -Et-6-Me-2-Py], [BI 1026; 4-Et-6-Et-2-Py], [BI 1027; 4-Et-6-Pr-2-Py], [BI 1028; 4-Et -6-i-Pr-2-Py !, [BI 1029; 4-i-Pr-5-Me-2-Py], [BI 1030; 4-i-Pr-5-Et-2-Py], [BI 1031] 4-i-Pr-5-Pr-2-Py !, [BI1032; 4-i-Pr-5-i-Pr-2-Py], [BI1033; 4-i-Pr-6-Me-2 -Py], [BI1034; 4-i-Pr-6-Et-2-Py], [BI1035; 4-i-Pr-6-Pr-2-Py], [BI1036; 4-i-Pr-6 -i-Pr-2-Py, [BI 1037; 5-Me-6-Me-2-Py], [BI 1038; 5-Me-6-Et-2-Py], [BI 1039; 5-Me-6 -Pr-2-Py], [BI 1040; 5-Me-6-i-Pr-2-Py], [BI 1 041; 5-Et-6-Me-2-Py], [BI1042; 5-Et-6-Et-2-Py], [BI1043; 5-Et-6-Pr-2-Py], [BI1044; 5-Et-6-i-Pr-2-Py !, [BI 1045; 5-Pr-6-Me-2-Py], [BI 1046; 5-Pr-6-Et-2-Py], [BI 1047; 5-Pr-6-Pr-2-Py], [BI1048; 5-Pr-6-i-Pr-2-Py], [BI1049; 5-i-Pr-6-Me-2-Py], BI 1050; 5-i-Pr-6-Et-2-Py], [BI 1051; 5-i-Pr-6-Pr-2-Py], [BI 1052; 5-i-Pr-6-i-Pr- 2-Py], [BI1053; 3-Me-4-Me-5-Me-2-Py], [BI1054; 3-Et-4-Me-5-Me-2-Py], [BI 1055; 3- Pr-4-Me-5-Me-2-Py], [BI 1056; 3-i-Pr-4-Me-5-Me-2-Py], [BI 1057; 3-Me-4-Me-6- 6 Me-2-Py !, [BI 1058; 3-Et-4-Me-6-Me-2-Py], [BI 1059; 3-Pr-4-Me-6-Me-2-Py], [BI 1060; 3-i-Pr-4-Me-6-Me-2-Py, [BI 1061; 3-Me-5-Me-6-Me-2-Py], [BI 1062; 3-Et-5-Me- 6-Me-2-Py, [BI1063; 3-Pr-5-Me-6-Me-2-Py], [BI1064; 3-Me-4-Et-5-Me-2-Py], BI 1065; 3-Me-4-Pr-5-Me-2-Py], [BI 1066; 3-Me-4-i-Pr-5-Me-2-Py], [BI 10 67; 4-Me-5- Me-6-Me-2-Py], [BI 1068; 4-Et-5-Me-6-Me-2-Py], [BI 1069; 4-Pr-5-Me-6-Me-2-Py] [BI 1070; 4-i-Pr-5-Me-6-Me-2-Py], [BI 1071; 4-Me-5-Et-6-Me-2-Py], [BI 1072; 4-Me- 5-Pr-6-Me-2-Py, [BI1073; 4-Me-5-i-Pr-6-Me-2-Py], [BI1074; 3-Me-4-Me-5-Et- 2-Py], [BI1075; 3-Me-4-Me-5-Pr-2-Py], [BI1076; 3-Me-4-Me-5-i-Pr- 2-Py], [BI 1077; 4-Me-5-Me-6-Et-2-Py], [BI 1078; 4-Me-5-Me-6-Pr-2-Py], [BI 1079; Me-5-Me-6-i-Pr-2-Py], [BI 1080; 3-Me-4-Me-6-Et-2-Py], [BI 1081; 3-Me-4-Me-6- 6 Pr-2-Py, [BI1082; 3-Me-4-Me-6-i-Pr-2-Py], [BI1083; 3-Me-5-Et-6-Me-2-Py], BI 1084; 3-Me-5-Pr-6-Me-2-Py], [BI 1085; 3-Me-5-i-Pr-6-Me-2-Py], [BI 1086; 3-Me-5- Me-6-Et-2-Py !, [BI 1087; 3-Me-5-Me-6-Pr-2-Py], [BI 1088; 3-Me-5-Me-6-i-Pr-2- Py], [BI1089; 3-Me-4-Me-5-Me-6-Me-2-Py], [BI1090; 3-F-2-Py], [BI1091; 3-Cl-2-Py] [BI1092; 3-Br-2-Py], [BI1093; 3-I-2-Py], [BI1094; 4-F-2-Py], [BI 1095; 4-Cl-2-Py], [BI 1094; BI 1096; 4-Br-2-Py], [BI 1097; 4-I-2-Py], [BI 1098; 5-F-2-Py], [BI 10 99; 5-Cl-2-Py], [BI 1100] 5-Br-2-Py],

[BI 1101; 5-I-2-Py], [BI 1102; 6-F-2-Py], [BI 1103; 6-Cl-2-Py], [BI 1104; 6-Br-2-Py], [BI 1 105] 6-I-2-Py !, [BI 1106; 3-Me-4-F-2-Py], [BI 1107; 3-Me-4-Cl-2-Py], [BI 1108; 3-Me-4 -Br-2-Py, [BI 1109; 3-Me-4-I-2-Py], [BI 1110; 3-Me-5-F-2-Py], [BI 1111; 3-Me-5-Cl -2-Py !, [BI 1112; 3-Me-5-Br-2-Py], [BI 1113; 3-Me-5-I-2-Py], [BI 1114; 3-Me-6-F-2 -Py], [BI 1115; 3-Me-6-Cl-2-Py], [BI 1116; 3-Me-6-Br-2-Py], [BI 1 117; 3-Me-6-I-2-Py ], [BI 1118; 3-Et-4-F-2-Py], [BI 1119; 3-Et-4-Cl-2-Py], [BI 1120; 3-Et-4-Br-2-Py], [BI 1121; 3-Et-4-I-2-Py], [BI 1122; 3-Et-5-F-2-Py], [BI 1123; 3-Et-5-Cl-2-Py], [BI 1 124] 3-Et-5-Br-2-Py !, [BI 1125; 3-Et-5-I-2-Py], [BI 1126; 3-Et-5-F-2-Py], [BI 1127; -Et-5-Cl-2-Py], [BI 1128; 3-Et-5-Br-2-Py], [BI 1129; 3-Et-5-I-2-Py], [BI 1130; 3-F -4-Me-2-Py !, [BI1131; 3-F-4-Et-2-Py], [BI1132; 3-F-4-F-2-Py], [BI 1133; 3-F-4] -Cl-2-Py, [BI 1134; 3-F-4-Br-2-Py], [BI 1 135; 3-F-4-I-2-Py], [BI 1136; 3-F-5-Me -2-Py, [BI 1137; 3-F-5-Et-2-Py], [BI 1138; 3-F-5-F-2-Py], [BI 1 139; 3-F-5-Cl-2 -Py], [BI 1140; 3-F-5-Br-2-Py], [BI 1141; 3-F-5-I-2-Py], [BI 1142; 3-F-6-Me-2-Py ], [BI 1143; 3-F-6-Et-2-Py], [BI 1144; 3-F-6-F-2-Py], [BI 1] 145; 3-F-6-Cl-2-Py !, [BI 1146; 3-F-6-Br-2-Py], [BI 1147; 3-F-6-I-2-Py], [BI 1148; 3-Cl-4-Me-2-Py !, [BI 1149; 3-Cl-4-Et-2-Py], [BI 1150; 3-Cl-4-F-2-Py], [BI 1151; Cl-4-Cl-2-Py !, [BI1152; 3-Cl-4-Br-2-Py], [BI1153; 3-Cl-4-I-2-Py], [BI 1154; 3-Cl- 5-Me-2-Py, [BI 1 155; 3-Cl-5-Et-2-Py], [BI 1156; 3-Cl-5-F-2-Py], [BI 1 157; 3-Cl-5- Cl-2-Py, [BI 1158; 3-Cl-5-Br-2-Py], [BI 1159; 3-Cl-5-I-2-Py], [BI 1 160; 3-Cl-6-Me- 2-Py], [BI1161; 3-Cl-6-Et-2-Py], [BI1162; 3-Cl-6-F-2-Py], [BI1163; 3-Cl-6-Cl-2-] Py], [BI 1164; 3-Cl-6-Br-2-Py], [BI 1165; 3-Cl-6-I-2-Py], [BI 1166; 3-Br-4-Me-2-Py] , [BI1167; 3-Br-4-Et-2-Py], [BI 1168; 3-Br-4-F-2-Py], [BI 1169; 3-Br-4-Cl-2-Py], [BI 1 16; BI1170; 3-Br-4-Br-2-Py], [BI1171; 3-Br-4-I-2-Py], [BI1172; 3-Br-5-Me-2-Py], [BI1173; 3-Br-5-Et-2-Py !, [BI 1174; 3-Br-5-F-2-Py], [BI 1175; 3-Br-5-Cl-2-Py], [BI 1176; 3- Br-5-Br-2-Py], [BI 1177; 3-Br-5-I-2-Py], [BI 1178; 3-Br-6-Me-2-Py], [BI 1179; 3-Br- 6-Et-2-Py, [BI 1180; 3-Br-6-F-2-Py], [BI 1181; 3-Br-6-Cl-2-Py], [BI 1182; 3-Br-6- Br-2-Py, [BI1183; 3-Br-6-I-2-Py], [BI 1184; 3-I-4-Me-2-Py], [BI 1185; 3-I-4-Et- 2-Py], [BI 1186; 3-I-4-F-2-Py], [BI 1187; 3-I-4-Cl -2-Py !, [BI 1188; 3-I-4-Br-2-Py], [BI 1189; 3-I-4-I-2-Py], [BI 1190; 3-I-5-Me-2 -Py], [BI1191; 3-I-5-Et-2-Py], [BI1192; 3-I-5-F-2-Py], [BI1193; 3-I-5-Cl-2-Py ], [BI 1194; 3-I-5-Br-2-Py], [BI 1195; 3-I-5-I-2-Py], [BI 1196; 3-I-6-Me-2-Py], [BI 1197; 3-I-6-Et-2-Py], [BI 1198; 3-I-6-F-2-Py], [BI 1199; 3-I-6-Cl-2-Py], [BI 1200] 3-I-6-Br-2-Py],

[BI 1201; 3-I-6-I-2-Py], [BI 1202; 4-Me-5-F-2-Py], [BI 1203; 4-Me-5-Cl-2-Py], [BI 1204] 4-Me-5-Br-2-Py !, [BI 1205; 4-Me-5-I-2-Py], [BI 1206; 4-Me-6-F-2-Py], [BI 1207; -Me-6-Cl-2-Py], [BI 1208; 4-Me-6-Br-2-Py], [BI 1209; 4-Me-6-I-2-Py], [BI 1210; 4-Et -5-F-2-Py !, [BI 1211; 4-Et-5-Cl-2-Py], [BI 1212; 4-Et-5-Br-2-Py], [BI 1213; 4-Et-5 -I-2-Py, [BI 1214; 4-Et-6-F-2-Py], [BI 1215; 4-Et-6-Cl-2-Py], [BI 1216; 4-Et-6-Br -2-Py, [BI 1217; 4-Et-6-I-2-Py], [BI 1218; 4-F-5-Me-2-Py], [BI 1219; 4-F-5-Et-2 -Py], [BI1220; 4-F-5-F-2-Py], [BI1221; 4-F-5-Cl-2-Py], [BI1222; 4-F-5-Br-2-Py] ], [BI1223; 4-F-5-I-2-Py], [BI1224; 4-F-6-Me-2-Py], [BI1225; 4-F-6-Et-2-Py], [BI1226; 4-F-6-F-2-Py], [BI1227; 4-F-6-Cl-2-Py], [BI1228; 4-F-6-Br-2-Py], [BI1229] 4-F-6-I-2-Py !, [BI 1230; 4-Cl-5-Me-2-Py], [BI 1231; 4-Cl-5-Et-2-Py], [BI 1232; 4] -Cl-5-F-2-Py], [BI 1233; 4-Cl-5-Cl-2-Py], [BI 1234; 4-Cl-5-Br-2-Py], [BI 1235; 4-Cl -4-I-2-Py, [BI 1236; 4-Cl-6-Me-2-Py], [BI 1237; 4-Cl-6-Et-2-Py], [BI 1238; 4-Cl-6 -F-2-Py, [BI 1239; 4-Cl-6-Cl-2-Py], [BI 1240; 4-Cl-6-Br-2-Py], [BI 1241; 4-Cl-6-I -2-Py, [BI 1242; 4-Br-5-Me-2-Py], [BI 1243; 4-Br-5-Et-2-Py ], [BI 1244; 4-Br-5-F-2-Py], [BI 1245; 4-Br-5-Cl-2-Py], [BI 1246; 4-Br-5-Br-2-Py], [BI 1247; 4-Br-5-I-2-Py], [BI 1248; 4-Br-6-Me-2-Py], [BI 1249; 4-Br-6-Et-2-Py], [BI 1 250] 4-Br-6-F-2-Py !, [BI 1251; 4-Br-6-Cl-2-Py], [BI 1252; 4-Br-6-Br-2-Py], [BI 1253; 5-Br-6-I-2-Py !, [BI 1254; 5-Me-6-F-2-Py], [BI 1 255; 5-Me-6-Cl-2-Py], [BI 1 256; 5-Me -6-Br-2-Py, [BI1257; 5-Me-6-I-2-Py], [BI 1258; 5-Et-6-F-2-Py], [BI 1259; 5-Et-6 -Cl-2-Py, [BI 1260; 5-Et-6-Br-2-Py], [BI 1261; 5-Et-6-I-2-Py], [BI 1262; 5-F-6-Me -2-Py !, [BI 1263; 5-F-6-Et-2-Py], [BI 1264; 5-F-6-F-2-Py], [BI 1265; 5-F-6-Cl-2] -Py], [BI1266; 5-F-6-Br-2-Py], [BI1267; 5-F-6-I-2-Py], [BI1268; 5-Cl-6-Me-2-Py] ], [BI 1269; 5-Cl-6-Et-2-Py], [BI 1270; 5-Cl-6-F-2-Py], [BI 1271; 5-Cl-6-Cl-2-Py], [BI 1272; 5-Cl-6-Br-2-Py], [BI 1273; 5-Cl-6-I-2-Py], [BI 1274; 5-Br-6-Me-2-Py], [BI 1275] 5-Br-6-Et-2-Py !, [BI 1276; 5-Br-6-F-2-Py], [BI 1277; 5-Br-6-Cl-2-Py], [BI 1278; 5] -Br-6-Br-2-Py], [BI 1279; 5-Br-6-I-2-Py], [BI 1280; 5-I-6-Me-2-Py], [BI 1281; 5-I -6-Et-2-Py !, [BI 1282; 5-I-6-F-2-Py], [BI 1283; 5-I-6-Cl-2-Py], [BI 1284; 5-I-6 -Br-2-Py, [BI 1285; 5-I-6-I-2-Py], [BI 1286; 3-F-4-F-5-. F-2-Py !, [BI 1287; 4-F-5-F-6-F-2-Py], [BI 1 288; 3-F-4-F-6-F-2-Py], [BI 1 289; 3-F-5-F-6-F-2-Py !, [BI 1290; 3-Me-4-F-6-Me-2-Py], [BI 1291; 3-Et-4-F-6- 6 Me-2-Py !, [BI1292; 3-F-4-F-6-Me-2-Py], [BI1293; 3-Cl-4-F-6-Me-2-Py], [BI1294; 3-Br-4-F-6-Me-2-Py], [BI 1295; 3-I-4-F-6-Me-2-Py], [BI 1296; 3-Me-5-F-6- 6 Me-2-Py, [BI 1297; 3-Et-5-F-6-Me-2-Py], [BI 1298; 3-F-5-F-6-Me-2-Py], [BI 1299; 3-Cl-5-F-6-Me-2-Py], [BI 1300; 3-Br-5-F-6-Me-2-Py],

[BI 1301; 3-I-5-F-6-Me-2-Py], [BI 1302; 3-Me-4-Me-5-Cl-2-Py], [BI 1303; 3-Et-4-Me -5-Cl-2-Py !, [BI1304; 3-F-4-Me-5-Cl-2-Py], [BI 1305; 3-Cl-4-Me-5-Cl-2-Py], [BI 1306; 3-Br-4-Me-5-Cl-2-Py], [BI 1307; 3-I-4-Me-5-Cl-2-Py], [BI 1308; 4-F-5-Me -6-Me-2-Py, [BI 1309; 4-F-5-Me-6-Et-2-Py], [BI 1310; 4-F-5-Me-6-F-2-Py], [BI1311; 4-F-5-Me-6-Cl-2-Py], [BI1312; 4-F-5-Me-6-Br-2-Py], [BI1313; 4-F-5-Me -4-I-2-Py, [BI 1314; 4-Me-5-F-6-Me-2-Py], [BI 1315; 4-Me-5-F-6-Et-2-Py], [BI 1316; 4-Me-5-F-6-F-2-Py], [BI 1317; 4-Me-5-F-6-Cl-2-Py], [BI 1318; 4-Me-5-F -6-Br-2-Py, [BI 1319; 4-Me-5-F-6-I-2-Py], [BI 1320; 4-Me-5-Cl-6-Et-2-Py], [BI 1321; 4-Et-5-Cl-6-Et-2-Py], [BI 1322; 4-F-5-Cl-6-Et-2-Py], [BI 1323; 4-Cl-5-Cl -4-Et-2-Py], [BI1324; 4-Br-5-Cl-6-Et-2-Py], [BI 1325; 4-I-5-Cl-6-Et-2-Py], [BI 1326; 2-PYM], [BI 1327; 4-Me-2-PYM], [BI 1328; 4-Et-2-PYM], [BI 1329; 4-Pr-2-PYM], [BI 1330; 4-i -Pr-2-PYM], [BI1331; 5-Me-2-PYM], [BI1332; 5-Et-2-PYM], [BI 1333; 5-Pr-2-PYM], [BI 1334; 5-i -Pr-2-PYM], [BI 1335; 4-Me-5-Me-2-PYM], [BI 1336; 4-Me-5-Et-2-PYM], [BI 1337; 4-Me-5-Pr -2-PYM], [BI1 338; 4-Me-5-i-Pr-2-PYM], [BI 1339; 4-Et-5-M e-2-PYM], [BI 1340; 4-Et-5-Et-2-PYM], [BI 1341; 4-Et-5-Pr-2-PYM], [BI 1342; 4-Et-5-i- Pr-2-PYM], [BI1343; 4-Pr-5-Me-2-PYM], [BI1344; 4-Pr-5-Et-2-PYM], [BI1345; 4-Pr-5-Pr- 2-PYM], [BI 1346; 4-Pr-5-i-Pr-2-PYM], [BI 1347; 4-i-Pr-5-Me-2-PYM], [BI 1348; 4-i-Pr- 5-Et-2-PYM], [BI 1349; 4-i-Pr-5-Pr-2-PYM], [BI 1350; 4-i-Pr-5-i-Pr-2-PYM], [BI 1351; 4-Me-6-Me-2-PYM], [BI1352; 4-Me-6-Et-2-PYM], [BI1353; 4-Me-6-Pr-2-PYM], [BI1354; Me-6-i-Pr-2-PYM], [BI 1355; 4-Et-6-Me-2-PYM], [BI 1356; 4-Et-6-Et-2-PYM], [BI 1 357; Et-6-Pr-2-PYM], [BI 1358; 4-Et-6-i-Pr-2-PYM], [BI 1359; 4-Pr-6-Me-2-PYM], [BI 1 360; Pr-6-Et-2-PYM], [BI1361; 4-Pr-6-Pr-2-PYM], [BI1362; 4-Pr-6-i-Pr-2-PYM], [BI1363; i-Pr-6-Me-2-PYM], [BI 1364; 4-i-Pr-6-Et-2-PYM], [BI 1365; 4-i-Pr-6-Pr-2-PYM], [BI 1 365; BI 1 366; 4-i-Pr-6-i-Pr-2-PYM], [BI 1367; 4-Me-5-Me-6-Me-2-PYM], [BI 1 368; 4-Me-5-Et- 6-Me-2-PYM], [BI1369; 4-Et-5-Me-6-Me-2-PYM], [BI1370; 4-Me-5-Pr-6-Me-2-PYM], [BI BI1371; 4-Pr-5-Me-6-Me-2-PYM], [BI1372; 4-Me-5-i-Pr-6-Me-2-PYM], [BI1373; 4-i-Pr- 5-Me-6-Me-2-PYM], [BI 1374; 4-F-2-PYM], [BI 1375; 4-Cl-2-PYM], [BI 1376; 4-Br-2-PYM], [BI 1 376; BI 1377; 4-I-2 -PYM], [BI 1378; 5-F-2-PYM], [BI 1379; 5-Cl-2-PYM], [BI 1 380; 5-Br-2-PYM], [BI 1381; 5-I-2-PYM] ], [BI1382; 4-Me-5-F-2-PYM], [BI1383; 4-Me-5-Cl-2-PYM], [BI1384; 4-Me-5-Br-2-PYM], [BI 1385; 4-Me-5-I-2-PYM], [BI 1386; 4-Et-5-F-2-PYM], [BI 1387; 4-Et-5-Cl-2-PYM], [BI 1388] 4-Et-5-Br-2-PYM], [BI1389; 4-Et-5-I-2-PYM], [BI1390; 4-F-5-F-2-PYM], [BI1391; -F-5-Cl-2-PYM], [BI1392; 4-F-5-Br-2-PYM], [BI1393; 4-F-5-I-2-PYM], [BI1394; 4-F -5-Me-2-PYM], [BI 1395; 4-Cl-5-F-2-PYM], [BI 1396; 4-Cl-5-Cl-2-PYM], [BI 1397; 4-Cl-5 -Br-2-PYM], [BI 1398; 4-Cl-5-I-2-PYM], [BI 1399; 4-Cl-5-Me-2-PYM], [BI 1400; 4-Cl-5-Et -2-PYM],

[BI 1401; 4-Br-5-F-2-PYM], [BI 1402; 4-Br-5-Cl-2-PYM], [BI 1403; 4-Br-5-Br-2-PYM], [BI 1404] 4-Br-5-I-2-PYM !, [BI 1405; 4-Br-5-Me-2-PYM], [BI 1406; 4-Br-5-Et-2-PYM], [BI 1407; -I-5-F-2-PYM], [BI 1408; 4-I-5-Cl-2-PYM], [BI 1409; 4-I-5-Br-2-PYM], [BI 1410; 4-I -5-I-2-PYM !, [BI 1411; 4-I-5-Me-2-PYM], [BI 1412; 4-I-5-Et-2-PYM], [BI 1413; 4-F-5. -F-6-F-2-PYM], [BI 1414; 4-Me-5-F-6-Me-2-PYM], [BI 1415; 4-Et-5-F-6-Me-2-PYM] ], [BI 1416; 4-F-5-F-6-Me-2-PYM], [BI 1417; 4-Cl-5-F-6-Me-2-PYM], [BI 14 18; 4-Me-5] -Cl-6-Me-2-PYM], [BI 1419; 4-Et-5-Cl-6-Me-2-PYM], [BI 1420; 4-Me-5-Br-6-Me-2-PYM ], [BI 1421; 4-Et-5-Br-6-Me-2-PYM], [BI 1422; 4-Me-5-I-6-Me-2-PYM], [BI 1423; 4-Et-5. -I-6-Me-2-PYM].

  In addition, the present compounds AJ1-BJ1 to AJ32-BJ366 can also be obtained according to the above-mentioned method.

The present compounds AJ1-BJ1 to AJ32-BJ366 are compounds represented by the following formula (AJBJ).

[Wherein, X ^{121 to} X ¹²⁸ each represent a substituent corresponding to each of the substituent numbers (MJ1) AJ 1 to AJ 32 shown below, wherein E ¹¹⁰ represents a substituent number (MJ 2) BJ 1 shown below ~ BJ 366 is represented. ]
For example, the present compound AJ1-BJ1, in the compounds of formula (AJBJ), X ¹²¹ ~X ¹²⁸ substituents ID ^{MJ1 (X 121, X 122,} X 125, X 126 and X ¹²⁷ is a hydrogen atom, X ¹²³ Is a sulfur atom, X ¹²⁸ is an oxygen atom, X ¹²⁴ is a fluorine, and E ¹¹⁰ is a compound in which the substituent number (MJ 2) is BJ 1 (phenyl group), and is represented by the following formula.

[Substituent group number ^{(MJ1); X 121, X} 122, X 123, X 124, X 125, X 126, X 127, X 128]: [AJ1; H, H, S, F, H, H, H, O], [AJ2; H, H, S, Cl, H, H, O], [AJ 3; H, H, S, Br, H, H, O], [AJ 4; H, H, S, I, H, H, H, O], [AJ 5; H, H, S, Me, H, H, H, O], [AJ 6; H, H, S, Et, H, H, H, H, O], [AJ7; H, H, S, Pr, H, H, H, O], [AJ 8; H, H, S, i-Pr, H, H, H, O], [AJ 9; H, H, S, Bu, H, H, H, O, [AJ10; H, H, S, i-Bu, H, H, H, O], [AJ 11; H, H, S, Sec-Bu, H, H, H, O], [AJ 12; H, H, S, t-Bu, H, H, H, O], [AJ 13; H, H, S, c-Pr, H, H, H, O], [AJ14; H, H, S, c-Bu, H, H, H, O], [AJ 15; H, H, S, OMe, H, H, H, O], [AJ 16; H, H, S, OEt, H, H, H, O, [AJ 17; H, H, S, OPr, H, H, H, O], [AJ 18; H, H, S, Oi-Pr, H, H, H, O], [AJ 19; H, H, S, OBu, H, H, H, O], [AJ 20; H, H, S, Oi-Bu, H, H, H, O], [AJ 20 AJ 21; H, H, S, O-sec-Bu, H, H, H, O], [AJ 22; H, H, S, Ot-Bu, H, H, H, O], [AJ 23; H, _{H, S, CH 2 F,} H, H, H, O], [AJ24; H, H, S, CHF 2, H, H, H, O], [AJ25; H, H, S, CF3, H , H, H, O], [AJ26; H, H, S, CH 2 CF 3, H, H, H, O], [AJ27; H, H, S, CH 2 CHF 2, H, H, H , O], [AJ28; H , H, S, OCH 2 F, H, H, H, O], [AJ29; H, H, S, OCHF 2, H, H, H, O], [AJ30; _{H, H, S, OCF 3} , H, H, H, O], [AJ31; H, H, S, OCH 2 CF 3, H, H, H, O], [AJ32; H, H, S, _{OCH 2 CHF 2, H, H} , H, O].

[Substituent number (MJ2); E ¹¹⁰ ]: [BJ1: Ph], [BJ 2: 2-F-Ph], [BJ 3: 3-F-Ph], [BJ 4: 4-F-Ph], [BJ 5 : 2-Cl-Ph], [BJ 6: 3-Cl-Ph], [BJ 7: 4-Cl-Ph], [BJ 8: 2-Br-Ph], [BJ 9: 3-Br-Ph], [BJ 10 : 4-Br-Ph, [BJ 11: 2-OMe-Ph], [BJ 12: 3-OMe-Ph], [BJ 13: 4-OMe-Ph], [BJ 14: 2-CF ₃ -Ph], [BJ 14: BJ15: 3-CF ₃ -Ph], [BJ 16: 4-CF ₃ -Ph], [BJ 17: 3-Py], [BJ 18: 2-F-3-Py], [BJ 19: 4-F-3-] Py], [BJ20: 5-F-3-Py], [BJ 21: 6-F-3-Py], [BJ 22: 2-Cl-3-Py], [BJ 23: 4-Cl-3-Py] , [BJ24: 5-Cl-3-Py], [BJ 25: 6-Cl-3-Py], [BJ 26: 2-Br-3-Py], [BJ 27: 4-Br-3-Py], [BJ 26: BJ28: 5-Br-3-Py], [BJ 29: 6-Br-3-Py], [BJ 30: 2-OMe-3-Py], [BJ 31: 4-OMe-3-Py], [BJ 32: 5-OMe-3-Py, [BJ33: 6-OMe-3-Py], [BJ 34: 2-CF ₃ -3-Py], [BJ 35: 4-CF ₃ -3-Py], [BJ 36: 5-CF ₃ -3-Py, [BJ 37: 6-CF ₃ -3-Py], [BJ 38: 2-OMe -3-Py], [BJ 39: 6-F -2-OMe -3- Py] , [BJ 40: 6-Cl-2-OMe-3-Py], [BJ 41: 6-Br-2-OMe-3-Py], [BJ 42: 6-Me-2-OMe-3-Py], BJ 43: 6-Et-2-OMe-3-Py], [BJ 44: 6-Pr-2-OMe-3-Py], [BJ 45: 6-i-Pr-2-OMe-3-Py], BJ 46: 6-CN-2-OMe-3-Py], [BJ 47: 6-CF ₃ -2-OMe-3-Py], [BJ 48: 2, 6-diOMe-3-Py], [BJ 49: 6] -OEt-2-OMe-3-Py], [BJ50: 6-OPr-2-OMe-3-Py], [BJ51: 6-i-OPr-2-OMe-3-Py], [BJ 52: 4] -F-2-OMe-3-Py], [BJ 53: 4, 6-diF-2-OMe- 3-Py], [BJ 54: 4-F-6-Cl-2-OMe-3-Py], [BJ 55: 4-F-6-Br-2-OMe-3-Py], [BJ 56: 4- F-6-Me-2-OMe-3-Py], [BJ 57: 4-F-6-Et-2-OMe-3-Py], [BJ 58: 4-F-6-Pr-2-OMe- 3-Py], [BJ59: 4-F-6-i-Pr-2-OMe-3-Py], [BJ60: 4-F-6-CN-2-OMe-3-Py], [BJ61: _{4-F-6-CF 3} -2-OMe-3-Py], [BJ62: 4-F-2,6-diOMe-3-Py], [BJ63: 4-F-6-OEt-2-OMe -3-Py, [BJ 64: 4-F-6-OPr-2-OMe-3-Py], [BJ 65: 4-F-6-i-OPr-2-OMe-3-Py], [BJ 66] : 4-Cl-2-OMe-3-Py], [BJ 67: 4-Cl-6-F-2-OMe-3-Py], [BJ 68: 4, 6-diCl-2-OMe-3-Py] ], [BJ69: 4-Cl-6-Br-2-OMe-3-Py], [BJ70: 4-Cl-6-Me-2-OMe-3-Py], [BJ 71: 4-Cl-6] -Et-2-OMe-3-Py], [BJ72: 4-Cl-6-Pr-2-OMe-3-Py], [BJ73: 4-Cl-6-i-Pr-2-OMe-3 -Py], [BJ74: 4- Cl-6-CN-2-OMe-3-Py], [BJ75: 4-Cl-6-CF 3 -2-OMe-3-Py], [BJ76: 4- Cl-2, 6-diOMe-3-Py], [BJ 77: 4-Cl-6-OEt-2-OMe-3-Py], [BJ 78: 4-Cl-6-OPr-2-OMe-3- 3 Py], [BJ 79: 4-Cl-6-i-OPr-2-OMe-3-Py], [BJ 80: 2,4-diOMe-3-Py], [BJ 81: 6-F-2,4- diOMe-3-Py], [BJ82: 6-Cl-2,4-diOMe-3-Py], [BJ 83: 6-Br-2,4-diOMe-3-Py], [BJ 84: 6-Me- 2,4-diOMe-3-Py], [BJ 85: 6-Et-2,4-diOMe-3-Py], [BJ 86: 6-Pr-2,4-diOMe-3-Py], [BJ 87: 6-i-Pr-2,4- diOMe-3-Py], [BJ88: 6-CN-2,4-diOMe-3-Py], [BJ89: 6-CF 3 -2,4-diOMe-3 -P y], [BJ90: 2,4,6-triOMe-3-Py], [BJ91: 6-OEt-2,4-diOMe-3-Py], [BJ92: 6-OPr-2,4-diOMe- 3-Py, [BJ 93: 6-i-OPr-2,4-diOMe-3-Py], [BJ 94: 5-F-2-OMe-3-Py], [BJ 95: 5, 6-diF- 2-OMe-3-Py], [BJ96: 5-F-6-Cl-2-OMe-3-Py], [BJ 97: 5-F-6-Br-2-OMe-3-Py], [BJ 97 BJ 98: 5-F-6-Me-2-OMe-3-Py], [BJ 99: 5-F-6-Et-2-OMe-3-Py], [BJ 100: 5-F-6-Pr- 2-OMe-3-Py],

[BJ 101: 5-F-6-i-Pr-2-OMe-3-Py], [BJ 102: 5-F-6-CN-2-OMe-3-Py], [BJ 103: 5-F-6] _{-CF 3 -2-OMe-3-} Py], [BJ104: 5-F-2,6-diOMe-3-Py], [BJ105: 5-F-6-OEt-2-OMe-3-Py] , [BJ106: 5-F-6-OPr-2-OMe-3-Py], [BJ107: 5-F-6-i-OPr-2-OMe-3-Py], [BJ108: 4, 5- diF-2-OMe-3-Py], [BJ109: 4,5,6-triF-2-OMe-3-Py], [BJ110: 4,5-diF-6-Cl-2-OMe-3-3] Py], [BJ 111: 4, 5-diF-6-Br-2-OMe-3-Py], [BJ 112: 4, 5-diF-6-Me-2-OMe-3-Py], [BJ 113: 4,5-diF-6-Et-2-OMe-3-Py], [BJ114: 4, 5-diF-6-Pr-2-OMe-3-Py], [BJ 115: 4, 5-diF- 6-i-Pr-2-OMe-3-Py], [BJ116: 4, 5-diF-6-CN-2-OMe-3-Py], [BJ 117: 4, 5-diF-6-CF ₃ -2-OMe-3-Py, [BJ118: 4, 5-diF-2, 6-diOMe-3-Py], [BJ 119: 4, 5-diF-6-OEt-2-OMe-3-Py ], [BJ120: 2-OEt-3-Py], [BJ 121: 6-F-2-OEt-3-Py], [BJ 122: 6-Cl-2-OEt-3-Py], [BJ 123: 6] -Br-2-OEt-3-Py], [BJ 124: 6-Me-2-OEt-3-Py], [BJ 125: 6-Et-2-OEt-3-Py], [BJ 126: 6-Pr -2-OEt-3-Py !, [BJ 127: 6-i-Pr-2-OEt-3-Py], [BJ 128: 6-CN-2-OEt-3-Py], [BJ 129: 6-CF] _{3 -2-OEt-3-Py} ], [BJ130: 6-OMe-2-OEt-3-Py], [BJ131: 2,6-diOEt-3-Py], [BJ132: 6-OPr-2- OEt-3-Py, [BJ133: 6-i-OPr-2-OEt-3-Py], [BJ 134: 4-F-2-OEt-3-Py], [BJ 135: 4, 6-diF- 2-OEt-3-Py], [BJ 136: 4-F-6-Cl-2-OEt-3- Py], [BJ 137: 4-F-6-Br-2-OEt-3-Py], [BJ 138: 4-F-6-Me-2-OEt-3-Py], [BJ 139: 4-F- 6-Et-2-OEt-3-Py], [BJ140: 4-F-6-Pr-2-OEt-3-Py], [BJ141: 4-F-6-i-Pr-2-OEt- 3-Py], [BJ142: 4-F-6-CN-2-OEt-3-Py], [BJ143: 4-F-6-CF 3 -2-OEt-3-Py], [BJ144: 4 -F-6-OMe-2-OEt-3-Py], [BJ145: 4-F-2, 6-diOEt-3-Py], [BJ 146: 4-F-6-OPr-2-OEt-3 -Py], [BJ 147: 4-F-6-i-OPr-2-OEt-3-Py], [BJ 148: 4-Cl-2-OEt-3-Py], [BJ 149: 4-Cl-6 -F-2-OEt-3-Py], [BJ150: 4, 6-diCl-2-OEt-3-Py], [BJ 151: 4-Cl-6-Br-2-OEt-3-Py], [BJ152: 4-Cl-6-Me-2-OEt-3-Py], [BJ 153: 4-Cl-6-Et-2-OEt-3-Py], [BJ 154: 4-Cl-6-Pr -2-OEt-3-Py !, [BJ 155: 4-Cl-6-i-Pr-2-OEt-3-Py], [BJ 156: 4-Cl-6-CN-2-OEt-3-Py ], [BJ157: 4-Cl -6-CF 3 -2-OEt-3-Py], [BJ158: 4-Cl-6-OMe-2-OEt-3-Py], [BJ159: 4-Cl- 2,6-diOEt-3-Py], [BJ160: 4-Cl-6-OPr-2-OEt-3-Py], [BJ161: 4-Cl-6-i-OPr-2-OEt-3- 3 Py], [BJ162: 4-OMe-2-OEt-3-Py], [BJ163: 6-F-4-OMe-2-OEt-3-Py], [BJ 164: 6-Cl-4-OMe- 2-OEt-3-Py], [BJ 165: 6-Br-4-OMe-2-OEt-3-Py], [BJ 166: 6-Me-4-OMe-2-OEt-3-Py], BJ 167: 6-Et-4-OMe-2-OEt-3-Py], [BJ 168: 6-Pr-4-OMe-2-OEt-3-Py], [BJ 169: 6-i-Pr-4- OMe-2-OEt-3-Py], [BJ 170: 6-CN-4-OMe-2-OEt-3-Py], [BJ 1 _{71: 6-CF 3 -4-} OMe-2-OEt-3-Py], [BJ172: 2,6-diOMe-2-OEt-3-Py], [BJ173: 4-OMe-2,6-diOEt -3-Py], [BJ 174: 6-OPr-4-OMe-2-OEt-3-Py], [BJ 175: 6-i-OPr-4-OMe-2-OEt-3-Py], [BJ 176] : 5-F-2-OEt-3-Py], [BJ177: 5, 6-diF-2-OEt-3-Py], [BJ 178: 5-F-6-Cl-2-OEt-3-Py] ], [BJ 179: 5-F-6-Br-2-OEt-3-Py], [BJ 180: 5-F-6-Me-2-OEt-3-Py], [BJ 181: 5-F-6] -Et-2-OEt-3-Py], [BJ 182: 5-F-6-Pr-2-OEt-3-Py], [BJ 183: 5-F-6-i-Pr-2-OEt-3 -Py], [BJ184: 5- F-6-CN-2-OEt-3-Py], [BJ185: 5-F-6-CF 3 -2-OEt-3-Py], [BJ186: 5- F-6-OMe-2-OEt-3-Py !, [BJ187: 5-F-2, 6-diOEt-3-Py], [BJ 188: 5-F-6-OPr-2-OEt-3- 3 Py], [BJ189: 5-F-6-i-OPr-2-OEt-3-Py], [BJ190: 4, 5-diF-2-OEt-3-Py], [BJ 191: 4, 5, 6 6-triF-2-OEt-3-Py !, [BJ192: 4, 5-diF-6-Cl-2-OEt-3-Py], [BJ 193: 4, 5-diF-6-Br-2-] OEt-3-Py], [BJ194: 4,5-diF-6-Me-2-OEt-3-Py], [BJ195: 4,5-diF-6-Et-2-OEt-3-Py] , [BJ 196: 4, 5-diF-6-Pr-2-OEt-3-Py], [BJ 197: 4, 5-diF-6-i-Pr-2-OEt-3-Py], [BJ 198: 4,5-diF-6-CN-2-OEt-3-Py], [BJ 199: 4, 5-diF-6-CF ₃ -2-OEt-3-Py], [BJ 200: 4, 5-diF -6-OMe-2-OEt-3-Py],

[BJ 201: 4, 5-diF-2, 6-diOEt-3-Py], [BJ 202: 2-OMe-Ph], [BJ 203: 4-F-2-OMe-Ph], [BJ 204: 4-Cl] -2-OMe-Ph !, [BJ 205: 4-Br-2-OMe-Ph], [BJ 206: 4-Me-2-OMe-Ph], [BJ 207: 4-Et-2-OMe-Ph], [BJ208: 4-Pr-2-OMe-Ph], [BJ209: 4-i-Pr-2-OMe-Ph], [BJ210: 4-CN-2-OMe-Ph], [BJ 211: 4-CF] ₃ -2-OMe-Ph !, [BJ 212: 2,4-diOMe-Ph], [BJ 213: 4-OEt-2-OMe-Ph], [BJ 214: 4-OPr-2-OMe-Ph], [BJ 214 BJ 215: 4-i-OPr-2-OMe-Ph], [BJ 216: 6-F-2-OMe-3-Py], [BJ 217: 4, 6-diF-2-OMe-Ph], [BJ 218: 4-F-4-Cl-2-OMe-Ph !, [BJ219: 6-F-4-Br-2-OMe-Ph], [BJ220: 6-F-4-Me-2-OMe-Ph] , [BJ 221: 6-F-4-Et-2-OMe-Ph], [BJ 222: 6-F-4-Pr-2-OMe-Ph], [BJ 223: 6-F-4-i-Pr- 2-OMe-Ph], [ BJ224: 6-F-4-CN-2-OMe-Ph], [BJ225: 6-F-4-CF 3 -2-OMe-Ph], [BJ226: 6-F -2,4-diOMe-Ph], [BJ 227: 6-F-4-OEt-2-OMe-Ph], [BJ 228: 6-F-4-OPr-2-OMe-Ph], [BJ 229: 6] -F-4-i-OPr-2-OMe-Ph], [BJ 230: 6-Cl-4-OMe-Ph], [BJ 231: 6-Cl-4-F-2-OMe-Ph], [BJ 232] 4,6-diCl-2-OMe-Ph !, [BJ233: 6-Cl-4-Br-2-OMe-Ph], [BJ234: 6-Cl-4-Me-2-OMe-Ph], [BJ 235: 6-Cl-4-Et-2-OMe-Ph], [BJ 236: 6-Cl-4-Pr-2-OMe-Ph], [BJ 237: 6-Cl-4-i-Pr-2 -OMe-Ph], [BJ238: 6-Cl-4-CN-2-OMe-Ph], [BJ239: 6-Cl-4-CF 3 -2-OMe-Ph], [BJ240: 6-Cl- 2,4-diOMe -Ph], [BJ241: 6-Cl-4-OEt-2-OMe-Ph], [BJ 242: 6-Cl-4-OPr-2-OMe-Ph], [BJ 243: 6-Cl-4-i -OPr-2-OMe-Ph], [BJ244: 2, 6-diOMe-Ph], [BJ 245: 4-F-2, 6-diOMe-Ph], [BJ 246: 4-Cl-2, 6-diOMe -Ph], [BJ 247: 4-Br-2, 6-diOMe-Ph], [BJ 248: 4-Me-2, 6-diOMe-Ph], [BJ 249: 4-Et-2, 6-diOMe-Ph] ], [BJ 250: 4-Pr-2, 6-diOMe-Ph], [BJ 251: 4-i-Pr-2, 6-diOMe-Ph], [BJ 252: 4-CN-2, 6-diOMe-Ph] ], [BJ 253: 4-CF ₃ -2, 6-diOMe-Ph], [BJ 254: 2, 4, 6-triOMe-Ph], [BJ 255: 4-OEt-2, 6-diOMe-Ph], [BJ 255 BJ 256: 4-OPr-2, 6-diOMe-Ph], [BJ 257: 4-i-OPr-2, 6-diOMe-Ph], [BJ 258: 5-F-2-OMe-Ph], [BJ 259: 4,5-diF-2-OMe-Ph], [BJ260: 5-F-4-Cl-2-OMe-Ph], [BJ261: 5-F-4-Br-2-OMe-Ph], [BJ 261 BJ 262: 5-F-4-Me-2-OMe-Ph], [BJ 263: 5-F-4-Et-2-OMe-Ph], [BJ 264: 5-F-4-Pr-2-OMe- Ph], [BJ 265: 5-F-4-i-Pr-2-OMe-Ph], [BJ 266: 5-F-4-CN-2-OMe-Ph], [BJ 267: 5-F-4- 4 _{CF 3 -2-OMe-Ph]} , [BJ268: 5-F-2,4-diOMe-Ph], [BJ269: 5-F-4-OEt-2-OMe-Ph], [BJ270: 5-F -4-OPr-2-OMe-Ph !, [BJ 271: 5-F-4-i-OPr-2-OMe-Ph], [BJ 272: 5, 6-diF-2-OMe-Ph], [BJ 273 : 4,5,6-triF-2-OMe-Ph], [BJ274: 5,6-diF-4-Cl-2-OMe-Ph], [BJ275: 5,6-diF-4-Br-2 -OMe-Ph], [BJ276: 5,6-diF-4-Me-2-OMe-Ph], [BJ 277: 5,6-diF-4-Et-2-OMe-Ph], [BJ J278: 5,6-diF-4-Pr-2-OMe-Ph], [BJ279: 5,6-diF-4-i-Pr-2-OMe-Ph], [BJ280: 5,6-diF- 4-CN-2-OMe- Ph], [BJ281: 5,6-diF-4-CF 3 -2-OMe-Ph], [BJ282: 5,6-diF-2,4-diOMe-Ph], [BJ283: 5,6-diF-4-OEt-2-OMe-Ph], [BJ284: 2-OEt-Ph], [BJ285: 4-F-2-OEt-Ph], [BJ 286: 4-Cl -2-OEt-Ph !, [B 287: 4-Br-2-OEt-Ph], [BJ 288: 4-Me-2-OEt-Ph], [BJ 289: 4-Et-2-OEt-Ph], [BJ290: 4-Pr-2-OEt-Ph], [BJ291: 4-i-Pr-2-OEt-Ph], [BJ292: 4-CN-2-OEt-Ph], [BJ293: 4-Ac -2-OEt-Ph !, [BJ 294: 4-CF ₃ -2-OEt-Ph], [BJ 295: 4-OMe-2-OEt-Ph], [BJ 296: 2,4-diOEt-Ph], [BJ 296 BJ 297: 4-OPr-2-OEt-Ph !, [BJ 298: 4-i-OPr-2-OEt-Ph], [BJ 299: 6-F-2-OEt-Ph], [BJ 300: 4, 6- diF-2-OEt-Ph],

[BJ301: 6-F-4-Cl-2-OEt-Ph], [BJ 302: 6-F-4-Br-2-OEt-Ph], [BJ 303: 6-F-4-Me-2-OEt -Ph], [BJ 304: 6-F-4-Et-2-OEt-Ph], [BJ 305: 6-F-4-Pr-2-OEt-Ph], [BJ 306: 6-F-4-i -Pr-2-OEt-Ph] , [BJ307: 6-F-4-CN-2-OEt-Ph], [BJ308: 6-F-4-CF 3 -2-OEt-Ph], [BJ309: 6-F-4-OMe-2-OEt-3-Ph !, [BJ310: 6-F-2,4-diOEt-Ph], [BJ 311: 6-F-4-OPr-2-OEt-Ph] , [BJ 312: 6-F-4-i-OPr-2-OEt-Ph], [BJ 313: 6-Cl-2-OEt-Ph], [BJ 314: 6-Cl-4-F-2-OEt- Ph], [BJ 315: 4, 6-diCl-2-OEt-Ph], [BJ 316: 6-Cl-4-Br-2-OEt-Ph], [BJ 317: 6-Cl-4- Me-2 OEt-Ph !, [BJ 318: 6-Cl-4-Et-2-OEt-Ph], [BJ 319: 6-Cl-4-Pr-2-OEt-Ph], [BJ 320: 6-Cl-4- i-Pr-2-OEt- Ph], [BJ321: 6-Cl-4-CN-2-OEt-Ph], [BJ322: 6-Cl-4-CF 3 -2-OEt-Ph], [BJ323 6-Cl-4-OMe-2-OEt-Ph !, [BJ324: 6-Cl-2,4-diOEt-Ph], [BJ325: 6-Cl-4-OPr-2-OEt-Ph], [BJ326: 6-Cl-4-i-OPr-2-OEt-Ph], [BJ 327: 6-OMe-2-OEt-Ph], [BJ 328: 4-F-6-OMe-2-OEt-Ph] ], [BJ 329: 4-Cl-6-OMe-2-OEt-Ph], [BJ 330: 4-Br-6-OMe-2-OEt-Ph], [BJ 331: 4-Me-6-OMe-2] -OEt-Ph, [BJ332: 4-Et-6-OMe-2-OEt-Ph], [BJ333: 4-Pr-6-OMe-2-OEt-Ph], [BJ334: 4-i-Pr -6-OMe-2-OEt-Ph !, [BJ 335: 4-CN-6-OMe-2-OEt-Ph], [BJ 336: 4-CF ₃ -6-OMe-2-OEt-Ph], BJ 337: 4, 6-diOMe- 2-OEt-Ph, [BJ 338: 6-OMe-2,4-diOEt-Ph], [BJ 339: 4-OPr-6-OMe-2-OEt-Ph], [BJ 340: 4-i-OPr- 6-OMe-2-OEt-Ph !, [BJ341: 5-F-2-OEt-Ph], [BJ 342: 4, 5-diF-2-OEt-Ph], [BJ 343: 5-F-4- 4 Cl-2-OEt-Ph !, [BJ 344: 5-F-4-Br-2-OEt-Ph], [BJ 345: 5-F-4-Me-2-OEt-Ph], [BJ 346: 5- F-4-Et-2-OEt-Ph !, [BJ347: 5-F-4-Pr-2-OEt-Ph], [BJ 348: 5-F-4-i-Pr-2-OEt-Ph] , [BJ 349: 5-F-4-CN-2-OEt-Ph], [BJ 350: 5-F-4-CF ₃ -2-OEt-Ph], [BJ 351: 5-F-4-OMe-2 -OEt-Ph, [BJ352: 5-F-2,4-diOEt-Ph], [BJ 353: 5-F-4-OPr-2-OEt-Ph], [BJ 354: 5-F-4-i -OPr-2-OEt-Ph], [BJ 355: 5, 6-diF-2-OEt-Ph], [BJ 356: 4, 5, 6 triF-2-OEt-Ph], [BJ 357: 5, 6 -diF-4-Cl-2-OEt-Ph], [BJ358: 5,6-diF-4-Br-2-OEt-Ph], [BJ 359: 5,6-diF-4-Me-2-OEt -Ph], [BJ360: 5,6-diF-4-Et-2-OEt-Ph], [BJ 361: 5,6-diF-4-Pr-2-OEt-Ph], [BJ 362: 5, 6 -diF-4-i-Pr-2-OEt-Ph], [BJ363: 5,6-diF-4-CN-2-OEt-Ph], [BJ 364: 5,6-diF-4-CF _3- 2-OEt-Ph], [BJ365: 5,6-diF-4-OMe-2-OEt-Ph], [BJ366: 5,6-diF-2,4-diOEt-Ph].

  Further, the present compounds AK1-BK1 to AK2688-BK846 can also be obtained according to the method described above.

The present compounds AK1-BK1 to AK2688-BK846 are compounds represented by the following formula (AKBK).
[Wherein, X ¹³⁰ to X ¹³⁹ are each respectively in the corresponding a substituent formula, E ¹¹¹ to substituent number (MK1) AK1~AK2688 shown below, substituents numbers shown below (MK2) BK1~ Each represents a substituent corresponding to BK 846. ]
For example, the AK1-BK1, wherein in the compound represented by (AKBK), X ¹³⁰ ~X ¹³⁹ substituents number AK1 (X ¹³⁴ is a sulfur atom, X ¹³⁹ is an oxygen atom, X ¹³⁰ to X ¹³³ and X ¹³⁵ to X ¹³⁸ represents a hydrogen atom, and E ¹¹¹ represents a compound in which the substituent number (MK2) is BK1 (pyrazol-1-yl group), and is represented by the following formula.

[Substituent group number ^{(MK1); X 130, X} 131, X 132, X 133, X 134, X 135, X 136, X 137, X 138, X 139]: [AK1; H, H, H, H, O, H, H, H, H, O], [AK2; H, H, H, H, H, O, F, H, H, O], [AK 3; H, H, H, H, O, Cl, H, H, H, O], [AK4; H, H, H, H, O, Br, H, H, H, O], [AK5; H, H, H, H, O, I, I, H, H, H, O], [AK6; H, H, H, H, O, Me, H, H, H, O], [AK7; H, H, H, H, H, O, Et, H, O] H, H, O], [AK 8; H, H, H, H, H, O, Pr, H, H, H, O], [AK 9; H, H, H, H, O, i-Pr, H, H, H, O], [AK10; H, H, H, H, H, O, Bu, H, H, H, O], [AK11; H, H, H, H, O, i-Bu, H, H H, H, O], [AK12; H, H, H, H, O, sec-Bu, H, H, H, O], [AK13; H, H, H, H, O, t-Bu, H, H, H, O], [AK 14; H, H, H, H, O, c-Pr, H, H, H, O], [AK 15; H, H, H, H, O, c- Bu, H, H, H, O], [AK 16; H, H, H, H, O, OBu, H, H, H, O], [AK 17; H, H, H, H, O, Oi- Bu, H, H, H, O], [AK 18; H, H, H, H, O, O-sec-Bu, H, H, H, O], [AK 19; H, H, H, H, O, _{O, CH 2 F, H,} H, H, O], [AK20; H, H, H, H, O, CHF 2, H, H, H, O], [AK21; H, H, H, H , O, CF ₃ , H, H, H, O], [AK 22; H, H, H, H, H, O, OCH ₂ F, H, H, H, O], [AK 23; H, H, H, H] _{H, O, OCHF 2, H} , H, H, O], [AK24; H, H, H, H, O, OCF 3, H, H, H, O], [AK25; H, H, H, Me, O, H, H, H, H, O, [AK26; H, H, H, Me, O, F, H, H, H, O], [AK 27; H, H, H, Me, O, Cl, H, H, H, O, [AK 28; H, H, H, Me, O, Br, H, H, H, O], [AK 29; H, H, H, Me, O, I, H, H, H, O] [AK30; H, H, H, Me, O, Me, H, H, H, O], [AK 31; H, H, H, Me, O, Et, H, H, H, O], [AK 32 H, H, H, H, Me, O, Pr, H, H, H, O], [AK33; H, H, H, Me, O, i-Pr, H, H, H, O], [AK34 H, H, H, H, Me, O, Bu, H, H, H, O], [AK 35; H, H, H, Me, O, i-Bu, H, H, H, O], [AK 36 H, H, H, H, Me, O, sec-Bu, H, H, H, O], [AK 37; H, H, H, Me, O, t-Bu, H, H, H, O], [AK 38; H, H, H, Me, O, c-Pr, H, H, H, O], [AK 39; H, H, H, Me, O, c-Bu, H, H, H, O , [AK40; H, H, H, Me, O, OBu, H, H, H, O], [AK 41; H, H, H, Me, O, Oi-Bu, H, H, H, O] H, H, H, Me, O, O-sec-Bu, H, H, H, O], [AK 43; H, H, H, Me, O, CH ₂ F, H, H] , H, O], [AK44 ; H, H, H, Me, O, CHF 2, H, H, H, O], [AK45; H, H, H, Me, O, CF 3, H, H , H, O], [AK 46; H, H, H, Me, O, OCH ₂ F, H, H, H, O], [AK 47; H, H, H, Me, O, OCHF ₂ , H, H, H, H, O], [ AK48; H, H, H, Me, O, OCF 3, H, H, H, O], [AK49; H, H, H, Me, O, OCF 3, H, H, H, O], [AK 50; H, H, H, Et, O, H, H, H, H, O], [AK 51; H, H, H, Et, O, F, H, H, H, H, O], [AK 52; H, H, H, Et, O, Cl, H, H, O], [AK 53; H, H, H, Et, O, Br, H, H, H, H, O], [AK 54; H, H, H, Et, O, I, H, H, H, O], [AK 55; H, H, H, Et, O, Me, H, H, H, O] [AK56; H, H, H, H, Et, O, Et, H, H, H, O], [AK57; H, H, H, Et, O, Pr, H, H, H, O], [AK56; AK58; H, H, H, H, Et, O, i-Pr, H, H, H, O], [AK59; H, H, H, Et, O, Bu, H, H, H, O], [[Ak59; AK60; H, H, H, Et, O , i-Bu, H, H, H, O], [AK 61; H, H, H, Et, O, sec-Bu, H, H, H, O], [AK 62; H, H, H, Et] , O, t-Bu, H, H, H, O], [AK 63; H, H, H, Et, O, c-Pr, H, H, H, O], [AK 64; H, H, H] , Et, O, c-Bu, H, H, H, O], [AK 65; H, H, H, Et, O, OBu, H, H, H, O], [AK 66; H, H, H] , Et, O, Oi-Bu, H, H, H, O], [AK 67; H, H, H, Et, O, O-sec-Bu, H, H, H, O], [AK 68; H , H, H, Et, O , CH 2 F, H, H, H, O], [AK69; H, H, H, Et, O, CHF 2, H, H, H, O], [AK70; H, H, H, Et, O, CF 3, H, H, H, O], [AK71; H, H, H, Et, O, OCH 2 F, H, H, H, O], [AK72 ; H, H, H, Et , O, OCHF 2, H, H, H, O], [AK73; H, H, H, Et, O, OCF 3, H, H, H, O], [AK74 ; H, H, H, Et , O, OCF 3, H, H, H, O], [AK75; H, H, H, Pr, O, H, H, H, H, O], [AK76; H, H, H, H, Pr, O, F, H, H, H, O], [AK 77; H, H, H, Pr, O, Cl, H, H, H, O], [AK 78; H, H, H, H, Pr, O, Br, H, H, H, O], [AK 79; H, H, H, Pr, O, I, H, H, H, O], [AK 80; H, H, H, H] H, Pr, O, Me, H, H, H, O], [AK 81; H, H, H, Pr, O, Et, H, H, H, O], [AK 82; H, H, H, H Pr, O, Pr, H, H, H, O], [AK 83; H, H, H, Pr, O, i-Pr, H, H, H, O], [AK 84; H, H, H, H] Pr, O, Bu, H, H, H, O], [AK 85; H, H, H, Pr, O, i-Bu, H, H, H, O], [AK 86; H, H, H, H] Pr, O, sec-Bu, H, H, H, O], [AK 87; H, H, H, Pr, O, t-Bu, H, H, H, O], [AK 88; H, H, H H, Pr, O, c-Pr, H, H, H, O], [AK 89; H, H, H, Pr, O, c-Bu, H, H, H, O], [AK 90; H, H, H H, H, Pr, O, OBu, H, H , H, O], [AK 91; H, H, H, H, Pr, O, Oi-Bu, H, H, H, O], [AK 92; H, H, H, H, Pr, O, O-sec-Bu , H, H, H, O ], [AK93; H, H, H, Pr, O, CH 2 F, H, H, H, O], [AK94; H, H, H, Pr, O, CHF _{2, H, H, H,} O], [AK95; H, H, H, Pr, O, CF 3, H, H, H, O], [AK96; H, H, H, Pr, O, OCH ₂ F, H, H, H, O], [AK 97; H, H, H, Pr, O, OCHF ₂ , H, H, H, O], [AK 98; H, H, H, Pr, O, OCF ₃ , H, H, H, O], [AK 99; H, H, H, H, Pr, O, OCF ₃ , H, H, H, O], [AK 100; H, H, H, i-Pr, O, H, H, H, H, O],

[AK101; H, H, H, i-Pr, O, F, H, H, O], [AK102; H, H, H, i-Pr, O, Cl, H, H, H, O , [AK103; H, H, H, i, Pr, O, Br, H, H, H, O], [AK104; H, H, H, i, Pr, O, I, H, H, H] , O], [AK 105; H, H, H, i-Pr, O, Me, H, H, H, O], [AK 106; H, H, H, i-Pr, O, Et, H, H , H, O], [AK 107; H, H, H, i-Pr, O, Pr, H, H, H, O], [AK 108; H, H, H, i-Pr, O, i-Pr , H, H, H, O], [AK109; H, H, H, i-Pr, O, Bu, H, H, H, O], [AK 110; H, H, H, i-Pr, O] , i-Bu, H, H, H, O], [AK 111; H, H, H, i-Pr, O, sec-Bu, H, H, H, O], [AK 112; H, H, H] , i-Pr, O, t-Bu, H, H, H, O], [AK113; H, H, H, i-Pr, O, c-Pr, H, H, H, O], [AK114 H, H, H, i-Pr, O, c-Bu, H, H, H, O], [AK115; H, H, H, i-Pr, O, OBu, H, H, H, O ], [AK116; H, H, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK117; H, H, H, i-Pr, O, O-sec-Bu , H, H, H, O ], [AK118; H, H, H, i-Pr, O, CH 2 F, H, H, H, O], [AK119; H, H, H, i-Pr , O, CHF ₂ , H, H, H, O], [AK 120; H, H, H, i-Pr, O, CF ₃ , H, H, H, O], [AK 121; H, H, H] , i-Pr, O, OCH 2 F, H, H, H, O], [AK122; H, H, H, i-Pr, O, OCHF 2, H, H, H, O], [AK123; H, H, H, i- Pr, O, OCF 3, H, H, H, O], [AK124; H, H, H, i-Pr, O, OCF 3, H, H, H, O] [AK 125; H, H, H, H, O, O, H, H, H, O], [AK 126; H, H, H, O, O, F, H, H, H, O], [A AK127; H, H, H, OMe, O, Cl, H, H, H, O], [AK 128; H, H, H, OMe, O, Br, H, H, H, O], [AK 129; H, H, H, H, OMe, O, I, H, H, O], [AK130; H, H, H, OMe, O, Me, H, H, H, O], [AK 131; H, H, H, H, OMe, O, Et, H, H, H, O], [AK132; H, H, H, OMe, O, Pr, H, H, H, O], [AK133; H, H, H, OMe, O, i-Pr, H, H, H, O], [AK134; H, H, H, OMe, O, Bu, H, H, H, O], [AK135; H, H, H, OMe, O, i-Bu, H, H, H, O], [AK 136; H, H, H, OMe, O, sec-Bu, H, H, H, O], [AK 137; H, H, H, H, OMe, O, t-Bu, H, H, H, O], [AK 138; H, H, H, OMe, O, c-Pr, H, H, H, O], [[ AK139; H, H, H, OMe, O, c-Bu, H, H, H, O], [AK 140; H, H, H, OMe, O, OBu, H, H, H, O], [AK 140; AK141; H, H, H, H, OMe, O, Oi-Bu, H, H, H, O], [AK142; H, H, H, OMe, O, O-sec-Bu, H, H, H, O], [AK143; H, H, H, OMe, O, CH 2 F, H, H, H, O], [AK144; H, H, H, OMe, O, CHF 2, H, H, H , O], [aK145; H , H, H, OMe, O, CF 3, H, H, H, O], [AK146; H, H, H, OMe, O, OCH 2 F, H, H, H, O], [AK 147; H, H, H, OMe, O, OCHF ₂ , H, H, H, O], [AK 148; H, H, H, OMe, O, OCF ₃ , H, H, H, O], [AK149; H, H, H, OMe, O, OCF 3, H, H, H, O], [AK150; H, H, H, F, O, H, H, H, H H, H, H, F, O, F, H, H, O], [AK152; H, H, H, F, O, Cl, H, H, H, O] ], [AK153; H, H, H, H, F, O, Br, H, H, O], [AK 154; H, H, H, F, O, I, H, H, H, O], [AK 155; H, H, H, F, O, Me, H, H, H, O], [AK 156; H, H, H, F, O, Et, H, H, H, O], [AK 157 H, H, H, H, F, O, Pr, H, H, H, O], [AK158; H, H, H, H F, O, i-Pr, H, H, H, O], [AK 159; H, H, H, F, O, Bu, H, H, H, O], [AK 160; H, H, H, H] F, O, i-Bu, H, H, H, O], [AK 161; H, H, H, F, O, sec-Bu, H, H, H, O], [AK 162; H, H, H, H] H, F, O, t-Bu, H, H, H, O], [AK 163; H, H, H, F, O, c-Pr, H, H, H, O], [AK 164; H, H, H, H, F, O, c-Bu, H, H, H, O], [AK165; H, H, H, F, O, OBu, H, H, H, O], [AK166; H, H, H, H, F, O, Oi-Bu, H, H, H, O], [AK 167; H, H, H, F, O, O-sec-Bu, H, H, H, O], [[A] AK168; H, H, H, F, O, CH 2 F, H, H, H, O], [AK169; H, H, H, F, O, CHF 2, H, H, H, O], [AK170; H, H, H , F, O, CF 3, H, H, H, O], [AK171; H, H, H, F, O, OCH 2 F, H, H, H, O] , [AK172; H, H, H, F, O, OCHF 2, H, H, H, O], [AK173; H, H, H, F, O, OCF 3, H, H, H, O] , [AK174; H, H, H, F, O, OCF 3, H, H, H, O], [AK175; H, H, H, Cl, O, H, H, H, H, O], [AK176; H, H, H, H, Cl, O, F, H, H, O], [AK 177; H, H, H, Cl, O, Cl, H, H, H, O], [AK178 H, H, H, H, Cl, O, Br, H, H, H, O], [AK 179; H, H, H, Cl, O, I, H, H, H, O], [AK 180; H , H, H, Cl, O, Me, H, H, H, O], [AK181; H, H, H, H, Cl, O, Et, H, H, H, O], [AK 182; H, H , H, Cl, O, Pr, H, H, H, O], [AK 183; H, H, H, Cl, O, i-Pr, H, H, H, O], [AK 184; H, H , H, Cl, O, Bu, H, H, H, O], [AK 185; H, H, H, Cl, O, i-Bu, H, H, H, O], [AK 186; H, H , H, Cl, O, sec-Bu, H, H, H, O], [AK 187; H, H, H, H, Cl, O, t-Bu, H, H, H, O], [AK 188; H , H , H, Cl, O, c-Pr, H, H, H, O], [AK 189; H, H, H, H, Cl, O, c-Bu, H, H, H, O], [AK190; H , H, H, Cl, O, OBu, H, H, H, O], [AK191; H, H, H, H, Cl, O, Oi-Bu, H, H, H, O], [AK192; H , H, H, Cl, O , O-sec-Bu, H, H, H, O], [AK193; H, H, H, Cl, O, CH 2 F, H, H, H, O], [AK194; H, H, H , Cl, O, CHF 2, H, H, H, O], [AK195; H, H, H, Cl, O, CF 3, H, H, H, O], [AK196; H, H, H , Cl, O, OCH 2 F, H, H, H, O], [AK197; H, H, H, Cl, O, OCHF 2, H, H, H, O] , [AK198; H, H, H, Cl, O, OCF 3, H, H, H, O], [AK199; H, H, H, Cl, O, OCF 3, H, H, H, O] [AK200; H, H, H, Br, O, H, H, H, H, O],

[AK201; H, H, H, H, Br, O, F, H, H, O], [AK 202; H, H, H, Br, O, Cl, H, H, H, O], [AK203 H, H, H, H, Br, O, Br, H, H, H, O], [AK 204; H, H, H, H, Br, O, I, H, H, H, O], [AK 205; H , H, H, Br, O, Me, H, H, H, O], [AK 206; H, H, H, H, Br, O, Et, H, H, H, O], [AK 207; H, H , H, Br, O, Pr, H, H, H, O], [AK208; H, H, H, Br, O, i-Pr, H, H, H, O], [AK209; H, H] , H, Br, O, Bu, H, H, H, O], [AK210; H, H, H, Br, O, i-Bu, H, H, H, O], [AK211; H, H , H, Br, O, sec-Bu, H, H, H, O], [AK 212; H, H, H, H, Br, O, t-Bu, H, H, H, O], [AK 213; H , H, H, Br, O, c-Pr, H, H, H, O], [AK214; H, H, H, H, Br, O, c-Bu, H, H, H, O], [AK215 H, H, H, H, Br, O, OBu, H, H, H, O], [AK 216; H, H, H, H, Br, O, Oi-Bu, H, H, H, O], [AK217 ; H, H, H, Br , O, O-sec-Bu, H, H, H, O], [AK218; H, H, H, Br, O, CH 2 F, H, H, H, O ], [AK219; H, H , H, Br, O, CHF 2, H, H, H, O], [AK220; H, H, H, Br, O, CF 3, H, H, H, O ], [AK221; H, H , H, Br, O, OCH 2 F, H, H, H, O], [AK222; H, H, H, Br, O, OCHF 2, H, H, H, O], [AK223; H, H, H, Br, O, OCF 3, H, H, H, O], [AK224; H, H, H, Br, O, OCF 3, H, H, H, O], [AK 225; H, Me, H, H, O, H, H, H, H, O], [AK 226; H, Me, H, H, O, F, H, H, H, O] [AK227; H, Me, H, H, O, Cl, H, H, H, O], [AK228; H, Me, H, H, O, Br, H, H, H, O], [AK227; AK229; H, Me, H, H, O, I, H, H, H, O], [AK230; H, Me, H, H, O, Me, H, H] , H, O], [AK 231; H, Me, H, H, O, Et, H, H, H, O], [AK 232; H, Me, H, H, O, Pr, H, H, H , O], [AK233; H, Me, H, H, O, i-Pr, H, H, H, O], [AK234; H, Me, H, H, O, Bu, H, H, H , O], [AK235; H, Me, H, H, O, i-Bu, H, H, H, O], [AK236; H, Me, H, H, O, sec-Bu, H, H , H, O], [AK 237; H, Me, H, H, O, t-Bu, H, H, H, O], [AK 238; H, Me, H, H, O, c-Pr, H , H, H, O], [AK 239; H, Me, H, H, O, c-Bu, H, H, H, O], [AK 240; H, Me, H, H, O, OBu, H] H, H, O], [AK241; H, Me, H, H, O, Oi-Bu, H, H, H, O], [AK 242; H, Me, H, H, O, O-sec -Bu, H, H, H, O], [AK243; H, Me, H, H, O, CH 2 F, H, H, H, O], [AK244; H, Me, H, H, O _{, CHF 2, H, H,} H, O], [AK245; H, Me, H, H, O, CF 3, H, H, H, O], [AK246; H, Me, H, H, O , OCH ₂ F, H, H, H, O], [AK247; H, Me, H, H, O, OCHF ₂ , H, H, H, O], [AK248; H, Me, H, H, O _{O, OCF 3, H, H} , H, O], [AK249; H, Me, H, Me, O, H, H, H, H, O], [AK250; H, Me, H, Me, O , F, H, H, H, O], [AK 251; H, Me, H, Me, O, Cl, H, H, H, O], [AK 252; H, Me, H, Me, O, Br] , H, H, H, O], [AK 253; H, Me, H, Me, O, I, H, H, H, O], [AK 254; H, Me, H, Me, O, Me, H] , H, H, O], [AK255; H, Me, H, Me, O, Et, H, H, H, O], [AK256; H, Me, H, Me, O, Pr, H, H] , H, O], [AK 257; H, Me, H, Me, O, i-Pr, H, H, H, O], [AK258; H, Me, H, Me, O, Bu, H, H] , H, O], [AK 259; H, Me, H, Me, O, i-Bu, H, H, H, O], [AK 260; H, Me, H, Me, O, sec-Bu, H, H, H, O], [AK 261; H, Me, H, Me, O, t-Bu, H, H, H, O] [AK262; H, Me, H, Me, O, c-Pr, H, H, H, O], [AK 263; H, Me, H, Me, O, c-Bu, H, H, H, H, O], [AK 264; H, Me, H, Me, O, OBu, H, H, H, O], [AK 265; H, Me, H, Me, O, Oi-Bu, H, H, H, O], [AK266; H, Me, H, Me, O, O-sec-Bu, H, H, H, O], [AK267; H, Me, H, Me, O, CH 2 F, H, H, H, O], [ AK268; H, Me, H, Me, O, CHF 2, H, H, H, O], [AK269; H, Me, H, Me, O, CF 3, H, H, H, O], [AK 270; H, Me, H, Me, O, OCH ₂ F, H, H, H, O], [AK 271; H, Me, H, Me, O, OCHF ₂ , H , H, H, O], [AK272; H, Me, H, Me, O, OCF 3, H, H, H, O], [AK273; H, Me, H, Me, O, OCF 3, H , H, H, O], [AK 274; H, Me, H, Et, O, H, H, H, H, O], [AK 275; H, Me, H, Et, O, F, H, H] , H, O], [AK 276; H, Me, H, Et, O, Cl, H, H, H, O], [AK 277; H, Me, H, Et, O, Br, H, H, H] H, Me, H, Et, O, I, H, H, H, O], [AK 279; H, Me, H, Et, O, Me, H, H, H, O] H, Me, H, Et, O, Et, H, H, H, O], [AK 281; H, Me, H, Et, O, Pr, H, H, H, O], [AK282; H, Me, H, Et, O, i-Pr, H, H, H, O], [AK 283; H, Me, H, Et, O, Bu, H, H, H, O], [AK284; H, Me, H, Et, O, i-Bu, H, H, H, O], [AK 285; H, Me, H, Et, O, sec-Bu, H, H, H, O H, Me, H, Et, O, t-Bu, H, H, H, O], [AK 287; H, Me, H, Et, O, c-Pr, H, H, H] , O], [AK 288; H, Me, H, Et, O, c- Bu, H, H, H, O], [AK 289; H, Me, H, Et, O, OBu, H, H, H, O], [AK 290; H, Me, H, Et, O, Oi − Bu, H, H, H, O], [AK 291; H, Me, H, Et, O, O-sec-Bu, H, H, H, O], [AK 292; H, Me, H, Et, Et _{O, CH 2 F, H,} H, H, O], [AK293; H, Me, H, Et, O, CHF 2, H, H, H, O], [AK294; H, Me, H, Et , O, CF ₃ , H, H, H, O], [AK 295; H, Me, H, Et, O, OCH ₂ F, H, H, H, O], [AK 296; H, Me, H, O _{Et, O, OCHF 2, H} , H, H, O], [AK297; H, Me, H, Et, O, OCF 3, H, H, H, O], [AK298; H, Me, H, _{Et, O, OCF 3, H} , H, H, O], [AK299; H, Me, H, Pr, O, H, H, H, H, O], [AK300; H, Me, H, Pr , O, F, H, H, H, O],

[AK301; H, Me, H, Pr, O, Cl, H, H, O], [AK302; H, Me, H, Pr, O, Br, H, H, H, O], [AK303 H, Me, H, Pr, O, I, H, H, H, O], [AK 304; H, Me, H, Pr, O, Me, H, H, H, O], [AK 305; H , Me, H, Pr, O, Et, H, H, O, [AK 306; H, Me, H, Pr, O, Pr, H, H, H, O], [AK 307; H, Me , H, Pr, O, i-Pr, H, H, H, O], [AK308; H, Me, H, Pr, O, Bu, H, H, H, O], [AK309; H, Me , H, Pr, O, i-Bu, H, H, H, O], [AK 310; H, Me, H, Pr, O, sec-Bu, H, H, H, O], [AK 311; H , Me, H, Pr, O, t-Bu, H, H, H, O], [AK 312; H, Me, H, Pr, O, c-Pr, H, H, H, O], [AK313 H, Me, H, Pr, O, c-Bu, H, H, H, O], [AK 314; H, Me, H, Pr, O, OBu, H, H, H, O], [AK 315 H, Me, H, Pr, O, Oi-Bu, H, H, H, O], [AK 316; H, Me, H, Pr, O, O-sec-Bu, H, H, H, O] H, Me, H, Pr, O, CH ₂ F, H, H, H, O], [AK 318; H, Me, H, Pr, O, CHF ₂ , H, H, H, H] O, [AK 319; H, Me, H, Pr, O, CF ₃ , H, H, O], [AK 320; H, Me, H, Pr, O, OCH ₂ F, H, H, H , O], [AK 321; H, Me, H, Pr, O, OCHF ₂ , H, H, H, O], [AK 322; H, Me, H, Pr, O, OCF ₃ , H, H, H , O], [AK323; H , Me, H, Pr, O, OCF 3, H, H, H, O], [AK324; H, Me, H, i-Pr, O, H, H, H, H, O], [AK 325; H, Me, H, i-Pr, O, F, H, H, H, O], [AK 326; H, Me, H, i-Pr, O, Cl, H, H, H, O], [AK 327; H, Me, H, i-Pr, O, Br, H, H, H, O], [AK 328; H, Me, H, i-Pr, O, I, H, H, H, O], [AK 329; H, Me, H, iP r, O, Me, H, H, H, O], [AK 330; H, Me, H, i-Pr, O, Et, H, H, H, O], [AK 331; H, Me, H, O] i-Pr, O, Pr, H, H, H, O, [AK332; H, Me, H, i-Pr, O, i-Pr, H, H, H, O], [AK333; H, Me, H, i-Pr, O, Bu, H, H, H, O], [AK 334; H, Me, H, i-Pr, O, i-Bu, H, H, H, O], [[ AK335; H, Me, H, i-Pr, O, sec-Bu, H, H, H, O], [AK336; H, Me, H, i-Pr, O, t-Bu, H, H, H H, O], [AK337; H, Me, H, i-Pr, O, c-Pr, H, H, H, O], [AK338; H, Me, H, i-Pr, O, c- Bu, H, H, H, O], [AK 339; H, Me, H, i-Pr, O, OBu, H, H, H, O], [AK 340; H, Me, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK 341; H, Me, H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK 342; H, H, Me, H, i-Pr, O, CH 2 F, H, H, H, O], [AK343; H, Me, H, i-Pr, O, CHF 2, H, H, H, O], [AK344; H, Me, H , i-Pr, O, CF 3, H, H, H, O], [AK345; H, Me, H, i-Pr, O, OCH 2 F, H, H, H, O], [AK346; H, Me, H, i-Pr, O, OCHF 2, H, H, H, O], [AK347; H, Me, H, i-Pr, O, OCF 3, H, H, H, O] , [AK348; H, Me, H, i-Pr, O, OCF 3, H, H, H, O], [AK349; H, Me, H, OMe, O, H H, H, H, O], [AK 350; H, Me, H, OMe, O, F, H, H, H, O], [AK 351; H, Me, H, OMe, O, Cl, H] H, H, O], [AK352; H, Me, H, OMe, O, Br, H, H, H, O], [AK 353; H, Me, H, OMe, O, I, H, H] , H, O], [AK 354; H, Me, H, OMe, O, Me, H, H, H, O], [AK 355; H, Me, H, OMe, O, Et, H, H, H , O], [AK 356; H, Me, H, OMe, O, Pr, H, H, H, O, [AK 357; H, Me, H, OMe, O, i-Pr, H, H, H, O], [AK 358; H, Me, H, OMe, O, Bu, H, H, H, O], [AK 359; H, Me, H, OMe, O, i-Bu, H, H, H, O], [AK 360; H, Me, H, OMe, O, sec-Bu, H, H, H, O], [AK 361; H, Me, H, OMe, O, t-Bu, H, H, H, O], [AK 362; H, Me, H, OMe, O, c-Pr, H, H, H, O], [AK 363; H, Me, H, OMe, O, c-Bu, H, H, H, O], [AK 364; H, Me, H, OMe, O, OBu, H, H, H, O], [AK365; H, Me, H, OMe, O, Oi-Bu, H, H, H, O], [AK 366; H, Me, H, OMe, O, O-sec- Bu, H, H, H, O], [AK 367; H, Me, H, OMe, O, CH ₂ F, H, H, H, O], [AK 368; H, Me, H, OMe, O, _{CHF 2, H, H, H} , O], [AK369; H, Me, H, OMe, O, CF 3, H, H, H, O], [AK370; H, Me, H, OMe, O, OCH ₂ F, H, H, H, O], [AK 371; H, Me, H, OMe, O, OCHF ₂ , H, H, H, O], [AK 372; H, Me, H, OMe, O , OCF ₃ , H, H, H, O], [AK 373; H, Me, H, OMe, O, OCF ₃ , H, H, H, O], [AK 374; H, Me, H, F, O , H, H, H, H, O], [AK 375; H, Me, H, F, O, F, H, H, H, O], [AK 376; H, Me, H, F, O, Cl , H, H, H, O], [AK 377; H, Me, H, F, O, Br, H, H, H, O], [AK 378; H, Me, H, F, O, I, H] H, H, O], [AK 379; H, Me, H, F, O, Me, H, H, H, O], [AK 380; H, Me, H, F, O, Et, H, H] , H, O], [AK 381; H, Me, H, F, O, Pr, H, H, H, O], [AK 382; H, Me, H, F, O, i-Pr, H, H , H, O], [AK 383; H, Me, H, F, O, Bu, H, H, H, O], [AK 384; H, Me, H, F, O, i-Bu, H, H] , H, O], [AK 385; H, Me , H, F, O, sec-Bu, H, H, H, O], [AK 386; H, Me, H, F, O, t-Bu, H, H, H, O], [AK 387; H , Me, H, F, O, c-Pr, H, H, H, O], [AK 388; H, Me, H, F, O, c-Bu, H, H, H, O], [AK 389] H, Me, H, F, O, OBu, H, H, H, O], [AK390; H, Me, H, F, O, Oi-Bu, H, H, H, O], [AK391] H, Me, H, F, O, O-sec-Bu, H, H, H, O], [AK 392; H, Me, H, F, O, CH ₂ F, H, H, H, O H, Me, H, F, O, CHF ₂ , H, H, H, O], [AK 394; H, Me, H, F, O, CF ₃ , H, H, H, O] H, Me, H, F, O, OCH ₂ F, H, H, H, O], [AK 396; H, Me, H, F, O, OCHF ₂ , H, H, H, O], [AK397; H, Me, H, F, O, OCF 3, H, H, H, O], [AK398; H, Me, H, F, O, OCF 3, H, H, H, O], [AK 399; H, Me, H, Cl, O, H, H, H, O], [AK 400; H, Me, H, Cl, O, F, H, H, H, O] ,

[AK 401; H, Me, H, Cl, O, Cl, H, H, O], [AK 402; H, Me, H, Cl, O, Br, H, H, H, O], [AK 403 H, Me, H, Cl, O, I, H, H, H, O], [AK 404; H, Me, H, Cl, O, Me, H, H, H, O], [AK 405; H , Me, H, Cl, O, Et, H, H, H, O], [AK 406; H, Me, H, Cl, O, Pr, H, H, H, O], [AK 407; H, Me , H, Cl, O, i-Pr, H, H, H, O], [AK 408; H, Me, H, Cl, O, Bu, H, H, H, O], [AK 409; H, Me , H, Cl, O, i-Bu, H, H, H, O], [AK 410; H, Me, H, Cl, O, sec-Bu, H, H, H, O], [AK 411; H , Me, H, Cl, O, t-Bu, H, H, H, O], [AK 412; H, Me, H, Cl, O, c-Pr, H, H, H, O], [AK 413 H, Me, H, Cl, O, c-Bu, H, H, H, O], [AK 414; H, Me, H, Cl, O, OBu, H, H, H, O], [AK 415 H, Me, H, Cl, O, Oi-Bu, H, H, H, O], [AK 416; H, Me, H, Cl, O, O-sec-Bu, H, H, H, O] ], [AK417; H, Me , H, Cl, O, CH 2 F, H, H, H, O], [AK418; H, Me, H, Cl, O, CHF 2, H, H, H, O], [AK419; H, Me, H, Cl, O, CF 3, H, H, H, O], [AK420; H, Me, H, Cl, O, OCH 2 F, H, H, H , O], [AK421; H , Me, H, Cl, O, OCHF 2, H, H, H, O], [AK422; H, Me, H, Cl, O, OCF 3, H, H, H , O], [AK423; H , Me, H, Cl, O, OCF 3, H, H, H, O], [AK424; H, Me, H, Br, O, H, H, H, H, O], [AK 425; H, Me, H, Br, O, F, H, H, O], [AK 426; H, Me, H, Br, O, Cl, H, H, H, O] [AK427; H, Me, H, Br, O, Br, H, H, O], [AK428; H, Me, H, Br, O, I, H, H, H, O], [AK 427; AK 429; H, Me, H, Br, O, Me, H, H, H H, Me, H, Br, O, Et, H, H, H, O], [AK 431; H, Me, H, Br, O, Pr, H, H, H, O] H, Me, H, Br, O, i-Pr, H, H, H, O], [AK 433; H, Me, H, Br, O, Bu, H, H, H, O] H, Me, H, Br, O, i-Bu, H, H, H, O], [AK 435; H, Me, H, Br, O, sec-Bu, H, H, H] H, Me, H, Br, O, t-Bu, H, H, H, O], [AK 437; H, Me, H, Br, O, c-Pr, H, H] , H, O], [AK 438; H, Me, H, Br, O, c-Bu, H, H, H, O], [AK 439; H, Me, H, Br, O, OBu, H, H] , H, O], [AK 440; H, Me, H, Br, O, Oi-Bu, H, H, H, O], [AK 441; H, Me, H, Br, O, O-sec-Bu , H, H, H, O], [AK 442; H, Me, H, Br, O, CH ₂ F, H, H, H, O], [AK 443; H, Me, H, Br, O, CHF _{2, H, H, H,} O], [AK444; H, Me, H, Br, O, CF 3, H, H, H, O], [AK445; H, Me, H, Br, O, OCH _{2 F, H, H, H} , O], [AK446; H, Me, H, Br, O, OCHF 2, H, H, H, O], [AK447; H, Me, H, Br, O, OCF ₃ , H, H, H, O], [AK 448; H, Me, H, Br, O, OCF ₃ , H, H, H, O], [AK 449; H, Et, H, H, O, H, H, H, H, O], [AK 450; H, Et, H, H, O, F, H, H, H, O], [AK 451; H, Et, H, H, O, Cl, H, H, H, O], [AK 452; H, Et, H, H, O, Br, H, H, H, O], [AK 453: H, Et, H, H, O, I, H, O H, H, O], [AK 454; H, Et, H, H, O, Me, H, H, H, O], [AK 455; H, Et, H, H, O, Et, H, H, H, H, O], [AK 456; H, Et, H, H, O, Pr, H, H, H, O], [AK 457; H, Et, H, H, O, i-Pr, H, H, H, H, O], [AK 458; H, Et, H, H, O, Bu, H, H, H, O], [AK 459; H, Et, H, H, O, i-Bu, H, H, H, O], [AK 460; H, Et, H, H, O, sec-Bu, H, H, H, H, O], [AK 461; H, Et, H, H, O, t, Bu, H, H, H, O], [AK 462; H, Et, H, H, O, c-Pr, H, H, H, O], [AK 463; H, Et, H, H, O, c, Bu, H, H, H, O], [AK 464; H, Et, H, H, O, O Bu, H, H, H, O], [AK 465; H, Et, H, H, O, Oi-Bu, H, H, H, O], [AK 466; H, Et, H, H, O, O-sec- Bu, H, H, H, O], [AK467; H, Et, H, H, O, CH 2 F, H, H, H, O], [AK468; H, Et, H, H, O, _{CHF 2, H, H, H} , O], [AK469; H, Et, H, H, O, CF 3, H, H, H, O], [AK470; H, Et, H, H, O, OCH ₂ F, H, H, H, O], [AK 471; H, Et, H, H, O, OCHF ₂ , H, H, H, O], [AK 472; H, Et, H, H, O] , OCF ₃ , H, H, H, O], [AK 473; H, Et, H, Me, O, H, H, H, H, O], [AK 474; H, Et, H, Me, O, F, H, H, H, O], [AK 475; H, Et, H, Me, O, Cl, H, H, H, O], [AK 476; H, Et, H, Me, O, Br, H, H, H, O], [AK 477; H, Et, H, Me, O, I, H, H, H, O], [AK 478; H, Et, H, Me, O, Me, H, H, H, O], [AK 479; H, Et, H, Me, O, Et, H, H, H, O], [AK 480; H, Et, H, Me, O, Pr, H, H, H H, O], [AK 481; H, Et, H, Me, O, i-Pr, H, H, H, O], [AK 482; H, Et, H, Me, O, Bu, H, H, H, H, O], [AK 483; H, Et, H, Me, O, i-Bu, H, H, H, O], [AK 484; H, Et, H, Me, O, sec-Bu, H, H H, H, O], [AK 485; H, Et, H, Me, O, t-Bu, H, H, H, O], [AK 486; H, Et, H, Me, O, c-Pr, H, H, H, O], [AK 487; H, Et, H, Me, O, c-Bu, H, H, H H, Et, H, Me, O, OBu, H, H, H, O], [AK 489; H, Et, H, Me, O, Oi-Bu, H, H, H] H, Et, H, Me, O, O-sec-Bu, H, H, H, O], [AK 491; H, Et, H, Me, O, CH ₂ F, H , H, H, O], [AK492; H, Et, H, Me, O, CHF 2, H, H, H, O], [AK493; H, Et, H, Me, O, CF 3, H , H, H, O], [AK 494; H, Et, H, Me, O, OCH ₂ F, H, H, H, O], [AK 495; H, Et, H, Me, O, OCHF ₂ , H, H, H, O] , [AK496; H, Et, H, Me, O, OCF 3, H, H, H, O], [AK497; H, Et, H, Me, O, OCF 3, H, H, H, O], [AK 498; H, Et, H, Et, O, H, H, H, H, O], [AK 499; H, Et, H, Et, O, F, H, H, H, H, O], [AK 500; H, Et, H, Et, O, Cl, H, H, H, O],

[AK501; H, Et, H, Et, O, Br, H, H, O], [AK 502; H, Et, H, Et, O, I, H, H, H, O], [AK503 H, Et, H, Et, O, Me, H, H, H, O], [AK 504; H, Et, H, Et, O, Et, H, H, H, O], [AK 505; H , Et, H, Et, O, Pr, H, H, H, O], [AK 506; H, Et, H, Et, O, i-Pr, H, H, H, O], [AK 507; H , Et, H, Et, O, Bu, H, H, H, O], [AK508; H, Et, H, Et, O, i-Bu, H, H, H, O], [AK509; H , Et, H, Et, O, sec-Bu, H, H, H, O], [AK510; H, Et, H, Et, O, t-Bu, H, H, H, O], [AK511 H, Et, H, Et, O, c-Pr, H, H, H, O], [AK512; H, Et, H, Et, O, c-Bu, H, H, H, O], [AK513; H, Et, H, Et, O, OBu, H, H, H, O], [AK514; H, Et, H, Et, O, Oi-Bu, H, H, H, O], [AK515; H, Et, H , Et, O, O-sec-Bu, H, H, H, O], [AK516; H, Et, H, Et, O, CH 2 F, H, H, H , O], [AK517; H , Et, H, Et, O, CHF 2, H, H, H, O], [AK518; H, Et, H, Et, O, CF 3, H, H, H , O], [AK519; H , Et, H, Et, O, OCH 2 F, H, H, H, O], [AK520; H, Et, H, Et, O, OCHF 2, H, H, H, O], [AK521; H, Et, H, Et, O, OCF 3, H, H, H, O], [AK522; H, Et, H, Et, O, OCF 3, H, H, H, O], [AK523; H, Et, H, Pr, O, H, H, H, H, O], [AK524; H, Et, H, Pr, O, F, H, H, H, H, O], [AK525; H, Et, H, Pr, O, Cl, H, H, O], [AK526; H, Et, H, Pr, O, Br, H, H, H, O] [AK527; H, Et, H, Pr, O, I, H, H, O], [AK528; H, Et, H, Pr, O, Me, H, H, H, O], [AK527; AK529; H, Et, H, Pr, O, Et, H, H, H H, Et, H, Pr, O, Pr, H, H, H, O], [AK 531; H, Et, H, Pr, O, i-Pr, H, H, H] H, Et, H, Pr, O, Bu, H, H, H, O], [AK 533: H, Et, H, Pr, O, i-Bu, H, H, H] H, Et, H, Pr, O, sec-Bu, H, H, H, O], [AK 535; H, Et, H, Pr, O, t-Bu, H, H] , H, O], [AK 536; H, Et, H, Pr, O, c-Pr, H, H, H, O], [AK 537; H, Et, H, Pr, O, c-Bu, H] H, H, O], [AK 538; H, Et, H, Pr, O, OBu, H, H, H, O], [AK 539; H, Et, H, Pr, O, Oi-Bu, H H, H, O], [AK 540; H, Et, H, Pr, O, O-sec-Bu, H, H, H, O], [AK 541; H, Et, H, Pr, O, CH _{2 F, H, H, H} , O], [AK542; H, Et, H, Pr, O, CHF 2, H, H, H, O], [AK543; H, Et, H, Pr, O, _{CF 3, H, H, H} , O], [AK544; H, Et, H, Pr, O, OCH 2 F, H, H, H, O], [AK545; H, Et, H, Pr, O _{, OCHF 2, H, H,} H, O], [AK546; H, Et, H, Pr, O, OCF 3, H, H, H, O], [AK547; H, Et, H, Pr, O , OCF ₃ , H, H, H, O], [AK 548; H, Et, H, i-Pr, O, H, H, H, H, O], [AK 549; H, Et, H, i- Pr, O, F, H, H, H, O], [AK 550; H, Et, H, i-Pr, O, Cl, H, H, H, O], [AK 551; H, Et, H, O] i-Pr, O, Br, H, H, H, O], [AK 552; H, Et, H, i-Pr, O, I, H, H, H, O], [AK 553: H, Et, H, i-Pr, O, Me, H, H, H, O], [AK 554; H, Et, H, i-Pr, O, Et, H, H, H, O], [AK 555; H, Et, H, i-Pr, O, Pr, H, H, H, O], [AK 556; H, Et, H, i-Pr, O, i-Pr, H, H, H, O], [[A] AK 557; H, Et, H, i-Pr, O, Bu, H, H, H, O] [AK 558; H, Et, H, i-Pr, O, i-Bu, H, H, H, O], [AK559; H, Et, H, i-Pr, O, sec-Bu, H, H , H, O], [AK 560; H, Et, H, i-Pr, O, t-Bu, H, H, H, O], [AK 561; H, Et, H, i-Pr, O, c -Pr, H, H, H, O], [AK 562; H, Et, H, i-Pr, O, c-Bu, H, H, H, O], [AK 563; H, Et, H, i] -Pr, O, OBu, H, H, H, O, [AK 564; H, Et, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK 565; H, Et , H, i-Pr, O , O-sec-Bu, H, H, H, O], [AK566; H, Et, H, i-Pr, O, CH 2 F, H, H, H, O ], [AK567; H, Et , H, i-Pr, O, CHF 2, H, H, H, O], [AK568; H, Et, H, i-Pr, O, CF 3, H, H , H, O], [AK569 ; H, Et, H, i-Pr, O, OCH 2 F, H, H, H, O], [AK570; H, Et, H, i-Pr, O, OCHF _{2, H, H, H,} O], [AK571; H, Et, H, i-Pr, O, OCF 3, H, H, H, O], [AK572; H, Et, H, i-Pr _{, O, OCF 3, H,} H, H, O], [AK573; H, Et, H, OMe, O, H, H, H, H, O], [AK574; H, Et, H, OMe, O, F, H, H, H, O], [AK575; H, Et, H, OMe, O, Cl, H, H, H, O], [AK 576; H, Et, H, OMe, O, Br, H, H, H, O], [AK577; H, Et, H, OMe, O, I, H, H, H, O], [AK 578; H, Et, H, OMe, O, Me, H, H, H, O], [AK579; H, Et, H, OMe, O, Et, H, H, H, O], [AK 580; H, Et, H, OMe, O, Pr, H, H, H, O], [AK 581; H, Et, H, OMe, O, i-Pr, H, H, H, O], [AK 582; H, Et, H, OMe, O, Bu, H, H, H, O], [AK 583; H, Et, H, OMe, O, i-Bu, H, H, H, O], [AK 584; H, Et, H, OMe, O, sec-Bu, H, H, H, O], [AK585; H, Et, H, OMe, O, t-Bu, H, H, H, O], [AK 586; H, Et, H, OMe, O, c-Pr, H, H, H, O], [AK 587; H, Et, H, OMe, O, c-Bu, H, H, H, O], [AK 588; H, Et, H, OMe, O, OBu, H, H, H, O], [AK 589; H, Et, H, OMe, O, Oi-Bu, H, H, H, O], [AK 590; H, Et, H, OMe, O, O-sec-Bu, H, H, H, O] , [AK591; H, Et, H, OMe, O, CH 2 F, H, H, H, O], [AK592; H, Et, H, OMe, O, CHF 2, H, H, H, O ], [AK593; H, Et , H, OMe, O, CF 3, H, H, H, O], [AK594; H, Et, H, OMe, O, OCH 2 F, H, H, H, O], [AK 595; H, Et, H, OMe, O, OCHF ₂ , H, H, H, O], [AK 596; H, Et, H, OMe, O, OCF ₃ , H, H, H, O], [AK597; H, Et, H, OMe, O, OCF 3, H, H, H, O], [AK598; H, Et, H, F, O, H, H, H, H, O H, Et, H, F, O, F, H, H, O], [AK600; H, Et, H, F, O, Cl, H, H, H, O],

[AK601; H, Et, H, F, O, Br, H, H, O], [AK602; H, Et, H, F, O, I, H, H, H, O], [AK603 H, Et, H, F, O, Me, H, H, H, O], [AK 604; H, Et, H, F, O, Et, H, H, H, O], [AK 605; H , Et, H, F, O, Pr, H, H, H, O], [AK 606; H, Et, H, F, O, i-Pr, H, H, H, O], [AK 607; H , Et, H, F, O, Bu, H, H, H, O], [AK 608; H, Et, H, F, O, i-Bu, H, H, H, O], [AK 609; H , Et, H, F, O, sec-Bu, H, H, H, O], [AK610; H, Et, H, F, O, t-Bu, H, H, H, O], [AK611 H, Et, H, F, O, c-Pr, H, H, H, O], [AK 612; H, Et, H, F, O, c-Bu, H, H, H, O], [AK613; H, Et, H, F, O, OBu, H, H, H, O], [AK614; H, Et, H, F, O, Oi-Bu, H, H, H, O], [AK615; H, Et, H , F, O, O-sec-Bu, H, H, H, O], [AK616; H, Et, H, F, O, CH 2 F, H, H, H , O], [AK617; H , Et, H, F, O, CHF 2, H, H, H, O], [AK618; H, Et, H, F, O, CF 3, H, H, H , O], [AK619; H , Et, H, F, O, OCH 2 F, H, H, H, O], [AK620; H, Et, H, F, O, OCHF 2, H, H, H, O], [AK621; H, Et, H, F, O, OCF 3, H, H, H, O], [AK622; H, Et, H, F, O, OCF 3, H, H, H, O], [AK 623; H, Et, H, Cl, O, H, H, H, H, O], [AK 624; H, Et, H, Cl, O, F, H, H, H, H, O], [AK 625; H, Et, H, Cl, O, Cl, H, H, H, O], [AK 626; H, Et, H, Cl, O, Br, H, H, H, O] [AK 627; H, Et, H, Cl, O, I, H, H, H, O], [AK 628; H, Et, H, Cl, O, Me, H, H, H, O], [AK 627; AK629; H, Et, H, Cl, O, Et, H, H, H, O], [AK630; H, Et, H, Cl , O, Pr, H, H, H, O], [AK 631; H, Et, H, Cl, O, i-Pr, H, H, H, O], [AK 632; H, Et, H, Cl , O, Bu, H, H, H, O], [AK 633; H, Et, H, Cl, O, i-Bu, H, H, H, O], [AK 634; H, Et, H, Cl , O, sec-Bu, H, H, H, O], [AK 635; H, Et, H, Cl, O, t-Bu, H, H, H, O], [AK 636; H, Et, H , Cl, O, c-Pr, H, H, H, O], [AK 637; H, Et, H, Cl, O, c-Bu, H, H, H, O], [AK 638; H, Et , H, Cl, O, OBu, H, H, H, O], [AK639; H, Et, H, Cl, O, Oi-Bu, H, H, H, O], [AK 640; H, Et] , H, Cl, O, O -sec-Bu, H, H, H, O], [AK641; H, Et, H, Cl, O, CH 2 F, H, H, H, O], [AK642 ; H, Et, H, Cl , O, CHF 2, H, H, H, O], [AK643; H, Et, H, Cl, O, CF 3, H, H, H, O], [AK644 ; H, Et, H, Cl , O, OCH 2 F, H, H, H, O], [AK645; H, Et, H, Cl, O, OCHF 2, H, H, H, O], [ AK646; H, Et, H, Cl, O, OCF 3, H, H, H, O], [AK647; H, Et, H, Cl, O, OCF 3, H, H, H, O], [ AK648; H, Et, H, Br, O, H, H, H, O], [AK 649; H, Et, H, Br, O, F, H, H, H, O], [AK 650; H, Et, H, Br, O, Cl, H, H, H, O], [AK651; H, Et, H, Br, O, Br, H, H, H, O], [AK652; H, H, Et, H, Br, O, I, H, H, H, O], [AK 653; H, Et, H, Br, O, Me, H, H, H, O], [AK 654; H, Et, H, Br, O, Et, H, H, H, O], [AK655; H, Et, H, Br, O, Pr, H, H, H, O], [AK656; H, Et, H, O] Br, O, i-Pr, H, H, H, O, [AK 657; H, Et, H, Br, O, Bu, H, H, H, O], [AK 658; H, Et, H, Br, O, i-Bu, H, H, H, O], [AK65 9; H, Et, H, Br, O, sec-Bu, H, H, H, O], [AK 660; H, Et, H, Br, O, t-Bu, H, H, H, O] [AK 661; H, Et, H, Br, O, c-Pr, H, H, H, O], [AK 662; H, Et, H, Br, O, c-Bu, H, H, H, H, O], [AK663; H, Et, H, Br, O, OBu, H, H, H, O], [AK664; H, Et, H, Br, O, Oi-Bu, H, H, H, O], [AK665; H, Et, H, Br, O, O-sec-Bu, H, H, H, O], [AK666; H, Et, H, Br, O, CH 2 F, H, H, H, O], [ AK667; H, Et, H, Br, O, CHF 2, H, H, H, O], [AK668; H, Et, H, Br, O, CF 3, H, H, H, O], [AK 669; H, Et, H, Br, O, OCH ₂ F, H, H, H, O], [AK 670; H, Et, H, Br, O, OCHF ₂ , H , H, H, O], [AK671; H, Et, H, Br, O, OCF 3, H, H, H, O], [AK672; H, Et, H, Br, O, OCF 3, H H, H, O], [AK673; H, Pr, H, H, O, H, H, H, H, O], [AK 674; H, Pr, H, H, O, F, H, H] , H, O], [AK 675; H, Pr, H, H, O, Cl, H, H, H, O], [AK 676; H, Pr, H, H, O, Br, H, H, H] , O], [AK 677; H, Pr, H, H, O, I, H, H, H, O], [AK 678; H, Pr, H, H, O, Me, H, H, H, O ], [AK 679; H, Pr, H, H, O, Et, H, H, H, O], [AK 680; H, Pr, H, H, O, Pr, H, H, H, O], [AK 681; H, Pr, H, H, O, i-Pr, H, H, H, O], [AK 682; H, Pr, H, H, O, Bu, H, H, H, O], [AK 683; H, Pr, H, H, O, i-Bu, H, H, H, O], [AK 684; H, Pr, H, H, O, sec-Bu, H, H, H, O ], [AK 685; H, Pr, H, H, O, t-Bu, H, H, H, O], [AK 686; H, Pr, H, H, O, c-Pr, H, H, H] , O], [AK 687; H, Pr, H, H, O, c-Bu, H, H, H, O], [AK 688; H, Pr, H, H, O, OBu, H, H, H, O], [AK 689; H, Pr, H, H, O, Oi-Bu, H, H, H, O], AK690; H, Pr, H, H, O, O-sec-Bu, H, H, H, O], [AK691; H, Pr, H, H, O, CH 2 F, H, H, H, O], [AK692; H, Pr, H, H, O, CHF 2, H, H, H, O], [AK693; H, Pr, H, H, O, CF 3, H, H, H, O], [AK 694; H, Pr, H, H, O, OCH ₂ F, H, H, H, O], [AK 695; H, Pr, H, H, O, OCHF ₂ , H, H, H , O], [AK696; H , Pr, H, H, O, OCF 3, H, H, H, O], [AK697; H, Pr, H, Me, O, H, H, H, H, O], [AK 698; H, Pr, H, Me, O, F, H, H, O], [AK 699; H, Pr, H, Me, O, Cl, H, H, H, O] [AK 700; H, Pr, H, Me, O, Br, H, H, H, O],

[AK 701; H, Pr, H, Me, O, I, H, H, O], [AK 702; H, Pr, H, Me, O, Me, H, H, H, O], [AK 703 H, Pr, H, Me, O, Et, H, H, H, O], [AK704; H, Pr, H, Me, O, Pr, H, H, H, O], [AK705; H , Pr, H, Me, O, i-Pr, H, H, H, O], [AK 706; H, Pr, H, Me, O, Bu, H, H, H, O], [AK 707; H , Pr, H, Me, O, i-Bu, H, H, H, O], [AK 708; H, Pr, H, Me, O, sec-Bu, H, H, H, O], [AK 709] H, Pr, H, Me, O, t-Bu, H, H, H, O], [AK 710; H, Pr, H, Me, O, c-Pr, H, H, H, O], [AK711; H, Pr, H, Me, O, c-Bu, H, H, H, O], [AK 712; H, Pr, H, Me, O, OBu, H, H, H, O], [AK713; H, Pr, H, Me, O, Oi-Bu, H, H, H, O], [AK714; H, Pr, H, Me, O, O-sec-Bu, H, H, H , O], [AK715; H , Pr, H, Me, O, CH 2 F, H, H, H, O], [AK716; H, Pr, H, Me, O, CHF 2, H, H, H, O], [AK717; H, Pr, H, Me, O, CF 3, H, H, H, O], [AK718; H, Pr, H, Me, O, OCH 2 F, H, H , H, O], [AK 719; H, Pr, H, Me, O, OCHF ₂ , H, H, H, O], [AK 720; H, Pr, H, Me, O, OCF ₃ , H, H , H, O], [AK721 ; H, Pr, H, Me, O, OCF 3, H, H, H, O], [AK722; H, Pr, H, Et, O, H, H, H, H, O], [AK 723; H, Pr, H, Et, O, F, H, H, H, O], [AK 724; H, Pr, H, Et, O, Cl, H, H, H, H, O], [AK 725; H, Pr, H, Et, O, Br, H, H, O], [AK 726; H, Pr, H, Et, O, I, H, H, H, O] [AK727; H, Pr, H, Et, O, Me, H, H, H, O], [AK 728; H, Pr, H, Et, O, Et, H, H, H, O], [[AK727; AK729; H, Pr, H, Et, O, Pr, H, H, H , O], [AK 730; H, Pr, H, Et, O, i-Pr, H, H, H, O], [AK 731; H, Pr, H, Et, O, Bu, H, H, H H, Pr, H, Et, O, i-Bu, H, H, H, O], [AK733; H, Pr, H, Et, O, sec-Bu, H, H] , H, O], [AK734; H, Pr, H, Et, O, t-Bu, H, H, H, O], [AK 735; H, Pr, H, Et, O, c-Pr, H H, H, O], [AK 736; H, Pr, H, Et, O, c-Bu, H, H, H, O], [AK 737; H, Pr, H, Et, O, OBu, H , H, H, O], [AK 738; H, Pr, H, Et, O, Oi-Bu, H, H, H, O], [AK 739; H, Pr, H, Et, O, O-sec -Bu, H, H, H, O], [AK740; H, Pr, H, Et, O, CH 2 F, H, H, H, O], [AK741; H, Pr, H, Et, O _{, CHF 2, H, H,} H, O], [AK742; H, Pr, H, Et, O, CF 3, H, H, H, O], [AK743; H, Pr, H, Et, O , OCH ₂ F, H, H, H, O], [AK 744; H, Pr, H, Et, O, OCHF ₂ , H, H, H, O], [AK 745; H, Pr, H, Et, _{O, OCF 3, H, H} , H, O], [AK746; H, Pr, H, Et, O, OCF 3, H, H, H, O], [AK747; H, Pr, H, Pr, O, H, H, H, H, O, [AK 748; H, Pr, H, Pr, O, F, H, H, H, O], [AK 749; H, Pr, H, Pr, O, Cl, H, H, H, O], [AK 750; H, Pr, H, Pr, O, Br, H, H, H, O], [AK 751; H, Pr, H, Pr, O, I, I, H, H, H, O], [AK 752; H, Pr, H, Pr, O, Me, H, H, H, O], [AK 753; H, Pr, H, Pr, O, Et, H, O] H, H, O], [AK 754; H, Pr, H, Pr, O, Pr, H, H, H, O], [AK 755; H, Pr, H, Pr, O, i-Pr, H, H, H, O], [AK 756; H, Pr, H, Pr, O, Bu, H, H, H, O], [AK757; H, Pr, H, Pr, O, i-Bu, H, H, H, O], [AK 758; H, Pr, H, Pr , O, sec-Bu, H, H, H, O], [AK 759; H, Pr, H, Pr, O, t-Bu, H, H, H, O], [AK 760; H, Pr, H , Pr, O, c-Pr, H, H, H, O], [AK 761; H, Pr, H, Pr, O, c-Bu, H, H, H, O], [AK 762; H, Pr , H, Pr, O, OBu, H, H, H, O], [AK 763; H, Pr, H, Pr, O, Oi-Bu, H, H, H, O], [AK 764; H, Pr , H, Pr, O, O -sec-Bu, H, H, H, O], [AK765; H, Pr, H, Pr, O, CH 2 F, H, H, H, O], [AK766 ; H, Pr, H, Pr , O, CHF 2, H, H, H, O], [AK767; H, Pr, H, Pr, O, CF 3, H, H, H, O], [AK768 H, Pr, H, Pr, O, OCH ₂ F, H, H, H, O], [AK 769; H, Pr, H, Pr, O, OCHF ₂ , H, H, H, O], [[ AK770; H, Pr, H, Pr, O, OCF 3, H, H, H, O], [AK771; H, Pr, H, Pr, O, OCF 3, H, H, H, O], [ AK772; H, Pr, H, i-Pr, O, H, H, H, H, O], [AK 773; H, Pr, H, i-Pr, O, F, H, H, H, O] [AK774; H, Pr, H, i-Pr, O, Cl, H, H, H, O], [AK775; H, Pr, H, i-Pr, O, Br, H, H, H, H, O], [AK 776; H, Pr, H, i-Pr, O, I, H, H, H, O], [AK 777; H, Pr, H, i-Pr, O, Me, H, H, H, H, O], [AK 778; H, Pr, H, i-Pr, O, Et, H, H, H, O], [AK 779; H, Pr, H, i-Pr, O, Pr, H, H, H, O], [AK 780; H, Pr, H, i-Pr, O, i-Pr, H, H, H, O], [AK 781; H, Pr, H, i-Pr, O, Bu, H, H, H, O], [AK 782; H, Pr, H, i-Pr, O, i-Bu, H, H, H, O], [AK 783; H, Pr, H, i- Pr, O, sec-Bu, H, H, H, O, [AK 784; H, Pr, H, i-Pr, O, t-Bu, H, H, H, O], [AK 785; H, Pr, H, i-Pr, O, c-Pr, H, H, H, O], [AK786 H, Pr, H, i-Pr, O, c-Bu, H, H, H, O], [AK 787; H, Pr, H, i-Pr, O, OBu, H, H, H, O] H, Pr, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK 789; H, Pr, H, i-Pr, O, O-sec-Bu] , H, H, H, O ], [AK790; H, Pr, H, i-Pr, O, CH 2 F, H, H, H, O], [AK791; H, Pr, H, i-Pr , O, CHF ₂ , H, H, H, O], [AK 792; H, Pr, H, i-Pr, O, CF ₃ , H, H, H, O], [AK 793; H, Pr, H , i-Pr, O, OCH 2 F, H, H, H, O], [AK794; H, Pr, H, i-Pr, O, OCHF 2, H, H, H, O], [AK795; H, Pr, H, i- Pr, O, OCF 3, H, H, H, O], [AK796; H, Pr, H, i-Pr, O, OCF 3, H, H, H, O] [AK 797; H, Pr, H, OMe, O, H, H, H, H, O], [AK 798; H, Pr, H, OMe, O, F, H, H, H, O], [AK 797; AK 799; H, Pr, H, OMe, O, Cl, H, H, H, O], [AK 800; H, Pr, H, OMe, O, Br, H, H, H, O],

[AK801; H, Pr, H, OMe, O, I, H, H, O], [AK802; H, Pr, H, OMe, O, Me, H, H, H, O], [AK803 H, Pr, H, OMe, O, Et, H, H, H, O], [AK 804; H, Pr, H, OMe, O, Pr, H, H, H, O], [AK 805; H , Pr, H, OMe, O, i-Pr, H, H, H, O], [AK 806; H, Pr, H, OMe, O, Bu, H, H, H, O], [AK 807; H , Pr, H, OMe, O, i-Bu, H, H, H, O], [AK 808; H, Pr, H, OMe, O, sec-Bu, H, H, H, O], [AK 809] H, Pr, H, OMe, O, t-Bu, H, H, H, O], [AK 810; H, Pr, H, OMe, O, c-Pr, H, H, H, O], [AK811; H, Pr, H, OMe, O, c-Bu, H, H, H, O], [AK 812; H, Pr, H, OMe, O, OBu, H, H, H, O], [AK813; H, Pr, H, OMe, O, Oi-Bu, H, H, H, O], [AK 814; H, Pr, H, OMe, O, O-sec-Bu, H, H, H , O], [AK815; H , Pr, H, OMe, O, CH 2 F, H, H, H, O], [AK816; H, Pr, H, OMe, O, CHF 2, H, H, H, O], [AK817; H, Pr, H, OMe, O, CF 3, H, H, H, O], [AK818; H, Pr, H, OMe, O, OCH 2 F, H, H , H, O], [AK 819; H, Pr, H, OMe, O, OCHF ₂ , H, H, H, O], [AK 820; H, Pr, H, OMe, O, OCF ₃ , H, H , H, O], [AK821 ; H, Pr, H, OMe, O, OCF 3, H, H, H, O], [AK822; H, Pr, H, F, O, H, H, H, H, O], [AK 823; H, Pr, H, F, O, F, H, H, H, O], [AK 824; H, Pr, H, F, O, Cl, H, H, H, H, O], [AK 825; H, Pr, H, F, O, Br, H, H, O], [AK 826; H, Pr, H, F, O, I, H, H, H, O] [AK827; H, Pr, H, F, O, Me, H, H, H, O], [AK 828; H, Pr, H, F, O, Et, H, H, H, O], [AK 827; AK829; H, Pr, H , F, O, Pr, H, H, H, O], [AK 830; H, Pr, H, F, O, i-Pr, H, H, H, O], [AK 831; H, Pr, H] , F, O, Bu, H, H, H, O], [AK 832; H, Pr, H, F, O, i-Bu, H, H, H, O], [AK 833; H, Pr, H] , F, O, sec-Bu, H, H, H, O], [AK 834; H, Pr, H, F, O, t-Bu, H, H, H, O], [AK 835; H, Pr , H, F, O, c-Pr, H, H, H, O], [AK 836; H, Pr, H, F, O, c-Bu, H, H, O], [AK 837; H , Pr, H, F, O, OBu, H, H, H, O], [AK 838; H, Pr, H, F, O, Oi-Bu, H, H, H, O], [AK 839; H , Pr, H, F, O , O-sec-Bu, H, H, H, O], [AK840; H, Pr, H, F, O, CH 2 F, H, H, H, O], [AK 841; H, Pr, H, F, O, CHF ₂ , H, H, H, O], [AK 842; H, Pr, H, F, O, CF ₃ , H, H, H, O], [AK843; H, Pr, H , F, O, OCH 2 F, H, H, H, O], [AK844; H, Pr, H, F, O, OCHF 2, H, H, H, O] , [AK845; H, Pr, H, F, O, OCF 3, H, H, H, O], [AK846; H, Pr, H, F, O, OCF 3, H, H, H, O] [AK 847; H, Pr, H, Cl, O, H, H, H, O], [AK 848; H, Pr, H, Cl, O, F, H, H, H, O], [AK 847; AK8 49; H, Pr, H, Cl, O, Cl, H, H, O], [AK850; H, Pr, H, Cl, O, Br, H, H, H, O], [AK 851; H, Pr, H, Cl, O, I, H, H, H, O], [AK 852; H, Pr, H, Cl, O, Me, H, H, H, O], [AK 853; H, Pr, H, Cl, O, Et, H, H, H, O], [AK 854; H, Pr, H, Cl, O, Pr, H, H, H, O], [AK 855; H, Pr, H, Cl, O, i-Pr, H, H, H, O], [AK 856; H, Pr, H, Cl, O, Bu, H, H, H, O], [AK 857; H, Pr, H, Cl, O, i-Bu, H, H, H, O], [AK 858; H, Pr, H, Cl, O, s ec-Bu, H, H, H, O], [AK 859; H, Pr, H, Cl, O, t-Bu, H, H, H, O], [AK 860; H, Pr, H, Cl, O, c-Pr, H, H, H, O], [AK 861; H, Pr, H, Cl, O, c-Bu, H, H, H, O], [AK 862; H, Pr, H, O] Cl, O, OBu, H, H, H, O], [AK863; H, Pr, H, Cl, O, Oi-Bu, H, H, H, O], [AK864; H, Pr, H, Cl, O, O-sec- Bu, H, H, H, O], [AK865; H, Pr, H, Cl, O, CH 2 F, H, H, H, O], [AK866; H, Pr, H, Cl, O, CHF 2, H, H, H, O], [AK867; H, Pr, H, Cl, O, CF 3, H, H, H, O], [AK868; H, Pr, H, Cl, O, OCH ₂ F, H, H, H, O], [AK 869; H, Pr, H, Cl, O, OCHF ₂ , H, H, H, O], [AK 870; H , Pr, H, Cl, O , OCF 3, H, H, H, O], [AK871; H, Pr, H, Cl, O, OCF 3, H, H, H, O], [AK872; H , Pr, H, Br, O, H, H, H, H, O], [AK 873; H, Pr, H, Br, O, F, H, H, H, O], [AK 874; H, Pr] , H, Br, O, Cl, H, H, H, O], [AK 875; H, Pr, H, Br, O, Br, H, H, H, O], [AK 876; H, Pr, H] , Br, O, I, H, H, H, O], [AK 877; H, Pr, H, Br, O, Me, H, H, H, O], [AK 878; H, Pr, H, Br] , O, Et, H, H, H, O], [AK 879; H, Pr, H, Br, O, Pr, H, H, H, O], [AK 880; H, Pr, H, Br, O] , i-Pr, H, H, H, O], [AK 881; H, Pr, H, Br, O, Bu, H, H, H, O], [AK 882; H, Pr, H, Br, O] , i-Bu, H, H, H, O], [AK 883; H, Pr, H, Br, O, sec-Bu, H, H, H, O], [AK 884; H, Pr, H, Br] , O, t-Bu, H, H, H, O], [AK 885; H, Pr, H, Br, O, c-Pr, H, H, H, O], [AK 886; H, Pr, H , Br, O, c-Bu, H, H, H, O], [AK 887; H, Pr, H, Br, O, OBu, H, H, H, O], [AK 888; H, Pr, H, Br, O, Oi-Bu, H, H, H, O], [A AK889; H, Pr, H, Br, O, O-sec-Bu, H, H, H, O], [AK890; H, Pr, H, Br, O, CH 2 F, H, H, H, O], [AK 891; H, Pr, H, Br, O, CHF ₂ , H, H, H, O], [AK 892; H, Pr, H, Br, O, CF ₃ , H, H, H, H, O], [AK 893; H, Pr, H, Br, O, OCH ₂ F, H, H, H, O], [AK 894; H, Pr, H, Br, O, OCHF ₂ , H, H, H , O], [AK895; H , Pr, H, Br, O, OCF 3, H, H, H, O], [AK896; H, Pr, H, Br, O, OCF 3, H, H, H , O], [AK897; H, i-Pr, H, H, O, H, H, H, H, O], [AK 898; H, i-Pr, H, H, O, F, H, H , H, O], [AK 899; H, i-Pr, H, H, O, Cl, H, H, H, O], [AK 900; H, i-Pr, H, H, O, Br, H , H, H, O],

[AK 901; H, i-Pr, H, H, O, I, H, H, H, O], [AK 902; H, i-Pr, H, H, O, Me, H, H, H, O , [AK 903; H, i-Pr, H, H, O, Et, H, H, H, O], [AK 904; H, i-Pr, H, H, O, Pr, H, H, H] H, i-Pr, H, H, O, i-Pr, H, H, H, O], [AK906; H, i-Pr, H, H, O, Bu, H , H, H, O], [AK 907; H, i-Pr, H, H, O, i-Bu, H, H, H, O], [AK 908; H, i-Pr, H, H, O] , sec-Bu, H, H, H, O], [AK 909; H, i-Pr, H, H, O, t-Bu, H, H, H, O], [AK 910; H, i-Pr , H, H, O, c-Pr, H, H, H, O], [AK911; H, i-Pr, H, H, O, c-Bu, H, H, H, O], [AK912 H, i-Pr, H, H, O, OBu, H, H, H, O], [AK 913; H, i-Pr, H, H, O, Oi-Bu, H, H, H, O H, i-Pr, H, H, O, O-sec-Bu, H, H, H, O], [AK 915; H, i-Pr, H, H, O, CH ₂ F] , H, H, H, O ], [AK916; H, i-Pr, H, H, O, CHF 2, H, H, H, O], [AK917; H, i-Pr, H, H, O, CF ₃ , H, H, H, O], [AK 918; H, i-Pr, H, H, O, OCH ₂ F, H, H, H, O], [AK 919; H, i-Pr , H, H, O, OCHF 2, H, H, H, O], [AK920; H, i-Pr, H, H, O, OCF 3, H, H, H, O], [AK921; H , i-Pr, H, Me, O, H, H, H, H, O], [AK 922; H, i-Pr, H, Me, O, F, H, H, H, O], [AK 923 H, i-Pr, H, Me, O, Cl, H, H, O], [AK 924; H, i-Pr, H, Me, O, Br, H, H, H, O], [AK 925; H, i-Pr, H, Me, O, I, H, H, H, O], [AK 926; H, i-Pr, H, Me, O, Me, H, H, H, O [AK 927; H, i-Pr, H, Me, O, Et, H, H, H, O], [AK 928; H, i-Pr, H, Me, O, Pr, H, H, H] , O], [AK 929; H, i-Pr, H, Me, O, i-Pr, H, H, H, O], [AK 930; H, i-Pr, H, Me, O, Bu, H, H, H, O], [AK 931; H, i-Pr, H, Me, O, i-Bu, H, H, H, O], [AK 932; H, i-Pr, H, Me, O, sec-Bu, H, H, H, O], [AK 933; H, i-Pr, H, Me, O, t-Bu, H, H, H, O], [AK 934; H, i-Pr, H, Me, O, c-Pr, H, H, H, O], [AK935; H, i-Pr, H, Me, O, c-Bu, H, H, H, O], [AK936; H, i-Pr, H, Me, O, OBu, H, H, H, O], [AK 937; H, i-Pr, H, Me, O, Oi-Bu, H, H, H, O] [AK 938; H, i-Pr, H, Me, O, O-sec-Bu, H, H, H, O], [AK 939; H, i-Pr, H, Me, O, CH ₂ F, H, H, H, O] , [AK940; H, i-Pr, H, Me, O, CHF 2, H, H, H, O], [AK941; H, i-Pr, H, Me, O , CF ₃ , H, H, H, O], [AK 942; H, i-Pr, H, Me, O, OCH ₂ F, H, H, H, O], [AK 943; H, i-Pr, _{H, Me, O, OCHF 2} , H, H, H, O], [AK944; H, i-Pr, H, Me, O, OCF 3, H, H, H, O], [AK945; H, i-Pr, H, Me, O, OCF 3, H, H, H, O], [AK946; H, i-Pr, H, Et, O, H, H, H, H, O], [AK947 H, i-Pr, H, Et, O, F, H, H, O], [AK 948; H, i-Pr, H, Et, O, Cl, H, H, H, O], [AK 949; H, i-Pr, H, Et, O, Br, H, H, O], [AK 950; H, i-Pr, H, Et, O, I, H, H, H, O H, i-Pr, H, Et, O, Me, H, H, H, O], [AK 952; H, i-Pr, H, Et, O, Et, H, H, H] , O], [AK953; H, i-Pr, H, Et, O, Pr, H, H, H, O], [AK 954; H, i-Pr, H, Et, O, i-Pr, H , H, H, O], [AK 955; H, i-Pr, H, Et, O, Bu, H, H, H, O] [AK956; H, i-Pr, H, Et, O, i-Bu, H, H, H, O], [AK957; H, i-Pr, H, Et, O, sec-Bu, H, H , H, O], [AK 958; H, i-Pr, H, Et, O, t-Bu, H, H, H, O], [AK 959; H, i-Pr, H, Et, O, c -Pr, H, H, H, O], [AK 960; H, i-Pr, H, Et, O, c-Bu, H, H, H, O], [AK 961; H, i-Pr, H , Et, O, OBu, H, H, H, O], [AK 962; H, i-Pr, H, Et, O, Oi-Bu, H, H, H, O], [AK963; H, i -Pr, H, Et, O, O-sec-Bu, H, H, H, O], [AK964; H, i-Pr, H, Et, O, CH 2 F, H, H, H, O ], [AK965; H, i -Pr, H, Et, O, CHF 2, H, H, H, O], [AK966; H, i-Pr, H, Et, O, CF 3, H, H , H, O], [AK 967; H, i-Pr, H, Et, O, OCH ₂ F, H, H, H, O], [AK 968; H, i-Pr, H, Et, O, OCHF _{2, H, H, H,} O], [AK969; H, i-Pr, H, Et, O, OCF 3, H, H, H, O], [AK970; H, i-Pr, H, Et _{, O, OCF 3, H,} H, H, O], [AK971; H, i-Pr, H, Pr, O, H, H, H, H, O], [AK972; H, i-Pr, H, Pr, O, F, H, H, H, O], [AK 973; H, i-Pr, H, Pr, O, Cl, H, H, H, O], [AK 974; H, i- Pr, H, Pr, O, Br, H, H, H, O], [AK 975; H, i-Pr, H, Pr, O, I, H, H, H, O], [AK 976; H, i-Pr, H, Pr, O, Me, H, H, H, O], [AK 977; H, i-Pr, H, Pr, O, Et, H, H, H, O], [AK 978; H, i-Pr, H, Pr, O, Pr, H, H, H, O], [AK979; H, i-Pr, H, Pr, O, i-Pr, H, H, H, O] [AK 980; H, i-Pr, H, Pr, O, Bu, H, H, H, O], [AK 981; H, i-Pr, H, Pr, O, i-Bu, H, H, H, O], [AK 982; H, i-Pr, H, Pr, O, sec-Bu, H, H, H, O] [AK983; H, i-Pr, H, Pr, O, t-Bu, H, H, H, O], [AK984; H, i-Pr, H, Pr, O, c-Pr, H, H, H, O], [AK 985; H, i-Pr, H, Pr, O, c-Bu, H, H, H, O], [AK 986; H, i-Pr, H, Pr, O, OBu, H, H, H, O], [AK 987; H, i-Pr, H, Pr, O, Oi-Bu, H, H, H, O], [AK 988; H, i-Pr, H, Pr, O, O-sec- Bu, H, H, H, O], [AK989; H, i-Pr, H, Pr, O, CH 2 F, H, H, H, O], [AK990; H, i-Pr, H, Pr, O, CHF 2, H, H, H, O], [AK991; H, i-Pr, H, Pr, O, CF 3, H, H, H, O] , [AK992; H, i- Pr, H, Pr, O, OCH 2 F, H, H, H, O], [AK993; H, i-Pr, H, Pr, O, OCHF 2, H, H , H, O], [AK994 ; H, i-Pr, H, Pr, O, OCF 3, H, H, H, O], [AK995; H, i-Pr, H, Pr, O, OCF 3 , H, H, H, O], [AK 996; H, i-Pr, H, i-Pr, O, H, H, H, H, O], [AK 997; H, i-Pr, H, i -Pr, O, F, H, H, H, O], [AK 998; H, i-Pr, H, i-Pr, O, Cl, H, H, H, O], [AK 999; H, i -Pr, H, i-Pr, O, Br, H, H, H, O], [AK1000; H, i-Pr, H, i-Pr, O, I, H, H, H, O],

[AK1001; H, i-Pr, H, i-Pr, O, Me, H, H, H, O], [AK1002; H, i-Pr, H, i-Pr, O, Et, H, H] , H, O], [AK 1003; H, i-Pr, H, i-Pr, O, Pr, H, H, H, O], [AK 1004; H, i-Pr, H, i-Pr, O , i-Pr, H, H, H, O], [AK 1005; H, i-Pr, H, i-Pr, O, Bu, H, H, H, O], [AK 1006; H, i-Pr , H, i-Pr, O, i-Bu, H, H, H, O], [AK 1007; H, i-Pr, H, i-Pr, O, sec-Bu, H, H, H, O H, i-Pr, H, i-Pr, O, t-Bu, H, H, H, O], [AK 1009; H, i-Pr, H, i-Pr, O, c] -Pr, H, H, H, O], [AK1010; H, i-Pr, H, i-Pr, O, c-Bu, H, H, H, O], [AK1011; H, i-Pr , H, i-Pr, O, OBu, H, H, H, O], [AK1012; H, i-Pr, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK1013; H, i-Pr, H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK1014; H, i-Pr, H, i-Pr, O, CH ₂ F, H, H, H, O], [AK 1015; H, i-Pr, H, i-Pr, O, CHF ₂ , H, H, H, O], [AK 1016; H, i-Pr, H, i-Pr, O, CF 3, H, H, H, O], [AK1017; H, i-Pr, H, i-Pr, O, OCH 2 F, H, H, H, O], [AK1018; H, i-Pr , H, i-Pr, O, OCHF 2, H, H, H, O], [AK1019; H, i-Pr, H, i-Pr, O, OCF 3, H , H, H, O], [AK1020; H, i-Pr, H, i-Pr, O, OCF 3, H, H, H, O], [AK1021; H, i-Pr, H, OMe, O, H, H, H, H, O], [AK 1022; H, i-Pr, H, OMe, O, F, H, H, H, O], [AK 1023; H, i-Pr, H, OMe, O, Cl, H, H, H, O], [AK 1024; H, i-Pr, H, OMe, O, Br, H, H, H, O], [AK1025; H, i-Pr, H, OMe, O, I, H, H, H, O], [AK10 26; H, i-Pr, H, OMe, O, Me, H, H, H, O], [AK1027; H, i-Pr, H, OMe, O, Et, H, H, H, O] [AK1028; H, i-Pr, H, OMe, O, Pr, H, H, H, O], [AK1029; H, i-Pr, H, OMe, O, i-Pr, H, H, H, O], [AK1030; H, i-Pr, H, OMe, O, Bu, H, H, H, O], [AK1031; H, i-Pr, H, OMe, O, i-Bu, H, H, H, O], [AK1032; H, i-Pr, H, OMe, O, sec-Bu, H, H, H, O], [AK1033; H, i-Pr, H, OMe, O, t-Bu, H, H, H, O], [AK 1034; H, i-Pr, H, OMe, O, c-Pr, H, H, H, O], [AK 10 35; H, i- Pr, H, OMe, O, c-Bu, H, H, H, O], [AK1036; H, i-Pr, H, OMe, O, OBu, H, H, H, O], [AK1037; H, i-Pr, H, OMe, O, Oi-Bu, H, H, H, O], [AK1038; H, i-Pr, H, OMe, O, O-sec-Bu, H, H, H, O], [AK1039; H, i-Pr, H, OMe, O, CH 2 F, H, H, H, O], [AK1040; H, i-Pr, H, OMe, O, CHF 2 , H, H, H, O ], [AK1041; H, i-Pr, H, OMe, O, CF 3, H, H, H, O], [AK1042; H, i-Pr, H, OMe, _{O, OCH 2 F, H,} H, H, O], [AK1043; H, i-Pr, H, OMe, O, OCHF 2, H, H, H, O], [AK1044; H, i-Pr , H, OMe, O, OCF 3, H, H, H, O], [AK1045; H, i-Pr, H, OMe, O, OCF 3, H, H, H, O], [AK1046; H , i-Pr, H, F, O, H, H, H, H, O], [AK1047; H, i-Pr, H, F, O, F, H, H, H, O], [AK1048 H, i-Pr, H, F, O, Cl, H, H, O], [AK1049; H, i-Pr, H, F, O, Br, H, H, H, O], [AK 1050; H, i-Pr, H, F, O, I, H, H, H, O], [AK 1051; H, i-Pr, H, F, O, Me, H, H, H, O ], [AK10 52; H, i-Pr, H, F, O, Et, H, H, H, O], [AK1053; H, i-Pr, H, F, O, Pr, H, H, H, O] [AK1054; H, i-Pr, H, F, O, i-Pr, H, H, H, O], [AK1055; H, i-Pr, H, F, O, Bu, H, H, H, O], [AK1056; H, i-Pr, H, F, O, i-Bu, H, H, H, O], [AK1057; H, i-Pr, H, F, O, sec- Bu, H, H, H, O], [AK 1058; H, i-Pr, H, F, O, t-Bu, H, H, H, O], [AK 1059; H, i-Pr, H, F, O, c-Pr, H, H, H, O, [AK 1060; H, i-Pr, H, F, O, c-Bu, H, H, O], [AK 1061; H, i-Pr, H, F, O, OBu, H, H, H, O], [AK1062; H, i-Pr, H, F, O, Oi-Bu, H, H, H, O], [[ AK1063; H, i-Pr, H, F, O, O-sec-Bu, H, H, H, O], [AK1064; H, i-Pr, H, F, O, CH 2 F, H, H, H, O], [AK 1065; H, i-Pr, H, F, O, CHF ₂ , H, H, H, O], [AK 1066; H, i-Pr, H, F, O, CF _{3, H, H, H,} O], [AK1067; H, i-Pr, H, F, O, OCH 2 F, H, H, H, O], [AK1068; H, i-Pr, H, _{F, O, OCHF 2, H} , H, H, O], [AK1069; H, i-Pr, H, F, O, OCF 3, H, H, H, O], [AK1070; H, i- Pr, H, F, O, OCF 3, H, H, H, O], [AK1071; H, i-Pr, H, Cl, O, H, H, H, H, O], [AK1072; H , i-Pr, H, Cl, O, F, H, H, H, O], [AK1073; H, i-Pr, H, Cl, O, Cl, H, H, H, O], [AK1074 H, i-Pr, H, Cl, O, Br, H, H, O], [AK1075; H, i-Pr, H, Cl, O, I, H, H, H, O], [AK1076; H, i-Pr, H, Cl, O, Me, H, H, H, O], [AK1077; H, i-Pr, H, Cl, O, Et, H, H, H, O ], [AK1078; H, i-Pr, H, Cl, O, Pr, H, H, H, O], [A K 1079; H, i-Pr, H, Cl, O, i-Pr, H, H, H, O], [AK 1080; H, i-Pr, H, Cl, O, Bu, H, H, H, H, O], [AK1081; H, i-Pr, H, Cl, O, i-Bu, H, H, H, O], [AK1082; H, i-Pr, H, Cl, O, sec-Bu, H, H, H, O], [AK1083; H, i-Pr, H, Cl, O, t-Bu, H, H, H, O], [AK1084; H, i-Pr, H, Cl, O, c-Pr, H, H, H, O], [AK1085; H, i-Pr, H, Cl, O, c-Bu, H, H, H, O], [AK1086; H, i- Pr, H, Cl, O, OBu, H, H, H, O], [AK1087; H, i-Pr, H, Cl, O, Oi-Bu, H, H, H, O], [AK1088; H, i-Pr, H, Cl, O, O-sec-Bu, H, H, H, O], [AK1089; H, i-Pr, H, Cl, O, CH 2 F, H, H, H, O], [AK 1090; H, i-Pr, H, Cl, O, CHF ₂ , H, H, H, O], [AK1091; H, i-Pr, H, Cl, O, CF ₃ , H, H, H, O] , [AK1092; H, i-Pr, H, Cl, O, OCH 2 F, H, H, H, O], [AK1093; H, i-Pr, H, Cl, _{O, OCHF 2, H, H} , H, O], [AK1094; H, i-Pr, H, Cl, O, OCF 3, H, H, H, O], [AK1095; H, i-Pr, _{H, Cl, O, OCF 3} , H, H, H, O], [AK1096; H, i-Pr, H, Br, O, H, H, H, H, O], [AK1097; H, i -Pr, H, Br, O, F, H, H, H, O], [AK1098; H, i-Pr, H, Br, O, Cl, H, H, H, O], [AK1099; H , i-Pr, H, Br, O, Br, H, H, H, O], [AK1100; H, i-Pr, H, Br, O, I, H, H, H, O],

[AK1101; H, i-Pr, H, Br, O, Me, H, H, H, O], [AK 1102; H, i-Pr, H, Br, O, Et, H, H, H, O H, i-Pr, H, Br, O, Pr, H, H, H, O], [AK 1104; H, i-Pr, H, Br, O, i-Pr, H, H] , H, O], [AK 1 105; H, i-Pr, H, Br, O, Bu, H, H, H, O], [AK 1106; H, i-Pr, H, Br, O, i-Bu , H, H, H, O], [AK 1107; H, i-Pr, H, Br, O, sec-Bu, H, H, H, O], [AK 1108; H, i-Pr, H, Br] , O, t-Bu, H, H, H, O], [AK 1109; H, i-Pr, H, Br, O, c-Pr, H, H, H, O], [AK1 110; H, i -Pr, H, Br, O, c-Bu, H, H, H, O], [AK1 111; H, i-Pr, H, Br, O, OBu, H, H, H, O], [AK 1112 H, i-Pr, H, Br, O, Oi-Bu, H, H, H, O], [AK1113; H, i-Pr, H, Br, O, O-sec-Bu, H, H , H, O], [AK 1114; H, i-Pr, H, Br, O, CH ₂ F, H, H, H, O], [AK 1115; H, i-Pr, H, Br, O, CHF _{2, H, H, H,} O], [AK1116; H, i-Pr, H, Br, O, CF 3, H, H, H, O], [AK1117; H, i-Pr, H, Br , O, OCH ₂ F, H, H, H, O], [AK 1118; H, i-Pr, H, Br, O, OCHF ₂ , H, H, H, O], [AK 1 119; H, i- Pr, H, Br, O, OCF 3, H, H, H, O], [AK1120; H, i-Pr, H, Br, O, OCF 3, H, H, H, O], [AK1121; H, F, H, H, O, H, H, H, H, O], [AK1122; H, F, H, H, O, F, H, H, O], [AK 1123; H, F, H, H, H, O, Cl, H, H, H, O], [AK 1 124; H, F, H, H, O, Br, H, H, O], [AK 1 125; H, F, H, H, O, I, H, H, H, O], [AK 1 126; H, F, H, H, O, Me, H, H, H, O], [AK 1 127; H, F, H, H, O, Et, H, H, H, O], [AK112 8; H, F, H, H, H, O, Pr, H, H, H, O], [AK 1129; H, F, H, H, O, i-Pr, H, H, H, O], [[1] AK1130; H, F, H, H, H, O, Bu, H, H, H, O], [AK1131; H, F, H, H, O, i-Bu, H, H, H, O], [A AK1132; H, F, H, H, H, O, sec-Bu, H, H, H, O], [AK 1133; H, F, H, H, O, t-Bu, H, H, H, O] [AK 1134; H, F, H, H, O, c-Pr, H, H, H, O], [AK 1 135; H, F, H, H, O, c-Bu, H, H, H, O], [AK 1136; H, F, H, H, O, OBu, H, H, H, O], [AK 1 137; H, F, H, H, O, Oi-Bu, H, H, H, O], [AK 1138; H, F, H, H, O, O-sec-Bu, H, H, H, O], [AK 1139; H, F, H, H, O, CH ₂ F, H, H, H, O], [ AK1140; H, F, H, H, O, CHF 2, H, H, H, O], [AK1141; H, F, H, H, O, CF 3, H, H, H, O], [ AK1142; H, F, H, H, O, OCH 2 F, H, H, H, O], [AK1143; H, F, H, H, O, OCHF 2, H , H, H, O], [AK1144; H, F, H, H, O, OCF 3, H, H, H, O], [AK1145; H, F, H, Me, O, H, H, H, H, O], [AK 1146; H, F, H, Me, O, F, H, H, H, O], [AK 1147; H, F, H, Me, O, Cl, H, H, H, O], [AK1148; H, F, H, Me, O, Br, H, H, H, O], [AK 1149; H, F, H, Me, O, I, H, H, H, H, O], [AK1150; H, F, H, Me, O, Me, H, H, H, O], [AK1151; H, F, H, Me, O, Et, H, H, H, O] [AK1152; H, F, H, Me, O, Pr, H, H, H, O], [AK1153; H, F, H, Me, O, i-Pr, H, H, H, O] [AK 1154; H, F, H, Me, O, Bu, H, H, H, O], [AK 1 155; H, F, H, Me, O, i-Bu, H, H, H, O] [AK 1156; H, F, H, Me, O, sec-Bu, H, H, H, O], [AK 1 157; H, F, H, Me, O, t-Bu, H, H, H, O], [AK1158; H, F, H, Me, O, c-Pr, H, H, H, O], [AK1 159; H, F, H, Me, O, c-Bu, H, H, H, O], [AK 1 160; H, F, H, Me, O, OBu, H, H, H, O], [AK 1161; H, F, H, Me, O, Oi-Bu, H, H, H, O], [AK1162; H, F, H, Me, O, O-sec-Bu, H, H, H, O], [[ AK1163; H, F, H, Me, O, CH 2 F, H, H, H, O], [AK1164; H, F, H, Me, O, CHF 2, H, H, H, O], [AK1165; H, F, H , Me, O, CF 3, H, H, H, O], [AK1166; H, F, H, Me, O, OCH 2 F, H, H, H, O] , [AK1167; H, F, H, Me, O, OCHF 2, H, H, H, O], [AK1168; H, F, H, Me, O, OCF 3, H, H, H, O] , [AK1169; H, F, H, Me, O, OCF 3, H, H, H, O], [AK1170; H, F, H, Et, O, H, H, H, H, O], [AK1171; H, F, H, Et, O, F, H, H, O], [AK1172; H, F, H, Et, O, Cl, H, H, H, O], [AK1173 H, F, H, Et, O, Br, H, H, O], [AK 1174; H, F, H, Et, O, I, H, H, H, O], [AK 1 175; H , F, H, Et, O, Me, H, H, H, O], [AK 1176; H, F, H, Et, O, Et, H, H, H, O], [AK1177; H, F , H, Et, O, Pr, H, H, H, O], [AK1178; H, F, H, Et, O, i-Pr, H, H, H, O], [AK1179; H, F , H, Et, O, Bu, H, H, H, O], [AK 1180; H, F, H, Et, O, i-Bu, H, H, H, O], [AK1181; H, F , H, Et, O, sec-Bu, H, H, H, O], [AK1182; H, F, H, Et, O, t-Bu, H, H, H, O], [AK1183; H , F, H, Et, O, c-Pr, H, H, H, O], [AK 1184; H, F, H, Et, O, c-Bu, H, H, H, O], [AK 1 185] H, F, H, Et, O, OBu, H, H, H, O] [AK1186; H, F, H, Et, O, Oi-Bu, H, H, H, O], [AK1187; H, F, H, Et, O, O-sec-Bu, H, H, H H, F, H, Et, O, CH ₂ F, H, H, H, O], [AK 1189; H, F, H, Et, O, CHF ₂ , H, H, H, O], [AK1190; H, F, H, Et, O, CF 3, H, H, H, O], [AK1191; H, F, H, Et, O, OCH 2 F, H, H , H, O], [AK1192 ; H, F, H, Et, O, OCHF 2, H, H, H, O], [AK1193; H, F, H, Et, O, OCF 3, H, H , H, O], [AK1194 ; H, F, H, Et, O, OCF 3, H, H, H, O], [AK1195; H, F, H, Pr, O, H, H, H, H, O], [AK1196; H, F, H, Pr, O, F, H, H, H, O], [AK 1197; H, F, H, Pr, O, Cl, H, H, H, H, O], [AK 1198; H, F, H, Pr, O, Br, H, H, O], [AK 1 199; H, F, H, Pr, O, I, H, H, H, O] [AK 1200; H, F, H, Pr, O, Me, H, H, H, O],

[AK1201; H, F, H, Pr, O, Et, H, H, H, O], [AK1202; H, F, H, Pr, O, Pr, H, H, H, O], [AK1203 H, F, H, Pr, O, i-Pr, H, H, H, O], [AK 1204; H, F, H, Pr, O, Bu, H, H, H, O], [AK 1205 H, F, H, Pr, O, i-Bu, H, H, H, O], [AK1206; H, F, H, Pr, O, sec-Bu, H, H, H, O], [AK1207; H, F, H, Pr, O, t-Bu, H, H, H, O], [AK 1208; H, F, H, Pr, O, c-Pr, H, H, H, O H, F, H, Pr, O, c-Bu, H, H, H, O], [AK 1210; H, F, H, Pr, O, OBu, H, H, H, O] H, F, H, Pr, O, Oi-Bu, H, H, H, O], [AK 1212; H, F, H, Pr, O, O-sec-Bu, H, H] , H, O], [AK 1213; H, F, H, Pr, O, CH ₂ F, H, H, H, O], [AK 1214; H, F, H, Pr, O, CHF ₂ , H, H, H, O], [AK 1215; H, F, H, Pr, O, CF ₃ , H, H, H, O], [AK 1216; H, F, H, Pr, O, OCH ₂ F, H , H, H, O], [AK1217; H, F, H, Pr, O, OCHF 2, H, H, H, O], [AK1218; H, F, H, Pr, O, OCF 3, H , H, H, O], [AK1219; H, F, H, Pr, O, OCF 3, H, H, H, O], [AK1220; H, F, H, i-Pr, O, H, H, H, H, O], [AK1221; H, F, H, i-Pr, O, F, H, H, H, O], [AK1222; H, F, H, i-Pr, O, Cl, H, H, H, O], [AK1223; H, F, H, i-Pr, O, Br, H, H, H, O], [AK1224; H, F, H, i-Pr, O, I, H, H, H, O], [AK 12 25; H, F, H, i-Pr, O, Me, H, H, H, O], [AK 1226; H, F, H, i- Pr, O, Et, H, H, H, O], [AK1227; H, F, H, i-Pr, O, Pr, H, H, H, O], [AK1228; H, F, H, i-Pr, O, i-Pr, H, H, H, O], [AK122 9; H, F, H, i-Pr, O, Bu, H, H, H, O], [AK1230; H, F, H, i-Pr, O, i-Bu, H, H, H, H O], [AK1231; H, F, H, i-Pr, O, sec-Bu, H, H, H, O], [AK1232; H, F, H, i-Pr, O, t-Bu, H, H, H, O], [AK1233; H, F, H, i-Pr, O, c-Pr, H, H, H, O], [AK1234; H, F, H, i-Pr, O, c-Bu, H, H, H, O], [AK1235; H, F, H, i-Pr, O, OBu, H, H, H, O], [AK1236; H, F, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK1237; H, F, H, i-Pr, O, O-sec-Bu, H, H, H, O], [[ AK1238; H, F, H, i-Pr, O, CH 2 F, H, H, H, O], [AK1239; H, F, H, i-Pr, O, CHF 2, H, H, H , O], [AK1240; H , F, H, i-Pr, O, CF 3, H, H, H, O], [AK1241; H, F, H, i-Pr, O, OCH 2 F, H, H, H, O] , [AK1242; H, F, H, i-Pr, O, OCHF 2, H, H, H, O], [AK1243; H, F, H, i-Pr, O , OCF ₃ , H, H, H, O], [AK 1244; H, F, H, i-Pr, O, OCF ₃ , H, H, H, O], [AK 1245; H, F, H, OMe , O, H, H, H, H, O], [AK 1246; H, F, H, OMe, O, F, H, H, H, O], [AK 1247; H, F, H, OMe, O , Cl, H, H, H, O], [AK 1248; H, F, H, OMe, O, Br, H, H, H, O], [AK 1249; H, F, H, OMe, O, I H, H, H, O], [AK 1 250; H, F, H, OMe, O, Me, H, H, H, O], [AK 1251; H, F, H, OMe, O, Et, H H, H, O], [AK 1252; H, F, H, OMe, O, Pr, H, H, H, O], [AK 1253; H, F, H, OMe, O, i-Pr, H , H, H, O], [AK1254; H, F, H, OMe, O, Bu, H, H, H, O], [AK1 255; H, F, H, OMe, O, i-Bu, H , H, H, O], [AK 1 256; H, F, H, OMe, O, sec-Bu, H, H, H, O], [AK1257; H, F, H, OMe, O, t-Bu, H, H, H, O], [AK1258; H, F, H, OMe, O, c-Pr, H, H, H, O], [AK 1259; H, F, H, OMe, O, c-Bu, H, H, H, O], [AK 1260; H, F, H, OMe, O, OBu, H, H, H, O], [AK 1261; H, F, H, OMe, O, Oi-Bu, H, H, H, O], [AK 1262; H, F, H, OMe, O, O-sec-Bu, H, H, H, O], [AK 1263; H, F, H, OMe, O, CH ₂ F, H, H, O, [AK 1264; H, F, H, OMe, O, CHF 2, H, H, H, O], [AK1265; H, F, H, OMe, O, CF 3, H, H, H, O], [AK1266; H, F, H, OMe, O, OCH 2 F, H, H, H, O], [AK1267; H, F, H, OMe, O, OCHF 2, H, H, H, O], [AK1268; H , F, H, OMe, O , OCF 3, H, H, H, O], [AK1269; H, F, H, OMe, O, OCF 3, H, H, H, O], [AK1270; H , F, H, F, O, H, H, H, H, O], [AK1271; H, F, H, F, O, F, H, H, O], [AK 1272; H, F , H, F, O, Cl, H, H, H, O], [AK1273; H, F, H, F, O, Br, H, H, H, O], [AK1274; H, F, H] , F, O, I, H, H, H, O], [AK 1275; H, F, H, F, O, Me, H, H, H, O], [AK 1276; H, F, H, F] , O, Et, H, H, H, O], [AK 1277; H, F, H, F, O, Pr, H, H, H, O], [AK 1 278; H, F, H, F, O , i-Pr, H, H, H, O], [AK 1279; H, F, H, F, O, Bu, H, H, H, O], [AK 1280; H, F, H, F, O] , i-Bu, H, H, H, O], [AK1281; H, F, H, F, O, sec-Bu, H, H, H, O], [AK1282; H, F, H, F] , O, t-Bu, H, H, H, O], [AK1283; H, F, H, F, O, c-Pr, H, H, H, O], [AK1284; H, F, H] , F, O, c-Bu, H, H, H, O], [AK1 H, F, H, F, O, O, OBu, H, H, H, O], [AK 1286; H, F, H, F, O, Oi-Bu, H, H, H, O], AK1287; H, F, H, F, O, O-sec-Bu, H, H, H, O], [AK1288; H, F, H, F, O, CH 2 F, H, H, H, O], [AK1289; H, F, H, F, O, CHF ₂ , H, H, H, O], [AK 1290; H, F, H, F, O, CF ₃ , H, H, H, O], [AK1291; H, F, H, F, O, OCH 2 F, H, H, H, O], [AK1292; H, F, H, F, O, OCHF 2, H, H, H , O], [AK1293; H , F, H, F, O, OCF 3, H, H, H, O], [AK1294; H, F, H, F, O, OCF 3, H, H, H , O], [AK 1295; H, F, H, Cl, O, H, H, H, H, O], [AK 1296; H, F, H, Cl, O, F, H, H, H, O H, F, H, Cl, O, Cl, H, H, H, O], [AK 1298; H, F, H, Cl, O, Br, H, H, H, O], [AK1299; H, F, H, Cl, O, I, H, H, O], [AK 1300; H, F, H, Cl, O, Me, H, H, H, O],

[AK1301; H, F, H, Cl, O, Et, H, H, H, O], [AK1302; H, F, H, Cl, O, Pr, H, H, H, O], [AK1303 H, F, H, Cl, O, i-Pr, H, H, H, O], [AK1304; H, F, H, Cl, O, Bu, H, H, H, O], [AK1 305 H, F, H, Cl, O, i-Bu, H, H, H, O], [AK 1306; H, F, H, Cl, O, sec-Bu, H, H, H, O], [AK1307; H, F, H, Cl, O, t-Bu, H, H, H, O], [AK1 308; H, F, H, Cl, O, c-Pr, H, H, H, O H, F, H, Cl, O, c-Bu, H, H, H, O], [AK 1310; H, F, H, Cl, O, OBu, H, H, H, O] H, F, H, Cl, O, Oi-Bu, H, H, H, O], [AK1312; H, F, H, Cl, O, O-sec-Bu, H, H] H, O, [AK 1313; H, F, H, Cl, O, CH ₂ F, H, H, H, O], [AK 1314; H, F, H, Cl, O, CHF ₂ , H, H, H, O], [ AK1315; H, F, H, Cl, O, CF 3, H, H, H, O], [AK1316; H, F, H, Cl, O, OCH 2 F, H , H, H, O], [AK1317; H, F, H, Cl, O, OCHF 2, H, H, H, O], [AK1318; H, F, H, Cl, O, OCF 3, H , H, H, O], [AK1319; H, F, H, Cl, O, OCF 3, H, H, H, O], [AK1320; H, F, H, Br, O, H, H, H, H, O], [AK1321; H, F, H, Br, O, F, H, H, H, O], [AK1322; H, F, H, Br, O, Cl, H, H, H, O], [AK1323; H, F, H, Br, O, Br, H, H, H, O], [AK1324; H, F, H, Br, O, I, H, H, H, O], [AK 1325; H, F, H, Br, O, Me, H, H, H, O], [AK 1326; H, F, H, Br, O, Et, H, H, H, O] [AK1327; H, F, H, Br, O, Pr, H, H, H, O], [AK1328; H, F, H, Br, O, i-Pr, H, H, H, O] [AK1329; H, F, H, Br, O, Bu, H, H, H, O], [AK1330; H, F, H, Br, O, i-Bu, H, H, H, O], [AK1331; H, F, H, Br, O, sec-Bu, H, H, H, O], [AK1332; H, F, H, Br, O, t-Bu, H, H, H, O], [AK1333; H, F, H, Br, O, c- Pr, H, H, H, O], [AK1334; H, F, H, Br, O, c-Bu, H, H, H, O], [AK 1335; H, F, H, Br, O, OBu, H, H, H, O], [AK1336; H, F, H, Br, O, Oi-Bu, H, H, H, O], [AK 1337; H, F, H, Br, O, O-sec-Bu, H, H, H, O], [AK1338; H, F, H, Br, O, CH 2 F, H, H, H, O], [AK1339; H, F, H, _{Br, O, CHF 2, H} , H, H, O], [AK1340; H, F, H, Br, O, CF 3, H, H, H, O], [AK1341; H, F, H, _{Br, O, OCH 2 F,} H, H, H, O], [AK1342; H, F, H, Br, O, OCHF 2, H, H, H, O], [AK1343; H, F, H _{, Br, O, OCF 3,} H, H, H, O], [AK1344; H, F, H, Br, O, OCF 3, H, H, H, O], [AK1345; H, Cl, H , H, O, H, H, H, H, O], [AK 1346; H, Cl, H, H, O, F, H, H, H, O], [AK 1347; H, Cl, H, H] , O, Cl, H, H, H, O], [AK1348; H, Cl, H, H, O, Br, H, H, H, O], [AK1 349; H, Cl, H, H, O] , I, H, H, H, O], [AK1 350; H, Cl, H, H, O, Me, H, H, H, O], [AK1351; H, Cl, H, H, O, Et] , H, H, H, O], [AK1352; H, Cl, H, H, O, Pr, H, H, H, O], [AK1353; H, Cl, H, H, O, i-Pr H, H, H, O], [AK1354; H, Cl, H, H, O, Bu, H, H, H, O], [AK1 355; H, Cl, H, H, O, i-Bu , H, H, H, O], [AK 1356; H, Cl, H, H, O, sec-Bu, H, H, H, O], [AK 1 357; H, Cl, H, H, O, t -Bu, H, H, H, O], [AK1358; H , Cl, H, H, O, c-Pr, H, H, H, O], [AK1359; H, Cl, H, H, O, c-Bu, H, H, H, O], [AK1360 H, Cl, H, H, H, O, OBu, H, H, H, O], [AK1361; H, Cl, H, H, O, Oi-Bu, H, H, H, O], [AK1362 ; H, Cl, H, H , O, O-sec-Bu, H, H, H, O], [AK1363; H, Cl, H, H, O, CH 2 F, H, H, H, O ], [AK1364; H, Cl , H, H, O, CHF 2, H, H, H, O], [AK1365; H, Cl, H, H, O, CF 3, H, H, H, O H, Cl, H, H, H, O, OCH ₂ F, H, H, H, O], [AK 1367; H, Cl, H, H, O, OCHF ₂ , H, H, H, O], [AK1368; H, Cl, H, H, O, OCF 3, H, H, H, O], [AK1369; H, Cl, H, Me, O, H, H, H, H, O H, Cl, H, Me, O, F, H, H, O], [AK1371; H, Cl, H, Me, O, Cl, H, H, H, O], [AK1372; H, Cl, H, Me, O, Br, H, H, O], [AK1373; H, Cl, H, Me, O, I, H, H, H, O], [AK1374 H, Cl, H, Me, O, Me, H, H, H, O], [AK 1375; H, Cl, H, Me, O, Et, H, H, H, O], [AK 1376; H , Cl, H, Me, O, Pr, H, H, H, O], [AK1 377; H, Cl, H, Me, O, i-Pr, H, H, H, O], [AK 1378; H , Cl, H, Me, O, Bu, H, H, H, O], [AK 1379; H, Cl, H, Me, O, i-Bu, H, H, H, O], [AK 1 380; H , Cl, H, Me, O, sec-Bu, H, H, H, O], [AK1381; H, Cl, H, Me, O, t-Bu, H, H, H, O], [AK1382 H, Cl, H, Me, O, c-Pr, H, H, H, O], [AK1383; H, Cl, H, Me, O, c-Bu, H, H, H, O], [AK1384; H, Cl, H, Me, O, OBu, H, H, H, O], [AK1 385; H, Cl, H, Me, O, Oi-Bu, H, H, H, O], [AK 1386; H, Cl, H , Me, O, O-sec -Bu, H, H, H, O], [AK1387; H, Cl, H, Me, O, CH 2 F, H, H, H, O], [AK1388; H , Cl, H, Me, O , CHF 2, H, H, H, O], [AK1389; H, Cl, H, Me, O, CF 3, H, H, H, O], [AK1390; H , Cl, H, Me, O , OCH 2 F, H, H, H, O], [AK1391; H, Cl, H, Me, O, OCHF 2, H, H, H, O], [AK1392; H, Cl, H, Me, O, OCF 3, H, H, H, O], [AK1393; H, Cl, H, Me, O, OCF 3, H, H, H, O], [AK1394; H, Cl, H, Et, O, H, H, H, H, O], [AK 1395; H, Cl, H, Et, O, F, H, H, H, O], [AK 1 396; H, Cl, H, Et, O, Cl, H, H, H, O], [AK 1397; H, Cl, H, Et, O, Br, H, H, H, O], [AK 1398; H, Cl, H, Et, O, I, H, H, H, O], [AK1399; H, Cl, H, Et, O, Me, H, H, H, O], [AK1400; H, Cl, H, Et, O, Et, H, H, H, O],

[AK 1401; H, Cl, H, Et, O, Pr, H, H, H, O], [AK 1402; H, Cl, H, Et, O, i-Pr, H, H, H, O], [AK 1403; H, Cl, H, Et, O, Bu, H, H, H, O], [AK 1404; H, Cl, H, Et, O, i-Bu, H, H, H, O], [AK1405; H, Cl, H, Et, O, sec-Bu, H, H, H, O], [AK 1406; H, Cl, H, Et, O, t-Bu, H, H, H, O H, Cl, H, Et, O, c-Pr, H, H, H, O], [AK 1408; H, Cl, H, Et, O, c-Bu, H, H, H] H, Cl, H, Et, O, OBu, H, H, H, O], [AK 1410; H, Cl, H, Et, O, Oi-Bu, H, H, H] H, Cl, H, Et, O, O-sec-Bu, H, H, H, O], [AK 1412; H, Cl, H, Et, O, CH ₂ F, H , H, H, O], [AK1413; H, Cl, H, Et, O, CHF 2, H, H, H, O], [AK1414; H, Cl, H, Et, O, CF 3, H H, H, O], [AK 1415; H, Cl, H, Et, O, OCH ₂ F, H, H, H, O], [AK 1416; H, Cl, H, Et, O, OCHF ₂ , H, H, H, O] , [AK1417; H, Cl, H, Et, O, OCF 3, H, H, H, O], [AK1418; H, Cl, H, Et, O, OCF 3, H, H, H, O], [AK 1419; H, Cl, H, Pr, O, H, H, H, H, O], [AK 1420; H, Cl, H, Pr, O, F, H, H, H, O], [AK1421; H, Cl, H, Pr, O, Cl, H, H, H, O], [AK1422; H, Cl, H, Pr, O, Br, H, H, H, H, O], [AK1423; H, Cl, H, Pr, O, I, H, H, H, O], [AK1424; H, Cl, H, Pr, O, Me, H, H, H, H, O], [AK 1425; H, Cl, H, Pr, O, Et, H, H, O], [AK 1426; H, Cl, H, Pr, O, Pr, H, H, H, O] [AK 1427; H, Cl, H, Pr, O, i-Pr, H, H, H, O], [AK 1428; H, Cl, H, Pr, O, Bu, H, H, H, O H, Cl, H, Pr, O, i-Bu, H, H, H, O], [AK 1430; H, Cl, H, Pr, O, sec-Bu, H, H, H] H, Cl, H, Pr, O, t-Bu, H, H, H, O], [AK 1432; H, Cl, H, Pr, O, c-Pr, H, H] , H, O], [AK 1433; H, Cl, H, Pr, O, c-Bu, H, H, H, O], [AK 1434; H, Cl, H, Pr, O, OBu, H, H] H, O], [AK1435; H, Cl, H, Pr, O, Oi-Bu, H, H, H, O], [AK1436; H, Cl, H, Pr, O, O-sec-Bu , H, H, H, O ], [AK1437; H, Cl, H, Pr, O, CH 2 F, H, H, H, O], [AK1438; H, Cl, H, Pr, O, CHF _{2, H, H, H,} O], [AK1439; H, Cl, H, Pr, O, CF 3, H, H, H, O], [AK1440; H, Cl, H, Pr, O, OCH _{2 F, H, H, H} , O], [AK1441; H, Cl, H, Pr, O, OCHF 2, H, H, H, O], [AK1442; H, Cl, H, Pr, O, OCF ₃ , H, H, H, O], [AK 1443; H, Cl, H, Pr, O, OCF ₃ , H, H, H, O], [AK 1444; H, Cl, H, i-Pr, O, H, H, H, H, O], [AK 1445; H, Cl, H, i-Pr, O, F, H, H, H, O], [AK 1446; H, Cl, H, i- Pr, O, Cl, H, H, H, O], [AK1447; H, Cl, H, i-Pr, O, Br, H, H, H, O], [AK 1448; H, Cl, H, i-Pr, O, I, H, H, H, O], [AK1449; H, Cl, H, i-Pr, O, Me, H, H, H, O], [AK 1450; H, Cl, H, i-Pr, O, Et, H, H, H, O], [AK1451; H, Cl, H, i-Pr, O, Pr, H, H, H, O], [AK1452; H, Cl, H, i-Pr, O, i-Pr, H, H, H, O], [AK1453; H, Cl, H, i-Pr, O, Bu, H, H, H, O], [[A] AK1454; H, Cl, H, i-Pr, O, i-Bu, H, H, H, O], [AK1455; H, Cl, H, i-Pr, O, sec-Bu, H, H, H, O] [AK1456; H, Cl, H, i-Pr, O, t-Bu, H, H, H, O], [AK1 457; H, Cl, H, i-Pr, O, c-Pr, H, H , H, O], [AK1458; H, Cl, H, i-Pr, O, c-Bu, H, H, H, O], [AK1459; H, Cl, H, i-Pr, O, OBu , H, H, H, O], [AK 1460; H, Cl, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK 1461; H, Cl, H, i-Pr , O, O-sec-Bu , H, H, H, O], [AK1462; H, Cl, H, i-Pr, O, CH 2 F, H, H, H, O], [AK1463; H , Cl, H, i-Pr , O, CHF 2, H, H, H, O], [AK1464; H, Cl, H, i-Pr, O, CF 3, H, H, H, O], [AK1465; H, Cl, H , i-Pr, O, OCH 2 F, H, H, H, O], [AK1466; H, Cl, H, i-Pr, O, OCHF 2, H, H, H, O], [AK1467; H, Cl, H, i-Pr, O, OCF 3, H, H, H, O], [AK1468; H, Cl, H, i-Pr, O, OCF 3, H, H, H, O], [AK1469; H, Cl, H, OMe, O, H, H, H, H, O], [AK 1470; H, Cl, H, OMe, O, F, H, H, H, O], [AK1471; H, Cl, H, OMe, O, Cl, H, H, H, O], [AK1472; H, Cl, H, OMe, O, Br, H, H, H, O], [AK 1 473; H, Cl, H, OMe, O, I, H, H, H, O], [AK 1 474; H, Cl, H, OMe, O, Me, H, H, H, O], [AK1475; H, Cl, H, OMe, O, Et, H, H, H, O], [AK1 476; H, Cl, H, OMe, O, Pr, H, H, H, O] [AK1477; H, Cl, H, OMe, O, i-Pr, H, H, H, O], [AK1478; H, Cl, H, OMe, O, Bu, H, H, H, O] [AK1479; H, Cl, H, OMe, O, i-Bu, H, H, H, O], [AK 1480; H, Cl, H, OMe, O, sec-Bu, H, H, H, O], [AK1481; H, Cl, H, OMe, O, t-Bu, H, H, H, O], [AK1482; H, Cl, H, OMe, O, c- Pr, H, H, H, O], [AK 1483; H, Cl, H, OMe, O, c-Bu, H, H, H, O], [AK 1484; H, Cl, H, OMe, O, OBu, H, H, H, O], [AK1485; H, Cl, H, OMe, O, Oi-Bu, H, H, H, O], [AK1486; H, Cl, H, OMe, O, O-sec-Bu, H, H, H, O], [AK 1487; H, Cl, H, OMe, O, CH ₂ F, H, H, H, O], [AK 1 488; H, Cl, H, _{OMe, O, CHF 2, H} , H, H, O], [AK1489; H, Cl, H, OMe, O, CF 3, H, H, H, O], [AK1490; H, Cl, H, _{OMe, O, OCH 2 F,} H, H, H, O], [AK1491; H, Cl, H, OMe, O, OCHF 2, H, H, H, O], [AK1492; H, Cl, H _{, OMe, O, OCF 3,} H, H, H, O], [AK1493; H, Cl, H, OMe, O, OCF 3, H, H, H, O], [AK1494; H, Cl, H , F, O, H, H, H, H, O], [AK 1495; H, Cl, H, F, O, F, H, H, H, O], [AK 1496; H, Cl, H, F] , O, Cl, H, H, H, O, [AK 1497; H, Cl, H, F, O, Br, H, H, H, O], [AK 1498; H, Cl, H, F, O , I, H, H, H, O], [AK 1499; H, Cl, H, F, O, Me, H, H, H, O], [AK 1500; H, Cl, H, F, O, Et , H, H, H, O],

[AK1501; H, Cl, H, F, O, Pr, H, H, H, O], [AK1502; H, Cl, H, F, O, i-Pr, H, H, H, O], [AK1503; H, Cl, H, F, O, Bu, H, H, H, O], [AK1504; H, Cl, H, F, O, i-Bu, H, H, H, O], [AK1505; H, Cl, H, F, O, sec-Bu, H, H, H, O], [AK1506; H, Cl, H, F, O, t-Bu, H, H, H, O H, Cl, H, F, O, c-Pr, H, H, H, O], [AK1508; H, Cl, H, F, O, c-Bu, H, H, H] H, Cl, H, F, O, OBu, H, H, H, O], [AK 1510; H, Cl, H, F, O, Oi-Bu, H, H, H] H, Cl, H, F, O, O-sec-Bu, H, H, H, O], [AK 1512; H, Cl, H, F, O, CH ₂ F, H H, H, O], [AK 1513; H, Cl, H, F, O, CHF ₂ , H, H, H, O], [AK 1514; H, Cl, H, F, O, CF ₃ , H H, H, O], [AK 1515; H, Cl, H, F, O, OCH ₂ F, H, H, H, O], [AK 1516; H, Cl, H, F, O, OCHF ₂ , H, H, H, O] , [AK1517; H, Cl, H, F, O, OCF 3, H, H, H, O], [AK1518; H, Cl, H, F, O, OCF 3, H, H, H, O], [AK 1519; H, Cl, H, Cl, O, H, H, H, H, O], [AK 1520; H, Cl, H, Cl, O, F, H, H, H, O], [AK1521; H, Cl, H, Cl, O, Cl, H, H, H, O], [AK1522; H, Cl, H, Cl, O, Br, H, H, H, O], [AK1523; H, Cl, H, Cl, O, I, H, H, H, O], [AK1524; H, Cl, H, Cl, O, Me, H, H, H, H, O], [AK1525; H, Cl, H, Cl, O, Et, H, H, H, O], [AK1526; H, Cl, H, Cl, O, Pr, H, H, H, O] [AK1527; H, Cl, H, Cl, O, i-Pr, H, H, H, O], [AK1 528; H, Cl, H, Cl, O, Bu, H, H, H, O] , [AK1529; H, Cl, H , Cl, O, i-Bu, H, H, H, O], [AK1530; H, Cl, H, Cl, O, sec-Bu, H, H, H, O], [AK 1531; H, Cl , H, Cl, O, t-Bu, H, H, H, O], [AK 1532; H, Cl, H, Cl, O, c-Pr, H, H, H, O], [AK 1533; H , Cl, H, Cl, O, c-Bu, H, H, H, O], [AK1534; H, Cl, H, Cl, O, OBu, H, H, H, O], [AK1535; H , Cl, H, Cl, O, Oi-Bu, H, H, H, O], [AK1536; H, Cl, H, Cl, O, O-sec-Bu, H, H, H, O], [AK1537; H, Cl, H , Cl, O, CH 2 F, H, H, H, O], [AK1538; H, Cl, H, Cl, O, CHF 2, H, H, H, O] , [AK1539; H, Cl, H, Cl, O, CF 3, H, H, H, O], [AK1540; H, Cl, H, Cl, O, OCH 2 F, H, H, H, O H, Cl, H, Cl, O, OCHF ₂ , H, H, H, O], [AK 1542; H, Cl, H, Cl, O, OCF ₃ , H, H, H, O] ], [AK1543; H, Cl , H, Cl, O, OCF 3, H, H, H, O], [AK1544; H, Cl, H, Br, O, H, H, H, H, O] [AK1545; H, Cl, H, Br, O, F, H, H, O], [AK1546; H, Cl, H, Br, O, Cl, H, H, H, O], AK1547; H, Cl, H, Br, O, Br, H, H, O], [AK1548; H, Cl, H, Br, O, I, H, H, H, O], [AK1 549; H, Cl, H, Br, O, Me, H, H, H, O], [AK1550; H, Cl, H, Br, O, Et, H, H, H, O], [AK1551; H, Cl, H, Br, O, Pr, H, H, H, O], [AK 1552; H, Cl, H, Br, O, i-Pr, H, H, H, O], [AK 1553; H, Cl, H, Br, O, Bu, H, H, H, O], [AK1554; H, Cl, H, Br, O, i-Bu, H, H, H, O], [AK1 555; H, Cl, H, Br, O, sec-Bu, H, H, H, O], [AK1556; H, Cl, H, Br, O, t-Bu, H, H, H, O], [AK1 557; H, Cl, H, Br, O, c-Pr, H, H, H, O], [AK 1 558; H, Cl, H, Br, O, c-Bu, H, H, H, O] [AK1559; H, Cl, H, Br, O, OBu, H, H, H, O], [AK 1560; H, Cl, H, Br, O, Oi-Bu, H, H, H, O] , [AK1561; H, Cl, H, Br, O, O-sec-Bu, H, H, H, O], [AK1562; H, Cl, H, Br, O, CH 2 F, H, H, H, O], [AK1563; H, Cl, H, Br, O, CHF 2, H, H, H, O], [AK1564; H, Cl, H, Br, O, CF 3, H, H, H, O], [AK1565; H, Cl, H, Br, O, OCH 2 F, H, H, H, O], [AK1566; H, Cl, H, Br, O, OCHF 2, H, H , H, O], [AK1567 ; H, Cl, H, Br, O, OCF 3, H, H, H, O], [AK1568; H, Cl, H, Br, O, OCF 3, H, H , H, O], [AK1569; H, Br, H, H, O, H, H, H, H, O], [AK 1570; H, Br, H, H, O, F, H, H, H] H, Br, H, H, O, Cl, H, H, O], [AK 1572; H, Br, H, H, O, Br, H, H, H, O] H, Br, H, H, O, I, H, H, H, O], [AK1 574; H, Br, H, H, O, Me, H, H, H, O], [AK1575; H, Br, H, H, O, Et, H, H, H, O], [AK1576; H, Br, H, H, O, Pr, H, H, H, O], [AK1577 H, Br, H, H, H, O, i-Pr, H, H, H, O], [AK1578; H, Br, H, H, O, Bu, H, H, H, O], [AK1579] H, Br, H, H, H, O, i-Bu, H, H, H, O], [AK1580; H, Br, H, H, O, sec-Bu, H, H, H, O], [AK 1581; H, Br, H, H, O, t-Bu, H, H, H, O], [AK 1582; H, Br, H, H, O, c-Pr, H, H, H, O H, Br, H, H, O, c-Bu, H, H, H, O], [AK 1584; H, Br, H, H, O, OBu, H, H, H, O] ], [AK1585; H, Br, H, H, O, Oi-Bu, H, H, H, O], [AK1586; H, Br, H, H, O, O-sec-Bu, H, H, H, O], [AK1587; H, Br, H, H, O, CH 2 F, H, H, H, O], [AK1588; H, Br, H, H, O, CHF 2, H, H, H, O], [AK1589 ; H, Br, H, H , O, CF 3, H, H, H, O], [AK1590; H, Br, H, H, O, OCH 2 F, H, H, H, O], [ AK1591; H, Br, H, H, O, OCHF 2, H, H, H, O], [AK1592; H, Br, H, H, O, OCF 3, H, H, H, O], [ AK1593; H, Br, H, Me, O, H, H, H, O], [AK1594; H, Br, H, Me, O, F, H, H, H, O], [AK1595; H, Br, H, Me, O, Cl, H, H, H, O], [AK1596; H, Br, H, Me, O, Br, H, H, H, O], [AK 1597; H, Br, H, Me, O, I, H, H, H, O], [AK 1598; H, Br, H, Me, O, Me, H, H, H, O], [AK 1 599; H, Br, H, Me, O, Et, H, H, H, O], [AK1600; H, Br, H, Me, O, Pr, H, H, H, O],

[AK1601; H, Br, H, Me, O, i-Pr, H, H, H, O], [AK1602; H, Br, H, Me, O, Bu, H, H, H, O], [AK1603; H, Br, H, Me, O, i-Bu, H, H, H, O], [AK1604; H, Br, H, Me, O, sec-Bu, H, H, H, O H, Br, H, Me, O, t-Bu, H, H, H, O], [AK 1606; H, Br, H, Me, O, c-Pr, H, H, H] H, Br, H, Me, O, c-Bu, H, H, H, O], [AK 1608; H, Br, H, Me, O, OBu, H, H, H] H, Br, H, Me, O, Oi-Bu, H, H, H, O], [AK 1610; H, Br, H, Me, O, O-sec-Bu, H] H, H, O], [AK 1611; H, Br, H, Me, O, CH ₂ F, H, H, H, O], [AK 1612; H, Br, H, Me, O, CHF ₂ , H, H, H, O], [AK 1613; H, Br, H, Me, O, CF ₃ , H, H, H, O], [AK 1614; H, Br, H, Me, O, OCH ₂ F , H, H, H, O ], [AK1615; H, Br, H, Me, O, OCHF 2, H, H, H, O], [AK1616; H, Br, H, Me, O, OCF 3 , H, H, H, O ], [AK1617; H, Br, H, Me, O, OCF 3, H, H, H, O], [AK1618; H, Br, H, Et, O, H, H, H, H, O], [AK1619; H, Br, H, Et, O, F, H, H, H, O], [AK 1620; H, Br, H, Et, O, Cl, H, H, H, O], [AK1621; H, Br, H, Et, O, Br, H, H, H, O], [AK1622; H, Br, H, Et, O, I, H, H, H, O], [AK1623; H, Br, H, Et, O, Me, H, H, H, O], [AK1624; H, Br, H, Et, O, Et, H, H, H, H, O, [AK1625; H, Br, H, Et, O, Pr, H, H, H, O], [AK1626; H, Br, H, Et, O, i-Pr, H, H, H, O], [AK1627; H, Br, H, Et, O, Bu, H, H, H, O], [AK1628; H, Br, H, Et, O, i-Bu, H, H, H] H, Br, H, Et, O, sec-Bu, H, H, H, O], [AK 1630; H, Br, H, Et, O, t-Bu, H, H] H, O], [AK1631; H, Br, H, Et, O, c-Pr, H, H, H, O], [AK1632; H, Br, H, Et, O, c-Bu, H H, H, O], [AK1633; H, Br, H, Et, O, OBu, H, H, H, O], [AK1634; H, Br, H, Et, O, Oi-Bu, H H, H, O], [AK 1635; H, Br, H, Et, O, O-sec-Bu, H, H, H, O], [AK 1636; H, Br, H, Et, O, CH _{2 F, H, H, H} , O], [AK1637; H, Br, H, Et, O, CHF 2, H, H, H, O], [AK1638; H, Br, H, Et, O, _{CF 3, H, H, H} , O], [AK1639; H, Br, H, Et, O, OCH 2 F, H, H, H, O], [AK1640; H, Br, H, Et, O _{, OCHF 2, H, H,} H, O], [AK1641; H, Br, H, Et, O, OCF 3, H, H, H, O], [AK1642; H, Br, H, Et, O , OCF ₃ , H, H, H, O], [AK 1643; H, Br, H, Pr, O, H, H, H, H, O], [AK 1644; H, Br, H, Pr, O, F, H, H, H, O], [AK1645; H, Br, H, Pr, O, Cl, H, H, H, O], [AK 1646; H, Br, H, Pr, O, Br, H, H, H, O], [AK1647; H, Br, H, Pr, O, I, H, H, H, O], [AK 1648; H, Br, H, Pr, O, Me, H, H, H, O], [AK1649; H, Br, H, Pr, O, Et, H, H, H, O], [AK1650; H, Br, H, Pr, O, Pr, H, H, H, H, O], [AK1651; H, Br, H, Pr, O, i-Pr, H, H, H, O], [AK1652; H, Br, H, Pr, O, Bu, H, H, H, O], [AK1653; H, Br, H, Pr, O, i-Bu, H, H, H, O], [AK1654; H, Br, H, Pr, O, sec-Bu, H, H, H, O], [AK 1 655; H, Br, H, Pr, O, t-Bu, H, H, H, O], [AK 1 656; H, Br, H, Pr, O, c-Pr, H, H, H, O], [AK1657; H, Br, H, Pr, O, c-Bu, H, H, H, O], [AK1658; H, Br, H, Pr, O, OBu, H, H, H, O], [AK 1659; H, Br, H, Pr, O, Oi-Bu, H, H, H, O], [AK 1660; H, Br, H, Pr, O, O-sec-Bu, H, H, H, O], [AK1661; H, Br, H, Pr, O, CH 2 F, H, H, H, O], [AK1662; H, Br, _{H, Pr, O, CHF 2} , H, H, H, O], [AK1663; H, Br, H, Pr, O, CF 3, H, H, H, O], [AK1664; H, Br, _{H, Pr, O, OCH 2} F, H, H, H, O], [AK1665; H, Br, H, Pr, O, OCHF 2, H, H, H, O], [AK1666; H, Br , H, Pr, O, OCF 3, H, H, H, O], [AK1667; H, Br, H, Pr, O, OCF 3, H, H, H, O], [AK1668; H, Br , H, i-Pr, O, H, H, H, H, O], [AK1669; H, Br, H, i-Pr, O, F, H, H, O], [AK 1670; H , Br, H, i-Pr, O, Cl, H, H, H, O], [AK1671; H, Br, H, i-Pr, O, Br, H, H, H, O], [AK1672 H, Br, H, i-Pr, O, I, H, H, H, O], [AK1673; H, Br, H, i-Pr, O, Me, H, H, H, O], [AK1674; H, Br, H, i-Pr, O, Et, H, H, H, O], [AK1 675; H, Br, H, i-Pr, O, Pr, H, H, H, O H, Br, H, i-Pr, O, i-Pr, H, H, H, O], [AK 1677; H, Br, H, i-Pr, O, Bu, H, H] , H, O], [AK1678; H, Br, H, i-Pr, O, i-Bu, H, H, H, O], [AK1679; H, Br, H, i-Pr, O, sec -Bu, H, H, H, O], [AK1680; H, Br, H, i-Pr, O, t-Bu, H, H, H, O], [AK1681; H, Br, H, i -Pr, O, c-Pr, H, H, H, O], [AK1682; H, Br, H, i-Pr, O, c-Bu, H, H, H, O], [AK 1683; H , Br, H, iP r, O, OBu, H, H, H, O], [AK1684; H, Br, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK1 685; H, Br, H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK1686; H, Br, H, i-Pr, O, CH 2 F, H, H, H, O] , [AK1687; H, Br, H, i-Pr, O, CHF 2, H, H, H, O], [AK1688; H, Br, H, i-Pr, O, CF 3, H, H, H, O], [AK 1689; H, Br, H, i-Pr, O, OCH ₂ F, H, H, H, O], [AK 1690; H, Br, H, i-Pr, O, OCHF ₂ , H, H, H, O ], [AK1691; H, Br, H, i-Pr, O, OCF 3, H, H, H, O], [AK1692; H, Br, H, i-Pr, _{O, OCF 3, H, H} , H, O], [AK1693; H, Br, H, OMe, O, H, H, H, H, O], [AK1694; H, Br, H, OMe, O , F, H, H, H, O], [AK 1695; H, Br, H, OMe, O, Cl, H, H, H, O], [AK 1 696; H, Br, H, OMe, O, Br] H, H, H, O], [AK 1697; H, Br, H, OMe, O, I, H, H, H, O], [AK 1698; H, Br, H, OMe, O, Me, H H, H, O], [AK1699; H, Br, H, OMe, O, Et, H, H, H, O], [AK1700; H, Br, H, OMe, O, Pr, H, H] , H, O],

[AK1701; H, Br, H, OMe, O, i-Pr, H, H, H, O], [AK1702; H, Br, H, OMe, O, Bu, H, H, H, O], [AK1703; H, Br, H, OMe, O, i-Bu, H, H, H, O], [AK1704; H, Br, H, OMe, O, sec-Bu, H, H, H, O H, Br, H, OMe, O, t-Bu, H, H, H, O], [AK 1706; H, Br, H, OMe, O, c-Pr, H, H, H] H, Br, H, OMe, O, c-Bu, H, H, H, O], [AK1 708; H, Br, H, OMe, O, OBu, H, H, H] H, Br, H, OMe, O, Oi-Bu, H, H, H, O], [AK 1710; H, Br, H, OMe, O, O-sec-Bu, H , H, H, O], [AK1711; H, Br, H, OMe, O, CH 2 F, H, H, H, O], [AK1712; H, Br, H, OMe, O, CHF 2, H, H, H, O] , [AK1713; H, Br, H, OMe, O, CF 3, H, H, H, O], [AK1714; H, Br, H, OMe, O, OCH 2 F , H, H, H, O ], [AK1715; H, Br, H, OMe, O, OCHF 2, H, H, H, O], [AK1716; H, Br, H, OMe, O, OCF 3 , H, H, H, O ], [AK1717; H, Br, H, OMe, O, OCF 3, H, H, H, O], [AK1718; H, Br, H, F, O, H, H, H, H, O], [AK1719; H, Br, H, F, O, F, H, H, H, O], [AK1720; H, Br, H, F, O, Cl, H, H, H, O], [AK1721; H, Br, H, F, O, Br, H, H, H, O], [AK1722; H, Br, H, F, O, I, H, H, H, O], [AK1723; H, Br, H, F, O, Me, H, H, H, O], [AK1724; H, Br, H, F, O, Et, H, H, H, H, O, [AK1725; H, Br, H, F, O, Pr, H, H, H, O], [AK1726; H, Br, H, F, O, i-Pr, H, H, H, O], [AK1727; H, Br, H, F, O, Bu, H, H, H, O], [AK1728; H, Br, H, F, O, i-Bu H, H, H, O], [AK1729; H, Br, H, F, O, sec-Bu, H, H, H, O], [AK1730; H, Br, H, F, O, t -Bu, H, H, H, O], [AK1731; H, Br, H, F, O, c-Pr, H, H, H, O], [AK 1732; H, Br, H, F, O , c-Bu, H, H, H, O], [AK1733; H, Br, H, F, O, OBu, H, H, H, O], [AK 1734; H, Br, H, F, O] , Oi-Bu, H, H, H, O], [AK1735; H, Br, H, F, O, O-sec-Bu, H, H, H, O], [AK1736; H, Br, H] _{, F, O, CH 2 F} , H, H, H, O], [AK1737; H, Br, H, F, O, CHF 2, H, H, H, O], [AK1738; H, Br, _{H, F, O, CF 3} , H, H, H, O], [AK1739; H, Br, H, F, O, OCH 2 F, H, H, H, O], [AK1740; H, Br , H, F, O, OCHF 2, H, H, H, O], [AK1741; H, Br, H, F, O, OCF 3, H, H, H, O], [AK1742; H, Br , H, F, O, OCF 3, H, H, H, O], [AK1743; H, Br, H, Cl, O, H, H, H, H, O], [AK1744; H, Br, H, Cl, O, F, H, H, H, O], [AK1 745; H, Br, H, Cl, O, Cl, H, H, H, O], [AK1 746; H, Br, H, Cl, O, Br, H, H, H, O, [AK1747; H, Br, H, Cl, O, I, H, H, H, O], [AK1 748; H, Br, H, Cl, O, Me, H, H, H, O], [AK 1749; H, Br, H, Cl, O, Et, H, H, H, O], [AK 1 750; H, Br, H, Cl, O, Pr, H, H, H, O], [AK1751; H, Br, H, Cl, O, i-Pr, H, H, H, O], [AK1752; H, Br, H, Cl, O, Bu, H, H, H, O], [AK1753; H, Br, H, Cl, O, i-Bu, H, H, H, O], [AK 1754; H, Br, H, Cl, O, sec-Bu, H, H, H, O], [AK1 755; H, Br, H, Cl, O, t-Bu, H, H, H, O], [AK1 756; H, Br, H, Cl, O, c-Pr, H, H , H, O], [AK1757; H, Br, H, Cl, O, c-Bu, H, H, H, O], [AK 1758; H, Br, H, Cl, O, OBu, H, H H, O], [AK 1759; H, Br, H, Cl, O, Oi-Bu, H, H, H, O], [AK 1760; H, Br, H, Cl, O, O-sec-Bu , H, H, H, O ], [AK1761; H, Br, H, Cl, O, CH 2 F, H, H, H, O], [AK1762; H, Br, H, Cl, O, CHF _{2, H, H, H,} O], [AK1763; H, Br, H, Cl, O, CF 3, H, H, H, O], [AK1764; H, Br, H, Cl, O, OCH ₂ F, H, H, H, O], [AK 1 765; H, Br, H, Cl, O, OCHF ₂ , H, H, H, O], [AK 1 766; H, Br, H, Cl, O, OCF ₃ , H, H, H, O], [AK 1767; H, Br, H, Cl, O, OCF ₃ , H, H, H, O], [AK 1768; H, Br, H, Br, O, H, H, H, H, O], [AK 1769; H, Br, H, Br, O, F, H, H, H, O], [AK 1 770; H, Br, H, Br, O, Cl, H, H, H, O], [AK1771; H, Br, H, Br, O, Br, H, H, H, O], [AK1772; H, Br, H, Br, O, I, H, H, H, O], [AK1773; H, Br, H, Br, O, Me, H, H, H, O], [AK1 774; H, Br, H, Br, O, Et, H, H, H, H, O], [AK1 775; H, Br, H, Br, O, Pr, H, H, H, O], [AK1 776; H, Br, H, Br, O, i-Pr, H, H, H, O], [AK 1 777; H, Br, H, Br, O, Bu, H, H, H, O], [AK 1778; H, Br, H, Br, O, i-Bu, H, H, H, O], [AK1779; H, Br, H, Br, O, sec-Bu, H, H, H, O], [AK1 780; H, Br, H, Br, O, t-Bu, H, H, H, O], [AK1781; H, Br, H, Br, O, c-Pr, H, H, H, O], [AK1782; H, Br, H, Br, O, c-Bu, H, H, H, O], [AK1783; H, Br, H, Br, O, OBu, H, H, H, O], [AK1784; H, Br, H, Br, O, O i-Bu, H, H, H, O], [AK1 785; H, Br, H, Br, O, O-sec-Bu, H, H, H, O], [AK1 786; H, Br, H, _{Br, O, CH 2 F,} H, H, H, O], [AK1787; H, Br, H, Br, O, CHF 2, H, H, H, O], [AK1788; H, Br, H _{, Br, O, CF 3,} H, H, H, O], [AK1789; H, Br, H, Br, O, OCH 2 F, H, H, H, O], [AK1790; H, Br, _{H, Br, O, OCHF 2} , H, H, H, O], [AK1791; H, Br, H, Br, O, OCF 3, H, H, H, O], [AK1792; H, Br, _{H, Br, O, OCF 3} , H, H, H, O], [AK1793; H, OMe, H, H, O, H, H, H, H, O], [AK1794; H, OMe, H , H, O, F, H, H, H, O], [AK 1795; H, OMe, H, H, O, Cl, H, H, H, O], [AK 1796; H, OMe, H, H] , O, Br, H, H, H, O], [AK1 797; H, OMe, H, H, O, I, H, H, H, O], [AK 1798; H, OMe, H, H, O] , Me, H, H, H, O], [AK1799; H, OMe, H, H, O, Et, H, H, H, O], [AK1800; H, OMe, H, H, O, Pr , H, H, H, O],

[AK1801; H, OMe, H, H, O, i-Pr, H, H, H, O], [AK1802; H, OMe, H, H, O, Bu, H, H, H, O], [AK1803; H, OMe, H, H, O, i-Bu, H, H, H, O], [AK1804; H, OMe, H, H, O, sec-Bu, H, H, H, O , [AK1805; H, OMe, H, H, O, t-Bu, H, H, H, O], [AK 1806; H, OMe, H, H, O, c-Pr, H, H, H] H, OMe, H, H, O, c-Bu, H, H, H, O], [AK 1808; H, OMe, H, H, O, OBu, H, H, H] H, OMe, H, H, O, Oi-Bu, H, H, H, O], [AK 1810; H, OMe, H, H, O, O-sec-Bu, H] H, H, O], [AK 1811; H, OMe, H, H, O, CH ₂ F, H, H, H, O], [AK 1812; H, OMe, H, H, O, CHF ₂ , H, H, H, O], [AK 1813; H, OMe, H, H, O, CF ₃ , H, H, H, O], [AK 1814; H, OMe, H, H, O, OCH ₂ F , H, H, H, O ], [AK1815; H, OMe, H, H, O, OCHF 2, H, H, H, O], [AK1816; H, OMe, H, H, O, OCF 3 , H, H, H, O], [AK1817; H, OMe, H, Me, O, H, H, H, H, O], [AK1818; H, OMe, H, Me, O, F, H] H, H, O], [AK1819; H, OMe, H, Me, O, Cl, H, H, H, O], [AK1820; H, OMe, H, Me, O, Br, H, H] H, O], [AK1821; H, OMe, H, Me, O, I, H, H, H, O], [AK1822; H, OMe, H, Me, O, Me, H, H, H] , O], [AK1823; H, OMe, H, Me, O, Et, H, H, H, O], [AK1824; H, OMe, H, Me, O, Pr, H, H, H, O H, OMe, H, Me, O, i-Pr, H, H, H, O], [AK 1826; H, OMe, H, Me, O, Bu, H, H, H, O] H, OMe, H, Me, O, i-Bu, H, H, H, O], [AK1 828; H, OMe, H, Me, O, sec-Bu, H, H, H, O], [AK 1829; H, OMe, H, Me, O, t-Bu, H, H, H, O], [AK 1830; H, OMe, H, Me, O, c-Pr, H, H, H, O], [AK 1831; H, OMe, H, Me, O, c-Bu, H, H, H, O], [AK 1832; H, OMe, H, Me, O, OBu, H, H, H, O], [AK1833; H, OMe, H, Me, O, Oi-Bu, H, H, H, O], [AK1834; H, OMe, H, O Me, O, O-sec- Bu, H, H, H, O], [AK1835; H, OMe, H, Me, O, CH 2 F, H, H, H, O], [AK1836; H, OMe, H, Me, O, CHF 2, H, H, H, O], [AK1837; H, OMe, H, Me, O, CF 3, H, H, H, O], [AK1838; H, OMe, H, Me, O, OCH 2 F, H, H, H, O], [AK1839; H, OMe, H, Me, O, OCHF 2, H, H, H, O], [AK1840; H , OMe, H, Me, O , OCF 3, H, H, H, O], [AK1841; H, OMe, H, Me, O, OCF 3, H, H, H, O], [AK1842; H , OMe, H, Et, O, H, H, H, H, O], [AK1843; H, OMe, H, Et, O, F, H, H, H, O], [AK 1844; H, OMe , H, Et, O, Cl, H, H, H, O], [AK 1845; H, OMe, H, Et, O, Br, H, H, H, O], [AK 1846; H, OMe, H , Et, O, I, H, H, H, O], [AK1 847; H, OMe, H, Et, O, Me, H, H, H, O], [AK1848; H, OMe, H, Et] , O, Et, H, H, H, O], [AK 1849; H, OMe, H, Et, O, Pr, H, H, H, O], [AK 1850; H, OMe, H, Et, O , i-Pr, H, H, H, O], [AK 1851; H, OMe, H, Et, O, Bu, H, H, H, O], [AK 1852; H, OMe, H, Et, O , i-Bu, H, H, H, O], [AK 1853; H, OMe, H, Et, O, sec-Bu, H, H, H, O], [AK 1 854; H, OMe, H, Et , O, t-Bu, H, H, H, O], [AK 1855; H, OMe, H, Et, O , c-Pr, H, H, H, O], [AK 1856; H, OMe, H, Et, O, c-Bu, H, H, H, O], [AK 1 857; H, OMe, H, Et , O, OBu, H, H, H, O], [AK 1858; H, OMe, H, Et, O, Oi-Bu, H, H, H, O], [AK 1859; H, OMe, H, Et , O, O-sec-Bu , H, H, H, O], [AK1860; H, OMe, H, Et, O, CH 2 F, H, H, H, O], [AK1861; H, OMe , H, Et, O, CHF 2, H, H, H, O], [AK1862; H, OMe, H, Et, O, CF 3, H, H, H, O], [AK1863; H, OMe , H, Et, O, OCH ₂ F, H, H, H, O], [AK 1864; H, OMe, H, Et, O, OCHF ₂ , H, H, H, O], [AK 1865; H, OMe, H, Et, O, OCF 3, H, H, H, O], [AK1866; H, OMe, H, Et, O, OCF 3, H, H, H, O], [AK1867; H, OMe, H, Pr, O, H, H, H, H, O], [AK1868; H, OMe, H, Pr, O, F, H, H, H, O], [AK1869; H, OMe, H, Pr, O, Cl, H, H, H, O], [AK 1 870; H, OMe, H, Pr, O, Br, H, H, H, O], [AK 1871; H, OMe, H, Pr, O, I, H, H, H, O], [AK1872; H, OMe, H, Pr, O, Me, H, H, H, O], [AK1 873; H, OMe, H, Pr, O, Et, H, H, H, O], [AK 1874; H, OMe, H, Pr, O, Pr, H, H, H, O], [AK 1875; H, OMe, H, Pr, O, i-Pr, H, H, H, O], [AK 1876; H, OMe, H, Pr, O, Bu, H, H, H, O], [AK 1877; H, OMe, H, Pr, O, i-Bu, H, H, H, O], [AK1 878; H, OMe, H, Pr, O, sec-Bu, H, H, H, O], [AK 1879; H, OMe, H, Pr, O, t-Bu, H, H, H, O], [AK1 880; H, OMe, H, Pr, O, c-Pr, H, H, H, O], [AK1881; H, OMe, H, Pr, O, c-Bu, H, H, H, O], [AK1882; H, OMe, H, Pr, O, OBu, H, H, H, O], [AK 1883; H, OMe, H, Pr, O, Oi-Bu, H, H, H, O], [AK 1 884; H, OMe, H, Pr, O, O-sec-Bu, H, H, H, O], [AK1885; H, OMe, H, Pr, O, CH 2 F, H, H, H, O], [AK1886; H, OMe, H, _{Pr, O, CHF 2, H} , H, H, O], [AK1887; H, OMe, H, Pr, O, CF 3, H, H, H, O], [AK1888; H, OMe, H, Pr, O, OCH ₂ F, H, H, H, O], [AK 1889; H, OMe, H, Pr, O, OCHF ₂ , H, H, H, O], [AK 1890; H, OMe, H _{, Pr, O, OCF 3,} H, H, H, O], [AK1891; H, OMe, H, Pr, O, OCF 3, H, H, H, O], [AK1892; H, OMe, H , i-Pr, O, H, H, H, H, O], [AK 1893; H, OMe, H, i-Pr, O, F, H, H, O], [AK 1894; H, OMe , H, i-Pr, O, Cl, H, H, H, O], [AK 1895; H, OMe, H, i-Pr, O, Br, H, H, H, O], [AK 1896; H , OMe, H, i-Pr, O, I, H, H, H, O], [AK 1897; H, OMe, H, i-Pr, O, Me, H, H, H, O], [AK 1898 H, OMe, H, i-Pr, O, Et, H, H, H, O], [AK1899; H, OMe, H, i-Pr, O, Pr, H, H, H, O], [AK1900; H, OMe, H, i-Pr, O, i-Pr, H, H, H, O],

[AK1901; H, OMe, H, i-Pr, O, Bu, H, H, H, O], [AK1902; H, OMe, H, i-Pr, O, i-Bu, H, H, H , O], [AK 1903; H, OMe, H, i-Pr, O, sec-Bu, H, H, H, O], [AK 1904; H, OMe, H, i-Pr, O, t-Bu H, H, H, O], [AK 1905; H, OMe, H, i-Pr, O, c-Pr, H, H, H, O], [AK 1906; H, OMe, H, i-Pr , O, c-Bu, H, H, H, O], [AK 1 907; H, OMe, H, i-Pr, O, OBu, H, H, H, O], [AK 1908; H, OMe, H] , i-Pr, O, Oi-Bu, H, H, H, O], [AK 1909; H, OMe, H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK 1910; H, OMe, H, i-Pr, O, CH ₂ F, H, H, H, O], [AK 1911; H, OMe, H, i-Pr, O, CHF ₂ , H, H, H, O], [AK1912; H, OMe, H, i-Pr, O, CF 3, H, H, H, O], [AK1913; H, OMe, H, i-Pr, O, OCH 2 F , H, H, H, O ], [AK1914; H, OMe, H, i-Pr, O, OCHF 2, H, H, H, O], [AK1915; H, OMe, H, i-Pr, _{O, OCF 3, H, H} , H, O], [AK1916; H, OMe, H, i-Pr, O, OCF 3, H, H, H, O], [AK1917; H, OMe, H, OMe, O, H, H, H, H, O], [AK1918; H, OMe, H, OMe, O, F, H, H, H, O], [AK1919; H, OMe, H, OMe, O, Cl, H, H, H, O], [AK 1920; H, OMe, H, OMe, O, Br, H, H, H, O], [AK1921; H, OMe, H, OMe, O, H, OMe, H, OMe, O, Me, H, H, H, O], [AK 1 923; H, OMe, H, OMe, O, Et, I, H, H, H, O], [AK 1 922; H, H, H, O], [AK 1 924; H, OMe, H, OMe, O, Pr, H, H, H, O], [AK 1 925; H, OMe, H, OMe, O, i-Pr, H, H, H, O], [AK 1926; H, OMe, H, OMe, O, Bu, H, H, H, O] [AK1 927; H, OMe, H, OMe, O, i-Bu, H, H, H, O], [AK 1 928; H, OMe, H, OMe, O, sec-Bu, H, H, H, O H, OMe, H, OMe, O, t-Bu, H, H, H, O], [AK1 930; H, OMe, H, OMe, O, c-Pr, H, H, H] , O], [AK1931; H, OMe, H, OMe, O, c-Bu, H, H, H, O], [AK1932; H, OMe, H, OMe, O, OBu, H, H, H] , O], [AK1933; H, OMe, H, OMe, O, Oi-Bu, H, H, H, O], [AK1 934; H, OMe, H, OMe, O, O-sec-Bu, H H, H, O], [AK 1935; H, OMe, H, OMe, O, CH ₂ F, H, H, H, O], [AK 1936; H, OMe, H, OMe, O, CHF ₂ , H, H, H, O] , [AK1937; H, OMe, H, OMe, O, CF 3, H, H, H, O], [AK1938; H, OMe, H, OMe, O, OCH 2 F H, H, H, O], [AK 1939; H, OMe, H, OMe, O, OCHF ₂ , H, H, H, O], [AK 1940; H, OMe, H, OMe, O, OCF ₃ , H, H, H, O ], [AK1941; H, OMe, H, OMe, O, OCF 3, H, H, H, O], [AK1942; H, OMe, H, F, O, H, H, H, H, O], [AK1943; H, OMe, H, F, O, F, H, H, H, O], [AK1 944; H, OMe, H, F, O, Cl, H, H, H, O], [AK 1 945; H, OMe, H, F, O, Br, H, H, H, O], [AK 1946; H, OMe, H, F, O, I, H, H, H, O], [AK 1947; H, OMe, H, F, O, Me, H, H, H, O], [AK 1948; H, OMe, H, F, O, Et, H, H, H, O], [AK1 949; H, OMe, H, F, O, Pr, H, H, H, O], [AK 1950; H, OMe, H, F, O, i-Pr, H, H, H, O], [AK1951; H, OMe, H, F, O, Bu, H, H, H, O], [AK1952; H, OMe, H, F, O, i-Bu, H, H, H, O], [AK1953; H, OMe, H, F, O, sec-Bu, H, H, H , O], [AK1954; H, OMe, H, F, O, t-Bu, H, H, H, O], [AK 1 955; H, OMe, H, F, O, c-Pr, H, H , H, O], [AK1956; H, OMe, H, F, O, c-Bu, H, H, H, O], [AK 1957; H, OMe, H, F, O, OBu, H, H H, O], [AK 1958; H, OMe, H, F, O, Oi-Bu, H, H, H, O], [AK1959; H, OMe, H, F, O, O-sec-Bu , H, H, H, O], [AK1960; H, OMe, H, F, O, CH ₂ F, H, H, H, O], [AK 1961; H, OMe, H, F, O, CHF _{2, H, H, H,} O], [AK1962; H, OMe, H, F, O, CF 3, H, H, H, O], [AK1963; H, OMe, H, F, O, OCH ₂ F, H, H, H, O], [AK 1964; H, OMe, H, F, O, OCHF ₂ , H, H, H, O], [AK 1 965; H, OMe, H, F, O, _{OCF 3, H, H, H} , O], [AK1966; H, OMe, H, F, O, OCF 3, H, H, H, O], [AK1967; H, OMe, H, Cl, O, H, H, H, H, O], [AK 1968; H, OMe, H, Cl, O, F, H, H, H, O], [AK 1969; H, OMe, H, Cl, O, Cl, H, H, H, O], [AK1970; H, OMe, H, Cl, O, Br, H, H, H, O], [AK 1971; H, OMe, H, Cl, O, I, H, H, H, O], [AK 1972; H, OMe, H, Cl, O, Me, H, H, H, O], [AK 1973; H, OMe, H, Cl, O, Et, H, H, H, O], [AK 1974; H, OMe, H, Cl, O, Pr, H, H, H, O], [AK1975; H, OMe, H, Cl, O, i-Pr, H, H, H, O], [AK1976; H, OMe, H, Cl, O, Bu, H, H, H, O], [AK1977; H, OMe, H, Cl, O, i-Bu, H, H, H, O], [AK1978; H, OMe, H, Cl, O, sec-Bu, H, H, H, O], [AK 1979; H, OMe, H, Cl, O, t-Bu, H, H, H, O], [AK1980; H, OMe, H, Cl, O, c-Pr, H, H, H, O], [AK1981; H, OMe, H, Cl, O, c-Bu, H, H, H, O], [AK1982; H, OMe, H, Cl, O, OBu, H, H, H, O], [AK1983; H, OMe, H, Cl, O, Oi-Bu, H, H, H, O], [AK1984; H, OMe, H, Cl, O, O-sec-Bu, H, H, H, O] , [AK1985; H, OMe, H, Cl, O, CH 2 F, H, H, H, O], [AK1986; H, OMe, H, Cl, O, CHF 2, H, H, H, O ], [AK1987; H, OMe , H, Cl, O, CF 3, H, H, H, O], [AK1988; H, OMe, H, Cl, O, OCH 2 F, H, H, H, O], [AK1989; H, OMe, H, Cl, O, OCHF 2, H, H, H, O], [AK1990; H, OMe, H, Cl, O, OCF 3, H, H, H, O], [AK1991; H, OMe, H, Cl, O, OCF 3, H, H, H, O], [AK1992; H, OMe, H, Br, O, H, H, H, H, O ], [AK1993; H, OMe, H, Br, O, F, H, H, O], [AK1994; H, OMe, H, Br, O, Cl, H, H, H, O], [AK1995; H, OMe, H, Br, O, Br, H, H, H, O], [AK1996; H, OMe, H, Br, O, I, H, H, H, O], [AK1997 H, OMe, H, Br, O, Me, H, H, H, O], [AK1998; H, OMe, H, Br, O, Et, H, H, H, O], [AK1999; H , OMe, H, Br, O, Pr, H, H, H, O], [AK 2000; H, OMe, H, Br, O, i-Pr, H, H, H, O],

[AK2001; H, OMe, H, Br, O, Bu, H, H, H, O], [AK2002; H, OMe, H, Br, O, i-Bu, H, H, H, O], [AK2003; H, OMe, H, Br, O, sec-Bu, H, H, H, O], [AK2004; H, OMe, H, Br, O, t-Bu, H, H, H, O ], [AK2005; H, OMe, H, Br, O, c-Pr, H, H, H, O], [AK2006; H, OMe, H, Br, O, c-Bu, H, H, H] , O], [AK2007; H, OMe, H, Br, O, OBu, H, H, H, O], [AK2008; H, OMe, H, Br, O, Oi-Bu, H, H, H] , O], [AK2009; H, OMe, H, Br, O, O-sec-Bu, H, H, H, O], [AK2010; H, OMe, H, Br, O, CH ₂ F, H , H, H, O], [AK2011; H, OMe, H, Br, O, CHF 2, H, H, H, O], [AK2012; H, OMe, H, Br, O, CF 3, H , H, H, O], [AK 2013; H, OMe, H, Br, O, OCH ₂ F, H, H, H, O], [AK 2014; H, OMe, H, Br, O, OCHF ₂ , H, H, H, O] , [AK2015; H, OMe, H, Br, O, OCF 3, H, H, H, O], [AK2016; H, OMe, H, Br, O, OCF 3, H, H, H, O], [AK 2017; H, OEt, H, H, O, H, H, H, H, O], [AK 2018; H, OE t, H, H, O, F, H, H, H, O], [AK 2019; H, OEt, H, H, O, Cl, H, H, H, O], [AK 2020; H, OE t, H, H, O, Br, H, H, H, O], [AK2021; H, OEt, H, H, O, I, H, H, H, O], [AK2022; H, OEt, H, H, O, Me, H, H, H, H, O], [AK2023; H, OEt, H, H, O, Et, H, H, H, O], [AK2024; H, OEt, H, H, O, Pr, H, H, H, O] [AK 2025; H, OEt, H, H, H, O, i-Pr, H, H, H, O], [AK 2026; H, OEt, H, H, O, Bu, H, H, H, O] [AK2027; H, OEt, H, H, O, i-Bu, H, H, H, O], [AK2028; H, OEt, H, H, O, sec-Bu, H, H, H, O], [AK 2029; H, OEt, H, H, O, t-Bu, H, H, H, O], [AK 2030; H, OEt, H, H, H, O, c-Pr, H, H, H, O], [AK2031; H, OEt, H, H, O, c-Bu, H, H, H, O], [AK2032; H, OEt, H, H, O, OBu, H, H, H, O], [AK2033; H, OEt, H, H, O, Oi-Bu, H, H, H, O], [AK2034; H, OEt, H, H, O, O-sec-Bu, H, H, H, O], [AK2035; H, OEt, H, H, O, CH 2 F, H, H, H, O] , [AK2036; H, OEt, H, H, O, CHF 2, H, H, H, O], [AK2037; H, OEt, H, H, O, CF 3, H, H, H, O] , [AK2038; H, OEt, H, H, O, OCH 2 F, H, H, H, O], [AK2039; H, OEt, H, H, O, OCHF 2, H, H, H, O ], [AK2040; H, OEt , H, H, O, OCF 3, H, H, H, O], [AK2041; H, OEt, H, Me, O, H, H, H, H, O] [AK2042; H, OEt, H, Me, O, F, H, H, O], [AK2043; H, OEt, H, Me, O, Cl, H, H, H, O], [AK 2043; AK2044; H, OEt, H, Me, O, Br, H, H, O], [AK 2045; H, OEt, H, Me, O, I, H, H, H, O], [AK2046; H, OEt, H, Me, O, Me, H, H, H, O], [AK 2047; H, OEt, H, Me, O, Et, H, H, H, O], [AK 2048; H, OEt, H, Me, O, Pr, H, H, H, O], [AK 2049; H, OEt, H, Me, O, i-Pr, H, H, H, O], [AK 2050; H, OEt, H, Me, O, Bu, H, H, H, O], [AK2051; H, OEt, H, Me, O, i-Bu, H, H, H, O], [AK2052; H, OEt, H, Me, O, sec-Bu, H, H, H, O], [AK2053; H, OEt, H, Me, O, t-Bu, H, H, H, O], [AK2054; H, OEt, H, Me, O, c-Pr, H, H, H, O], [AK2055; H, OEt, H, Me, O, c-Bu, H, H, H, O], [AK2056; H, OEt, H, Me, O, OBu, H, H, H, O], [AK 2057; H, OEt, H, Me, O, Oi-Bu, H, H, H, O], [AK2058; H, OEt, H, Me, O, O-sec-Bu, H, H, H, O], [AK 2059; H, OEt, H, Me, O, CH ₂ F, H, H, H, O], [AK2060; H, OEt, H, Me, O, CHF 2, H, H, H, O], [AK2061; H, OEt, H, Me, O, CF _{3, H, H, H,} O], [AK2062; H, OEt, H, Me, O, OCH 2 F, H, H, H, O], [AK2063; H, OEt, H, Me, O, _{OCHF 2, H, H, H} , O], [AK2064; H, OEt, H, Me, O, OCF 3, H, H, H, O], [AK2065; H, OEt, H, Me, O, _{OCF 3, H, H, H} , O], [AK2066; H, OEt, H, Et, O, H, H, H, H, O], [AK2067; H, OEt, H, Et, O, F , H, H, H, O], [AK 2068; H, OEt, H, Et, O, Cl, H, H, H, O], [AK 2069; H, OEt, H, Et, O, Br, H , H, H, O], [AK2070; H, OEt, H, Et, O, I, H, H, H, O], [AK2071; H, OEt, H, Et, O, Me, H, H] H, O], [AK2072; H, OEt, H, Et, O, Et, H, H, H, O], [AK 2073; H, OEt, H, Et, O, Pr, H, H, H] H, OEt, H, Et, O, i-Pr, H, H, H, O], [AK 2075; H, OEt, H, Et, O, Bu, H, H, H] , O], [AK 2076; H, OEt, H, Et, O, i, Bu, H, H, H, O], [AK 2077; H, OEt, H, Et, O, sec-Bu, H, H , H, O], [AK 2078; H, OEt, H, Et, O, t-Bu, H, H, H, O], [AK 2079; H, OE t, H, Et, O, c-Pr, H H, H, O], [AK2080; H, OEt, H, Et, O, c-Bu, H, H, H, O], [AK2081; H, OEt, H, Et, O, OBu, H] , H, H, O], [AK2082; H, OEt, H, Et, O, Oi-Bu, H, H H, O], [AK 2083; H, OEt, H, Et, O, O-sec-Bu, H, H, H, O], [AK 2084; H, OE t, H, Et, O, CH ₂ F , H, H, H, O], [AK 2085; H, OEt, H, Et, O, CHF ₂ , H, H, H, O], [AK 2086; H, OE t, H, Et, O, CF ₃ , H, H, H, O], [AK 2087; H, OEt, H, Et, O, OCH ₂ F, H, H, H, O], [AK 2088; H, OE t, H, Et, O, OCHF _{2, H, H, H,} O], [AK2089; H, OEt, H, Et, O, OCF 3, H, H, H, O], [AK2090; H, OEt, H, Et, O, OCF ₃ , H, H, H, O], [AK2091; H, OEt, H, Pr, O, H, H, H, H, O], [AK2092; H, OEt, H, Pr, O, F, H, H, H, O], [AK 2093; H, OEt, H, Pr, O, Cl, H, H, H, O], [AK 2094; H, OE t, H, Pr, O, Br, H, H, H, O], [AK 2095; H, OEt, H, Pr, O, I, H, H, H, O], [AK 2096; H, OE t, H, Pr, O, Me, H, H, H, O], [AK 2097; H, OEt, H, Pr, O, Et, H, H, H, O], [AK 2098; H, OE t, H, Pr, O, Pr, H, H, H, O], [AK 2099; H, OEt, H, Pr, O, i-Pr, H, H, H, O], [AK 2 100; H, OEt, H, Pr, O, Bu, H, H, H, O],

[AK2101; H, OEt, H, Pr, O, i-Bu, H, H, H, O], [AK2 102; H, OEt, H, Pr, O, sec-Bu, H, H, H, O H, OEt, H, Pr, O, t-Bu, H, H, H, O], [AK 2104; H, OEt, H, Pr, O, c-Pr, H, H, H] H, OEt, H, Pr, O, c-Bu, H, H, H, O], [AK 2106; H, OEt, H, Pr, O, OBu, H, H, H] , O], [AK 2107; H, OEt, H, Pr, O, Oi-Bu, H, H, H, O], [AK 2108; H, OEt, H, Pr, O, O-sec-Bu, H H, H, O], [AK 2109; H, OEt, H, Pr, O, CH ₂ F, H, H, H, O], [AK 2 110; H, OEt, H, Pr, O, CHF ₂ , H, H, H, O] , [AK2111; H, OEt, H, Pr, O, CF 3, H, H, H, O], [AK2112; H, OEt, H, Pr, O, OCH 2 F H, H, H, O], [AK 2 113; H, OEt, H, Pr, O, OCHF ₂ , H, H, H, O], [AK 2 114; H, OE t, H, Pr, O, OCF ₃ , H, H, H, O ], [AK2115; H, OEt, H, Pr, O, OCF 3, H, H, H, O], [AK2116; H, OEt, H, i-Pr, O, H, H, H, H, O], [AK 2 117; H, OEt, H, i-Pr, O, F, H, H, H, O], [AK 2 118; H, OE t, H, i-Pr, O, Cl, H, H, H, O], [AK 2119; H, OEt, H, i-Pr, O, Br, H, H, H, O], [AK 2 120; H, OEt, H, i- Pr, O, I, H, H, H, O], [AK2121; H, OEt, H, i-Pr, O, Me, H, H, H, O], [AK 2122; H, OEt, H, i-Pr, O, Et, H, H, H, O], [AK 2 123; H, OEt, H, i-Pr, O, Pr, H, H, H, O], [AK 2 124; H, OE t, H, i-Pr, O, i-Pr, H, H, H, O], [AK 2 125; H, OEt, H, i-Pr, O, Bu, H, H, H, O], [AK 2 126; H, OEt, H, i-Pr, O, i-Bu, H, H, H, O], [AK2127; H, OEt, H, i-Pr, O, sec-Bu, H, H, H, O], [AK 2 128; H, OEt, H, i-Pr, O, t-Bu, H, H, H, O], [AK 2 129; H, OEt, H, i-Pr, O, c-Pr, H, H, H, O], [AK 2130; H, OEt, H, i-Pr, O, c-Bu, H, H, H, O], [AK2131; H, OEt, H, i-Pr, O, OBu, H, H, H, O], [AK2132; H, OEt, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK 2133; H, OEt, H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK 2 134; H, OE t, H, i-Pr, _{O, CH 2 F, H,} H, H, O], [AK2135; H, OEt, H, i-Pr, O, CHF 2, H, H, H, O], [AK2136; H, OEt, H , i-Pr, O, CF 3, H, H, H, O], [AK2137; H, OEt, H, i-Pr, O, OCH 2 F, H, H, H, O], [AK2138; H, OEt, H, i- Pr, O, OCHF 2, H, H, H, O], [AK2139; H, OEt, H, i-Pr, O, OCF 3, H, H, H, O] , [AK2140; H, OEt, H, i-Pr, O, OCF 3, H, H, H, O], [AK2141; H, OEt, H, OMe, O, H, H, H, H, O H, OEt, H, OMe, O, F, H, H, O], [AK 2143; H, OEt, H, OMe, O, Cl, H, H, H, O], [AK2144; H, OEt, H, OMe, O, Br, H, H, H, O], [AK2145; H, OEt, H, OMe, O, I, H, H, H, O], [AK2146 H, OEt, H, OMe, O, Me, H, H, H, O], [AK 2147; H, OEt, H, OMe, O, Et, H, H, H, O], [AK 2 148; H , OEt, H, OMe, O, Pr, H, H, H, O], [AK 2149; H, OEt, H, OMe, O, i-Pr, H, H, H, O], [AK 2 150; H , OEt, H, OMe, O, Bu, H, H, H, O], [AK2151; H, OEt, H, OMe, O, i-Bu, H, H, H, O], [AK2152; H , OEt, H, OMe, O, sec-Bu, H, H, H, O], [AK2153; H, OE t, H, OMe, O, t-Bu, H, H, H, O], [AK 2154; H, OE t, H, OMe, O, c-Pr, H, H, H, O], [AK 2 155; H, OEt, H, OMe, O, c-Bu, H, H, H, O], [AK 2156; H, OEt, H, OMe, O, OBu, H, H, H, O], [AK 2 157; H, OEt, H, OMe, O, Oi-Bu, H, H, H, O], [AK 2158; H, OEt, H, OMe, O, O-sec-Bu, H, H, H, O] , [AK2159; H, OEt, H, OMe, O, CH 2 F, H, H, H, O], [AK2160; H, OEt, H, OMe, O, CHF 2, H, H, H, O ], [AK2161; H, OEt , H, OMe, O, CF 3, H, H, H, O], [AK2162; H, OEt, H, OMe, O, OCH 2 F, H, H, H, O], [AK2163; H, OEt, H, OMe, O, OCHF 2, H, H, H, O], [AK2164; H, OEt, H, OMe, O, OCF 3, H, H, H, O], [AK2165; H, OEt, H, OMe, O, OCF 3, H, H, H, O], [AK2166; H, OEt, H, F, O, H, H, H, H, O H, OEt, H, F, O, F, H, H, O], [AK 2 168; H, OEt, H, F, O, Cl, H, H, H, O], [AK2169; H, OEt, H, F, O, Br, H, H, H, O], [AK 2170; H, OEt, H, F, O, I, H, H, H, O], [AK2171 H, OEt, H, F, O, Me, H, H, H, O], [AK2172; H, OEt, H, F, O, Et, H, H, H, O], [AK 2173; H , OEt, H, F, O, Pr, H, H, H, O], [AK 2174; H, OEt, H, F, O, i-Pr, H, H, H, O], [AK 2 175; H , OEt, H, F, O, Bu, H, H, H, O], [AK 2176; H, OEt, H, F, O, i-Bu, H, H, H, O], [AK 2177; H , OEt, H, F, O, sec-Bu, H, H, H, O], [AK2178; H, OEt, H, F, O, t-Bu, H, H, H, O], [AK2179 H, OEt, H, F, O, c-Pr, H, H, H, O], [AK2180; H, OEt, H, F, O, c-Bu, H, H, H, O, [AK2181; H, OEt, H, F, O, OBu, H, H, H, O], [AK2182; H, OEt, H, F, O, Oi-Bu, H, H, H, O], [AK 2183; H, OEt, H, F, O, O-sec-Bu, H, H, H, O], [AK 2 184; H, OEt, H, F, O, CH 2 F, H, H, H, O], [AK2185; H, OEt, H, F, O, CHF 2, H, H, H, O], [AK2186 H, OEt, H, F, O, CF ₃ , H, H, H, O], [AK 2187; H, OEt, H, F, O, OCH ₂ F, H, H, H, O], [[ AK2188; H, OEt, H, F, O, OCHF 2, H, H, H, O], [AK2189; H, OEt, H, F, O, OCF 3, H, H, H, O], [ AK2190; H, OEt, H, F, O, OCF 3, H, H, H, O], [AK2191; H, OEt, H, Cl, O, H, H, H, H, O], [AK2192 H, OEt, H, Cl, O, F, H, H, H, O], [AK 2193; H, OEt, H, Cl, O, Cl, H, H, H, O], [AK 2 194; H , OEt, H, Cl, O, Br, H, H, H, O], [AK2195; H, OEt, H, Cl, O, I, H, H, H, O], [AK 2196; H, OEt , H, Cl, O, Me, H, H, H, O], [AK 2 197; H, OEt, H, Cl, O, Et, H, H, H, O], [AK 2198; H, OE t, H , Cl, O, Pr, H, H, H, O], [AK 2199; H, OEt, H, Cl, O, i-Pr, H, H, H, O], [AK 2200; H, OE t, H] , Cl, O, Bu, H, H, H, O],

[AK2201; H, OEt, H, Cl, O, i-Bu, H, H, H, O], [AK 2202; H, OEt, H, Cl, O, sec-Bu, H, H, H, O H, OEt, H, Cl, O, t-Bu, H, H, H, O], [AK 2 204; H, OEt, H, Cl, O, c-Pr, H, H, H] , O], [AK2205; H, OEt, H, Cl, O, c-Bu, H, H, H, O], [AK 2206; H, OEt, H, Cl, O, OBu, H, H, H] H, OEt, H, Cl, O, Oi-Bu, H, H, H, O], [AK 2208; H, OEt, H, Cl, O, O-sec-Bu, H] , H, H, O], [AK2209; H, OEt, H, Cl, O, CH 2 F, H, H, H, O], [AK2210; H, OEt, H, Cl, O, CHF 2, H, H, H, O] , [AK2211; H, OEt, H, Cl, O, CF 3, H, H, H, O], [AK2212; H, OEt, H, Cl, O, OCH 2 F , H, H, H, O ], [AK2213; H, OEt, H, Cl, O, OCHF 2, H, H, H, O], [AK2214; H, OEt, H, Cl, O, OCF 3 , H, H, H, O ], [AK2215; H, OEt, H, Cl, O, OCF 3, H, H, H, O], [AK2216; H, OEt, H, Br, O, H, H, H, H, O], [AK2217; H, OEt, H, Br, O, F, H, H, H, O], [AK2218; H, OEt, H, Br, O, Cl, H, H, H, O], [AK2219; H, OEt, H, Br, O, Br, H, H, H, O], [AK2220; H, OEt, H, Br, O, I, H, H, H, O], [AK 2221; H, OEt, H, Br, O, Me, H, H, H, O], [AK 2222; H, OE t, H, Br, O, Et, H, H, H, O, [AK2223; H, OEt, H, Br, O, Pr, H, H, H, O], [AK2224; H, OEt, H, Br, O, i-Pr, H, H, H, O], [AK2225; H, OEt, H, Br, O, Bu, H, H, H, O], [AK 2226; H, OEt, H, Br, O, i-Bu, H, H, H, O], [AK 2 227; H, OEt, H, Br, O, sec-Bu, H, H, H, O] [AK 2 228; H, OEt, H, Br, O, t-Bu, H, H, H, O], [AK 2 229; H, OEt, H, Br, O, c-Pr, H, H, H, O H, OEt, H, Br, O, c-Bu, H, H, H, O], [AK 2 231; H, OEt, H, Br, O, OBu, H, H, H, O] H, OEt, H, Br, O, Oi-Bu, H, H, H, O], [AK 2233; H, OEt, H, Br, O, O-sec-Bu, H, H] , H, O], [AK2234 ; H, OEt, H, Br, O, CH 2 F, H, H, H, O], [AK2235; H, OEt, H, Br, O, CHF 2, H, H, H, O], [ AK2236; H, OEt, H, Br, O, CF 3, H, H, H, O], [AK2237; H, OEt, H, Br, O, OCH 2 F, H H, H, O], [AK 2238; H, OEt, H, Br, O, OCHF ₂ , H, H, H, O], [AK 2239; H, OEt, H, Br, O, OCF ₃ , H , H, H, O], [AK 2240; H, OEt, H, Br, O, OCF ₃ , H, H, H, O], [AK 2241; H, CHF ₂ , H, H, O, H, H , H, H, O], [AK2242; H, CHF 2, H, H, O, F, H, H, H, O], [AK2243; H, CHF 2, H, H, O, Cl, H , H, H, O], [AK ₂ 244; H, CHF ₂ , H, H, O, Br, H, H, H, O], [AK ₂ 245; H, CHF ₂ , H, H, O, I, H H, H, O], [AK 2246; H, CHF ₂ , H, H, O, Me, H, H, H, O], [AK ₂ 247; H, CHF ₂ , H, H, O, Et, H , H, H, O], [AK2248; H, CHF 2, H, H, O, Pr, H, H, H, O], [AK2249; H, CHF 2, H, H, O, i-Pr H, H, H, O], [AK ₂ 250; H, CHF ₂ , H, H, O, Bu, H, H, H, O], [AK 2251; H, CHF ₂ , H, H, O, i -Bu, H, H, H, O], [AK 2252; H, CHF ₂ , H, H, O, sec-Bu, H, H, H, O], [AK ₂ 253; H, CHF ₂ , H, H , O, t-Bu, H, H, H, O], [AK 2254; H, C HF ₂ , H, H, H, O, c-Pr, H, H, H, O], [AK ₂ 255; H, CHF ₂ , H, H, O, c-Bu, H, H, H, O], [[ _{AK2256; H, CHF 2, H} , H, O, OBu, H, H, H, O], [AK2257; H, CHF 2, H, H, O, Oi-Bu, H, H, H, O] _{, [AK2258; H, CHF 2} , H, H, O, O-sec-Bu, H, H, H, O], [AK2259; H, CHF 2, H, H, O, CH 2 F, H, H, H, O], [AK ₂ 260; H, CHF ₂ , H, H, O, CHF ₂ , H, H, H, O], [AK 2261; H, CHF ₂ , H, H, O, CF ₃ , H, H, H, O] , [AK2262; H, CHF 2, H, H, O, OCH 2 F, H, H, H, O], [AK2263; H, CHF 2, H, H, O, OHF ₂ , H, H, H, O], [AK ₂ 264; H, CHF ₂ , H, H, H, O, OCF ₃ , H, H, H, O], [AK ₂ 265; H, CHF ₂ , H, Me, O, H, H, H, H, O], [AK 2266; H, CHF ₂ , H, Me, O, F, H, H, H, O], [AK ₂ 267; H, CHF ₂ , H, Me, O, Cl, H, H, H, O], [AK 2268; H, CHF ₂ , H, Me, O, Br, H, H, H, O], [AK 2269; H, CHF ₂ , H, Me, O, I, H, H, H, O], [AK2270; H, CHF 2, H, Me, O, Me, H, H, H, O], [AK2271; H, CHF 2, H, Me, O, Et, H, H, H, O], [AK2272; H, CHF 2, H, Me, O, Pr, H, H, H, O], [AK2273; H, CHF 2, H, Me, O, i-Pr, H, H, H, O], [AK 2274; H, CHF ₂ , H, Me, O, Bu, H, H, H, O], [AK 2275; H, CHF ₂ , H, Me, O, i-Bu, H, H, H, O, [AK 2276; H, CHF ₂ , H, Me, O, sec-Bu, H, H, H, O], [AK 2277; H, CHF ₂ , H, Me, O, t-Bu, H, H, H, O], [AK ₂ 278; H, CHF ₂ , H, Me, O, c-Pr, H, H, H, O], [AK 2279 H, CHF ₂ , H, Me, O, c-Bu, H, H, H, O], [AK2280; H, CHF 2, H, Me, O, OBu, H, H, H, O], [AK2281; H, CHF 2, H, Me, O, Oi-Bu, H, H, H, O], [AK2282; H, CHF 2, H, Me, O, O-sec-Bu, H, H, H, O], [AK2283; H, CHF _{2, H, Me, O,} CH 2 F, H, H, H, O], [AK2284; H, CHF 2, H, Me, O, CHF 2, H, H, H, O], [AK2285; H, CHF ₂ , H, Me, O, CF ₃ , H, H, H, O], [AK 2286; H, CHF ₂ , H, Me, O, OCH ₂ F, H, H, H, O], _{[AK2287; H, CHF 2,} H, Me, O, OCHF 2, H, H, H, O], [AK2288; H, CHF 2, H, Me, O, OCF 3, H, H, H, O H, CHF ₂ , H, Me, O, OCF ₃ , H, H, H, O], [AK ₂ 290; H, CHF ₂ , H, Et, O, H, H, H, H, O], [AK2291; H, CHF 2, H, Et, O, F, H, H, H, O], [AK2292; H, CHF 2, H, Et, O, Cl, H, H, H, O], [AK 2293; H, CHF ₂ , H, Et, O, Br, H, H, H, O], [AK ₂ 294; H, CHF ₂ , H, Et, O, I, H, H, H, H, O], [AK2295; H, CHF 2, H, Et, O, Me, H, H, H, O], [AK2296; H, CHF 2, H, Et, O, Et, H, H, H, O], [AK 2297; H, CHF ₂ , H, Et, O, Pr, H, H, H, O], [AK 2298; H, CHF ₂ , H, Et, O, i-Pr, H, H, H, O], [AK ₂ 299; H, CHF ₂ , H, Et, O, Bu, H, H, H, O], [AK ₂ 300; H, CHF ₂ , H, Et, O, i-Bu, H, H, H, O],

_{[AK2301; H, CHF 2,} H, Et, O, sec-Bu, H, H, H, O], [AK2302; H, CHF 2, H, Et, O, t-Bu, H, H, H , O], [AK2303; H , CHF 2, H, Et, O, c-Pr, H, H, H, O], [AK2304; H, CHF 2, H, Et, O, c-Bu, H , H, H, O], [AK ₂ 305; H, CHF ₂ , H, Et, O, OBu, H, H, H, O], [AK 2306; H, CHF ₂ , H, Et, O, Oi-Bu H, H, H, O], [AK 2307; H, CHF ₂ , H, Et, O, O-sec-Bu, H, H, H, O], [AK ₂ 308; H, CHF ₂ , H, Et] _{, O, CH 2 F, H} , H, H, O], [AK2309; H, CHF 2, H, Et, O, CHF 2, H, H, H, O], [AK2310; H, CHF 2, _{H, Et, O, CF 3} , H, H, H, O], [AK2311; H, CHF 2, H, Et, O, OCH 2 F, H, H, H, O], [AK2312; H, _{CHF 2, H, Et, O} , OCHF 2, H, H, H, O], [AK2313; H, CHF 2, H, Et, O, OCF 3, H, H, H, O], [AK2314; _{H, CHF 2, H, Et} , O, OCF 3, H, H, H, O], [AK2315; H, CHF 2, H, Pr, O, H, H, H, H, O], [AK2316 _{; H, CHF 2, H,} Pr, O, F, H, H, H, O], [AK2317; H, CHF 2, H, Pr, O, Cl, H, H, H, O], [AK2318 _{; H, CHF 2, H,} Pr, O, Br, H, H, H, O], [AK2319; H, CHF 2, H, Pr, O, I, H, H, H, O], [AK2320 H, CHF ₂ , H, Pr, O, Me, H, H, H, O], [AK2321; H, CHF ₂ , H, Pr, O, Et, H, H, H, O], [AK2322 _{; H, CHF 2, H,} Pr, O, Pr, H, H, H, O], [AK2323; H, CHF 2, H, Pr, O, i-Pr, H, H, H, O], _{[AK2324; H, CHF 2,} H, Pr, O, Bu, H, H, H, O], [AK2325; H, CHF 2, H, Pr, O, i-Bu, H, H, H, O ], _{[AK2326; H, CHF 2,} H, Pr, O, sec-Bu, H, H, H, O], [AK2327; H, CHF 2, H, Pr, O, t-Bu, H, H, H , O], [AK2328; H , CHF 2, H, Pr, O, c-Pr, H, H, H, O], [AK2329; H, CHF 2, H, Pr, O, c-Bu, H , H, H, O], [AK2330; H, CHF 2, H, Pr, O, OBu, H, H, H, O], [AK2331; H, CHF 2, H, Pr, O, Oi-Bu , H, H, H, O ], [AK2332; H, CHF 2, H, Pr, O, O-sec-Bu, H, H, H, O], [AK2333; H, CHF 2, H, Pr , O, CH ₂ F, H, H, H, O], [AK 2334; H, CHF ₂ , H, Pr, O, CHF ₂ , H, H, H, O], [AK ₂ 335; H, CHF ₂ , H, Pr, O, CF ₃ , H, H, H, O], [AK 2336; H, CHF ₂ , H, Pr, O, OCH ₂ F, H, H, O, [AK 2 337; H, CHF ₂ , H, Pr, O, OCHF ₂ , H, H, H, O], [AK ₂ 338; H, CHF ₂ , H, Pr, O, OCF ₃ , H, H, H, O], [AK 2339; _{H, CHF 2, H, Pr} , O, OCF 3, H, H, H, O], [AK2340; H, CHF 2, H, i-Pr, O, H, H, H, H, O], _{[AK2341; H, CHF 2,} H, i-Pr, O, F, H, H, H, O], [AK2342; H, CHF 2, H, i-Pr, O, Cl, H, H, H , O], [AK 2343; H, CHF ₂ , H, i-Pr, O, Br, H, H, H, O], [AK 2344; H, CHF ₂ , H, i-Pr, O, I, H H, H, O], [AK 2345; H, CHF ₂ , H, i-Pr, O, Me, H, H, H, O], [AK 2346; H, CHF ₂ , H, i-Pr, O , Et, H, H, H , O], [AK2347; H, CHF 2, H, i-Pr, O, Pr, H, H, H, O], [AK2348; H, CHF 2, H, i -Pr, O, i-Pr, H, H, H, O], [AK 2349; H, CHF ₂ , H, i-Pr, O, Bu, H, H, H, O], [AK 2 350; H, CHF ₂ , H, i -Pr, O, i-Bu, H, H, H, O], [AK2351; H, CHF 2, H, i-Pr, O, sec-Bu, H, H, H, O], [AK2352; _{H, CHF 2, H, i} -Pr, O, t-Bu, H, H, H, O], [AK2353; H, CHF 2, H, i-Pr, O, c-Pr, H, H, H, O], [AK 2354; H, CHF ₂ , H, i-Pr, O, c-Bu, H, H, H, O], [AK ₂ 355; H, CHF ₂ , H, i-Pr, O, OBu, H, H, H, O], [AK 2356; H, CHF ₂ , H, i-Pr, O, Oi-Bu, H, H, H, O], [AK ₂ 357; H, CHF ₂ , H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK ₂ 358; H, CHF ₂ , H, i-Pr, O, CH ₂ F, H, H, H, O], [AK 2359; H, CHF ₂ , H, i-Pr, O, CHF ₂ , H, H, H, O], [AK ₂ 360; H, CHF ₂ , H, i-Pr, O, CF ₃ , H, H , H, O], [AK2361 ; H, CHF 2, H, i-Pr, O, OCH 2 F, H, H, H, O], [AK2362; H, CHF 2, H, i-Pr, O _{, OCHF 2, H, H,} H, O], [AK2363; H, CHF 2, H, i-Pr, O, OCF 3, H, H, H, O], [AK2364; H, CHF 2, H , i-Pr, O, OCF ₃ , H, H, H, O], [AK 2365; H, CHF ₂ , H, OMe, O, H, H, H, H, O], [AK 2 366; H, CHF ₂ , H, OMe, O, F, H, H, H, O], [AK2367; H, CHF ₂ , H, OMe, O, Cl, H, H, H, O], [AK 2368; H, CHF ₂ , H, OMe, O, Br, H, H, H, O], [AK 2369; H, CHF ₂ , H, OMe, O, I, H, H, H, O], [AK 2370; H, CHF _{2, H, OMe, O,} Me, H, H, H, O], [AK2371; H, CHF 2, H, OMe, O, Et, H, H, H, O], [AK2372; H, CHF ₂ , H, OMe, O, Pr, H, H, H, O], [AK 2373; H, CHF ₂ , H, OMe, O, i-Pr, H, H, H, O], [AK 2374; H , CHF ₂ , H, OMe, O, Bu, H, H, H, O], [AK 2375; H, CHF ₂ , H, OMe, O, i-Bu, H, H, H, O], [AK ₂ 376; H, CHF ₂ , H, OMe, O, sec- Bu, H, H, H, O], [AK2377; H, CHF 2, H, OMe, O, t-Bu, H, H, H, O], [AK2378; H _{, CHF 2, H, OMe,} O, c-Pr, H, H, H, O], [AK2379; H, CHF 2, H, OMe, O, c-Bu, H, H, H, O], _{[AK2380; H, CHF 2,} H, OMe, O, OBu, H, H, H, O], [AK2381; H, CHF 2, H, OMe, O, Oi-Bu, H, H, H, O ], [AK2382; H, CHF 2, H, OMe, O, O-sec-Bu, H, H, H, O], [AK2383; H, CHF 2, H, OMe, O, CH 2 F, H , H, H, O], [AK 2384; H, CHF ₂ , H, OMe, O, CHF ₂ , H, H, H, O], [AK 2385; H, CHF ₂ , H, OMe, O, CF ₃ H, H, H, O], [AK 2386; H, CHF ₂ , H, OMe, O, OCH ₂ F, H, H, H, O], [AK 2387; H, CHF ₂ , H, OMe, O _{, OCHF 2, H, H,} H, O], [AK2388; H, CHF 2, H, OMe, O, OCF 3, H, H, H, O], [AK2389; H, CHF 2, H, OMe _{, O, OCF 3, H,} H, H, O], [AK2390; H, CHF 2, H, F, O, H, H, H, H, O], [AK2391; H, CHF 2, H, F, O, F, H, H, H, O], [AK2392; H, CHF 2, H, F, O, Cl, H, H, H, O], [AK2393; H, CHF 2, H, F, O, Br, H, H, H, O], [AK2394; H, CHF 2, H, F, O, I, H, H, H, O], [AK2395; H, CHF 2, H, F, O, Me, H, H, H, O], [AK 2396; H, CHF ₂ , H, F, O, Et, H, H, H, O], [AK 2397; H, CHF ₂ , H, F, O, Pr, H, H, H, O, [AK 2398; H, CHF ₂ , H, F, O, i-Pr, H, H, H, O], [AK 2399; H, CH F ₂ , H, F, O, Bu, H, H, H, O], [AK2400; H, CHF ₂ , H, F, O, i-Bu, H, H, H, O],

_{[AK2401; H, CHF 2,} H, F, O, sec-Bu, H, H, H, O], [AK2402; H, CHF 2, H, F, O, t-Bu, H, H, H , O], [AK2403; H , CHF 2, H, F, O, c-Pr, H, H, H, O], [AK2404; H, CHF 2, H, F, O, c-Bu, H , H, H, O], [AK ₂ 405; H, CHF ₂ , H, F, O, OBu, H, H, H, O], [AK 2406; H, CHF ₂ , H, F, O, Oi-Bu , H, H, H, O], [AK 2407; H, CHF ₂ , H, F, O, O-sec-Bu, H, H, H, O], [AK ₂ 408; H, CHF ₂ , H, F _{, O, CH 2 F, H} , H, H, O], [AK2409; H, CHF 2, H, F, O, CHF 2, H, H, H, O], [AK2410; H, CHF 2, _{H, F, O, CF 3} , H, H, H, O], [AK2411; H, CHF 2, H, F, O, OCH 2 F, H, H, H, O], [AK2412; H, _{CHF 2, H, F, O} , OCHF 2, H, H, H, O], [AK2413; H, CHF 2, H, F, O, OCF 3, H, H, H, O], [AK2414; _{H, CHF 2, H, F} , O, OCF 3, H, H, H, O], [AK2415; H, CHF 2, H, Cl, O, H, H, H, H, O], [AK2416 _{; H, CHF 2, H,} Cl, O, F, H, H, H, O], [AK2417; H, CHF 2, H, Cl, O, Cl, H, H, H, O], [AK2418 _{; H, CHF 2, H,} Cl, O, Br, H, H, H, O], [AK2419; H, CHF 2, H, Cl, O, I, H, H, H, O], [AK2420 _{; H, CHF 2, H,} Cl, O, Me, H, H, H, O], [AK2421; H, CHF 2, H, Cl, O, Et, H, H, H, O], [AK2422 _{; H, CHF 2, H,} Cl, O, Pr, H, H, H, O], [AK2423; H, CHF 2, H, Cl, O, i-Pr, H, H, H, O], _{[AK2424; H, CHF 2,} H, Cl, O, Bu, H, H, H, O], [AK2425; H, CHF 2, H, Cl, O, i-Bu, H, H, H, O ], [AK 2426; H, CHF _{2, H, Cl, O,} sec-Bu, H, H, H, O], [AK2427; H, CHF 2, H, Cl, O, t-Bu, H, H, H, O], [AK2428 _{; H, CHF 2, H,} Cl, O, c-Pr, H, H, H, O], [AK2429; H, CHF 2, H, Cl, O, c-Bu, H, H, H, O ], [AK2430; H, CHF 2, H, Cl, O, OBu, H, H, H, O], [AK2431; H, CHF 2, H, Cl, O, Oi-Bu, H, H, H , O], [AK2432; H , CHF 2, H, Cl, O, O-sec-Bu, H, H, H, O], [AK2433; H, CHF 2, H, Cl, O, CH 2 F , H, H, H, O ], [AK2434; H, CHF 2, H, Cl, O, CHF 2, H, H, H, O], [AK2435; H, CHF 2, H, Cl, O, _{CF 3, H, H, H} , O], [AK2436; H, CHF 2, H, Cl, O, OCH 2 F, H, H, H, O], [AK2437; H, CHF 2, H, Cl , O, OCHF ₂ , H, H, H, O], [AK 2438; H, CHF ₂ , H, Cl, O, OCF ₃ , H, H, H, O], [AK 2439; H, CHF ₂ , H _{, Cl, O, OCF 3,} H, H, H, O], [AK2440; H, CHF 2, H, Br, O, H, H, H, H, O], [AK2441; H, CHF 2, H, Br, O, F, H, H, H, O], [AK2442; H, CHF 2, H, Br, O, Cl, H, H, H, O], [AK2443; H, CHF 2, H, Br, O, Br, H, H, H, O], [AK2444; H, CHF 2, H, Br, O, I, H, H, H, O], [AK2445; H, CHF 2, H, Br, O, Me, H, H, H, O], [AK2446; H, CHF 2, H, Br, O, Et, H, H, H, O], [AK2447; H, CHF 2, H, Br, O, Pr, H, H, H, O], [AK 2448; H, CHF ₂ , H, Br, O, i-Pr, H, H, H, O], [AK 2449; H, CHF _{2, H, Br, O,} Bu, H, H, H, O], [AK2450; H, CHF 2, H, Br, O, i-Bu, H, H, H, O], [AK2451; H , CHF _{2, H, Br, O,} sec-Bu, H, H, H, O], [AK2452; H, CHF 2, H, Br, O, t-Bu, H, H, H, O], [AK2453 _{; H, CHF 2, H,} Br, O, c-Pr, H, H, H, O], [AK2454; H, CHF 2, H, Br, O, c-Bu, H, H, H, O ], [AK2455; H, CHF 2, H, Br, O, OBu, H, H, H, O], [AK2456; H, CHF 2, H, Br, O, Oi-Bu, H, H, H , O], [AK2457; H , CHF 2, H, Br, O, O-sec-Bu, H, H, H, O], [AK2458; H, CHF 2, H, Br, O, CH 2 F , H, H, H, O ], [AK2459; H, CHF 2, H, Br, O, CHF 2, H, H, H, O], [AK2460; H, CHF 2, H, Br, O, _{CF 3, H, H, H} , O], [AK2461; H, CHF 2, H, Br, O, OCH 2 F, H, H, H, O], [AK2462; H, CHF 2, H, Br _{, O, OCHF 2, H,} H, H, O], [AK2463; H, CHF 2, H, Br, O, OCF 3, H, H, H, O], [AK2464; H, CHF 2, H _{, Br, O, OCF 3,} H, H, H, O], [AK2465; H, CF 3, H, H, O, H, H, H, H, O], [AK2466; H, CF 3, H, H, O, F, H, H, H, O], [AK2467; H, CF 3, H, H, O, Cl, H, H, H, O], [AK2468; H, CF 3, H, H, O, Br, H, H, H, O], [AK 2469; H, CF ₃ , H, H, O, I, H, H, H, O], [AK 2 470; H, CF ₃ , H, H, O, Me, H, H, H, O], [AK2471; H, CF 3, H, H, O, Et, H, H, H, O], [AK2472; H, CF 3, H, H, O, Pr, H, H, H, O], [AK 2 473; H, CF ₃ , H, H, O, i-Pr, H, H, H, O], [AK 2 474; H, CF _{3, H, H, O,} Bu, H, H, H, O], [AK2475; H, CF 3, H, H, O, i-Bu, H, H, H, O], [AK2476; H , CF ₃ , H, H, O, sec-Bu, H, H, H, O ], [AK2477; H, CF 3, H, H, O, t-Bu, H, H, H, O], [AK2478; H, CF 3, H, H, O, c-Pr, H, H , H, O], [AK 2479; H, CF ₃ , H, H, O, c-Bu, H, H, H, O], [AK 2 480; H, CF ₃ , H, H, O, OBu, H , H, H, O], [AK2481; H, CF 3, H, H, O, Oi-Bu, H, H, H, O], [AK2482; H, CF 3, H, H, O, O -sec-Bu, H, H, H, O], [AK2483; H, CF 3, H, H, O, CH 2 F, H, H, H, O], [AK2484; H, CF 3, H _{, H, O, CHF 2,} H, H, H, O], [AK2485; H, CF 3, H, H, O, CF 3, H, H, H, O], [AK2486; H, CF 3 , H, H, O, OCH 2 F, H, H, H, O], [AK2487; H, CF 3, H, H, O, OCHF 2, H, H, H, O], [AK2488; H , CF ₃ , H, H, O, OCF ₃ , H, H, H, O], [AK 2489; H, CF ₃ , H, Me, O, H, H, H, H, O], [AK 2490; _{H, CF 3, H, Me} , O, F, H, H, H, O], [AK2491; H, CF 3, H, Me, O, Cl, H, H, H, O], [AK2492; _{H, CF 3, H, Me} , O, Br, H, H, H, O], [AK2493; H, CF 3, H, Me, O, I, H, H, H, O], [AK2494; _{H, CF 3, H, Me} , O, Me, H, H, H, O], [AK2495; H, CF 3, H, Me, O, Et, H, H, H, O], [AK2496; _{H, CF 3, H, Me} , O, Pr, H, H, H, O], [AK2497; H, CF 3, H, Me, O, i-Pr, H, H, H, O], [ _{AK2498; H, CF 3, H} , Me, O, Bu, H, H, H, O], [AK2499; H, CF 3, H, Me, O, i-Bu, H, H, H, O] _{, [AK2500; H, CF 3} , H, Me, O, sec-Bu, H, H, H, O],

_{[AK2501; H, CF 3,} H, Me, O, t-Bu, H, H, H, O], [AK2502; H, CF 3, H, Me, O, c-Pr, H, H, H , O], [AK2503; H , CF 3, H, Me, O, c-Bu, H, H, H, O], [AK2504; H, CF 3, H, Me, O, OBu, H, H , H, O], [AK2505 ; H, CF 3, H, Me, O, Oi-Bu, H, H, H, O], [AK2506; H, CF 3, H, Me, O, O-sec -Bu, H, H, H, O], [AK 2507; H, CF ₃ , H, Me, O, CH ₂ F, H, H, H, O], [AK 2508; H, CF ₃ , H, Me , O, CHF ₂ , H, H, H, O], [AK 2509; H, CF ₃ , H, Me, O, CF ₃ , H, H, H, O], [AK 2510; H, CF ₃ , H] , Me, O, OCH ₂ F, H, H, H, O], [AK 2511; H, CF ₃ , H, Me, O, OCHF ₂ , H, H, H, O], [AK 2512; H, CF _{3, H, Me, O,} OCF 3, H, H, H, O], [AK2513; H, CF 3, H, Me, O, OCF 3, H, H, H, O], [AK2514; H , CF ₃ , H, Et, O, H, H, H, H, O], [AK 2515; H, CF ₃ , H, Et, O, F, H, H, H, O], [AK 2516; H _{, CF 3, H, Et,} O, Cl, H, H, H, O], [AK2517; H, CF 3, H, Et, O, Br, H, H, H, O], [AK2518; H _{, CF 3, H, Et,} O, I, H, H, H, O], [AK2519; H, CF 3, H, Et, O, Me, H, H, H, O], [AK2520; H , CF ₃ , H, Et, O, Et, H, H, H, O], [AK 2521; H, CF ₃ , H, Et, O, Pr, H, H, H, O], [AK 2522; H _{, CF 3, H, Et,} O, i-Pr, H, H, H, O], [AK2523; H, CF 3, H, Et, O, Bu, H, H, H, O], [AK2524 _{; H, CF 3, H,} Et, O, i-Bu, H, H, H, O], [AK2525; H, CF 3, H, Et, O, sec-Bu, H, H, H, O ], [AK2526; H, CF 3, H, Et, O, t- Bu, H, H, H, O], [AK2527; H, CF 3, H, Et, O, c-Pr, H, H, H, O], [AK2528; H, CF 3, H, Et, O, c-Bu, H, H, H, O], [AK 2529; H, CF ₃ , H, Et, O, OBu, H, H, H, O], [AK 2530; H, CF ₃ , H, Et, O, Oi-Bu, H, H, H, O], [AK2531; H, CF 3, H, Et, O, O-sec-Bu, H, H, H, O], [AK2532; H , CF ₃ , H, Et, O, CH ₂ F, H, H, H, O], [AK 2533; H, CF ₃ , H, Et, O, CHF ₂ , H, H, H, O], [[ _{AK2534; H, CF 3, H} , Et, O, CF 3, H, H, H, O], [AK2535; H, CF 3, H, Et, O, OCH 2 F, H, H, H, O ], [AK2536; H, CF 3, H, Et, O, OCHF 2, H, H, H, O], [AK2537; H, CF 3, H, Et, O, OCF 3, H, H, H H, CF ₃ , H, Et, O, OCF ₃ , H, H, H, O], [AK 2 539; H, CF ₃ , H, Pr, O, H, H, H, H H, O], [AK2540; H, CF 3, H, Pr, O, F, H, H, H, O], [AK2541; H, CF 3, H, Pr, O, Cl, H, H, H, O], [AK2542; H, CF 3, H, Pr, O, Br, H, H, H, O], [AK2543; H, CF 3, H, Pr, O, I, H, H, H, O], [AK2544; H, CF 3, H, Pr, O, Me, H, H, H, O], [AK2545; H, CF 3, H, Pr, O, Et, H, H, H, O], [AK 2546; H, CF ₃ , H, Pr, O, Pr, H, H, H, O], [AK 2547; H, CF ₃ , H, Pr, O, i-Pr, H, H, H, O], [ AK2548; H, CF 3, H, Pr, O, Bu, H, H, H, O], [AK2549; H, CF 3, H, Pr, O, i-Bu, H, H, H, O] , [AK2550; H, CF 3, H, Pr, O, sec-Bu, H, H, H, O], [AK2551; H, CF 3, H, Pr, O, t-Bu, H, H, H, O], [AK2552; H, C F ₃ , H, Pr, O, c, Pr, H, H, H, O], [AK2553; H, CF ₃ , H, Pr, O, c, Bu, H, H, H, O], [[ AK 2554; H, CF ₃ , H, Pr, O, OBu, H, H, H, O], [AK 2 555; H, CF ₃ , H, Pr, O, Oi-Bu, H, H, H, O] _{, [AK2556; H, CF 3} , H, Pr, O, O-sec-Bu, H, H, H, O], [AK2557; H, CF 3, H, Pr, O, CH 2 F, H, H, H, O], [ AK2558; H, CF 3, H, Pr, O, CHF 2, H, H, H, O], [AK2559; H, CF 3, H, Pr, O, CF 3, H, H, H, O] , [AK2560; H, CF 3, H, Pr, O, OCH 2 F, H, H, H, O], [AK2561; H, CF 3, H, Pr, O, _{OCHF 2, H, H, H} , O], [AK2562; H, CF 3, H, Pr, O, OCF 3, H, H, H, O], [AK2563; H, CF 3, H, Pr, _{O, OCF 3, H, H} , H, O], [AK2564; H, CF 3, H, i-Pr, O, H, H, H, H, O], [AK2565; H, CF 3, H , i-Pr, O, F, H, H, H, O], [AK 2566; H, CF ₃ , H, i-Pr, O, Cl, H, H, O], [AK 2 567; H, _{CF 3, H, i-Pr} , O, Br, H, H, H, O], [AK2568; H, CF 3, H, i-Pr, O, I, H, H, H, O], [ AK 2569; H, CF ₃ , H, i-Pr, O, Me, H, H, H, O], [AK 2570; H, CF ₃ , H, i-Pr, O, Et, H, H, H, O], [AK2571; H, CF 3, H, i-Pr, O, Pr, H, H, H, O], [AK2572; H, CF 3, H, i-Pr, O, i-Pr, H, H, H, O] , [AK2573; H, CF 3, H, i-Pr, O, Bu, H, H, H, O], [AK2574; H, CF 3, H, i-Pr, O, i-Bu, H, H, H, O], [AK2575; H, CF 3, H, i-Pr, O, sec-Bu, H, H, H, O], [AK2576; H, CF ₃ , H, i-Pr, O, t-Bu, H, H, H, O], [AK 2577; H, CF ₃ , H, i-Pr, O, c-Pr, H, H, H, O], [AK 2578; H, CF ₃ , H, i-Pr, O, c-Bu, H, H, H, H, O], [AK2579; H, CF 3, H, i-Pr, O, OBu, H, H, H, O], [AK2580; H, CF 3, H, i-Pr, O, Oi-Bu, H, H, H, O], [AK 2581; H, CF ₃ , H, i-Pr, O, O-sec-Bu, H, H, H, O], [AK 2582; H, CF ₃ , H, _{i-Pr, O, CH 2} F, H, H, H, O], [AK2583; H, CF 3, H, i-Pr, O, CHF 2, H, H, H, O], [AK2584; _{H, CF 3, H, i} -Pr, O, CF 3, H, H, H, O], [AK2585; H, CF 3, H, i-Pr, O, OCH 2 F, H, H, H , O], [AK2586; H , CF 3, H, i-Pr, O, OCHF 2, H, H, H, O], [AK2587; H, CF 3, H, i-Pr, O, OCF 3 , H, H, H, O ], [AK2588; H, CF 3, H, i-Pr, O, OCF 3, H, H, H, O], [AK2589; H, CF 3, H, OMe, O, H, H, H, H, O], [AK2590; H, CF 3, H, OMe, O, F, H, H, H, O], [AK2591; H, CF 3, H, OMe, O, Cl, H, H, H, O], [AK2592; H, CF 3, H, OMe, O, Br, H, H, H, O], [AK2593; H, CF 3, H, OMe, O, I, H, H, H, O], [AK2594; H, CF 3, H, OMe, O, Me, H, H, H, O], [AK2595; H, CF 3, H, OMe, O, Et, H, H, H, O], [AK2596; H, CF 3, H, OMe, O, Pr, H, H, H, O], [AK2597; H, CF 3, H, OMe, O, i-Pr, H, H, H, O], [AK2598; H, CF 3, H, OMe, O, Bu, H, H, H, O], [AK2599; H, CF 3, H, OMe, O, i-Bu, H, H, H, O], [AK 2600; H, CF ₃ , H, OMe, O, sec-Bu, H, H, H, O],

_{[AK2601; H, CF 3,} H, OMe, O, t-Bu, H, H, H, O], [AK2602; H, CF 3, H, OMe, O, c-Pr, H, H, H , O], [AK 2603; H, CF ₃ , H, OMe, O, c-Bu, H, H, H, O], [AK 2 604; H, CF ₃ , H, OMe, O, OBu, H, H , H, O], [AK2605 ; H, CF 3, H, OMe, O, Oi-Bu, H, H, H, O], [AK2606; H, CF 3, H, OMe, O, O-sec -Bu, H, H, H, O], [AK 2607; H, CF ₃ , H, OMe, O, CH ₂ F, H, H, H, O], [AK 2 608; H, CF ₃ , H, OMe _{, O, CHF 2, H,} H, H, O], [AK2609; H, CF 3, H, OMe, O, CF 3, H, H, H, O], [AK2610; H, CF 3, H , OMe, O, OCH ₂ F, H, H, H, O], [AK 2611; H, CF ₃ , H, OMe, O, OCHF ₂ , H, H, H, O], [AK 2612; H, CF _{3, H, OMe, O,} OCF 3, H, H, H, O], [AK2613; H, CF 3, H, OMe, O, OCF 3, H, H, H, O], [AK2614; H _{, CF 3, H, F,} O, H, H, H, H, O], [AK2615; H, CF 3, H, F, O, F, H, H, H, O], [AK2616; H , CF ₃ , H, F, O, Cl, H, H, H, O], [AK 2617; H, CF ₃ , H, F, O, Br, H, H, O], [AK 2618; H _{, CF 3, H, F,} O, I, H, H, H, O], [AK2619; H, CF 3, H, F, O, Me, H, H, H, O], [AK2620; H _{, CF 3, H, F,} O, Et, H, H, H, O], [AK2621; H, CF 3, H, F, O, Pr, H, H, H, O], [AK2622; H _{, CF 3, H, F,} O, i-Pr, H, H, H, O], [AK2623; H, CF 3, H, F, O, Bu, H, H, H, O], [AK2624 _{; H, CF 3, H,} F, O, i-Bu, H, H, H, O], [AK2625; H, CF 3, H, F, O, sec-Bu, H, H, H, O , [AK 2626; H, CF ₃ , H, F, O, t − Bu, H, H, H, O], [AK2627; H, CF 3, H, F, O, c-Pr, H, H, H, O], [AK2628; H, CF 3, H, F, O, c-Bu, H, H, H, O], [AK 2629; H, CF ₃ , H, F, O, OBu, H, H, H, O], [AK 2630; H, CF ₃ , H, F, O, Oi-Bu, H, H, H, O], [AK2631; H, CF 3, H, F, O, O-sec-Bu, H, H, H, O], [AK2632; H , CF ₃ , H, F, O, CH ₂ F, H, H, H, O], [AK 2633; H, CF ₃ , H, F, O, CHF ₂ , H, H, H, O], [[ _{AK2634; H, CF 3, H} , F, O, CF 3, H, H, H, O], [AK2635; H, CF 3, H, F, O, OCH 2 F, H, H, H, O H, CF ₃ , H, F, O, OCHF ₂ , H, H, H, O], [AK 2637; H, CF ₃ , H, F, O, OCF ₃ , H, H, H] H, CF ₃ , H, F, O, OCF ₃ , H, H, H, O], [AK 2639; H, CF ₃ , H, Cl, O, H, H, H, H H, O], [AK2640; H, CF 3, H, Cl, O, F, H, H, H, O], [AK2641; H, CF 3, H, Cl, O, Cl, H, H, H, O], [AK2642; H, CF 3, H, Cl, O, Br, H, H, H, O], [AK2643; H, CF 3, H, Cl, O, I, H, H, H, O], [AK2644; H, CF 3, H, Cl, O, Me, H, H, H, O], [AK2645; H, CF 3, H, Cl, O, Et, H, H, H, O], [AK 2646; H, CF ₃ , H, Cl, O, Pr, H, H, H, O], [AK 2647; H, CF ₃ , H, Cl, O, i-Pr, H, H, H, O], [ AK2648; H, CF 3, H, Cl, O, Bu, H, H, H, O], [AK2649; H, CF 3, H, Cl, O, i-Bu, H, H, H, O] , [AK2650; H, CF 3, H, Cl, O, sec-Bu, H, H, H, O], [AK2651; H, CF 3, H, Cl, O, t-Bu, H, H, H, O], [AK2652; H, CF 3, H, Cl, O, c-Pr, H, H, H, O], [AK2653; H, CF 3, H, Cl, O, c-Bu, H, H, H, O], [AK2654; H, CF 3, H, Cl, O, OBu, H, H, H, O], [AK2655; H, CF 3, H, Cl, O, Oi-Bu, H, H, H, O], [AK2656; H, CF 3, H, Cl, O, O- sec-Bu, H, H, H, O], [AK2657; H, CF 3, H, Cl, O, CH 2 F, H, H, H, O], [AK2658 _{; H, CF 3, H,} Cl, O, CHF 2, H, H, H, O], [AK2659; H, CF 3, H, Cl, O, CF 3, H, H, H, O], _{[AK2660; H, CF 3,} H, Cl, O, OCH 2 F, H, H, H, O], [AK2661; H, CF 3, H, Cl, O, OCHF 2, H, H, H, O], [AK2662; H, CF 3, H, Cl, O, OCF 3, H, H, H, O], [AK2663; H, CF 3, H, Cl, O, OCF 3, H, H, H, O], [AK 2664; H, CF ₃ , H, Br, O, H, H, H, H, O], [AK 2 665; H, CF ₃ , H, Br, O, F, H, H, H, H, O], [AK 2 666; H, CF ₃ , H, Br, O, Cl, H, H, H, O], [AK 2 667; H, CF ₃ , H, Br, O, Br, H, H, H, H, O], [AK 2668; H, CF ₃ , H, Br, O, I, H, H, H, O], [AK 2 669; H, CF ₃ , H, Br, O, Me, H, H, H H, O], [AK2670; H, CF 3, H, Br, O, Et, H, H, H, O], [AK2671; H, CF 3, H, Br, O, Pr, H, H, H, O], [AK2672; H, CF 3, H, Br, O, i-Pr, H, H, H, O], [AK2673; H, CF 3, H, Br, O, Bu, H, H, H, O], [AK 2 674; H, CF ₃ , H, Br, O, i-Bu, H, H, H, O], [AK 2 675; H, CF ₃ , H, Br, O, sec- Bu, H, H, H, O], [AK 2 676; H, CF ₃ , H, Br, O, t-Bu, H, H, H, O], [AK 2677; H, CF ₃ , H, Br, O, c-Pr, H, H, H, O], [AK2678; H _{, CF 3, H, Br,} O, c-Bu, H, H, H, O], [AK2679; H, CF 3, H, Br, O, OBu, H, H, H, O], [AK2680 _{; H, CF 3, H,} Br, O, Oi-Bu, H, H, H, O], [AK2681; H, CF 3, H, Br, O, O-sec-Bu, H, H, H , O], [AK2682; H , CF 3, H, Br, O, CH 2 F, H, H, H, O], [AK2683; H, CF 3, H, Br, O, CHF 2, H, H, H, O], [ AK2684; H, CF 3, H, Br, O, CF 3, H, H, H, O], [AK2685; H, CF 3, H, Br, O, OCH 2 F H, H, H, O], [AK 2 686; H, CF ₃ , H, Br, O, OCHF ₂ , H, H, H, O], [AK 2687; H, CF ₃ , H, Br, O, OCF ₃ , H, H, H, O], [AK 2688; H, CF ₃ , H, Br, O, OCF ₃ , H, H, H, O].

[Substituent number (MK2); E ¹¹¹ ]: [BK1; 3-Me-1-PYR], [BK2; 3-Me-4-F-1-PYR], [BK3; 3-Me-4-Cl -1-PYR !, [BK4; 3-Me-4-Br-1-PYR], [BK5; 3-Me-4-Me-1-PYR], [BK6; 3-Me-4-Et-1 -PYR], [BK7; 3-Me-4-OMe-1-PYR], [BK8; 3-Me-4-OEt-1-PYR], [BK9; 3-Me-4-CN-1-PYR ], [BK10; 3-Me -4-CHF 2 -1-PYR], [BK11; 3-Me-4-CF 3 -1-PYR], [BK12; 3-Me-4-OCHF 2 -1- PYR], [BK13; 3- Me-4-OCF 3 -1-PYR], [BK14; 3-Me-5-F-1-PYR], [BK15; 3-Me-5-Cl-1-PYR ], [BK16; 3-Me-5-Br-1-PYR], [BK17; 3-Me-5-Me-1-PYR], [BK18; 3-Me-5-Et-1-PYR], [BK19; 3-Me-5-OMe-1-PYR], [BK20; 3-Me-5-OEt-1-PYR], [BK21; 3-Me-5-CN-1-PYR], [BK22 3-Me-5-CHF ₂ -1-PYR], [BK23; 3-Me-5-CF ₃ -1-PYR], [BK 24; 3-Me-5-OCHF ₂ -1-PYR], [BK BK25; 3-Me-5- OCF 3 -1-PYR], [BK26; 3-Me-4-F-5-F-1-PYR], [BK27; 3-Me-4-F-5-Cl -1-PYR], [BK28; 3-Me-4-F-5-Br-1-PYR], [BK29; 3-Me-4-F-5-Me-1-PYR], [BK30; 3 -Me-4-F-5-Et-1-PYR], [BK31; 3-Me-4-F-5-OMe-1-PYR], [BK32; 3-Me-4-F-5-OEt -1-PYR !, [BK 33; 3-Me-4-F-5-CN-1-PYR], [BK 34; 3-Me-4-F-5-CHF ₂ -1-PYR], [BK 35; 3-Me-4-F- 5-CF 3 -1-PYR], [BK36; 3-Me-4-F-5-OCHF 2 -1-PYR], [BK37; 3-Me-4-F- 5-OCF ₃ -1-PYR], [BK 38; 3-Me-4-Cl-5-F-1-PYR], [B K39; 3-Me-4-Cl-5-Cl-1-PYR], [BK40; 3-Me-4-Cl-5-Br-1-PYR], [BK41; 3-Me-4-Cl- 5-Me-1-PYR], [BK 42; 3-Me-4-Cl-5-Et-1-PYR], [BK 43; 3-Me-4-Cl-5-OMe-1-PYR], [BK BK44; 3-Me-4-Cl-5-OEt-1-PYR], [BK45; 3-Me-4-Cl-5-CN-1-PYR], [BK46; 3-Me-4-Cl- 5-CHF ₂ -1-PYR], [BK 47; 3-Me-4-Cl-5-CF ₃ -1-PYR], [BK 48; 3-Me-4-Cl-5-OCHF ₂ -1-PYR ], [BK49; 3-Me -4-Cl-5-OCF 3 -1-PYR], [BK50; 3-Me-4-Br-5-F-1-PYR], [BK51; 3-Me- 4-Br-5-Cl-1-PYR], [BK52; 3-Me-4-Br-5-Br-1-PYR], [BK53; 3-Me-4-Br-5-Me-1-l PYR], [BK 54; 3-Me-4-Br-5-Et-1-PYR], [BK 55; 3-Me-4-Br-5-OMe-1-PYR], [BK 56; 3-Me- 4-Br-5-OEt-1-PYR], [BK57; 3-Me-4-Br-5-CN-1-PYR], [BK58; 3-Me-4-Br-5-CHF ₂ -1 -PYR], [BK59; 3- Me-4-Br-5-CF 3 -1-PYR], [BK60; 3-Me-4-Br-5-OCHF 2 -1-PYR], [BK61; 3 -Me-4-Br-5- OCF 3 -1-PYR], [BK62; 3-Me-4-Me-5-F-1-PYR], [BK63; 3-Me-4-Me-5- Cl-1-PYR], [BK 64; 3-Me-4-Me-5-Br-1-PYR], [BK 65; 3-Me-4-Me-5-Me-1-PYR], [BK 66; 3-Me-4-Me-5-Et-1-PYR], [BK67; 3-Me-4-Me-5-OMe-1-PYR], [BK68; 3-Me-4-Me-5-5 OEt-1-PYR], [BK69; 3-Me-4-Me-5-CN-1-PYR], [BK70; 3-Me-4-Me-5-CHF ₂ -1-PYR], [BK71 ; 3-Me-4-Me -5-CF 3 -1-PYR], [BK72; 3-Me-4-Me-5-OCHF 2 -1-PYR], [B K73; 3-Me-4- Me-5-OCF 3 -1-PYR], [BK74; 3-Me-4-Et-5-F-1-PYR], [BK75; 3-Me-4-Et -5-Cl-1-PYR], [BK 76; 3-Me-4-Et-5-Br-1-PYR], [BK 77; 3-Me-4-Et-5-Me-1-PYR], [BK 78; 3-Me-4-Et-5-Et-1-PYR], [BK 79; 3-Me-4-Et-5-OMe-1-PYR], [BK 80; 3-Me-4-Et -5-OEt-1-PYR], [BK 81; 3-Me-4-Et-5-CN-1-PYR], [BK 82; 3-Me-4-Et-5-CHF ₂ -1-PYR] , [BK 83; 3-Me-4-Et-5-CF ₃ -1-PYR], [BK 84; 3-Me-4-Et-5-OCHF ₂ -1-PYR], [BK 85; 3-Me- _{4-Et-5-OCF 3} -1-PYR], [BK86; 3-Me-4-OMe-5-F-1-PYR], [BK87; 3-Me-4-OMe-5-Cl-1 -PYR], [BK 88; 3-Me-4-OMe-5-Br-1-PYR], [BK 89; 3-Me-4-OMe-5-Me-1-PYR], [BK 90; 3-Me -4-OMe-5-Et-1-PYR], [BK 91; 3-Me-4-OMe-5-OMe-1-PYR], [BK 92; 3-Me-4-OMe-5-OEt-1 -PYR], [BK93; 3- Me-4-OMe-5-CN-1-PYR], [BK94; 3-Me-4-OMe-5-CHF 2 -1-PYR], [BK95; 3- Me-4-OMe-5- CF 3 -1-PYR], [BK96; 3-Me-4-OMe-5-OCHF 2 -1-PYR], [BK97; 3-Me-4-OMe-5- OCF ₃ -1-PYR], [BK 98; 3-Me-4-OEt-5-F-1-PYR], [BK 99; 3-Me-4-OEt-5-Cl-1-PYR], [BK 100] 3-Me-4-OEt-5-Br-1-PYR],

[BK101; 3-Me-4-OEt-5-Me-1-PYR], [BK102; 3-Me-4-OEt-5-Et-1-PYR], [BK103; 3-Me-4-OEt -5-OMe-1-PYR], [BK104; 3-Me-4-OEt-5-OEt-1-PYR], [BK105; 3-Me-4-OEt-5-CN-1-PYR], [BK106; 3-Me-4 -OEt-5-CHF 2 -1-PYR], [BK107; 3-Me-4-OEt-5-CF 3 -1-PYR], [BK108; 3-Me-4 -OEt-5-OCHF ₂ -1-PYR], [BK109; 3-Me-4-OEt-5-OCF ₃ -1-PYR], [BK110; 3-Me-4-CN-5-F-1 -PYR], [BK111; 3-Me-4-CN-5-Cl-1-PYR], [BK112; 3-Me-4-CN-5-Br-1-PYR], [BK113; 3-Me -4-CN-5-Me-1-PYR], [BK114; 3-Me-4-CN-5-Et-1-PYR], [BK115; 3-Me-4-CN-5-OMe-1 -PYR], [BK116; 3-Me-4-CN-5-OEt-1-PYR], [BK117; 3-Me-4-CN-5-CN-1-PYR], [BK118; 3-Me -4-CN-5-CHF ₂ -1-PYR], [BK119; 3-Me-4-CN-5-CF ₃ -1-PYR], [BK120; 3-Me-4-CN-5-OCHF _{2 -1-PYR], [BK121} ; 3-Me-4-CN-5-OCF 3 -1-PYR], [BK122; 3-Me-4-CHF 2 -5-F-1-PYR], [ BK123; 3-Me-4- CHF 2 -5-Cl-1-PYR], [BK124; 3-Me-4-CHF 2 -5-Br-1-PYR], [BK125; 3-Me-4- _{CHF 2 -5-Me-1-} PYR], [BK126; 3-Me-4-CHF 2 -5-Et-1-PYR], [BK127; 3-Me-4-CHF 2 -5-OMe-1 -PYR], [BK128; 3- Me-4-CHF 2 -5-OEt-1-PYR], [BK129; 3-Me-4-CHF 2 -5-CN-1-PYR], [BK130; 3 -Me-4-CHF ₂ -5-CHF ₂ -1-PYR], [BK 131; 3-Me 4-CHF ₂ -5-CF ₃ -1-PYR], [BK 132; 3- _{Me-4-CHF 2 -5-} OCHF 2 -1-PYR], [BK133; 3-Me-4-CHF 2 -5-OCF 3 -1-PYR], [BK134; 3-Me-4-CF 3 -5-F-1-PYR], [BK 135; 3-Me-4-CF ₃ -5-Cl-1-PYR], [BK 136; 3-Me-4-CF ₃ -5-Br-1-PYR ], [BK137; 3-Me -4-CF 3 -5-Me-1-PYR], [BK138; 3-Me-4-CF 3 -5-Et-1-PYR], [BK139; 3-Me -4-CF ₃ -5-OMe-1-PYR !, [BK 140; 3-Me-4-CF ₃ -5-OEt-1-PYR], [BK 141; 3-Me-4-CF ₃ -5- CN-1-PYR], [ BK142; 3-Me-4-CF 3 -5-CHF 2 -1-PYR], [BK143; 3-Me-4-CF 3 -5-CF 3 -1-PYR] , [BK144; 3-Me- 4-CF 3 -5-OCHF 2 -1-PYR], [BK145; 3-Me-4-CF 3 -5-OCF 3 -1-PYR], [BK146; 3- _{Me-4-OCHF 2 -5-} F-1-PYR], [BK147; 3-Me-4-OCHF 2 -5-Cl-1-PYR], [BK148; 3-Me-4-OCHF 2 -5 -Br-1-PYR], [ BK149; 3-Me-4-OCHF 2 -5-Me-1-PYR], [BK150; 3-Me-4-OCHF 2 -5-Et-1-PYR], [BK151; 3-Me-4 -OCHF 2 -5-OMe-1-PYR], [BK152; 3-Me-4-OCHF 2 -5-OEt-1-PYR], [BK153; 3-Me-4 _{-OCHF 2 -5-CN-1-} PYR], [BK154; 3-Me-4-OCHF 2 -5-CHF 2 -1-PYR], [BK155; 3-Me-4-OCHF 2 -5-CF _{3 -1-PYR], [BK156} ; 3-Me-4-OCHF 2 -5-OCHF 2 -1-PYR], [BK157; 3-Me-4-OCHF 2 -5-OCF 3 -1-PYR] , [BK158; 3-Me- 4-OCF 3 -5-F-1-PYR], [BK159; 3-Me-4-OCF 3 -5-Cl-1-PYR], [BK160; 3-Me- _{4-OCF 3 -5-Br-} 1-PYR], [BK161; 3-M _{e-4-OCF 3 -5-} Me-1-PYR], [BK162; 3-Me-4-OCF 3 -5-Et-1-PYR], [BK163; 3-Me-4-OCF 3 -5 -OMe-1-PYR], [ BK164; 3-Me-4-OCF 3 -5-OEt-1-PYR], [BK165; 3-Me-4-OCF 3 -5-CN-1-PYR], [BK166; 3-Me-4 -OCF 3 -5-CHF 2 -1-PYR], [BK167; 3-Me-4-OCF 3 -5-CF 3 -1-PYR], [BK168; 3-Me _{-4-OCF 3 -5-OCHF 2} -1-PYR], [BK169; 3-Me-4-OCF 3 -5-OCF 3 -1-PYR], [BK170; 1-PYR], [BK171; 1 -Me-3-PYR], [BK 172; 1-Me-4-F-3-PYR], [BK 173; 1-Me-4-Cl-3-PYR], [BK 174; 1-Me-4-Br -3-PYR], [BK175; 1-Me-4-Me-3-PYR], [BK176; 1-Me-4-Et-3-PYR], [BK177; 1-Me-4-OMe-3 -PYR], [BK178; 1- Me-4-OEt-3-PYR], [BK179; 1-Me-4-CN-3-PYR], [BK180; 1-Me-4-CHF 2 -3- PYR], [BK181; 1- Me-4-CF 3 -3-PYR], [BK182; 1-Me-4-OCHF 2 -3-PYR], [BK183; 1-Me-4-OCF 3 -3 -PYR], [BK184; 1-Me-5-F-3-PYR], [BK185; 1-Me-5-Cl-3-PYR], [BK186; 1-Me-5-Br-3-PYR ], [BK187; 1-Me-5-Me-3-PYR], [BK188; 1-Me-5-Et-3-PYR], [BK189; 1-Me-5-OMe-3-PYR], [BK190; 1-Me-5 -OEt-3-PYR], [BK191; 1-Me-5-CN-3-PYR], [BK192; 1-Me-5-CHF 2 -3-PYR], [ BK193; 1-Me-5- CF 3 -3-PYR], [BK194; 1-Me-5-OCHF 2 -3-PYR], [BK195; 1-Me-5-OCF 3 -3-PYR], [BK 196; 1-Me-4-F-5-F-3-PYR], [BK 197; 1-Me-4-F-5-Cl-3-PY R], [BK 198; 1-Me-4-F-5-Br-3-PYR], [BK199; 1-Me-4-F-5-Me-3-PYR], [BK200; 1-Me- 4-F-5-Et-3-PYR],

[BK201; 1-Me-4-F-5-OMe-3-PYR], [BK202; 1-Me-4-F-5-OEt-3-PYR], [BK203; 1-Me-4-F -5-CN-3-PYR], [BK 204; 1-Me-4-F-5-CHF ₂ -3-PYR], [BK 205; 1-Me-4-F-5-CF ₃ -3-PYR ], [BK206; 1-Me -4-F-5-OCHF 2 -3-PYR], [BK207; 1-Me-4-F-5-OCF 3 -3-PYR], [BK208; 1-Me -4-Cl-5-F-3-PYR], [BK209; 1-Me-4-Cl-5-Cl-3-PYR], [BK210; 1-Me-4-Cl-5-Br-3 -PYR], [BK211; 1-Me-4-Cl-5-Me-3-PYR], [BK212; 1-Me-4-Cl-5-Et-3-PYR], [BK213; 1-Me -4-Cl-5-OMe-3-PYR], [BK 214; 1-Me-4-Cl-5-OEt-3-PYR], [BK 215; 1-Me-4-Cl-5-CN-3 -PYR], [BK216; 1- Me-4-Cl-5-CHF 2 -3-PYR], [BK217; 1-Me-4-Cl-5-CF 3 -3-PYR], [BK218; 1 -Me-4-Cl-5-OCHF ₂ -3-PYR !, [BK 219; 1-Me -4-Cl -5-OCF ₃ -3-PYR], [BK 220; 1-Me-4-Br-5 -F-3-PYR], [BK221; 1-Me-4-Br-5-Cl-3-PYR], [BK222; 1-Me-4-Br-5-Br-3-PYR], [BK223] 1-Me-4-Br-5-Me-3-PYR], [BK224; 1-Me-4-Br-5-Et-3-PYR], [BK225; 1-Me-4-Br-5 -OMe-3-PYR], [BK226; 1-Me-4-Br-5-OEt-3-PYR], [BK227; 1-Me-4-Br-5-CN-3-PYR], [BK228] ; 1-Me-4-Br -5-CHF 2 -3-PYR], [BK229; 1-Me-4-Br-5-CF 3 -3-PYR], [BK230; 1-Me-4-Br -5-OCHF ₂ -3-PYR !, [BK 231; 1-Me-4-Br-5-OCF ₃ -3-PYR], [BK 232; 1-Me-4-Me-5-F-3-PYR ], [BK 233; 1-Me-4-Me-5-Cl-3-PYR] , [BK234; 1-Me-4-Me-5-Br-3-PYR], [BK235; 1-Me-4-Me-5-Me-3-PYR], [BK236; 1-Me-4- 4 Me-5-Et-3-PYR], [BK 237; 1-Me-4-Me-5-OMe-3-PYR], [BK 238; 1-Me-4-Me-5-OEt-3-PYR] , [BK 239; 1-Me-4-Me-5-CN-3-PYR], [BK 240; 1-Me-4-Me-5-CHF ₂ -3-PYR], [BK 241; 1-Me-4 _{-Me-5-CF 3 -3-} PYR], [BK242; 1-Me-4-Me-5-OCHF 2 -3-PYR], [BK243; 1-Me-4-Me-5-OCF 3 - 3-PYR], [BK244; 1-Me-4-Et-5-F-3-PYR], [BK245; 1-Me-4-Et-5-Cl-3-PYR], [BK246; 1- Me-4-Et-5-Br-3-PYR], [BK 247; 1-Me-4-Et-5-Me-3-PYR], [BK 248; 1-Me-4-Et-5-Et- 3-PYR], [BK 249; 1-Me-4-Et-5-OMe-3-PYR], [BK 250; 1-Me-4-Et-5-OEt-3-PYR], [BK 251; Me-4-Et-5-CN-3-PYR], [BK 252; 1-Me-4-Et-5-CHF ₂ -3-PYR], [BK 253; 1-Me-4-Et-5-CF _{3 -3-PYR], [BK254} ; 1-Me-4-Et-5-OCHF 2 -3-PYR], [BK255; 1-Me-4-Et-5-OCF 3 -3-PYR], [ BK 256; 1-Me-4-OMe-5-F-3-PYR], [BK 257; 1-Me-4-OMe-5-Cl-3-PYR], [BK 258; 1-Me-4-OMe- 5-Br-3-PYR], [BK 259; 1-Me-4-OMe-5-Me-3-PYR], [BK 260; 1-Me-4-OMe-5-Et-3-PYR], [BK BK 261; 1-Me-4-OMe-5-OMe-3-PYR], [BK 262; 1-Me-4-OMe-5-OEt-3-PYR], [BK 263; 1-Me-4-OMe- 5-CN-3-PYR], [BK 264; 1-Me-4-OMe-5-CHF ₂ -3-PYR], [BK 265; 1-Me-4-OMe-5-CF ₃ -3-PYR] , [BK 266; 1-Me-4-OMe- _{5-OCHF 2 -3-PYR]} , [BK267; 1-Me-4-OMe-5-OCF 3 -3-PYR], [BK268; 1-Me-4-OEt-5-F-3-PYR] , [BK 269; 1-Me-4-OEt-5-Cl-3-PYR], [BK 270; 1-Me-4-OEt-5-Br-3-PYR], [BK 271; 1-Me-4- 4 OEt-5-Me-3-PYR], [BK 272; 1-Me-4-OEt-5-Et-3-PYR], [BK 273; 1-Me-4-OEt-5-OMe-3-PYR] , [BK 274; 1-Me-4-OEt-5-OEt-3-PYR], [BK 275; 1-Me-4-OEt-5-CN-3-PYR], [BK 276; 1-Me-4- _{OEt-5-CHF 2 -3-} PYR], [BK277; 1-Me-4-OEt-5-CF 3 -3-PYR], [BK278; 1-Me-4-OEt-5-OCHF 2 -3 -PYR], [BK279; 1- Me-4-OEt-5-OCF 3 -3-PYR], [BK280; 1-Me-4-CN-5-F-3-PYR], [BK281; 1- Me-4-CN-5-Cl-3-PYR], [BK282; 1-Me-4-CN-5-Br-3-PYR], [BK 283; 1-Me-4-CN-5-Me- 3-PYR], [BK284; 1-Me-4-CN-5-Et-3-PYR], [BK 285; 1-Me-4-CN-5-OMe-3-PYR], [BK 286; Me-4-CN-5-OEt-3-PYR], [BK 287; 1-Me-4-CN-5-CN-3-PYR], [BK 288; 1-Me-4-CN-5-CHF ₂ -3-PYR], [BK 289; 1-Me-4-CN-5-CF ₃ -3-PYR], [BK 290; 1-Me-4-CN-5-OCHF ₂ -3-PYR], [BK 291 ; 1-Me-4-CN -5-OCF 3 -3-PYR], [BK292; 1-Me-4-CHF 2 -5-F-3-PYR], [BK293; 1-Me-4-CHF _{2 -5-Cl-3-PYR} ], [BK294; 1-Me-4-CHF 2 -5-Br-3-PYR], [BK295; 1-Me-4-CHF 2 -5-Me-3- PYR], [BK 296; 1-Me-4-CHF ₂ -5-Et-3-PYR], [BK 297; 1-Me-4-CHF ₂ -5-OMe-3-PYR], [BK 298; 1- _{Me-4-CHF 2 -5-} OEt-3-PYR], [BK299; 1-Me-4-CHF 2 -5-CN-3-PYR], [BK300; 1-Me-4-CHF 2 -5 -CHF ₂ -3-PYR],

[BK301; 1-Me-4 -CHF 2 -5-CF 3 -3-PYR], [BK302; 1-Me-4-CHF 2 -5-OCHF 2 -3-PYR], [BK303; 1-Me _{-4-CHF 2 -5-OCF 3} -3-PYR], [BK304; 1-Me-4-CF 3 -5-F-3-PYR], [BK305; 1-Me-4-CF 3 -5 -Cl-3-PYR], [ BK306; 1-Me-4-CF 3 -5-Br-3-PYR], [BK307; 1-Me-4-CF 3 -5-Me-3-PYR], [BK308; 1-Me-4 -CF 3 -5-Et-3-PYR], [bK309; 1-Me-4-CF 3 -5-OMe-3-PYR], [BK310; 1-Me-4 _{-CF 3 -5-OEt-3-} PYR], [BK311; 1-Me-4-CF 3 -5-CN-3-PYR], [BK312; 1-Me-4-CF 3 -5-CHF 2 -3-PYR], [BK313; 1-Me-4-CF 3 -5-CF 3 -3-PYR], [BK314; 1-Me-4-CF 3 -5-OCHF 2 -3-PYR], [BK315; 1-Me-4 -CF 3 -5-OCF 3 -3-PYR], [BK316; 1-Me-4-OCHF 2 -5-F-3-PYR], [BK317; 1-Me- _{4-OCHF 2 -5-Cl-} 3-PYR], [BK318; 1-Me-4-OCHF 2 -5-Br-3-PYR], [BK319; 1-Me-4-OCHF 2 -5-Me -3-PYR], [BK320; 1-Me-4-OCHF 2 -5-Et-3-PYR], [BK321; 1-Me-4-OCHF 2 -5-OMe-3-PYR], [BK322 ; 1-Me-4-OCHF 2 -5-OEt-3-PYR], [BK323; 1-Me-4-OCHF 2 -5-CN-3-PYR], [BK324; 1-Me-4-OCHF ₂ -5-CHF ₂ -3-PYR !, [BK 325; 1-Me 4-OCHF ₂ -5-CF ₃ -3-PYR], [BK 326; 1-Me-4-OCHF ₂ -5-OCHF ₂ -3-PYR], [BK 327; 1-Me-4-OCHF ₂ -5-OCF ₃ -3-PYR], [BK 328; 1-Me-4-OCF ₃ -5-F-3-PYR], [BK BK329; 1-Me-4- OCF 3 -5-Cl-3-PYR ], [BK330; 1-Me -4-OCF 3 -5-Br-3-PYR], [BK331; 1-Me-4-OCF 3 -5-Me-3-PYR], [BK332; 1-Me _{-4-OCF 3 -5-Et-} 3-PYR], [BK333; 1-Me-4-OCF 3 -5-OMe-3-PYR], [BK334; 1-Me-4-OCF 3 -5- OEt-3-PYR], [ BK335; 1-Me-4-OCF 3 -5-CN-3-PYR], [BK336; 1-Me-4-OCF 3 -5-CHF 2 -3-PYR], [BK337; 1-Me-4 -OCF 3 -5-CF 3 -3-PYR], [BK338; 1-Me-4-OCF 3 -5-OCHF 2 -3-PYR], [BK339; 1-Me _{-4-OCF 3 -5-OCF 3} -3-PYR], [BK340; 2-Me-3-PYR], [BK341; 2-Me-4-F-3-PYR], [BK342; 2-Me -4-Cl-3-PYR !, [BK 343; 2-Me-4-Br-3-PYR], [BK 344; 2-Me-4-Me-3-PYR], [BK 345; 2-Me-4 -Et-3-PYR], [BK346; 2-Me-4-OMe-3-PYR], [BK347; 2-Me-4-OEt-3-PYR], [BK 348; 2-Me-4-CN -3-PYR], [BK349; 2-Me-4-CHF 2 -3-PYR], [BK350; 2-Me-4-CF 3 -3-PYR], [BK351; 2-Me-4-OCHF _{2 -3-PYR], [BK352} ; 2-Me-4-OCF 3 -3-PYR], [BK353; 2-Me-5-F-3-PYR], [BK354; 2-Me-5-Cl -3-PYR], [BK 355; 2-Me-5-Br-3-PYR], [BK 356; 2-Me-5-Me-3-PYR], [BK 357; 2-Me-5-Et-3 -PYR], [BK 358; 2-Me-5-OMe-3-PYR], [BK 359; 2-Me-5-OEt-3-PYR], [BK 360; 2-Me-5-CN-3-PYR ], [BK361; 2-Me -5-CHF 2 -3-PYR], [BK362; 2-Me-5-CF 3 -3-PYR], [BK363; 2-Me-5-OCHF 2 -3- PYR], [BK364; 2- Me-5-OCF 3 -3-PYR], [BK365; 2-Me-4-F-5-F-3 -PYR], [BK 366; 2-Me-4-F-5-Cl-3-PYR], [BK 367; 2-Me-4-F-5-Br-3-PYR], [BK 368; 2-Me -4-F-5-Me-3-PYR], [BK369; 2-Me-4-F-5-Et-3-PYR], [BK370; 2-Me-4-F-5-OMe-3 -PYR], [BK 371; 2-Me-4-F-5-OEt-3-PYR], [BK 372; 2-Me-4-F-5-CN-3-PYR], [BK 373; 2-Me _{-4-F-5-CHF 2} -3-PYR], [BK374; 2-Me-4-F-5-CF 3 -3-PYR], [BK375; 2-Me-4-F-5-OCHF _2-3 -PYR], [BK 376; 2-Me-4-F-5-OCF ₃ -3-PYR], [BK 377; 2-Me-4-Cl-5-F-3-PYR], [BK 378 2-Me-4-Cl-5-Cl-3-PYR], [BK379; 2-Me-4-Cl-5-Br-3-PYR], [BK380; 2-Me-4-Cl-5 -Me-3-PYR], [BK 381; 2-Me-4-Cl-5-Et-3-PYR], [BK 382; 2-Me-4-Cl-5-OMe-3-PYR], [BK 383] 2-Me-4-Cl-5-OEt-3-PYR], [BK 384; 2-Me-4-Cl-5-CN-3-PYR], [BK 385; 2-Me-4-Cl-5 _{-CHF 2 -3-PYR], [} BK386; 2-Me-4-Cl-5-CF 3 -3-PYR], [BK387; 2-Me-4-Cl-5-OCHF 2 -3-PYR] , [BK388; 2-Me- 4-Cl-5-OCF 3 -3-PYR], [BK389; 2-Me-4-Br-5-F-3-PYR], [BK390; 2-Me-4 -Br-5-Cl-3-PYR], [BK 391; 2-Me-4-Br-5-Br-3-PYR], [BK 392; 2-Me-4-Br-5-Me-3-PYR ], [BK 393; 2-Me-4-Br-5-Et-3-PYR], [BK 394; 2-Me-4-Br-5-OMe-3-PYR], [BK 395; 2-Me-4 -Br-5-OEt-3-PYR], [BK 396; 2-Me-4-Br-5-CN-3-PYR], [BK 397; 2-Me-4-Br-5-CHF ₂ -3- PYR], [BK 398; 2-Me-4-Br-5-CF ₃ -3-PYR], [BK 39 9; 2-Me-4- Br-5-OCHF 2 -3-PYR], [BK400; 2-Me-4-Br-5-OCF 3 -3-PYR],

[BK 401; 2-Me-4-Me-5-F-3-PYR], [BK 402; 2-Me-4-Me-5-Cl-3-PYR], [BK 403; 2-Me-4-Me -5-Br-3-PYR], [BK 404; 2-Me-4-Me-5-Me-3-PYR], [BK 405; 2-Me-4-Me-5-Et-3-PYR], [BK406; 2-Me-4-Me-5-OMe-3-PYR], [BK407; 2-Me-4-Me-5-OEt-3-PYR], [BK408; 2-Me-4-Me -5-CN-3-PYR], [BK 409; 2-Me-4-Me-5-CHF ₂ -3-PYR], [BK 410; 2-Me-4-Me-5-CF ₃ -3-PYR ], [BK411; 2-Me -4-Me-5-OCHF 2 -3-PYR], [BK412; 2-Me-4-Me-5-OCF 3 -3-PYR], [BK413; 2-Me -4-Et-5-F-3-PYR], [BK 414; 2-Me-4-Et-5-Cl-3-PYR], [BK 415; 2-Me-4-Et-5-Br-3 -PYR], [BK 416; 2-Me-4-Et-5-Me-3-PYR], [BK 417; 2-Me-4-Et-5-Et-3-PYR], [BK 418; 2-Me -4-Et-5-OMe-3-PYR], [BK 419; 2-Me-4-Et-5-OEt-3-PYR], [BK 420; 2-Me-4-Et-5-CN-3 -PYR], [BK421; 2- Me-4-Et-5-CHF 2 -3-PYR], [BK422; 2-Me-4-Et-5-CF 3 -3-PYR], [BK423; 2 -Me-4-Et-5- OCHF 2 -3-PYR], [BK424; 2-Me-4-Et-5-OCF 3 -3-PYR], [BK425; 2-Me-4-OMe-5 -F-3-PYR], [BK 426; 2-Me-4-OMe-5-Cl-3-PYR], [BK 427; 2-Me-4-OMe-5-Br-3-PYR], [BK 428] 2-Me-4-OMe-5-Me-3-PYR], [BK 429; 2-Me-4-OMe-5-Et-3-PYR], [BK 430; 2-Me-4-OMe-5 -OMe-3-PYR], [BK 431; 2-Me-4-OMe-5-OEt-3-PYR], [BK 432; 2-Me-4-OMe-5-CN-3-PYR], [BK 433] 2-Me-4-OMe-5-CHF ₂ -3- PYR], [BK434; 2- Me-4-OMe-5-CF 3 -3-PYR], [BK435; 2-Me-4-OMe-5-OCHF 2 -3-PYR], [BK436; 2- Me-4-OMe-5- OCF 3 -3-PYR], [BK437; 2-Me-4-OEt-5-F-3-PYR], [BK438; 2-Me-4-OEt-5-Cl -3-PYR !, [BK 439; 2-Me-4-OEt-5-Br-3-PYR], [BK 440; 2-Me-4-OEt-5-Me-3-PYR], [BK 441; -Me-4-OEt-5-Et-3-PYR], [BK 442; 2-Me-4-OEt-5-OMe-3-PYR], [BK 443; 2-Me-4-OEt-5-OEt -3-PYR !, [BK 444; 2-Me-4-OEt-5-CN-3-PYR], [BK 445; 2-Me-4-OEt-5-CHF ₂ -3-PYR], [BK 446; 2-Me-4-OEt- 5-CF 3 -3-PYR], [BK447; 2-Me-4-OEt-5-OCHF 2 -3-PYR], [BK448; 2-Me-4-OEt- _{5-OCF 3 -3-PYR]} , [BK449; 2-Me-4-CN-5-F-3-PYR], [BK450; 2-Me-4-CN-5-Cl-3-PYR], [BK 451; 2-Me-4-CN-5-Br-3-PYR], [BK 452: 2-Me-4-CN-5-Me-3-PYR], [BK 453; 2-Me-4-CN -5-Et-3-PYR], [BK 454; 2-Me-4-CN-5-OMe-3-PYR], [BK 455; 2-Me-4-CN-5-OEt-3-PYR], [BK 456; 2-Me-4-CN-5-CN-3-PYR], [BK 457; 2-Me-4-CN-5-CHF ₂ -3-PYR], [BK 458; _{CN-5-CF 3 -3-} PYR], [BK459; 2-Me-4-CN-5-OCHF 2 -3-PYR], [BK460; 2-Me-4-CN-5-OCF 3 -3 -PYR], [BK461; 2- Me-4-CHF 2 -5-F-3-PYR], [BK462; 2-Me-4-CHF 2 -5-Cl-3-PYR], [BK463; 2 _{-Me-4-CHF 2 -5-} Br-3-PYR], [BK464; 2-Me-4-CHF 2 -5-Me-3-PYR], [BK465; 2-Me-4-CHF 2 -5-Et-3-PYR], [BK 466; 2-Me-4-CHF ₂ -5-OMe-3-PYR], [BK 467; 2-Me-4-CHF ₂ -5-OEt-3-PYR ], [BK468; 2-Me -4-CHF 2 -5-CN-3-PYR], [BK469; 2-Me-4-CHF 2 -5-CHF 2 -3-PYR], [BK470; 2- _{Me-4-CHF 2 -5-} CF 3 -3-PYR], [BK471; 2-Me-4-CHF 2 -5-OCHF 2 -3-PYR], [BK472; 2-Me-4-CHF 2 _{-5-OCF 3 -3-PYR]} , [BK473; 2-Me-4-CF 3 -5-F-3-PYR], [BK474; 2-Me-4-CF 3 -5-Cl-3- PYR], [BK475; 2- Me-4-CF 3 -5-Br-3-PYR], [BK476; 2-Me-4-CF 3 -5-Me-3-PYR], [BK477; 2- _{Me-4-CF 3 -5-} Et-3-PYR], [BK478; 2-Me-4-CF 3 -5-OMe-3-PYR], [BK479; 2-Me-4-CF 3 -5 -OEt-3-PYR], [ BK480; 2-Me-4-CF 3 -5-CN-3-PYR], [BK481; 2-Me-4-CF 3 -5-CHF 2 -3-PYR] , [BK482; 2-Me- 4-CF 3 -5-CF 3 -3-PYR], [BK483; 2-Me-4-CF 3 -5-OCHF 2 -3-PYR], [BK484; 2- _{Me-4-CF 3 -5-} OCF 3 -3-PYR], [BK485; 2-Me-4-OCHF 2 -5-F-3-PYR], [BK486; 2-Me-4-OCHF 2 - 5-Cl-3-PYR] , [BK487; 2-Me-4-OCHF 2 -5-Br-3-PYR], [BK488; 2-Me-4-OCHF 2 -5-Me-3-PYR] , [BK 489; 2-Me-4-OCHF ₂ -5-Et-3-PYR], [BK 490; 2-Me-4-OCHF ₂ -5-OMe-3-PYR], [BK 491; _{4-OCHF 2 -5-OEt-} 3-PYR], [BK492; 2-Me-4-OCHF 2 -5-CN-3-PYR], [BK493; 2-Me-4-OCHF 2 -5-CHF ₂ -3-PYR], [BK 494; 2-Me-4-OCHF ₂ -5-CF _{3 -3-PYR], [BK495} ; 2-Me-4-OCHF 2 -5-OCHF 2 -3-PYR], [BK496; 2-Me-4-OCHF 2 -5-OCF 3 -3-PYR] , [BK497; 2-Me- 4-OCF 3 -5-F-3-PYR], [BK498; 2-Me-4-OCF 3 -5-Cl-3-PYR], [BK499; 2-Me- _{4-OCF 3 -5-Br-} 3-PYR], [BK500; 2-Me-4-OCF 3 -5-Me-3-PYR],

[BK501; 2-Me-4 -OCF 3 -5-Et-3-PYR], [BK502; 2-Me-4-OCF 3 -5-OMe-3-PYR], [BK503; 2-Me-4 _{-OCF 3 -5-OEt-3-} PYR], [BK504; 2-Me-4-OCF 3 -5-CN-3-PYR], [BK505; 2-Me-4-OCF 3 -5-CHF 2 -3-PYR], [BK506; 2-Me-4-OCF 3 -5-CF 3 -3-PYR], [BK507; 2-Me-4-OCF 3 -5-OCHF 2 -3-PYR], [BK508; 2-Me-4 -OCF 3 -5-OCF 3 -3-PYR], [BK509; 1-Me-4-PYR], [BK510; 1-Me-3-F-4-PYR], [BK511; 1-Me-3-Cl-4-PYR], [BK512; 1-Me-3-Br-4-PYR], [BK513; 1-Me-3-Me-4-PYR], [BK514] 1-Me-3-Et-4-PYR], [BK515; 1-Me-3-OMe-4-PYR], [BK516; 1-Me-3-OEt-4-PYR], [BK517; 1 -Me-3-CN-4- PYR], [BK518; 1-Me-3-CHF 2 -4-PYR], [BK519; 1-Me-3-CF 3 -4-PYR], [BK520; 1 -Me-3-OCHF ₂ -4-PYR], [BK 521; 1-Me-3-OCF ₃ -4-PYR], [BK 522; 1-Me-5-F-4-PYR], [BK 523; 1 -Me-5-Cl-4-PYR], [BK 524; 1-Me-5-Br-4-PYR], [BK 525; 1-Me-5-Me-4-PYR], [BK 526; 1-Me -5-Et-4-PYR], [BK 527; 1-Me-5-OMe-4-PYR], [BK 528; 1-Me-5-OEt-4-PYR], [BK 529; 1-Me-5 -CN-4-PYR], [ BK530; 1-Me-5-CHF 2 -4-PYR], [BK531; 1-Me-5-CF 3 -4-PYR], [BK532; 1-Me-5 -OCHF ₂ -4-PYR], [BK 533; 1-Me-5-OCF ₃ -4-PYR], [BK 534; 1-Me-3-F-5-F-4-PYR], [BK 535; 1 -Me-3-F-5-Cl-4-PYR], [BK 536; 1-Me-3-F-5-Br-4-PYR], [BK 537] 1-Me-3-F-5-Me-4-PYR], [BK 538; 1-Me-3-F-5-Et-4-PYR], [BK 539; 1-Me-3-F-5 -OMe-4-PYR], [BK 540; 1-Me-3-F-5-OEt-4-PYR], [BK 541; 1-Me-3-F-5-CN-4-PYR], [BK 542] 1-Me-3-F-5-CHF ₂ -4-PYR !, [BK 543; 1-Me-3-F-5-CF ₃ -4-PYR], [BK 544; 1-Me-3-F -5-OCHF ₂ -4-PYR], [BK 545; 1-Me-3-F-5-OCF ₃ -4-PYR], [BK 546; 1-Me-3-Cl-5-F-4-PYR ], [BK 547; 1-Me-3-Cl-5-Cl-4-PYR], [BK 548; 1-Me-3-Cl-5-Br-4-PYR], [BK 549; 1-Me-3] -Cl-5-Me-4-PYR], [BK 550; 1-Me-3-Cl-5-Et-4-PYR], [BK 551; 1-Me-3-Cl-5-OMe-4-PYR ], [BK 552; 1-Me-3-Cl-5-OEt-4-PYR], [BK 553; 1-Me-3-Cl-5-CN-4-PYR], [BK 554; 1-Me-3 -Cl-5-CHF ₂ -4-PYR], [BK 555; 1-Me-3-Cl-5-CF ₃ -4-PYR], [BK 556; 1-Me-3-Cl-5-OCHF _2- 4-PYR], [BK557; 1-Me-3-Cl-5-OCF 3 -4-PYR], [BK558; 1-Me-3-Br-5-F-4-PYR], [BK559; 1 -Me-3-Br-5-Cl-4-PYR], [BK 560; 1-Me-3-Br-5-Br-4-PYR], [BK 561; 1-Me-3-Br-5-Me -4-PYR !, [BK 562; 1-Me-3-Br-5-Et-4-PYR], [BK 563; 1-Me-3-Br-5-OMe-4-PYR], [BK 564; 1 -Me-3-Br-5-OEt-4-PYR], [BK 565; 1-Me-3-Br-5-CN-4-PYR], [BK 566; 1-Me-3-Br-5-CHF ₂ -4-PYR], [BK 567; 1-Me-3-Br-5-CF ₃ -4-PYR], [BK 568; 1-Me-3-Br-5-OCHF ₂ -4-PYR], BK569; 1-Me-3- Br-5-OCF 3 -4-PYR], [BK570 1-Me-3-Me-5-F-4-PYR], [BK 571; 1-Me-3-Me-5-Cl-4-PYR], [BK 572; 1-Me-3-Me-5 -Br-4-PYR], [BK 573; 1-Me-3-Me-5-Me-4-PYR], [BK 574; 1-Me-3-Me-5-Et-4-PYR], [BK 575] 1-Me-3-Me-5-OMe-4-PYR], [BK 576; 1-Me-3-Me-5-OEt-4-PYR], [BK577; 1-Me-3-Me-5 -CN-4-PYR], [BK 578; 1-Me-3-Me-5-CHF ₂ -4-PYR], [BK 579; 1-Me-3-Me-5-CF ₃ -4-PYR], [BK 580; 1-Me-3-Me-5-OCHF ₂ -4-PYR], [BK 581; 1-Me-3-Me-5-OCF ₃ -4-PYR], [BK 582; 1-Me-3 -Et-5-F-4-PYR], [BK 583; 1-Me-3-Et-5-Cl-4-PYR], [BK 584; 1-Me-3-Et-5-Br-4-PYR ], [BK 585; 1-Me-3-Et-5-Me-4-PYR], [BK 586; 1-Me-3-Et-5-Et-4-PYR], [BK 587; 1-Me-3 -Et-5-OMe-4-PYR], [BK 588; 1-Me-3-Et-5-OEt-4-PYR], [BK 589; 1-Me-3-Et-5-CN-4-PYR ], [BK 590; 1-Me-3-Et-5-CHF ₂ -4-PYR], [BK 591; 1-Me-3-Et-5-CF ₃ -4-PYR], [BK 592; 1-Me -3-Et-5-OCHF ₂ -4-PYR !, [BK 593; 1-Me-3-Et-5-OCF ₃ -4-PYR], [BK 594; 1-Me-3-OMe-5-F -4-PYR], [BK 595; 1-Me-3-OMe-5-Cl-4-PYR], [BK 596; 1-Me-3-OMe-5-Br-4-PYR], [BK 597; 1 -Me-3-OMe-5-Me-4-PYR], [BK 598; 1-Me-3-OMe-5-Et-4-PYR], [BK 599; 1-Me-3-OMe-5-OMe -4-PYR], [BK600; 1-Me-3-OMe-5-OEt-4-PYR],

[BK 601; 1-Me-3-OMe-5-CN-4-PYR], [BK 602; 1-Me-3-OMe-5-CHF ₂ -4-PYR], [BK 603; 1-Me-3- _{OMe-5-CF 3 -4-} PYR], [BK604; 1-Me-3-OMe-5-OCHF 2 -4-PYR], [BK605; 1-Me-3-OMe-5-OCF 3 -4 -PYR], [BK 606; 1-Me-3-OEt-5-F-4-PYR], [BK 607; 1-Me-3-OEt-5-Cl-4-PYR], [BK 608; 1-Me -3-OEt-5-Br-4-PYR], [BK 609; 1-Me-3-OEt-5-Me-4-PYR], [BK 610; 1-Me-3-OEt-5-Et-4 -PYR], [BK611; 1-Me-3-OEt-5-OMe-4-PYR], [BK612; 1-Me-3-OEt-5-OEt-4-PYR], [BK613; 1-Me -3-OEt-5-CN-4-PYR], [BK 614; 1-Me-3-OEt-5-CHF ₂ -4-PYR], [BK 615; 1-Me-3-OEt-5-CF ₃ -4-PYR], [BK 616; 1-Me-3-OEt-5-OCHF ₂ -4-PYR], [BK 617; 1-Me-3-OEt-5-OCF ₃ -4-PYR], [BK 618] 1-Me-3-CN-5-F-4-PYR !, [BK 619; 1-Me-3-CN-5-Cl-4-PYR], [BK 620; 1-Me-3-CN-5; -Br-4-PYR], [BK 621; 1-Me-3-CN-5-Me-4-PYR], [BK 622; 1-Me-3-CN-5-Et-4-PYR], [BK 623] 1-Me-3-CN-5-OMe-4-PYR], [BK 624; 1-Me-3-CN-5-OEt-4-PYR], [BK 625; 1-Me-3-CN-5; -CN-4-PYR], [BK 626; 1-Me-3-CN-5-CHF ₂ -4-PYR], [BK 627; 1-Me-3-CN-5-CF ₃ -4-PYR], [BK 628; 1-Me-3-CN-5-OCHF ₂ -4-PYR], [BK 629; 1-Me-3-CN-5-OCF ₃ -4-PYR], [BK 630; 1-Me-3 _{-CHF 2 -5-F-4-} PYR], [BK631; 1-Me-3-CHF 2 -5-Cl-4-PYR], [BK632; 1-Me-3-CHF 2 -5-Br- Four -PYR], [BK 633; 1-Me-3-CHF ₂ -5-Me-4-PYR], [BK 634; 1-Me-3-CHF ₂ -5-Et-4-PYR], [BK 635; 1 _{-Me-3-CHF 2 -5-} OMe-4-PYR], [BK636; 1-Me-3-CHF 2 -5-OEt-4-PYR], [BK637; 1-Me-3-CHF 2 - 5-CN-4-PYR, [BK 638; 1-Me-3-CHF ₂ -5-CHF ₂ -4-PYR], [BK 639; 1-Me-3-CHF ₂ -5-CF ₃ -4- PYR], [BK 640; 1-Me-3-CHF ₂ -5-OCHF ₂ -4-PYR], [BK 641; 1 Me-3-CHF ₂ -5-OCF ₃ -4-PYR], [BK 642; _{1-Me-3-CF 3} -5-F-4-PYR], [BK643; 1-Me-3-CF 3 -5-Cl-4-PYR], [BK644; 1-Me-3-CF 3 -5-Br-4-PYR], [BK 645; 1-Me-3-CF ₃ -5-Me-4-PYR], [BK 646; 1-Me-3-CF ₃ -5-Et-4-PYR ], [BK647; 1-Me -3-CF 3 -5-OMe-4-PYR], [BK648; 1-Me-3-CF 3 -5-OEt-4-PYR], [BK649; 1-Me -3-CF ₃ -5-CN-4-PYR !, [BK 650; 1-Me-3-CF ₃ -5-CHF ₂ -4-PYR], [BK 651; 1-Me-3-CF ₃ -5 _{-CF 3 -4-PYR], [} BK652; 1-Me-3-CF 3 -5-OCHF 2 -4-PYR], [BK653; 1-Me-3-CF 3 -5-OCF 3 -4- PYR], [BK 654; 1-Me-3-OCHF ₂ -5-F-4-PYR], [BK 655; 1-Me-3-OCHF ₂ -5-Cl-4-PYR], [BK 656; 1- _{Me-3-OCHF 2 -5-} Br-4-PYR], [BK657; 1-Me-3-OCHF 2 -5-Me-4-PYR], [BK658; 1-Me-3-OCHF 2 -5 -Et-4-PYR], [ BK659; 1-Me-3-OCHF 2 -5-OMe-4-PYR], [BK660; 1-Me-3-OCHF 2 -5-OEt-4-PYR], [BK 661; 1-Me-3-OCHF ₂ -5-CN-4-PYR], [BK 66 2; 1-Me-3-OCHF ₂ -5-CHF ₂ -4-PYR !, [BK 663; 1-Me-3-OCHF ₂ -5-CF ₃ -4-PYR], [BK 664; 1-Me- _{3-OCHF 2 -5-OCHF 2} -4-PYR], [BK665; 1-Me-3-OCHF 2 -5-OCF 3 -4-PYR], [BK666; 1-Me-3-OCF 3 -5 -F-4-PYR], [ BK667; 1-Me-3-OCF 3 -5-Cl-4-PYR], [BK668; 1-Me-3-OCF 3 -5-Br-4-PYR], [BK669; 1-Me-3 -OCF 3 -5-Me-4-PYR], [BK670; 1-Me-3-OCF 3 -5-Et-4-PYR], [BK671; 1-Me-3 _{-OCF 3 -5-OMe-4-} PYR], [BK672; 1-Me-3-OCF 3 -5-OEt-4-PYR], [BK673; 1-Me-3-OCF 3 -5-CN- 4-PYR], [BK 674; 1-Me-3-OCF ₃ -5-CHF ₂ -4-PYR], [BK 675; 1-Me-3-OCF ₃ -5-CF ₃ -4-PYR], [BK BK676; 1-Me-3- OCF 3 -5-OCHF 2 -4-PYR], [BK677; 1-Me-3-OCF 3 -5-OCF 3 -4-PYR], [BK678; 2-Me- 4-PYR], [BK 679; 2-Me-3-F-4-PYR], [BK 680; 2-Me-3-Cl-4-PYR], [BK 681; 2-Me-3-Br-4- PYR], [BK 682; 2-Me-3-Me-4-PYR], [BK 683; 2-Me-3-Et-4-PYR], [BK 684; 2-Me-3-OMe-4-PYR] , [BK 685; 2-Me-3-OEt-4-PYR], [BK 686; 2-Me-3-CN-4-PYR], [BK 687; 2-Me-3-CHF ₂ -4-PYR], [BK688; 2-Me-3 -CF 3 -4-PYR], [BK689; 2-Me-3-OCHF 2 -4-PYR], [BK690; 2-Me-3-OCF 3 -4-PYR] , [BK691; 2-Me-5-F-4-PYR], [BK692; 2-Me-5-Cl-4-PYR], [BK693; 2-Me-5-Br-4-PYR], [BK692; BK694; 2-Me-5-Me-4-PYR], [BK 695; 2-Me-5-Et-4-PY R], [BK 696; 2-Me-5-OMe-4-PYR], [BK 697; 2-Me-5-OEt-4-PYR], [BK 698; 2-Me-5-CN-4-PYR] , [BK 699; 2-Me-5-CHF ₂ -4-PYR], [BK 700; 2-Me-5-CF ₃ -4-PYR],

[BK 701; 2-Me-5-OCHF ₂ -4-PYR], [BK 702; 2-Me-5-OCF ₃ -4-PYR], [BK 703; 2-Me-3-F-5-F-4 -PYR], [BK 704; 2-Me-3-F-5-Cl-4-PYR], [BK 705; 2-Me-3-F-5-Br-4-PYR], [BK 706; 2-Me -3-F-5-Me-4-PYR], [BK 707; 2-Me-3-F-5-Et-4-PYR], [BK 708; 2-Me-3-F-5-OMe-4 -PYR], [BK 709; 2-Me-3-F-5-OEt-4-PYR], [BK 710; 2-Me-3-F-5-CN-4-PYR], [BK 711; 2-Me -3-F-5-CHF ₂ -4-PYR !, [BK 712; 2-Me-3-F-5-CF ₃ -4-PYR], [BK 713; 2-Me-3-F-5-OCHF ₂ -4-PYR], [BK 714; 2-Me-3-F-5-OCF ₃ -4-PYR], [BK 715; 2-Me-3-Cl-5-F-4-PYR], [BK 716] 2-Me-3-Cl-5-Cl-4-PYR], [BK717; 2-Me-3-Cl-5-Br-4-PYR], [BK 718; 2-Me-3-Cl-5 -Me-4-PYR], [BK 719; 2-Me-3-Cl-5-Et-4-PYR], [BK 720; 2-Me-3-Cl-5-OMe-4-PYR], [BK 721 2-Me-3-Cl-5-OEt-4-PYR !, [BK 722; 2-Me-3-Cl-5-CN-4-PYR], [BK 723; 2-Me-3-Cl-5 _{-CHF 2 -4-PYR], [} BK724; 2-Me-3-Cl-5-CF 3 -4-PYR], [BK725; 2-Me-3-Cl-5-OCHF 2 -4-PYR] , [BK 726; 2-Me-3-Cl-5-OCF ₃ -4-PYR], [BK 727; 2-Me34-Br-5-F-4-PYR], [BK 728; 2-Me-3-Br -5-Cl-4-PYR], [BK 729; 2-Me-3-Br-5-Br-4-PYR], [BK 730; 2-Me-3-Br-5-Me-4-PYR], [BK 731; 2-Me-3-Br-5-Et-4-PYR], [BK 732; 2-Me-3-Br-5-OMe-4-PYR], [BK 733; 2-Me-3-Br -5-OEt-4-PYR], [BK 734; 2-Me-3-Br-5-CN -4-PYR], [BK735; 2-Me-3-Br-5-CHF 2 -4-PYR], [BK736; 2-Me-3-Br-5-CF 3 -4-PYR], [BK737 2-Me-3-Br-5-OCHF ₂ -4-PYR !, [BK 738; 2-Me-3-Br-5-OCF ₃ -4-PYR], [BK 739; 2-Me-3-Me -5-F-4-PYR], [BK 740; 2-Me-3-Me-5-Cl-4-PYR], [BK 741; 2-Me-3-Me-5-Br-4-PYR], [BK 742; 2-Me-3-Me-5-Me-4-PYR], [BK 743; 2-Me-3-Me-5-Et-4-PYR], [BK 744; 2-Me-3-Me -5-OMe-4-PYR], [BK 745; 2-Me-3-Me-5-OEt-4-PYR], [BK 746; 2-Me-3-Me-5-CN-4-PYR], [BK 747; 2-Me-3-Me-5-CHF ₂ -4-PYR], [BK 748; 2-Me-3-Me-5-CF ₃ -4-PYR], [BK 749; 2-Me-3 -Me-5-OCHF ₂ -4-PYR], [BK 750; 2-Me-3-Me-5-OCF ₃ -4-PYR], [BK 751; 2-Me-3-Et-5-F-4 -PYR], [BK 752; 2-Me-3-Et-5-Cl-4-PYR], [BK 753; 2-Me-3-Et-5-Br-4-PYR], [BK 754; 2-Me -3-Et-5-Me-4-PYR], [BK 755; 2-Me-3-Et-5-Et-4-PYR], [BK 756; 2-Me-3-Et-5-OMe-4 -PYR], [BK 757; 2-Me-3-Et-5-OEt-4-PYR], [BK 758; 2-Me-3-Et-5-CN-4-PYR], [BK 759; 2-Me -3-Et-5-CHF ₂ -4-PYR !, [BK 760; 2-Me-3-Et-5-CF ₃ -4-PYR], [BK 761; 2-Me-3-Et-5-OCHF ₂ -4-PYR], [BK 762; 2-Me-3-Et-5-OCF ₃ -4-PYR], [BK 763; 2-Me-3-OMe-5-F-4-PYR], [BK 764] 2-Me-3-OMe-5-Cl-4-PYR !, [BK 765; 2-Me-3-OMe-5-Br-4-PYR], [BK766; 2-Me-3-OMe-5 -Me-4-PYR], [BK 767; 2-Me -3-OMe-5-Et-4-PYR], [BK 768; 2-Me-3-OMe-5-OMe-3-PYR], [BK 769; 2-Me-3-OMe-5-OEt-4 -PYR], [BK 770; 2-Me-3-OMe-5-CN-4-PYR], [BK 771; 2-Me-3-OMe-5-CHF _2-4 -PYR], [BK 772; Me-3-OMe-5- CF 3 -4-PYR], [BK773; 2-Me-3-OMe-5-OCHF 2 -4-PYR], [BK774; 2-Me-3-OMe-5- OCF ₃ -4-PYR], [BK 775; 2-Me-3-OEt-5-F-4-PYR], [BK 776; 2-Me-3-OEt-5-Cl-4-PYR], [BK 777] 2-Me-3-OEt-5-Br-4-PYR !, [BK 778; 2-Me-3-OEt-5-Me-4-PYR], [BK 779; 2-Me-3-OEt-5; -Et-4-PYR], [BK 780; 2-Me-3-OEt-5-OMe-4-PYR], [BK 781; 2-Me-3-OEt-5-OEt-4-PYR], [BK 782 ; 2-Me-3-OEt -5-CN-4-PYR], [BK783; 2-Me-3-OEt-5-CHF 2 -4-PYR], [BK784; 2-Me-3-OEt- _{5-CF 3 -4-PYR]} , [BK785; 2-Me-3-OEt-5-OCHF 2 -4-PYR], [BK786; 2-Me-3-OEt-5-OCF 3 -4-PYR ], [BK 787; 2-Me-3-CN-5-F-4-PYR], [BK 788; 2-Me-3-CN-5-Cl-4-PYR], [BK 789; 2-Me-3] -CN-5-Br-4-PYR], [BK 790; 2-Me-3-CN-5-Me-4-PYR], [BK 791; 2-Me-3-CN-5-Et-4-PYR ], [BK 792; 2-Me-3-CN-5-OMe-4-PYR], [BK 793; 2-Me-3-CN-5-OEt-4-PYR], [BK 794; 2-Me-3 -CN-5-CN-4- PYR], [BK795; 2-Me-3-CN-5-CHF 2 -4-PYR], [BK796; 2-Me-3-CN-5-CF 3 -4 -PYR], [BK 797; 2-Me-3-CN-5-OCHF ₂ -4-PYR], [BK 798; 2-Me-3-CN-5-OCF ₃ -4-PYR], [BK 799; -Me -3-CHF ₂ -5-F-4-PYR], [BK 800; 2-Me-3-CHF ₂ -5-Cl-4-PYR],

[BK801; 2-Me-3 -CHF 2 -5-Br-4-PYR], [BK802; 2-Me-3-CHF 2 -5-Me-4-PYR], [BK803; 2-Me-3 -CHF ₂ -5-Et-4-PYR], [BK 804; 2-Me-3-CHF ₂ -5-OMe-4-PYR], [BK 805; 2-Me-3-CHF ₂ -5-OEt- 4-PYR], [BK 806; 2-Me-3-CHF ₂ -5-CN-4-PYR], [BK 807; 2-Me-3-CHF ₂ -5-CHF ₂ -4-PYR], [BK 808] ; 2-Me-3-CHF 2 -5-CF 3 -4-PYR], [BK809; 2-Me-3-CHF 2 -5-OCHF 2 -4-PYR], [BK810; 2-Me-3 _{-CHF 2 -5-OCF 3 -4-} PYR], [BK811; 2-Me-3-CF 3 -5-F-4-PYR], [BK812; 2-Me-3-CF 3 -5-Cl -4-PYR], [BK813; 2-Me-3-CF 3 -5-Br-4-PYR], [BK814; 2-Me-3-CF 3 -5-Me-4-PYR], [BK815 ; 2-Me-3-CF 3 -5-Et-4-PYR], [BK816; 2-Me-3-CF 3 -5-OMe-4-PYR], [BK817; 2-Me-3-CF _{3 -5-OEt-4-PYR} ], [BK818; 2-Me-3-CF 3 -5-CN-4-PYR], [BK819; 2-Me-3-CF 3 -5-CHF 2 -4 -PYR], [BK 820; 2-Me-3-CF ₃ -5-CF ₃ -4-PYR], [BK 821; 2-Me-3-CF ₃ -5-OCHF ₂ -4-PYR], [BK 822] ; 2-Me-3-CF 3 -5-OCF 3 -4-PYR], [BK823; 2-Me-3-OCHF 2 -5-F-4-PYR], [BK824; 2-Me-3- OCHF ₂ -5-Cl-4-PYR], [BK 825; 2-Me-3-OCHF ₂ -5-Br-4-PYR], [BK 826; 2-Me-3-OCHF ₂ -5-Me-4 -PYR], [BK 827; 2-Me-3-OCHF ₂ -5-Et-4-PYR], [BK 828; 2-Me-3-OCHF ₂ -5-OMe-4-PYR], [BK 829; -Me-3-OCHF ₂ -5-OEt-4-PYR], [BK 830; 2-Me- _{3-OCHF 2 -5-CN-} 4-PYR], [BK831; 2-Me-3-OCHF 2 -5-CHF 2 -4-PYR], [BK832; 2-Me-3-OCHF 2 -5- CF ₃ -4-PYR !, [BK 833; 2-Me-3-OCHF ₂ -5-OCHF ₂ -4-PYR], [BK 834; 2-Me-3-OCHF ₂ -5-OCF ₃ -4-PYR ], [BK835; 2-Me -3-OCF 3 -5-F-4-PYR], [BK836; 2-Me-3-OCF 3 -5-Cl-4-PYR], [BK837; 2-Me _{-3-OCF 3 -5-Br-} 4-PYR], [BK838; 2-Me-3-OCF 3 -5-Me-4-PYR], [BK839; 2-Me-3-OCF 3 -5- Et-4-PYR], [ BK840; 2-Me-3-OCF 3 -5-OMe-4-PYR], [BK841; 2-Me-3-OCF 3 -5-OEt-4-PYR], [ BK842; 2-Me-3- OCF 3 -5-CN-4-PYR], [BK843; 2-Me-3-OCF 3 -5-CHF 2 -4-PYR], [BK844; 2-Me-3 _{-OCF 3 -5-CF 3 -4-} PYR], [BK845; 2-Me-3-OCF 3 -5-OCHF 2 -4-PYR], [BK846; 2-Me-3-OCF 3 -5- OCF ₃ -4-PYR].

E12 and E13 representing E ¹¹¹ in BK 847 to BK 1285 represent the following structures.
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[Substituent number (MK2); E ¹¹¹ : [BK 848; E 12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 849: E 12, X ¹⁴¹ : Me, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 850; E12, X ¹⁴¹ : H, X ¹⁴² : Me, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 851; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : Me, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 852; E12, X ¹⁴¹ : Et, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 853; E12, X ¹⁴¹ : H, X ¹⁴² : Et, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 854; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : Et, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 855; E12, X ¹⁴¹ : F, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 856; E12, X ¹⁴¹ : H, X ¹⁴² : F, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 857; E12, X ¹⁴¹ : H, ^{X 142: H, X 143:} F, X 144: H, X 145: H], [BK858; E12, X 141: Cl, X 142: H, X 143: H, X 144: H, X 145: H ], [BK 859; E12, X ¹⁴¹ : H, X ¹⁴² : Cl, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 860; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ^143] : Cl, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 861; E12, X ¹⁴¹ : Br, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 862; E12, X ¹⁴¹ : H, X ¹⁴² : Br, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 863; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : Br, X ¹⁴⁴ : H , X ¹⁴⁵ : H], [BK 864; E 12, X ¹⁴¹ : CN, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 865; E12, X ¹⁴¹ : H, X ¹⁴² : CN, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 866; E12, X ¹⁴¹ : H , X ¹⁴² : H, X ¹⁴³ : CN, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 867; E12, X ¹⁴¹ : OMe, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 868; E12, X ¹⁴¹ : H, X ¹⁴² : OMe, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 869; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : OMe, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 870; E12, X ¹⁴¹ : OEt, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 871; E12 , X ¹⁴¹ : H, X ¹⁴² : OEt, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 872; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : OE t, X ¹⁴⁴ : ^{H, X 145: H],} [BK873; E12, X 141: CF 3, X 142: H, X 143: H, X 144: H, X 145: H, X 144: H, X 145: H], ^{[BK874; E12, X 141:} H, X 142: CF 3, X 143: H, X 144: H, X 145: H], [BK875; E12, X 141: H, X 142: H, X 143: ^{_{CF 3, X 144: H,}} X 145: H], [BK876; E12, X 141: CHF 2, X 142: H, X 143: H, X 144: H, X 145: H], [BK877; E12 , X ¹⁴¹ : H, X ¹⁴² : CHF ₂ , X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 878; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : CHF ₂ , X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 879; E12, X ¹⁴¹ : Me, X ¹⁴² : Me, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 880; E12, X ¹⁴¹ : Me , X ¹⁴² : H, X ¹⁴³ : Me, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 881; E12, X ¹⁴¹ : Cl, X ¹⁴² : Cl, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 882; E12, X ¹⁴¹ : Cl, X ¹⁴² : H, X ¹⁴³ : Cl, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 883; E12, X ¹⁴¹ : H, X ¹⁴² : Me, X ¹⁴³ : Me, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 884; E12, X ¹⁴¹ : H, ^{X 142: Cl, X 143:} Cl, X 144: H, X 145: H], [BK885; E12, X 141: OMe, X 142: H, X 143: Cl, X 144: H, X 145: H ], [BK 886; E12, X ¹⁴¹ : OMe, X ¹⁴² : H, X ¹⁴³ : CN, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 887; E12, X ¹⁴¹ : OMe, X ¹⁴² : H, X ^143] : F, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 888; E12, X ¹⁴¹ : F, X ¹⁴² : H, X ¹⁴³ : Cl, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 889; E 12, X ¹⁴¹ : F, X ¹⁴² : H, X ¹⁴³ : CN, X ¹⁴⁴ : H, X ¹⁴⁵ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 890; E12 , X ¹⁴¹ : F, X ¹⁴² : H, X ¹⁴³ : F, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 891; E12, X ¹⁴¹ : H, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H], [BK 892; E12, X ¹⁴¹ : Me, X ¹⁴² : H, X ¹⁴³ : H, X ¹⁴⁴ : H, X ¹⁴⁵ : H] [BK 893; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 894; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 895; E 13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 896; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 897; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 898; E13, X ¹⁵¹ : Me, X ^{15 2} : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 899; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 900; E 13, X ¹⁵¹ : Me , X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 901; E 13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 902; E 13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 903; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Me], [BK 904; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 905; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 906; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 907; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Me], [, BK 908; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : Me, X ¹⁵⁴ : Me], [BK 909; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : Me, X ¹⁵⁴ : Me] , [BK 910; E 13, X ¹⁵¹ : Me, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 911; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 912; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 913; E13, X ¹⁵¹ : Me, X ¹⁵² : F, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 914; E13, X ¹⁵¹ : Me, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 915; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : F , X ¹⁵⁴ : F], [BK 916; E 13, X ¹⁵¹ : Me, X ¹⁵² : F, X ¹⁵³ : F, X ¹⁵⁴ : F], [BK 917; E 13, X ¹⁵¹ : F, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 918; E 13, X ¹⁵¹ : H, X ¹⁵² : M e, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 919; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 920; E13, X ¹⁵¹ : F, X ¹⁵² : Me, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 921; E13, X ¹⁵¹ : F, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 922; E13, X ¹⁵¹ : H , X ¹⁵² : Me, X ¹⁵³ : F, X ¹⁵⁴ : F], [BK 923; E 13, X ¹⁵¹ : F, X ¹⁵² : Me, X ¹⁵³ : F, X ¹⁵⁴ : F], [BK 924; E 13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 925; E 13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 926; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : F], [BK 927; E13, X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 928; E13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : F], [BK 929; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : Me, X ¹⁵⁴ : F], [ BK930; E13, X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : Me, X ¹⁵⁴ : F], [BK 931; E13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Me] [BK 932; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 933; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : Me], [BK 934; E13, X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 935; E13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : Me], [BK 936; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : F, X ¹⁵⁴ : Me], [BK 937; E13, X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : F , X ¹⁵⁴ : Me], [BK 938; E 13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : F, X ¹⁵⁴ : H ], [BK 939; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 940; E13, X ¹⁵¹ : Me, X ¹⁵² : F, X ¹⁵³ : Me, X ^154] : H], [BK 941; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : F], [BK 942; E13, X ¹⁵¹ : Me, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 943; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : Me], [BK 944; E 13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 945; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 946; E13, X ¹⁵¹ : Me, X ¹⁵² : Cl, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 947; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Cl], [BK 948; E13, X ¹⁵¹ : Me, X ¹⁵² : Cl , X ¹⁵³ : H, X ¹⁵⁴ : Me],

[BK 949; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : Me], [BK 950; E13, X ¹⁵¹ : Me, X ¹⁵² : Cl, X ¹⁵³ : H, X ¹⁵⁴ : H ], [BK 951: E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 952; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : H, X ^154] : Cl], [BK 953; E13, X ¹⁵¹ : Me, X ¹⁵² : Cl, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 954; E13, X ¹⁵¹ : Me, X ¹⁵² : Cl, X ¹⁵³ : H, ^{X 154: Cl], [BK955} ; E13, X 151: Me, X 152: H, X 153: Cl, X 154: Cl], [BK956; E13, X 151: Cl, X 152: Me, X 153: H, X ¹⁵⁴ : H], [BK 957; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 958; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 959; E13, X ¹⁵¹ : Cl, X ¹⁵² : Me, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 960; E13, X ¹⁵¹ : Cl, X ¹⁵² : Me , X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 961; E 13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : Cl, X ¹⁵⁴ : Cl], [BK 962; E 13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 963; E 13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 964; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Cl], [BK 965; E 13, X ¹⁵¹ : Cl, X ¹⁵² : Cl, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 966; E 13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Cl], [BK 967; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : Me, X ¹⁵⁴ : Cl], [BK 968; E13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 969; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 970; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Cl , X ¹⁵⁴ : Me], [BK 971; E 13, X ¹⁵¹ : Cl, X ¹⁵² : Cl, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 972; E 13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : Me], [BK 973; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : Cl, X ¹⁵⁴ : Me], [BK 974; E13, X ¹⁵¹ : Me, X ¹⁵² : Br, ^{X 153: H, X 154:} H], [BK975; E13, X 151: Me, X 152: H, X 153: Br, X 154: H], [BK976; E13, X 151: Me, X 152: H, X ¹⁵³ : H, X ¹⁵⁴ : Br], [BK 977; E13, X ¹⁵¹ : Br, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 978; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : Br, X ¹⁵⁴ : H], [BK 979; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Br], [BK 980; E13, X ¹⁵¹ : Br , X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 981; E 13, X ¹⁵¹ : H, X ¹⁵² : Br, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 982; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Br], [BK 983; E13, X ¹⁵¹ : Br, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 984; E 13, X ¹⁵¹ : H, X ¹⁵² : Br, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 985; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Br, X ¹⁵⁴ : Me], [BK 986; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : Br, X ¹⁵⁴ : H], [BK 987; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Br], [ BK 988; E 13, X ¹⁵¹ : Me, X ¹⁵² : Br, X ^{15 3} : Me, X ¹⁵⁴ : H], [BK 989; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Br], [BK 990; E13, X ¹⁵¹ : Me, X ¹⁵² : Br , X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 991; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Br, X ¹⁵⁴ : Me], [BK 992; E 13, X ¹⁵¹ : Me, X ¹⁵² : CN, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 993; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : CN, X ¹⁵⁴ : H], [BK 994; E 13, X ¹⁵¹ : Me, ^{X 152: H, X 153:} H, X 154: CN], [BK995; E13, X 151: CN, X 152: Me, X 153: H, X 154: H], [BK996; E13, X 151: H, X ¹⁵² : Me, X ¹⁵³ : CN, X ¹⁵⁴ : H], [BK 997; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : CN], [BK 998; E 13, X ¹⁵¹ : CN, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 999; E13, X ¹⁵¹ : H, X ¹⁵² : CN, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 1000; E 13 ^{, X 151: H, X 152} : H, X 153: Me, X 154: CN], [BK1001; E13, X 151: CN, X 152: H, X 153: H, X 154: Me], [BK1002 E13, X ¹⁵¹ : H, X ¹⁵² : CN, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 1003; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : CN, X ¹⁵⁴ : Me], [BK1004: E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : CN, X ¹⁵⁴ : H], [BK 1005; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : CN ], [BK 1006; E13, X ¹⁵¹ : Me, X ¹⁵² : CN, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 1007; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ^154] : CN], [BK 1008; E13, X ¹⁵¹ : ^{Me, X 152: CN, X} 153: H, X 154: Me], [BK1009; E13, X 151: Me, X 152: H, X 153: CN, X 154: Me], [BK1010; E13, X ^{151: Me, X 152: OMe} , X 153: H, X 154: H], [BK1011; E13, X 151: Me, X 152: H, X 153: OMe, X 154: H], [BK1012; E13 , X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : OMe], [BK 1013; E13, X ¹⁵¹ : OMe, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1014 E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : OMe, X ¹⁵⁴ : H], [BK 1015; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : OMe], ^{[BK1016; E13, X 151:} OMe, X 152: H, X 153: Me, X 154: H], [BK1017; E13, X 151: H, X 152: OMe, X 153: Me, X 154: H ], [BK1018; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : OMe], [BK 10 19; E13, X ¹⁵¹ : OMe, X ¹⁵² : H, X ¹⁵³ : H, X ^154] : Me], [BK 1020; E13, X ¹⁵¹ : H, X ¹⁵² : OMe, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 1021; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : OMe, X ¹⁵⁴ : Me], [BK 1022; E 13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : OMe, X ¹⁵⁴ : H], [BK 1023; E 13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : OMe], [BK 1024; E13, X ¹⁵¹ : Me, X ¹⁵² : OMe, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 1025; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : OMe], [BK 1026; E13, X ¹⁵¹ : Me, X ¹⁵² : OMe, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK 1027; E13, X ¹⁵¹ : Me, X ^{15 2} : H, X ¹⁵³ : OMe, X ¹⁵⁴ : Me], [BK 1028; E13, X ¹⁵¹ : Me, X ¹⁵² : OEt, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1029; E13, X ¹⁵¹ : Me ^{, X 152: H, X 153} : OEt, X 154: H], [BK1030; E13, X 151: Me, X 152: H, X 153: H, X 154: OEt], [BK1031; E13, X 151 ^{: OEt, X 152: Me,} X 153: H, X 154: H], [BK1032; E13, X 151: H, X 152: Me, X 153: OEt, X 154: H], [BK1033; E13, ^{X 151: H, X 152:} Me, X 153: H, X 154: OEt], [BK1034; E13, X 151: OEt, X 152: H, X 153: Me, X 154: H], [BK1035; E13, X ¹⁵¹ : H, X ¹⁵² : OEt, X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 1036; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : OE t], [ ^{BK1037; E13, X 151: OEt} , X 152: H, X 153: H, X 154: Me], [BK1038; E13, X 151: H, X 152: OEt, X 153: H, X 154: Me] , [BK1039; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : OEt, X ¹⁵⁴ : Me], [BK 1040; E13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : OE t, X ¹⁵⁴ : H], [BK1041; E13, X 151: Me, X 152: Me, X 153: H, X 154: OEt], [BK1042; E13, X 151: Me, X 152: OEt, X 153: Me, X ^{154: H], [BK1043;} E13, X 151: Me, X 152: H, X 153: Me, X 154: OEt], [BK1044; E13, X 151: Me, X 152: OEt, X 153: H , X ¹⁵⁴ : Me], [BK 1045; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : OEt, X ¹⁵⁴ : Me], [BK 1046; E 13, X ¹⁵¹ : Me, X ¹⁵² : Et , X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1047; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1048; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Et],

[BK1049; E13, X ¹⁵¹ : Et, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1050; E13, X ¹⁵¹ : H, X ¹⁵² : Me, X ¹⁵³ : Et, X ¹⁵⁴ : H ], [BK1051; E13, X 151: H, X 152: Me, X 153: H, X 154: Et], [BK1052; E13, X 151: Et, X 152: H, X 153: Me, X 154 : H], [BK1053; E13 , X 151: H, X 152: Et, X 153: Me, X 154: H], [BK1054; E13, X 151: H, X 152: H, X 153: Me, ^{X 154: Et], [BK1055} ; E13, X 151: Et, X 152: H, X 153: H, X 154: Me], [BK1056; E13, X 151: H, X 152: Et, X 153: ^{H, X 154: Me],} [BK1057; E13, X 151: H, X 152: H, X 153: Et, X 154: Me], [BK1058; E13, X 151: Me, X 152: Me, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1059; E 13, X ¹⁵¹ : Me, X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1060; E13, X ¹⁵¹ : Me, X ¹⁵² : Et , X ¹⁵³ : Me, X ¹⁵⁴ : H], [BK 1061; E 13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : Et], [BK 1062; E 13, X ¹⁵¹ : Me, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : Me], [BK1063; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : Me], [BK 1064; E13, X ¹⁵¹ : Me, _{^{X 152: CF 3, X 153}} : H, X 154: H], [BK1065; E13, X 151: Me, X 152: H, X 153: CF 3, X 154: H], [BK1066; E13, X ¹⁵¹ : Me, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : CF ₃ ], [BK 1067; E 13, X ¹⁵¹ : CF ₃ , X ¹⁵² : Me, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1068 E13, X ^{151: H, X 152: Me} , X 153: CF 3, X 154: H], [BK1069; E13, X 151: H, X 152: Me, X 153: H, X 154: CF 3], [BK1070 _{^{; E13, X 151: CF 3}} , X 152: H, X 153: Me, X 154: H], [BK1071; E13, X 151: H, X 152: CF 3, X 153: Me, X 154: H ], [BK1072; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Me, X ¹⁵⁴ : CF ₃ ], [BK 1073; E13, X ¹⁵¹ : CF ₃ , X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵³ : H, ^{X 154: Me], [BK1074} ; E13, X 151: H, X 152: CF 3, X 153: H, X 154: Me], [BK1075; E13, X 151: H, X 152: H, X 153 : CF ₃ , X ¹⁵⁴ : Me], [BK 1076; E 13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1077; E 13, X ¹⁵¹ : H, X ¹⁵² : Et , X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1078; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1079; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1080; E13, X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1081; E13, X ¹⁵¹ : Et, ^{X 152: H, X 153:} Et, X 154: H], [BK1082; E13, X 151: Et, X 152: H, X 153: H, X 154: Et], [BK1083; E13, X 151: H, X ¹⁵² : Et, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1084; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1085; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : Et], [BK 1086; E13, X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1087; E 13 , X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1088; E13, X ¹⁵¹ : Et, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1089; E13, X ¹⁵¹ : Et , X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1090; E 13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 109 1; E 13, X ¹⁵¹ : Et, X ¹⁵² : F, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK1092; E13, X ¹⁵¹ : Et, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 1093; E13, ^{X 151: Et, X 152:} H, X 153: F, X 154: F], [BK1094; E13, X 151: F, X 152: Et, X 153: H, X 154: H], [BK1095; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1096; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : F], [ BK1097; E13, X ¹⁵¹ : F, X ¹⁵² : Et, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1098; E13, X ¹⁵¹ : F, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : F] ^{, [BK1099; E13, X 151} : H, X 152: Et, X 153: F, X 154: F], [BK1100; E13, X 151: F, X 152: H, X 153: Et, X 154: H], [BK1 101; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1102; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : F], [BK 1 103; E13, X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1104; E13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : Et , X ¹⁵⁴ : F], [BK 1105; E 13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : Et, X ¹⁵⁴ : F], [BK 1106; E 13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1107; E 13, X ¹⁵¹ : H, ^{X 152: F, X 153:} H, X 154: Et], [BK1108; E13, X 151: H, X 152: H, X 153: F, X 154: Et], [BK1109; E13, X 151: ^{F, X 152: F, X} 153: H, X 154: Et], [BK1110; E13, X 151: F, X 152: H, X 153: F, X 154: Et], [BK1111; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : F, X ¹⁵⁴ : Et], [BK 11 12; E13, X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 11 13; E 13 , X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 1114; E 13, X ¹⁵¹ : Et, X ¹⁵² : F, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1115 E13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : F], [BK 1116; E13, X ¹⁵¹ : Et, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK1 117; E13, X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 1 118; E13, X ¹⁵¹ : Et, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : Cl ], [BK 1119; E13, X ¹⁵¹ : Et, X ¹⁵² : Cl, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1 120; E13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : Et, X ^154] : Cl], [BK1121; E13 , X 151: Et, X 152: Cl, X 153: H, X 154: Et], [BK1122; E13, X 151: Et, X 152: H, X 153: Cl, X ¹⁵⁴ : Et], [BK 1123; E 13, X ¹⁵¹ : Et, X ¹⁵² : Cl, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1 124; E 13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 1 125; E13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 1 126; E13, X ¹⁵¹ : Et, X ¹⁵² : Cl, X ¹⁵³ : Cl, X ¹⁵⁴ : H] ^{, [BK1127; E13, X 151} : Et, X 152: Cl, X 153: H, X 154: Cl], [BK1128; E13, X 151: Et, X 152: H, X 153: Cl, X 154: Cl], [BK 1129; E13, X ¹⁵¹ : Cl, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1130; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 1131; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 1132; E13, X ¹⁵¹ : Cl, X ¹⁵² : Et, X ¹⁵³ : Cl ¹⁵³ , X ¹⁵⁴ : H], [BK 1133; E 13, X ¹⁵¹ : Cl, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 1134; E 13, X ¹⁵¹ : H, X ¹⁵² : Et, X ^{153 : Cl, X 154: Cl]} , [BK1135; E13, X 151: Cl, X 152: H, X 153: Et, X 154: H], [BK1136; E13, X 151: H, X 152: Cl, ^{X 153: Et, X 154:} H], [BK1137; E13, X 151: H, X 152: H, X 153: Et, X 154: Cl], [BK1138; E13, X 151: Cl, X 152: Cl, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1139; E 13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : Cl], [BK 1 140; E 13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : Et, X ¹⁵⁴ : Cl], [BK 1141; E13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1142; E13, X ¹⁵¹ : H ^{, X 152: Cl, X 153} : H, X 154: Et], [BK1143; E13, X 151: H, X 152: H, X 153: Cl, X 154: Et], [BK1144; E13, X 151 ^{: Cl, X 152: Cl,} X 153: H, X 154: Et], [BK1145; E13, X 151: Cl, X 152: H, X 153: Cl, X 154: Et], [BK1146; E13, X ¹⁵¹ : H ^{, X 152: Cl, X 153} : Cl, X 154: Et], [BK1147; E13, X 151: Et, X 152: CN, X 153: H, X 154: H], [BK1148; E13, X 151 : Et, X ¹⁵² : H, X ¹⁵³ : CN, X ¹⁵⁴ : H],

[BK1149; E13, X ¹⁵¹ : Et, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : CN], [BK 1 150; E13, X ¹⁵¹ : CN, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : H ], [BK1151; E13, X 151: H, X 152: Et, X 153: CN, X 154: H], [BK1152; E13, X 151: H, X 152: Et, X 153: H, X 154 : CN], [BK 1153; E13, X ¹⁵¹ : CN, X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : H], [BK 1 ¹⁵⁴ ; E13, X ¹⁵¹ : H, X ¹⁵² : CN, X ¹⁵³ : Et, ^{X 154: H], [BK1155} ; E13, X 151: H, X 152: H, X 153: Et, X 154: CN], [BK1156; E13, X 151: CN, X 152: H, X 153: H, X ¹⁵⁴ : Et], [BK 1 157; E13, X ¹⁵¹ : H, X ¹⁵² : CN, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1158; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ^{153: CN, X 154: Et} ], [BK1159; E13, X 151: Et, X 152: CF 3, X 153: H, X 154: H], [BK1160; E13, X 151: Et, X 152: _{^{H, X 153: CF 3,}} X 154: H], [BK1161; E13, X 151: Et, X 152: H, X 153: H, X 154: CF 3], [BK1162; E13, X 151: CF ^{_{3, X 152: Et, X}} 153: H, X 154: H], [BK1163; E13, X 151: H, X 152: Et, X 153: CF 3, X 154: H], [BK1164; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : CF ₃ ], [BK 1165; E 13, X ¹⁵¹ : CF ₃ , X ¹⁵² : H, X ¹⁵³ : Et, X ¹⁵⁴ : H], [ ^{BK1166; E13, X 151: H} , X 152: CF 3, X 153: Et, X 154: H], [BK1167; E13, X 151: H, X 152: H, X 153: Et, X 154: CF ₃ ], [BK1 ^{168; E13, X 151: CF} 3, X 152: H, X 153: H, X 154: Et], [BK1169; E13, X 151: H, X 152: CF 3, X 153: H, X 154: Et], [BK1170; E13, X 151: H, X 152: H, X 153: CF 3, X 154: Et], [BK1171; E13, X 151: Et, X 152: OMe, X 153: H, ^{X 154: H], [BK1172} ; E13, X 151: Et, X 152: H, X 153: OMe, X 154: H], [BK1173; E13, X 151: Et, X 152: H, X 153: H, X ¹⁵⁴ : OMe], [BK 1174; E13, X ¹⁵¹ : OMe, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1175; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : OMe, X ¹⁵⁴ : H], [BK 1176; E13, X ¹⁵¹ : H, X ¹⁵² : Et, X ¹⁵³ : H, X ¹⁵⁴ : OMe], [BK 1177; E13, X ¹⁵¹ : OMe, X ¹⁵² : H ^{, X 153: Et, X 154} : H], [BK1178; E13, X 151: H, X 152: OMe, X 153: Et, X 154: H], [BK1179; E13, X 151: H, X 152 : H, X ¹⁵³ : Et, X ¹⁵⁴ : OMe], [BK 1180; E13, X ¹⁵¹ : OMe, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Et], [BK 1181; E13, X ¹⁵¹ : H, ^{X 152: OMe, X 153:} H, X 154: Et], [BK1182; E13, X 151: H, X 152: H, X 153: OMe, X 154: Et], [BK1183; E13, X 151: F, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1184; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1 185; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1186; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 1187; E 13 , X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1188; E13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1189; E13, X ¹⁵¹ : F , X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 1190; E 13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1191; E 13, X ^{151 : H, X 152: F,} X 153: H, X 154: F], [BK1192; E13, X 151: H, X 152: H, X 153: F, X 154: F], [BK1193; E13, ^{X 151: F, X 152:} F, X 153: F, X 154: H], [BK1194; E13, X 151: F, X 152: H, X 153: F, X 154: F], [BK1195; E13, X ¹⁵¹ : F, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 1196; E13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [ ^{BK1197; E13, X 151: H} , X 152: Cl, X 153: H, X 154: H], [BK1198; E13, X 151: H, X 152: H, X 153: Cl, X 154: H] ^{, [BK1199; E13, X 151} : H, X 152: H, X 153: H, X 154: Cl], [BK1200; E13, X 151: Cl, X 152: Cl, X 153: H, X 154: H], [BK1201; E13, X 151: Cl, X 152: H, X 153: Cl, X 154: H], [BK1202; E13, X 151: Cl, X 152: H, X 153: H, X ¹⁵⁴ : Cl], [BK 1203; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 1204; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : H , X ¹⁵⁴ : Cl], [BK 1205; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : Cl], [BK 1206; E 13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : Cl], [BK 1207; E 13, X ¹⁵¹ : Cl, X ¹⁵² : Cl, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 1208; E13, X ¹⁵¹ : Cl, X ¹⁵² : Cl, X ¹⁵³ : Cl, X ¹⁵⁴ : H], [BK 1 209; E13, X ¹⁵¹ : F ^{, X 152: Cl, X 153} : H, X 154: H], [BK1210; E13, X 151: F, X 152: H, X 153: Cl, X 154: H], [BK1211; E13, X 151 : F, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : Cl], [BK 1212; E13, X ¹⁵¹ : Cl, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1213; E 13, ^{X 151: H, X 152:} F, X 153: Cl, X 154: H], [BK1214; E13, X 151: H, X 152: F, X 153: H, X 154: Cl], [BK1215; E13, X ¹⁵¹ : Cl, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1216; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : F, X ¹⁵⁴ : H], [ ^{BK1217; E13, X 151: H} , X 152: H, X 153: F, X 154: Cl], [BK1218; E13, X 151: Cl, X 152: H, X 153: H, X 154: F] ^{, [BK1219; E13, X 151} : H, X 152: Cl, X 153: H, X 154: F], [BK1220; E13, X 151: H, X 152: H, X 153: Cl, X 154: F], [BK1221; E13, X 151: n-propyl, X 152: H, X 153: H, X 154: H], [BK1222; E13, X 151: H, X 152: n-propyl, X 153 ^{: H, X 154: H]} , [BK1223; E13, X 151: H, X 152: H, X 153: n-propyl, X 154: H], [BK1224; E13, X 151: H, X 152: ^{H, X 153: H, X} 154: n-propyl], [BK1225; E13, X 151: isopropyl, X 152: H, X 153: H, X 154: H], [BK1226; E13, X 151: H , X ¹⁵² : isopropyl, ^{X 153: H, X 154:} H], [BK1227; E13, X 151: H, X 152: H, X 153: isopropyl, X 154: H], [BK1228; E13, X 151: H, X 152: ^{H, X 153: H, X} 154: isopropyl], [BK1229; E13, X 151: OMe, X 152: H, X 153: H, X 154: H], [BK1230; E13, X 151: H, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : OMe], [BK 1231; E13, X ¹⁵¹ : OMe, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1232: E13, X ¹⁵¹ : OMe , X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1233; E 13, X ¹⁵¹ : H, X ¹⁵² : OMe, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1234; E 13, X ^{151 : H, X 152: H,} X 153: OMe, X 154: H], [BK1235; E13, X 151: H, X 152: H, X 153: H, X 154: OMe], [BK1236; E13, ^{X 151: OMe, X 152:} F, X 153: H, X 154: H], [BK1237; E13, X 151: OMe, X 152: H, X 153: F, X 154: H], [BK1238; E13, X ¹⁵¹ : OMe, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : F], [BK 1239; E13, X ¹⁵¹ : F, X ¹⁵² : OMe, X ¹⁵³ : H, X ¹⁵⁴ : H], [ BK1240; E13, X ¹⁵¹ : H, X ¹⁵² : OMe, X ¹⁵³ : F, X ¹⁵⁴ : H], [BK 1241; E13, X ¹⁵¹ : H, X ¹⁵² : OMe, X ¹⁵³ : H, X ¹⁵⁴ : F] ^{, [BK1242; E13, X 151} : F, X 152: H, X 153: OMe, X 154: H], [BK1243; E13, X 151: H, X 152: F, X 153: OMe, X 154: H], [BK 1244; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : OMe, X ¹⁵⁴ : F], [BK 1245; E13, X ¹⁵¹ : F, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : OMe], ^{[BK1246; E13, X 151:} H, X 152: F, X 153: H, X 154: OMe], [BK1247; E13, X 151: H, X 152: H, X 153: F, X 154: OMe ], [BK1248; E13, X 151: OMe, X 152: Cl, X 153: H, X 154: H],

^{[BK1249; E13, X 151:} OMe, X 152: H, X 153: Cl, X 154: H], [BK1250; E13, X 151: OMe, X 152: H, X 153: H, X 154: Cl ], [BK1251; E13, X 151: Cl, X 152: OMe, X 153: H, X 154: H], [BK1252; E13, X 151: H, X 152: OMe, X 153: Cl, X 154 : H], [BK1253; E13 , X 151: H, X 152: OMe, X 153: H, X 154: Cl], [BK1254; E13, X 151: Cl, X 152: H, X 153: OMe, ^{X 154: H], [BK1255} ; E13, X 151: H, X 152: Cl, X 153: OMe, X 154: H], [BK1256; E13, X 151: H, X 152: H, X 153: ^{OMe, X 154: Cl],} [BK1257; E13, X 151: Cl, X 152: H, X 153: H, X 154: OMe], [BK1258; E13, X 151: H, X 152: Cl, X ¹⁵³ : H, X ¹⁵⁴ : OMe], [BK 1259; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Cl, X ¹⁵⁴ : OMe], [BK 1260; E13, X ¹⁵¹ : CN, X ¹⁵² : H , X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1261; E 13, X ¹⁵¹ : H, X ¹⁵² : CN, X ¹⁵³ : H, X ¹⁵⁴ : H], [BK 1262; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : CN, X ¹⁵⁴ : H], [BK 1263; E 13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : H, X ¹⁵⁴ : CN], [BK 1264; E 13, X ¹⁵¹ : CN, ^{X 152: F, X 153:} H, X 154: H], [BK1265; E13, X 151: CN, X 152: H, X 153: F, X 154: H], [BK1266; E13, X 151: ^{CN, X 152: H, X} 153: H, X 154: F], [BK1267; E13, X 151: F, X 152: CN, X 153: H, X 154: H], [BK1268; E13, X ¹⁵¹ : H, X ¹⁵² : ^{CN, X 153: F, X} 154: H], [BK1269; E13, X 151: H, X 152: CN, X 153: H, X 154: F], [BK1270; E13, X 151: F, X ¹⁵² : H, X ¹⁵³ : CN, X ¹⁵⁴ : H], [BK 1271; E13, X ¹⁵¹ : H, X ¹⁵² : F, X ¹⁵³ : CN, X ¹⁵⁴ : H], [BK 1272; E13, X ¹⁵¹ : H ^{, X 152: H, X 153} : CN, X 154: F], [BK1273; E13, X 151: F, X 152: H, X 153: H, X 154: CN], [BK1274; E13, X 151 : H, X ¹⁵² : F, X ¹⁵³ : H, X ¹⁵⁴ : CN], [BK 1275; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : F, X ¹⁵⁴ : CN], [BK 1276; E 13, ^{X 151: CN, X 152:} Cl, X 153: H, X 154: H], [BK1277; E13, X 151: CN, X 152: H, X 153: Cl, X 154: H], [BK1278; ^{E13, X 151: CN, X} 152: H, X 153: H, X 154: Cl], [BK1279; E13, X 151: Cl, X 152: CN, X 153: H, X 154: H], [ ^{BK1280; E13, X 151: H} , X 152: CN, X 153: Cl, X 154: H], [BK1281; E13, X 151: H, X 152: CN, X 153: H, X 154: Cl] ^{, [BK1282; E13, X 151} : Cl, X 152: H, X 153: CN, X 154: H], [BK1283; E13, X 151: H, X 152: Cl, X 153: CN, X 154: H], [BK1284; E13, X 151: H, X 152: H, X 153: CN, X 154: Cl], [BK1285; E13, X 151: Cl, X 152: H, X 153: H, X ¹⁵⁴ : CN], [BK 1286; E13, X ¹⁵¹ : H, X ¹⁵² : Cl, X ¹⁵³ : H, X ¹⁵⁴ : CN], [BK 1287; E13, X ¹⁵¹ : H, X ¹⁵² : H, X ¹⁵³ : Cl , X ¹⁵⁴ : CN].

  The composition of the present invention usually contains the present compound in an amount of 0.01 to 99% by weight.

  The composition of the present invention comprises the present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E and Group F.

The components of the bactericide included in group A include, for example, (1) DMI bactericide (demethylation inhibitor)
Azaconazole (azaconazole), bitertanol (bitertanol), bromuconazole (bromuconazole), cyproconazole (cyproconazole), difenoconazole (difenoconazole), diniconazole, diniconazole M (diniconazole-M), epoxyconazole (epoxiconazole) (Etaconazole), phenarimol (fenarimol), fenbuconazole (fenbuconazole), fluquinconazole (fluquinconazole), quinconazole (quinconazole), flusilazole (flusilazole), flutriaphor (flutriafol), hexaconazole (hexaconazole), imazaryl ( imazalil), imibenconazole (imibenconazole), ipconazole (ipconazole), metconazole (metconazole), microbutanil (myclobutanil), nuarimol (nuarimol), oxisoconazole (oxpoconazole), o Spoconazole fumarate (oxpoconazole fumarate), pefrazoate (pefurazoate), penconazole (penconazole), prochloraz (prochloraz), propiconazole (propiconazole), prothioconazole (prothioconazole), pyriphenox (pyrifoxazole) ), Simeconazole (simeconazole), tebuconazole (tebuconazole), tetraconazole (tetraconazole), triadimefon (triadimefon), triadimenol (triadimenol), triflumisole (triflumisole), triphorin (triforine), trichiconazole (triticonazole), α- [3- (4-Chloro-2-fluorophenyl) -5- (2,4-difluorophenyl) -4-isoxazolyl] -3-pyridinemethanol (CAS Registry No. 1229605-96-2), (αS) -[3- (4-chloro-2-ful Rophenyl) -5- (2,4-difluorophenyl) -4-isoxazolyl] -3-pyridinemethanol (CAS Registry No. 1229606-46-5), (αR)-[3- (4-chloro-2-fluorophenyl) ) -5- (2,4-Difluorophenyl) -4-isoxazolyl] -3-pyridinemethanol (CAS Registry Number 1229606-02-3), 2-{[3- (2-chlorophenyl) -2- (2 ,, 4-Difluorophenyl) oxiran-2-yl] methyl} -2,4-dihydro-3H-1,2,4-triazole-3-thione (CAS Registry Number 1342260-19-8), 2-{[(2R) , 3S) -3- (2-Chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] methyl} -2,4-dihydro-3H-1,2,4-triazole-3-thione (CAS registration number 1638897-70-7), 2-{[(2S, 3R) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -2,4-dihydro- 3H-1,2,4-triazole-3-thione (CAS Registry Number 1638897-71-8),
2-{[(2R, 3R) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -2,4-dihydro-3H-1,2,4 Triazole-3-thione (CAS Registry No. 1638897-72-9), 2-{[(2S, 3S) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] ] -Methyl} -2,4-dihydro-3H-1,2,4-triazole-3-thione (CAS Registry Number 1638897-73-0), 1-{[3- (2-chlorophenyl) -2- (2) , 4-Difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4-triazol-5-yl thiocyanato (CAS Registry Number 1342260-26-7), 1-{[(2R, 3S)- 3- (2-chlorophenyl) -2- (2,4-diful) Orophenyl) oxirane-2-yl] methyl} -1H-1,2,4-triazol-5-yl thiocyanato (CAS Registry No. 1638897-82-1), 1-{[(2S, 3R) -3- (2) -Chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] methyl} -1H-1,2,4-triazol-5-yl thiocyanate (CAS Registry No. 1638897-84-3), 1- {[(2R, 3R) -3- (2-Chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4-triazol-5-yl thiocyanate ( CAS Registry Number 1638897-86-5), 1-{[(2S, 3S) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -1H-1 , 2,4-tria 5-yl thiocyanato (CAS Registry Number 1638897-89-8), 5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole-1) -Ilmethyl) cyclopentanol (CAS Reg. No. 1394057-11-4), (1R, 2S, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,5) 2,4-Triazol-1-ylmethyl) cyclopentanol (CAS Registry No. 1801930-06-2), (1S, 2R, 5R) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl- 1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry No. 1801930-07-3), (1R, 2R, 5R) -5- (4-chlorobenzyl) -2- Chloromethyl-2-methyl-1- (1H- , 2,4-Triazol-1-ylmethyl) cyclopentanol (CAS Registry Number 1801919-53-8), (1S, 2S, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl -1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry No. 1801919-54-9), (1R, 2R, 5S) -5- (4-chlorobenzyl) -2 -Chloromethyl-2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS registration number 1801919-55-0), (1S, 2S, 5R) -5- (5) 4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS registration number 1801919-56-1), (1R, 2S) , 5R) -5- (4-chloro N-diyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS registration number 1801919-57-2), (1S, 2R, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry Number 1801919-58-3), Methyl 3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanecarboxylate (CAS Registry Number 1791398-02 1), methyl = (1R, 2S, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopente Tan carboxylate, methyl = (1S, 2R, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) Cyclopentane carboxylate, methyl = (1R, 2R, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl ) Cyclopentanecarboxylate, methyl = (1S, 2S, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazole-1) Ylmethyl) cyclopentane carboxylate, methyl = (1R, 2R, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2 (1H-1,2,4-triazol-1-ylmethyl) cyclopentanecarboxylate, methyl = (1S, 2S, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2 -(1H-1,2,4-triazol-1-ylmethyl) cyclopentane carboxylate, methyl = (1R, 2S, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl- 2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentane carboxylate, methyl = (1S, 2R, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl -2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentane carboxylate, 2-chloromethyl-5- (4-fluoro) Ndidyl) -2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry No. 1394057-13-6), (1R, 2S, 5S) -2-chloromethyl -5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry No. 1801930-08-4), (1S, 2R, 5R) -2-Chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry Number 1801930-09-5) ), (1R, 2R, 5R) -2-chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS) Registration number 1638898-08-4) , (1S, 2S, 5S) -2-Chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanol (CAS Registry) No. 1638898-10-8), (1R, 2R, 5S) -2-chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,4-triazol-1-ylmethyl) ) Cyclopentanol (CAS Registry No. 1638898-13-1), (1S, 2S, 5R) -2-chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,5) 4-Triazol-1-ylmethyl) cyclopentanol (CAS Registry No. 1638898-16-4), (1R, 2S, 5R) -2-chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1,2,4-triazole 1-ylmethyl) cyclopentanol (CAS Registry No. 1638898-20-0), (1S, 2R, 5S) -2-chloromethyl-5- (4-fluorobenzyl) -2-methyl-1- (1H-1) , 2,4-Triazol-1-ylmethyl) cyclopentanol (CAS Registry Number 1638898-24-4), 2- [2-chloro-4- (4-chlorophenoxy) phenyl] -1- (1,2,2,7 4-Triazol-1-yl) pent-3-yn-2-ol (CAS Registry No. 1419875-41-4), 2- [4- (4-chlorophenoxy) -2- (trifluoromethyl) phenyl]- 1- (1,2,4-triazol-1-yl) propan-2-ol (CAS Registry No. 1417782-03-6), 1- [4- (4-chlorophenoxy) -2- (trifluoromethyl) Phenyl] -1-cyclopropyl-2- ( , 2,4-Triazol-1-yl) ethanol (CAS Registry No. 1417782-09-2), 2- [4- (4-Chlorophenoxy) -2- (trifluoromethyl) phenyl] -3-methyl-1 -(1,2,4-triazol-1-yl) butan-2-ol (CAS Registry No. 1417782-08-1), (R) -2- [2-chloro-4- (4-chlorophenoxy) phenyl -1- (1,2,4-triazol-1-yl) pent-3-yn-2-ol (CAS Registry No. 1801919-59-4), (R) -2- [4- (4-chloro) Phenoxy) -2- (trifluoromethyl) phenyl] -1- (1,2,4-triazol-1-yl) propan-2-ol (CAS Registry No. 1616236-94-2), (R) -1- [4- (4-Chlorophenoxy) -2- (trifluoromethyl) phenyl] -1 Cyclopropyl-2- (1,2,4-triazol-1-yl) ethanol (CAS Registry Number 1801919-60-7, (R) -2- [4- (4-chlorophenoxy) -2- (tri) Fluoromethyl) phenyl] -3-methyl-1- (1,2,4-triazol-1-yl) butan-2-ol (CAS Registry No. 1801919-61-8), Difenodiconazole (Difenodiconazole CAS Registry No.) 930581-38-7), Pyrisoxazole (pyrisoxazole CAS Registry Number 291771-83-0), 3- [5- (4-chlorophenyl) -2,3-dimethyl-1,2-oxazolidin-3-yl] pyridine (CAS Registration number 847749-37-5) etc.

(2) Aminic fungicide aldimorph, dodemorph, fenpropidin, fenpropimorph, piperaline, pirazrin, spiroxamine, tridemorph and the like.

(3) Benzimidazole fungicides benamyl, carbendazim, fuberidazole, thiabendazole, thiophanate, thiophanate methyl and the like.

(4) Dicarboximide fungicide clozolinate (chlozolinate), iprodione (iprodione), procymidone (procymidone), vinclozolin and the like.

(5) Anilinopyrimidine fungicides cyprodinil, mepanipyrim, pyrimethanil etc.
(6) Phenylpyrrole fungicide fenpiclonil, fludioxonil and the like.

(7) QoI disinfectant (Qo inhibitor)
Azoxystrobin (azoxystrobin), spider oxystrobin (coumoxystrobin), dimoxystrobin (dimoxystrobin), enoxastrobin (enoxastrobin), famoxadone (famoxadone), fenamidonone (fenamidone), phenaminstrobin (fenaminstrobin), full Phenoxystrobin (flufenoxystrobin), fluoxastrobin (fluoxastrobin), kresoxim-methyl (kresoxim-methyl), mandestorobin (mandestrobin), metominostrobin (metominostrobin), orysastrobin (orysastrobin), picoxystrobin (picoxystrobin) , Pyraclostrobin, pyrametostrobin, pyraoxystrobin, pyribencarb, triclopyricarb, trifloxystrobin and the like.

(8) PA fungicide (phenylamide fungicide)
Benalaxyl (benalaxyl), Benalaxyl M or chiralaxyl (benalaxyl-M or kiralaxyl), fralaxyl (furalaxyl), metalaxyl (metalaxyl), metalaxyl M or mefenoxam (metalaxyl-M or mefenoxam), oxadixil (oxadixil)

(9) Carboxylic acid amide based fungicide dimethomorph, flumorph, pyrimorph, benthiavalicarab, benthiavalicca isopropyl (benthivalicarb-isopropyl), iprovaricarb (iprovalicarb), mandipropamide ( mandipropamid), varifenalate etc.

(10) SDHI fungicide (succinic acid dehydrogenase inhibitor)
Benodanil (benodanil), benzobindiflupyr (benzovindiflupyr), bixafen (bixafen), boscalid (boscalid), carboxin (carboxin), fenfuram (fenfuram), fluopyram (fluopyram), flutolanil (flutolanil), fluxapiroxad (fluxapiroxad) ), Furametopyr (furametpyr), isofetamide (isofetamid), isopyrazam (isopyrazam), mepronil (mepronil), oxycarboxin (oxycarboxin), penthiopyrade (penthiopyrad), penflufen (penflufen), sedaxane, thifluzamide (thiflumimide) (Pyraziflumid, CAS Registry No. 942515-63-1), N-Cyclopropyl-3- (difluoromethyl) -5-fluoro-N- (2-isopropylbenzyl) -1-methyl-1H-pyrazole-4-carboxamide ( CAS registration No. 1255733-83-5), N-Cyclopropyl-3- (difluoromethyl) -5-fluoro-N- (5-chloro-2-isopropylbenzyl) -1-methyl-1H-pyrazole-4-carboxamide (CAS) Registration number 1255734-28-1), pydiflumetofen (CAS reg. 1228284-64-7), 3-difluoromethyl-N-methoxy-1-methyl-N-[(1R) -1-methyl- 2- (2,4,6-trichlorophenyl) ethyl] pyrazole-4-carboxamide (CAS Registry No. 1639015-48-7), 3-difluoromethyl-N-methoxy-1-methyl-N-[(1S)- 1-methyl-2- (2,4,6-trichlorophenyl) ethyl] pyrazole-4-carboxamide (CAS registry number 1639015-49-8), 3-difluoromethyl-1-methyl-N- (1,1, 3-to Methylindan-4-yl) pyrazole-4-carboxamide (CAS Registry Number 141573-94-6), 3-Difluoromethyl-1-methyl-N-[(3R) -1,1,3-trimethylindan-4- [Yl] pyrazole-4-carboxamide (CAS Registry No. 1352994-67-2), 3-difluoromethyl-N- (7-fluoro-1,1,3-trimethylindan-4-yl) -1-methylpyrazole-4 -Carboxamide (CAS Registry Number 1383809-87-7), 3-Difluoromethyl-N-[(3R) -7-fluoro-1,1,3-trimethylindan-4-yl] -1-methylpyrazole-4- Carboxamide (CAS registration number 1513466-73-3) etc.

(11) Dithiocarbamate fungicides ferbam (ferbam), mancozeb or manzeb (mancozeb or manzeb), maneb (maneb), methiram (metiram), propineb (propineb), thiuram (thiram), zineb (zineb), ziram (ziram) )etc.

(12) MBI-R agent (reductase-inhibited melanin biosynthesis inhibitor)
Phthalide (phthalide or phthalide), piroquilone (pyroquilone), tricyclazole (tricyclazole) and the like.

(13) MBI-D agent (Citalon dehydrating enzyme-inhibited melanin synthesis inhibitor)
Carpropamide (carpropamide), diclocymet (diclocymet), phenoxanyl (fenoxanil) and the like.

(14) Other fungicides acibenzolar S-methyl (acibenzolar-S-methyl), ametoctradine (ametoctradin), amisulblom (amisulbrom), anilazine (anilazine), biphenyl (biphenyl), blastsaidin S (basticidin-S), bupirimate bupirimate, captaphor, captan, quinomethionate or quinomethionate, chloroneb, chlorothalonil, bromothalonil, cyazofamide ), Dichlofluanid, diclomezine, dichloran, dietofrancarb, diethofencarb, diflumetorim, dimethirimol, dinocap, ditianano). (Dithianon), dodine (dodine), ecromezole or etridiazole (echlomezol or etridiazole), edifenphos (edifenphos), ethaboxam (ethaboxam), etiymol (ethirimol), fenhexamid (fenhexamid), fenpyrazamine (fenpyrazamine), triphenyl tin acetate fentin acetate, triphenyltin chloride, fentin hydroxide, fenmin hydroxide, ferimzone, fluazinam, fluopicolide, fluoroimide, fluulfamide, flutinil (flutinil) flutianil), phorpet (folpet), fluorophorpet (fluorofolpet), fosetyl (fosetyl), guazatine (guazatine), hymexazole (hymexazol), iminoctadine (iminoctadine), iminoctadine triacetate (iminoctadine triacetate) , Iodocarb (iodocarb), iprobenphos (iprobenfos), isoprothiolane (isoprothiolane), isotianil (isotianil), kasugamycin (kasugamycin), laminarin (laminarin), meptyldinocap, methasulfocarb (methasulfocarb), mephene metraphenone , Octilinone, oxathiapiprolin (oxathiapiprolin), oxolinic acid (oxolinic acid), oxytetracycline (oxytetracycline), pencicuron (pencycuron), picalbutrazox (picarbutrazox), phosphorous acid (phosphorous acid), phosphorous acid Acid sodium salt (sodium phosphate), ammonium phosphite (ammonium phosphate), potassium phosphite (potassium phosphate), polyoxins (polyoxins), probenazole (probenazole), propamocarb (propamocarb), proquio Zido (proquinazid), prothiocarb (prothiocarb), pyrazophos (pyrazophos), pyributicarb (pyributicarb), pyriofenone (pyriofenone), quinoxyfen (quinoxyfen), quintozene (quintozene), streptomycin, tebufloquine (tebufoloquine) Teknazen (tecnazene), thiazinyl (tiadinil), tolclophos-methyl (tolclofos-methyl), tolfenpyrad (tolfenpyrad), tolylfluanid (tolylfluanid), tolprocarb (tolprocarb), triazoxide (triazole), validamycin A (validamycinazoxamide, ), Propamidine (propamidine), thymol (Thymol), garlic extract (extract of Allium sativum), Quillaja plant extract (Quillaja extract), veratrine (Veratrine), kaurenguka extract (extract o) f Tropaeolum majus), oak leaves and bark (leaves and bark of Quercus), mustard powder (Yellow mustard powder), extractive extract of Equisetum arvense, chitin (Chitin), saponin of quinoa (Saponins of Chenopodium quinoa) , Basic copper chloride, cupric hydroxide, basic copper sulfate, dodecylbenzenesulfonic acid bisethylenediamine copper complex salt [II] (dodecylbenzenesulfonic acid bisethylenediamine copper [II] salt, DBEDC), organic copper, sulfur (3) -Chloro-5-phenyl-6-methyl-4- (2,6-difluorophenyl) pyridazine (CAS registration number 1358061-55-8), 3-cyano-5-phenyl-6-methyl-4- (2, 6-Difluorophenyl) pyridazine (CAS registration number 1358061-60-5), the following formula (a)

A compound represented by the formula (CAS registration number 517875-34-2), the following formula (b)

Compound represented by (CAS registration number 167173-85-5), the following formula (c)

Of the compound represented by the formula (CAS registration number 1202946-82-4), dipimethitrone (dipymetitrone, CAS registration number 16114-35-5), N '-[4-({3-[(4-chlorophenyl) methyl] -1 , 2,4-thiadiazol-5-yl} oxy) -2,5-dimethylphenyl] -N-ethyl-N-methylmethaneimidamide (CAS registration number 1202781-91-6), 3- (4,4- Difluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl) quinoline (CAS Registry Number 861647-84-9), 2- {3- [2- (1-{[3,5-bis ( Difluoromethyl) -1H-pyrazol-1-yl] acetyl} piperidin-4-yl) -1,3-thiazol-4-yl] -4,5-dihydro-1,2-oxazol-5-yl} -3 -Chlorophenyl = methanesulfonate (CAS registration No. 1360819-11-9), 4- (2-bromo-4-fluorophenyl) -N- (2-chloro-6-fluorophenyl) -1,3-dimethyl-1H-pyrazol-5-amine (CAS registration No.) 136247 7-26), 3- (3,4-Dichloroisothiazol-5-ylmethoxy) -benzoisothiazole 1, 1-dioxide (CAS Registry No. 95714 4-77-3), 2, 2-dimethyl-9- Fluoro-5- (quinolin-3-yl) -2,3-dihydro-benzo [f] [1,4] oxazepine (CAS Registry Number 1207749-50-5), 2- [6- (3-fluoro-4) -Methoxyphenyl) -5-methylpyridin-2-yl] quinazoline (CAS Registry Number 1257056-97-5), 5-fluoro-2-[(4-methylphenyl) methoxy] -4-pyrimidinamine (CAS Registry Number) 1174376-25-0), 5-fluoro -4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2 (1H) -one (CAS Registry No. 1616664-98-2), N '-(2,5-dimethyl-4-phenoxyphenyl) ) -N-Ethyl-N-methylmethanimidamide (CAS Registry No. 10526288-31-9), phenamacryl (phenamacril CAS Registry No. 3336-69-4), (2Z) -3-amino-2-cyano-3-cyano-3- Ethyl phenylacrylate (CAS Registry No. 39491-78-6), N-[(2-Chlorothiazol-5-yl) methyl] -N-ethyl-6-methoxy-3-nitropyridin-2-amine (CAS Registry) No. 1446247-98-8) etc. is mentioned.

As components of insecticides and acaricides included in Group B, for example, (1A) carbamate-based acetylcholine esterase inhibitor alanical (alanycarb), aldicarb (aldicarb), bendioo carub (bendiocarb), benfracarb (benfuracarb), butto Carboxim (butocarboxim), butoxycarboxim (butoxycarboxim), carbaryl (carbaryl: NAC), carbofuran (carbofuran), carbosulfan (carbosulfan), ethiophene carb (ethiofencarb), fenobucarb (fenobucarb: BPMC), hormenate (formetanate), frathiocarb (Furathiocarb), isoprocarb (isoprocarb: MIPC), methiocarb (methiocarb), methomil (methomyl), metolcarb (metolcarb), oxamyl (oxamyl), pyrimicarb (pirimicarb), propoxur (propoxur: PHC), thiodicarb (thiodicarb) b) Thiofanox, triazamate, trimethacarb, XMC, xylylcarb and the like.

(1B) Organophosphorus acetylcholinesterase inhibitors acephate, azamethiphos, azinphos-ethyl, azinphos-methyl, cadusafos, chlorethoxiphos, chlorfenvinphos (chlorfenvinphos) ), Chlormephos (chlormephos), chlorpyrifos (chlorpyrifos), chlorpyrifos-methyl (chlorpyrifos-methyl), coumaphos (coumaphos), cyanophos (cyanophos: CYAP), demeton-S-methyl (demeton-S-methyl), diazinon (diazinon), Dichlorvos (DDVP), dicrotophos, dimethoate, dimethoate, dimethylvinphos, disulfoton (disulfoton), EPN, ethion, ethoprophos (ethoprophos), fenfur (famphur), fenamimi Scan (fenamiphos), fenitrothion (MEP), fenthion (MPP), phosthiazate (fosthiazate), heptenophos (heptenophos), imiciaphos (imicyafos), isofenphos (isofenphos), isopropyl-O- (methoxyaminothiophosphoryl) salicylate Or isocarbophos (isopropylaminothiophosphoryl) salicylate or isocarbophos), isoxathion (isoxathion), malathion (malathion), mecarbam (mecarbam), methamidophos (methamidophos), methidathion (DM), methinphos monocrotophos), nared (BRP), omethoate, oxydemeton-methyl, parathion, parathion-methyl or parathion-methyl or methyl parathion, Phenthoate (PAP), phorate (phorate), phosalone (phosalone), phosmet (phosmet) (PMP), phosphamidon (phosphamidon), phoxim (phoxim), pirimiphos-methyl (pirimiphos-methyl), profenophos (profenofos), propetamphos (propetamphos) Prothiofos, pyraclofos, pyridaphenthion, quinalphos, sulphotep, tebupirimphos, temephos, temphos, terbufos, tetrachlorvin phos (Thiometon), triazophos (triazophos), trichlorfon (trichlorfon: DEP), vamidothion and the like.

(2) GABAergic chloride channel blocker ethiprole, fipronil (fipronil), flufiprole (flufiprole), chlordane (chlordane), endosulfan (endosulfan), alpha endosulfan (alpha-endosulfan) and the like.

(3) GABAergic Chloride Channel Allosteric Modulator Afoxorana (afoxalaner), fluralaner (fluralaner), brofuranilide (broflanilide), fluxamethamide (fluxametamide) and the like.

(4) Sodium Channel Modulators Achrinathrin (acrinathrin), allethrin (allethrin), bifenthrin (bifenthrin), kappa bifenthrin (kappa-bifenthrin), bioallethrin (bioallethrin), bioresmethrin (bioresmethrin), cycloprothrin (cycloprothrin), cyfluthrin (cyfluthrin) ), Beta cyfluthrin (beta-cyfluthrin), cyhalothrin (cyhalothrin), gamma cyhalothrin (gamma-cyhalothrin), lambda cyhalothrin (lambda-cyhalothrin), cypermethrin (cypermethrin), alpha cypermethrin (alpha-cypermethrin) , Betacypermethrin (beta-cypermethrin), theta-cypermethrin (theta-cypermethrin), zetacypermethrin (zeta-cypermethrin), sigmacypermethrin (sigma-cypermethrin), cypenothrin (cyphenothrin), deltamethrin (deltamethrin) ), Empenthrin, esfenvalerate, etofenprox, fenpropathrin, fenvalerate, flucythrinate, flumethrin, fluvalinate (fluvalinate) ), Taufluvalinate (Tau-fluvalinate), Halfenprox (halfenprox), Heptafluthrin (Heptafluthrin), Imiprothrin (imiprothrin), Kadethrin (kadethrin), Meperfluthrin (meperfluthrin), Monfluorothrin (momfluorthrin), Permethrin (permethrin) ), Phenothrin (phenothrin), prarethrin (prallethrin), pyrethrin (pyrethrins), resmethrin (resmethrin), silafluofen (silafluofen), tefluthrin (tefluthrin), kappa tefluthrin (kappa-tefluthrin), Tramethrin (tetramethrin), tetramethylfluthrin (tetramethylfluthrin), tralomethrin (tralomethrin), transfluthrin (transfluthrin), benfluthrin (benfluthrin), flufenprox (flufenoprox), flumethrin (flumethrin), framethrin (furamethrin), methofutrin (metofluthrin) ), Profluthrin (profluthrin), dimefluthrin (dimefluthrin), epsilon methofluthrin (epsilon-metofluthrin), 2,3,5,6-tetrafluoro-4-methylbenzyl (EZ)-(1 RS, 3 RS; 1 RS, 3 SR) 2,2-Dimethyl-3-prop-1-enylcyclopropane carboxylate, 2,3,5,6-tetrafluoro-4- (methoxymethyl) benzyl (1 RS, 3 RS; 1 RS, 3 SR) -2, 2 -Dimethyl-3- (2-methyl) 1-propenyl) cyclopropanecarboxylate, epsilon Mont fluoro Trinh (epsilon-momfluorothrin), methoxychlor (methoxychlor), and the like.

(5) Nicotinic acetylcholine receptor competitive modulator acetamiprid (acetamiprid), clothianidin (clothianidin), dinotefuran (dinotefuran), imidacloprid (imidacloprid), nitenpyram (nitenpyram), thiacloprid (thiacloprid), thiamethoxam (sulfathiofloxa) (Flupyradifurone), triflumezopyrin (triflumezopyrim), dichloro mesothias (dicloromezotiaz), cycloxaprid (cycloxaprid), the following formula (d)

And the like (CAS registration number 1363400-41-2) and the like.

(6) Glutamatergic Chloride Channel Allosteric Modulator Abamectin (abamectin), emamectin benzoate (emamectin-benzoate), lepimectin (lepimectin), milbemectin and the like.

(7) Juvenile hormone analogues hydroprene (hydroprene), kinoprene (kinoprene), methoprene (methoprene), fenoxycarb, pyriproxyfen and the like.

(8) Other nonspecific (multisite) inhibitors methyl bromide, chloropicrin, sulfuryl fluoride, borax, boric acid, octaboric acid Disodium acid (disodium octaborate), sodium borate (sodium borate), sodium metaborate (sodium metaborate), tartaric acid (tartar emetic), dazomet (dazomet), metam (metam) and the like.

(9) Acaricide Growth Inhibitor Clofenthezine, hexythiazox, diflovidazin, etoxazole and the like.

(10) Mitochondrial ATP synthetase inhibitor diafenthiuron (diafenthiuron), azocyclotin (azocyclotin), cyhexatin (cyhexatin), fenbutatin oxide oxidized, propargite (propargite), tetradiphone (tetradifon) and the like.

(11) Oxidative phosphorylation uncoupling agent chlorfenapyr (DN), DNOC, sulfluramid etc.

(12) Nicotinic acetylcholine receptor channel blocker bensultap, cartap (cartap), cartap hydrochloride (cartap hydrochloride), thiocyclam (thiocyclam), thiosultap-2 sodium salt or bisultap (thiosultap-disodium or bisultap), thiosultap- Monosodium salt or monosultap (thiosultap-monosodium or monosultap) and the like.

(13) Benzoylurea-based chitin biosynthesis inhibitors bistrifluron (bistrifluron), chlorfluazuron (chlorfluazuron), diflubenzuron (diflubenzuron), fluazuron (fluazuron), flucycloxron (flucycloxuron), flufenoxuron , Hexaflumuron, lufenuron, novallon, noviflumuron, teflubenzuron, triflumuron and the like.

(14) Moulting hormone (ecdysone) receptor agonist chromafenozide, halofenozide, methoxyfenozide, tebufenozide and the like.

(15) Mitochondrial electron transport complex III inhibitor hydramethylnon (hydramethylnon), acequinocyl (acequinocyl), fluacripyrim (fluacrypyrim), bifenazate etc.

(16) Mitochondrial electron transport complex I inhibitor phenazaquin (fenazaquin), fenpyroximate, pyridaben (pyridaben), pyrimidifen (pyrimidifen), tebufenpyrad (tebufenpyrad), tolfenpyrad (tolfenpyrad), rotenone (rotenone) and the like.

(17) Acetyl-CoA carboxylase inhibitor spirodyclofen, spiromesifen, spirotetramat and the like.

(18) Mitochondrial electron transport complex IV inhibitor aluminum phosphide, calcium phosphide, hydrogen phosphine, phosphine, zinc phosphide, calcium cyanide , Potassium cyanide (potassium cyanide), sodium cyanide (sodium cyanide) and the like.

(19) Mitochondrial electron transport complex II inhibitor cienopyraphen (cyenopyrafen), ciflumethofen (cyflumetofen), pyflubumide etc.

(20) Ryanodine receptor modulators chlorantraniliprole (cyanoraniliprole), cyanantranilprole (cyantraniliprole), cyclaniliprole (cycliliporole), flubendiamide (flubendiamide), tetraniliprole (tetraniliprole), cyhalodiamide (cyhalodiamide), Formula (e)

And the like (SYP-9080; CAS Registry No. 1104384-14-6) and the like.

(21) Natural Insecticides Nicotine (nicotine), Nicotine Sulfate (nicotine-sulfate), Neem oil (Neem tree (Azadirachta indica) oil), Shrimp nigrum wood extract (wood extract of Quasisia amara), Rianodine (Ryanodine), Extract of Mistletoe extract (extract of Viscum album), Extract of Tansy extract (Extract of Tanacetum vulgare), Extract of Artemisia absinthium, Extract of Stinging Nettle (extract of Urtica dioica), Extract of Symbitum of extract , Citrus seed oil (oil of the seeds of Chenopodium anthelminticum), dried leaves of dried leaves (dried leaves of Dryopteris filix-mas), Celastrus angulatus bark (bark of Celastrus angulatus), extract of Citrus oryzae (natural extracts or simulated bound of Chenopodium ambrosioides), Cassia nigricans extract (extract of Cassia nigricans) etc.

(24) Other Insecticides / Acaricides / Nematocides Spinetoram (Spinetoram), Spinosad (Spinosad), Pimetrozine (Pymetrozine), Pyrifluquinazone (Pyrifluquinazone), Buprofezin (buprofezin), Cyromazine (Cyromazine), Amitraz (amitraz), India Xacarb (indoxacarb), metaflumizone (metaflumizone), flonicamid (flonicamid), azadirachtin (azadirachtin), benzoximate (benzoxiate), bromopropyrate (bromopropylate), quinomethionate (chinomethionat), dicofol (dicofol), pyridaryl, Lime-sulfur combination (lime sulfur), sulfur (sulfur), afidopyropene, fluazaindolizine (fluazaindolizine), fluenesulfone (fluensulfone), flomethoquin (flometoquin), methoxadiazon (metoxadiazone), pyriminostroline Down (pyriminostrobin), Chiokisazafen (tioxazafen), machine oil (machine oil), aluminum fluoride sodium (sodium aluminium fluoride or chiolite), the following formula (f)

And the stereoisomers thereof, the following formula (g):

Embedded image (CAS registration number 1118626-57-5) and its stereoisomer, the following formula (h)

A compound represented by the following formula (CAS registration number 1239276-34-6), the following formula (i)

A compound represented by the formula (CAS registration number 1204608-98-9), the following formula (j)

Compound (CAS registration number 1353559-47-3), the following formula (k)

A compound represented by the formula (CAS registration number 1229023-00-0), the following formula (I)

A compound represented by the formula (CAS registration number 1477919-27-9), the following formula (m)

And the stereoisomers thereof, the compound represented by the following formula (n):

A compound represented by the formula (CAS registration number 1429513-53-0), the following formula (o)

A compound represented by the formula (CAS registration No. 1609007-65-9), the following formula (p)

A compound represented by the formula (CAS registration number 885026-50-6), the following formula (q)

And the like.

(16) synergist Piperonyl butoxide, sesamex, sulfoxide, N- (2-ethylhexyl) -8,9,10-trinorlborn-5-ene-2,3-dicarboxy Imide (MGK 264), N-declyimidazole (N-declyimidazole), WARF-antiresistant (WARF-antiresistant), TBPT (S, S, S, S-tributyl phosphorothioate), TPP (triphenyl phosphate), IBP Diisopropyl S-benzyl phosphorothiolate, PSCP (phenyl saligenin cyclic phosphonate), methyl iodide (CH ₃ I), t-phenylbutenone (t-phenylbutone), diethyl maleate (diethylmaleate), DMC (1,1-bis-) (p-chloro-phenyl) methyl carbinol), FDMC (bis- (p-chlorophenyl) -trifluoromethyl caxbinol), ETP (1,1,1-trichloro-2,3-expoxypropane), ETN (1,2-epoxy-) 1,2,3,4-tetrahydronapthale ne) etc.

The components of the herbicides included in Group C include, for example, clodinafop, clodinafop-propargyl, cyhalofop, cyhalofop-butyl, diclofop, diclofop Hop methyl (diclofop-methyl), fenoxaprop (fenoxaprop), fenoxaprop-ethyl (fenoxaprop-ethyl), fenoxaprop P (fenoxaprop-P), fenoxaprop P-ethyl (fenoxaprop-P-ethyl), fluazifop ( fluazifop), fluazifop-butyl, fluazifop-P, fluazifop-P-butyl, haloxyfop, haloxyfop-methyl, haloxyfop P haloxyfop-P), haloxyfop P-methyl (haloxyfop-P-methyl), metamifop , Propaquizafop, quizalohop (quizalofop), quizalohop-ethyl (quizalofop-ethyl), quizalo-hop P (quizalofop-P), quizalo-hop P ethyl (quizalofop-P-ethyl), alloxydim (alloxydim), butroxydim (butroxydim) ), Clethodim, cycloxydim, propoxydim, profoxydim, cetoxydim, tepraloxydim, tralkoxydim, pinoxaden, amidosulfuron, amidulsulfuron azimsulfuron), bensulfuron (bensulfuron), bensulfuron methyl (bensulfuron-methyl), chlorimuron (chlorimuron), chlorimuron ethyl (chlorimuron-ethyl), chlorsulfuron (chlorosfurfuron), chinosulfuron (cinosulfuron), cyclosulfamuron ( cyclosulfam uron), etamethsulfuron (ethamethsulfuron), etamethsulfuron-methyl (ethamethsulfuron-methyl), ethoxysulfuron (ethoxysulfuron), flazasulfuron (flazasulfuron), flucetosulfuron (flucetosulfuron), flupyrsulfuron (flupyrsulfuron), flupyrus Ruflon methyl sodium (flupyrsulfuron-methyl-sodium), phoramsulfuron (foramsulfuron), halosulfuron (halosulfuron), halosulfuron methyl (halosulfuron-methyl), imazosulfuron (imazosulfuron), iodosulfuron (iodosulfururon), iodosulfuron methyl sodium (Iodosulfuron-methyl-sodium), iofensulfuron (iofensulfuron), iofensulfuron sodium (iofensulfuron-sodium), mesosulfuron (mesosulfuron), mesosulfuron methyl (mesosulfuron-methyl), metazosulfuron (metazosulfuron) ), Methsulfuron (metsulfuron), methsulfuron methyl (metsulfuron-methyl), nicosulfuron (nicosulfuron), orthosulfamuron (orthosulfamuron), oxasulfuron (oxasulfuron), primisulfuron (primisulfuron), primisulfuron methyl (primisulfuron) -methyl), propyrisulfuron, prosulfuron (prosulfuron), pyrazosulfuron (pyrazosulfuron), pyrazosulfuron-ethyl (pyrazosulfuron-ethyl), rimsulfuron (rimsulfuron), sulfometuron, sulfometuron methyl (sulfometuron- methyl), sulfosulfuron (sulfosulfuron), thifensulfuron (thifensulfuron), thifensulfuron-methyl (thifensulfuron-methyl), triasulfuron (triasulfuron), tribenuron (tribenuron), tribenuron methyl (tribenuron-methyl), Rifuloxysulfuron sodium salt (trifloxysulfuron-sodium), trifloxysulfuron (trifloxysulfuron), triflusulfuron (triflusulfuron), triflusulfuron methyl (triflusulfuron-methyl), tritosulfuron (tritosulfuron), imazapic (imazapic), imimapic Thepic ammonium salt (imazapic-ammonium), imazamethabenz (imazamethabenz), imazamethabenzmethyl (imazamethabenz-methyl), imazamox (imazamox), imazamox ammonium salt (imazamox-ammonium), imazapyr (imazapyr), imazapyr Isopropyl ammonium salt (imazapyr-isopropylammonium), imazaquin (imazaquin), imazaquin ammonium salt (imazaquin-ammonium), imazethapyr, imazethapyr ammonium salt (imazethapyr-ammonium), cloransulam, cloransulam Methyl (cloransulam-methyl), diclosulam, florasulam, flumetsulam, flumetsulam, metosulam, penoxsulam, pyroxsulam, pyroxisulam, bispyribac Sodium salt (bispyribac-sodium), pyribenzoxim, pyriphthalide, pyriminobac, pyriminobac-methyl, pyrithiobac, pyrithiobac sodium salt, pyrithiobac-sodium, pyrithiobac-sodium Misulfan (pyrimisulfan), triafamone (triafamone), flucarbazone (flucarbazone), flucarbazone sodium salt (flucarbazone-sodium), propoxycarbazone (propoxycarbazone), propoxycarbazone sodium salt (propo xycarbazone-sodium, thiencarbazone, thiencarbazone-methyl, ametrine, atrazine, atrazine, cyanazine, cyanazine, desmetryn, dimethamethrin, prometon, promethon Promethrin (prometryn), propazine (propazine), simazine (simazine), simetryn (simetryn), terubumeton (terbumeton), terbutylazine (terbuthylazine), terbutrin (terbutryn), trietadine (trietazine), hexazinone (hexazinone), metamitrone, Metribuzin (metribuzin), amicarbazone (amicarbazone), bromacil (bromacil), lenacil (lenacil), terbacil (terbacil), chloridazon (chloridazon), desmedipham (desmedipham), phenmedipham, crodida Bromron (chlorobromuron), Chlorotoluron, chloroxuron, dimefron (dimefuron), diuron (diuron), etidimuron (ethidimuron), phenuron (fenuron), fluometuron, isoproturon (isoproturon) Linuron (linuron), benzthiazuron, benzthiazuuron (methabenzthiazuron), metobromuron (metobromuron), metoxuron (metoxuron), monolinuron (monolinuron), nebron (neburon), siduron (siduron), tebutiuron (tebutiruon) (Propanil), pentanochlor (pentanochlor), bromophenoxim (bromofenoxim), bromoxynil (bromoxynil), bromoxynil octanoate (bromoxynil-octanoate), ioxynil (ioxynil), Oxynyl octanoate (ioxynil-octanoate), bentazone (bentazon), cyclopyrimorate (cyclopyrorate), pyridate (pyridate), pyridafol (pyridafol), diquat (diquat), diquat dibromide (diquat-dibromide), paraquat (paraquat (diquat) paraquat), paraquat-dichloride, acifluorfen (acifluorfen), acifluorfen sodium salt (acifluorfen-sodium), bifenox (bifenox), chloromethoxyphen (chlomethoxyfen), ethoxyphenethyl (ethoxyfen-ethyl), Fluoroglycophene ethyl (flouroglycofen-ethyl), fomesafen (fomesafen), fomesafen sodium (fomesafen-sodium), halosafene (halosafen), lactofen (lactofen), oxyfluorfen (oxyfluorfen), fluazolate (fluazolate), pyraflufene (Pyraflufen-ethyl), cinidone (cinidon), cinidone ethyl (cinidon-ethyl), flumicrolac (flumiclorac), flumicrolac pentyl (flumiclorac-pentyl), flumioxazin (flumioxazin), fluthiaset (fluthiacet), fluthiaset Methyl (fluthiacet-methyl), thidiazimin (thidiazimin), oxadiazone (oxadiazon), oxadiargyl (oxadiargyl), azaphenidine (azafenidin), bencarbazone (bencarbazone), carfentrazone (carfentrazone), carfentrazone ethyl (carfentrazone-ethyl) , Sulfentrazone (sulfentrazone), pentoxazone (pentoxazone), benzphendizone (benzfendizone), butafenacil (butafenacil), saflufenacil (saflufenacil), tiafenacil (tiafenacil), pyraclonil (pyraclonil), proflua zoole (profluazo) l) flufenpyr (flufenpyr), flufenpyrethyl (flufenpyr-ethyl), trifludimoxazine (trifludimoxazin), norflurazon (norflurazon), diflufenican (diflufenican), pyrocolinafen (picolinafen), beflubutamide (beflubutamido), fluridone (fluridone) fluridone, flurochloridone, flurtamone, fenquinotrione, mesotrione, mesotrione, sulcotrione, tefuryltrione, tebotrione, isoxachlorol ( isoxachlortole), isoxaflutole, benzofenap, pyrasulfotole, pyrazolynate, pyrazoloxifen, topramezone, topramezone, benzobicyclon benzobicyclone), bicyclopyrone, tolpyralate, tolpyralate, amitrole, aclonifen, aclonifen, clomazone, glyphosate, glyphosate isopropylamine salt, glyphosate isopropylamine salt, trisodium salt salt Glyphosate-trimethylsulfonium), Glyphosate ammonium salt (glyphosate-ammonium), Glyphosate diammonium salt (glyphosate-diammonium), Glyphosate sodium salt (glyphosate-sodium), Glyphosate potassium salt (glyphosate-potassium), Glyphosate guanidine derivative salt (metallic electrolyte) Glyphosate choline salt, Glyphosate BAPMA (glyphosate N, N-Bis (3-aminopropyl) methylamine salt), glufosinate, glufosinate ammonium salt Salt (glufosinate-ammonium), glufosinate P (glufosinate-P), glufosinate P sodium salt (glufosinate-P-sodium), glufosinate P ammonium salt (glufosinate-P-ammonium), bialaphos (bialafosbialaphos), asulam (asulam), benfluraline (Benfluralin), butoralin (butralin), dinitramine (dinitramine), etalfluralin (ethalfluralin), oryzalin (oryzalin), pendimethalin (pendimethalin), trifluralin (trifluralin), amiprofos methyl (amiprophos-methyl), butamiphos ( butamifos), dithiopyr (thiazolopyr), prodiamine (prodiamine), propizamide (propyzamide), tebutam, DCPA (chlorothal-dimethyl), chlorprofam (chlorpropham), profam (propham) ), Carbetamide (carbetam) ide), flumprop-M, acetochlor, alachlor, alachlor, butachlor, butachlor, dimethachlor, dimethenamid, dimethenamid P, dimethenamid-P, metazachlor metazachlor), metolachlor, S-metolachlor, pethoxamid, pettiloxal, pretilachlor, propachlor, propisochlor, propyochlor, thenylchlor, diphenamide ), Napropamide (napropamide), Napropamide M (napropamide-M), Naproanilide (naproanilide), Flufenacet (flufenacet), Mefenacet (mefenacet), Fentrazamide (fentrazamide), Ipfencarbazone (ipfencarbazone), Anilofos (anilofos) Fencetrol (cafenstrole), piperophos (piperophos), pyroxasulfone (pyroxasulfone), fenoxasulfone (fenoxasulfone), diclobenil (dichlobenil), chlorthiamide (chlorthiamide), isoxaben (isoxaben), flupoxam (flupoxam), indaziflam (indaziflam) Triaziflam (triaziflam), DNOC (2-methyl-4,6-dinitrophenol), dinoseb, dinoterb (dinoterb), butyrate (butylate), cycloate (cycloate), dialate (di-allate), dimepiperate (dimepiperate), EPTC (S-ethyl N, N-dipropylcarbathioate), esprocarb (esprocarb), molinate (molinate), orbencarb (orbencarb), pebulate (pebulate), prosulcarb (prosulfocarb), benthiocarb (benthiocarb), thiocal basil (tiocarbazil) tri-al late, vernolate, bensulide, benfuresate, benfuresate, ethofumesate, TCA (2,2,2-trichloroacetic acid), dalapone (dalapon), flupropanate, chromeprop ( clomeprop), 2,4-D (2- (2,4-dichlorophenoxy) acetic acid), 2,4-D ammonium (2,4-D-ammonium, ammonium 2- (2,4-dichlorophenoxy) acetate), 2,4-D-Butyl (2,4-D-butyl, 2-butoxyethyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D 2-butoxypropyl (2,4-D-2-butoxypropyl, 2-butoxypropyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D 3-butoxypropyl (2,4-D-3-butoxypropyl, 3-butoxypropyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D-butyl (2,4-D-butyl, butyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D-diethylammonium (2,4-D-diethylammonium, 2- (2,4 (2,4) -dichlorophenoxy) acetic acid compound with N-ethylethanamine (1: 1), 2,4-D-dimethylammonium, 2- (2,4-dichlorophenoxy) acetic acid compound with N-methylmethanamine (1: 1) ), 2,4-D diol amine salt (2,4-D-diolamine, 2- (2,4-dichlorophenoxy) acetic acid compound with 2,2'-iminobis [ethanol] (1: 1)), 2, 4-D-dodecylammonium (2,4-D-dodecyl lammonium, 2- (2,4-dichlorophenoxy) acetic acid compound with 1-dodecanamine (1: 1)), 2,4-D-ethyl (2,4-D- ethyl, ethyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D 2-ethylhexyl (2,4-D-2-ethylhexyl, 2-ethylhexyl 2- (2,4-dichlorophenoxy) acetate), 2 , 4-D heptyl ammonium (2,4-D-heptalammonium, 2- (2,4-dichlorophenoxy) acetic acid compound with 1-heptanamine (1: 1)), 2,4-D isobutyl (2,4-D) -isobutyl, 2-methylpropyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D isooctyl (2,4-D-isooctyl, isoocty) l 2- (2,4-dichlorophenoxy) acetate), 2,4-D isopropyl (2,4-D-isopropyl, 1-methylethyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D isopropyl ammonium (2,4-D-isopropylammonium, 2- (2,4-dichlorophenoxy) acetic acid compound with 2-propanamine (1: 1)), 2,4-D lithium (2,4-D-lithium, lithium 2-) (2,4-dichlorophenoxy) acetate), 2,4-D-meptyl (2,4-D-meptyl, 1-methylheptyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D-methyl (2,4 (dichlorophenoxy) acetate) -D-methyl, methyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D-octyl (2,4-D-octyl, octyl 2- (2,4-dichlorophenoxy) acetate), 2,4- D pentyl (2,4-D-pentyl, pentyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D-propyl (2,4-D-propyl, propyl 2- (2,4-dichlorophenoxy) acetate ), 2,4-D sodium salt (2,4-D-sodium, sodium 2- (2,4-dichlorophenoxy) acetate), 2,4-D tefuryl (2,4-D-tefuryl, (tetrahydro-2) -furanyl) methyl 2- (2,4-dichlorophenoxy) acetate), 2,4-D tetradecyl ammonium (2,4-D-tetradecylcylammonium, 2- (2,4-dichlorophenoxy) acetic acid compound with 1-tetradecacanamine (1: 1)), 2,4-D triethylammonium (2- (2,4-dichlorophenoxy) acetic acid compound with N, N-diethylethanamine (1: 1)), 2,4-D tris (2- Hydroxypropyl) ammonium (2,4-D-tris (2-hydroxypropyl) ammonium, 2- (2,4-dichlorophenoxy) acetic acid compound with 1,1 ′, 1 ′ ′-nitrilotris [2-propanol] (1: 1 ), 2,4-D trolamine salt (2,4-D-trolamine salt, 2- (2,4-dichlorophenoxy) acetic acid compound with 2,2 ′, 2 ′ ′-nitrilotris [ethanol] (1: 1) ), 2,4-D choline salt (2,4-D choline salt, 2- (2,4-dichlorophenoxy) acetic acid compound with 2-hydroxy-N, N, N-trimethylethanamine (1: 1)), 2,4-D BAPMA salt (2,4-DN, N-bis- (3-aminopropyl) methylamine salt, 2- (2,4-dichlorophenoxy) acetic acid compo und with N, N-bis- (3-aminopropyl) methylamine (1: 1)), 2,4-DB (4- (2,4-dichlorophenoxy) butanoic acid), 2,4-DB dimethyl ammonium (2, 2, 3) 4-DB-dimethylammonium, 4- (2,4-dichlorophenoxy) butanoic acid compound with N-methylmethanamine (1: 1), 2,4-DB isooctyl (2,4-DB-isooctyl, isooctyl 4- (2, 4-dichlorophenoxy) butanol), 2,4-DB butyl (2,4-DB-butyl, butyl 4- (2,4-dichlorophenoxy) butanoate), 2,4-DB sodium salt (2,4-DB-sodium) Sodium, 4- (2,4-dichlorophenoxy) butanoate, 2,4-DB potassium salt (2,4-DB-potassium, potassium 4- (2,4-dichlorophenoxy) butanoate), 2,4-DB choline salt (2,4-DB choline salt, 4- (2,4-dichlorophenoxy) butanoic acid compound with 2-hydroxy-N, N, N-trimethylethanamine (1: 1)), 2,4-DB BAPMA salt (2 ,, 4-DB N, N-bis- (3-aminopropyl) methylamine salt, 4- (2,4-dichlorophenoxy) butanolic acid compound with N, N-bis- (3-aminopropyl) methylam ine (1: 1), MCPA (2- (4-chloro-2-methylphenoxy) acetic acid), MCPA dimethylammonium (MCPA-dimethylammonium, 2- (4-chloro-2-methylphenoxy) acetic acid compound with N- methylmethanamine (1: 1), MCPA 2-ethylhexyl (MCPA-2-ethylhexyl, 2-ethylhexyl 2- (4-chloro-2-methylphenoxy) acetate), MCPA isooctyl (MCPA-isoctyl, isooctyl 2- (4-chloro) -2-methylphenoxy) acetate), MCPA butytyl (MCPA-butyl, 2-butoxyethyl 2- (4-chloro-2-methylphenoxy) acetate), MCPA butyl (MCPA-butyl, butyl 2- (4-chloro-2-methylphenoxy) ) acetate), MCPA diolamine salt (MCPA diolamine salt, 2- (4-chloro-2-methylphenoxy) acetic acid compound with 2,2'-iminobis [ethanol] (1: 1)), MCPA ethyl (MCPA-ethyl) , Ethyl 2- (4-chloro-2-methylphenoxy) acetate), MCPA isobutyl (MCPA-isobutyl, 2-methylpropyl 2- (4-chloro-2-methylphenoxy) acetate), MCPA isopropyl (MCPA -isopropyl, 1-methylethyl 2- (4-chloro-2-methylphenoxy) acetate), MCPA methyl (MCPA-methyl, methyl 2- (4-chloro-2-methylphenoxy) acetate), MCPA allamine salt (MCPA olamine salt , 2- (4-chloro-2-methylphenoxy) acetic acid compound with 2-aminoethanol (1: 1), MCPA sodium salt (MCPA-sodium, sodium 2- (4-chloro-2-methylphenoxy) acetate), MCPA Trollamine salt (MCPA trolamine salt, 2- (4-chloro-2-methylphenoxy) acetic acid compound with 2,2 ′, 2 ′ ′-nitrotritis [ethanol] (1: 1)), MCPA choline salt (MCPA choline salt, 2- (4-chloro-2-methylphenoxy) acetic acid compound with 2-hydroxy-N, N, N-trimethylethanamine (1: 1), MCPA BAPMA salt (MCPA N, N-bis- (3-aminopropyl) methylamine salt, 2- (4-chloro-2-methylphenoxy) acetic acid compound with N, N-bis- (3-aminopropyl) methylamine (1: 1)), MCPB (4- (4-chloro-2-methylphenoxy) butanolic acid, MCPB ethyl (MCPB-ethyl, ethyl 4- (4-chloro-2-methyl) phenoxy) butanolate, MCPB methyl (MCPB-methyl, methyl 4- (4-chloro-2-methylphenoxy) butanoate), MCPB sodium salt (MCPB-sodium, sodium 4- (4-chloro-2-methylphenoxy) butanoate), MCPB choline salt (MCPB choline salt, sodium 4- (4-chloro-2-methylphenoxy) butanoic acid compound with 2-hydroxy-N, N, N-trimethylethanamine (1: 1)), MCPB BAPMA salt (MCBP N, N -bis- (3-aminopropyl) methylamine salt, sodium 4- (4-chloro-2-methylphenoxy) butanoic acid compound N, N-bis- (3-aminopropyl) methylamine (1: 1)), mecoprop (mecoprop), Mecoprop-dimethylammonium, mecoprop diolamine salt, mecoprop-ethadyl, mecoprop-2-ethylhexyl, mecoprop-isocyl (mecoprop-isoctyl) ), Mecoprop methyl (mecoprop-methyl), mecoprop Lilium salt (mecoprop-potassium), mecoprop sodium salt (mecoprop-sodium), mecoprop trolamine salt, mecoprop choline salt, mecoprop P (mecoprop-P), mecoprop P dimethyl Ammonium (mecoprop-P-dimethylammonium), mecoprop P-ethylhexyl (mecoprop-P-2-ethylhexyl), mecoprop-P-isobutyl (mecoprop-P-isobutyl), mecoprop-P potassium salt (mecoprop-P-potassium), mecoprop-P choline salt (Mecoprop-P choline salt), mecoprop BAPMA salt (mecoprop-N, N-bis- (3-aminopropyl) methylamine salt), dicloprop (dichlorprop), dicloprop buttyl (dichlorprop-butotyl), dicloprop dimethylammonium ( dichlorprop-dimethylammonium), dicloprop ethylammonium (dichlorprop-ethylammonium), Dicloprop 2-ethylhexyl (dichlorprop-2-ethylhexyl), dicloprop isoctyl (dichlorprop-isoctyl), dicloprop methyl (dichlorprop-methyl), dicloprop potassium salt (dichlorprop-potassium), dicloprop sodium salt (dichlorprop-sodium) , Dichlorprop choline salt, dicloprop BAPMA salt (dichlorprop N, N-bis- (3-aminopropyl) methylamine salt), dicloprop P (dichlorprop-P), dicloprop P dimethyl ammonium (dichlorprop-P) -dimethylammonium), dicloprop P-diethylprophyl (dichlorprop-P-2-ethylhexyl), dicloprop-P choline salt, dicloprop P-BAPMA salt (dichlorprop-P N, N-bis- (3- aminopropyl) methylamine salt), chloramben, dicamba, dicamba dichloramine (Dicamba diglycolamine salt), dicamba dimethylammonium (dicamba-dimethylammonium), dicambadiol amine salt (dicamba diololate salt), dicamba isopropyl ammonium (dicamba-isopropylammonium), dicamba methyl (dicamba-methyl), dicambaol amine salt (dicamba olamine salt), dicamba potassium salt (dicamba-potassium), dicamba sodium salt (dicamba-sodium), dicamba trolamine salt, dicamba choline salt, dicamba choline salt, dicamba BAPMA salt (dicamba N, N-bis- (3-aminopropyl) methylamine salt), 2,3, 6-TBA (2, 3, 6-trichlorobenzoic acid), 2, 3, 6-TBA dimethyl ammonium (2, 3, 6-TBA-dimethylamm)
onium, 2,3,6-trichlorobenzoic acid compound with N-methylmethanamine (1: 1), 2,3,6-TBA lithium (2,3,6-TBA-lithium, lithium 2,3,6-trichlorobenzoate) 2,3,6-TBA potassium salt (2,3,6-TBAS-potassium, potassium 2,3,6-trichlorobozoate), 2,3,6-TBA sodium salt (2,3,6-TBA-sodium) Sodium, 2, 3, 6-trichlorobozoate, triclopyr, triclopyr-butotyl, triclopyr-ethyl, triclopyr-triethylammonium, triazopyr, Fluoxypyr (fluroxypyr), fluoxypyrmeptyl (fluroxypyr-meptyl), aminopyralid (aminopyralid), aminopyralid potassium salt (aminopyralid-potassium), aminopyralid tris (2-hydroxypropyl) ammonium (aminopyralid-tris (2-hydroxypropyl) ammonium ), A) Nopyralid choline salt (aminopyralid choline salt), clopyralid (clopyralid), clopyralid methyl (clopyralid olamine salt), clopyralid potassium salt (clopyralid-potassium), clopyralid tris (2-hydroxypropyl) ammonium -tris (2-hydroxypropyl) ammonium), clopyralid choline salt, quinclorac, quinmerac, benazolin ethyl (benazolin-ethyl), napthalam (naptalam), diflufenzopyr (diflufenzopyr) , Diflufenzopyr-sodium salt, diphenzoquat (diphenzoquat), DSMA (disodium As-methylarsonate), MSMA (sodium hydrogen As-methylarsonate), bromobutide, bromonide, flurenol, synmethylin ( Cinmethylin, cumyluron, dazomet, daimuron, methyl-daymuron, etobenzanide, etobenzanid, fosamine, indanofan, indanofan, metam, oxaziclomefone , Oleic acid, pelargonic acid, pelibutonic acid, pyributicarb; methiozolin, phenisopham, swep, aminocyclopyrachlor, aminocyclopyrachlor methyl -methyl), aminocyclopyrachlor potassium (aminocyclopyrachlor-potassium), difenoxuron, didinoxuron, tridiphane, maleic hydrazide, ACN (2-amino-3-chloro-1, 4-naphthoquinone), Harauxi E emissions (halauxifen), Halau Shiki Fen methyl (halauxifen-methyl)
Etc.

  The components of the safeners to be included in group D include, for example, benoxacor, cloquintocet-mexyl, ciometrinil, dichlormid, fenchlorazole-ethyl. Fenclorim (fenclorim), flurazole (flurazole), furilazole (furilazole), mefenpyr-diethyl (mefenpyr-diethyl), MG191 (2- (dichloromethyl) -2-methyl-1,3-dioxolane), oxabetrinil (oxabetrinil), Arididol (allidochlor), isoxadiphen-ethyl (isoxadifen-ethyl), cyprosulfamide (cyprosulfamide), fluxophenim (fluxofenim), 1,8- naphthalic anhydride (1,8-naphthalic anhydride), AD-67 ( 4- (dichloroacetyl) -1-oxa-4-azospiro [4.5] decane) and the like.

  Examples of components of plant growth regulators included in Group E include indole butyric acid (4-indol-3-ylbutyric acid), ethychlozate, 1-naphthylacetamide (2- (1-naphthyl) acetamide), 4-CPA (4-chlorophenoxyacetic acid), dichlorprop (trolamine), 1-sodium naphthalene acetate (sodium 1-naphthaleneacetate), MCPB (4- (4-chloro-o-tolyoxy) butyric acid), maleic acid Hydrazide (Maleic hydrazide), Ethephon (ethephon), AVG (aminoethoxyvinylglycine), 1-methylcyclopropene (1-methylcyclopropene), chlormequat (chlormequat-chloride), mepiquat (mepiquat-chloride), gibberellin A3 (Gibberellin A3) Gibberellin A, uniconazole-P, paclobutrazol, flurprimidol, prohexadione cal Sium (prohexandione-calcium), trinexapac-ethyl (trinexapac-ethyl), daminozide (daminozide), abscisic acid (abscisic acid), kinetin (Kinetin), benzyl adenine (benzyladenine), 1,3-diphenylurea, forchlorphenuron (Forchlorfenuron), thidiazuron, prohydrojasmon (prohydrojasmon), aminolevulinic acid acid hydrochloride (5-aminolevulinic acid hydrochloride), pendimethalin (pendimethalin), decyl alcohol (decyl alcohol), butoralin (butralin), asymidol (acymidol) ), Mefluidide (mefluidide), calcium peroxide (caicium peroxide), hydroxy isoxazole (hymexazol), isoprothiolane (isoprothiolane), choline (choline chloride), cyanamide (cyanamide), pyraflufenyl (pyraflufen-ethyl), Diquat diquat dibromide, streptomycin, sodium cyanate, calcium polysilfide, calcium chloride, calcium sulfate, calcium carbonate, calcium formate , 4-oxo-4- (2-phenylethyl) aminobutyric acid, 5- (trifluoromethyl) benzo [b] thiophene-2-carboxylate methyl, 5- (trifluoromethyl) benzo [b] thiophene-2- Carboxylic acid etc. are mentioned.

Examples of components of the microbial material included in the group F include, for example, Bacillus films (Bacillus firmus, CNCM I-1582 etc.), Bacillus megaterium, Hirsutella rhossiliensis, and Hilstera.・ Minesotensis (Hirsutella minnesotensis), Monaclospora phymatopagus (Monacrosporium phymatopagus), Pasteuria nishizawae (Pasteuria nishizawae, Pn-1 strain etc.), Pasteuria penetrans (Pasteuria penetrans), Pasteuria usgarium (Pus.・ Chlamid sporium (Verticillium chlamydosporium), harpin protein (Harpin protein, Harpin protein derived from Erwinia amylovora, etc.), Bacillus thuringiensis (Bacillus thuringiensis, strain BD # 32, strain AQ52, etc., Aizawai subspecies (subsp) aizawai, ABTS-1857 shares etc.) Kuris Starch subspecies (subsp. Kurstaki, HD-1 strain, BMP 123 strain, etc.), Tenebriosis subspecies (subsp. Tenebriosis, NB 176 strain, etc.), Israeli cis variety (var. Israelensis), aegypti variant (var. Aegypti) , Colmel variant (var. Colmeri), varm stadiensis variant (var. Darmstadiensis), dendrimus variant (var. Dendrolimus), galeria variant (var. Galleriae), japonensis variant (var. Japonensis), Morisoni subspecies (subsp. Subsp.) Morrisoni), San Diego variant (var. San diego), thuringiensis subspecies (subsp. Thuringiensis, strain MPPL 002, etc.), variant 7216 (var. 7216), variant T36 (var. T36)), Bacillus sp. , AQ175 strain, AQ177 strain, AQ178 strain, etc.), Bacillus sphaericus (Bacillus sphaericus), Bacillus subtilis (Bacillus subtilis, QST713 strain, AQ743 strain, AQ153 strain, FQB24 strain, MBI600 strain, D747 strain, HAI0404 strain, Y1336 strain , QST3 0002 / AQ30002 strain, QST30004 / AQ30004 strain, Bacillus amyloliquefaciens (Bacillus amyloliquefaciens (strain IN93a, strain FZB42, strain FZB24, strain B3), Bacillus simplex (strain Bacillus simplex, strain CGF2856, etc.), Bacillus Pumirus (Bacillus pumilus, strain GB34, strain QST2808, strain AQ717, etc.), Bacillus acidocaldarius, Bacillus acidoterrestris, Bacillus algri, Bacillus alboriactis (Bacillus) Albolactis), Bacillus alcalophilus, Bacillus alvei, Bacillus aminoglucosidicus, Bacillus aminovorans, Bacillus amylolyticus, Bacillus・ Aneurolithus (Bacillus aneuri nolyticus), Bacillus atrophaeus, Bacillus azotoformans, Bacillus badius, Bacillus cereus (Bacillus cereus, strain CNCM 1-1562, etc.), Bacillus chitinosporus (Bacillus chitinosporus) , AQ 746, etc.), Bacillus circulans (Bacillus circulans), Bacillus coagulans (Bacillus coagulans), bacillus fortidiosus (Bacillus fastidiosus), bacillus lacticola (Bacillus lacticola), bacillus lactimorbus, Bacillus lactis, Bacillus laterosporus, Bacillus lautus, Bacillus lentimorbus, Bacillus lentus, Bacillus lichenif Rumis (Bacillus licheniformis), Bacillus marocanus (Bacillus maroccanus), Varioborax paradox (Variovorax paradox, CGF 4526 strain, etc.), Bacillus methiens (Bacillus methiens), Bacillus myoides (Bacillus mycoides, AQ 726 strain, J (BMJ) Strains, etc.), Bacillus natto, Bacillus nematocida, Bacillus nigrificans, Bacillus nigrum, Bacillus pantothenticus, Bacillus popiriae (Bacillus pantothenticus) popilliae), Bacillus psychrosaccharolyticus, Bacillus siamensis, Bacillus smithii, Bacillus uniflagellate, Brevibacillus b. revis, SS86-3 strain, SS86-4 strain, SS86-5 strain, 2904 strain etc., Brevibacillus laterosporus (Brevibacillus laterosporus, 64 strains, 1111 strain, 1645 strains, 1647 strains etc.), Beauveria bassiana (Beauveria bassiana) , ATCC 74040 strain, GHA strain etc.), Beauveria brongniartii (Beauvelia brongniartii), Pequilomyces fumosoroseus (Paecilomyces fumosoroseus, Apopka 97 strain etc.), Pequilomyces lilacinus (Paecilomyces lilacinus, 251 strain etc.), Pequirometes Pequilomyces variotii (Paecilomyces variotii, Q-09 etc.), Trichoderma harzianum (Trichoderma harzianum, T39, T22, DSM 14944, DB 104, DB 104, 21, kd, SF, ESALQ-1306, etc. ESALQ-1303 strain, IIHR-Th-2 strain etc.), Trichoderma atroviride (Trichoderma atroviride, SKT-1 strain etc.), Trichoderma album (Trichoderma album) , Trichoderma asperellum (Trichoderma asperellum, strain ICC012 etc.), Trichoderma atriloviride (Trichoderma atroviride, CNCM 1-1237 strain, etc.), Trichoderma gumsii (Trichoderma gamsii, strain ICC080 etc.), Lignoram (Trichoderma lignorum), Trichoderma polysporum (Trichoderma polysporum, strain EVII 206039 etc.), Trichoderma virens (Trichoderma virens, strain G-41 etc.), Trichoderma spp. (Trichoderma spp., Trade name: Excalibur ^TM SA, Excalibur-SA, ^{TM, Graph-Ex SA TM,} naturall TM, SabrEx TM), Verticillium potassium-Rekani (Verticillium lecani), Verticillium potassium-Aruboatoramu (Verticillium alboatrum, WCS850 strain, etc.), Verticillium potassium Kula bromide sports potassium (Verticillium chlamydosporium , Verticillium Darjee (Verti) C. cillia dahliae), live spores and produced crystal toxins derived from Pasteuria penetrans, live spores and produced crystal toxins, (Pseudomonas fluorescens, strain G7090, etc.), Pseudomonas aeruginosa, Pseudomonas aureofaciens, Pseudomonas cepacia (Pseudomonas cepacia, M54 strain, J82 strain) , MA 342 strain, etc.), Pseudomonas proradix (Pseudomonas proradix), Pseudomonas putida (Pseudomonas putida), Pseudomonas resinovolans (Pseudomonas resinovorans), Pseudomonas syringae (Pseudomonas syrin) gae), Talaromyces flavus (Talaromyces flavus, strain SAY-Y-94-01, etc.), Bradyrhizobium japonicum, Brady rhizobium elkani (Bradyrhizobium elkani), Rhizobium legminosarum bv. (Rhizobium leguminosarum bv. Trifolii), Rhizobium legumino salm bv. Phazeo (Rhizobium leguminosarum bv. Phaseoli), Rhizobium leguminosaum bv. Rhizobium leguminosarum bv. ., trade ^{name: Excalibre-SA TM, Graph-} Ex SA TM, MegaPack TM), Anperomaisesu-Kisukarisu (Ampelomyces quisqualis, AQ10 shares, etc.), Aureobasidium pullulans (Aureobasidium pullulans, DSM14940 strain, DSM14941 shares, etc.), Asher Sonia Allyrodes (Aschersonia aleyrode) s), chromobacterium subsp. moth (Chromobacterium subtsugae, PRAA4-1T strain, etc.), Delftia acidovorans (Delftia acidovorans, RAY 209 strain, etc.), Lactobacillus acidophilus (Lactobacillus acidophilus), Lysobacter antibiotics (Lysobacter antibioticus, 13-1 strain, Lysobacter enzymogenes (C3 strain etc.), Paenibacillus alvei (Paenibacillus alvei, III3DT-1A strain, III2E strain, 46C3 strain, 2771 strain etc.), Paenibacillus polymyxa [Paenibacillus polymyxa] Paenibacillus popilliae (Paenibacillus popilliae), Pantoea agglomerans, Pectobacterium carotovorum, Rhodococcus globerulus (strain AQ 719, etc.), Serratia entomophila (Serreria) A. marcescens (Serratia marcescens, SRM strain, R35 strain etc.), Streptomyces candidus (Streptomyces candidus), Streptomyces colombiensis, Streptomyces galbus (Streptomyces galbus, K61 strain, QST 6047 strain) Etc.), Streptomyces goshikiensis, Streptomyces griseoviridis, Streptomyces lavendulae, Streptomyces lydicus, WYEC108 strain, etc. , Streptomyces prasinus, Streptomyces rimosus, Streptomyces saraceticus, Streptomyces venezuelae, strike P.myces sp. (Streptomyces sp. NRRL B-30145), Xanthomonas campestris, Xenolabdasu luminescens, Xenorhabdus nematophila, Aspergillus flavus Robotris spermatova (Arthrobotrys superba), Candida oleophila (Candida oleophila, O strain etc.), Ketomium cupreum (Chaetomium cupreum), Cladsporium cladosporioides (Cladosporium cladosporioides (H39 strain etc.), conidiobolus) Obscuras (Conidiobolus obscurus), Coniosidium minitans (Coniothyrium minitans, CON / M / 91-8 strain), Dirophosphora alopecuri, Entomophthora virulenta, Fusarium oxys Lam (Fusarium oxysporum, strain Fo47, etc.), gliocladium catenulatam (Gliocladium catenulatum, strain J1446), Hirstela thompsonii (Hirsutella thompsonii), Lagenidium gigantium (Lagenidium giganteum), Recanicillium L. lucii ), Metarhizium anisopliae (Metarhizium anisopliae, F52 strain, etc., Acridam variant (var. Acridum)), Metarhizium flavoviride (Metarhizium flavoviride), Metichnikowia fructicola (NRRLY-30752), M. ochracea), Mucor hiemalis (Mucor hiemalis), Muscodor albus (Muscodor albus (QST 20799 strain, 620 strains etc.), Muscodor roseus (Muscodor roseus, strain A3-5 etc.), Myrothecium verrucaria (Myrothecium verrucaria, AARC- 0255 shares etc), Laea Lily (Nomuraea rileyi, SA86101, GU87401, SR86151, CG128, VA9101 etc.), Ophiostoma piliferum (Ophiostoma piliferum, D97 etc.), Pandora delphacis (Pandora delphacis), Penicillium bilai (Penicillium bilaii , ATCC 22348, etc.), Penicillium vermiculatum, Phlebiopsis gigantea, Pichia anomala (Pichia anomala, WRL-076 etc.), Poconia chlamydosporia, Phlocuroza sp. (Pseudozyma flocculosa, PF-A22UL strain, etc.), Pythium oligondrum (Pythium oligodrum, DV74 strain, etc.), Sporothrix insectorum, Tsukamurella paurometabola (Tsukamurella paurometabola), urocladium oodemidium i), Zuhoftra radicans (Zoophtora radicans), Nozema rokustae (Nosema locustae), Telohania solenopsis (Thelohania solenopsis), Bailimorpha spp. granulosis virus (GV), Agrotis segetum nuclear polyhedrosis virus (NPV), Anticalcia gemataris nuclear polyhedrosis virus (Anticarsia gemmatalis mNPV), autographa california nuclear polyhedrosis virus (Autographa californica mNPV), Biston-Supresaria nuclear polyhedrosis virus (Biston suppressaria NPV), Bombyx-Mori nuclear polyhedrosis virus (Bombyx mori NPV), Cryptofrebbia leukotreta granular disease virus (Cryptophlebia leucotreta GV), Shijia-Ponnera granular disease virus Cydia pomonella GV), Dendolimus punctatus cytosolic virus (Dendrolimus punctatus cypovirus), Helicoverpa armigera NPV, Helicoverpa zea nuclear polyhedrosis virus (Helicoverpa zea NPV) Polyhedra disease virus (Leucoma salicis NPV), Lymantria dispar nuclear polyhedrosis virus (Lymantria dispar NPV), Neodiplion abientis nuclear polyhedrosis virus (Neodiprion abietis NPV), Neodiprion recontei nuclear polyhedrosis virus (Neodiprion lecontei NPV), Neodiprion sertifer nuclear polyhedrosis virus (Neodiprion sertifer NPV), Orgia pseudotosugata nuclear polyhedrosis virus (Orgyia pseudotsugata NPV), Stromaea operculella granulosa virus (Phthorimaea operculella GV) Pieris rapae granulosis virus (Pieris rapae GV), Plutella xylostella granulosis virus (Plutella xylostella GV), Spodoptera albra nuclear polyhedrosis virus (Spodoptera albula mNPV), Spodoptera exulpum nuclear polyhedrosis virus (Spodoptera exemplar mNPV) ), Spodoptera exigua nuclear polyhedrosis virus (Spodoptera exigua mNPV), Spodoptera frugiperta nuclear polyhedrosis virus (Spodoptera frugiperda mNPV), Spodoptera littoralis nuclear polyhedrosis virus (Spodoptera littoralis mNPV), Disease virus (Spodoptera litura NPV), Abrevita caucasica, aquaria spp. (Acuaria spp.), Agamelmis decaudata (Agamermis decaudata), Allantoma spp. .), Bedin Gia Silydicola (Beddingia siridicola), Bobienema spp. (Bovienema spp.), Cameronia spp. spp. (Culicimermis spp.), deprotolize spp. (Diplotriaena spp.), Empidomermis spp. (Gongylonema spp.), Gynopoecilia pseudovipara, Heterolabditis bacteriophora, Heterolabditis baujardi, Heterolabditis heliotizitehitivehe Itis indica (Heterorhabditis indica), heterolabditis malereitas (Heterorhabditis marelatus), heterolabditis megidis (Heterorhabditis megidis), heterolabditis zealandica (Heterorhabditis zealandica), hexamermis spp. (Hydromermis spp.), isomelmis spp. (Isomermis spp.), limomelmis spp. (Limnomermis spp.), Maupasina weissi, Malypas nigrescens (Mermis nigrescens), mesomermis spp. (Mesomermis spp. ., Neomesomermis spp. (Neomesomermis spp.), Neoparasatirengus ragrossi (Neoparasitylenchus rugulosi), Octoomyo mermis spp. Ditis spp. ( Parasitatorhabditis spp., Parasity lenchus spp., Perutilimermis culicis, Phasmarhabditis hermaphrodita, Physalupta spp. (Protrellatus spp.), Ptereligo dermatitus spp. (Pterygodermatites spp.), Romanomelmis spp. (Romanomermis spp.), Souretum cadarachense (Seuratum cadarachense), Sphael laryopsis spp. ), Spyrura gaianensis (Spirura guianensis), Steinernema carpocapsae (Steinernema carpocapsae), Steinernema fertiae (Steinernema feltiae), Steinernema glaseri (Steinernema glaseri), Steinernema crasei (Steinernemakrainese) Maa Riobrabe (Steinernema riobrave), Stainanema scupteris (Steinernema scapterisci), Stainenema scalabaei (Steinernema scarabaei), Stainenema siamkayai (Steinernema siamkayai), Strelco bimmel Miss Putel Sivelvegetal And Sulpletilex elongitus, Tetrameres spp., And the like.

  Each component included in the above-mentioned group A, group B, group C, group D, group E and group F is known, for example, “THE PESTICIDE MANUAL-16th EDITION (BCPC publication) ISBN 978-1- 901396-86-7. These compounds can be produced by the methods described in the patent documents or non-patent documents cited in "THE PESTICIDE MANUAL", or their related documents, or can be obtained from commercially available preparations.

  Among the components selected from the group consisting of Group A, Group B, Group C, Group D, Group E and Group F, the components described in the following abbreviation correspondence table are described as PP1 to PP1537.

Abbreviation correspondence table [abbreviation: component]
[PP1: mandestorobin], [PP2: 3-chloro-5-phenyl-6-methyl-4- (2,6-difluorophenyl) pyridazine], [PP3: 3-cyano-5-phenyl-6-methyl] -4- (2,6-difluorophenyl) pyridazine], [PP4: 3-difluoromethyl-1-methyl-N-[(3R) -1,1,3-trimethylindan-4-yl] pyrazole-4- Carboxamide], [PP5: cyclaniliprole], [PP6: tetraniliprole], [PP7: cyhalodiamide], [PP8: 4-oxo-4- (2-phenylethyl) aminobutyric acid], [PP9: imidacloprid] , [PP10: clothianidin], [PP11: thiamethoxam], [PP12: dinotefuran], [PP13: acetamiprid], [PP14: thiacloprid], [PP15: nitenpyram], [PP16: acrinatrin [PP17: bifenthrin], [PP18: cycloprotoline], [PP19: cyfluthrin], [PP20: beta cyfluthrin], [PP21: cyhalothrin], [PP22: lambda cyhalothrin], [PP23: gamma cyhalo] [Trin], [PP24: cypermethrin], [PP25: alpha cypermethrin], [PP26: beta cypermethrin], [PP27: theta cypermethrin], [PP28: zeta cypermethrin], [PP29: deltamethrin], [PP31 : Fenpropatrin], [PP32: fenvalerate], [PP33: esfenvalerate], [PP34: flucitrate], [PP35: fluvalinate], [PP36: taufluvalinate], [PP38: permethrin], [PP39: silafluofen], [PP40: tefluthrin], [PP41: tralomethrin], [PP43: fipronil], [PP44: ethiprole] [PP49: Abamectin], [PP51: Emamectin benzoate], [PP52: Milbemectin], [PP53: Doramectin], [PP54: Lepimectin], [PP55: Flubendiamide], [PP56: Chlorantranyriprole], [PP57: cyantraniriprole], [PP58: pimetrozine], [PP59: pyridalyl], [PP60: pyriproxyfen], [PP61: spirotetramat], [PP62: sulfoxaflor], [PP63: flupyradifluro], [PP PP64: Acephate], [PP65: Chlorpyrifos], [PP66: Chlorpyrifos methyl], [PP67: Kazusaphos], [PP68: Diazinon], [PP69: Etoprophos], [PP70: Fenamiphos], [PP71: Fossiazate], [PP72 : Isofenphos], [PP73: imiciaphos], [PP74: isoxathion], [PP75: fenitrothion], [PP76 : Folate: [PP 77: Hosmet], [PP 78: Hoxim], [PP 79: Terbuphos], [PP 80: Quinalphos], [PP 81: Pyraclophos], [PP 82: Monocrotophos], [PP 83: Dicrotophos], [PP 84: Carbofuran], [PP 85: Carbosulfan], [PP 86: Aldicarb], [PP 87: Thiodicarb], [PP 88: Methiocarb], [PP 89: Oxamyl], [PP 90: Mesomil], [PP 91: Pyrimicarb], [PP 92: Benfrukarubu], [PP93: pyrethrin], [PP94: allethrin], [PP95: buprofezin], [PP96: tolfenpyrado], [PP97: thiocyclam], [PP98: cartap hydrochloride], [PP99: bensultap], [PP100: Furonicamide], [PP101: Indoxacarb], [PP102: Metaflumizone], [PP103: Chromafenozide], [PP104: Methoxyfenozide [PP105: halofenozide], [PP106: tebufenozide], [PP107: diflubenzuron], [PP108: teflubenzuron], [PP109: chlorfluazuron], [PP110: ruffenuron], [PP111: novaluron], [PP112: full Phenoxlon], [PP113: chlorfenapyr], [PP114: pyrifluquinazone], [PP115: cyromazine], [PP116: diafenthiuron], [PP117: etoxazole], [PP118: spirodiclofen], [PP119: spiromesi] Phen], [PP120: fenpyroxymate], [PP121: pyridaben], [PP122: pyrimidiphen], [PP123: tebufenpyrado], [PP124: acequinosyl], [PP125: biphenazate], [PP126: fluacripyrim], [PP127: sheenopyraphen] , [PP128: ciflumethofen], [PP129: piflubumid], [PP130 [Imidaclotiz], [PP 131: cycloxaprid], [PP 132: tebuconazole], [PP 133: metconazole], [PP 134: difenoconazole], [PP 135: triticonazole], [PP 136: imazalil], [PP 137: triadimenol], [PP PP 138: Fluquinconazole], [PP 139: Prochloraz], [PP 140: Prothioconazole], [PP 141: Diniconazole], [PP 142: Diniconazole M], [PP 143: Ciproconazole], [PP 144: Tetraconazole], [PP145: ipconazole], [PP146: triphorin], [PP147: pyriphenox], [PP148: phenarimol], [PP149: nuarimol], [PP150: oxosconazole fumarate], [PP151: peflazoate], [PP152: triflumizole], [PP153: azaconazole], [PP154: bitertanol], [PP155: brom Conazole], [PP156: Epoxyconazole], [PP157: Fenbuconazole], [PP158: Flusilazole], [PP159: Flutriahol], [PP160: Hexaconazole], [PP161: Imibenconazole], [PP PP 162: microbutanyl], [PP 163: penconazole], [PP 164: propiconazole], [PP 165: simeconazole], [PP 166: triadimefon], [PP 167: kresoxim methyl], [PP 168: azoxystrobin], [PP 169: pyra Clostrobin], [PP 170: Picoxystrobin], [PP 171: Enestrobin], [PP 172: Trifloxystrobin], [PP 173: Dimoxystrobin], [PP 174: Fluoxastrobin], [PP 175: Orysastrobin ], [PP176: oxathiapiproline], [PP177: phenamidone], [PP178: metominostrobin], [PP179: Taraxil], [PP180: Metalaxyl M], [PP181: Fullaxyl], [PP182: Fullaxyl M], [PP183: Benalaxyl], [PP184: Benalaxyl M], [PP185: Offrace], [PP186: Oxadixil], [PP187 : Probenazole], [PP188: Thiazinyl], [PP189: Tricyclazole], [PP190: Pyroxolone], [PP191: Kasugamycin], [PP192: Ferrimzone], [PP193: Isothianyl], [PP194: Phthalide], [PP195: Tephofloquine] ], [PP 196: Pencclone], [PP 197: Flamethopyr], [PP 198: Validamycin A], [PP 199: Carboxin], [PP 200: Flutolanil], [PP 201: Penthiopyrad], [PP 202: Fluopyram], [PP 203: Penfulfen ], [PP 204: Sedaxane], [PP 205: Fluxapiroxide], [PP 206: Fludioxonil] [PP 207: Etaboxam], [PP 208: Torclophos methyl], [PP 209: Captan], [PP 210: Benomyl], [PP 211: Carbendazim], [PP 212: Pyradiflumid], [PP 213: Thiophanate Methyl], [PP 214: Thiabendazole], [PP 215: dietophene carb], [PP 216: zoxamide], [PP 217: fluopicolide], [PP 218: thifluzamide], [PP 219: boscalid], [PP 220: bixaphen], [PP 221: isopyrazam], [PP 222: enoxastrobin], [PP223: famoxadone], [PP224: pyribencarb], [PP225: pyraxtorobin], [PP226: pyramethostrobin], [PP227: spider oxystrobin], [PP228: fluphenoxystrobin], [PP229: Triclopyricarb], [PP230: phenaminostrobin], [PP231: Cyazofamid], [PP23 2: Amisulblom], [PP233: Ametoclazine], [PP234: Binapakryl], [PP235: Fluazinam], [PP236: Silthiofam], [PP237: Pyrimethanyl], [PP238: Ciprodinil], [PP239: Blastsaidin S], [PP 240: procymidone], [PP 241: iprodione], [PP 242: quinoxyphene], [PP 243: proquinazide], [PP 244: fenpyrazamine], [PP 245: isoprothiolane], [PP 246: iprobenphos], [PP 247: eginphos], [PP 248 : Pyrazophos], [PP 249: Quintozen], [PP 250: Fenpropimorph], [PP 251: Fenpropidine], [PP 252: Spiroxamine], [PP 253: Fenhexamide], [PP 254: Dodine], [PP 255: Resid Benzolar S methyl], [PP256: Mankozeb], [PP257: Folpet], [PP258: Chlorothalonil], PP 259: Thiuram], [PP 260: Diclocymet], [PP 261: Carpropamide], [PP 262: Oxolinic acid], [PP 263: Isophetamide], [PP 264: Pasteuria penetrans fungus], [PP 265: Dichlormid], [PP 266: Bacillus • Thuringiensis bacteria], [PP266-1-1: Bacillus thuringiensis strain BD # 32], [PP 266-1-2: Bacillus thuringiensis bacteria AQ 52], [PP 266-2: Bacillus thuringiensis bacteria Aizawai Subspecies], [PP 266-2-1: Bacillus thuringiensis bacteria Aizawai subspecies ABTS-1857 strain], [PP 266-3: Bacillus thuringiensis Bacillus subtilis subspecies], [PP 266-3-1: Bacillus thuringia C. cistoea cristae subsp. Strain HD-1], [PP 266-3-2: Bacillus thuringiensis sp. Cristola sp. BMP 123 strain], [PP 266-4: Bacillus thuri] N. gonorrhoeae subsp. Spp. [PP 266-4-1: Bacillus thuringiensis subsp. Tenebriosis subsp. NB 176 strain], [PP 266-5: Bacillus thuringiensis israeliensis variant], [PP 266-6: Bacillus sp. Thuringiensis spp. Aedipti variant], [PP266-7: Bacillus thuringiensis kolmeri variant], [PP 266-8: Bacillus thuringiensis dermstasis variant], [PP 266-9: Bacillus thuringiensis dendolimus variant ], [PP266-10: Bacillus thuringiensis galleria variant], [PP266-11: Bacillus thuringiensis japonensis variant], [PP266-12: Bacillus thuringiensis morizoni subspecies], [PP266-13: Bacillus thuringiensis bacteria San Diego variant], [PP 266-14: Bacillus thuringi [Genus Bacillus thuringiensis subspecies], [PP 266-14-1: Bacillus thuringiensis strain thuringiensis subspecies MPPL 002 strain], [PP 266-15: Bacillus thuringiensis strain 7216 variant], [PP 266-16: Bacillus thuringia Cis microbe T36 variant], [PP 267: Bacillus film bacillus], [PP 267-1: Bacillus bacillus microbe CNCM I-1582 strain], [PP 268: oxycarboxin], [PP 269: triazoxide], [PP 270: Anthraquinone], [PP 271: Himexazole], [PP 272: Shimoxanil], [PP 273: Fluensulfone], [PP 274: Gibberellin A3], [PP 275: Etaconazole], [PP 276: Uniconazole], [PP 277: 3-Difluoromethyl-N -(7-fluoro-1,1,3-trimethylindan-4-yl) -1-methylpyrazole-4-carboxamide], [PP 277- : 3-Difluoromethyl-N-[(3R) -7-fluoro-1,1,3-trimethylindan-4-yl] -1-methylpyrazole-4-carboxamide], [PP278: benodanyl], [PP279: Fenfram], [PP280: organic copper], [PP281: tridemorph], [PP282: dodemorph], [PP 283: piperaline], [PP284: mepanipyrim], [PP 285: fenpiclonyl], [PP 286: vinclozolin], [PP 287: fuberidazole] ], [PP 288: thiophanate], [PP 289: dimethomorph], [PP 290: iprobaricarb], [PP 291: benchavaricab isopropyl], [PP 292: mandipropamide], [PP 293: varifenalate (varifenal)], [PP 294: Fulmorph], [PP 295: 3- (3,4-dichloroisothiazol-5-ylmethoxy) -benzoisothiazo 1,1-Dioxide], [PP 296: picalbutrazox], [PP 297: focetylaluminum], [PP 298: potassium salt of phosphorous acid], [PP 299: propamocarb hydrochloride], [PP 300: flusulfamide], [PP 2 PP 301: Metraphenone], [PP 302: Pyrophenone], [PP 303: Cifluphenamide], [PP 304: Laminarin], [PP 305: Tolprocarb], [PP 306: Diclomedin], [PP 307: Streptomycin]
[PP309: Oxytetracycline], [PP310: Quillaraceae plant extract], [PP312: Iminoctadine acetate], [PP313: Sulfur], [PP314: Basic copper chloride], [PP315: Cupric hydroxide] [PP 316: basic copper sulfate], [PP 318: diclofluanid], [PP 319: phenoxanyl], [PP 320: anilazine], [PP 321: betoxazine], [PP 322: biphenyl], [PP 323: bupyrimate], [PP 324 : Captaphor], [PP 325: chloroneb], [PP 326: dichloran], [PP 327: diflumetrime], [PP 328: dimesilymol], [PP 329: dinocap], [PP 330: dithianone], [PP 332: ethydiazole], [PP 333: Triphenyltin acetate], [PP334: triphenyltin hydroxide], [PP335: felbum], [PP336: flumetober], [PP337: fluoroimide], [PP338: fluthiani ], [PP 339: Flumecyclox], [PP 340: Iodocarb], [PP 341: Meptyldino Cap], [PP 342: Metasulfocarb], [PP 343: Methylam], [PP 344: Naftifine], [PP 345: Occirinone], [ PP 346: phosphorous acid, [PP 347: sodium salt of phosphorous acid], [PP 348: ammonium salt of phosphorous acid], [PP 349: polyoxin], [PP 350: propineb], [PP 351: prothiocarb], [PP 352: Pyributycarb], [PP 353: pyrrolnitrin], [PP 354: TCNB], [PP 355: teclophthalam], [PP 356: terbinafine], [PP 357: tolyl fluanide], [PP 358: triarimol], [PP 359: triazoloxide], [ PP 361: Zineb], [PP 362: Zillam], [PP 363: a compound represented by the above formula (b)], [PP 364: a compound represented by the above formula (a)], [PP 365: N ′-[4-] ( {3-[(4-Chlorophenyl) methyl] -1,2,4-thiadiazol-5-yl} oxy) -2,5-dimethylphenyl] -N-ethyl-N-methylmethanimidamide], [PP 366: Dipimetictron], [PP 367: 3- (4, 4-Difluoro-3, 3-dimethyl-3,4-dihydroisoquinolin-1-yl) quinoline], [PP 368: 2- {3- [2- (1- {{ [3,5-Bis (difluoromethyl) -1H-pyrazol-1-yl] acetyl} piperidin-4-yl) -1,3-thiazol-4-yl] -4,5-dihydro-1,2-oxazole -5-yl} -3-chlorophenyl = methanesulfonate], [PP 369: 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2 (1H) -one], [PP370: α- [3- 4-chloro-2-fluorophenyl) -5- (2,4-difluorophenyl) -4-isoxazolyl] -3-pyridinemethanol], [PP 371: (αS)-[3- (4-chloro-2-fluoro) Phenyl) -5- (2,4-difluorophenyl) -4-isoxazolyl] -3-pyridinemethanol], [PP 372: (αR)-[3- (4-chloro-2-fluorophenyl) -5- (2 , 4-Difluorophenyl) -4-isoxazolyl] -3-pyridinemethanol], [PP 373: 2-{[3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl } -2,4-Dihydro-3H-1,2,4-triazole-3-thione], [PP 374: phenchlorazole ethyl], [PP 375: phenclorim], [PP 376: 2-{[(2R, 3) ) -3- (2-Chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] methyl} -2,4-dihydro-3H-1,2,4-triazole-3-thione], [PP 377: 2-{[(2S, 3R) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -2,4-dihydro-3H-1, 2,4-Triazole-3-thione], [PP 378: 2-{[(2R, 3R) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -2,4-dihydro-3H-1,2,4-triazole-3-thione], [PP 379: 2-{[(2S, 3S) -3- (2-chlorophenyl) -2- (2,4-) Difluorophenyl) oxirane-2-yl] methyl} -2,4- Dihydro-3H-1,2,4-triazole-3-thione], [PP 380: 1-{[3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4-triazole-5-thiol], [PP 381: flurazole], [PP 382: furilazole], [PP 383: 1-{[(2R, 3S) -3- (2-chlorophenyl) -2] -(2,4-Difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4-triazole-5-thiol], [PP384: 1-{[(2S, 3R) -3- (2) -Chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] methyl} -1H-1,2,4-triazole-5-thiol, [PP 385: 1-{[(2R, 3R)] -3- (2-chlorophenyl)- -(2,4-Difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4-triazole-5-thiol], [PP 386: 1-{[(2S, 3S) -3- (2) -Chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] methyl} -1H-1,2,4-triazole-5-thiol, [PP 387: 1-{[3- (2-) Chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-yl] methyl} -1H-1,2,4-triazol-5-ylthiocyanato], [PP 388: mefenpyr diethyl], [PP 389: MG 191], [PP 390: 1-{[(2R, 3S) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4 -Triazole-5-i Thiocyanato], [PP 391: 1-{[(2S, 3R) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -1H-1,2,4 -Triazol-5-yl thiocyanato], [PP 392: 1-{[(2R, 3R) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxiran-2-yl] methyl} -1H -1,2,4-triazol-5-ylthiocyanato], [PP 393: 1-{[(2S, 3S) -3- (2-chlorophenyl) -2- (2,4-difluorophenyl) oxirane-2-] [Ill] methyl} -1H-1,2,4-triazol-5-yl thiocyanate], [PP 394: 5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2 , 4-Triazole-1-i Methyl) cyclopentanol], [PP 395: (1RS, 2SR, 5SR) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole-1 -Ylmethyl) cyclopentanol], [PP 396: (1RS, 2RS, 5RS) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole- 1-ylmethyl) cyclopentanol], [PP397: (1RS, 2RS, 5SR) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole] -1-ylmethyl) cyclopentanol], [PP 398: (1RS, 2SR, 5RS) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1, 2,4-) Triaza -1-ylmethyl) cyclopentanol], [PP 399: (1R, 2S, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-) Triazol-1-ylmethyl) cyclopentanol], [PP 400: (1S, 2R, 5R) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4 -Triazol-1-ylmethyl) cyclopentanol], [PP 401: (1R, 2R, 5R) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,6 4-Triazol-1-ylmethyl) cyclopentanol], [PP 402: (1S, 2S, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2 , 4-Triazol-1-ylme Ethyl) cyclopentanol], [PP 403: (1R, 2R, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole-1 -Ylmethyl) cyclopentanol], [PP 404: (1S, 2S, 5R) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole- 1-ylmethyl) cyclopentanol], [PP 405: (1R, 2S, 5R) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-triazole] -1-ylmethyl) cyclopentanol], [PP 406: (1S, 2R, 5S) -5- (4-chlorobenzyl) -2-chloromethyl-2-methyl-1- (1H-1,2,4-) Triazol-1-ylmethyl) cyclo Ethanol], [PP 407: methyl 3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentane carboxylate], [PP408: methyl = (1R, 2S, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclo Pentane carboxylate], [PP 409: methyl = (1S, 2R, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazole- 1-ylmethyl) cyclopentanecarboxylate], [PP410: methyl 3- (1R, 2R, 3R)-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl -2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanecarboxylate], [PP 411: methyl = (1S, 2S, 3S) -3-[(4-chlorophenyl) methyl] -2- Hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanecarboxylate], [PP 412: methyl = (1R, 2R, 3S) -3-[(4-chlorophenyl)] Methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentanecarboxylate], [PP 413: methyl = (1S, 2S, 3R) -3- [ (4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentane carboxylate], PP 414: methyl = (1R, 2S, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) cyclopentane Carboxylate], [PP 415: methyl = (1S, 2R, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- [1H-1,2,4-triazole-1 -Ylmethyl] cyclopentane carboxylate], [PP 416: flusophenim], [PP 417: 1,8-naphthalic anhydride], [PP 418: AD-67], [PP 419: indole butyric acid], [PP 420: ethychlozate], [PP PP 421: 1-Naphthylacetamide], [PP 422: 4-CPA], [PP 424: Aridochlor], [PP 425: Oxabetrinyl], [PP 426: Cyprosulfamide], [PP 427: Isoxadiphe Ethyl, [PP 428: 2, 2-dimethyl-9-fluoro-5- (quinolin-3-yl) -2,3-dihydro-benzo [f] [1,4] oxazepine, [PP 429: N-cyclo Propyl-3- (difluoromethyl) -5-fluoro-N- (2-isopropylbenzyl) -1-methyl-1H-pyrazole-4-carboxamide], [PP 430: N-cyclopropyl-3- (difluoromethyl)- 5-fluoro-N- (5-chloro-2-isopropylbenzyl) -1-methyl-1H-pyrazole-4-carboxamide], [PP 431: 1-naphthaleneacetic acid sodium], [PP432: 1-methylcyclopropene], [PP 433: Chlormecoat], [PP 434: Mepicoat], [PP 435: Uniconazole P], [PP 436: Paclobutrazol], [PP 437: Flurprimidol], [PP 438: Kaine Chin], [
PP 439: 1,3-Diphenylurea], [PP 440: Forchlorphenuron], [PP 441: Decyl alcohol], [PP 442: Pidiflumethophene], [PP 443: 3-Difluoromethyl-N-methoxy-1-methyl- N-[(1R) -1-methyl-2- (2,4,6-trichlorophenyl) ethyl] pyrazole-4-carboxamide], [PP 444: 3-difluoromethyl-N-methoxy-1-methyl-N- [(1S) -1-Methyl-2- (2,4,6-trichlorophenyl) ethyl] pyrazole-4-carboxamide], [PP 445: 2- [6- (3-fluoro-4-methoxyphenyl) -5 -Methylpyridin-2-yl] quinazoline], [PP446: 5-fluoro-2-[(4-methylphenyl) methoxy] -4-pyrimidinamine], [PP 447: iometrinil], [PP448 Azamethyphos], [PP 449: azinphos ethyl], [PP 450: azinphos methyl], [PP 451: chlorethoxyphos], [PP 452: chlorfenvinphos], [PP 453: chlormephos], [PP 454: lime sulfur], [PP 455: coumaphos], [ PP 456: Cyanophos !, [PP 457: Demeton-S-Methyl], [PP 458: Dichlorvos], [PP 459: Dimethoate], [PP 460: Dimethylvinphos], [PP 461: Disulfoton], [PP 462: EPN], [PP 463: Ethion], [PP 464: Funful], [PP 465: Phenthion], [PP 466: Heptenophos], [PP 467: Isopropyl-O- (methoxyaminothiophosphoryl) salicylate or isocarbophos], [PP 468: Malathion], [PP 469: Mecarbam ], [PP 470: methamidophos], [PP 471: methidathion], [PP 472: mevinphos], [PP 473: nared], PP 474: omethoate], [PP 475: oxydimethone methyl], [PP 476: parathion], [PP 477: parathion methyl or methyl parathion], [PP 478: phentoate], [PP 479: fosarone], [PP 480: phosphamidone], [PP 481: pyrimiphos methyl] ], [PP 482: profenophos], [PP 483: propetamphos], [PP 484: prothiophos], [PP 485: pyridafenthion], [PP 486: sulfotep], [PP 487: tebupilimphos], [PP 488: temephos], [PP 489: tetrachlorvin Phos], [PP 490: thiomethone], [PP 491: triazophos], [PP 492: trichlorfon], [PP 493: Vamidothion], [PP 494: alanicarb], [PP 495: bendadiocarb], [PP 496: butocarboxim], [ PP 497: butoxy carboxime], [PP 498: carbaryl], [PP 499: ethiofe [Carb], [PP500: Fenobucarb], [PP501: Holmetanate], [PP 502: Frathiocarb], [PP 503: Isoproph], [PP504: Metorcarb], [PP505: Propokisul], [PP506: Thiophanox], [PP507: Triazamate], [PP508: Trimetacarb], [PP509: XMC], [PP510: Xylylcarb], [PP511: Thiosultap-2 sodium salt or bislutap], [PP512: Thiosultap-1 sodium salt or monosultap], [PP 513: Bistrifl Ron], [PP514: Flucycloxlon], [PP515: Hexaflumuron], [PP516: Nobiflumuron], [PP517: Triflumuron], [PP518: Flufiprol], [PP519: Chlorden], [PP520: Endosulfan ], [PP 521: Alpha Endosulfan], [PP 522: Benoxaco ], [PP 523: Cloquintocetmexyl], [PP 524: Machine oil], [PP 525: Nicotine Sulfate], [PP 526: Rotenone], [PP 527: Bacillus sphaericus], [PP 528: Pseudomonas resinvolans], [PP 529: Bovelia Bronniati], [PP 530: Pekilomices fumosoroseus], [PP 530-1: Pekilomices fumosoroseus Apopka 97], [PP 531: Pekilomices lyracinas], [PP 531-1: Pekilomices lyracinas 251], [PP 532: Pekilomices -Tenuipes], [PP 533: Trichoderma harzianum], [PP 533-1: Trichoderma harzianum T39 strain], [PP 533-2: Trichoderma harzianum strain T22], [PP 533-3: Trichoderma harzianum strain DSM 14944 strain, PP 533-4: Trichoderma harzianum DB 104 strain], [PP 533-5: Trichoderma ha Gianam 21 strain], [PP 533-6: Trichoderma harzianum kd strain], [PP 533-7: Trichoderma harzianum SF strain], [PP 533-8: Trichoderma harzianum strain ESALQ-1306], [PP 533-9: Trichoderma strain Harsianum ESALQ-1303 strain], [PP 533-10: Trichoderma harzianum IIHR-Th-2 strain], [PP 534: Verticillium lecani], [PP 535: Dazomet], [PP 536: ACN], [PP 537: Pseudomonas • Puchida], [PP 538: Liquorice stone], [PP 539: Thioxazaphene], [PP 541: Bacillus megaterium], [PP 542: Hilstera rossiliensis], [PP 543: Hilstera minesotensis], [PP 544: Monacrosporium • Figmatopagum], [PP 545: Pasteuria nishizawae], [PP545-1: Pasteuria nishizawae Pn-1 strain], [PP546: Pasteuria usgae], [PP 545: PP547: pyraflufenayl], [PP548: harpin protein], [PP548-1: harpin protein from Erwinia amylovora], [PP549: 5- (trifluoromethyl) benzo [b] thiophene-2-carboxylic acid Acid methyl], [PP550: 5- (trifluoromethyl) benzo [b] thiophene-2-carboxylic acid], [PP551: amitraz], [PP552: benzoximate], [PP553: bromopropilate], [PP554] : Quinomethionate], [PP 555: clophenthezin], [PP 556: cyhexatin], [PP 557: dicophor], [PP 558: phenazaquin], [PP 559: fenbutatin oxide], [PP 560: fluazulon], [PP 561: hydroxyisoxazole] ], [PP 562: Hexythiazox], [PP 563: Propargite], [PP 564: Pyriminostrobin], [PP 565: Tetradiphone], [PP 566: Affidopirino] Pen], [PP567: aluminum phosphide], [PP568: calcium phosphide], [PP569: hydrogen phosphide], [PP570: zinc phosphide], [PP571: thidiazuron], [PP572: chlorpicrin], [PP573: DNOC], [PP 574: Phenoxycarb), [PP 575: Furometoquine], [PP 576: Hydramethylnon], [PP 577: Hydroprene], [PP 578: Quinoprene], [PP 579: Metoprene], [PP 580: Methoxychlor], [PP 581 : Methyl bromide], [PP 582: methoxadiazone], [PP 583: prohydrojasmone], [PP 584: aluminum fluoride sodium], [PP 585: sulphuramide], [PP 586: sulphuryl fluoride], [PP 587: triflumesopyrim] [PP 588: methyl 5- (trifluoromethyl) benzo [b] thiophene-2-carboxylate, [PP 589: 5- (trifluoromethyl) benzo [ Thiophene-2-carboxylic acid], [PP 590: 2,4-D], [PP 591: 2, 4-DB], [PP 592: acetochlor], [PP 593: acifluorphen], [PP 594: alachlor] [PP 595: ametrine], [PP 596: amicarbazone], [PP 597: aminopyralid], [PP 598: atrazine], [PP 600: bentazone], [PP 601: bromoxynil], [PP 602: carfentrazone], [PP 603: cal Fentrazone ethyl], [PP 604: chloran lam], [PP 605: chlorimuron], [PP 606: chlorimuron ethyl], [PP 607: chloridazone], [PP 608: cretodym], [PP 609: clodinafop], [PP 610: chromazone] , [PP 611: clopyralid], [PP 612: chloran lam methyl], [PP 613: desmedi famem], [PP 614: dicamba], [PP 615: diclophop], [PP 616: dich Roslam], [PP 617: diflufenzopyr], [PP 618: dimethenamide], [PP 620: diuron], [PP 621: EPTC], [PP 622: etalfluraline], [PP 623: ethofumesate], [PP 624: fenoxaprop ], [PP 625: fenoxaprop-P-ethyl], [PP 626: florus lam], [PP 627: fluazifop P-butyl], [PP 628: flufenaset], [PP 629: flumethoslam], [PP 630: full microlac], [PP 631: flumioxazine], [PP 632: fluthiaset], [PP 633: fomethafen], [PP 634: foramsulfuron], [PP 635: glufosinate], [PP 636: glufosinate ammonium salt], [PP 637: glyphosate], [PP 638 : Glyphosate trimesium salt], [PP 639: Glyphosate potassium salt], [PP 640: Glyphosate isopropylamine Salt], [PP 641: halosulfuron], [PP 642: halosulfuron methyl], [PP 643: haloxy hop P methyl], [PP 644: hexaazinone], [PP 645: imazamox], [PP 646: imazapic], [PP 647: imazaquin], [PP 648: imazethapyr], [PP 650: isoxaflutole], [PP 651: lactofen], [PP 652: renacil], [PP 653: linuron], [PP 654: mesosulfuron], [PP 655: meso trione], [PP 656: metam] [PP 657: metamitrone], [PP 658: metolachlor], [PP 659: metrivudine], [PP 660: methosulfurone], [PP 661: MPCA], [PP 662: MSMA], [PP 663: nicosulfuron], [PP 664: orizarin] , [PP 665: oxyfluorphen], [PP 666: paraquat], [PP 667: pendimethalin], [PP 668: fenmedifam], [PP 669: Chloram], [PP 670: Pyrimisulfuron], [PP 671: Pinoxaden], [PP 672: Promethrin], [PP 673: Pyraflufen Ethyl], [PP 674: Pyrithiobac], [PP 676: Pyroxasulfone], [PP 679: Cetoxidim ], [PP 680: simazine], [PP 681: sulfentrazone], [PP 682: tebutyuron], [PP 683: Tevotrione], [PP 684: tepraloxydim], [PP 685: thifensulfuron], [PP 686: tribe [Neuron methyl], [PP 687: triclopyr], [PP 688: trifloxysulfuron], [PP 689: trifluralin], [PP 690: triflusulfuron methyl], [PP 691: benzobin diflupyr], [PP 692: halalachus kifen Methyl], [PP 693: 2- [2-chloro-4- (4-chlorophenoxy) phenyl] -1- (1,2,4-triazol-1-yl) [Le) pent-3-yn-2-ol], [PP 694: 2- [4- (4-chlorophenoxy) -2- (trifluoromethyl) phenyl] -1- (1,2,4-triazole-1) -Yl) propan-2-ol], [PP 695: 1- [4- (4-chlorophenoxy) -2- (trifluoromethyl) phenyl] -1-cyclopropyl-2- (1,2,4-triazole) -1-yl) ethanol], [PP 696: 2- [4- (4-chlorophenoxy) -2- (trifluoromethyl) phenyl] -3-methyl-1- (1,2,4-triazole-1-) [Ill) butan-2-ol], [PP 697: (R) -2- [2-chloro-4- (4-chlorophenoxy) phenyl] -1- (1,2,4-triazol-1-yl) pentene -3-yn-2-ol], [PP 698: (R) -2- [ 4- (4-chlorophenoxy) -2- (trifluoromethyl) phenyl] -1- (1,2,4-triazol-1-yl) propan-2-ol], [PP 699: (R) -1-] [4- (4-Chlorophenoxy) -2- (trifluoromethyl) phenyl] -1-cyclopropyl-2- (1,2,4-triazol-1-yl) ethanol], [PP700: (R)- 2- [4- (4-chlorophenoxy) -2- (trifluoromethyl) phenyl] -3-methyl-1- (1,2,4-triazol-1-yl) butan-2-ol], [PP 702 : 3-difluoromethyl-1-methyl-N-[(1S) -1,1,3-trimethylindan-4-yl] pyrazole-4-carboxamide], [PP703: 3-difluoromethyl-1-methyl-N -(1,1,3-trimethy Indan-4-yl) pyrazole-4-carboxamide], [PP704: AVG], [PP 705: MCPB], [PP 706: Agrobacterium radiobacter], [PP 707: Asimidol], [PP 708: Abscisic acid], [PP 708: Abscisic acid], [PP. PP 709: Aminolevulinic acid hydrochloride], [PP 710: Aldimorph], [PP 711: Indolebutyric acid], [PP 712: Ethicolate], [PP 713: Ethephon], [PP 714: Erwinia carotobola], [PP714-1: Erwinia carotobola CGE234M403 stock],
[PP 715: Calcium formate], [PP 716: Guazatine], [PP 717: Clozolinate], [PP 718: Chlormecoat], [PP 719: Choline], [PP 720: Cyanamide], [PP 721: Cyanic acid], [PP 722: Dichlorprop ], [PP 723: Pseudomonas fluorescens], [PP 723-1: Pseudomonas fluorescens G7090 strain], [PP 724: Daminozide], [PP 725: Talaromyces flavasus], [PP725-1: Talaromyces flavasus SAY-Y- 94-01 strain], [PP 726: decyl alcohol], [PP 727: Trichoderma atroviride], [PP 727-1: Trichoderma atroviride SKT-1], [PP 728: trinexapac ethyl], [PP 729: Paclobutra [PP 730: Bacillus subtilis], [PP 730-1: Bacillus subtilis QST 713 strain], [PP 730-2: Bacillus subtilis AQ 743 strain], [PP 730] 730-3: Bacillus subtilis AQ153 strain], [PP 730-4: Bacillus subtilis FZB24 strain], [PP 730-5: Bacillus subtilis MBI 600 strain], [PP 730-6: Bacillus subtilis D747 strain], [PP 730- 7: Bacillus subtilis HAI 0404 strain, [PP 730-8: Bacillus subtilis strain Y 1336], [PP 730-9: Bacillus subtilis QST 30002 / AQ 30002 strain], [PP 730-10: Bacillus subtilis QST 30004 / AQ 30004 strain], [PP PP 731: Bacillus amyloliquefaciens], [PP 731-1: Bacillus amyloliquefaciens strain IN937a], [PP 731-2: Bacillus amyloliquefaciens strain FZB 42], [PP 731-3: Bacillus amyloliquefaciens Ensu FZB24 strain], [PP731-4: Bacillus amyloliquefaciens B3 strain], [PP732: Bacillus symplex], [PP732-1: Bacillus simplex CGF2856 strain], [PP733: Bacillus pumil ], [PP733-1: Bacillus pumilus GB34 strain], [PP733-2: Bacillus pumilus strain QST2808], [PP733-3: Bacillus pumilus strain AQ717], [PP734: varioborac paradox], [PP734] -1: Variovorax paradox CGF 4526 strain], [PP 735: Pyrisoxazole], [PP 736: Pirimorph], [PP 737: Flurprimidol], [PP 738: Prohexadione calcium], [PP 739: Bencha calilab], [PP 740: mefluidide], [PP 741: calcium chloride], [PP 742: triphenyltin chloride], [PP 743: calcium peroxide], [PP 744: calcium carbonate], [PP 745: calcium sulfate], [PP 746: bradyrhizobi] Umm Japonicum], [PP 747: Rhizobium leguminosalum bv. Trifoli], [PP 748: Rhizobium leguminosalum bv. Phazeo], [PP 749: Rhizobium] Legminino salm bv. Visiae], [PP 750: Sinolysobium • meliloti], [PP 751: Amperomyces xis calis], [PP 751-1: Amperomyces xis calis AQ10], [PP 752: aureobasidium pullulans], [PP 75 2-1: aureo Vasidium pullulans strain DSM 14 940], [PP 752-2: Aureobasidium pullulans strain DSM 14941], [PP 753: Achelsonia alleiroides], [PP 754: Bacillus sp.], [PP 754-1: Bacillus sp. Strain AQ 175] [PP 754-2: Bacillus sp. Strain AQ177], [PP 754-3: Bacillus sp. Strain AQ 178], [PP 755: Bacillus acidocaldarius], [PP 756: Bacillus acido terestris], [PP757: Bacillus sp. Alguri], [PP758: Bacillus alboractis], [PP759: Bacillus alcaliphilus], [PP760: Bacillus albay], [PP761: ba Tylus aminoglucosidicus], [PP 762: Bacillus aminoboranes], [PP 763: Bacillus amiloriticus], [PP 764: Bacillus aneurolithus], [PP 765: Bacillus atrophaeus], [PP 766: Bacillus [Azo Performance], [PP 767: Bacillus badius], [PP 768: Bacillus cereus], [PP 768-1: Bacillus cereus strain CNCM 1-1562], [PP 769: Bacillus chinosporus], [PP 769-1: Bacillus] -Kitinosporus strain AQ746], [PP 770: Bacillus circulans], [PP 771: Bacillus coagulans], [PP 772: Bacillus phostidiosas], [PP 773: Bacillus lacticola], [PP 774: Bacillus lactimulbas], [PP 775: Bacillus lactis], [PP 776: Bacillus laterosporus], [PP 777: Batil]・ Lautus], [PP 778: Bacillus lentimorphs], [PP 779: Bacillus lentus], [PP 780: Bacillus licheniformis], [PP 781: Bacillus malocanus], [PP 782: Bacillus methiens], [PP 783: Bacillus mycoides] ], [PP 783-1: Bacillus mycoides AQ 726 strain], [PP 783-2: Bacillus mycoides J (BMJ) strain], [PP 784: Bacillus natto], [PP 785: Bacillus nigrificans], [PP 786: Bacillus n. Two grams], [PP 787: Bacillus pantothenicus], [PP 788: Bacillus popiliae], [PP 789: Bacillus cyclosaccharolyticus], [PP 790: Bacillus siamentis], [PP 791: Bacillus smithii], [PP 792 B. uniflagellate], [PP 793: Brevibacillus brevis], [PP 793-1: Brevibacillus b. Levis SS 86-3 strain], [PP 793-2: Brevibacillus brevis SS 86-4 strain], [PP 793-3: Brevibacillus brevis SS 86-5 strain], [PP 793-4: Brevibacillus brevis 2904 strain], [PP 794: Brevibacillus laterosporus], [PP794-1: Brevibacillus laterosporus 64], [PP 794-2: Brevibacillus laterosporus 1111], [PP 794-3: Brevibacillus laterosporus 1645], [PP 794] -4: Brevibacillus laterosporus strain 1647], [PP795: Chromobacteria subcutae], [PP795-1: Chromobacteria subcutae PRAA4-1T], [PP796: Delfthia acidoboranes], [PP796-1: Delphithia acidoboranes RAY 209], [PP 797: Lactobacillus acidophilus], [PP 798: Lysobacter antibiotics], [PP 798-1: Lysobacter anti Ioticus 13-1 strain], [PP 799: Rhizobacthrase enzymogenes], [PP 799-1: Rhizobacthrase enzymogenes C3 strain], [PP800: Paenibacillus alvai], [PP800-1: Paenibacillus alvai III3DT-1A strain], [PP800 PP 800-2: Paenibacillus albay strain III2E], [PP 800-3: Paenibacillus albay 46C3 strain], [PP 800-4: Paenibacillus albay 2771 strain], [PP 801: paenibacillus polymixer], [PP 802: paenibacillus popilia]] [PP 803: Pantoea agglomerans], [PP 804: Pectobacterium carotobolum], [PP 805: Pseudomonas aeruginosa], [PP 806: Pseudomonas fluorescens], [PP 807: Pseudomonas aureofaciens], [PP 808: Pseudomonas cepacia], [PP 808-1: Pseudomonas cepacia M54 strain], [PP 808-2: Pseudomonas cepacia J 82], [PP 809: Pseudomonas chlorolafis], [PP 809-1: Pseudomonas chlorolaphys MA 342], [PP 810: Pseudomonas proradix], [PP 811: Pseudomonas syringae], [PP 812: Rhodococcus globulus], [PP 812-1: Rhodococcus globulus AQ 719], [PP 813: Serratia entomophila], [PP 814: Serratia marcesens], [PP 814-1: Serratia marcescens] SRM strain], [PP 814-2: Serratia marcescens R 35 strain], [PP 815: Streptomyces candidas], [PP 816: Streptomyces columbiensis], [PP 817: Streptomyces gallus], [PP 817- 1: Streptomyces gallus K61 strain], [PP 817-2: Streptomyces gallus QST 6047 strain [PP 818: Streptomyces goshikiensis], [PP 819: Streptomyces griseoviridis], [PP 820: Streptomyces la benzre], [PP 821: Streptomyces lidicus], [PP 821-1: Streptomyces.・ Lydicus WYCD108 strain], [PP 821-2: Streptomyces lyzicus WYEC 108], [PP 822: Streptomyces plasticinas], [PP 823: Streptomyces saraceticus], [PP 824: Streptomyces venezuela], [PP 825: Xanthomonas campestris], [PP 826: Xenolabdas luminescence], [PP 827: Xenolabdas nematophila], [PP 828: Aspergillus flavus], [PP 828-1: Aspergillus flavus NRRL 21 882 strain], [PP 829: Als Robotris・ Sperva], [PP 830: Boberia Basiana [PP830-1: Bovelia basiana ATCC 74040 strain], [PP 830-2: Bovelia basiana GHA strain], [PP 831: Candida oleofa], [PP 831-1: Candida oleofa O strain], [PP 832: ketomium. Cupleum], [PP 833: cladosporium cladosporoides], [PP 833-1: cladosporium cladosporoides H39 strain], [PP 834: conidioborus obscuras], [PP 835: coniosilium minitoss] [PP 835-1: Coniocillus minitans CON / M / 91-8 strain], [PP 836: Dirophosphora alopekri], [PP 837: Entomoftora billenta], [PP 838: Fusarium oxysporum], [PP 838-1: Fusarium • Oxysporum Fo47 strain], [PP839: Gliocladium catenulatam], [PP 839-1: Gliocladium catenulatam J1446 ], [PP 840: Hilstera thompsoni], [PP 841: Lagenidium giganteum], [PP 842: Recanicillium recani], [PP 842-1: Recanicillium recani KV 01], [PP 843: Metallidium anisopliae], [PP 843-1] : Metallidium anisopliae F 52 strain, [PP 843-2: Metaridium anisopriae achrydam variant], [PP 844: methalidium flavoviride], [PP 845: methynikobia fructicola], [PP 846: Microsphaelopsis ochracea], [PP 847: Mucor Heemaris], [PP 848: Muscodor Albus], [PP 848-1: Muscodor Albus QST 20799 stock], [PP 848-2: Muscodor Albus 620 stock], [PP 849: Muscodor Roseus], [PP 849-1 : Muscodor Roseus A3-5], [PP 850: Myrotesium vercaria], [PP 850-1: Mi Tesium Verkalia AARC-0255 stock, [PP 851: Nomura Air Lily], [PP 851-1: Nomura Air Lily SA 86 101 stock, [PP 851-2: Nomura Air Lily GU 87401 stock], [PP 851-3: Nomura Air Lily SR 86 151 Inc., [PP 851-4: Nomuraea Lily CG128 stock], [PP 851-5: Nomuraea Lily VA 9101 stock], [PP 852: Ophiostoma pyliferum], [PP 852-1: Ophiostoma piriferum D97 stock], [PP 853: [Pecilomyces valiotti], [PP 853-1: Pequilomyces valiotti Q-09 stock], [PP 854: Pandora delphasis], [PP 855: Penicillium bilayi], [PP 855-1: Penicillium bilayi ATCC 22348 strain], [PP PP 856: Penicillium vermiculatam], [PP 857: Frebiopsis gigantea], [PP 858: Pichia anomala], [PP 858-1: Pichia anomala WRL -076 strain], [PP 859: Poconia chlamydropia], [PP 860: pseudo zyma flocurosa], [PP 860-1: pseudo zyma flocculosa PF-A 22 UL strain], [PP 861: picium o ligandum], [PP 861-1: picium・ Oligand Rum DV 74], [PP 862: Sporotricus insectome], [PP 863: Trichoderma arbum], [PP 864: Trichoderma asperomem], [PP 864-1: Trichoderma asperomem ICC 012], [PP 865: Trichoderma atorioviride] ], [PP865-1: Trichoderma atriloviride CNCM 1-1237 strain], [PP866: Trichoderma gumcycii], [PP866-1: Trichoderma gumcycillus ICC 080], [PP867: Trichoderma koningi], [PP868: Trichoderma vibrense] Lignoram], [PP869: Trichoderma polysporum], [PP869-1: Trichoderma. Lisporum EVII 206039 strain], [PP 870: Trichoderma villens], [PP 870-1: Trichoderma villens G-41 strain], [PP 871: Zukamella paulometabola], [PP 872: Urocladium oudemansii], [PP 873: Vertisi Libert Albotram], [P
P873-1: Verticillium alboatramus WCS 850 stock], [PP 874: Verticillium chlamydsporium], [PP 875: Verticillium darje], [PP 876: Zuftra Radicans], [PP 877: Nozema Roxtae ], [PP 878: Telojania sorenopsis], [PP 879: Bailimorpha spp.], [PP 879-1: Bailimorpha spp. Q-09 strain], [PP 880: Adxophiles orana granule disease virus], [PP 881: Agrotis segegium core Polyhedrosis virus], [PP 882: Anticalcia gemataris nuclear polyhedrosis virus], [PP 883: Autographa california nuclear polyhedrosis virus], [PP 884: Bison suppressor nuclear polyhedrosis virus], [PP 885] : Bombyx-Mori nuclear polyhedrosis virus], [PP 886: Cryptofrebbia leukotleta granular disease virus], [PP 887: Shidia pomo. Nella granule disease virus], [PP 888: dendolimus punctatus cytosolic polyhedrosis virus], [PP 889: Helicoverpa armigera nuclear polyhedrosis virus], [PP 890: Helicoverpa zea nuclear polyhedrosis virus] [PP 891: Leukoma salicis nuclear polyhedrosis virus], [PP 892: Lumantria dispar nuclear polyhedrosis virus], [PP 893: neodiplion avientis nuclear polyhedrosis virus], [PP 894: neodiprion recontei Nuclear polyhedrosis virus], [PP 895: Neodiplion-Selfifer nuclear polyhedrosis virus], [PP 896: Orgia pseudo-Tsugata nuclear polyhedrosis virus], [PP897: Stromaea operculella granule disease virus], [PP898: PIERIS LAPEAE Granulosis Virus], [PP 899: Plutera xylostella granules Viruses], [PP 900: Spodoptera albra nuclear polyhedrosis virus], [PP 901: Spodoptera exulpum nuclear polyhedrosis virus], [PP 902: Spodoptera exiqua nuclear polyhedrosis virus], [PP 903: Spodoptera fulgiperta nuclear polyhedra Body disease virus], [PP 904: Spodoptera ritritalis nuclear polyhedrosis virus], [PP 905: Spodoptera ritula nuclear polyhedrosis virus], [PP 906: Ablebita coccia], [PP 907: aquaria spp.], [PP 908: Agamel Miss Decauda], [PP 909: Allantonem spp.], [PP 910: Anfimel miss spp.], [PP 911: Veginia syllidola], [PP 912: Bobienema spp.], [PP 913: Camelonia spp.], [PP 914: Kitto Woodyella obofilamenta], [PP 915: Contr. Tenkas spp.], [PP 916: Kori Shimer mis s pp.], [PP 917: Deprotolize spp.], [PP 918: Empidomel miss spp.], [PP 919: Filippivebaim rape sanda], [PP 920: Gastromel miss spp.], [PP 921: Gongiro Nema spp.], [PP 922 : [Jinopoesia shubadubapara], [PP 923: heterolabditis bacterifolia], [PP 924: heterolabditis boujardi], [PP 925: heterolabditis heliothisis], [PP 926: heterolabditis indica], [PP 927: Heterolabditis malereitas], [PP 928: Heterolabditis megidis], [PP 929: Heterolabditis zealandica], [PP 930: Hexamel miss spp.], [PP 931: Hydromer Miss spp.], [PP 932 : Isomel miss spp.], [PP 933: limomel miss spp.], [PP 934: maupasina way ], [PP 935: Melmis naigressense], [PP 936: mesomel miss spp.], [PP 937: neomesomel miss spp.], [PP 938: Neoparasity lensus ragrossi], [PP 939: octomi o mer mis spp.], [PP 940: Paralacita Ferenx spp.], [PP 941: Parasite Rehab ditis spp.], [PP 942: Paracitic Rex spp.], [PP 943: Pertili Melmis curicis], [PP 944: Fasu Marab Ditis hermaphrodita], [PP 945: Physioptra spp.], [PP 946: Protollera spp.], [PP 947: Pterigigo del Matitas spp.], [PP 948: Romanomel miss spp.], [PP 949: Souretam kay Dalachens], [PP 950: Sphaerella liarensis spp.], [PP 951: Spirula gaianensis], [PP 952: Steinernema Capocapsae], [PP 9 53: Steiner Nema Fertariae], [PP 954: Steiner Nema Gracelai], [PP 955: Steiner Nema Crushay], [PP 956: Steiner Nema Riobrabe], [PP 957: Steiner Nema Scapteris], [PP 958: Steiner Nema Scarabaei], [PP 959 : [Stainanema Siamuka Yai], [PP 960: Strelco Baimermis putter Seni], [PP 961: Subaru la spp.], [PP 962: Salpretilex elongitas], [PP 963: Tetrameles spp.], [PP 964: Thymol] [PP 965: Neem oil], [PP 966: Azadirachtin], [PP 967: Shrimp nigrum wood extract], [PP 968: Garlic extract], [PP 969: veratrin], [PP 970: Ryanosine], [PP 971: Mistletoe ], [PP 972: Tansy extract], [PP 973: Niyomogi extract] [PP 974: Alveolaris extract component], [PP 975: Calendula extract component], [PP 976: Oak leaf and bark], [PP 977: American red root seed oil], [PP 978: Celastrus angulatus bark], [PP 9 7 9 Leaves], [PP 980: mustard powder], [PP 981: Japanese horseradish extract], [PP 982: chitin], [PP 983: Chinese lichen extract], [PP 984: quinoa saponin], [PP 985: quinconazole], [PP 986: Fluorophorpet], [PP 987: Propamidine], [PP 988: Cassia nigricans extract], [PP 989: Brady rhizobium elkani], [PP 990: Rhizobium spp.], [PP 991: Trichoderma spp], [PP 992: Above Compound represented by Formula (c), [PP993: Compound represented by Formula (d)], [PP994: Compound represented by Formula (e)], [PP995: Compound represented by Formula (f) Compounds to be expressed], [ PP 996: brofuranilide], [PP 997: fluazaindolizine], [PP 998: compound represented by the above formula (g)], [PP 999: compound represented by the above formula (h)], [PP 1000: piperonyl butoxide], [PP1001: sesomax], [PP1002: sulfoxide], [PP1003: N- (2-ethylhexyl) -8,9,10-trinorborn-5-ene-2,3-dicarboximide], [PP1004: N -Decuriimidazole], [PP1005: WARF-Anti-Resistant], [PP1006: TBPT], [PP1007: TPP], [PP1008: IBP], [PP1009: PSCP], [PP1010: Methyl iodide], [PP1011 : T-phenylbutenone], [PP1012: diethyl maleate], [PP1013: DMC], [PP1014: FDMC], [PP1015: ETP], [PP1016: ETN], [PP1017: fluralanel], [PP1018: pyrisoqui , [PP1019: kappa bifenthrin], [PP 1020: capatefluthrin], [PP 1021: dichloro mesothias], [PP 1022: fluxamethamide], [PP 1023: a compound represented by the above formula (i)], [PP 1024 : Compound represented by the above formula (j)], [PP1025: compound represented by the above formula (k)], [PP1026: compound represented by the above formula (1)], [PP1027: above formula (m) Compounds], [PP1028: compounds represented by the above formula (n)], [PP1029: compounds represented by the above formula (o)], [PP1030: represented by the above formula (p) Compound], [PP1031: compound represented by the above formula (q)], [PP1032: oxpoconazole], [PP1033: methyl = (1R, 2R, 3R) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazol-1-ylmethyl) Cyclopentane carboxylate], [PP1034: methyl = (1S, 2S, 3S) -3-[(4-chlorophenylmethyl] -2-hydroxy-1-methyl-2- (1H-1,2,4-triazole) 1-ylmethyl) cyclopentanecarboxylate], [PP1035: methyl = (1S, 2R, 3S) -3-[(4-chlorophenyl) methyl] -2-hydroxy-1-methyl-2- (1H-1,2 , 4-Triazol-1-ylmethyl) cyclopentanecarboxylate], [PP 1036: clozolinate], [PP 1037: phenamidone], [PP 1038: phenamine strobin], [PP 1039: mepronil], [PP 1040: acibenzolar S methyl], [PP1041: Edifenphos], [PP1042: Ethylymol], [PP1043: Iminoctadine], [PP1044: Iminoctadine triacetate], PP1045: Iodocarb], [PP 1046: Octylinone], [PP 1047: Technazen], [PP 1048: Bisethylenediamine copper complex salt of dodecylbenzenesulfonic acid [II], [PP 1049: Dipimethytron], [PP 1050: 2- {3- [2-] (1-{[3,5-bis (difluoromethyl) -1H-pyrazol-1-yl] acetyl} piperidin-4-yl) -1,3-thiazol-4-yl] -4,5-dihydro-1 , 2-Oxazol-5-yl} -3-chlorophenyl = methanesulfonato], [PP 1051: 4- (2-bromo-4-fluorophenyl) -N- (2-chloro-6-fluorophenyl) -1,3-dimethylphenol] Dimethyl-1H-pyrazole-5-amine], [PP1052: 2,2-Dimethyl-9-fluoro-5- (quinolin-3-yl) -2,3-dihydro-benzo [f] [1,4] Oxazepin], [PP1053: 2- [6- (3-fluoro-4-methoxyphenyl) -5-methylpyridin-2-yl] quinazoline], [PP1054: N '-(2,5-dimethyl-4-phenoxy] Phenyl) -N-ethyl-N-methylmethaneimidamide], [PP 1055: N '-[4-({3-[(4-chlorophenyl) methyl] -1,2,4-thiadiazol-5-yl} oxy] ), 2,5-Dimethylphenyl] -N-ethyl-N-methylmethanimidamide], [PP1056: Folate], [PP1057: Bioallethrin], [PP1058: Bioresmethrin], [PP1059: Cypenothrin], [PP1060] : Enpentrin], [PP1061: Etophenprox], [PP1062: Flumethrin], [PP1063: Halfenprox], [PP1064: Heptafluthrin], [PP1065: Imiprotri] ], [PP1066: cadestrin], [PP1067: meperfluthrin], [PP1068: monfluorothrin], [PP1069: phenothrin], [PP1070: prarethrin], [PP1071: resmethrin], [PP1072: tetramethrin], [PP1073: tetramethrin] Methylfluthrin], [PP1074: Transfluthrin], [PP1075: Benfluthrin], [PP1076: Flufenprox], [PP1077: Flumethrin], [PP1078: Sigmacypermethrin], [PP1079: Flamethrin], [PP1080: Metofluthrin], [PP1081: profluthrin], [PP1082: dimefluthrin], [PP1083: epsilon-methoflthrin], [PP1084: 2,3,5,6-tetrafluoro-4-methylbenzyl (EZ)-(1RS, 3RS; 1RS, 3SR) -2,2-Dimethyl-3-prop-1-enylcyclopropanecarbo Sylate], [PP1085: 2,3,5,6-tetrafluoro-4- (methoxymethyl) benzyl (1RS, 3RS; 1RS, 3SR) -2,2-dimethyl-3- (2-methyl-1-propenyl) ) Cyclopropanecarboxylate], [PP1086: epsilon mont fluorotrithrin], [PP1087: Cartap], [PP1088: Thiosultap-2 sodium salt or bislutapt], [PP1089: Thiosultap-1 sodium salt or monosultap], [PP1090: rufenuron] ], [PP1091: Stinging nettle extract], [PP1092: spinosad], [PP1093: triflumesopyrin], [PP1094: clodinafop propargyl], [PP1095: cyhalofop], [PP1096: cyhalofop butyl], [PP109: PP 1097: Diclohop methyl], [PP 1098: Fenoxaprop ethyl], [PP 10 99: Fenoxaprop P], [PP1100: fluazifop], [PP1101: fluazifop butyl], [PP1102: fluazifop P], [PP1103: haloxyfop], [PP1104: haloxyfop methyl], [PP1105: haloxyhop P], [PP 1106: haloxyfop P methyl], [PP 1107: metamihop], [PP 1108: propacihop], [PP 1109: Qizaro hop], [PP 1110: Qizalo hop ethyl], [PP 1111: Qizalo hop P], [PP 1112: Qizalo hop P ethyl ], [
PP 1113: Alloxydim], [PP 1114: Butoxydimm], [PP 1115: Cycloxydim], [PP 1116: Propoxydim], [PP 1117: Tralkoxidim], [PP 1118: Amidosulfuron], [PP 1119: Aziimsulfuron], [PP 1120: Bensulfuron ], [PP1121: bensulfuron methyl], [PP1122: chlorsulfuron], [PP1123: cinosulfuron], [PP1124: cyclosulfamuron], [PP1125: etamethsulfuron], [PP1126: etamethsulfuron methyl], [PP1127: ethoxysulfuron], [PP1128: flazasulfuron], [PP1129: flucetosulfuron], [PP1130: flupyrsulfuron], [PP1131: flupyrsulfuron methyl sodium], [PP1132: holamsulfuron], [PP1133: imazosulfuron], [PP1134: iodosulfuron], [PP1135: iodosulfuron Chill sodium], [PP1136: iodine sulfuron], [PP1137: sodium ionsulfuron], [PP1138: mesosulfuron methyl], [PP1139: methazosulfuron], [PP1140: methsulfuron methyl], [PP1141: orthosulfamuron ], [PP1142: Oxasulfuron], [PP1143: Primisulfuron], [PP1144: Primisulfuron methyl], [PP1145: Propyrisulfuron], [PP1146: Prosulfuron], [PP1147: Pyrazosulfuron], [PP1148] [Pylazosulfuron ethyl], [PP1149: rimsulfuron], [PP1150: sulfometuron], [PP1151: sulfometuron methyl], [PP1152: sulfosulfuron], [PP1153: thifensulfuron methyl], [PP1154: trias Ruflon], [PP1 155: tribenuron], [PP 1156: tribenuron methyl], [PP 1 157 Trifloxysulfuron sodium salt], [PP1158: triflusulfuron], [PP1159: tritosulfuron], [PP1160: imazapic ammonium salt], [PP1161: imazamethabenz], [PP1162: imazamethabenzmethyl], [PP1163: imazamox], [PP1164: imazamox ammonium salt], [PP1165: imazapyr], [PP1166: imazapyr isopropylammonium salt], [PP1167: imazaquin ammonium salt], [PP1168: imazethapyr ammonium] Salt], [PP1169: flumetsulam], [PP1170: methoslam], [PP1171: penoxsulam], [PP1172: pyroxyslam], [PP1173: bispyribac], [PP1174: bispyribac sodium salt], [PP1175: pyribenzoxime], [PP1175: pyribenzoxim], PP1176: Pyriphthalide], [PP1177: Pyriminobac], [PP1178: Pyriminobac [Methyl], [PP1179: pyrithiobac sodium salt], [PP1180: pyrimisulfan], [PP1181: triafamone], [PP1182: flucarbazone], [PP1183: flucarbazone sodium salt], [PP1184: propoxycarbazone] [PP1185: Propoxycarbazone sodium salt], [PP1186: Thienecarbazone], [PP1187: Thienecarbazone methyl], [PP1188: Cyanazine], [PP1189: Desmethrin], [PP1190: Dimetamethrin], [PP1191: Prometon], [PP1192: Propazine], [PP1193: Simetryne], [PP1194: Terbumetone], [PP1195: Terbutyrazine], [PP1196: Terbutrin], [PP1 197: Trietadine], [PP1198: Bromacil], [PP1 199: Tabacil], [PP 1200] : Fenmedifam], [PP1201: chlorbromuron], [PP1202: chlorotoluron [PP1203: chloroxuron], [PP 1204: dimeflon], [PP 1205: ethidimolone], [PP 1206: phenuron], [PP 1207: isouron], [PP 1208: isoproturon], [PP 1209: fluomethuron], [PP 1210: benzthiazlon], [PP 1210: PP1211: methabenzthiazuuron], [PP1212: methoxuron], [PP1213: methobromron], [PP1214: nebron], [PP1215: siduron], [PP1216: monolinuron], [PP1217: propanil], [PP1218: pentano] Kroll], [PP1219: Ioxynyl], [PP1220: Bromophenoxyme], [PP1221: Bromoxinyl Octanoate], [PP1222: Ioxynyl Octanoate], [PP1223: Cyclopyrimolate], [PP1224 : Piridaphor], [PP1225: Pyridate], [PP1226: Diquat], [PP1227: Paraquat dichloride [PP1228: diquat dibromide], [PP1229: biphenox], [PP1230: acifluorfen sodium salt], [PP1231: chloromethoxyphen], [PP1232: fluoroglycophene ethyl], [PP1233: ethoxyphenethyl], [PP 1234: fomethafen], [PP 1235: fomethafen sodium], [PP 1236: halosaphene], [PP 1237: fluazolate], [PP 1238: sinidone], [PP 1239: sinidone ethyl], [PP 1240: flumicrolac pentyl], [PP 1241 : Fluthiaset methyl], [PP1242: thidiazimine], [PP1243: oxadiazone], [PP1244: oxadiargyl], [PP1245: bencarbazone], [PP1246: azaphenidine], [PP1247: pentoxazone], [PP1248: butafenacil], [PP1249 : Benzphendizone], [PP1250: saflufenacil], [ PP1251: Profluazole], [PP1252: Pyraclonyl], [PP1253: Thiafenacil], [PP1254: Flufenpyr], [PP1255: Flufenpyrethyl], [PP1256: Trifludimoxazine], [PP1257: Diflufenican], PP1258: norflurazon], [PP1259: beflubutamide], [PP1260: pyrocolinaphen], [PP1261: flurochloridon], [PP1262: fluridone], [PP1263: phenquinotrione], [PP1264: flurutamon], [PP1265: Sulcotrione], [PP1266: tefuryltrione], [PP1267: isoxachlortol], [PP1268: benzophenap], [PP1269: pyrasulfotol], [PP1270: pyrazolinate], [PP1271: benzobicyclone] [PP1272: topramezone], [PP1273: pyrazoloxifene], [PP1274: bicyclopyrone], [PP 1275: tolpi Rate], [PP1276: Acroniphen], [PP1277: Amitrole], [PP1278: Glyphosate Ammonium Salt], [PP1279: Glyphosate Diammonium Salt], [PP1280: Glyphosate Sodium Salt], [PP1281: Glyphosate Guanidine Derivative Salt], [ PP1282: glyphosate choline salt], [PP1283: glyphosate BAPMA salt], [PP1284: glufosinate P], [PP1285: glufosinate P sodium salt], [PP1286: glufosinate P ammonium salt], [PP1287: bialaphos], [PP1288: ashram ], [PP1289: Benfluralin], [PP1290: Butoralin], [PP1291: Dinitramine], [PP1292: Pendimethalin], [PP1293: Trifluralin], [PP1294: Dithiopyr], [PP1295: Butamiphos], [PP1296: Ami] Prophos methyl], [PP1297: thiazopyr], [PP 1298: tebutam], [PP1 299: propyzamide], [PP1300: prodiamine], [PP1301: DCPA], [PP1302: chlorprofam], [PP1303: profam], [PP1304: calbetamide], [PP 1305: flumplop M ], [PP1306: Butacrol], [PP1307: Dimethacrol], [PP1308: Dimethenamide P], [PP1309: Metazachlor], [PP1310: S-Metrachlor], [PP1311: Petoxamide], [PP1312: Pretilacrole], PP 1313: Propacrol], [PP 1314: Propysochlor], [PP 1315: Diphenamide], [PP 1316: Tenil Kroll], [PP 1317: Napropamide], [PP 1318: Napropamide M], [PP 1319: Naproanilide], [PP 1320: Mefena Set] [PP1321: Fentrazamide], [PP1322: Ipphencarbazone], [PP1323: Anilophos], [PP1324: Caffenstrol], [PP 1325: piperophos], [PP 1326: piroxasulfone], [PP 1327: phenoxasulfone], [PP 1328: diclovenyl], [PP 1329: chlorthiamide], [PP 1330: isoxabene], [PP 1331: flupoxam], [ PP1332: Indadifram], [PP1333: Triadifram], [PP1334: dinoseb], [PP1335: dinoterb], [PP1336: butyrate], [PP1337: cycloate], [PP1338: dialate], [PP1339: dimepiperate], [PP1340: Esprocarb], [PP1341: molinate], [PP1342: orbencarb], [PP1343: pebrate], [PP1344: prosulfb], [PP1345: benthiocarb], [PP1346: thiocal basil], [PP1347: trialate], [PP1348: barna] Rate], [PP1349: bensulide], [PP1350: benfresate], [PP1351: CA], [PP1352: darapon], [PP1353: full propanate], [PP1354: chromeprop], [PP1355: 2,4-D ammonium], [PP1356: 2,4-D butytyl], [PP1357: 2, 4-D 2-Butoxypropyl], [PP 1358: 2,4-D 3-Butoxypropyl], [PP 1359: 2,4-D-butyl], [PP 1360: 2,4-D diethylammonium], [PP 1361: 2 , 4-D dimethyl ammonium], [PP1362: 2,4-D diol amine salt], [PP 1363: 2,4-D dodecyl ammonium], [PP 1364: 2,4-D ethyl], [PP 1 365: 2, 4 -D 2-ethylhexyl], [PP 1366: 2,4-D heptyl ammonium], [PP 1367: 2,4-D isobutyl], [PP 1 368: 2,4-D isooctyl], [PP 1369: 2,4-D isopropyl ], [PP 1370: 2,4-D isopropyl Ammonium], [PP1371: 2, 4-D lithium], [PP1372: 2, 4-D-meptyl], [PP1373: 2, 4-D-methyl], [PP1 374: 2, 4-D-octyl], [PP1 375: 2,4-D pentyl], [PP 1376: 2,4-D propyl], [PP 1377: 2,4-D sodium salt], [PP 1378: 2,4-D tefuryl], [PP 1379: 2,4-D Tetradecylammonium], [PP1380: 2,4-D triethylammonium], [PP1381: 2, 4-D tris (2-hydroxypropyl) ammonium], [PP1382: 2,4-D tololamine salt], [PP1383 : [2,4-D choline salt], [PP1 384: 2,4-D BAPMA salt], [PP 1385: 2, 4-DB dimethyl ammonium], [PP 1 386: 2, 4-DB isooctyl], [PP 1387: 2, 2, 3 4-DB butyl], [PP1388: 2,4-DB sodium salt], [PP138 9: 2,4-DB potassium salt], [PP1390: 2,4-DB choline salt], [PP1391: 2, 4-DB BAPMA salt], [PP1392: MCPA], [PP1393: MCPA dimethyl ammonium], [PP1392: MCPA] PP1394: MCPA 2-ethylhexyl], [PP 1395: MCPA isooctyl], [PP 1396: MCPA butytyl], [PP 1397: MCPA butyl], [PP 1398: MCPA diamine amine salt], [PP 1399: MCPA ethyl], [PP1400: MCPA isobutyl] ], [PP 1401: MCPA isopropyl], [PP 1402: MCPA methyl], [PP 1403: MCPA all amine salt], [PP 1404: MCPA sodium salt], [PP 1405: MCPA traolamine salt], [PP 1406: MCPA choline salt], [PP 1407: MCPA BAPMA salt], [PP 1408: MCPB], [PP 1409: MCPB et al], [PP 1410: MCPB methyl], [PP1 14 PP 1411: MCPB sodium salt], [PP 1412: MCPB choline salt], [PP 1413: MCPB BAPMA salt], [PP 1414: mecoprop], [PP 1415: mecoprop dimethylammonium], [PP 1416: mecopropiolamine salt], [PP 1417 : Mecoprop etazyl], [PP1418: Mecoprop 2-ethylhexyl], [PP 1419: Mecoprop isobutyl], [PP 1420: Mecoprop methyl], [PP 1421: Mecoprop potassium salt], [PP 1422: Mecoprop sodium salt], [PP1423: Mecoproptrol amine salt], [PP1424: Mecoprop choline salt], [PP1425: Mecoprop P], [PP1426: Mecoprop P dimethylammonium], [PP1427: Mecoprop P2 ethylhexyl], [PP1428: Mecoprop P isobutyl ], [PP1429: Mecoprop P potassium salt], [PP 1430: mecoprop P choline salt], [PP 1431: mecoprop BAPMA salt], [PP 1432: dicloprop butchi], [PP 1433: dicloprop], [PP 1434: dicloprop dimethyl ammonium], [PP 1435: dicloprop ethyl ammonium], [PP 1436: dicloprop 2 ethyl hex
Syl], [PP1437: dicloprop isoctyl], [PP1438: dicloprop methyl], [PP1439: dicloprop potassium salt], [PP1440: dicloprop sodium salt], [PP1441: dicloprop choline salt (], [PP1442 : Dicloprop BAPMA salt], [PP 1443: dicloprop P dimethyl ammonium], [PP 1444: dicloprop P], [PP 1445: dicloprop P 2 ethylhexyl], [PP 1446: dicloprop P choline salt], [PP 1447: dicloprop PBAPMA salt], [PP1448: chloramine], [PP1449: dicamba dimethylammonium], [PP1450: dicambadichloramine salt], [PP1451: dicambadiolamine salt], [PP1452: dicamba isopropylammonium], PP1453: dicamba methyl], [PP1454: dicambaol amine salt], [PP 1455: dicamba potassium salt], [PP 1456: dicamba sodium salt], [PP 1457: dicambatrol amine salt], [PP 1458: dicamba choline salt], [PP 1459: dicamba BAPMA salt], [PP 1460: 2, 3, 6 -TBA dimethylammonium], [PP1461: 2,3,6-TBA lithium], [PP1462: 2,3,6-TBA potassium salt], [PP1463: 2,3,6-TBA sodium salt], [PP1464: Triclopyropistyl], [PP1465: Triclopyrethyl], [PP1466: Triclopyrtriethylammonium], [PP1467: Fluoxypyr], [PP1468: Fluoxypyrmeptyl], [PP1469: Aminopyralid potassium salt], [PP1469: PP1470: aminopyralid tris (2hydroxypropyl) ammonium], [PP1471: aminopyralidcholine salt], [PP1472: clopyralidmethyl], [PP147 3: Clopyralidolamine salt], [PP1474: Clopyralid potassium salt], [PP1475: clopyralid tris (2-hydroxypropyl) ammonium], [PP1476: clopyralidcholine salt], [PP1477: quinclorac], [PP1478: quinmelac] [PP1479: Benazoline ethyl], [PP1480: Naptalam], [PP1481: Diflufenzopyr-sodium salt], [PP1482: Diphenzocoat], [PP1483: DSMA], [PP1484: Bromobutide], [PP1485: Flurenol], [PP1484: PP1486: Synmethylin], [PP1487: Cumirolon], [PP1488: Dimron], [PP1489: Methyldimuron], [PP1490: Etobenzanide], [PP1491: Indanofan], [PP1492: Hosamine], [PP1493: Oxadichromephone], [PP1494 : Oleic acid], [PP1495: methiozoline], [PP1496: pelargon ], [PP1497: phenisochamm], [PP1498: Suep], [PP1499: aminocyclopyracrole], [PP1500: aminocyclopyracrolet methyl], [PP1501: aminocyclopyracrole potassium], [PP1502: difenoxuron], PP 1503: Tridiphane], [PP 1504: Maleic Hydrazide], [PP 1505: Halauxifene], [PP 1506: Difenodiconazole], [PP 1507: 3- [5- (4-Chlorophenyl) -2,3-dimethyl- 1,2-oxazolidin-3-yl] pyridine], [PP1508: bromothalonyl], [PP1509: phenamacryl], [PP1510: ethyl (2Z) -3-amino-2-cyano-3-phenylacrylate], [PP1511 : N-[(2-chlorothiazol-5-yl) methyl] -N-ethyl-6-methoxy-3-nitropyridin-2-amine], [[ PP1512: afoxolanel], [PP1513: borax], [PP1514: boric acid], [PP1515: disodium octaborate], [PP1516: sodium borate], [PP1517: sodium metaborate], [PP1518: diflovidazine] [PP1519: azocyclotine], [PP1520: calcium cyanide], [PP1521: potassium cyanide], [PP1522: sodium cyanide], [PP1523: nicotine].

  The composition of the present invention preferably contains 1 to 7 components selected from group A, group B, group C, group D, group E and group F.

  In the control method of the present invention, the mixing ratio (weight ratio) of the present compound to one or more components selected from Group A, Group B, Group C, Group D, Group E and Group F is the ratio of the plant to be protected Depending on the type, the type and frequency of occurrence of the pest to be controlled, the formulation form, the application time, the application method, the application method, the application place, the weather conditions, etc. When the compound is applied, the compound contained in group A is (the present compound) / (one or more components selected from group A) = 1/100 to 10000/1, regardless of the presence or absence of other components. With respect to the compounds contained in B, regardless of the presence or absence of other components, (the present compound) / (one or more components selected from group B) = 1/10 to 100/1 and the components contained in group C With or without other components (the present compound) / (group 1 or more components selected from 1/10 to 100/1, with regard to the components contained in group D regardless of the presence or absence of other components (this compound) / (1 or more components selected from group D) (The present compound) / (one or more components selected from group E), regardless of the presence or absence of other components, for the components contained in group E) = 1/100 to 10000 With respect to the components contained in / 1 and the group F, regardless of the presence or absence of other components, (the present compound) / (one or more components selected from the group F) = 1/100 to 10000/1.

  Examples of the composition of the present invention include the following.

A pest control composition containing the present compound and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (I) and one or more compounds selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (II) and one or more compounds selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (III) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IV) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of the group (V) and one or more compounds selected from the group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VI) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VII) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VIII) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IX) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (X) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of the group (XI) and one or more compounds selected from the group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (XII) and one or more compounds selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (XIII) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XIV) and one or more compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XV) and one or more compounds selected from group (A).
A pest control composition containing the aromatic compound according to any one of the group (XVI) and one or more compounds selected from the group (A).
A pest control composition comprising the aromatic compound according to any of group (XVII) and one or more compounds selected from group (A).
A pest control composition containing the aromatic compound according to any of group (XVIII) and one or more compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XIX) and one or more compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XX) and one or more compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XXI) and one or more compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XXII) and one or more compounds selected from group (A).
A pest control composition containing the carbamate compound according to any one of group (XXIII) and one or more compounds selected from group (A).

A pest control composition containing the present compound and a compound selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (I) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (II) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (III) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IV) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (V) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VI) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VII) and a compound selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (VIII) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IX) and a compound selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (X) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XI) and a compound selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XII) and a compound selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (XIII) and a compound selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of the group (XIV) and a compound selected from the group (A).
A pest control composition comprising the tetrazolinone compound according to any one of the group (XV) and a compound selected from the group (A).
A pest control composition containing the aromatic compound according to any of group (XVI) and a compound selected from group (A).
A pest control composition comprising the aromatic compound according to any of group (XVII) and a compound selected from group (A).
A pest control composition containing the aromatic compound according to any of group (XVIII) and a compound selected from group (A).
A pest control composition containing the carbamate compound according to any of group (XIX) and a compound selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XX) and a compound selected from group (A).
A pest control composition containing the carbamate compound according to any one of group (XXI) and a compound selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XXII) and a compound selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XXIII) and a compound selected from group (A).

A pest control composition containing the present compound and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (I) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (II) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (III) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IV) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (V) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VI) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VII) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VIII) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IX) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (X) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XI) and two compounds selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (XII) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XIII) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XIV) and two compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of the group (XV) and two compounds selected from the group (A).
A pest control composition comprising the aromatic compound according to any of group (XVI) and two compounds selected from group (A).
A pest control composition containing the aromatic compound according to any of group (XVII) and two compounds selected from group (A).
A pest control composition comprising the aromatic compound according to any of group (XVIII) and two compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XIX) and two compounds selected from group (A).
A pest control composition containing the carbamate compound according to any of group (XX) and two compounds selected from group (A).
A pest control composition containing the carbamate compound according to any of group (XXI) and two compounds selected from group (A).
A pest control composition containing the carbamate compound according to any of group (XXII) and two compounds selected from group (A).
A pest control composition containing the carbamate compound according to any one of group (XXIII) and two compounds selected from group (A).

A pest control composition containing the present compound and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (I) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (II) and three compounds selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (III) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IV) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (V) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VI) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VII) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (VIII) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (IX) and three compounds selected from group (A).
The pest control composition containing the tetrazolinone compound in any one of group (X), and three types of compounds chosen from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XI) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XII) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XIII) and three compounds selected from group (A).
A pest control composition containing the tetrazolinone compound according to any one of group (XIV) and three compounds selected from group (A).
A pest control composition comprising the tetrazolinone compound according to any one of group (XV) and three compounds selected from group (A).
A pest control composition containing the aromatic compound according to any of group (XVI) and three compounds selected from group (A).
A pest control composition containing the aromatic compound according to any of group (XVII) and three compounds selected from group (A).
A pest control composition comprising the aromatic compound according to any of group (XVIII) and three compounds selected from group (A).
A pest control composition containing the carbamate compound according to any of group (XIX) and three compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XX) and three compounds selected from group (A).
A pest control composition comprising the carbamate compound according to any of group (XXI) and three compounds selected from group (A).
A pest control composition containing the carbamate compound according to any of group (XXII) and three compounds selected from group (A).
A pest control composition containing the carbamate compound according to any one of group (XXIII) and three compounds selected from group (A).

A pest control composition containing the present compound and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (I) and a compound selected from group (B).
A pest control composition containing the tetrazolinone compound according to any one of group (II) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (III) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (IV) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (V) and a compound selected from group (B).
A pest control composition containing the tetrazolinone compound according to any one of group (VI) and a compound selected from group (B).
A pest control composition containing the tetrazolinone compound according to any one of group (VII) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (VIII) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (IX) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (X) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (XI) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (XII) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of group (XIII) and a compound selected from group (B).
A pest control composition comprising the tetrazolinone compound according to any one of the group (XIV) and a compound selected from the group (B).
A pest control composition containing the tetrazolinone compound according to any one of group (XV) and a compound selected from group (B).
A pest control composition containing the aromatic compound according to any one of the group (XVI) and a compound selected from the group (B).
A pest control composition containing the aromatic compound according to any of group (XVII) and a compound selected from group (B).
A pest control composition containing the aromatic compound according to any of group (XVIII) and a compound selected from group (B).
A pest control composition containing the carbamate compound according to any of group (XIX) and a compound selected from group (B).
A pest control composition comprising the carbamate compound according to any of group (XX) and a compound selected from group (B).
A pest control composition comprising the carbamate compound according to any of group (XXI) and a compound selected from group (B).
A pest control composition comprising the carbamate compound according to any of group (XXII) and a compound selected from group (B).
A pest control composition comprising the carbamate compound according to any of group (XXIII) and a compound selected from group (B).

  Examples of the composition of the present invention also include the following.

That is, the composition of the present invention, wherein the combination of the present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E and Group F is the following combination:
“The present compound AA1-BA1 to AA319-BA6365, the present compound AB1-BB1 to AB119-BB511, the present compound AB1-BB1001 to AB119-BB3016, the present compound AC1-BC1 to AC10200-BC5278, the present compound AD1-BD1 to AD2160-BD558 The present compound AE1-BE1 to AE5220-BE5982, the present compound AF1-BF1 to AF360-BF1300, the present compound AG1-BG1 to AG327-BG6699, the present compound AH1-BH1 to AH3780-BH4501, the present compound AI1-BI1 to AI6096-BI1423 The present compound AJ1-BJ1 to AJ32-BJ366 and the present compounds AK1-BK1 to AK2688-BK1287 (hereinafter, described as any one of the compounds AA1-BA1 to AK2688-BK1287) and “PP1” (mixing ratio) 1:10 to 10: 1) (Composition A1); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP2” (mixing ratio 1:10 to 10: 1) (Composition A2 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP3" (mixing ratio 1:10 to 10: 1) (Composition A3); "Compounds AA1-BA1 to AK2688-BK1287" Any one " Combination with PP 4 "(mixture ratio 1: 10 to 10: 1) (Composition A 4);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP5 "(mixture ratio 1: 1 to 1: 100) (Composition A5); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP6” (mixing ratio 1: 1 to 1: 100) (Composition A6); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP7” (mixing ratio 1: 1 to 1: 100) (Composition A7); “any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP8” (mixture ratio 1:10 to 10: 1) (composition A8); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP9” (mixture ratio 1: 1 to 1: 100) (Composition A 9); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 10” (mixing ratio 1: 1 to 1: 100) (Composition A 10); " Any one of AA1 -BA1 to AK2688-BK1287 "and" PP11 "(mixing ratio 1: 1 to 1: 100) (composition A11);" any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition A12” with “PP12” (composition A12); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP13” (mixture 1) "Composition A13";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP14" (mixing ratio 1: 1 to 1: 100) (Composition A14) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP15” (mixing ratio 1: 1 to 1: 100) (Composition A15); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP16” (mixture ratio 1:10 to 10: 1) (Composition A16); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP17” (Mixing ratio 1:10 to 10: 1) (Composition A17); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP18” (Mixing ratio 1:10 to 10: 1) (Composition A17) “Composition A18);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP19 ”(mixing ratio 1:10 to 10: 1) (Composition A19);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP20” (mixture ratio 1:10 to 10: 1) (composition A20); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP21” Combination (mixture ratio 1:10 to 10: 1) (composition A21); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP22” (mixture ratio 1:10 to 10: 1 (Composition A22); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP23” in combination (mixing ratio 1:10 to 10: 1) (Composition A23); “Compound AA1 to BA1 ~ Any one of AK2688-BK1287 "and" PP24 "(mixture ratio 1:10 to 10: 1) (Composition A24);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP25 (Mixture ratio 1:10 to 10: 1) (composition A 25); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP26” (mixture ratio 1:10 to 10) "Composition A26";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP27" (mixing ratio 1:10 to 10: 1) (Composition A27); "Compound AA1 Any one of “BA1 to AK2688-BK1287” and “PP28” (mixture ratio 1:10 to 10: 1) (composition A28); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP29” (mixture ratio 1:10 to 10: 1) (Composition A 29); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP31” 1:10 to 10: 1) (Composition A30); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP32” (mixing ratio 1:10 to 10: 1) (Composition A31 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP33" (mixing ratio 1:10 to 10: 1) (Composition A32); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and PP34 (mixture ratio 1:10 to 10: 1) (Composition A33); Combination of any one of Compounds AA1-BA1 to AK2688-BK1287 and PP35 (Composition A33) Mixing ratio 1:10 to 10: 1) (Composition A34); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP36" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP38” (mixing ratio 1:10 to 10: 1) (composition A36); “compound AA1 to BA1 to AK2688” B A combination of “one of K1287” and “PP39” (mixture ratio 1:10 to 10: 1) (composition A 37); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP40” Combination (mixture ratio 1:10 to 10: 1) (Composition A 38); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP41" (mixture ratio 1:10 to 10: 1) (Composition A39); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP43” (mixing ratio 1: 1 to 1: 100) (Composition A40); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP44” (mixture ratio 1: 1 to 1: 100) (composition A41); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP49” (Combination ratio 1: 1 to 1: 100) (composition A 42); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP51” (mixture ratio 1: 1) "Composition A43";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP52" (mixing ratio 1:10 to 10: 1) (Composition A44); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP53” (mixture ratio 1:10 to 10: 1) (composition A45); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP54” (mixture ratio 1:10 to 10: 1) (composition A46); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP55” (mixture ratio 1 “Composition A47);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP56 ”(mixing ratio 1: 1 to 1: 100) (Composition A48) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP57” (mixing ratio 1: 1 to 1: 100) (Composition A49); “Compound AA1-BA1 to AK2688-BK1287 Combination of “one or more” and “PP58” (mixture ratio 1:10 to 10: 1) (composition A50); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP59” Mixing ratio 1:10 to 10: 1) (Composition A51); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP60" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP61” (mixing ratio 1:10 to 10: 1) (composition A53); “compound AA1-BA1 to AK2688- Any one of BK1287 and PP62 (mixture ratio 1: 1 to 1: 100) (composition A 54); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP63” Combination (mixture ratio 1: 1 to 1: 100) (Composition A 55); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP64” (mixture ratio 1:10 to 10 "Composition A56";"Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP65" (mixing ratio 1:10 to 10: 1) (Composition A57); "Compound AA1 -Any one of “BA66 to AK2688-BK1287” and “PP66” (mixture ratio 1:10 to 10: 1) (composition A58); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP67” (mixture ratio 1:10 to 10: 1) (Composition A59); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP68” (mixture ratio 1:10 “Composition A60);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP69 ”(mixing ratio 1:10 to 10: 1) (Composition A61); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP70” (mixture ratio 1:10 to 10: 1) (Composition A 62); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP71” (mixture ratio 1:10 to 10: 1) (composition A63); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP72” (mixture "Composition A64";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP 73" (mixing ratio 1:10 to 10: 1) (Composition A65) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP74” (mixing ratio 1:10 to 10: 1) (Composition A66); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1:75 to 10: 1” (composition A67) with “PP75” (composition A67); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP76” (Composition ratio 1:10 to 10: 1) (Composition A 68); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP77” (mixture ratio 1:10 to 10: 1) Composition A69); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP78” (mixing ratio 1:10 to 10: 1) (Composition A70); “Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP79” (mixture ratio 1:10 to 10: 1) (composition A71); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP80” Combination (mixture ratio 1:10 to 10: 1) (composition A 72); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP81” (mixture ratio 1:10 to 10: 1 (Composition A73); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP82” (mixing ratio 1:10 to 10: 1) (Composition A74); “Compound AA1-BA1” ~ A combination of one of “AK2688-BK1287” and “PP83” (mixture ratio 1:10 to 10: 1) (composition A75); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP84” (mixture ratio 1: 1 to 1: 100) (Composition A 76); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP85” (mixture ratio 1:10 “Composition A 77);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 86 ”(mixing ratio 1: 1 to 1: 100) (Composition A 78); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP87” (mixture ratio 1:10 to 10: 1) (composition A79); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 88” (mixture ratio 1:10 to 10: 1) (Composition A 80); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP89” (mixture ratio 1 "Composition A81);" Any one of Compounds AA1-BA1-AK2688-BK1287 "and" PP90 "(mixing ratio 1:10 to 10: 1) (Composition A) 82) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP91” (mixture ratio 1:10 to 10: 1) (Composition A 83); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1: 92 to 10: 1” with “PP 92” (composition A 84) (composition A 84); “combination of any one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 93” (Composition ratio 1:10 to 10: 1) (Composition A 85); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP94” (mixture ratio 1:10 to 10: 1) “Composition A86);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP95 ”(mixture ratio 1:10 to 10: 1) (Composition A87);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP96” (mixture ratio 1:10 to 10: 1) (composition A 88); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP97 Combination of (mixing ratio 1: 10 to 10:
1) (Composition A 89); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP98” (mixing ratio 1:10 to 10: 1) (Composition A90); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP99” (mixture ratio 1:10 to 10: 1) (composition A91); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 100 "(mixture ratio 1:10 to 10: 1) (Composition A 92);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP101 "(mixture ratio 1:10 to 10) 10: 1) (Composition A93); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP102” (mixing ratio 1:10 to 10: 1) (Composition A94); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP103” (mixture ratio 1:10 to 10: 1) (composition A95); “any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP104” (mixture ratio 1:10 to 10: 1) (composition A 96); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP105” (mixture “Composition A 97);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP106 ”(mixing ratio 1:10 to 10: 1) (Composition A98); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP107” (mixing ratio 1:10 to 10: 1) (Composition A99); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1:10 to 10: 1” (composition A 100) with “PP108” (composition A 100); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP109” (Composition ratio 1:10 to 10: 1) (Composition A101); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP110” (mixture ratio 1:10 to 10) 1) (Composition A102); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP111” (mixing ratio 1:10 to 10: 1) (Composition A103); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP112” (mixture ratio 1:10 to 10: 1) (composition A104); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 113 "(mixture ratio 1:10 to 10: 1) (Composition A 105);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP114 "(mixture ratio 1:10 to 10) 10: 1) (Composition A106); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP115” (mixing ratio 1:10 to 10: 1) (Composition A107); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP116” (mixture ratio 1:10 to 10: 1) (composition A108); “compound AA1-BA1 to AK2688-BK1287 Combination of “one or more” and “PP117” (mixture ratio 1:10 to 10: 1) (composition A 109); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP118” Mixing ratio 1:10 to 10: 1) (Composition A110); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP119" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP120” (mixing ratio 1:10 to 10: 1) (composition A112); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP121” (mixture ratio 1:10 to 10: 1) (composition A113); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP122” Combination (mixture ratio 1:10 to 10: 1) (Composition A114); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP123” (mixture ratio 1: 0 to 10: 1) (Composition A115); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP124” (mixing ratio 1:10 to 10: 1) (Composition A116); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP125” (mixture ratio 1:10 to 10: 1) (Composition A 117); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP126” (mixture ratio 1:10 to 10: 1) (Composition A 118); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP127” (mixture ratio 1:10 to 10: 1) (Composition A119); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP128” (mixing ratio 1:10 to 10: 1) (Composition A120) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP129" (mixing ratio 1:10 to 10: 1) (Composition A121); "Compounds AA1-BA1 to AK2" Any one of 688-BK1287 and “PP130” (mixture ratio 1:10 to 10: 1) (composition A122); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP131” (Combination ratio 1:10 to 10: 1) (composition A123); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” (mixture ratio 1:10 to 10: 1) (Composition A124); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” (mixing ratio 1:10 to 10: 1) (Composition A125); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP134” (mixture ratio 1:10 to 10: 1) (composition A 126); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP135 "(mixture ratio 1:10 to 10: 1) (Composition A127);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP136 "(Composition A127) Combination ratio 1:10 to 10: 1) (Composition A 128); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 137" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP138” (mixing ratio 1:10 to 10: 1) (composition A130); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP139” (mixture ratio 1:10 to 10: 1) (composition A131); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP140” Combination (mixture ratio 1:10 to 10: 1) (Composition A 132); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP141" (mixture ratio 1:10 to 10: 1) (Composition A133); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP142” (mixing ratio 1:10 to 10: 1) (Composition A134); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP143” (mixture ratio 1:10 to 10: 1) (composition A 135); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP144” (mixture ratio 1:10 to 10: 1) (Composition A 136); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP145” (mixture ratio 1: 10 to 10: 1) (Composition A 137); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 146” (mixing ratio 1:10 to 10: 1) (Composition A 138); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP147” (mixing ratio 1:10 to 10: 1) (Composition A 139); “Any of Compounds AA1-BA1 to AK2688-BK1287 “One” and “PP148” (mixture ratio 1:10 to 10: 1) (composition A 140); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP149” Combination (mixture ratio 1:10 to 10: 1) (Composition A 141); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP150" (mixture ratio 1:10 to 10: 1) (Composition A142); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP151” (mixing ratio 1:10 to 10: 1) (Composition A143); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP152” (mixture ratio 1:10 to 10: 1) (composition A 144); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP153” (Combination ratio 1:10 to 10: 1) (composition A145); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP154” (mixture ratio 1:10 to 10: 1) (Composition A 146); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 155” (mixing ratio 1:10 to 10: 1) (Composition A 147) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” (mixing ratio 1:10 to 10: 1) (Composition A 148); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 157” (mixture ratio 1:10 to 10: 1) (Composition A 149); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP158” (Mixed "Composition A150";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP159" (mixing ratio 1:10 to 10: 1) (Composition A 151) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP160” (mixture ratio 1:10 to 10: 1) (Composition A152); “Compounds AA1-BA1 to AK2688-BK1287 And “PP 161” (mixture ratio 1:10 to 10: 1) (composition A153); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with "PP162" (mixture ratio 1:10 to 10: 1) (Composition A 154); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP163" (mixture ratio 1:10 “Composition A 155);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 164 ”(mixing ratio 1:10 to 10: 1) (Composition A 156); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP165” (mixture ratio 1:10 to 10: 1) (composition A 157); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP166” (mixture ratio 1:10 to 10: 1) (Composition A 158); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP167” (mixture ratio 1 “Composition A159);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP168 ”(mixing ratio 1:10 to 10: 1) “Composition A160);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP169 ”(mixing ratio 1:10 to 10: 1) (Composition A161);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP170” (mixture ratio 1:10 to 10: 1) (composition A162); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP171” Combination (mixture ratio 1:10 to 10: 1) (composition A 163); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP172” (mixture ratio 1:10 to 10: 1 (Composition A 164); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 173” in combination (mixing ratio 1: 10 to 10: 1) (Composition A 165); “Compound AA 1-BA 1 ~ Any one of “AK2688-BK1287” and “PP174” (mixing ratio 1:10 to 10: 1) (Composition A 166); “Compound AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP175” (mixture ratio 1:10 to 10: 1) (Composition A 167); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP176” (mixture ratio 1:10 to 10: 1) (Composition A 168); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP177” (mixing ratio 1:10 to 10: 1) (Composition A169) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP178" (mixing ratio 1:10 to 10: 1) (Composition A170); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and PP179 (mixture ratio 1:10 to 10: 1) (Composition A 171); Combination of any one of Compounds AA1-BA1 to AK2688-BK1287 and PP180 (Composition A 171) Mixing ratio 1:10 to 10: 1) (Composition A 172); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP181" (mixing ratio 1:10 to 10) 0: 1) (Composition A 173); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 182” in combination (mixing ratio 1: 10 to 10: 1) (Composition A 174); Any one of AA1-BA1 to AK2688-BK1287 and “PP183” (mixture ratio 1:10 to 10: 1) (composition A175); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP184” (mixture ratio 1:10 to 10: 1) (Composition A 176); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP185” (mixture ratio 1: 10 to 10: 1) (Composition A 177); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 186” (mixing ratio 1: 10 to 10: 1) (Composition A 178); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP187” (mixing ratio 1:10 to 10: 1) (Composition A 179); “Compounds AA1-BA1 to AK2688-BK1287 Of “one of the two” and “PP188”
Combination (mixture ratio 1:10 to 10: 1) (Composition A 180); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP189” (mixture ratio 1:10 to 10: 1) (Composition A181); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP190” (mixing ratio 1:10 to 10: 1) (Composition A182); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP191” (mixture ratio 1:10 to 10: 1) (composition A183); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP192” (Combination ratio 1:10 to 10: 1) (composition A 184); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP193” (mixture ratio 1:10 to 10: 1) (Composition A185); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP194” (mixing ratio 1:10 to 10: 1) (Composition A186); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP195” (mixture ratio 1:10 to 10: 1) (Composition A 187); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP196” (mixture ratio 1:10 to 10: 1) (Composition A 188); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP197” (mixture ratio 1:10 to 10: 1) (Composition A 189); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP198” (mixing ratio 1:10 to 10: 1) (Composition A190 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP199" (mixing ratio 1:10 to 10: 1) (Composition A191); "Compounds AA1-BA1 to AK2688-BK1287" “Any one” and “PP200” in combination (mixture ratio 1:10 to 10: 1) (composition A 192); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP “Composition A 193) in combination with 201” (composition A 193); “any one of compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 202” (mixture ratio 1: 10 to 10) 10: 1) (Composition A194); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP203” (mixing ratio 1:10 to 10: 1) (Composition A195); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP204” (mixture ratio 1:10 to 10: 1) (composition A 196); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP205” (mixture ratio 1:10 to 10: 1) (Composition A 197); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP206” (mixture ratio 1: 10 to 10: 1) (Composition A198); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP207" (mixing ratio 1:10 to 10: 1) (pair A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP208” (mixing ratio 1:10 to 10: 1) (composition A200); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP209” (mixture ratio 1:10 to 10: 1) (composition A201); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP210” Combination (mixture ratio 1:10 to 10: 1) (Composition A 202); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP211" (mixture ratio 1:10 to 10: 1) (Composition A203); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP212” (mixing ratio 1:10 to 10: 1) (Composition A204); “Compound AA1 to BA1” Any one of AK2688-BK1287 and “PP213” (mixture ratio 1:10 to 10: 1) (composition A205); “any one of compounds AA1-BA1 to AK2688-BK1287” (Composition A 206); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP215” (mixture ratio) 1:10 to 10: 1) (Composition A207); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP216” (mixing ratio 1:10 to 10: 1) (Composition A208 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP217" (mixture ratio 1:10 to 10: 1) (Composition A 209); "Compounds AA1-BA1 to AK2688-BK1287 “Any one” and “PP 218” in combination (mixture ratio 1:10 to 10: 1) (Composition A 210); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP219” Mixing ratio 1:10 to 10: 1) (Composition A 211); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP220" (Mixing ratio 1:10 to 10) 1) (Composition A212); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP221” (mixing ratio 1:10 to 10: 1) (Composition A213); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP222” (mixture ratio 1:10 to 10: 1) (composition A 214); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 223 "(mixture ratio 1:10 to 10: 1) (Composition A 215);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP224 "(mixture ratio 1:10 to 10) 10: 1) (Composition A216); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP225” (mixing ratio 1:10 to 10: 1) (Composition A217); “Compound Any one of AA1-BA1-AK2688-BK1287 and “PP226” (mixture ratio 1:10 to 10: 1) (composition A 218); “compound AA1-BA1 to AK2688-BK1287 Combination of “any one” and “PP227” (mixture ratio 1:10 to 10: 1) (composition A 219); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP228” Mixing ratio 1:10 to 10: 1) (Composition A 220); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 229" (Mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP230” (mixing ratio 1:10 to 10: 1) (composition A222); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP231” (mixture ratio 1:10 to 10: 1) (composition A 223); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP232” Combination (mixture ratio 1:10 to 10: 1) (Composition A 224); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP233” (mixture ratio 1: 0 to 10: 1) (Composition A 225); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP234” (mixing ratio 1:10 to 10: 1) (Composition A 226); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP235” (mixture ratio 1:10 to 10: 1) (Composition A 227); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP236” (mixture ratio 1:10 to 10: 1) (Composition A 228); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP237” (mixture ratio 1:10 to 10: 1) (Composition A 229); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP238” (mixing ratio 1:10 to 10: 1) (Composition A230 A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 239” (mixture ratio 1:10 to 10: 1) (composition A 231); “compound AA1 to BA1 to AK2”; Any one of 688-BK1287 and “PP240” (mixture ratio 1:10 to 10: 1) (composition A 232); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP241” (Combination ratio 1:10 to 10: 1) (composition A233); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP242” (mixture ratio 1:10 to 10: 1) (Composition A234); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP243” (mixing ratio 1:10 to 10: 1) (Composition A235); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP244” (mixture ratio 1:10 to 10: 1) (composition A 236); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP245 "(mixture ratio 1:10 to 10: 1) (Composition A 237);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP246 " Composition ratio 1:10 to 10: 1) (Composition A 238); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 247” (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP248” (mixing ratio 1:10 to 10: 1) (composition A240); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP249” (mixture ratio 1:10 to 10: 1) (composition A 241); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP250” Combination (mixture ratio 1:10 to 10: 1) (Composition A 242); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 251" (mixture ratio 1:10 to 10: 1) (Composition A243); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP252” (mixing ratio 1:10 to 10: 1) (Composition A244); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP253” (mixture ratio 1:10 to 10: 1) (composition A245); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP254” (mixture ratio 1:10 to 10: 1) (Composition A 246); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP255” (mixture ratio 1: 10 to 10: 1) (Composition A 247); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 256” (mixing ratio 1: 10 to 10: 1) (Composition A 248); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP257” (mixing ratio 1:10 to 10: 1) (Composition A 249); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP258” (mixture ratio 1:10 to 10: 1) (composition A 250); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP259” Combination (mixture ratio 1:10 to 10: 1) (Composition A 251); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP260" (mixture ratio 1:10 to 10: 1) (Composition A 252); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP261” (mixture ratio 1:10 to 10: 1) (Composition A253); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP262” (mixture ratio 1:10 to 10: 1) (composition A 254); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP263” Combination (mixture ratio 1:10 to 10: 1) (composition A255); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP264” (mixture ratio 1:10 to 10: 1) (Composition A 256); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 266” (mixing ratio 1:10 to 10: 1) (Composition A 257) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP266-1-1" (mixing ratio 1:10 to 10: 1) (Composition A 258); "Compound AA1 -BA1 to AK2688 Any one of “-BK1287” and “PP266-1-2” (mixture ratio 1:10 to 10: 1) (composition A 259); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP266-2” (mixture ratio 1:10 to 10: 1) (Composition A 260); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP266-2-1” (Mixing ratio 1:10 to 10: 1) (Composition A 261); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP266-3” (Mixing ratio 1:10 to 10: 1 “Composition A262);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP 266-3-1 ”(mixing ratio 1:10 to 10: 1) (Composition A263); Any of the compounds AA1-BA1 to AK2688-BK1287 “Composition” (composition A 264); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 266-4”. (Composition A 265); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 266-4-1” (mixture ratio 1) “Composition A 266);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP 266-5 ”(mixing ratio 1:10 to 10: 1) (Composition A267) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP266-6” (mixture ratio 1:10 to 10: 1) (Composition A 268); “Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP266-7” (mixture ratio 1:10 to 10: 1) (composition A269); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP266 Combination with “-8” Total ratio 1:10 to 10: 1) (
Composition A270); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP266-9” (mixing ratio 1:10 to 10: 1) (Composition A271); “Compound AA1 to BA1 -Any one of AK2688-BK1287 'and' PP266-10 '(mixture ratio 1:10 to 10: 1) (Composition A 272); “any one of Compounds AA1-BA1 to AK2688-BK1287” Combination with “PP266-11” (mixture ratio 1:10 to 10: 1) (Composition A 273); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP266-12” “Composition A 274);“ Any one of the compounds AA1-BA1 to AK2688-BK1287 ”and“ PP266-13 ”(mixing ratio 1:10 to 10: 1) (composition A 274) Composition A275); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP266-14” (mixing ratio 1:10 to 10: 1) (Composition A276); “Compound AA1 to BA1 ~ AK2688-BK128 “Any one of 7” and “PP 266-14-1” (mixture ratio 1:10 to 10: 1) (composition A 277); “any one of compounds AA1-BA1 to AK2688-BK1287” and “composition A277” Combination with PP 266-15 "(mixture ratio 1:10 to 10: 1) (Composition A 278);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP266-16 "(mixture ratio 1:10 to 10: 1) (Composition A 279); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 267” (mixing ratio 1:10 to 10: 1) (Composition A 280 A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP267-1” (mixing ratio 1:10 to 10: 1) (composition A 281); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP268” (mixture ratio 1:10 to 10: 1) (composition A282); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP269” combination (Composition ratio 1:10 to 10: 1) (Composition A 283); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP270” (mixture ratio 1:10 to 10: 1) (Composition A 283) “Composition A284);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP271 ”(mixing ratio 1:10 to 10: 1) (Composition A285);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP272” (mixture ratio 1:10 to 10: 1) (composition A 286); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP273” Combination (mixture ratio 1:10 to 10: 1) (composition A 287); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP274” (mixture ratio 1:10 to 10: 1 (Composition A 288); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP 275” (mixing ratio 1:10 to 10: 1) (Composition A 289); Any one of Compound AA1-BA1 to AK2688-BK1287 and “PP276” (mixing ratio 1:10 to 10: 1) (Composition A 290); “Compound AA1 to BA1 to AK2688-BK1287 Combination of “One” and “PP 277” (mixture ratio 1:10 to 10: 1) (Composition A 291); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP277-1” Mixing ratio 1:10 to 10: 1) (Composition A292); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 278" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP279” (mixing ratio 1:10 to 10: 1) (composition A294); “compound AA1 to BA1 to AK2688” “Any one of BK1287” and “PP280” in combination (mixture ratio 1:10 to 10: 1) (Composition A 295); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP281 (Combination ratio 1:10 to 10: 1) (composition A 296); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP282” (mixture ratio 1:10 to 10: 1) (Composition A 297); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 283” (mixture ratio 1: 10 to 10: 1) (Composition A 298); Any one of BA1 to AK2688-BK1287 and “PP284” (mixture ratio 1:10 to 10: 1) (composition A 299); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 285 "(mixture ratio 1:10 to 10: 1) (Composition A 300);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP 286 "(mixture ratio 1:10 to 10) 10: 1) (Composition A301); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP287” (mixing ratio 1:10 to 10: 1) (Composition A302); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP288” (mixing ratio 1:10 to 10: 1) (Composition A303); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the above and “PP 289” (mixture ratio 1:10 to 10: 1) (Composition A 304); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP290” (Composition ratio 1:10 to 10: 1) (Composition A 305); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP 291” (mixture ratio 1:10 to 10: 1) “Composition A306);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP292 ”(mixing ratio 1:10 to 10: 1) (Composition A307);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP293” (mixture ratio 1:10 to 10: 1) (composition A 308); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP294” (mixture ratio 1:10 to 10: 1) (Composition A 309); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP295” (mixture ratio 1 “Composition A310);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP296 ”(mixing ratio 1:10 to 10: 1) (Composition A311) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP297” (mixing ratio 1:10 to 10: 1) (Composition A312); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 298” (mixture ratio 1:10 to 10: 1) (Composition A 313); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 299” "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP300" (mixing ratio 1:10 to 10: 1 to 10: 1) (Composition A 314); (Composition A 315); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP301” (mixing ratio 1:10 to 10: 1) (Composition A316); “Compound AA1 to BA1” ~ Any one of AK2688-BK1287 "and" PP302 "(mixture ratio 1:10 to 10: 1) (Composition A 317);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP303 (Mixture ratio 1:10 to 10: 1) (Composition A 318); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP304” (mixture ratio 1:10 to 10) "Composition A319";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP305" (mixing ratio 1:10 to 10: 1) (Composition A320); "Compound AA1 Any one of “-BA1 to AK2688-BK1287” and “PP306” (mixture ratio 1:10 to 10: 1) (Composition A 321); “Attachment of Compound AA1-BA1 to AK2688-BK1287 Combination of “one piece” and “PP307” (mixture ratio 1:10 to 10: 1) (composition A 322); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP309” (composition A322) Mixing ratio 1:10 to 10: 1) (Composition A 323); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP310" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP312” (mixing ratio 1:10 to 10: 1) (composition A 325); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP313” (mixture ratio 1:10 to 10: 1) (composition A326); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP314” Combination (mixture ratio 1:10 to 10: 1) (Composition A 327); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP315" (mixture ratio 1: 1 “Composition A 328);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 316 ”(mixing ratio 1: 10 to 10: 1) (Composition A 329); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP318” (mixture ratio 1:10 to 10: 1) (composition A330); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 319” (mixture ratio 1:10 to 10: 1) (Composition A 331); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP320” (mixture ratio 1 "Composition A332";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP 321" (mixing ratio 1:10 to 10: 1) (Composition A333) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP322” (mixture ratio 1:10 to 10: 1) (Composition A334); “Compound AA1 to BA1 to AK2688- A combination of “one of BK1287” and “PP323” (mixture ratio 1:10 to 10: 1) (composition A 335); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP324” Combination (mixture ratio 1:10 to 10: 1) (Composition A 336); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 325" (mixture ratio 1:10 to 10: 1) (Composition A 337); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 326” (mixing ratio 1:10 to 10: 1) (Composition A 338); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP327” (mixture ratio 1:10 to 10: 1) (composition A 339); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP328” Combination (mixture ratio 1:10 to 10: 1) (composition A340); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP329” "Composition A341";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP330" (mixing ratio 1:10 to 10: 1) (Composition A 342); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP332” (mixture ratio 1:10 to 10: 1) (Composition A343); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following “composition of 1 to 10: 1” with “PP 333” (composition A 344) (composition A 344); “a combination of any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP334” (Composition ratio 1:10 to 10: 1) (Composition A 345); “Any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 335” (mixture ratio 1:10 to 10: 1) (Composition A 345) “Composition A346);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP336 ”(mixing ratio 1:10 to 10: 1) (Composition A347);“ Compound AA Any one of 1-BA1 to AK2688-BK1287 and “PP 337” (mixture ratio 1:10 to 10: 1) (composition A 348); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP338” (mixture ratio 1:10 to 10: 1) (Composition A 349); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP339” (mixture ratio 1: 10 to 10: 1) (Composition A 350); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 340” (mixing ratio 1: 10 to 10: 1) (Composition A 351); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP341” (mixture ratio 1:10 to 10: 1) (Composition A 352); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP342” (mixture ratio 1:10 to 10: 1) (composition A 353); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP343” Combination (mixture ratio 1:10 to 10: 1) (Composition A 354); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP344” (mixture ratio 1:10 to 10: 1) (Composition A355); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP345” (mixing ratio 1:10 to 10: 1) (Composition A356); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP346” (mixture ratio 1:10 to 10: 1) (composition A 357); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP347” (Combination ratio 1:10 to 10: 1) (Composition A 358); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP348” (mixture ratio 1:10 to 10: 1) (Composition A 359); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 349” (mixing ratio 1:10 to 10: 1) (Composition A 360) "Compound AA1-BA1~AK2688-B
A combination of “one of K1287” and “PP350” (mixture ratio 1:10 to 10: 1) (composition A 361); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP351” Combination (mixture ratio 1:10 to 10: 1) (Composition A 362); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 352" (mixture ratio 1:10 to 10: 1) (Composition A 363); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 353” (mixing ratio 1:10 to 10: 1) (Composition A 364); “Compound AA 1-BA1 “Any one of AK2688-BK1287” and “PP354” (mixture ratio 1:10 to 10: 1) (composition A 365); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP355” Combination (mixture ratio 1:10 to 10: 1) (composition A 366); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 356” (mixture "Composition A367);" Any one of Compounds AA1-BA1-AK2688-BK1287 "and" PP 357 "(mixing ratio 1:10 to 10: 1) (Composition A368); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP358” (mixture ratio 1:10 to 10: 1) (Composition A369); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following “composition of 1 to 10: 1” with “PP 359” (composition A 370) (composition A 370); “one of the compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 361” (Composition ratio 1:10 to 10: 1) (Composition A 371); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP362” (mixture ratio 1:10 to 10: 1) Composition A372); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP363” (mixture ratio 1:10 to 10: 1) (Composition A 373); “Compound AA1 -Any one of “BA1 to AK2688-BK1287” and “PP364” (mixture ratio 1:10 to 10: 1) (composition A 374); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP365” (mixture ratio 1:10 to 10: 1) (Composition A 375); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP366” (mixture ratio 1:10 "Composition A 376";"Any one of Compounds AA1-BA 1 to AK 2688-BK 1287" and "PP 367" (mixing ratio 1:10 to 10: 1) (Composition A 377); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP368” (mixture ratio 1:10 to 10: 1) (composition A378); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 369” (mixture ratio 1:10 to 10: 1) (Composition A 379); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370” Combination (mixture ratio 1:10 to 10: 1) (Composition A 380); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP371” (mixture ratio 1:10 to 10: 1) (Composition A 381); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 372” (mixing ratio 1:10 to 10: 1) (Composition A 382); “Compound AA 1-BA 1 “Any one of AK2688-BK1287” and “PP 373” (mixture ratio 1:10 to 10: 1) (Composition A 383); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP376” (Combination ratio 1:10 to 10: 1) (composition A 384); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 377” (mixture ratio 1:10 to 10: 1) (Composition A 385); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP378” (mixing ratio 1:10 to 10: 1) (Composition A 386); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP379” (mixing ratio 1:10 to 10: 1) (Composition A 387); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP380” (mixture ratio 1:10 to 10: 1) (Composition A 388); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP383” (mixture ratio 1:10 to 10: 1) (Composition A 389); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP384” (mixing ratio 1:10 to 10: 1) (Composition A 390) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP385" (mixture ratio 1:10 to 10: 1) (Composition A391); "Compounds AA1-BA1 to AK2688-BK1287" “Any one” and “PP 386” in combination (mixture ratio 1:10 to 10: 1) (composition A 392); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP “Composition A393”; “Any one of compounds AA1-BA1 to AK2688-BK1287” and “PP390” (mixture ratio 1:10 to 10) 10: 1) (Composition A394); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP391” (mixing ratio 1:10 to 10: 1) (Composition A395); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP392” (mixture ratio 1:10 to 10: 1) (composition A 396); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP393” (mixture ratio 1:10 to 10: 1) (Composition A397); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394” (mixture ratio 1: 10 to 10: 1) (Composition A 398); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 395” (mixing ratio 1:10 to 10: 1) (combination A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP396” (mixing ratio 1:10 to 10: 1) (composition A400); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP397” (mixture ratio 1:10 to 10: 1) (composition A 401); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP398” Combination (mixture ratio 1:10 to 10: 1) (Composition A 402); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP399" (mixture ratio 1:10 to 10: 1) (Composition A403); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP400” (mixing ratio 1:10 to 10: 1) (Composition A404); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP401” (mixture ratio 1:10 to 10: 1) (Composition A 405); “Compound AA 1-BA 1 to AK 2688-BK 1287” (Composition A 406); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP403” (mixture ratio) 1: 10 to 10: 1) (Composition A 407); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 404” (mixing ratio 1: 10 to 10: 1) (Composition A 408 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP405" (mixing ratio 1:10 to 10: 1) (Composition A409); "Compounds AA1-BA1 to AK2688-BK1287" “Any one” and “PP406” in combination (mixture ratio 1:10 to 10: 1) (Composition A 410); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” Mixing ratio 1:10 to 10: 1) (Composition A411); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP408" (mixing ratio 1:10 to 10) 1) (Composition A412); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP409” (mixing ratio 1:10 to 10: 1) (Composition A413); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP410” (mixture ratio 1:10 to 10: 1) (composition A 414); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 411 "(mixture ratio 1: 10 to 10: 1) (Composition A 415);" Any one of Compounds AA1-BA 1 to AK 2688-BK 1287 "and" PP 412 "(mixture ratio 1: 10 to 10 10: 1) (Composition A 416); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 413” in combination (mixing ratio 1:10 to 10: 1) (Composition A 417); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP 414” (mixture ratio 1:10 to 10: 1) (composition A418); “compound AA1-BA1 to AK2688-BK1287 Combination of “one or more” and “PP 415” (mixture ratio 1:10 to 10: 1) (composition A 419); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP428” Mixing ratio 1:10 to 10: 1) (Composition A420); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 429" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP430” (mixing ratio 1:10 to 10: 1) (composition A 422); “compound AA1 to BA1 to AK2688” “Any one of BK1287” and “PP 431” (mixture ratio 1:10 to 10: 1) (Composition A 423); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP432” Combination (mixture ratio 1:10 to 10: 1) (Composition A 424); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 433” (mixture ratio 1: 0 to 10: 1) (Composition A 425); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 434” (mixing ratio 1: 10 to 10: 1) (Composition A 426); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP435” (mixture ratio 1:10 to 10: 1) (Composition A 427); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP436” (mixture ratio 1:10 to 10: 1) (Composition A 428); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP437” (mixture ratio 1:10 to 10: 1) (Composition A 429); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP438” (mixing ratio 1:10 to 10: 1) (Composition A 430) A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP439” (mixing ratio 1:10 to 10: 1) (composition A 431); “compound AA1 to BA1 to AK2” Any one of 688-BK1287 and “PP440” (mixture ratio 1:10 to 10: 1) (composition A432); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP441” (Combination ratio 1:10 to 10: 1) (composition A 433); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 442” (mixture ratio 1:10 to 10: 1) (Composition A 434); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP 443” (mixing ratio 1:10 to 10: 1) (Composition A 435); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP444” (mixture ratio 1:10 to 10: 1) (composition A 436); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 445 "(mixture ratio 1: 10 to 10: 1) (Composition A 437);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP 446 " Combination ratio 1:10 to 10: 1) (Composition A 438); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP448" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP449” (mixing ratio 1:10 to 10: 1) (composition A440); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP450” (mixture ratio 1:10 to 10: 1) (composition A441); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP451” Combination (mixture ratio 1:10 to 10: 1) (Composition A 442); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP452" (mixture ratio 1:10 to 10: 1) (Composition A 443); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 453” (mixing ratio 1:10 to 10: 1) (Composition A 444); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP454” (mixture ratio 1:10 to 10: 1) (composition A445); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP455” (mixture ratio 1:10 to 10: 1) (composition A446); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP456” (mixture ratio 1: 10 to 10: 1) (Composition A 447); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 457” (mixing ratio 1:10 to 10: 1) (Composition A448); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP458” (mixing ratio 1:10 to 10: 1) (Composition A 449); “Any of Compounds AA1-BA1 to AK2688-BK1287 “One” and “PP 459” (mixture ratio 1:10 to 10: 1) (composition A 450); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP460” Combining (mixing ratio 1: 10 to 10: 1)
(Composition A 451); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 461” (mixing ratio 1:10 to 10: 1) (Composition A452); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP462” in combination (mixture ratio 1:10 to 10: 1) (composition A 453); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP463” (Combination ratio 1:10 to 10: 1) (composition A454); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP464” (mixture ratio 1:10 to 10: 1) (Composition A455); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP465” (mixing ratio 1:10 to 10: 1) (Composition A456); “Compound AA1− A combination of “one of BA1 to AK2688-BK1287” and “PP466” (mixture ratio 1:10 to 10: 1) (composition A 457); “any of compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 467” (mixture ratio 1:10 to 10: 1) (Composition A 458); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP468” (mixture ratio 1:10 to 10: 1) (Composition A 459); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 469” (mixing ratio 1:10 to 10: 1) (Composition A 460 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP470" (mixture ratio 1:10 to 10: 1) (Composition A 461); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and PP 471 (mixture ratio 1:10 to 10: 1) (Composition A 462); Combination of any one of Compounds AA1-BA1 to AK2688-BK1287 and PP472 ” Mixing ratio 1:10 to 10: 1) (Composition A463); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 473" (mixing ratio 1:10 to 10) 10: 1) (Composition A 464); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 474” (mixing ratio 1:10 to 10: 1) (Composition A 465); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP475” (mixture ratio 1:10 to 10: 1) (composition A 466); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 476” (mixture ratio 1:10 to 10: 1) (Composition A 467); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 477” (mixture ratio 1: 10 to 10: 1) (Composition A 468); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 478” (mixing ratio 1:10 to 10: 1) (Composition A 469); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP479” (mixing ratio 1:10 to 10: 1) (Composition A 470); “Compounds AA1-BA1 to AK2688-BK12 A combination of “any one of 87” and “PP 480” (mixture ratio 1:10 to 10: 1) (composition A 471); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP481” Combination (mixture ratio 1:10 to 10: 1) (Composition A 472); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP482" (mixture ratio 1:10 to 10: 1) (Composition A 473); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP483” in combination (mixing ratio 1:10 to 10: 1) (Composition A 474); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP484” in combination (mixture ratio 1:10 to 10: 1) (Composition A 475); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP485” (Combination ratio 1:10 to 10: 1) (composition A 476); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 486” (mixing ratio 1:10 to 10: 1) (Composition A 477); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP487” (mixing ratio 1:10 to 10: 1) (Composition A 478) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP488" (mixture ratio 1:10 to 10: 1) (Composition A 479); "Compounds AA1-BA1 to AK2688-BK1287 “Any one” and “PP 489” (mixture ratio 1:10 to 10: 1) (Composition A 480); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP490” (Composition A 480) Mixing ratio 1:10 to 10: 1) (Composition A 481); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 491" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 492” (mixing ratio 1:10 to 10: 1) (composition A483); “compound AA1-BA”; Any one of 1 to AK2688-BK1287 "and" PP493 "(mixture ratio 1:10 to 10: 1) (composition A 484);" any one of compounds AA1-BA1 to AK2688-BK1287 "and" composition “Composition A 485” in combination with “PP 494” (mixture ratio 1:10 to 10: 1); “Any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 495” (mixture ratio 1:10 to 10) 10: 1) (Composition A 486); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 496” in combination (mixing ratio 1:10 to 10: 1) (Composition A487); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP 497” (mixture ratio 1:10 to 10: 1) (composition A 488); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 498” (mixture ratio 1:10 to 10: 1) (composition A 489); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP499” “Composition ratio 1:10 to 10: 1” (composition A 490); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP500” (mixture ratio 1:10 to 10: 1) (Composition A491); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP501” (mixing ratio 1:10 to 10: 1) (Composition A492); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP502” (mixture ratio 1:10 to 10: 1) (composition A493); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP503” (Combination ratio 1:10 to 10: 1) (composition A494); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP504” (mixture ratio 1:10 to 10: 1) (Composition A 495); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 505” (mixing ratio 1:10 to 10: 1) (Composition A 496); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP506” (mixture ratio 1:10 to 10: 1) (composition A 497); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 507” (mixture ratio 1:10 to 10: 1) (Composition A 498); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP508” (mixture ratio 1 "Composition A 499";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP 509" (mixing ratio 1:10 to 10: 1) (Composition A 500) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP510” (mixing ratio 1:10 to 10: 1) (Composition A 501); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP511” (mixture ratio 1:10 to 10: 1) (composition A 502); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP512 (Mixture ratio 1:10 to 10: 1) (Composition A 503); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP513” (mixture ratio 1:10 to 10) "Composition A504";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 514" in combination (mixing ratio 1:10 to 10: 1) (Composition A505); "Compound AAl Any one of “BA1 to AK2688-BK1287” and “PP515” (mixture ratio 1:10 to 10: 1) (composition A506); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP516” (mixture ratio 1:10 to 10: 1) (Composition A 507); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP517” (mixture ratio 1:10 ~ 10: 1) (Composition A 508); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 518" (mixing ratio 1:10 to 10: 1) (Composition A 509) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP519” (mixing ratio 1:10 to 10: 1) (Composition A510); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1:50 to 10: 1” (composition A 511) with “PP520” (composition A 511); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP521” (Composition ratio 1:10 to 10: 1) (Composition A 512); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP524” (mixture ratio 1:10 to 10: 1) “Composition A513);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP525 ”(mixing ratio 1:10 to 10: 1) (Composition A514);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP526” (mixture ratio 1:10 to 10: 1) (composition A515); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP 527” (mixture ratio 1:10 to 10: 1) (Composition A 516); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP528” (mixture ratio 1 “Composition A517);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP529 ”(mixing ratio 1:10 to 10: 1) (Composition A518) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP530” (mixing ratio 1:10 to 10: 1) (Composition A519); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 530-1” (mixture ratio 1:10 to 10: 1) (Composition A 520); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP531” (Composition ratio 1:10 to 10: 1) (Composition A 521); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP 531-1” (mixture ratio 1:10 to 10) 1) (Composition A 522); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 532” in combination (mixture ratio 1: 10 to 10: 1) (Composition A 523); Any one of “-BA1 to AK2688-BK1287” and “PP533” (mixing ratio 1:10 to 10: 1) (composition A 524); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP533-1” (mixture ratio 1:10 to 10: 1) (Composition A 525); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP533-2” "Composition A526";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP 533-3" (mixing ratio 1:10 to 10: 1) (Composition A 526) Composition A527); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 533-4” (mixing ratio 1:10 to 10: 1) (Composition A 528); “Compound AA1 to BA1 ~ AK 2688-BK “One of 1287” and “PP 533-5” in combination (mixture ratio 1:10 to 10: 1) (composition A529); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP533- 6) (mixture ratio 1:10 to 10: 1) (Composition A 530); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP533-7” (mixture ratio 1: 10 to 10: 1) (Composition A 531); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 533-8” (mixing ratio 1: 10 to 10: 1) (Composition A 532) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP533-9" (mixing ratio 1:10 to 10: 1) (Composition A533); "Compounds AA1-BA1 to AK2688-" “Any one of BK1287” and “PP533-10” in combination (mixture ratio 1:10 to 10: 1) (Composition A 534); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP534” Union with “Composition ratio 1:10 to 10: 1” (composition A 535); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP 535” (mixture ratio 1:10 to 10: 1) (Composition A536); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP537” (mixing ratio 1:10 to 10: 1) (Composition A537); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP538” (mixture ratio 1:10 to 10: 1) (composition A 538); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP539” (Combination ratio 1:10 to 10: 1) (composition A 539); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 541” (mixture ratio 1:10 to 10: 1) (Composition A 540); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 542” (mixing ratio 1:10 to 10: 1) (Composition A 541); Compounds AA1-BA1 to AK2688-BK1287
Any one of the following “composition of 1 to 10: 1” with “PP 543” (composition A 542) (composition A 542); “one of the compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 544” (Composition ratio 1:10 to 10: 1) (Composition A 543); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP545” (Mixing ratio 1:10 to 10: 1) (Composition A 543) “Composition A 544);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP545-1 ”(mixing ratio 1:10 to 10: 1) (Composition A545);“ Compound AA1 to BA1 ~ Any one of AK2688-BK1287 'and' PP546 '(mixture ratio 1:10 to 10: 1) (composition A 546);' any one of compounds AA1-BA1 to AK2688-BK1287 'and' PP547 (Mixture ratio 1:10 to 10: 1) (composition A547); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP548” (mixture ratio 1:10 to 10: 1) (Composition A 548); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP548-1” (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP551” (mixture ratio 1:10 to 10: 1) (composition A550); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP552” (mixture ratio 1:10 to 10: 1) (composition A 551); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP553” Combination (mixture ratio 1:10 to 10: 1) (Composition A 552); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP554" (mixture ratio 1:10 to 10: 1) (Composition A553); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP555” (mixing ratio 1:10 to 10: 1) (Composition A 554); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP 556” (mixture ratio 1:10 to 10: 1) (composition A 555); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 557 "(mixture ratio 1:10 to 10: 1) (Composition A 556);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP558 "(mixture ratio 1:10 to 10) 10: 1) (Composition A 557); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP559” (mixing ratio 1:10 to 10: 1) (Composition A 558); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP560” (mixture ratio 1:10 to 10: 1) (composition A559); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 562” (mixture ratio 1:10 to 10: 1) (Composition A 560); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP563” (Composition ratio 1:10 to 10: 1) (composition A 561); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 564” (mixture ratio 1:10 to 10: 1) (Composition A 562); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 565” (mixture ratio 1: 10 to 10: 1) (Composition A 563); “Compound AA 1-BA 1 “Any one of AK2688-BK1287” and “PP566” (mixture ratio 1:10 to 10: 1) (composition A 564); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP567” (Combination ratio 1:10 to 10: 1) (composition A 565); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP568” (mixture ratio 1:10 to 10: 1) (Composition A 566); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP569” (mixing ratio 1:10 to 10: 1) (Composition A 567); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP570” (mixture ratio 1:10 to 10: 1) (composition A 568); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 571” (mixture ratio 1:10 to 10: 1) (Composition A 569); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP572” (mixture ratio 1 “Composition A570);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP 573 ”(mixing ratio 1:10 to 10: 1) (Composition A 571) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP574” (mixture ratio 1:10 to 10: 1) (Composition A572); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP575” (mixture ratio 1:10 to 10: 1) (composition A 573); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP5 76 "(mixture ratio 1:10 to 10: 1) (Composition A 574);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP577 "(mixture ratio 1:10 to 10) 10: 1) (Composition A 575); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 578” (mixing ratio 1: 10 to 10: 1) (Composition A 576); Any one of AA1-BA1 to AK2688-BK1287 and “PP579” (mixture ratio 1:10 to 10: 1) (composition A577); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP580” (mixture ratio 1:10 to 10: 1) (Composition A 578); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP581” (mixture ratio 1: 10 to 10: 1) (Composition A 579); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP582” (mixing ratio 1:10 to 10: 1) (combination A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP583” (mixture ratio 1:10 to 10: 1) (composition A581); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP584” (mixture ratio 1:10 to 10: 1) (composition A 582); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP585” Combination (mixture ratio 1:10 to 10: 1) (Composition A583); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP586" (mixture ratio 1:10 to 10: 1) (Composition A 584); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 587” (mixing ratio 1:10 to 10: 1) (Composition A585); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP 588” (mixture ratio 1:10 to 10: 1) (Composition A 586); “Compounds AA1-BA1 to AK2688-BK1287” (Composition A 587); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 590” (mixture ratio) 1:10 to 10: 1) (Composition A 588); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 591” (mixing ratio 1:10 to 10: 1) (Composition A 589) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP592" (mixture ratio 1:10 to 10: 1) (Composition A 590); "Compound AA1 -BA1 to AK2688-BK1287 Combination of any one of them and “PP593” (mixture ratio 1:10 to 10: 1) (Composition A591); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP594” (Composition A591) Mixing ratio 1:10 to 10: 1) (Composition A 592); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 595" (Mixing ratio 1:10 to 10) 1) (Composition A593); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP596” (mixing ratio 1:10 to 10: 1) (Composition A 594); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP 597” (mixture ratio 1:10 to 10: 1) (composition A 595); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition A 596” in combination with “PP 598” (composition A 596); “Any one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 600” (mixture ratio 1: 10 to 10) 10: 1) (Composition A 597); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP601” in combination (mixing ratio 1:10 to 10: 1) (Composition A 598); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP602” (mixture ratio 1:10 to 10: 1) (composition A599); “compound AA1-BA1 to AK2688-BK1287 Combination of “any one” and “PP603” (mixture ratio 1:10 to 10: 1) (composition A 600); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP604” Mixing ratio 1:10 to 10: 1) (Composition A 601); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 605" (Mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP606” (mixing ratio 1:10 to 10: 1) (composition A 603); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP607” (mixture ratio 1:10 to 10: 1) (composition A 604); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP608” Combination (mixture ratio 1:10 to 10: 1) (Composition A 605); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP609” (mixture ratio 1: 0 to 10: 1) (Composition A 606); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 610” (mixing ratio 1:10 to 10: 1) (Composition A 607); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 611” (mixture ratio 1:10 to 10: 1) (Composition A 608); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 612” (mixture ratio 1:10 to 10: 1) (Composition A 609); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP613” (mixture ratio 1:10 to 10: 1) (Composition A610); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 614” (mixing ratio 1:10 to 10: 1) (Composition A 611) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 615" (mixture ratio 1:10 to 10: 1) (Composition A 612); "Compounds AA1-BA1 to AK26" “Any one of 88-BK1287” and “PP 616” (mixture ratio 1:10 to 10: 1) (composition A 613); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP617” (Combination ratio 1:10 to 10: 1) (composition A 614); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 618” (mixture ratio 1:10 to 10: 1) (Composition A 615); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP 620” (mixing ratio 1:10 to 10: 1) (Composition A 616); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP 621” (mixture ratio 1:10 to 10: 1) (composition A 617); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 622 (mixture ratio 1: 10 to 10: 1) (Composition A 618); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 623” (Composition A 618) Combination ratio 1:10 to 10: 1) (Composition A 619); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 624" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP625” (mixture ratio 1:10 to 10: 1) (composition A621); “compound AA1-BA1 to AK2688- A combination of “one of BK1287” and “PP626” (mixture ratio 1:10 to 10: 1) (composition A 622); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP627” Combination (mixture ratio 1:10 to 10: 1) (Composition A 623); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 628" (mixture ratio 1:10 to 10: 1) (Composition A 624); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP629” in combination (mixing ratio 1:10 to 10: 1) (Composition A 625); Any one of AA1-BA1 to AK2688-BK1287 and “PP630” (mixture ratio 1:10 to 10: 1) (composition A 626); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 631” (mixture ratio 1:10 to 10: 1) (Composition A 627); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 632” (mixture ratio 1: 10 to 10: 1) (Composition A 628); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 633” (mixing ratio 1:10 to 10: 1) (Composition A629); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP634” (mixing ratio 1:10 to 10: 1) (Composition A 630); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP635” (mixture ratio 1:10 to 10: 1) (composition A 631); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP636” Combining (mixing ratio 1: 10 to 10: 1)
(Composition A 632); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP637” (mixing ratio 1:10 to 10: 1) (Composition A633); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP638” (mixture ratio 1:10 to 10: 1) (composition A 634); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP639” (Combination ratio 1:10 to 10: 1) (Composition A 635); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP 640” (mixture ratio 1:10 to 10: 1) (Composition A 636); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 641” (mixing ratio 1:10 to 10: 1) (Composition A 637); “Compound AA1− A combination of “one of BA1 to AK2688-BK1287” and “PP 642” (mixing ratio 1:10 to 10: 1) (composition A 638); “any of compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP643” (mixture ratio 1:10 to 10: 1) (Composition A 639); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP644” (mixture ratio 1:10 to 10: 1) (Composition A 640); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 645” (mixing ratio 1:10 to 10: 1) (Composition A 641) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP646" (mixing ratio 1:10 to 10: 1) (Composition A 642); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and “PP 647” (mixture ratio 1:10 to 10: 1) (Composition A 643); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP648” Mixing ratio 1:10 to 10: 1) (Composition A 644); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP650" (mixing ratio 1:10 to 10) 10: 1) (Composition A645); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 651” (mixing ratio 1:10 to 10: 1) (Composition A 646); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP652” (mixture ratio 1:10 to 10: 1) (composition A 647); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP653” (mixture ratio 1:10 to 10: 1) (Composition A 648); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP654” (mixture ratio 1: 10 to 10: 1) (Composition A 649); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP655” (mixing ratio 1:10 to 10: 1) (Composition A 650); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP656” (mixing ratio 1:10 to 10: 1) (Composition A 651); “Compounds AA1-BA1 to AK2688-BK12 Any one of 87 and a combination of “PP657” (mixture ratio 1:10 to 10: 1) (composition A 652); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP658” Combination (mixture ratio 1:10 to 10: 1) (Composition A653); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP659" (mixture ratio 1:10 to 10: 1) (Composition A654): “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP660” (mixing ratio 1:10 to 10: 1) (Composition A655); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP 661” (mixture ratio 1:10 to 10: 1) (composition A 656); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP662” (Combination ratio 1:10 to 10: 1) (composition A 657); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP663” (mixture ratio 1:10 to 10: 1) (Composition A 658); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP664” (mixing ratio 1:10 to 10: 1) (Composition A659) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP665" (mixing ratio 1:10 to 10: 1) (Composition A660); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and “PP666” (mixture ratio 1:10 to 10: 1) (Composition A 661); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP667” Mixing ratio 1:10 to 10: 1) (Composition A 662); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP668" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP669” (mixture ratio 1:10 to 10: 1) (composition A664); “compound AA1-BA”; “Any one of 1 to AK 2688-BK 1287” and “PP 670” (mixture ratio 1:10 to 10: 1) (composition A 665); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 671 "(mixture ratio 1: 10 to 10: 1) (Composition A 666);" Any one of Compounds AA1-BA 1 to AK 2688-BK 1287 "and" PP 672 "(mixture ratio 1: 10 to 10 10: 1) (Composition A 667); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 673” in combination (mixing ratio 1:10 to 10: 1) (Composition A 668); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP 674” (mixture ratio 1:10 to 10: 1) (Composition A 669); “any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP676” (mixture ratio 1:10 to 10: 1) (composition A 670); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP679” “Composition ratio 1:10 to 10: 1” (composition A 671); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 680” (mixture ratio 1:10 to 10: 1) (Composition A 672); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 681” (mixing ratio 1:10 to 10: 1) (Composition A673); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP682” (mixture ratio 1:10 to 10: 1) (composition A 674); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP683” (Combination ratio 1:10 to 10: 1) (Composition A 675); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP684” (mixture ratio 1:10 to 10: 1) (Composition A 676); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 685” (mixing ratio 1:10 to 10: 1) (Composition A 677); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP686” (mixture ratio 1:10 to 10: 1) (composition A 678); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP687” (mixture ratio 1:10 to 10: 1) (Composition A 679); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP688” (mixture ratio 1 "Composition A680);" Any one of Compounds AA1-BA1-AK2688-BK1287 "and" PP689 "(mixing ratio 1:10 to 10: 1) (Composition A 681) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP690” (mixing ratio 1:10 to 10: 1) (Composition A 682); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “Kone” and “PP691” (mixture ratio 1:10 to 10: 1) (composition A683); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP693 (Combination ratio 1:10 to 10: 1) (composition A 684); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP694” (mixture ratio 1:10 to 10) 1) (Composition A 685); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 695” in combination (mixing ratio 1:10 to 10: 1) (Composition A 686); “Compound AA1 Any one of “-BA1 to AK2688-BK1287” and “PP696” (mixture ratio 1:10 to 10: 1) (composition A687); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with "PP 697" (mixture ratio 1:10 to 10: 1) (Composition A 688); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP698" (mixture ratio 1:10 ~ 10: 1) (Composition A 689); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP699" (mixing ratio 1:10 to 10: 1) (Composition A690); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP700” (mixing ratio 1:10 to 10: 1) (Composition A691); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1:70 to 10: 1” (composition A692) of “PP702” (composition A692); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP703” (Composition ratio 1:10 to 10: 1) (Composition A693); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP704” (mixture ratio 1:10 to 10: 1) “Composition A694);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP705 ”(mixing ratio 1:10 to 10: 1) (Composition A695);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP706” (mixture ratio 1:10 to 10: 1) (composition A 696); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP 707” (mixing ratio 1:10 to 10: 1) (Composition A 697); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP708” (mixing ratio 1 “Composition A 698);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 709 ”(mixture ratio 1: 10 to 10: 1) (Composition A 699) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP710” (mixture ratio 1:10 to 10: 1) (Composition A700); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP711” (mixture ratio 1:10 to 10: 1) (Composition A 701); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP712” (Mixed “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 713” (mixture ratio 1:10 to 10: 1 to 10: 1) (Composition A 702); (Composition A703); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP714” (mixing ratio 1:10 to 10: 1) (Composition A704); “Compound AA1-BA1” -Any one of AK2688-BK1287 and 'PP714-1' (mixture ratio 1:10 to 10: 1) (Composition A705); “any one of Compounds AA1-BA1 to AK2688-BK1287” Combination with “PP715” (mixture ratio 1:10 to 10: 1) (Composition A 706); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP716” (mixture ratio 1:10 "Composition A 707";"Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287" and "PP 717" (mixing ratio 1: 10 to 10: 1) (Composition A 708); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP718” (mixing ratio 1:10 to 10: 1) (composition A 709); “compound AA1-BA1 to AK2688-BK1287 Combination of “one or more” and “PP719” (mixture ratio 1:10 to 10: 1) (composition A 710); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP720” (composition Mixing ratio 1:10 to 10: 1) (Composition A711); "Any one of the compounds AA1-BA1 to AK2688-BK1287" and "PP 721" (mixing ratio 1:10 to 10: 1) (composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP722” (mixing ratio 1:10 to 10: 1) (composition A 713); “compound AA1 to BA1 to AK2688” “Any one of BK1287” and “PP 723” in combination (mixture ratio 1:10 to 10: 1) (composition A 714); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP723-1” (Combination ratio 1:10 to 10: 1) (composition A 715); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP724” (mixture ratio 1: 10 to 10: 1) (Composition A 716); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 725” (mixing ratio 1:10 to 10: 1) (Composition A 717); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP725-1” (mixture ratio 1:10 to 10: 1) (Composition A 718); “Compound AA1-BA1 to AK2688-BK1287 Combination of any one of them and “PP 726” (mixture ratio 1:10 to 10: 1) (Composition A 719); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP727” Mixing ratio 1:10 to 10: 1) (Composition A 720); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP727-1" (mixing ratio 1:10 to 10: 1) (Composition A 721); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 728” (mixing ratio 1:10 to 10: 1) (Composition A 722); “Compound AA 1-BA1 Any one of the AK2688-BK1287 "
And “PP729” (mixture ratio 1:10 to 10: 1) (Composition A 723); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP730” (mixture ratio 1: 10 to 10: 1) (Composition A 724); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 730-1” (mixing ratio 1:10 to 10: 1) (Composition A 725) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 730-2" (mixing ratio 1:10 to 10: 1) (Composition A 726); "Compounds AA1-BA1 to AK2688-" “Any one of BK1287” and “PP 730-3” in combination (mixture ratio 1:10 to 10: 1) (composition A 727); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP730- 4 "(mixture ratio 1:10 to 10: 1) (Composition A 728);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP 730-5 "(mixture ratio 1: 10 to 1 1) (Composition A 729); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 730-6” (mixing ratio 1: 10 to 10: 1) (Composition A 730); Any one of compounds AA1-BA1 to AK2688-BK1287 and “PP 730-7” (mixture ratio 1:10 to 10: 1) (composition A 731); “any of compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP 730-8” (mixture ratio 1:10 to 10: 1) (composition A 732); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP730-9” Combination (mixture ratio 1:10 to 10: 1) (composition A 733); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 730-10” (mixture ratio 1:10 to 10) "Composition A734";"Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP 731" (mixing ratio 1:10 to 10: 1) (Composition A 735); "Compound AAl -BA1 to AK26 “Any one of 88-BK1287” and “PP 731-1” (mixture ratio 1:10 to 10: 1) (composition A 736); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 731-2 "(mixture ratio 1:10 to 10: 1) (Composition A 737);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP731-3 "(mixture ratio 1:10 to 10: 1) (Composition A 738); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP731-4” (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP732” (mixture ratio 1:10 to 10: 1) (composition A 740); “compound AA1 to BA1 to AK2688” “Any one of BK1287” and “PP732-1” in combination (mixture ratio 1:10 to 10: 1) (Composition A 741); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP733” Pair with “Composition ratio 1:10 to 10: 1” (composition A 742); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP733-1” (mixture ratio 1:10 to 10: 1) (Composition A 743); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 733-2” (mixing ratio 1:10 to 10: 1) (Composition A 744); Any one of AA1-BA1 to AK2688-BK1287 and “PP733-3” (mixture ratio 1:10 to 10: 1) (composition A745); “any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP734” (mixture ratio 1:10 to 10: 1) (Composition A 746); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP734-1” Mixing ratio 1:10 to 10: 1) (Composition A 747); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 735" (mixing ratio 1:10 to 10: 1) (Composition Object A74 8) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP736” (mixture ratio 1:10 to 10: 1) (Composition A 749); “Compounds AA1-BA1 to AK2688-BK1287 Of “any one of” and “PP737” (mixture ratio 1:10 to 10: 1) (composition A 750); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP738” (Composition ratio 1:10 to 10: 1) (Composition A 751); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP739” (mixture ratio 1:10 to 10: 1) (Composition A 751) “Composition A 752”; “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 740” (mixture ratio 1:10 to 10: 1) (Composition A753); “Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP741” (mixture ratio 1:10 to 10: 1) (composition A 754); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP 742” (mixture ratio 1: 10 to 10: 1) (Composition A 755); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 743” (mixture ratio 1: 10 “Composition A756);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP744 ”(mixing ratio 1:10 to 10: 1) (Composition A757); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP745” (mixture ratio 1:10 to 10: 1) (composition A758); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP746” (mixture ratio 1:10 to 10: 1) (Composition A759); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP747” (mixture ratio 1 "Composition A760);" Any one of Compounds AA1-BA1-AK2688-BK1287 "and" PP 748 "(mixing ratio 1:10 to 10: 1) (Composition A 761); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 749” in combination (mixing ratio 1:10 to 10: 1) (Composition A 762); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP750” (mixture ratio 1:10 to 10: 1) (composition A 763); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP751” (Combination ratio 1:10 to 10: 1) (composition A764); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP751-1” (mixture ratio 1:10 to 10) 10: 1) (Composition A 765); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 752” (mixing ratio 1:10 to 10: 1) (Composition A 766); “Compound A combination of any one of AA1-BA1 to AK2688-BK1287 with “PP 752-1” (mixture ratio 1:10 to 10: 1) (Composition A 767); “A respectively of compounds AA1-BA1 to AK2688-BK1287 A combination of 1) and “PP 752-2” (mixture ratio 1:10 to 10: 1) (composition A 768); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP753” Combination (mixture ratio 1:10 to 10: 1) (Composition A 769); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP754" (mixture ratio 1:10 to 10: 1) (Composition A 770); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP754-1” (mixing ratio 1:10 to 10: 1) (Composition A771); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP 754-2” (mixture ratio 1:10 to 10: 1) (composition A 772); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 754-3” (mixture ratio 1:10 to 10: 1) (Composition A 773); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP755” (mixture ratio 1 "Composition A 774";"Any one of the compounds AA1-BA1-AK2688-BK1287" and "PP 756" (mixing ratio 1:10 to 10: 1) (Composition A 775) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP757” (mixing ratio 1:10 to 10: 1) (Composition A 776); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP758” (mixture ratio 1:10 to 10: 1) (Composition A 777); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP759” “Composition A 778);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 760 ”(mixture ratio 1: 10 to 10: 1) (Composition A779); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP761” (mixture ratio 1:10 to 10: 1) (Composition A 780); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP762” (mixture ratio 1:10 to 10: 1) (composition A 781); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP763” (Combination ratio 1:10 to 10: 1) (Composition A 782); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP764” (mixture ratio 1:10 to 10: 1) (Composition A 783); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP765” (mixing ratio 1:10 to 10: 1) (Composition A 784); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP766” (mixing ratio 1:10 to 10: 1) (composition A 785); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 767 "(mixture ratio 1: 10 to 10: 1) (Composition A 786);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP768 " (Composition ratio 1:10 to 10: 1) (Composition A 787); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP768-1” (Mixing ratio 1:10 to 10: 1 (Composition A 788); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP769” (mixing ratio 1:10 to 10: 1) (Composition A 789); “Compound AA1 to BA1” -A combination of “one of AK2688-BK1287” and “PP769-1” (mixture ratio 1:10 to 10: 1) (composition A 790); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP 770” (mixture ratio 1:10 to 10: 1) (Composition A 791); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP771” (mixture ratio 1:10 ~ 10: 1) (Composition A 792); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 772" in combination (mixing ratio 1:10 to 10: 1) (Composition A 793); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP773” (mixture ratio 1:10 to 10: 1) (composition A 794); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP774” (mixture ratio 1:10 to 10: 1) (Composition A795); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP775” (mixture ratio 1 "Composition A796);" Any one of Compounds AA1-BA1-AK2688-BK1287 "and" PP 776 "(mixing ratio 1:10 to 10: 1) (Composition A 797) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP777” (mixing ratio 1:10 to 10: 1) (Composition A798); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP778” (mixture ratio 1:10 to 10: 1) (composition A 799); “any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP77 9 (combination ratio 1:10 to 10: 1) (composition A 800); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP780” (mixture ratio 1:10 to 10) 10: 1) (Composition A801); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP781” (mixing ratio 1:10 to 10: 1) (Composition A 802); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP782” (mixture ratio 1:10 to 10: 1) (composition A 803); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP783” (mixture ratio 1:10 to 10: 1) (Composition A 804); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP783-1” (mixture ratio 1:10 to 10: 1) (Composition A 805); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP783-2” (mixing ratio 1:10 to 10: 1) “Composition A806);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP784 ”(mixing ratio 1:10 to 10: 1) (Composition A 807);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP785” (mixture ratio 1:10 to 10: 1) (composition A 808); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP786” Combination (mixture ratio 1:10 to 10: 1) (composition A 809); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP787” (mixture ratio 1:10 to 10: 1 (Composition A810); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP788” in combination (mixing ratio 1:10 to 10: 1) (Composition A811); “Compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287” and “PP789” (mixture ratio 1:10 to 10: 1) (composition A812); “any one of compounds AA1-BA1 to AK2688-BK1287 "Tosu" and "PP 790"
Combination (mixture ratio 1:10 to 10: 1) (composition A813); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP791” (mixture ratio 1:10 to 10: 1 (Composition A 814); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 792” (mixing ratio 1:10 to 10: 1) (Composition A815); “Compound AA1 to BA1” ~ Any one of AK2688-BK1287 "and" PP 793 "(mixture ratio 1:10 to 10: 1) (Composition A 816);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP793 " -1 (combination ratio 1:10 to 10: 1) (composition A 817); "any one of compounds AA1-BA1 to AK2688-BK1287" and "PP 793-2" (mix ratio 1 "Composition A 818";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP 793-3" (mixing ratio 1:10 to 10: 1) (Composition A819); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP793-4” (mixing ratio 1:10 to 10: 1) (Composition A820); “Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP794” (mixture ratio 1:10 to 10: 1) (composition A 821); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP794-1 (Mixture ratio 1:10 to 10: 1) (Composition A 822); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP794-2” (mixture ratio 1:10 ~ 10: 1) (Composition A 823); "Any one of Compounds AA1-BA 1 to AK 2688-BK 1287" and "PP 794-3" (mixing ratio 1: 10 to 10: 1) (Composition A 824) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP794-4” (mixing ratio 1:10 to 10: 1) (Composition A 825); “Compounds AA1-BA1 to AK2688-BK1287 Any of Combination of “one” and “PP795” (mixture ratio 1:10 to 10: 1) (Composition A 826); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP795-1” Mixing ratio 1:10 to 10: 1) (Composition A 827); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP796" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP796-1” (mixing ratio 1:10 to 10: 1) (composition A829); “compound AA1 to BA1”; “Any one of AK2688-BK1287” and “PP 797” (mixture ratio 1:10 to 10: 1) (composition A 830); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP798” (Combination ratio 1:10 to 10: 1) (composition A 831); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP798-1” (mixture ratio 1:11 0 to 10: 1) (Composition A 832); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 799” (mixing ratio 1:10 to 10: 1) (Composition A 833); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP799-1” (mixture ratio 1:10 to 10: 1) (composition A 834); “compound AA1-BA1 to AK2688-BK1287 Combination of any one of them and “PP800” (mixture ratio 1:10 to 10: 1) (composition A 835); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP800-1” Combination (mixture ratio 1:10 to 10: 1) (Composition A 836); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP800-2” (mixture ratio 1:10 to 10: 1) (Composition A837); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP800-3” in combination (mixing ratio 1:10 to 10: 1) (Composition A 838); “Compound AA1-BA1 -Any one of AK2688-BK1287 'and' PP800-4 '(mixture ratio 1:10 to 10: 1) (Composition A839);' any one of Compounds AA1-BA1 to AK2688-BK1287 ' Combination with “PP801” (mixture ratio 1:10 to 10: 1) (Composition A 840); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP802” (mixture ratio 1:10 “Composition A 841);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 803 ”(mixing ratio 1: 10 to 10: 1) (Composition A 842); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP804” (mixture ratio 1:10 to 10: 1) (composition A 843); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 805” (mixture ratio 1:10 to 10: 1) (Composition A 844); “Any one of Compound AA1-BA1 to AK2688-BK1287” and “PP 806” “Composition ratio 1:10 to 10: 1” (composition A845); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 807” (mixture ratio 1:10 to 10: 1) (Composition A 846); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP808” (mixing ratio 1:10 to 10: 1) (Composition A 847); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP808-1” (mixture ratio 1:10 to 10: 1) (composition A 848); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 808-2 (mixture ratio 1: 10 to 10: 1) (Composition A 849); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 809” (mixture ratio 1: 10 to 10: 1) (Composition A 850); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 809-1” (mixing ratio 1: 10 to 10: 1) (Composition A 851) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP810” (mixture ratio 1:10 to 10: 1) (Composition A 852); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP811” (mixture ratio 1:10 to 10: 1) (Composition A 853); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP812” (mixture "Composition A 854";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP812-1" (mixing ratio 1:10 to 10: 1) (Composition A 854) “Composition A855);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP813 ”(mixture ratio 1:10 to 10: 1) (Composition A856);“ Compounds AA1-BA1 to AK2688 -Any one of BK1287 'and' PP814 '(mixture ratio 1:10 to 10: 1) (composition A 857);' any one of compounds AA1-BA1 to AK2688-BK1287 ' Combination with “PP814-1” (mixture ratio 1:10 to 10: 1) (Composition A 858); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP814-2” “Composition A 859);“ Any one of Compounds AA1-BA 1 to AK 2688-BK 1287 ”and“ PP 815 ”(mixing ratio 1:10 to 10: 1) (Composition A860); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP816” (mixture ratio 1:10 to 10: 1) (Composition A861); “Compounds AA1-BA1 to AK2688-BK1287 And “PP 817” (mixture ratio 1:10 to 10: 1) (composition A 862); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP817-1” Combination (mixture ratio 1:10 to 10: 1) (composition A 863); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 817-2” (mixture ratio 1:10 to 10) 1) (Composition A864); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 818” in combination (mixing ratio 1:10 to 10: 1) (Composition A865); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP 819” (mixture ratio 1:10 to 10: 1) (composition A866); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 820 ′ ′ (mixture ratio 1: 10 to 10: 1) (Composition A 867); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 821” (mixture ratio 1: 10 to 10: 1) (Composition A 868); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 821-1” (mixing ratio 1:10 to 10: 1) (Composition A869); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP821-2” (mixture ratio 1:10 to 10: 1) (Composition A 870); “Compounds AA1-BA1 to AK2688-BK1287 “Any one” and “PP 822” in combination (mixture ratio 1:10 to 10: 1) (Composition A 871); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP823” Mixing ratio 1:10 to 10: 1) (Composition A 872); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 824" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP825” (mixing ratio 1:10 to 10: 1) (composition A 874); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP826” (mixture ratio 1:10 to 10: 1) (composition A 875); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP827” Combination (mixture ratio 1:10 to 10: 1) (Composition A 876); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 828” (mixture ratio 1 10 to 10: 1) (Composition A 877); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 828-1” (mixing ratio 1:10 to 10: 1) (Composition A 878) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP829" (mixture ratio 1:10 to 10: 1) (Composition A879); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and “PP830” (mixture ratio 1:10 to 10: 1) (composition A 880); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP830-1” Combination (mixture ratio 1:10 to 10: 1) (Composition A 881); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP830-2” (mixture ratio 1:10 to 10: 1) (Composition A 882); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 831” (mixing ratio 1:10 to 10: 1) (Composition A 883); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP 831-1” (mixture ratio 1:10 to 10: 1) (composition A 884); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 832” (mixture ratio 1:10 to 10: 1) (Composition A 885); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP833” (mixture ratio 1: 10 to 10: 1) (Composition A 886); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP833-1” (mixing ratio 1:10 to 10: 1) (Composition A 887) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 834" (mixture ratio 1:10 to 10: 1) (Composition A 888); "Compounds AA1-BA1 to AK2688-BK1287 “Any one” and “PP 835” in combination (mixture ratio 1:10 to 10: 1) (composition A 889); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP835-1” Combination (mixture ratio 1:10 to 10: 1) (Composition A 890); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP836" (mixture ratio 1:10 to 10: 1) (Composition A891); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP837” (mixing ratio 1:10 to 10: 1) (Composition A892); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP838” in combination (mixture ratio 1:10 to 10: 1) (composition A 893); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP838- 1 (combination ratio 1:10 to 10: 1) (composition A 894); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP839” (mixture ratio 1:10 to 10) 10: 1) (Composition A 895); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 839-1” (mixing ratio 1:10 to 10: 1) (Composition A 896) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP840” (mixture ratio 1:10 to 10: 1) (Composition A897); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1: 84 to 10: 1) (composition A 898) with“ PP 841 ”(composition A 898);“ combination of any one of compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 842 ” (Mixing ratio 1:10 to 10: 1) (Composition A 899); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP842-1” (Mixing ratio 1:10 to 10: 1 (Composition A900); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP843” (mixture ratio 1:10 to 10: 1) (Composition A901); “Compound AA1 to BA1” ~ A combination of “any one of AK2688-BK1287” and “PP843-1” (mixture ratio 1:10 to 10: 1) (Composition A 902); “Compound AA 1-BA 1 to AK 2688-BK 1287 any one of "And" PP843-2 "
(Combination ratio 1:10 to 10: 1) (composition A 903); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP844” (mixture ratio 1:10 to 10: 1) (Composition A 904); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP845” (mixing ratio 1:10 to 10: 1) (Composition A 905); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP 846” (mixture ratio 1:10 to 10: 1) (composition A 906); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition A 907” with “PP 847” (mixture ratio 1:10 to 10: 1); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP848” (mixture ratio 1:10 to 10) 10: 1) (Composition A 908); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP848-1” (mixing ratio 1:10 to 10: 1) (Composition A 909); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP848-2” (mixing ratio 1:10 to 10: 1) (Composition A 910); “Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP849” (mixture ratio 1:10 to 10: 1) (composition A 911); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP849-1 (Mixture ratio 1:10 to 10: 1) (Composition A 912); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP850” (mixture ratio 1:10 to 10: 1) 1) (Composition A 913); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 850-1” (mixing ratio 1: 10 to 10: 1) (Composition A 914); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP851” (mixture ratio 1:10 to 10: 1) (composition A 915); “any one of the compounds AA1-BA1 to AK2688-BK1287 “Composition” and “PP 851-1” (mixture ratio 1:10 to 10: 1) (composition A 916); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP851-2” Combination (mixture ratio 1:10 to 10: 1) (Composition A 917); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 851-3” (mixture ratio 1:10 to 10) 1) (Composition A 918); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 851-4” (mixing ratio 1: 10 to 10: 1) (Composition A 919); Any one of compounds AA1-BA1 to AK2688-BK1287 and “PP 851-5” (mixture ratio 1:10 to 10: 1) (composition A920); “any of compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 852” (mixture ratio 1:10 to 10: 1) (Composition A 921); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP852-1” (Mixing ratio 1: 0 to 10: 1) (Composition A 922); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 853” (mixing ratio 1:10 to 10: 1) (Composition A 923); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP853-1” (mixture ratio 1:10 to 10: 1) (Composition A 924); “Compound AA1-BA1 to AK2688-BK1287 Combination of any one of them and “PP 854” (mixture ratio 1:10 to 10: 1) (Composition A 925); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP855” (Composition A925) Mixing ratio 1:10 to 10: 1) (Composition A 926); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 855-1" (Mixing ratio 1:10 to 10: 1) (Composition A 927); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 856” (mixture ratio 1:10 to 10: 1) (Composition A 928); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP 857” in combination (mixture ratio 1:10 to 10: 1) (Composition A 929); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP858” (Combination ratio 1:10 to 10: 1) (composition A 930); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP858-1” (mixture ratio 1:10 to 10) 10: 1) (Composition A 931); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP859” (mixing ratio 1:10 to 10: 1) (Composition A 932); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP860” (mixture ratio 1:10 to 10: 1) (Composition A 933); “any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP860-1” (mixture ratio 1:10 to 10: 1) (Composition A 934); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP861” “Composition ratio 1:10 to 10: 1” (composition A 935); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 861-1” (mixture ratio 1:10 to 10: 1) (Composition A 936); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 862” (mixing ratio 1:10 to 10: 1) (Composition A 937); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP863” (mixture ratio 1:10 to 10: 1) (composition A 938); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition A939” with “PP 864” (mixture ratio 1:10 to 10: 1); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP864-1” (mixture ratio 1: 10 to 10: 1) (Composition A 940); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP865” (mixing ratio 1:10 to 10: 1) (Composition A 941) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP865-1” (mixture ratio 1:10 to 10: 1) (Composition A942); “Compound AA1-BA1 to AK2688-BK1287 Combination of any one of them and “PP866” (mixture ratio 1:10 to 10: 1) (Composition A943); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP866-1” Combination (mixture ratio 1:10 to 10: 1) (Composition A 944); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP867" (mixture ratio 1:10 to 10: 1) (Composition A 945); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP868” (mixture ratio 1:10 to 10: 1) (Composition A 946); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP869” in combination (mixture ratio 1:10 to 10: 1) (composition A947); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP869-1” (mixture ratio 1:10 to 10: 1) (Composition A 948); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP870” (mixture ratio 1 “Composition A 949);“ Any one of the compounds AA1-BA1 to AK2688-BK1287 ”and“ PP870-1 ”(mixing ratio 1:10 to 10: 1) (composition A950); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP871” (mixing ratio 1:10 to 10: 1) (Composition A 951); “Compounds AA1-BA1 to AK2688-BK1287 Of “any one of” and “PP 872” (mixture ratio 1:10 to 10: 1) (composition A 952); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP873” (Composition ratio 1:10 to 10: 1) (Composition A953); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP873-1” (mixture ratio 1:10 to 10: (Composition A954); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP874” in combination (mixing ratio 1:10 to 10: 1) (Composition A955); “Compound AA1-BA1” ~ Any one of AK2688-BK1287 "and" PP875 "(mixture ratio 1:10 to 10: 1) (Composition A956);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP876 " (Combination ratio 1:10 to 10: 1) (composition A 957); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP877” (mixture ratio 1:10 to 10) "Composition A958";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 878" in combination (mixing ratio 1:10 to 10: 1) (Composition A 959); "Compound AA1 Any one of “BA1 to AK2688-BK1287” and “PP879” (mixture ratio 1:10 to 10: 1) (composition A 960); “any of compounds AA1-BA1 to AK2688-BK1287 A combination of 1) and “PP 879-1” (mixture ratio 1:10 to 10: 1) (composition A 961); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP880” Combination (mixture ratio 1:10 to 10: 1) (Composition A 962); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP881" (mixture ratio 1:10 to 10: 1) (Composition A963); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP882” (mixing ratio 1:10 to 10: 1) (Composition A964); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP883” (mixture ratio 1:10 to 10: 1) (composition A965); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP884” (Composition ratio 1:10 to 10: 1) (composition A 966); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP885” (mixture ratio 1:11 0 to 10: 1) (Composition A 967); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP886” (mixing ratio 1:10 to 10: 1) (Composition A 968); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP887” (mixture ratio 1:10 to 10: 1) (Composition A 969); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP888” (mixture ratio 1:10 to 10: 1) (Composition A 970); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP889” (mixture ratio 1:10 to 10: 1) (Composition A 971); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 890” (mixing ratio 1:10 to 10: 1) (Composition A 972) A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP891” (mixture ratio 1:10 to 10: 1) (composition A 973); “compound AA1 to BA1 to AK268” “Any one of 8-BK1287” and “PP 892” in combination (mixture ratio 1:10 to 10: 1) (composition A 974); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP893” (Combination ratio 1:10 to 10: 1) (composition A 975); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 894” (mixture ratio 1:10 to 10: 1) (Composition A976); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP895” (mixing ratio 1:10 to 10: 1) (Composition A977); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP896” (mixture ratio 1:10 to 10: 1) (composition A 978); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 897 "(mixing ratio 1:10 to 10: 1) (Composition A 979);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP898 "(Mixed Combination ratio 1:10 to 10: 1) (Composition A 980); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP899" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP900” (mixture ratio 1:10 to 10: 1) (composition A 982); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP901” (mixture ratio 1:10 to 10: 1) (composition A 983); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP902” Combination (mixture ratio 1:10 to 10: 1) (Composition A 984); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 903" (mixture ratio 1:10 to 10: 1) (Composition A985): “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP 904” (mixing ratio 1:10 to 10: 1) (Composition A 986); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP905” (mixture ratio 1:10 to 10: 1) (composition A 987); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 906” (mixture ratio 1:10 to 10: 1) (Composition A 988); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP 907” (mix ratio 1: 10 to 10: 1) (Composition A 989); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 908” (mixing ratio 1:10 to 10: 1) (Composition A 990); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP909” (mixing ratio 1:10 to 10: 1) (Composition A 991); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP 910” (mixture ratio 1:10 to 10: 1) (composition A 992); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP911” Combination (mixing ratio 1:10 to
10: 1) (Composition A 993); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 912” (mixing ratio 1:10 to 10: 1) (Composition A 994); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP913” (mixture ratio 1:10 to 10: 1) (composition A995); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 914” (mixture ratio 1:10 to 10: 1) (Composition A 996); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 915” (mixture ratio 1: 10 to 10: 1) (Composition A 997); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 916” (mixing ratio 1:10 to 10: 1) (Composition A 998); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP917” (mixture ratio 1:10 to 10: 1) (Composition A 999); “Compounds AA1-BA1 to AK2688-BK12 “Any one of 87” and “PP 918” in combination (mixture ratio 1:10 to 10: 1) (composition A 1000); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP919” Combination (mixture ratio 1:10 to 10: 1) (Composition A1001); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP920" (mixture ratio 1:10 to 10: 1) (Composition A1002); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 921” (mixing ratio 1:10 to 10: 1) (Composition A1003); “Compound AA1 to BA1” “Any one of AK2688-BK1287” and “PP 922” (mixture ratio 1:10 to 10: 1) (composition A 1004); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP923” Combination (mixture ratio 1:10 to 10: 1) (composition A 1005); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 924” Composition ratio 1:10 to 10: 1) (Composition A 1006); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 925" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP926” (mixing ratio 1:10 to 10: 1) (composition A1008); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP 927” (mixture ratio 1:10 to 10: 1) (composition A 1009); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP928” Combination (mixture ratio 1:10 to 10: 1) (Composition A1010); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 929" (mixture ratio 1:10 to 10: 1) (Composition A1011): “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 930” (mixing ratio 1:10 to 10: 1) (Composition A1012); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP931” (mixing ratio 1:10 to 10: 1) (composition A1013); “any one of compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 932” (mixture ratio 1:10 to 10: 1) (Composition A 1014); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 933” (mixture ratio 1:10 to 10: 1) (Composition A1015); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP934” (mixing ratio 1:10 to 10: 1) (Composition A1016) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP935" (mixing ratio 1:10 to 10: 1) (Composition A1017); "Compounds AA1-BA1 to AK2688-BK1287" “Any one” and “PP 936” in combination (mixture ratio 1:10 to 10: 1) (composition A1018); “any one of compounds AA1-BA1 to AK2688-BK1287” and “P “Composition A1019) with“ P937 ”(mixture ratio 1:10 to 10: 1);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP938 ”(mixture ratio 1:10 to 10) 10: 1) (Composition A1020); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP939” in combination (mixing ratio 1:10 to 10: 1) (Composition A1021); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP940” (mixture ratio 1:10 to 10: 1) (Composition A 1022); “any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP 941” (mixture ratio 1:10 to 10: 1) (Composition A 1023); “Any one of Compound AA1-BA1 to AK2688-BK1287” and “PP942” (mixture ratio 1: 10 to 10: 1) (Composition A 1024); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP943” (mixing ratio 1:10 to 10: 1) (Composition A1025); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 944” in combination (mixing ratio 1:10 to 10: 1) (Composition A1026); “Compounds AA1-BA1 “Any one of AK2688-BK1287” and “PP 945” in combination (mixture ratio 1:10 to 10: 1) (composition A1027); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP946” (Combination ratio 1:10 to 10: 1) (composition A1028); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP947” (mixture ratio 1:10 to 10: 1) (Composition A1029); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP948” (mixing ratio 1:10 to 10: 1) (Composition A1030); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP949” (mixture ratio 1:10 to 10: 1) (composition A1031); “compound AA1-BA1 to AK2688-BK1287” Combination of “one or more” and “PP950” (mixture ratio 1:10 to 10: 1) (composition A1032); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP951” Mixing ratio 1:10 to 10: 1) (Composition A1033); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 952" (Mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP953” (mixing ratio 1:10 to 10: 1) (composition A1035); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP954” (mixture ratio 1:10 to 10: 1) (composition A1036); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP955” Combination (mixture ratio 1:10 to 10: 1) (Composition A1037); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP956” (mixture ratio “Composition A1038);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP957 ”(mixing ratio 1:10 to 10: 1) (Composition A1039) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP958” (mixing ratio 1:10 to 10: 1) (Composition A1040); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP 959” (mixture ratio 1:10 to 10: 1) (Composition A 1041); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP960” (Mixed “Composition A1042);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP961 ”(mixing ratio 1:10 to 10: 1) (Composition A1043); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP962” (mixing ratio 1:10 to 10: 1) (Composition A1044); “Compound A Any one of A1-BA1 to AK2688-BK1287 and “PP963” (mixture ratio 1:10 to 10: 1) (composition A1045); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP964” (mixture ratio 1:10 to 10: 1) (Composition A 1046); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP965” (mixture ratio 1: 10-10: 1) (Composition A1047); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP966” (mixing ratio 1:10 to 10: 1) (Composition A1048); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP967” (mixing ratio 1:10 to 10: 1) (Composition A1049); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP968” (mixture ratio 1:10 to 10: 1) (composition A1050); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP969” Combination (mixture ratio 1:10 to 10: 1) (composition A 1051); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 970” (mixture ratio 1:10 to 10: 1 (Composition A1052); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP971” (mixing ratio 1:10 to 10: 1) (Composition A1053); “Compound AA1-BA1” ~ Any one of AK2688-BK1287 "and" PP972 "(mixture ratio 1:10 to 10: 1) (composition A1054);" any one of compounds AA1-BA1 to AK2688-BK1287 "and" PP973 " (Composition ratio A1055); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP974” (mixture ratio 1:10 to 10) "Composition A1056";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP975" (mixing ratio 1:10 to 10: 1) (combination A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP976” (mixing ratio 1:10 to 10: 1) (composition A1058); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP977” (mixture ratio 1:10 to 10: 1) (composition A1059); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP978” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1060); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP979" (mixture ratio 1:10 to 10: 1) (Composition A1061); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP980” (mixture ratio 1:10 to 10: 1) (Composition A1062); “Compound AA1 to BA1-1 “Any one of AK2688-BK1287” and “PP981” (mixture ratio 1:10 to 10: 1) (Composition A1063); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP982” (mixture ratio 1:10 to 10: 1) (Composition A 1064); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP983” (mixture ratio 1: 10 to 10: 1) (Composition A 1065); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 984” (mixing ratio 1: 10 to 10: 1) (Composition A 1066) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP985" (mixing ratio 1:10 to 10: 1) (Composition A1067); "Compounds AA1-BA1 to AK2688-BK1287" “Any one” and “PP986” in combination (mixture ratio 1:10 to 10: 1) (Composition A1068); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP987” Mixing ratio 1:10 to 10: 1) (Composition A1069); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP988" (mixing ratio 1: 1) “Composition A 1070);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”and“ PP 989 ”(mixing ratio 1: 10 to 10: 1) (Composition A 1071); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP990” (mixture ratio 1:10 to 10: 1) (composition A1072); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 991” (mixture ratio 1:10 to 10: 1) (Composition A 1073); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP992” (mixture ratio 1 "Composition A1074" (Composition A1075); "Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP993" (mixing ratio 1:10 to 10: 1) (Composition A1075) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP994" (mixing ratio 1:10 to 10: 1) (Composition A1076); "Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP995” (mixture ratio 1:10 to 10: 1) (composition A1077); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP996” (Combination ratio 1:10 to 10: 1) (composition A 1078); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP997” (mixture ratio 1:10 to 10: 1) (Composition A1079); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP998” (mixing ratio 1:10 to 10: 1) (Composition A1080); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP 999” (mixture ratio 1:10 to 10: 1) (composition A1081); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1000 "(mixture ratio 1: 10 to 10: 1) (composition A 1082);" any one of compounds AA1-BA1 to AK2688-BK1287 "and" PP1001 " Combined (mixed
Combination ratio 1:10 to 10: 1) (Composition A1083); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1002" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1003” (mixing ratio 1:10 to 10: 1) (composition A1085); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1004” (mixture ratio 1:10 to 10: 1) (composition A1086); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1005” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1087); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1006" (mixture ratio 1:10 to 10: 1) (Composition A1088); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1007” (mixing ratio 1:10 to 10: 1) (Composition A1089) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1008” (mixing ratio 1:10 to 10: 1) (Composition A 1090); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP1009” (mixture ratio 1:10 to 10: 1) (Composition A1091); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1010” (mixture ratio 1:10 to 10: 1) (Composition A1092); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1011” (mixing ratio 1:10 to 10: 1) (Composition A1093) A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1012” (mixture ratio 1:10 to 10: 1) (composition A1094); “compound AA1-BA1 to AK2688-BK1287” A combination of “one one” and “PP1013” (mixture ratio 1:10 to 10: 1) (composition A1095); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP1014” (mixture ratio 1:10 to 10: 1) (Composition A1096); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1015” (mixture ratio 1 “Composition A1097);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1016 ”(mixing ratio 1:10 to 10: 1) (Composition A1098) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1017” (mixing ratio 1:10 to 10: 1) (Composition A1099); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1018” (mixture ratio 1:10 to 10: 1) (composition A1100); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1019” (mixture Ratio 1:10 to 10: 1) (Composition A1101); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1020" (mixing ratio 1: 1 “Composition A1102);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1021 ”(mixing ratio 1:10 to 10: 1) (Composition A1103); Any one of compounds AA1-BA1 to AK2688-BK1287 and “PP1022” (mixing ratio 1:10 to 10: 1) (composition A1104); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP 1023” (mixture ratio 1:10 to 10: 1) (Composition A1105); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1024” (mixture ratio 1 "Composition A1106);" Any one of Compounds AA1-BA1-AK2688-BK1287 "and" PP1025 "(mixing ratio 1:10 to 10: 1) (Composition A1107) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1026” (mixing ratio 1:10 to 10: 1) (Composition A1108); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1027” (mixing ratio 1:10 to 10: 1) (composition A1109); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1028 "(mixture ratio 1:10 to 10: 1) (Composition A 1110);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1029 "(mixture ratio 1:10 to 10: 1) (Composition A1111); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1030” (mixing ratio 1:10 to 10: 1) (Composition A1112); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1031” (mixture ratio 1:10 to 10: 1) (composition A1113); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1032” (mixture ratio 1:10 to 10: 1) (composition A1114); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1033 (Combination ratio 1:10 to 10: 1) (composition A1115); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1034” (mixture ratio 1:10 to 10) “Composition A1116);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1035 ”(mixing ratio 1:10 to 10: 1) (Composition A1117);“ Compound AA1 Any one of “BA1 to AK2688-BK1287” and “PP1036” (mixing ratio 1:10 to 10: 1) (composition A1118); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with "PP1037" (mixture ratio 1:10 to 10: 1) (Composition A1119); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1038" (mixture ratio 1:10 ~ 10: 1) (Composition A1120); "Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP1039" (mixing ratio 1:10 to 10: 1 (Composition A1121); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1040” (mixing ratio 1:10 to 10: 1) (Composition A1122); “Compound AA1 to BA1-2” “Any one of AK2688-BK1287” and “PP1041” (mixture ratio 1:10 to 10: 1) (composition A1123); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1042” (Combination ratio 1:10 to 10: 1) (composition A1124); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1043” (mixture ratio 1:10 to 10: 1) (Composition A1125); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1044” (mixing ratio 1:10 to 10: 1) (Composition A1126); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP1045” (mixing ratio 1:10 to 10: 1) (composition A1127); “compound AA1-BA1 to AK2688-BK12 “Any one of 87” and “PP 1046” in combination (mixture ratio 1:10 to 10: 1) (composition A1128); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1047” Combination (mixture ratio 1:10 to 10: 1) (Composition A1129); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1048" (mixture ratio 1:10 to 10: 1) (Composition A1130); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1049” (mixing ratio 1:10 to 10: 1) (Composition A1131); “Compound AA1 to BA1-1” “Any one of AK2688-BK1287” and “PP1050” in combination (mixture ratio 1:10 to 10: 1) (composition A1132); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1051” (Combination ratio 1:10 to 10: 1) (composition A1133); “combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP1052 ” (Composition ratio 1:10 to 10: 1) (Composition A1134); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1053” (mixture ratio 1:10 to 10: 1) (Composition A1 134) “Composition A1135);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1054 ”(mixing ratio 1:10 to 10: 1) (Composition A1136);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP1055” (mixture ratio 1:10 to 10: 1) (composition A1137); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1056” Combination (mixture ratio 1:10 to 10: 1) (composition A1138); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1057” (mixture ratio 1:10 to 10: 1 (Composition A1139); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1058” (mixing ratio 1:10 to 10: 1) (Composition A11) 40) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1059” (mixing ratio 1:10 to 10: 1) (Composition A1141); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1: 10 to 10: 1” with “PP 1060” (composition A 1142) (composition A 1142); “any one of compounds AA 1 -BA 1 to AK 2688-BK 1287” and “PP 1061” (Composition ratio 1:10 to 10: 1) (Composition A1143); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1062” (mixture ratio 1:10 to 10: 1) “Composition A1144);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1063 ”(mixing ratio 1:10 to 10: 1) (Composition A1145);“ Compounds AA1 to BA1 to AK2688 -Any one of -BK1287 "and" PP1064 "(mixture ratio 1:10 to 10: 1) (composition A1146);" any of compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP1065” (mixture ratio 1:10 to 10: 1) (Composition A1147); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1066” (mixture ratio 1:10 to 10: 1) (Composition A1148); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1067” (mixing ratio 1:10 to 10: 1) (Composition A1149 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1068" (mixing ratio 1:10 to 10: 1) (Composition A1150); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and PP1069 (mixture ratio 1:10 to 10: 1) (Composition A 1151); Combination of any one of Compounds AA1-BA1 to AK2688-BK1287 and PP1070 (Composition A 1151) Mixing ratio 1:10 to 10: 1) (Composition A1152); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1071" (mixing ratio 1 10 to 10: 1) (Composition A 1153); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1072” (mixing ratio 1:10 to 10: 1) (Composition A1154); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1073” (mixing ratio 1:10 to 10: 1) (Composition A1155); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP1074” (mixture ratio 1:10 to 10: 1) (Composition A1156); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1075” (mixture ratio 1:10 to 10: 1) (Composition A1157); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1076” (mixing ratio 1:10 to 10: 1) (Composition A1158 A combination of “any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP1077” (mixing ratio 1:10 to 10: 1) (composition A 1159); “compound Any one of AA1 -BA1 to AK2688-BK1287 "and" PP1078 "(mixing ratio 1:10 to 10: 1) (composition A1160);" any one of Compounds AA1 to BA1 to AK2688-BK1287 And “PP1079” (mixture ratio 1:10 to 10: 1) (Composition A1161); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1080” (mixture ratio 1 “Composition A1162);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1081 ”(mixing ratio 1:10 to 10: 1) (Composition A1163) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1082” (mixing ratio 1:10 to 10: 1) (Composition A 1164); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1083” (mixture ratio 1:10 to 10: 1) (composition A1165); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP1084 (mixture ratio 1:10 to 10: 1) (Composition A1166); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1085” (mixture ratio 1:10 to 10: 1) (Composition A1167); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1086” in combination (mixing ratio 1:10 to 10: 1) (Composition A1168); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1087” (mixture ratio 1:10 to 10: 1) (composition A1169); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1088” (mixture ratio 1:10 to 10: 1) (Composition A1170); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1089” (mixture ratio 1: 10 to 10: 1) (Composition A 1171); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1090” (mixing ratio 1
“Composition A1172);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1091 ”(mixing ratio 1:10 to 10: 1) (Composition A1173) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1092” (mixing ratio 1:10 to 10: 1) (Composition A1174); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1093” (mixture ratio 1:10 to 10: 1) (composition A1175); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1094” (mixture “Composition A1176);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1095 ”(mixing ratio 1:10 to 10: 1) (Composition A1177); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1096” (mixing ratio 1:10 to 10: 1) (Composition A1178); Any one of AA1 -BA1 to AK2688-BK1287 "and" PP1097 "(mixture ratio 1:10 to 10: 1) (composition A1179);" any one of Compounds AA1 -BA1 to AK2688-BK1287 And “PP 1098” (mixture ratio 1:10 to 10: 1) (Composition A 1180); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1099” (mixture ratio 1 “Composition A1181);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1100 ”(mixing ratio 1:10 to 10: 1) (Composition A1182) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1101” (mixing ratio 1:10 to 10: 1) (Composition A1183); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP 1102” (mixture ratio 1:10 to 10: 1) (composition A1184); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP1103 "(mixture ratio 1:10 to 10: 1) (Composition A1185);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1104 "(mixture ratio 1:10 to 10) 10: 1) (Composition A1186); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1105” (mixing ratio 1:10 to 10: 1) (Composition A1187); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1106” (mixture ratio 1:10 to 10: 1) (composition A1188); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1107” (mixture ratio 1:10 to 10: 1) (Composition A1189); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1108” (mixture ratio 1: 10 to 10: 1) (Composition A1190); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1109” (mixing ratio 1:10 to 1) "Composition A1191";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1110" (mixing ratio 1:10 to 10: 1) (Composition A1192); "Compound A1 1 -Any one of “BA1 to AK2688-BK1287” and “PP1111” (mixture ratio 1:10 to 10: 1) (composition A1193); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with "PP1112" (mixture ratio 1:10 to 10: 1) (Composition A1194); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1113" (mixture ratio 1:10 “Composition A1195);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1114 ”(mixing ratio 1:10 to 10: 1) (Composition A1196); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP1115” (mixture ratio 1:10 to 10: 1) (composition A1197); “compound AA1-BA1 to AK2 Any one of 688-BK1287 and “PP1116” (mixture ratio 1:10 to 10: 1) (composition A1198); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1117” (Combination ratio 1:10 to 10: 1) (composition A 1199); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1118” (mixture ratio 1:10 to 10: 1) (Composition A1200); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1119” in combination (mixing ratio 1:10 to 10: 1) (Composition A1201); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1120” (mixing ratio 1:10 to 10: 1) (composition A1202); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP1121 (mixture ratio 1:10 to 10: 1) (Composition A1203); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1122” Combination (mixture ratio 1:10 to 10: 1) (Composition A1204); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1123" (mixture ratio 1:10 to 10: 1) (Composition A1205); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1124” (mixing ratio 1:10 to 10: 1) (Composition A1206); “Compound AA1 to BA1” “Any one of AK2688-BK1287” and “PP1125” (mixture ratio 1:10 to 10: 1) (composition A1207); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1126” (Combination ratio 1:10 to 10: 1) (composition A1208); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1127” (mixture ratio 1:10 to 10: 1) (Composition A1209); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1128” (mixing ratio 1:10 to 10: 1) (pair A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1129” (mixing ratio 1:10 to 10: 1) (composition A1211); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1130” (mixture ratio 1:10 to 10: 1) (composition A1212); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1131” Combination (mixture ratio 1:10 to 10: 1) (Composition A1213); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1132" (mixture ratio 1:10 to 10: 1) (Composition A1214); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP1133” (mixing ratio 1:10 to 10: 1) (Composition A1215); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP1134” (mixture ratio 1:10 to 10: 1) (composition A 1216) (composition AA1-BA1 to AK2688-BK1287) Combination of “one” and “PP1135” (mixture ratio 1:10 to 10: 1) (composition A1217); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1136” Mixing ratio 1:10 to 10: 1) (Composition A1218); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1137" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1138” (mixing ratio 1:10 to 10: 1) (composition A1220); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1139” (mixture ratio 1:10 to 10: 1) (composition A1221); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1140” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1222); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1141” "Composition A1223";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1142" (mixing ratio 1:10 to 10: 1) (Composition “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1143” (mixing ratio 1:10 to 10: 1) (Composition A1225); “Compounds AA1-BA1 to AK2688-BK1287 Any one of “a” and “PP1144” (mixture ratio 1:10 to 10: 1) (Composition A1226); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1145” (Composition ratio 1:10 to 10: 1) (Composition A1227); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1146” (mixture ratio 1:10 to 10: 1) (Composition A1227) “Composition A1228);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1147 ”(mixing ratio 1:10 to 10: 1) (Composition A1229); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP1148” (mixing ratio 1:10 to 10: 1) (composition A1230); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 1149” (mixture ratio 1:10 to 10: 1) (Composition A 1231); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1150” (mixture ratio 1 “Composition A1232);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1151 ”(mixing ratio 1:10 to 10: 1) (Composition A1233) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1152” (mixing ratio 1:10 to 10: 1) (Composition A 1234); “Any of Compounds AA1-BA1 to AK2688-BK1287 Or “PP1153” (mixture ratio 1:10 to 10: 1) (composition A1235); “any one of compounds AA1-BA1 to AK2688-BK1287 “Composition A1236” (composition A1236); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1155” (mixture ratio 1) "Composition A1237" (Composition A1237); "Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP1156" (mixing ratio 1:10 to 10: 1) (Composition A1238) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1157” (mixing ratio 1:10 to 10: 1) (Composition A1239); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1158” (mixture ratio 1:10 to 10: 1) (composition A1240); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1159” (mixture Ratio 1:10 to 10: 1) (Composition A 1241); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1160” (mixing ratio 1:10 10: 1) (Composition A 1242); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1161” (mixing ratio 1:10 to 10: 1) (Composition A 1243); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1162” (mixture ratio 1:10 to 10: 1) (composition A1244); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1163” (mixture ratio 1:10 to 10: 1) (Composition A1245); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1164” (mixture ratio 1: 10 to 10: 1) (Composition A 1246); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1165” (mixing ratio 1:10 to 10: 1) (Composition A1247); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1166” (mixture ratio 1:10 to 10: 1) (Composition A1248); “Compound AA1-BA Any one of 1 to AK2688-BK1287 and a combination of “PP1167” (mixture ratio 1:10 to 10: 1) (composition A1249); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1168 "(mixture ratio 1:10 to 10: 1) (Composition A1250);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1169 "(mixture ratio 1:10 to 10: 1) (Composition A 1251); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 1170” (mixing ratio 1:10 to 10: 1) (Composition A 1252); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1171” (mixture ratio 1:10 to 10: 1) (composition A1253); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1172” (mixture ratio 1:10 to 10: 1) (composition A1254); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1173 (Combination ratio 1:10 to 10: 1) (composition A1255); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1174” (mixture ratio 1:10 to 10: 1) (Composition A1256); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1175” (mixing ratio 1:10 to 10: 1) (Composition A1257); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1176” (mixing ratio 1:10 to 10: 1) (composition A1258); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1177 (mixing ratio 1:10 to 10: 1) (Composition A 1259); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1178” (mixing ratio 1:10 to 10: 1) (Composition A 1260); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1179” (mixing ratio 1:10
“Composition A1261);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1180 ”(mixing ratio 1:10 to 10: 1) (Composition A1262); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP1181” (mixing ratio 1:10 to 10: 1) (composition A 1263); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP1182” (mixture ratio 1:10 to 10: 1) (Composition A1264); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1183” (mixture ratio 1 “Composition A1265);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1184 ”(mixing ratio 1:10 to 10: 1) (Composition A1266) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1185" (mixing ratio 1:10 to 10: 1) (Composition A1267); "Compound AA1-B “Any one of A1 to AK2688-BK1287” and “PP1186” (mixing ratio 1:10 to 10: 1) (composition A1268); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1187 (mixing ratio 1:10 to 10: 1) (Composition A 1269); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1188” (mixing ratio 1:10 to 10: 1) (Composition A1270); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1189” (mixing ratio 1:10 to 10: 1) (Composition A1271); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1190” (mixture ratio 1:10 to 10: 1) (composition A1272); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1191” (mixture ratio 1:10 to 10: 1) (composition A1273); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1192 (Combination ratio 1:10 to 10: 1) (composition A1274); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1193” (mixture ratio 1:10 to 10: 1) (Composition A1275); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1194” (mixing ratio 1:10 to 10: 1) (Composition A1276); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1195” (mixing ratio 1:10 to 10: 1) (composition A1277); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition A1278” in combination with “PP1196” (composition A1278); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1197” (mixture ratio 1:10 to 10: 1) (Composition A1279); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1198” (mixing ratio 1:10 to 10: 1 (Composition A 1280); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1199” (mixing ratio 1:10 to 10: 1) (Composition A 1281); “Compound AA1 to BA1-1” “Any one of AK2688-BK1287” and “PP1200” (mixture ratio 1:10 to 10: 1) (composition A 1282); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1201” (Combination ratio 1:10 to 10: 1) (composition A1283); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1202” (mixture ratio 1:10 to 10: 1) (Composition A1284); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1203” (mixing ratio 1:10 to 10: 1) (Composition A1285); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP1204” (mixing ratio 1:10 to 10: 1) (composition A1286); “compound AA1-BA1 to AK2688-BK128 A combination of “one of 7” and “PP 1205” (mixture ratio 1:10 to 10: 1) (composition A1287); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1206” Combination (mixture ratio 1:10 to 10: 1) (Composition A1288); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1207" (mixture ratio 1:10 to 10: 1) (Composition A1289); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1208” in combination (mixing ratio 1:10 to 10: 1) (Composition A1290); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP1209” (mixture ratio 1:10 to 10: 1) (composition A1291); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1210” (Combination ratio 1:10 to 10: 1) (composition A1292); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP1211” (Composition ratio 1:10 to 10: 1) (Composition A1293); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1212” (mixture ratio 1:10 to 10: 1) (Composition A 1293) “Composition A1294);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1213 ”(mixing ratio 1:10 to 10: 1) (Composition A1295);“ Compounds AA1 to BA1 to AK2688 Any one of “-BK1287” and “PP1214” (mixture ratio 1:10 to 10: 1) (composition A1296); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1215” Combination (mixture ratio 1:10 to 10: 1) (composition A 1297); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1216” (mixture ratio 1:10 to 10: 1 (Composition A1298); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1217” (mixing ratio 1:10 to 10: 1) (Composition A129) 9); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1218” (mixing ratio 1:10 to 10: 1) (Composition A1300); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the above and “PP1219” (mixture ratio 1:10 to 10: 1) (Composition A 1301); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1220” (Composition ratio 1:10 to 10: 1) (Composition A1302); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1221” (mixture ratio 1:10 to 10: 1) (Composition A 1302) “Composition A1303);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1222 ”(mixing ratio 1:10 to 10: 1) (Composition A1304);“ Compounds AA1-BA1 to AK2688 -Any one of BK1287 'and' PP1223 '(mixture ratio 1:10 to 10: 1) (composition A1305); any of compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1224” (mixture ratio 1:10 to 10: 1) (composition A1306); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1225” (mixture “Composition A1307);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1226 ”(mixing ratio 1:10 to 10: 1) (Composition A1308) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1227” (mixing ratio 1:10 to 10: 1) (Composition A1309); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the above and “PP1228” (mixture ratio 1:10 to 10: 1) (Composition A1310); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1229” (Composition ratio 1:10 to 10: 1) (Composition A1311); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1230” (Composition ratio 1 10 to 10: 1) (Composition A1312); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1231” (mixing ratio 1:10 to 10: 1) (Composition A1313); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1232” (mixing ratio 1:10 to 10: 1) (Composition A 1314); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP1233” (mixture ratio 1:10 to 10: 1) (Composition A 1315); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1234” (mixture ratio 1:10 to 10: 1) (Composition A 1316); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1235” (mixing ratio 1:10 to 10: 1) (Composition A1317 A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1236” (mixing ratio 1:10 to 10: 1) (composition A 1318); “compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1237” (mixture ratio 1:10 to 10: 1) (composition A1319); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1238” (mixture ratio 1:10 to 10: 1) (Composition A1320); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1239” (mixture ratio 1: 10 to 10: 1) (Composition A 1321); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 1240” (mixing ratio 1:10 to 10: 1) (Composition A 1322); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1241” (mixing ratio 1:10 to 10: 1) (Composition A1323); “Compounds AA1-BA1 to AK2688-BK1287 “One” and “PP1242” (mixture ratio 1:10 to 10: 1) (composition A1324); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1243 "(mixture ratio 1:10 to 10: 1) (Composition A 1325);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1244 "(mixture ratio 1:10 to 10: 1) (Composition A1326); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1245” (mixing ratio 1:10 to 10: 1) (Composition A1327); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1246” (mixture ratio 1:10 to 10: 1) (composition A1328); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1247” (mixture ratio 1:10 to 10: 1) (Composition A1329); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1248” (mixture ratio 1: 10 to 10: 1) (Composition A 1330); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1249” (mixing ratio 1:10 to 10) 1) (Composition A1331); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1250” (mixing ratio 1:10 to 10: 1) (Composition A1332); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1251” (mixture ratio 1:10 to 10: 1) (composition A1333); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1252 (mixture ratio 1: 10 to 10: 1) (Composition A 1334); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 1253” (mixture ratio 1: 10 to 10: 1) (Composition A1335); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1254” (mixing ratio 1:10 to 10: 1) (Composition A1336); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1255” (mixture ratio 1:10 to 10: 1) (composition A1337); “compound AA1-BA1 to AK268” “Any one of 8-BK1287” and “PP1256” in combination (mixture ratio 1:10 to 10: 1) (composition A1338); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1257” (Combination ratio 1:10 to 10: 1) (composition A1339); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1258” (mixture ratio 1:10 to 10: 1) (Composition A1340); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1259” (mixing ratio 1:10 to 10: 1) (Composition A1341); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1260” (mixing ratio 1:10 to 10: 1) (composition A 1342); “any one of compounds AA1-BA1 to AK2688-BK1287” In combination with PP 1261 (mixture ratio 1:10 to 10: 1) (composition A 1343); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1262” Combination (mixing ratio 1:10 to 10: 1) (Composition A 1344); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1263” (mixing ratio 1:10 to 10: 1) (Composition A1345); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1264” (mixing ratio 1:10 to 10: 1) (Composition A1346); “Compound AA1 to BA1” “Any one of AK2688-BK1287” and “PP1265” in combination (mixture ratio 1:10 to 10: 1) (composition A 1347); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1266” (Combination ratio 1:10 to 10: 1) (composition A1348); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1267” (mixture ratio 1:10 to 10: 1) (Composition A1349); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1268” (mixing ratio 1:10 to 10
"Composition A1350";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1269" (mixing ratio 1:10 to 10: 1) (Composition A1351); "Compound AA1 -Any one of “BA1 to AK2688-BK1287” and “PP1270” (mixture ratio 1:10 to 10: 1) (composition A1352); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP1271” (mixture ratio 1:10 to 10: 1) (Composition A1353); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1272” (mixture ratio 1:10 “Composition A1354);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1273 ”(mixing ratio 1:10 to 10: 1) (Composition A1355); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP1274” (mixing ratio 1:10 to 10: 1) (composition A1356); “compound AA1 to BA1 to AK26 “Any one of 88-BK1287” and “PP1275” in combination (mixing ratio 1:10 to 10: 1) (composition A1357); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1276” (Combination ratio 1:10 to 10: 1) (composition A1358); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1277” (mixture ratio 1:10 to 10: 1) (Composition A1359); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1278” (mixing ratio 1:10 to 10: 1) (Composition A1360); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1279” (mixing ratio 1:10 to 10: 1) (composition A 1361); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition A 1362) with“ PP 1280 ”(composition ratio 1:10 to 10: 1);“ any one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1281 ” Combination (mixture ratio 1:10 to 10: 1) (Composition A1363); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1282” (mixture ratio 1:10 to 10: 1) (Composition A1364): A combination of “any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1283” (mixing ratio 1:10 to 10: 1) (Composition A1365); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP1284” (mixture ratio 1:10 to 10: 1) (composition A1366); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1285” (Combination ratio 1:10 to 10: 1) (composition A 1367); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1286” (mixture ratio 1:10 to 10: 1) (Composition A1368); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1287” (mixing ratio 1:10 to 10: 1) (combination A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1288” (mixing ratio 1:10 to 10: 1) (composition A1370); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1289” (mixture ratio 1:10 to 10: 1) (composition A1371); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1290” Combination (mixture ratio 1:10 to 10: 1) (Composition A1372); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1291" (mixture ratio 1:10 to 10: 1) (Composition A1373); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1292” (mixing ratio 1:10 to 10: 1) (Composition A1374); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP1293” (mixture ratio 1:10 to 10: 1) (Composition A1375); “Compound AA1-BA1 to AK2688-BK1287” Combination of “one piece” and “PP1294” (mixture ratio 1:10 to 10: 1) (composition A1376); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1295” Mixing ratio 1:10 to 10: 1) (Composition A1377); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1296" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1297” (mixture ratio 1:10 to 10: 1) (composition A 1379); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1298” (mixture ratio 1:10 to 10: 1) (composition A1380); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1299” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1381); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1300” “Composition A1382);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1301 ”(mixing ratio 1:10 to 10: 1) (Composition A1383); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1302” (mixing ratio 1:10 to 10: 1) (Composition A1384); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “combination of 1: 1 to 10: 1” (composition A1385) of “PP1303” (composition A1385); “combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1304” (Composition ratio 1:10 to 10: 1) (Composition A1386); “Any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP1305” (mixture ratio 1:10 to 10: 1) (Composition A1386) “Composition A1387);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1306 ”(mixing ratio 1:10 to 10: 1) (Composition A1388); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP1307” (mixture ratio 1:10 to 10: 1) (composition A1389); “any one of the compounds AA1-BA1 to AK2688-BK1287 And “PP 1308” (mixture ratio 1:10 to 10: 1) (Composition A1390); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1309” (mixture ratio 1 “Composition A1391);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1310 ”(mixing ratio 1:10 to 10: 1) (Composition A1392) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1311” (mixing ratio 1:10 to 10: 1) (Composition A1393); “Any of Compounds AA1-BA1 to AK2688-BK1287 Or “PP1312” (mixture ratio 1:10 to 10: 1) (composition A 1394); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP1313” (mixture ratio 1:10 to 10: 1) (Composition A1395); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1314” (mixture ratio 1: 10-10: 1) (Composition A1396); “Any one of Compounds AA1-BA1-AK2688-BK1287” and “PP1315” (mixing ratio 1: 10-10: 1) (Composition A1397); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1316” (mixing ratio 1:10 to 10: 1) (Composition A1398); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1317” (mixing ratio 1:10 to 10: 1) (Composition A1399); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1318” (mixing ratio 1:10 to 10: 1) (Composition A1400); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1319” (mixing ratio 1:10 10: 1) (Composition A 1401); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 1320” (mixing ratio 1:10 to 10: 1) (Composition A 1402); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1321” (mixture ratio 1:10 to 10: 1) (Composition A 1403); “any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP1322” (mixture ratio 1:10 to 10: 1) (Composition A1404); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1323” (mixture ratio 1: 10-10: 1) (Composition A1405); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1324” (mixing ratio 1:10 to 10: 1) (Composition A1406); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1325” (mixing ratio 1:10 to 10: 1) (Composition A1407); “Compound AA1 to BA1 ~ Any one of AK2688-BK1287 "and" PP1326 "(mixture ratio 1:10 to 10: 1) (Composition A1408);" any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1327 (Combination ratio 1:10 to 10: 1) (composition A1409); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1328” (mixture ratio 1:10 to 10) "Composition A1410";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 1329" (mixing ratio 1:10 to 10: 1) (Composition A1411); "Compound AA1 -Any one of “BA1 to AK2688-BK1287” and “PP1330” (mixing ratio 1:10 to 10: 1) (composition A1412); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with “PP1331” (mixture ratio 1:10 to 10: 1) (Composition A1413); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1332” (Combination ratio 1:10 to 10: 1) (composition A 1414); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1333” (mixture ratio 1:10 to 10: 1) (Composition A1415); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1334” (mixing ratio 1:10 to 10: 1) (Composition A1416); “Compound AA1- “Any one of BA1 to AK2688-BK1287” and “PP1335” (mixing ratio 1:10 to 10: 1) (composition A1417); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP1336 "(mixture ratio 1:10 to 10: 1) (Composition A1418);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1337 "(mixture ratio 1:10 to 10: 1) (Composition A1419); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1338” (mixing ratio 1:10 to 10: 1) “Composition A1420);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1339 ”(mixing ratio 1:10 to 10: 1) (Composition A1421);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP1340” (mixture ratio 1:10 to 10: 1) (composition A1422); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1341” Combination (mixture ratio 1:10 to 10: 1) (composition A1423); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1342” (mixture ratio 1:10 to 10: 1 (Composition A1424); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1343” (mixing ratio 1:10 to 10: 1) (Composition A1425); “Compound AA1-BA1” ~ Any one of AK2688-BK1287 "and" PP1344 "(mixture ratio 1:10 to 10: 1) (Composition A1426);" Compound AA1-BA1 to AK2688-BK1287 Combination of any one of them and “PP1345” (mixture ratio 1:10 to 10: 1) (Composition A1427); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1346” Mixing ratio 1:10 to 10: 1) (Composition A1428); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 1347" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1348” (mixing ratio 1:10 to 10: 1) (composition A1430); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1349” (mixture ratio 1:10 to 10: 1) (composition A1431); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1350” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1432); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1351" Mixing ratio 1:10 to 10: 1) (Composition A 1433); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1352" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1353” (mixing ratio 1:10 to 10: 1) (composition A1435); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1354” (mixture ratio 1:10 to 10: 1) (composition A1436); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1355” Combination (mixture ratio 1:10 to 10: 1) (Composition A1437); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1356" (mixture ratio 1:10 to 10: 1) (Composition A1438); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1357” (mixing ratio 1:10 to 10: 1)
(Composition A1439); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1358” in combination (mixing ratio 1:10 to 10: 1) (Composition A1440); “Compound AA1 to BA1” “Any one of AK2688-BK1287” and “PP1359” (mixture ratio 1:10 to 10: 1) (composition A 1441); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1360” (Combination ratio 1:10 to 10: 1) (composition A 1442); “any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP1361” (mixture ratio 1:10 to 10: 1) (Composition A1443); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1362” (mixing ratio 1:10 to 10: 1) (Composition A1444); “Compound AA1− Any one of BA1 to AK2688-BK1287 and “PP1363” (mixture ratio 1:10 to 10: 1) (composition A1445); “compound AA1-BA1 to AK2688-BK1287 Any one of “a” and “PP1364” (mixture ratio 1:10 to 10: 1) (Composition A1446); “a combination of any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1365” (Composition ratio 1:10 to 10: 1) (Composition A1447); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1366” (mixture ratio 1:10 to 10: 1) (Composition A1447) “Composition A1448);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1367 ”(mixing ratio 1:10 to 10: 1) (Composition A1449);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP1368” (mixture ratio 1:10 to 10: 1) (composition A1450); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1369” Combination (mixture ratio 1:10 to 10: 1) (composition A1451); “combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP1370 ” Mixing ratio 1:10 to 10: 1) (Composition A1452); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1371" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1372” (mixing ratio 1:10 to 10: 1) (composition A1454); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1373” (mixture ratio 1:10 to 10: 1) (composition A1455); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1374” Combination (mixture ratio 1:10 to 10: 1) (Composition A1456); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1375" (mixture ratio 1:10 to 10: 1) (Composition A1457); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1376” (mixing ratio 1:10 to 10: 1) (Composition A1458 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1377" (mixing ratio 1:10 to 10: 1) (Composition A1459); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and “PP1378” (mixture ratio 1:10 to 10: 1) (Composition A 1460); Combination of “any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1379” (Composition A1460) Mixing ratio 1:10 to 10: 1) (Composition A 1461); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 1380" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1381” (mixing ratio 1:10 to 10: 1) (composition A1463); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1382” (mixture ratio 1:10 to 10: 1) (composition A1464); “any of compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP1383” (mixture ratio 1:10 to 10: 1) (composition A1465); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1384” (mixture "Composition A1466";"Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1385" (mixing ratio 1:10 to 10: 1) (Composition A1467) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1386” (mixture ratio 1:10 to 10: 1) (Composition A1468); “Compounds AA1-BA1 to AK2688-BK1287 Any one of “a” and “PP1387” (mixture ratio 1:10 to 10: 1) (Composition A1469); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1388” (Composition ratio 1:10 to 10: 1) (Composition A1470); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1389” (Composition ratio 1: 10 to 10: 1) (Composition A 1471); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 1390” (mixing ratio 1: 10 to 10: 1) (Composition A 1472); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1391” (mixing ratio 1:10 to 10: 1) (Composition A1473); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “One” and “PP1392” (mixture ratio 1:10 to 10: 1) (Composition A1474); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1393” (mixture ratio 1:10 to 10: 1) (Composition A1475); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1394” (mixing ratio 1:10 to 10: 1) (Composition A1476 A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1395” (mixing ratio 1:10 to 10: 1) (composition A1477); “compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1396” (mixture ratio 1:10 to 10: 1) (composition A1478); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1397” (mixture ratio 1:10 to 10: 1) (Composition A1479); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1398” (mixture ratio 1: 10-10: 1) (Composition A1480); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1399” (mixing ratio 1:10 to 10: 1) (Composition A1481); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1400” (mixing ratio 1:10 to 10: 1) (Composition A1482); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP 1401” (mixture ratio 1:10 to 10: 1) (composition A 1483); “any one of compounds AA1-BA1 to AK2688-BK1287” and “P Combination with P1402 (mixture ratio 1:10 to 10: 1) (Composition A1484); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1403” (mixture ratio 1:10 to 10: 1) (Composition A1485); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 1404” (mixing ratio 1:10 to 10: 1) (Composition A1486); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1405” (mixture ratio 1:10 to 10: 1) (composition A1487); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1406” (mixture ratio 1:10 to 10: 1) (Composition A1488); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1407” (mixture ratio 1: 10 to 10: 1) (Composition A 1489); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1408” (mixing ratio 1:10 to 10) 1) (Composition A1490); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP1409” (mixing ratio 1:10 to 10: 1) (Composition A1491); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1410” (mixture ratio 1:10 to 10: 1) (composition A1492); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1411 "(mixing ratio 1:10 to 10: 1) (Composition A 1493);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1412 "(mixing ratio 1:10 to 10) 10: 1) (Composition A1494); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1413” (mixing ratio 1:10 to 10: 1) (Composition A1495); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1414” (mixture ratio 1:10 to 10: 1) (composition A1496); “compound AA1-BA1 to AK2688 Any one of “-BK1287” and “PP1415” (mixture ratio 1:10 to 10: 1) (composition A1497); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1416” Combination (mixture ratio 1:10 to 10: 1) (composition A1498); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1417” (mixture ratio 1:10 to 10: 1 (Composition A1499); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1418” (mixing ratio 1:10 to 10: 1) (Composition A1500); “Compound AA1-BA1” ~ Any one of AK2688-BK1287 and PP 1419 (mixture ratio 1:10 to 10: 1) (Composition A 1501); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1420 (Mixture ratio 1:10 to 10: 1) (Composition A1502); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1421” Combination (mixing ratio 1:10 to 10: 1) (Composition A 1503); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1422” (mixing ratio 1:10 to 10: 1) (Composition A1504); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1423” (mixing ratio 1:10 to 10: 1) (Composition A1505); “Compound AA1 to BA1” “Any one of AK2688-BK1287” and “PP1424” (mixture ratio 1:10 to 10: 1) (composition A1506); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1425” (Combination ratio 1:10 to 10: 1) (composition A1507); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1426” (mixture ratio 1:10 to 10: 1) (Composition A1508); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1427” (mixing ratio 1:10 to 10: 1) (composition A1509) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1428” (mixing ratio 1:10 to 10: 1) (Composition A1510); “Compounds AA1-BA1 to AK2688-BK1287 Any one of “a” and “PP1429” (mixture ratio 1:10 to 10: 1) (Composition A1511); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1430” (Composition ratio 1:10 to 10: 1) (Composition A1512); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1431” (mixture ratio 1:10 to 10: 1) "Composition A1513);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1432 "(mixing ratio 1:10 to 10: 1) (Composition A1514);" Compounds AA1-BA1 to AK2688 " Any one of “-BK1287” and “PP1433” (mixture ratio 1:10 to 10: 1) (composition A1515); “all of compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP 1434” (mixture ratio 1:10 to 10: 1) (composition A 1516); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1435” (mixture “Composition A1517);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1436 ”(mixing ratio 1:10 to 10: 1) (Composition A1518); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1437” (mixture ratio 1:10 to 10: 1) (Composition A1519); “Compounds AA1-BA1 to AK2688-BK1287 Any one of “a” and “PP1438” (mixture ratio 1:10 to 10: 1) (Composition A 1520); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1439” (Composition ratio 1:10 to 10: 1) (Composition A1521); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1440” 1:10 to 10: 1) (Composition A1522); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1441” (mixing ratio 1:10 to 10: 1) (Composition A1523) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1442" (mixing ratio 1:10 to 10: 1) (Composition A1524); "Compounds AA1-BA1 to AK2688-BK1287" Combination of any one of them and PP 1443 (mixture ratio 1:10 to 10: 1) (Composition A1525); Combination of any one of Compounds AA1-BA1 to AK2688-BK1287 and PP1444 Mixing ratio 1:10 to 10: 1) (Composition A1526); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1445" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1446” (mixing ratio 1:10 to 10: 1) (composition
A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1447” (mixing ratio 1:10 to 10: 1) (composition A1529); “compound AA1 to BA1 to AK2688” Any one of BK1287 and “PP1448” (mixture ratio 1:10 to 10: 1) (composition A1530); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1449” Combination (mixture ratio 1:10 to 10: 1) (Composition A1531); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 1450" (mixture ratio 1:10 to 10: 1) (Composition A1532); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1451” (mixing ratio 1:10 to 10: 1) (Composition A1533); “Compound AA1-BA1 “Any one of AK2688-BK1287” and “PP1452” (mixture ratio 1:10 to 10: 1) (composition A1534) (composition AA1-BA1 to AK2688-BK1287) Combination of “one piece” and “PP1453” (mixture ratio 1:10 to 10: 1) (composition A1535); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1454” Mixing ratio 1:10 to 10: 1) (Composition A1536); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1455" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1456” (mixing ratio 1:10 to 10: 1) (composition A1538); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1457” (mixture ratio 1:10 to 10: 1) (composition A1539); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1458” Combination (mixture ratio 1:10 to 10: 1) (Composition A1540); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1459” 1:10 to 10: 1) (Composition A1541); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 1460” (mixing ratio 1:10 to 10: 1) (Composition A1542) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1461" (mixing ratio 1:10 to 10: 1) (Composition A1543); "Compound AA1-BA1 to AK2688-BK1287" Combination of any one of them and “PP1462” (mixture ratio 1:10 to 10: 1) (Composition A1544); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1463” Mixing ratio 1:10 to 10: 1) (Composition A1545); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 1464" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1465” (mixing ratio 1:10 to 10: 1) (Composition A1547); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP1466” (mixing ratio 1:10 to 10: 1) (composition A1548); “any one of the compounds AA1-BA1 to AK2688-BK1287 “Composition A1549” (composition A1549); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1468” (mixture ratio 1) "Composition A1550";"Any one of Compounds AA1-BA1-AK2688-BK1287" and "PP1469" (mixing ratio 1:10 to 10: 1) (Composition A 1551) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1470” (mixing ratio 1:10 to 10: 1) (Composition A 1552); “Any of Compounds AA1-BA1 to AK2688-BK1287 Or “PP1471” (mixture ratio 1:10 to 10: 1) (composition A 1553); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP1472” (mixture ratio 1:10 to 10: 1) (Composition A1554); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1473” (mixture ratio 1: 10-10: 1) (Composition A1555); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1474” (mixing ratio 1:10 to 10: 1) (Composition A1556); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1475” (mixture ratio 1:10 to 10: 1) (Composition A1557); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one” and “PP1476” (mixture ratio 1:10 to 10: 1) (Composition A1558); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1477” (mixture ratio 1:10 to 10: 1) (Composition A 1559); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1478” (mixing ratio 1:10 to 10: 1) (Composition A1560); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1479” (mixing ratio 1:10 to 10: 1) (Composition A 1561); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1480” (mixture ratio 1:10 to 10: 1) (composition A1562); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP1481” (mixture ratio 1:10 to 10: 1) (Composition A 1563); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1482” (mixture ratio 1: 10 to 10: 1) (Composition A 1564); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1483” (mixing ratio 1:10 to 10: 1) (Composition A1565); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1484” (mixing ratio 1:10 to 10: 1) (Composition A1566); “Compound AA1 to BA1 “Any one of AK2688-BK1287” and “PP1485” (mixture ratio 1:10 to 10: 1) (composition A1567); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1486” (Combination ratio 1:10 to 10: 1) (composition A1568); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1487” (mixture ratio 1:10 to 10: 1) (Composition A1569); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1488” in combination (mixing ratio 1:10 to 10: 1) (Composition A1570); “Compound AA1− “Any one of BA1 to AK2688-BK1287” and “PP1489” (mixing ratio 1:10 to 10: 1) (composition A 1571); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination with PP 1490 "(mixture ratio 1:10 to 10: 1) (Composition A 1572);" any one of compounds AA1-BA1 to AK2688-BK1287 "and" PP1491 " Combination (mixture ratio 1:10 to 10: 1) (Composition A 1573); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1492” (mixture ratio 1:10 to 10: 1 (Composition A1574); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1493” (mixing ratio 1:10 to 10: 1) (Composition A1575); “Compound AA1-BA1” ~ Any one of AK2688-BK1287 "and" PP1494 "(mixture ratio 1:10 to 10: 1) (composition A1576);" any one of compounds AA1-BA1 to AK2688-BK1287 "and" PP1495 (Combination ratio 1:10 to 10: 1) (composition A1577); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1496” (mixture ratio 1:10 to 10) "Composition A1578";"Any one of Compounds AA1-BA1-AK2688-BK1287" in combination with "PP1497" (mixing ratio 1:10 to 10: 1) “Composition A1579);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1498 ”(mixing ratio 1:10 to 10: 1) (Composition A1580);“ Compounds AA1-BA1 to AK2688 Any one of “-BK1287” and “PP1499” (mixture ratio 1:10 to 10: 1) (composition A1581); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1500” Combination (mixture ratio 1:10 to 10: 1) (composition A1582); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1501” (mixture ratio 1:10 to 10: 1 "Composition A1583);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP1502 "(mixing ratio 1:10 to 10: 1) (Composition A1584);" Compound AA1-BA1 " ~ Any one of AK2688-BK1287 "and" PP1503 "(mixture ratio 1:10 to 10: 1) (Composition A1585);" Compound AA1-BA1 to AK2688-BK1287 Combination of any one of them and PP1504 (mixture ratio 1:10 to 10: 1) (Composition A1586); Combination of any one of Compounds AA1-BA1 to AK2688-BK1287 and PP1505 Mixing ratio 1:10 to 10: 1) (Composition A1587); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1506" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1507” (mixing ratio 1:10 to 10: 1) (composition A1589); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1508” (mixing ratio 1:10 to 10: 1) (composition A1590); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1509” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1591); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1510” Mixing ratio 1:10 to 10: 1) (Composition A1592); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1511" (mixing ratio 1:10 to 10: 1) (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP1512” (mixing ratio 1:10 to 10: 1) (composition A1594); “compound AA1 to BA1 to AK2688” A combination of “one of BK1287” and “PP1513” (mixing ratio 1:10 to 10: 1) (composition A1595); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1514” Combination (mixture ratio 1:10 to 10: 1) (Composition A 1596); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP1515" (mixture ratio 1:10 to 10: 1) (Composition A1597); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1516” (mixing ratio 1:10 to 10: 1) (Composition A 1598) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1517” (mixing ratio 1:10 to 10: 1) (Composition A1599); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one” and “PP 1518” (mixture ratio 1:10 to 10: 1) (composition A1600); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1519” (mixture “Composition A 1601);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1520 ”(mixing ratio 1:10 to 10: 1) (Composition A 1602); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1521” (mixing ratio 1:10 to 10: 1) (Composition A1603); “Compounds AA1-BA1 to AK2688-BK1287 Any one of the following: “a combination of 1:10 to 10: 1” (composition A1604) of “PP1522” (composition A1604); “any one of compounds AA1-BA1 to AK2688-BK1287 Combinations of One "and" PP1523 "(mixing ratio 1: 10 to 10: 1) (composition A1605);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP145” (Composition B1); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” Combination with “PP133” (Composition B2); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP134” (Composition B3); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP10” and “PP132” (composition B4); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP140” “Composition B5);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP10 ”and“ PP138 ”(Composition B6);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP10” and “PP135” (Composition B7); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP136” (Composition B8); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP10” and “PP196” (Composition B9); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” Combination with “PP139” (Composition B10); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP169” (Composition B11); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP10” and “PP168” (composition B12); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP172” “Composition B13);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP10 ”and“ PP179 ”(Composition B14);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP10” and “PP180” (Composition B15); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP206” (Composition B1 6) “combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP10 ”and“ PP259 ”(composition B17);“ any one of compounds AA1-BA1 to AK2688-BK1287 ” A combination of PP10 "and" PP256 "(Composition B18);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and a combination of" PP10 "and" PP200 "(Composition B19);" Compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP10” and “PP204” (composition B20); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP203” (Composition B21); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP205” (Composition B22); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP10” and “PP267” (composition B23); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP264” (combination “Composition B24);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP10 ”and“ PP49 ”(Composition B25);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP10” and “PP87” (Composition B26); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP208” (Composition B27); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP10” and “PP207” (composition B28); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP4” (Composition B29); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP2” (Composition B30); “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one of compounds”, “PP10” and “PP3” (composition B31); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP1” A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP8” (composition B33); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP10” and “PP180” (Composition B34); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP10” and “PP193” (Composition B35); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP10” and “PP187” (composition B36); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP260” (Composition B37); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP10” and “PP197” (Composition B38); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP9” and “PP145” (Composition B39); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP133” “Compound B40);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP9 ”and“ PP134 ”(Composition B41);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP9” and “PP132” (Composition B42); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP140” (Composition B43); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP9” and “PP138” (composition B44); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP135” (Composition B45); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP136” (Composition B46); “Compound AA1-BA1 to AK2688-BK1287 “One of the following”, “PP9” and “PP196” (composition B47); “one of the compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP139” “Compound B48);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP9 ”and“ PP207 ”(Composition B49);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP9” and “PP168” (Composition B50); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP172” (Composition B51); “Compound Any one of AA1-BA1 to AK2688-BK1287, and a combination of “PP9” and “PP179” (Composition B52); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9”, and “PP180” (Composition B53); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP206” (Composition B54); “Compound AA1-BA1 to AK2688-BK1287 Any one of “PP9” and “PP259” (Composition B55); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP256” (Composition B 55) “Composition B56);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP9 ”and“ PP200 ”(Composition B57);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP9” and “PP204” (composition B58); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP203” (composition B59); “compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP9” and “PP205” (Composition B60); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP267” (Composition B61); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP264” (Composition B62); “Compounds AA1-BA1 to AK2688-BK1287 Combination of “one of compounds”, “PP9” and “PP49” (composition B63); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP87” “Composition B64);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP9 ”and“ PP208 ”(Composition B65);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP9” and “PP207” (Composition B66); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP4” (Composition B67); “Compound Any one of AA1-BA1 to AK2688-BK1287 and a combination of “PP9” and “PP2” (Composition B 68); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP3” (Composition B69); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP9” and “PP1” (Composition B70); “Compounds AA1-BA1 to AK2688-BK1287” Of “any one of”, “PP9” and “PP8” (composition B71); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP175” (composition B72 "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP9" and "PP193" (Composition B 73); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP9" And “PP187” (Composition B74); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP9” and “PP260” (Composition B75); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP9” and “PP197” (composition B76); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP145” (Composition B 77); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP11” and “PP133” (Composition B78); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP11” and “PP134” (Composition B79); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP132” (Composition B80) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP11” and “PP140” (Composition B81); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “B. A combination of PP11 "and" PP138 "(Composition B82);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and a combination of" PP11 "and" PP135 "(Composition B83);" Compound AA1- " Any one of BA1 to AK2688-BK1287 and a combination of “PP11” and “PP136” (Composition B84); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP196” (Composition B85); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP139” (Composition B86); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP11” and “PP169” (composition B 87); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP168” “Compound B 88);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP11 ”and“ PP172 ”(Composition B 89);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP11” and “PP179” (Composition B90); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP180” (Composition B91); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP11” and “PP206” (Composition B 92); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP259” (Composition B93); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP256” (Composition B94); “Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP11” and “PP200” (Composition B 95); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, and a union of “PP11” and “PP204” “Composition B96);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP11 ”and“ PP203 ”(Composition B97);“ Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP11” and “PP205” (composition B98); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP267” (composition B99); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP11” and “PP264” (Composition B100); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP11” Combination with “PP49” (Composition B101); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP87” (Composition B102); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP11” and “PP208” (composition B103); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP207” (Composition B104); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP4” (Composition B105); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP11” and “PP2” (composition B106); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP3” (composition B107) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP11” and “PP1” (Composition B108); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “P
A combination of P11 "and" PP8 "(Composition B109);" Any one of Compounds AA1-BA1 to AK2688-BK1287 ", a combination of" PP11 "and" PP175 "(Composition B110); Any one of BA1 to AK2688-BK1287 and a combination of “PP11” and “PP193” (composition B111); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP187” (Composition B112); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP11” and “PP260” (Composition B113); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP11” and “PP197” (composition B114); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP20” and “PP145” (composition B115) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP20 ”and“ PP133 ”(composition B116);“ any one of compounds AA1-BA1 to AK2688-BK1287 ” And “PP20” and “PP134” (Composition B117); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP20” and “PP132” (Composition B118); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP20” and “PP140” (Composition B119); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP20” Combination with “PP138” (Composition B120); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP20” and “PP135” (Composition B121); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP20” and “PP136” (composition B122); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP20” and “PP196” “Composition B123);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP20 ”and“ PP139 ”(Composition B124);“ Compound AA1-BA1 to AK2688-BK1287 A combination of “PP20” and “PP169” (Composition B 125); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP20” and “PP168” (Composition B 126) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP20" and "PP172" (Composition B127); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP20"; And “PP 179” (Composition B 128); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 20” and “PP 180” (Composition B 129); “Compound AA 1-BA 1 ~ A combination of “any one of AK2688-BK1287”, “PP20” and “PP206” (composition B130); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP20” and “PP259” Combination (Composition B131); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP20” and “PP256” (Composition B132); “Compound AA1-BA1 to A A combination of “one of K2688-BK1287”, “PP20” and “PP200” (composition B 133); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP20” and “PP204” (Composition B134); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP20” and “PP203” (Composition B135); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B136);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP20 ”and“ PP267 ”(composition B137); Any one of the compounds AA1-BA1 to AK2688-BK1287 "," PP20 "and" PP264 "in combination (Composition B 138);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "," PP20 "and" “Composition B139);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP20 ”and“ PP87 ”(Composition B140);“ Compound Any one of AA1 -BA1 to AK2688-BK1287 "," PP20 "and" PP208 "(Composition B 141);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "," PP20 "and" “Composition B142);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP20 ”and“ PP4 ”(Composition B143);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP20” and “PP2” (composition B 144); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP20” and “PP3” (composition Substance B145); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP20” and “PP1” (composition B146); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP20” and “PP8” (Composition B 147); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP145” (Composition B 148); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP49” and “PP133” (composition B149); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “PP149” “Composition B150);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP49 ”and“ PP132 ”(Composition B151);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP49” and “PP140” (composition B152); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP138” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP135” (composition B154); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP49” and “PP136” (Composition B 155); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP196” (Composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “PP139” (composition B 157); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP49” and “PP169” (Composition B 158); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP168” (Composition B 159); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP49” and “PP172” (composition B 160); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “PP179” (Composition B161); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “PP180” (Composition B162); “Compound AA1-BA1 to AK2688-BK1287 “A combination of any one of“ PP49 ”and“ PP206 ”(composition B 163);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP49 ”and“ PP259 ” Combination (Composition B164); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “PP256” (Composition B165); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP49” and “PP200” (composition B166); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP204” (composition B167); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP49” and “PP203” (Composition B 168); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP49” Combination with “PP205” (Composition B169); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “PP267” (Composition B170); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP49” and “PP264” (composition B 171); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP49” and “P “Composition B172);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP49 ”and“ PP208 ”(Composition B173);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP49” and “PP207” (composition B 174); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP4” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP2” (composition B176); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP49” and “PP3” (Composition B 177); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP49” and “PP1” (Composition B 178); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP49” and “PP8” (composition B 179); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP87” Combination with “PP145” (Composition B 180); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP87” and “PP133” (Composition B181); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP87” and “PP134” (composition B 182); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP132” "Composition B183);" Any one of Compounds AA1-BA1-AK2688-BK1287 "," PP87 "and" PP140 "(Composition B184);" Any one of Compounds AA1-BA1-AK2688-BK1287 " And “PP87” and “PP138” (Composition B 185); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP135” (Composition B 186); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP87” and “PP136” (Composition B 187); “Any one of Compounds AA1-BA1 to AK2688-BK1287 And “PP 87” and “PP 196” (Composition B 188); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 87” and “PP 139” (Composition B 189); Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP87” and “PP169” (Composition B190); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP87” and “PP168” (Composition B191); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP87” and “PP172” (Composition B192); “Compounds AA1-BA1 to AK2688-BK1287” Of “any one of”, “PP87” and “PP179” (composition B 193); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP180” (composition B194) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP87” and “PP206” (Composition B 195); “Attachment of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one”, “PP 87” and “PP 259” (composition B 196); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 87” and “PP 256” (composition B 197) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP200” (Composition B198); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP87” And “PP204” (Composition B199); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP203” (Composition B200); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP87” and “PP205” (Composition B 201); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP87” and “PP267” (Composition B202); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP87” and “PP264” (Composition B203); “Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP87” and “PP208” (composition B 204); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP207” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP4” (composition B206); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP87” and “PP2” (Composition B 207); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP87” and “PP3” (Composition B 208); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP87” and “PP1” (composition B 209); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP87” and “PP8” (Composition B210); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP87” and “PP197” (Composition B211); “Compound AA1-BA1 to A Any one of K2688-BK1287, a combination of “PP179” and “PP145” (Composition B 212); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP179” and “PP133” (Composition B 213); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP179” and “PP134” (Composition B214); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “PP179” and “PP132” (composition B 215); “any one of compounds AA1-BA1 to AK2688-BK1287” and “P
“Combination of P179” and “PP140” (composition B216); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP179” and “PP138” (composition B217); “compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP179” and “PP135” (Composition B 218); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP179” and “PP136” (Composition B 219); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP179” and “PP196” (Composition B220); Any one of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP 179” and “PP 139” (composition B 221); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 179” and “PP 169” (composition B 222) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP179” and “PP168” in combination (Composition B 223); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of “one”, “PP179” and “PP172” (composition B224); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP179” and “PP206” (composition B225) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP179" and "PP259" (Composition B 226); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP179" And “PP200” (Composition B227); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP179” and “PP204” (Composition B228); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP179” and “PP203” (Composition B 229); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP179” and “PP205” (Composition B230); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP179” and “PP267” (Composition B231); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP179” and “PP264” (composition B 232); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP179” and “PP208” (Composition B233); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP179” and “PP207” (Composition B234); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B235);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP179 ”and“ PP2 ”(composition B236); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP179” and “PP3” (composition B 237); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP179” and “PP3” Combination with PP 1 "(Composition B 238);" Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 "," PP 179 "and" PP 8 "(Composition B 239); Any one of AA 1-BA 1 to AK 2688-BK 1287, “PP 179” and “PP 197” (composition B 240); “any one of compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 180” and “ “Composition B241);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP180 ”and“ PP133 ”(Composition B242);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP180” and “PP134” (composition B 243); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP132” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP140” (composition B245); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP180” and “PP138” (Composition B 246); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP135” “Composition B247);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP180 ”and“ PP136 ”(Composition B248);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP180” and “PP196” (Composition B249); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP139” (Composition B250); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP180” and “PP169” (Composition B 251); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP168” (Composition B252); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP172” (Composition B253); “Compound AA1-BA1 to AK2688-BK1287” “One of the compounds”, “PP180” and “PP206” (composition B 254); “one of the compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP259” (Composition B255); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP200” (Composition B256); “Compound AA1-BA1 to AK2688-BK1287 Any one of “PP180” and “PP204” (Composition B 257); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP203” (Composition B258); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP205” (Composition B259); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “B. A combination of PP 180 ′ ′ and “PP 267” (Composition B 260); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 180” and “PP 264” (Composition B 261); Any one of BA1 to AK2688-BK1287 and a combination of “PP180” and “PP208” (Composition B 262); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP180” and “PP207” (Composition B263); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP4” (Composition B264); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP180” and “PP2” (composition B 265); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP3” (Composition B266); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP180” and “PP1” (Composition B267); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP180” and “PP8” (Composition B 268); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP180” and “PP197” (Composition B269 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP206" and "PP145" (Composition B 270); Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP206” and “PP133” (composition B271); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP134” (composition B272); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP206” and “PP132” (Composition B 273); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP206” Combination with “PP 140” (Composition B 274); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 206” and “PP 138” (Composition B 275); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP206” and “PP135” (composition B 276); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP136” “Composition B 277);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”,“ PP 206 ”and“ PP 196 ”(Composition B 278);“ Compounds AA 1-BA 1 to AK 2 Any one of 688-BK1287 and a combination of “PP206” and “PP139” (Composition B 279); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP169” (Composition B 280); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP206” and “PP168” (Composition B 281); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B282);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP206 ”and“ PP259 ”(composition B283); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP206” and “PP200” (composition B 284); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP206” and “PP200” “Composition B 285”; “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 206” and “PP 203” (Composition B 286); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP206” and “PP205” (composition B 287); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP206” and “PP206” “Composition B 288”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 206” and “PP 264” (Composition B 289); “Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP206” and “PP208” (composition B 290); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP206” and “PP207” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP4” (composition B292); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP206” and “PP2” (Composition B 293); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP3” “Compound B 294)” “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP1” (Composition B 295); “Any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP206” and “PP8” (Composition B 296); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP206” and “PP197” (Composition B 297); Any one of AA1-BA1 to AK2688-BK1287 and “PP145” and “PP169” (composition B 298); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP145” and “PP168” (Composition B299); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP145” and “PP172” (Composition B300); “Compound AA1-BA1 to AK2688-BK1287” “One of the following”, “PP145” and “PP259” (composition B301); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP145” and “PP200” (Composition B302); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP145” and “PP204” (Composition B303); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP145” and “PP203” (composition B304); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP145” and “PP205” (composition B305) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP145" and "PP9" (Composition B 306); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP145" And “PP264” (Composition B307); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP145” and “PP208” (Composition B308); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP145” and “PP207” (Composition B 309); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “P “Combination of P145” and “PP4” (composition B310); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP145” and “PP2” (composition B311); “compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP145” and “PP3” (composition B312); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP145” and “PP1” (Composition B313); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP145” and “PP8” (Composition B314); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP133” and “PP169” (composition B 315); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP168” (composition B316) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP172” (Composition B 317); “Compound AA1-BA1 to AK2688-BK1287” And “PP133” and “PP259” (Composition B318); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP200” (Composition B319); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP133” and “PP204” (Composition B 320); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” Combination with “PP203” (composition B 321); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP
133 "and" PP205 "(Composition B322);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP133 "and" PP267 "(Composition B323);" Compound AA1- " Any one of BA1 to AK2688-BK1287 and a combination of “PP133” and “PP264” (composition B324); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP208” (Composition B325); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP207” (Composition B326); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP133” and “PP4” (composition B 327); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP2” (composition B 328) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” in combination with “PP3” (Composition B 329); “Any of Compounds AA1-BA1 to AK2688-BK1287 “Combination of“ one ”,“ PP133 ”and“ PP1 ”(composition B330);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP133 ”and“ PP8 ”(composition B331) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP132" and "PP169" (Composition B332); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP132" And “PP168” (Composition B333); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP172” (Composition B334); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP132” and “PP259” (Composition B 335); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP200” (Composition B336); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP204” (Composition B337); “Compound AA1-BA1 to AK2688-BK1 Any one of 287, “PP132” and “PP203” (composition B 338); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP205” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP267” (composition B340); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP132” and “PP264” (Composition B 341); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP208” (Composition B342); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP132” and “PP207” (composition B 343); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP4” (Composition B 344); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 132” and “PP 2” (Composition B 345); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP132” and “PP3” (composition B346); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP1” (Composition B347); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP8” (Composition B348); “Compound AA1-BA1 to AK2688-BK1287 Any one of “PP134” and “PP169” (Composition B 349); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP168” (Composition B350); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP172” (Composition B351); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “B. Combination of PP134 "and" PP259 "(Composition B 352);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "," PP134 "and" PP200 "(Composition B 353) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP204” (Composition B 354); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” And “PP203” (Composition B355); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP205” (Composition B356); “Compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP134” and “PP267” (composition B 357); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP264” Combination (Composition B 358); Any one of “Compounds AA1-BA1 to AK2688-BK1287”, “PP 134” and “PP 208” (Composition B 359); Any of “Compounds AA 1-BA 1 to AK 2688-BK 1287 A combination of “one”, “PP134” and “PP207” (composition B 360); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP4” “Composition B 361”; “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 134” and “PP 2” (Composition B 362); “Compounds AA 1-BA 1 to AK 2688-BK 1287” “Combination of one”, “PP134” and “PP3” (composition B363); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP1” (composition B364); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP134” and “PP8” (Composition B 365); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP140” Combination with “PP 169” (Composition B 366); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 140” and “PP 168” (Composition B 367); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP140” and “PP172” (composition B 368); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP “Composition B369);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP140 ”and“ PP200 ”(Composition B370);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP140” and “PP204” (composition B371); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP203” (composition Substance B372); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP140” and “PP205” (composition B 373); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP140” and “PP267” (Composition B 374); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP264” (Composition B375); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP140” and “PP208” (composition B 376); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP140” and “PP207” (Composition B 377); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP4” (Composition B378); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP140” and “PP2” (Composition B379); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP3” (Composition B380); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP1” (Composition B381); “Compounds AA1-BA1 to AK2688-BK1287” Any one of the above, “PP 140” and “PP 8” (Composition B 382);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP133” (Composition B 383); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” “Composition B 384”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 132” and “PP 139” (Composition B 385); “Compound AA 1-BA 1 to AK 2688 Any one of “-BK1287”, “PP132” and “PP140” (composition B 386); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP143” “Composition B 387);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP132 ”and“ PP155 ”(Composition B 388);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” , “PP132” and “PP156” (Composition B 389); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP164” (Composition B390); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP370” (Composition B391); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B392”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP380” (composition B393); “Any one of compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP387” (composition B394); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “ “Composition B395);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP132 ”and“ PP407 ”(Composition B396);“ Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP132” and “PP693” (Composition B397); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” “Composition B 398);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 132 ”and“ PP 695 ”(Composition B 399);“ Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP132” and “PP696” (composition B 400); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP134” (composition B41) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP133” and “PP139” (Composition B402); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP133” and “PP140” (Composition B403); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP143” (Composition B404); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP133” and “PP155” (composition B 405); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP133” and “PP156” (Composition B406); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP164” (Composition B407); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP133” and “PP370” (Composition B 408); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” “Composition B409);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP380 ”(Composition B410);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP133” and “PP387” (composition B411); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP394” “Composition B412);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP407 ”(Composition B413);“ Compounds AA1-BA1 to AK2688-BK1 “One of 287”, “the combination of“ PP133 ”and“ PP693 ”(composition B 414);“ the combination of any one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP694 ”(composition "Any one of Compounds AA1-BA1 to AK2688-BK1287" and a combination of "PP133" and "PP695" (Composition B 416); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP133” and “PP696” (Composition B417); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP139” (Composition B418); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP134” and “PP140” (composition B419); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP143” (Composition B420); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP155” (Composition B421); Any one of compounds AA1-BA1 to AK2688-BK1287 and “PP134” and “PP156” (composition B 422); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP134” “Composition B423);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP370 ”(Composition B424);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP134” and “PP373” (composition B 425); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP380” (composition "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP134" and "PP387" (Composition B 427); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP134” and “PP394” (Composition B 428); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP407” “Compound B429);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP693 ”(Composition B430);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP134” and “PP694” (Composition B 431); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP695” (Composition B432); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP134” and “PP696” (Composition B 433); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP140” (Composition B 434); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 139” and “PP 143” (Composition B 435); “Compound AA 1-BA 1 to AK 2688-BK1287” “One of the compounds”, “PP139” and “PP155” (composition B 436); “one of the compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP156” (Composition B 437); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 139” and “PP 164” (Composition B 438); “Compound AA 1-BA 1 to AK 2688-BK 1287 Any one of the combinations of “PP139” and “PP370” (Composition B 439); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP373” (Composition B440 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP139" and "PP380" (Composition B441); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP139" And “PP387” (Composition B 442); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP394” (Composition B 443); “Compound AA1-BA1” ~ A combination of one of “AK2688-BK1287”, “PP139” and “PP407” (Composition B 444); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP139” and “PP693” (Composition B445); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP694” (Composition B446); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP139” and “PP695” (composition B 447); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP696” (Composition B448); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP143” (Composition B449); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP140” and “PP155” (Composition B450); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP156” (Composition B451 "Any one of Compounds AA1-BA1-AK2688-BK1287", "PP140" and "PP164" (Composition B 452); "Compound AA1-BA1-AK2688-BK1287 Combination of “one or more”, “PP140” and “PP370” (composition B 453); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP373” (composition B454) "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP140" and "PP380" (Composition B 455); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP140" “Composition B456”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP394” (composition B457); “compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP140” and “PP407” (composition B 458); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP693” Combination (Composition B459); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP694” (Composition B460); “Compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP140” and “PP695” (Composition B 461); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP696” (Composition B462); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP155” (Composition B463); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP143” and “PP156” (composition B464); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP164” (composition B465) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP143" and "PP370" (Composition B 466); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP143" And “PP373” (Composition B 467); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP380” (Composition B4 68) “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP387” (Composition B 469); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Combination of PP143” and “PP394” (composition B470); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP407” (composition B471); “compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP143” and “PP693” (composition B 472); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP694” (Composition B 473); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 143” and “PP 695” (Composition B 474); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP143” and “PP696” (composition B 475); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP156” Combination (Composition B 476); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 155” and “PP 164” (Composition B 477); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP155” and “PP370” (composition B 478); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP373” (composition B 479); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP155” and “PP380” (Composition B 480); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” Combination with “PP 387” (Composition B 481); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 155” and “PP 394” (Composition B 482); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP155” and “PP407” (composition B483); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP15 5 "and" PP693 "(Composition B 484);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP 155 "and" PP694 "(Composition B 485);" Compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP155” and “PP695” (Composition B 486); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP696” A combination of (composition B487); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP15
6 "and" PP 164 "(Composition B 488);" Any one of Compounds AA1-BA1 to AK 2688-BK 1287 "and" PP 156 "and" PP 370 "(Composition B 489);" Compound AA 1- " Any one of BA1 to AK2688-BK1287 and a combination of “PP156” and “PP373” (Composition B 490); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP380” Combination of “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP387” (composition B492); any one of “compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP156” and “PP394” (composition B493); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP407” (composition B494) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP693” in combination (Composition B 495); “Any of Compounds AA1-BA1 to AK2688-BK1287 “Combination of one”, “PP156” and “PP694” (Composition B 496); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP695” (Composition B 497); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP156” and “PP696” (Composition B 498); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP164” “Composition B 499”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 164” and “PP 373” (Composition B 500); “Compound AA 1-BA 1 to AK 2688 Any one of “-BK1287”, “PP164” and “PP380” (composition B501); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP387” "Composition B502);" Any one of Compounds AA1-BA1-AK2688-BK1287 "," PP164 "and" PP394 "(Composition B503);" Compound AA1-BA1-AK " Any one of 2688-BK1287 and a combination of “PP164” and “PP407” (Composition B 504); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP693” (Composition B 505); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP164” and “PP694” (Composition B506); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B507);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP164 ”and“ PP696 ”(composition B508); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP370” and “PP373” (composition B 509); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP370” “Composition B510);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP370 ”and“ PP387 ”(Composition B511); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP394” (Composition B512); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370” Combination with “PP 407” (Composition B 513); “Any one of Compounds AA1-BA 1-AK 2688-BK 1287”, “PP 370” and “PP 693” (Composition B 514); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP370” and “PP694” (composition B515); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP370” and “PP695” “Composition B516);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP370 ”and“ PP696 ”(Composition B517);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP 373” and “PP 380” (Composition B 518); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 387” (Composition B519); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP373” and “PP394” (Composition B520); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B521);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP373 ”and“ PP693 ”(composition B522); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP373” and “PP694” (composition B 523); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “ “Composition B 524”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 696” (Composition B 525); “Compound AA 1-BA 1 to AK 2688- Any one of BK1287, a combination of “PP380” and “PP387” (Composition B 526); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380” “Composition B 527”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 380” and “PP 407” (Composition B 528); “Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP380” and “PP693” (composition B529); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP694” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP695” (composition B 531); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP380” and “PP696” (Composition B532); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP394” (Composition B533); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP387” and “PP407” (composition B 534); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP 387” and “PP 693” (composition B 535); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 387” and “PP 694” (composition B 536); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP387” and “PP695” (Composition B 537); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP387” “Composition B538);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP394 ”and“ PP407 ”(Composition B539);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP394” and “PP693” (composition B 540); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP694” “Composition B 541);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP394 ”and“ PP695 ”(Composition B 542);“ Compound AA1-BA1 to AK2688-BK1 Combination of “one of 287”, “PP394” and “PP696” (composition B 543); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP693” (composition B44) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP694” (Composition B545); “Any one of Compounds AA1-BA1 to AK2688-BK1287” A combination of “PP407” and “PP695” (Composition B 546); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP696” (Composition B547); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP693” and “PP694” (composition B 548); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP695” (Composition B549); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP696” (Composition B550); Any one of AA 1-BA 1 to AK 2688-BK 1287, “PP 694” and “PP 695” (composition B 551); “any one of compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 694” and “PP “Composition B 552”; “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 695” and “PP 696” (Composition B 553);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP1” (Composition B 554); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” “Composition B 555”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 132” and “PP 168” (Composition B 556); “Compound AA 1-BA 1 to AK 2688 Any one of “-BK1287”, “PP132” and “PP169” (composition B 557); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP170” "Composition B558);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "," PP132 "and" PP172 "(Composition B559);" Any one of Compounds AA1-BA1 to AK2688-BK1287 " And “PP132” and “PP173” (Composition B 560); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP174” (Composition B 561); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP1” (Composition B 562); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B563”; “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP168” (composition B564); “composition B564”; “composition B564”; Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP133” and “PP169” (composition B 565); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP133”, and “Composition B566);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP172 ”(Composition B567);“ Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP133” and “PP173” (Composition B 568); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP “Composition B569);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP1 ”(Composition B570);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP134” and “PP167” (composition B 571); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP168” (composition Substance B572): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP134” and “PP169” (composition B 573); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP134” and “PP170” (Composition B 574); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP172” (Composition B575); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP134” and “PP173” (composition B 576); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP134” and “PP174” (Composition B577); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP1” (Composition B578); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP139” and “PP167” (composition B579); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP168” (Composition B580); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP169” (Composition B581); “Compound AA1-BA1 to AK2688-BK1287” Any one of “PP139” and “PP170” (Composition B 582); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP172” (Composition B583); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP173” (Composition B584); “Compound AA1-BA1 to AK2688-BK1287 Combination of “one or more”, “PP139” and “PP174” (composition B585); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP1” (composition B586) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP140" and "PP167" (Composition B 587); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP140" And “PP168” (Composition B 588); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 140” and “PP169” (Composition B 589); “Compound AA 1-BA 1 ~ A combination of “any one of AK2688-BK1287”, “PP140” and “PP170” (composition B 590); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP172” Combination (Composition B591); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP173” (Composition B592); “Compound AA1-BA Any one of 1 to AK2688-BK1287 and a combination of “PP140” and “PP174” (Composition B593); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP1” (Composition B 594); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 143” and “PP 167” (Composition B 595); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP143” and “PP168” (composition B596); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP169” (composition B 597) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP143" and "PP170" (Composition B 598); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP143" And “PP172” (Composition B599); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP173” (Composition B600 "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP143" and "PP174" (Composition B601); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP155" And “PP1” (Composition B602); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP167” (Composition B603); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP155” and “PP168” (Composition B 604); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP169” (Composition B 605); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP155” and “PP170” (Composition B 606); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP155” and “PP172” (composition B 607); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP173” “Composition B 608);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP155 ”and“ PP174 ”(Composition B 609);“ Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP156” and “PP1” (composition B610); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP167” (composition B611); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP156” and “PP168” (Composition B 612); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” Combination with “PP169” (Composition B 613); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP170” (Composition B614); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP156” and “PP172” (composition B 615); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP156” Combination with PP 173 "(Composition B 616);" Any one of Compounds AA1-BA1-AK2688-BK1287 "," PP 156 "and" PP 174 "(Composition B 617);" Compound AA 1-BA 1-AK 2688- A combination of “one of BK1287”, “PP164” and “PP1” (composition B 618); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP167” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP168” (composition B620); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP164” and “PP169” (Composition B 621); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP170” (Composition B 622); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP164” and “PP172” (composition B 623); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B624);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP164 ”and“ PP174 ”(composition B625); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP370” and “PP1” (composition B 626); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP370”, and “Composition B627);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP370 ”and“ PP168 ”(Composition B628);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP370” and “PP169” (Composition B629); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370” and “PP170” (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP172” (composition B631); “compound AA1-BA1 to AK2688-BK1287”; Combination of any one of “PP370” and “PP173” (Composition B 632); Combination of “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP174” (Composition B 633 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 373" and "PP 1" (Composition B 634); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP 373 “Composition B635);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP373 ”and“ PP168 ”(composition B636),“ compound AA1-BA1 ” ~ A combination of “any one of AK2688-BK1287”, “PP373” and “PP169” (composition B 637); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP170” Combination (Composition B 638); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 172” (Composition B 639); “Compound AA Any one of 1-BA1 to AK2688-BK1287 and a combination of “PP373” and “PP173” (Composition B 640); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP174” (Composition B641); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP1” (Composition B642); “Compound AA1-BA1 to AK2688-BK1287” Of “any one of”, “PP380” and “PP167” (composition B 643); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP168” (composition B644) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP380” and “PP169” (Composition B645); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “B. “Combination of PP380” and “PP170” (composition B646); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP172” (composition B6) 47) “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP173” (Composition B648); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Combination of PP 380” and “PP 174” (composition B 649); “one of compounds AA1-BA1 to AK 2688-BK 1287”, “PP 387” and “PP 1” (composition B 650); “compound AA 1− Any one of BA1 to AK2688-BK1287 and a combination of “PP387” and “PP167” (Composition B 651); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP168” Combination of “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP169” (composition B653); any one of “compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP387” and “PP170” (composition B 654); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP172” Combination (Composition B655); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP173” (Composition B656); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP387” and “PP174” (composition B 657); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP1” (composition B658); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP394” and “PP167” (Composition B659); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394” Combination with “PP168” (Composition B 660); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP394” and “PP169” (Composition B 661); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP394” and “PP170” (composition B662); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” And “PP172” (Composition B663); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP394” and “PP173” (Composition B664); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP394” and “PP174” (Composition B 665); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP1” (Composition B666); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP167” (Composition B667); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B668);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP407 ”and“ PP169 ”(composition B669);“ composition B669 ”;“ composition B669 ”; Any one of the compounds AA1-BA1 to AK2688-BK1287, “PP407” and “PP170” (composition B 670); “any one of the compounds AA1-BA1 to AK2688-BK1287” And “PP 407” and “PP 172” (Composition B 671); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 407” and “PP 173” (Composition B 672); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP174” (Composition B 673); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” Combination with “PP1” (Composition B 674); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP167” (Composition B 675); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP693” and “PP168” (composition B 676); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP169” “Composition B677);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP693 ”and“ PP170 ”(Composition B678);“ Compound AA1-BA1 to AK2688-BK1 "One of 287", a combination of "PP693" and "PP172" (composition B 679); a combination of "any one of compounds AA1-BA1 to AK2688-BK1287", "PP693" and "PP173" (composition Substance B 680); “any one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP693” and “PP174” (composition B 681); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP694” and “PP1” (Composition B 682); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP694” and “PP167” (Composition B683); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP694” and “PP168” (composition B 684); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP169” (Composition B 685); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP170” (Composition B 686); Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP694” and “PP172” (Composition B687); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP173” (Composition B688); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP174” (Composition B689); “Compound AA1-BA1 to AK2688-BK1287” Of “any one of”, “PP 695” and “PP 1” (composition B 690); “one of compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 695” and “PP 167” (composition B691); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP168” in combination (composition B692); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition of PP 695” and “PP 169” (Composition B 693); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 695” and “PP 170” (Composition B694); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP695” and “PP172” (Composition B695); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Combination of PP 695” and “PP 173” (composition B 696); “any one of compounds AA1-BA1 to AK 2688-BK 1287” and “PP 695” and “PP 174” (composition B 697); Any one of BA1 to AK2688-BK1287 and a combination of “PP696” and “PP1” (composition B698); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP167” (Composition B699); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP168” (Composition B700); Any one of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP696” and “PP169” (composition B 701); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP170” Combination (Composition B702); Any one of “Compounds AA1-BA1 to AK2688-BK1287” and “PP696” and “PP172” (Composition B703); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP696” and “PP173” (composition B704); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP174” (composition B705);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP4” (Composition B 706); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” “Composition B 707);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 132 ”and“ PP 205 ”(Composition B 708);“ Compound AA 1-BA 1 to AK 2688 Any one of “-BK1287”, “PP132” and “PP220” (composition B 709); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP221” “Composition B710);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP132 ”and“ PP691 ”(Composition B711);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP132” and “PP202” (Composition B 712); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP212” (Composition B 713); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP263” (Composition B714); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B715);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP132 ”and“ PP204 ”(composition B716); Any one of the compounds AA1-BA1 to AK2688-BK1287 and the combination of “PP132” and “PP201” (composition B 717); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “ “Composition B 718”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 132” and “PP 430” (Composition B 719); “Compound AA 1-BA 1 to AK 2688- "Any one of BK1287", a combination of "PP132" and "PP442" (Composition B 720); "Any one of Compounds AA1-BA1-AK2688-BK1287", "PP132" and " “Composition B 721”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 132” and “PP 702” (Composition B 722); “Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP132” and “PP703” (composition B 723); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP277” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP277-1” (composition B 725); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B726);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP219 ”(composition B727); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP133” and “PP205” (composition B 728); “any one of the compounds AA1-BA1 to AK2688-BK1287” And “PP133” and “PP220” (Composition B 729); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP221” (Composition B730); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP133” and “PP691” (Composition B 731); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” Combination with “PP 202” (Composition B 732); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 133” and “PP 212” (Composition B 733); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP133” and “PP263” (composition B734); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP203” “Composition B735);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP204 ”(Composition B736);“ Compound AA1-BA1 to AK2688-B Combination of “one of K1287”, “PP133” and “PP201” (composition B 737); “combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP429” (composition B738) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP133” and “PP430” (Composition B739); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP133” and “PP442” (Composition B 740); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP701” (Composition B 741); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP133” and “PP702” (composition B 742); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP703” (Composition B 743); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 133” and “PP 277” (Composition B 744); Any one of the compounds AA1-BA1 to AK2688-BK1287 and the combination of “PP133” and “PP277-1” (Composition B 745); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134 And “PP4” (Composition B746); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP219” (Composition B747); “Compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP134” and “PP205” (composition B 748); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP220” Combination (Composition B 749); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 134” and “PP 221” (Composition B 750); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “One”, “PP134” and “PP691” (Composition B 751); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP202” (Composition B 752): “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP134” and “PP212” (Composition B753); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B754);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP203 ”(composition B755); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP134” and “PP204” (Composition B 756); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP204” “Composition B757);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP429 ”(Composition B758);“ Compound AA1-BA1 to AK2688- "Any one of BK1287", a combination of "PP134" and "PP430" (Composition B759); "Any one of Compounds AA1-BA1-AK2688-BK1287", "PP134" and " “Composition B760);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP701 ”(Composition B761);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP134” and “PP702” (composition B 762); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP703” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP277” (composition B764); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP134” and “PP277-1” (Composition B 765); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP4” (Composition B766); Any one of the compounds AA1-BA1 to AK2688-BK1287, “PP139” and “PP219” (composition B 767); “any one of the compounds AA1-BA1 to AK2688-BK1287” And “PP139” and “PP205” (Composition B 768); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP220” (Composition B769); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP139” and “PP221” (Composition B 770); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” “Composition B771);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP139 ”and“ PP202 ”(Composition B772);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP139” and “PP212” (composition B 773); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP263” “Composition B774);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP139 ”and“ PP203 ”(Composition B775);“ Compound AA1-BA1 to AK2688-B Combination of “one of K1287”, “PP139” and “PP204” (Composition B 776); “Composition of any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP201” (Composition Substance B777); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP139” and “PP429” (composition B778); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP139” and “PP430” (Composition B779); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP442” (Composition B780); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP139” and “PP701” (composition B 781); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP702” (Composition B 782); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 139” and “PP 703” (Composition B 783); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP139” and “PP277” (composition B784); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP139” Combination with “PP 277-1” (Composition B 785); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 140” and “PP 4” (Composition B 786); “Compound AA 1-BA 1 ~ A combination of “any one of AK2688-BK1287”, “PP140” and “PP219” (composition B 787); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP205” Combination (Composition B 788); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP220” (Composition B 789); Any one of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “One”, “PP140” and “PP221” (Composition B 790); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP691” (Composition B 791); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP140” and “PP202” (Composition B 792); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B793);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP140 ”and“ PP263 ”(composition B794); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP140” and “PP203” (composition B795); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP140”, and “PP140” “Composition B796);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP140 ”and“ PP201 ”(Composition B797);“ Compound AA1-BA1 to AK2688- "Any one of BK1287", a combination of "PP140" and "PP429" (Composition B798); "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP140" and " Combination with PP 430 "(Composition B 799);" Any one of Compounds AA1-BA1-AK2688-BK1287 "," PP 140 "and" PP 442 "(Composition B 800);" Compound AA 1-BA 1-AK 2688- A combination of “one of BK1287”, “PP140” and “PP701” (Composition B 801); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP702” (Composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP703” (composition B 803); “any one of compounds AA1-BA1 to AK2688-BK1287” A combination of “PP140” and “PP277” (Composition B 804); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP277-1” (Composition B 805); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP143” and “PP4” (composition B 806); “any one of the compounds AA1-BA1 to AK2688-BK1287” And “PP 143” and “PP 219” (Composition B 807); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 143” and “PP 205” (Composition B 808); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP143” and “PP220” (Composition B 809); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” Combination with “PP 221” (Composition B 810); “Any one of Compounds AA1-BA1 to AK2688-BK1287”
And “PP143” and “PP691” (Composition B811); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP202” (Composition B812); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP143” and “PP212” (Composition B 813); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP263” (Composition B 814); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 143” and “PP 203” (Composition B 815); “Compounds AA1-BA1 to AK2688-BK1287” Of “one of compounds”, “PP143” and “PP204” (composition B 816); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP201” (composition B817); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP143” and “PP429” (Composition B 818); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP143” and “PP430” (Composition B 819); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP442” (Composition B820 “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP701” (Composition B 821); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” And “PP702” (Composition B822); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP703” (Composition B823); “Compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP143” and “PP277” (composition B 824); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP277-1” (Composition B 825); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 155” and “PP 4” (Composition B 826); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP155” and “PP219” (Composition B 827); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP205” (Composition B 828); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 155” and “PP 220” (Composition B 829); “Compound AA 1-BA 1-AK 2688-BK 1287 Any one of “PP155” and “PP221” (Composition B 830); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP691” (Composition B831); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP202” in combination (composition B 832); “any one of compounds AA1-BA1 to AK2688-BK1287” “Combination of PP 155” and “PP 212” (composition B 833); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 155” and “PP 263” (pair “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP203” (Composition B 835); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 155” and “PP 204” (Composition B 836); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 155” and “PP 201” (Composition B 837); Any one of “-BA1 to AK2688-BK1287” and “PP155” and “PP429” (Composition B 838); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP430” (Composition B839); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP442” (Composition B840); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP 155” and “PP 701” (Composition B 841); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 155” and “PP 702” (Composition B842); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP703” (Composition B843); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP155” and “PP277” (Composition B844); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP277-1” A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP4” (composition B 846); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP156” and “PP219” (Composition B 847); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP205” (Composition B848); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP156” and “PP220” (composition B849); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP156” and “PP221” (Composition B850); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP691” (Composition B851); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP156” and “PP202” (Composition B 852); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP212” (Composition B853); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP263” (Composition B854); “Compound AA1-BA1 to AK2688-BK1287” Any one of “PP156” and “PP203” (Composition B 855); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP204” (Composition B856); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP156” and “PP201” (Composition B 857); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP156” and “PP429” (Composition B 858); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP430” (Composition B859 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP156" and "PP442" (Composition B 860); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP156" And “PP 701” (Composition B 861); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 156” and “PP 702” (Composition B 862); “Compound AA 1-BA 1 ~ A combination of “one of AK2688-BK1287”, “PP156” and “PP703” (Composition B 863); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP277” Combination (Composition B864); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP277-1” (Composition B865); Any one of AA 1-BA 1 to AK 2688-BK 1287 and “PP 164” and “PP 4” (composition B 866); “any one of Compound AA 1-BA 1 to AK 2688-BK 1287”, “PP 164” and “PP4” “Composition B867);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP164 ”and“ PP205 ”(Composition B868);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP164” and “PP220” (composition B869); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP221” (composition Substance B 870): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP164” and “PP691” (composition B871); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP164” and “PP202” (Composition B 872); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP212” "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP164" and "PP263" (Composition B874); "Any one of Compounds AA1-BA1 to AK2688-BK1287" A combination of “PP164” and “PP203” (Composition B 875); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and a combination of “PP164” and “PP204” (Composition B 876); Any one of “-BA1 to AK2688-BK1287” and “PP164” and “PP201” (Composition B 877); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP164” and “PP429” (Composition B 878); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 164” and “PP 430” (Composition B 879); “Compounds AA 1-BA 1-AK 2688-BK 1287 “Any one”, a combination of “PP164” and “PP442” (composition B 880); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP164” and “PP701” (Composition B 881); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 164” and “PP 702” (Composition B 882); “Compound AA 1-BA 1-AK 2688-BK 1287 Combination of any one of “PP 164” and “PP 703” (Composition B 883); “Composition of any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 164” and “PP 277” (Composition B 884 "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP164" and "PP277-1" (Composition B885); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP370” and “PP4” (Composition B886); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP219” (Composition B887); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP370” and “PP205” (composition B 888); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP370” and “PP220” (Composition B889); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370” and “PP221” (Composition B890); “Compound Combination of any one of AA1-BA1 to AK2688-BK1287 with “PP370” and “PP691” (Composition B 891); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP202” (Composition B 892); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 370” and “PP 212” (Composition B 893); “Compound AA 1-BA 1 to AK 2688-BK1287” Any one of “PP370” and “PP263” (Composition B 894); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370” and “PP203” (Composition “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP204” (Composition B896); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP370” and “PP201” (Composition B 897); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370” and “PP429” (Composition B898 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP370" and "PP430" (Composition B 899); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP370". And “PP 442” (Composition B 900); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 370” and “PP 701” (Composition B 901); “Compound AA 1-BA 1 ~ A combination of “one of AK2688-BK1287”, “PP370” and “PP702” (Composition B 902); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP703” Combination (Composition B 903); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 370” and “PP 277” (Composition B 904); “Compound AA Any one of 1-BA1 to AK2688-BK1287, a combination of “PP370” and “PP277-1” (composition B 905); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP373” Combination with “PP4” (Composition B 906); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 373” and “PP 219” (Composition B 907); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP373” and “PP205” (composition B 908); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP373” and “PP220” Composition B 909); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 221” (Composition B 910); “Any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP 373” and “PP 691” (Composition B 911); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 373” and “PP 202” A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP373” and “PP212” (composition B 913); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 373” and “PP 263” (Composition B 914); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 373” and “PP 203” (Composition B 915); Any one of “-BA1 to AK2688-BK1287”, “PP 373” and “PP 204” in combination (Composition B 916)
"Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP373" and "PP201" (Composition B 917); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP373" And “PP 429” (Composition B 918); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 373” and “PP 430” (Composition B 919); “Compound AA 1-BA1 “Any one of AK2688-BK1287”, a combination of “PP373” and “PP442” (Composition B 920); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP701” (Composition B 921); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP373” and “PP702” (Composition B 922); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP 373” and “PP 703” (Composition B 923); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 277” (Composition B 924); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 277-1” (Composition B 925); “Compound AA 1-BA 1 to AK 2688-BK 1287 Any one of the combinations of “PP380” and “PP4” (Composition B 926); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP219” (Composition B 927) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP205” (Composition B 928); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380 And “PP220” (Composition B 929); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP221” (Composition B930); “Compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP380” and “PP691” (composition B 931); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP380 And “PP 202” (Composition B 932); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 380” and “PP 212” (Composition B 933); “Compound AA 1-BA 1 ~ A combination of one of “AK2688-BK1287”, “PP380” and “PP263” (Composition B 934); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP203” Combination (Composition B935); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP204” (Composition B936); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP380” and “PP201” (Composition B 937); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP429” (Composition B938); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP430” (Composition B939); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP380” and “PP442” (composition B940); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP380” and “PP701” (composition B941); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP380” and “PP702” (Composition B942); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380” “Composition B943);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP380 ”and“ PP277 ”(Composition B944);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP380” and “PP277-1” (composition B 945); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP4” Combination (Composition B 946); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 387” and “PP 219” (Composition B 947); “Compound AA 1-BA 1 “Any one of AK2688-BK1287”, a combination of “PP387” and “PP205” (composition B948); “a combination of any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP220” (Composition B 949): “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP387” and “PP221” (Composition B950); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B 951”; “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 387” and “PP 202” (Composition B 952); “Composition B 951”; Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP387” and “PP212” (composition B953); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP387” “Composition B954);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP387 ”and“ PP203 ”(Composition B955) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP387" and "PP204" (Composition B956); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP387" And “PP201” (Composition B 957); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 387” and “PP429” (Composition B 958); “Compound AA 1-BA1 Any one of AK2688-BK1287, a combination of “PP387” and “PP430” (Composition B 959); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP387” and “PP442” (Composition B 960); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP 387” and “PP 701” (Composition B 961); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP 387” and “PP 702” (Composition B 962); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 387” and “PP 703” “Composition B963);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP387 ”and“ PP277 ”(Composition B964);“ Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP387” and “PP277-1” (Composition B 965); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP4” (Composition B966 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP394" and "PP219" (Composition B 967); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP394" And “PP205” (Composition B968); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP220” (Composition B969); “Compound AA1-BA1” ~ Any one of “AK2688-BK1287”, a combination of “PP394” and “PP221” (Composition B 970); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394 “Composition B971);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP394 ”and“ PP202 ”(composition B972);“ compound AA1-BA1 ” ~ A combination of “one of AK2688-BK1287”, “PP394” and “PP212” (Composition B 973); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP394” and “PP263” Combination (Composition B 974); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP394” and “PP203” (Composition B 975); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP394” and “PP204” (Composition B976); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP201” (Composition B977); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP394” and “PP429” (Composition B 978); “Any of Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP394” and “PP430” (composition B979); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP442” (composition B980); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP394” and “PP701” (Composition B 981); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP394” “Composition B982);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP394 ”and“ PP703 ”(Composition B983);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP394” and “PP277” (composition B 984); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP394” and “PP277-1” Combination (Composition B985); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP4” (Composition B986); “Compound AA1-BA1 “Any one of AK2688-BK1287”, “a combination of“ PP407 ”and“ PP219 ”(composition B 987);“ a combination of any one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP407 ”and“ PP205 ” (Composition B 988); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP220” (Composition B 989); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B990);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP407 ”and“ PP691 ”(composition B991); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP407” and “PP202” (composition B 992); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP407” and Combination with PP 212 "(Composition B 993);" Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 "," PP 407 "and" PP 263 "(Composition B 994) "Any one of Compounds AA1-BA1 to AK2688-BK1287", a combination of "PP407" and "PP203" (Composition B 995); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP407" And “PP204” (Composition B996); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP201” (Composition B997); “Compound AA1-BA1 Any one of AK2688-BK1287, a combination of “PP407” and “PP429” (Composition B 998); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP430” (Composition B 999); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP442” (Composition B1000); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP 407” and “PP 701” (Composition B 1001); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 407” and “PP 702” Combination (Composition B1002); Any one of “Compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP703” (Composition B1003); “Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP407” and “PP277” (Composition B 1004); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP277-1” (Composition B 1005 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP693" and "PP4" (Composition B1006); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP693" “Composition B1007);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP693 ”and“ PP205 ”(composition B1008);“ compound AA1-BA1 ” ~ A combination of one of “AK2688-BK1287”, “PP693” and “PP220” (Composition B 1009); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP693” and “PP221” (Composition B1010); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP691” (Composition B1011); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP693” and “PP202” (composition B1012); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP212” (Composition B1013); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP263” (Composition B1014); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP693” and “PP203” (Composition B1015); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP204” (Composition B1016 A combination of “one of compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP201” (composition B1017); “compound AA1-BA1 to AK2688-BK” Combination of “one of 1287”, “PP693” and “PP429” (composition B1018); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP430” (composition Substance B1019): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP693” and “PP442” (composition B1020); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP693” and “PP701” (Composition B 1021); “Compounds AA1-BA1 to AK268
Any one of 8-BK1287, a combination of “PP693” and “PP702” (composition B 1022); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP703” (Composition B 1023); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP693” and “PP277” (Composition B 1024); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP693” and “PP277-1” (Composition B1025); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP694” and “PP4” (Composition B1026) "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP694" and "PP219" in combination (Composition B1027); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP694" And “PP205” (Composition B1028); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP220” (Composition B1 “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP221” (Composition B1030); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Combination of PP694” and “PP691” (composition B1031); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP694” and “PP202” (composition B1032); “compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP694” and “PP212” (Composition B 1033); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP263” (Composition B1034); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP203” (Composition B1035); Any of “Compounds AA1-BA1 to AK2688-BK1287” “Composition B1036);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP694 ”and“ PP201 ” (Composition B1037); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP429” (Composition B1038); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP694” and “PP430” (Composition B1039); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP694” and “PP442” (Composition B1040 "Any one of Compounds AA1-BA1 to AK2688-BK1287", a combination of "PP694" and "PP701" (Composition B1041); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP694". And “PP702” (Composition B1042); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP694” and “PP703” (Composition B1043); “Compound AA1-BA1” ~ A combination of one of “AK2688-BK1287”, “PP694” and “PP277” (Composition B1044); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP694” and “PP277-1” (Composition B1045); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP695” and “PP4” (Composition B1046) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP695” and “PP219” (Composition B1047); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP695 And “PP205” (Composition B1048); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP695” and “PP220” (Composition B1049); “Compound AA1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP695” and “PP221” (composition B1050); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP691” Combination (Composition B 1051); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 695” and “PP 202” (Composition B 1052); “Compound AA 1-BA 1 “Any one of AK2688-BK1287”, a combination of “PP695” and “PP212” (composition B1053); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP263” (Composition B1054); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP695” and “PP203” (Composition B1055); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1056);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP695 ”and“ PP201 ”(Composition B1057); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP695” and “PP429” (composition B1058); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP695” and Combination with PP 430 "(Composition B 1059);" Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 "," PP 695 "and" PP 44 2 "(Composition B1060); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP695” and “PP701” (composition B1061); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B1062) of“ PP 695 ”and“ PP 702 ”;“ Composition B 1063 ”of“ any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 695 ”and“ PP 703 ”(Compound B1063); Any one of BA1 to AK2688-BK1287, a combination of “PP695” and “PP277” (Composition B 1064); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP277-1 (Composition B 1065); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 696” and “PP 4” (Composition B 1066); “Compounds AA 1-BA 1 to AK 2688-BK 1287 Of “any one of” and “PP696” and “PP219” (composition B1067); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP696” “Composition B1068);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP696 ”and“ PP220 ”(Composition B1069);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP696” and “PP221” (composition B 1070); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP691” (composition Substance B1071); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP696” and “PP202” (composition B1072); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B 1073) of“ PP 696 ”and“ PP 212 ”; A combination of“ PP 696 ”and“ PP 26 3 ”with“ any one of Compounds AA1-BA1 to AK2688-BK1287 ”(Composition B 1074); Any one of “-BA1 to AK2688-BK1287”, “PP696” and “PP203” (composition B1075); any one of “compound AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP696” and “PP204” (composition B1076); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP696” and “PP201” (composition B1077); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP696” and “PP429” (Composition B1078); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP696” “Composition B1079);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP696 ”and“ PP442 ”(Composition B1080);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP696” and “PP701” (composition B1081); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP696” and “PP702” “Composition B1082);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP696 ”and“ PP703 ”(Composition B1083);“ Compound AA1-B Any one of A1 to AK2688-BK1287, a combination of “PP696” and “PP277” (composition B1084); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP696”, and “PP277-1 In combination with (composition B 1085);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP209” (Composition B1086); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” “Composition B1087);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP132 ”and“ PP257 ”(Composition B1088);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP132” and “PP258” (composition B1089); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP366” “Composition B1090);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP132 ”and“ PP250 ”(Composition B1091);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP132” and “PP251” (Composition B1092); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP252” Combination (Composition B1093); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP132” and “PP363” (Composition B1094); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP132” and “PP364” (composition B1095); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP132” and “PP2” (composition B1096); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP132” and “PP3” (Composition B1097); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP132” “Composition B1098);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP132 ”and“ PP1054 ”(Composition B1099);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287” and “PP132” and “PP1055” (composition B1100); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B1101) of“ PP 133 ”and“ PP 209 ”;“ Composition of any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP133 ”and“ PP256 ”(Composition B1102);“ Compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP133” and “PP257” (Composition B1103); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP258” (Composition B1104); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP366” (Composition B1105); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP133” and “PP250” (composition B1106); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP251” (composition B1107) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP133 ”and“ PP252 ”(composition B1108);“ compound AA1-BA1 to AK2688-BK128 7) of “one of 7”, “PP133” and “PP363” (composition B1109); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP364” (composition Substance B1110); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP133” and “PP2” in combination (composition B1111); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP133” and “PP3” (Composition B1112); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP1051” (Composition B1113); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP133” and “PP1054” (composition B1114); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP133” and “PP1055” (Composition B1115); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP209” (Composition B1116); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP134” and “PP256” (composition B1117); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP134” “Composition B1118);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP258 ”(Composition B1119);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP134” and “PP366” (composition B1120); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP134” and “PP250” (composition Substance B1121); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP251” in combination (composition B1122); “any one of compounds AA1-BA1 to AK2688-BK1287” A combination of “PP134” and “PP252” (composition B1123); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP134” and “PP363” “Composition B1124);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP134 ”and“ PP364 ”(Composition B1125);“ Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP134” and “PP2” (composition B1126); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP134” and “PP3” (composition B1127); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP134” and “PP1051” (Composition B1128); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP134” “Composition B1129” with “PP1054”; “Any one of Compounds AA1-BA1 to AK2688-BK1287” with “PP134” and “PP1055” (Composition B1130); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP139” and “PP209” (composition B 1131); “one of compounds AA1-BA1 to AK2688-BK1287” and “P “Composition B1132) of“ P139 ”and“ PP256 ”;“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP139 ”and“ PP257 ”(Composition B1133);“ Compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP139” and “PP258” (composition B1134); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP366” (Composition B1135); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP139” and “PP250” (Composition B1136); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP139” and “PP251” (composition B1137); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP252” (composition B1138) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP139 ”and“ PP363 ”(composition B1139);“ compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP139” and “PP364” (Composition B1140); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP139” and “PP2” (Composition B1141 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP139" and "PP3" (Composition B1142); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP139". “Composition B1143);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP139 ”and“ PP1054 ”(composition B1144);“ compound AA1-BA1 ” ~ A combination of “any one of AK2688-BK1287”, “PP139” and “PP1055” (composition B1145); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP209” Combination (Composition B1146); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP256” (Composition B1147); Any one of the compounds AA1-BA1 to AK2688-BK1287 and a combination of “PP140” and “PP257” (composition B1148); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP140” “Composition B1149);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP140 ”and“ PP366 ”(Composition B1150);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP140” and “PP250” (composition B 1151); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP140” and “PP251” “Composition B1152);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP140 ”and“ PP252 ”(Composition B1153);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP140” and “PP363” (Composition B1154); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP364” (Composition B1155); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP2” (Composition B1156); “Compound AA1-BA1 to AK2688-BK1287 “Composition B1157);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP140 ”and“ PP1051 ”(composition B1158); “Any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP1054” (composition B1159); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP140” and “PP140” “Composition B1160);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP143 ”and“ PP209 ”(Composition B1161);“ Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP143” and “PP256” (Composition B1162); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP14 3 "and" PP 257 "(Composition B1163);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP 143 "and" PP258 "(Composition B 1164);" Compound AA 1- " Any one of BA1 to AK2688-BK1287 and a combination of “PP143” and “PP366” (composition B1165); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP143”, and “PP250” (Composition B1166); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP251” (Composition B1167); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP143” and “PP252” (composition B1168); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP363” (composition B1169) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP364” (Composition B1170); “Compound AA1-BA1 to AK2688-BK1287 A combination of “PP143” and “PP2” (composition B1171); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP143” and “PP3” (composition B1172) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP143" and "PP1051" (Composition B1173); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP143" “Composition B1174”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP143” and “PP1055” (composition B1175); “compound AA1-BA1” ~ A combination of one of “AK2688-BK1287”, “PP155” and “PP209” (Composition B1176); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP256” Combination (Composition B1177); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP155” and “PP257” (Composition B1178); Any one of AA1 -BA1 to AK2688-BK1287 "," PP155 "and" PP258 "(Composition B1179);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "," PP155 "and" “Composition B1180);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP155 ”and“ PP250 ”(Composition B1181);“ Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP155” and “PP251” (Composition B1182); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP252” (Composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP363” (composition B1184); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP155” and “PP364” (Composition B1185); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP2” “Composition B1186);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP155 ”and“ PP3 ”(Composition B1187);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP155” and “PP1051” (Composition B1188); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP155” and “PP1054” (Composition B1189); “Compound Any one of AA1-BA1 to AK2688-BK1287 and "PP155"
“Composition B1190);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP156 ”and“ PP209 ”(composition B1191);“ compound AA1-BA1 ” ~ A combination of “any one of AK2688-BK1287”, “PP156” and “PP256” (composition B1192); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP257” Combination (Composition B 1193); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP258” (Composition B1194); Any one of “Compounds AA1-BA1 to AK2688-BK1287” “Combination of one”, “PP156” and “PP366” (composition B1195); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP250” (composition B1196); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP251” in combination (Composition B1197); “Compound AA1-BA1 to AK2688-BK1287 Combination of “one or more”, “PP156” and “PP252” (composition B1198); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP363” (composition B1199) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” and “PP364” (Composition B1200); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP156” “Composition B1201);“ any one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP156 ”and“ PP3 ”(composition B1202);“ compound AA1-BA1 ” ~ A combination of “one of AK2688-BK1287”, “PP156” and “PP1051” (Composition B 1203); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP156” and “PP1054” Combination (Composition B 1204); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 156” and “PP 1055” (Composition B 1205); “Compound Any one of AA1 -BA1 to AK2688-BK1287 "," PP164 "and" PP209 "(composition B1206);" any one of Compounds AA1 -BA1 to AK2688-BK1287 "," PP164 "and" PP1 " “Composition B 1207);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 164 ”and“ PP 257 ”(Composition B 1208);“ Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP164” and “PP258” (composition B1209); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP164” and “PP366” (composition Substance B1210): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP164” and “PP250” (composition B1211); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 164” and “PP 251” (Composition B 1212); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 164” and “PP 252” (Composition B1213); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP164” and “PP363” (Composition B1214); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1215);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP164 ”and“ PP2 ”(composition B1216);“ composition B1216) ” Any one of the compounds AA1-BA1 to AK2688-BK1287 and the combination of “PP164” and “PP3” (composition B1217); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP164” and “Composition B1218”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP164” and “PP1054” (Composition B1219); “Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP164” and “PP1055” (Composition B1220); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP370 And “PP 209” (Composition B 1221); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 370” and “PP 256” (Composition B 1222); “Compound AA 1-BA 1 “Any one of AK2688-BK1287”, a combination of “PP370” and “PP257” (Composition B1223); “a combination of any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP258” (Composition B1224); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP370” and “PP366” (Composition B1225); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1226”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP251” (composition B1227); Any one of Compounds AA1-BA1 to AK2688-BK1287, “PP370” and “PP252” (Composition B1228); “Compound AA1-BA1 to AK2688-BK1287” Combination of “one piece”, “PP370” and “PP363” (composition B1229); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP370” and “PP364” (composition B1230) "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP370" and "PP2" (Composition B 1231); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP370". “Composition B1232);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP370 ”and“ PP1051 ”(composition B1233);“ compound AA1-BA1 ” ~ A combination of one of “AK2688-BK1287”, “PP370” and “PP1054” (composition B 1234); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP370” and “PP1055” Combination (Composition B 1235); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 373” and “PP 209” (Composition B 1236); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP373” and “PP256” (Composition B1237); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP257” (Composition B1238); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 373” and “PP258” (Composition B1239); “Compound AA1-BA1 to AK2688-BK1287 Any one of “PP 373” and “PP 366” (Composition B 1240); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 373” and “PP 250” (Composition B1241); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP251” (composition B 1242); “any one of compounds AA1-BA1 to AK2688-BK1287” “Combination of PP373” and “PP252” (composition B 1243); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP373” to “PP363” “Composition B1244);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP373 ”and“ PP364 ”(Composition B1245);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP 373” and “PP 2” (Composition B 1246); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 373” and “PP 3” (Composition B 1247); Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP373” and “PP1051” (composition B1248); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP1054 (Composition B1249); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP373” and “PP1055” (Composition B1250); “Compound AA1-BA1 to AK2688-BK1287” “One of the combinations”, “PP380” and “PP209” (composition B 1251); “one of the compounds AA1-BA1 to AK2688-BK1287” and “PP380” “Composition B1252);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP380 ”and“ PP257 ”(Composition B1253);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP380” and “PP258” (composition B1254); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP366” “Composition B1255);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP380 ”and“ PP250 ”(Composition B1256);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP380” and “PP251” (Composition B1257); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP252” (Composition B1258); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP380” and “PP363” (composition B1259); “any of compounds AA1-BA1 to AK2688-BK1287 Combination of “one”, “PP380” and “PP364” (composition B1260); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP380” and “PP2” (composition B1261) "Any one of Compounds AA1-BA1 to AK2688-BK1287", a combination of "PP380" and "PP3" (Composition B 1262); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP380" And “PP 1051” (Composition B 1263); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 380” and “PP 1054” (Composition B 1264); “Compound AA 1-BA 1 “Any one of AK2688-BK1287”, a combination of “PP380” and “PP1055” (composition B1265); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP209” (Composition B1266); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP256” (Composition B1267); “Compound AA1 Any one of “-BA1 to AK2688-BK1287” and “PP387” and “PP257” (Composition B1268); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP258” (Composition B1269); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP366” (Composition B1270); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP387” and “PP250” (Composition B 1271); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP387” and “PP251” (Composition B1272 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP387" and "PP252" (Composition B1273); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP387". “Composition B1274”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP364” (combination “Compound B1275);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP387 ”and“ PP2 ”(Composition B1276);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP387” and “PP3” (Composition B1277); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP387” and “PP1051” (Composition B1278); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP387” and “PP1054” (composition B1279); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP387” and “PP1055” (Composition B 1280); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 394” and “PP 209” (Composition B 1281); “Compound AA 1-BA 1-AK 2688-BK 1287 Of “one of compounds”, “PP394” and “PP256” (composition B 1282); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” “Composition B1283);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP394 ”and“ PP258 ”(Composition B1284);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP394” and “PP366” (composition B1285); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP394” and “PP250” (composition Substance B 1286): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP394” and “PP251” (composition B1287); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 394” and “PP 252” (Composition B 1288); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 394” and “PP 363” (Composition B 1289); Any one of “-BA1 to AK2688-BK1287”, “PP394” and “PP364” (composition B1290); “any of compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP394” and “PP2” (composition B1291); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP394” and “PP3” (composition B1292); “Any one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” and “PP1051” (composition B1293); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP394” Combination with “PP1054” (Composition B1294); “Compound AA1-BA1
~ A combination of “any one of AK2688-BK1287”, “PP394” and “PP1055” (composition B1295); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP209” Combination (Composition B1296); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP256” (Composition B1297); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP407” and “PP257” (composition B1298); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP258” (composition B1299); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP366” (Composition B1300); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” Combination with “PP 250” (Composition B 1301); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 407” and “PP 251” (Composition Substance B1302); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP407” and “PP252” (composition B1303); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP407” and “PP363” (Composition B1304); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP407” and “PP364” (Composition B1305); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP407” and “PP2” (composition B1306); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP3” (Composition B1307); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP1051” (Composition B1308); “Compound AA1-BA1 to AK2688-BK1287 “Any one”, a combination of “PP407” and “PP1054” (composition B1309); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP407” and “PP1 “Composition B1310);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP693 ”and“ PP209 ”(Composition B1311);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP693” and “PP256” (composition B1312); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP257” (composition Substance B1313); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP693” and “PP258” (composition B1314); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP693” and “PP366” (Composition B1315); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP250” (Composition B1316); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP693” and “PP251” (composition B1317); “any one of compounds AA1-BA1 to AK2688-BK1287 “Composition”, “PP693” and “PP252” (composition B1318); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP363” (composition B1319) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP364” (Composition B1320); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” And “PP2” (Composition B1321); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP693” and “PP3” (Composition B1322); “Compound AA1-BA1 Combination of “one of AK2688-BK1287”, “PP693” and “PP1051” (composition B1323); “combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP1054” (Composition B1324); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP693” and “PP1055” (Composition B1325); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP694” and “PP209” (composition B1326); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP256” (Composition B1327); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP257” in combination (Composition B1328); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1329”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP366” (composition B1330); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP694” and “PP250” (composition B1331); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “Composition B1332);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP694 ”and“ PP252 ”(Composition B1333); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP363” in combination (Composition B1334); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Combination of PP694” and “PP364” (composition B1335); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP694” and “PP2” (composition B1336); “compound AA1- Any one of BA1 to AK2688-BK1287, a combination of “PP694” and “PP3” (composition B1337); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP1051” (Composition B1338); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP694” and “PP1054” (Composition B1339); Any one of “Compounds AA1-BA1 to AK2688-BK1287” “Composition B1340”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP209” (Composition B1341); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP256” (Composition B1342); “Compound AA1-BA1 to AK2688-BK1287” Of “any one of”, “PP695” and “PP257” (composition B1343); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP695” and “PP258” (composition B1344) “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP366” in combination (Composition B1345); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Composition of PP695” and “PP250” (Composition B1346); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP695” and “PP251” (Composition B1347); “Compound AA1− Any one of BA1 to AK2688-BK1287, a combination of “PP695” and “PP252” (composition B1348); “any one of compounds AA1-BA1 to AK2688-BK1287” And “PP 695” and “PP 363” (Composition B 1349); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 695” and “PP 364” (Composition B 1350); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP695” and “PP2” (Composition B 1351); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP695” Combination with “PP3” (Composition B1352); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP695” and “PP1051” (Composition B1353); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP695” and “PP1054” (composition B1354); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP695” and “PP1055” “Composition B1355);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP696 ”and“ PP209 ”(Composition B1356);“ Compound AA1-BA1 to AK Any one of 2688-BK1287, a combination of “PP696” and “PP256” (composition B1357); “a combination of any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP257” (Composition B1358); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP696” and “PP258” (Composition B1359); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1360);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP696 ”and“ PP250 ”(composition B1361);“ composition B1361 ”; Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP696” and “PP251” (composition B1362); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP696” and Combination with PP 252 "(Composition B 1363);" Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 "," PP 696 "and" PP 36 3 "(Composition B 13 64) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP696” and “PP364” (Composition B1365); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Composition of PP696” and “PP2” (Composition B1366); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP696” and “PP3” (Composition B1367); “Compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP696” and “PP1051” (composition B1368); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP696” and “PP1054” “Composition B1369);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP696 ”and“ PP1055 ”(Composition B1370);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP1” and “PP4” (Composition B1371); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1” Combination with “PP 219” (Composition B 1372); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 1” and “PP 205” (Composition B 1373); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP1” and “PP220” (composition B1374); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP221” “Composition B1375);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP1 ”and“ PP691 ”(Composition B1376);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP1” and “PP202” (Composition B1377); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP212” (Composition Substance B1378); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP263” in combination (composition B1379); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP1” and “PP203” (Composition B1380); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP204” (Composition B1381); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP1” and “PP201” (composition B1382); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP429” (Composition B1383); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP430” (Composition B1384); “Compound AA1-BA1 to AK2688-BK1287 “A combination of any one”, “PP1” and “PP 442” (composition B1385); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP701” Combination (Composition B1386); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP702” (Composition B1387); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP1” and “PP703” (composition B1388); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP277” (composition B1389); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP277-1” (Composition B1390); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1 “Composition B1391);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP1 ”and“ PP256 ”(composition B1392);“ compound AA1-BA1 ” ~ A combination of one of “AK2688-BK1287”, “PP1” and “PP257” (Composition B1393); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1” Combination with “PP258” (Composition B 1394); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP366” (Composition B1395); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP1” and “PP250” (composition B1396); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP251” "Composition B1397);" Any one of Compounds AA1-BA1-AK2688-BK1287 "," PP1 "and" PP252 "(Composition B1398);" Any one of Compounds AA1-BA1-AK2688-BK1287 " And “PP1” and “PP363” (Composition B1399); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP364” (Composition B1400); “Compound Any one of AA1-BA1 to AK2688-BK1287 and a combination of “PP1” and “PP2” (Composition B 1401); “Any one of Compounds AA1-BA1 to AK2688-BK1287 And “PP1” and “PP3” (composition B1402); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP1” and “PP1051” (composition B1403); “compound Any one of AA1-BA1 to AK2688-BK1287 and “PP1” and “PP1054” (composition B1404); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP1” and “PP1055” (Composition B1405); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP167” and “PP4” (Composition B1406); “Compound AA1-BA1 to AK2688-BK1287” Of “any one of”, “PP167” and “PP219” (composition B1407); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP167” and “PP205” (composition B1408) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP167” and “PP220” (Composition B1409); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP 167” and “PP 221” (Composition B 1410); “One of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 167” and “PP 691” (Composition B 1411 “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP167” and “PP202” (Composition B1412); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP167 And “PP 212” (Composition B 1413); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 167” and “PP 263” (Composition B 1414); “Compound AA 1-BA 1 ~ A combination of “any one of AK2688-BK1287”, “PP167” and “PP203” (composition B1415); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP167” and “PP204” Combination (Composition B 1416); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 167” and “PP 201” (Composition B 1417); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP167” and “PP429” (composition B1418); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP167” Combination with “PP 430” (Composition B 1419); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 167” and “PP 442” (Composition B 1420); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP167” and “PP701” (composition B 1421); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP167” and “PP702” “Composition B1422);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP167 ”and“ PP703 ”(Composition B1423);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP 167” and “PP 277” (Composition B 1424); “One of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 167” and “PP 277-1” Combination (Composition B1425); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP167” and “PP209” (Composition B1426); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP167” and “PP256” (composition B1427); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP167” and “PP257” (composition B1428); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP167” and “PP258” (Composition B1429); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP167” Combination with “PP 366” (Composition B1430); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 167” and “PP 250” (Composition B 1431); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “combination of“ PP167 ”and“ PP251 ”(composition B 1432);“ any one of compounds AA1-BA1 to AK2688-BK1287 ” Combination of “PP 167” and “PP 252” (Composition B 1433); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 167” and “PP 363” (Composition B 1434); Any one of “-BA1 to AK2688-BK1287”, “PP167” and “PP364” (composition B1435); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP167” and “PP2” (Composition B1436); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP167” and “PP3” (Composition B1437); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP167” and “PP1051” (Composition B1438); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP167” and “PP1054” (Composition B1439) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP167 ”and“ PP1055 ”(composition B1440);“ compound AA1-BA1 to AK2688-BK128 ” Combination of “one of 7”, “PP168” and “PP4” (composition B 1441); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP219” (composition Substance B1442); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP168” and “PP205” (composition B1443); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP168” and “PP220” (Composition B1444); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP221” (Composition B1445); “Compound AA1 Any one of “-BA1 to AK2688-BK1287” and “PP168” and “PP691” (composition B1446); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP168” and “PP202” (Composition B1447); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP168” and “PP212” (Composition B1448); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP168” and “PP263” (composition B1449); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP168” “Composition B1450);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP168 ”and“ PP204 ”(Composition B1451);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP168” and “PP201” (composition B1452); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP429” "Composition B1453);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "," PP168 "and" PP430 "(Composition B1454);" Any one of Compounds AA1-BA1 to AK2688-BK1287 " And “PP168” and “PP442” (Composition B1455); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP168” and “PP701” “Composition B1456);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP168 ”and“ PP702 ”(Composition B1457);“ Compounds AA1-BA1 to AK2688-BK1287 A combination of “one”, “PP168” and “PP703” (composition B1458); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP168” and “PP277” (composition B1459); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP277-1” (Composition B1460); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP168 “Composition B1461);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP168 ”and“ PP256 ”(composition B1462);“ compound AA1-BA1 ” ~ Any one of AK2688-BK1287 ", a combination of" PP168 "and" PP257 "(Composition B 1463);" Any one of Compounds AA1-BA1-AK2688-BK1287 " Combination of “PP168” and “PP258” (Composition B1464); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP366” (Composition B1465); “Compound AA1 Any one of “-BA1 to AK2688-BK1287” and “PP168” and “PP250” (Composition B1466); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP168” and “PP251” (Composition B1467); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP168” and “PP252” (Composition B1468); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP168” and “PP363” (Composition B1469); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP364” (Composition B1470) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP168 ”and“ PP2 ”(composition B1471);“ compound AA1-BA1 to AK2688-BK12 ” Combination of “one of 87”, “PP168” and “PP3” (composition B1472); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP1051” (composition Substance B1473); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP168” and “PP1054” in combination (composition B1474); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP168” and “PP1055” (Composition B 1475); “Compound AA 1-BA 1-A
A combination of “one of K2688-BK1287”, “PP169” and “PP4” (composition B1476); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP219” (Composition B1477); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP169” and “PP205” (Composition B1478); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1479”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP221” (composition B1480); “Any one of compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP691” (composition B1481); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP169” “Composition B1482);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”and“ PP169 ”and“ PP212 ”(Composition B148) 3); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “a combination of“ PP169 ”and“ PP263 ”(Composition B1484);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” “Combination of PP169” and “PP203” (composition B1485); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP169” and “PP204” (composition B1486); “compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP169” and “PP201” (composition B1487); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP429” (Composition B1488); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP430” (Composition B1489); Any of “Compounds AA1-BA1 to AK2688-BK1287” “Combination of K 1”, “PP 169” and “PP 44 2” (composition B 1490); “any one of compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 169” and “PP 701” (Composition B1491); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP702” (Composition B1492); “Compound AA1-BA1 to AK2688-BK1287 Combination of any one of “PP169” and “PP703” (Composition B 1493); “Composition of any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP277” (Composition B1494) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP169" and "PP277-1" (Composition B1495); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP169” and “PP209” (Composition B1496); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP169” and “PP256” (Composition B1497); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP169” and “PP257” (composition B1498); “any one of compounds AA1-BA1 to AK2688-BK1287 "Combination of Tosu", "PP169" and "PP258" (Composition B1499); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP169" and "PP366" (Composition B1500) “Combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP169” and “PP250” (composition B1501); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP169” And “PP251” (Composition B1502); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP252” (Composition B1503); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP169” and “PP363” (Composition B 1504); “a combination of any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP364” (Composition B1505); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP169” and “PP2” (Composition B1506); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP169” and “PP3” (composition B1507); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP169” and “PP1051” (Composition B1508); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP169” and “PP1054” (Composition B1509); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1510);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP170 ”and“ PP4 ”(composition B1511);“ composition B1511) ” Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP170” and “PP219” (composition B1512); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP170”, and “PP170” “Composition B 1513);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”,“ PP 170 ”and“ PP 220 ”(Composition B 1 514) combination of “any one of compounds AA1-BA1 to AK2688-BK1287” with “PP170” and “PP221” (composition B1515); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B 1516) of“ PP 170 ”and“ PP 691 ”;“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”,“ PP 170 ”and“ PP 202 ”(Composition B 1517); Any one of BA1 to AK2688-BK1287 and a combination of “PP170” and “PP212” (Composition B1518); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP263” (Composition B1519); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP203” (Composition B1520); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP170” and “PP204” (composition B1521); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP201” (Composition B1522); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP429” (Composition B1523); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP170” and “PP430” (Composition B1524); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP170” and “PP442” (Composition B1525 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP170" and "PP701" (Composition B1526); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP170". And “PP702” (Composition B1527); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP170” and “PP703” (Composition B1528); “Compound AA1-BA1” ~ A combination of one of “AK2688-BK1287”, “PP170” and “PP277” (Composition B1529); “Any one of Compounds AA1-BA1-AK2688-BK1287 , “PP170” and “PP277-1” (Composition B1530); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP170” and “PP209” (Composition B1531 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP170" and "PP256" (Composition B1532); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP170". And “PP 257” (Composition B1533); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP170” and “PP258” (Composition B1534); “Compound AA1 to BA1” ~ A combination of “any one of AK2688-BK1287”, “PP170” and “PP366” (composition B1535); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP250” Combination (Composition B1536); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP251” (Composition B1537); “Compound AA1-BA Any one of 1 to AK2688-BK1287 and a combination of “PP170” and “PP252” (Composition B1538); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP363” (Composition B1539); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP364” (Composition B1540); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP170” and “PP2” (composition B1541); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP170” and “PP3” (composition B1542) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP170" and "PP1051" (Composition B1543); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP170" And “PP1054” (composition B1544); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP170” and “PP1055” (composition B1545); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP4” (Composition B1546); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Combination of PP172” and “PP219” (composition B1547); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP172” and “PP205” (composition B1548); “compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP172” and “PP220” (composition B1549); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP221” (Composition B1550); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP691” (Composition B1551); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP172” and “PP202” (Composition B 1552); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP21” 2) (Composition B 1553); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 172” and “PP 263” (Composition B 1554); “Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP172” and “PP203” (composition B1555); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP172” and “PP204” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP201” (composition B1557); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP172” and “PP429” (Composition B1558); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP172” and “PP430” (Composition B1559); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP172” and “PP442” (composition B1560); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B1561);“ any one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP172 ”and“ PP702 ”(composition B1562); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP172” and “PP703” (Composition B 1563); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP172” Combination with “PP 277” (Composition B 1564); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 172” and “PP 277-1” (Composition B 1565); “Compound AA 1-BA 1 ~ A combination of “any one of AK2688-BK1287”, “PP172” and “PP209” (composition B1566); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP256” Combination (Composition B1567); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP257” (Composition B1568); “Compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP172” and “PP258” (Composition B 1569); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP366” (Composition B1570); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP250” (Composition B1571); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP172” and “PP251” (composition B 1572); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 172” and “PP 252” (composition B 1573) "Any one of Compounds AA1-BA1 to AK2688-BK1287", a combination of "PP172" and "PP363" (Composition B1574); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP172" And “PP364” (Composition B1575); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP2” (Composition "Any one of Compounds AA1-BA1 to AK2688-BK1287" and a combination of "PP172" and "PP3" (Composition B1577); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP172” and “PP1051” (Composition B1578); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP172” and “PP1054” (Composition B1579); “Compound AA1 Any one of “-BA1 to AK2688-BK1287” and “PP172” and “PP
1055 ”(Composition B 1580);“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”,“ PP 173 ”and“ PP 4 ”(Composition B 1581);“ Compound AA 1-BA 1 to AK 2688- A combination of “one of BK1287”, “PP173” and “PP219” (composition B1582); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP205” (composition A combination of “one of compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP220” (composition B1584); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP173” and “PP221” (Composition B 1585); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP691” (Composition B1586); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP173” and “PP202” (composition B1587); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP173” and “PP212” (composition B1588); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP263” (composition B1589) "Any one of Compounds AA1-BA1 to AK2688-BK1287", a combination of "PP173" and "PP203" (Composition B1590); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP173" And “PP204” (Composition B1591); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP201” (Composition B1592); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP173” and “PP429” (composition B 1593); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP173” and “PP430” (Composition B1594); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP173” and “PP442” (Composition B1595); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP173” and “PP701” (composition B1596); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP173” and “PP702” (Composition B1597); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP173” and “PP703” (Composition B1598); “Any one of Compounds AA1-BA1 to AK2688-BK1287 , “PP173” and “PP277” (Composition B1599); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP277-1” (Composition B1600) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP209” in combination (Composition B1601); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP173” And “PP256” (Composition B 1602); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP173” and “PP257” “Compound B1603);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP173 ”and“ PP258 ”(Composition B1604);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP 173” and “PP 366” (Composition B 1605); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 173” and “PP 250” (Composition B 1606); Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP173” and “PP251” (composition B1607); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP173” and “PP252” (Composition B1608); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP173” and “PP363” (Composition B1609); “Compound AA1-BA1 to AK2688-BK1287” “One of the compounds”, “PP173” and “PP364” (composition B1610); “one of the compounds AA1-BA1 to AK2688-BK1287” and “PP173” “Composition B 1611);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP173 ”and“ PP3 ”(Composition B1612);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP173” and “PP1051” (composition B1613); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP173” and “PP1054” (composition Substance B1614); “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP173” and “PP1055” (composition B1615); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP174” and “PP4” (Composition B1616); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP174” and “PP219” (Composition B1617); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP174” and “PP205” (Composition B1618); “Compound AA1-BA1 to AK2688-BK1287 Combination of “one”, “PP174” and “PP220” (composition B1619); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP174” and “PP221” (composition B1620) “Combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP174” and “PP691” (composition B1621); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP174” And “PP202” (Composition B1622); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP174” and “PP212” (Composition B1623); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP174” and “PP263” (composition B1624); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP174” and “PP203” (Composition B1625); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP174” and “PP204” (Composition B1626); “Compound AA1-BA1 ~ A combination of “any one of AK2688-BK1287”, “PP174” and “PP201” (composition B1627); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP174” and “PP429” Combination (Composition B1628); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP174” and “PP430” (Composition B1629); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP174” and “PP442” (composition B1630); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP174” and “PP701” (composition B1631); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP174” and “PP702” (Composition B1632); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP174” Combination with “PP 703” (Composition B1633); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP174” and “PP277” (Composition B1634); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP174” and “PP277-1” (Composition B1635); “Any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP174” and “PP209” (Composition B1636); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP174” and “PP256” (Composition B1637); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP174” and “PP257” (composition B1638); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP174” and “PP258” (Composition B1639); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP174” and “PP366” (Composition B1640); “Compound AA1-BA1 to AK2688-BK1287” “One of the combinations”, “PP174” and “PP250” (composition B 1641); “one of the compounds AA1-BA1 to AK2688-BK1287” and “PP174” Combination with “PP 251” (Composition B 1642); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 174” and “PP 252” (Composition B 1643); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “the combination of“ PP174 ”and“ PP363 ”(composition B1644);“ the combination of any one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP174 ”and“ PP364 ” “Composition B1645);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP174 ”and“ PP2 ”(Composition B1646);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP174” and “PP3” (Composition B1647); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP174” and “PP1051” (Composition B1648); “Compound Any one of AA1-BA1 to AK2688-BK1287 and a combination of “PP174” and “PP1054” (Composition B1649); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of one, "and" PP174 "and" PP1055 "(composition B1650);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP4” and “PP209” (Composition B 1651); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP4” “Composition B1652);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP4 ”and“ PP257 ”(Composition B1653);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP4” and “PP258” (composition B1654); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP4” and “PP366” “Composition B1655);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP4 ”and“ PP250 ”(Composition B1656);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” , “PP4” and “PP251” (Composition B1657); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP4” and “PP252” B1658) “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP4” and “PP363” in combination (composition B1659); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP4” and “PP364” (Composition B1660); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP4” and “PP2” (Composition B1661); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP4” and “PP3” (composition B1662); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP4” and “PP1051” (Composition B1663); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP4” and “PP1054” (Composition B1664); “Compound AA1-BA1 to AK2688-BK1287 “Any one”, a combination of “PP4” and “PP1055” (composition B1665); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP219” and “PP209” Combination (Composition B1666); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP219” and “PP256” (Composition B1667); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP219” and “PP257” (composition B1668); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP219” and “PP258” (composition B1669); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP219” and “PP366” (Composition B1670); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP219” Combination with “PP250” (Composition B 1671); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP219” and “PP251” (Composition B 1672); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP219” and “PP252” (composition B 1673); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 219” and “PP 363” (Composition B 1674); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 219” and “PP 364” (Composition B 1675); Any one of “-BA1 to AK2688-BK1287”, “PP219” and “PP2” (composition B1676); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP219” and “PP3” (Composition B 1677); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 219” and “PP 1051” (Composition B 1678); “Compound AA 1-BA 1-AK 2688-BK 1287 Any one of the combinations of “PP 219” and “PP1054” (Composition B1679); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP219” and “PP1055” (Composition B1680) “Combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP205” and “PP209” (composition B1681); “compound AA1-BA1 to AK2688-BK12” Combination of “one of 87”, “PP205” and “PP256” (composition B1682); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP205” and “PP257” (composition “Combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP205” and “PP258” (composition B1684); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP205” and “PP366” (Composition B1685); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP205” and “PP250” (Composition B1686); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP205” and “PP251” (composition B1687); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP205” and “PP252” (Composition B1688); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP205” and “PP363” (Composition B1689); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP205” and “PP364” (composition B1690); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP205” and “PP205” “Composition B1691);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP205 ”and“ PP3 ”(Composition B1692);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP205” and “PP1051” (composition B 1693); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP205” and “PP1054” (composition "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP205" and "PP1055" (Composition B1695); "Any one of Compounds AA1-BA1 to AK2688-BK1287" A combination of “PP220” and “PP209” (composition B1696); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP220” and “PP256” Combination (Composition B 1697); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP220” and “PP257” (Composition B1698); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP220” and “PP258” (composition B1699); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” and “PP220” and “PP366” (composition B1700); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP220” and “PP250” (Composition B1701); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP220” Combination with “PP 251” (Composition B 1702); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 220” and “PP 252” (Composition B 1703); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP220” and “PP363” (composition B1704); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B1705) of“ PP 220 ”and“ PP 364 ”;“ Composition B 1706 ”of“ any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 220 ”and“ PP2 ”(Compound B1706); Any one of BA1 to AK2688-BK1287 and a combination of “PP220” and “PP3” (composition B1707); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP220”, and “PP1051” (Composition B1708); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP220” and “PP1054” (Composition B1709); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP220” and “PP1055” (composition B1710); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP221” and “PP209” (composition B1711) “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP221” and “PP256” (Composition B1712); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP221” and “PP257” (Composition B 1713); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP221” and “PP258” (Composition B1714 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP221" and "PP366" (Composition B1715); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP221" And “PP 250” (Composition B1716); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 221” and “PP 251” (Composition B1717); “Compound AA 1-BA1” ~ A combination of “any one of AK2688-BK1287”, “PP221” and “PP252” (composition B1718); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP221” and “PP363” Combination (Composition B1719); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP221” and “PP364” (Composition B1720); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP221” and “PP2” (composition B1721); “any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP221” Combination with “PP3” (Composition B1722); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP221” and “PP1051” (Composition B1723); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP221” and “PP1054” (composition B1724); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP221” and “PP1055” “Composition B1725);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP691 ”and“ PP209 ”(Composition B1726);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP 691” and “PP 256” (Composition B 1727); “One of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 691” and “PP 257” “Composition B1728);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP691 ”and“ PP258 ”(Composition B1729); Any one of“ Compounds AA1-BA1 to AK2688-BK1287 ” A combination of “one”, “PP691” and “PP366” (composition B1730); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP691” and “PP250” (composition B1731); “Any one of the compounds AA1-BA1 to AK2688-BK1287” in combination with “PP691” and “PP251” (composition B1732); “any one of the compounds AA1-BA1 to AK2688-BK1287” and “PP691” “Composition B1733);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP691 ”and“ PP363 ”(Composition B1734);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP691” and “PP364” (composition B1735); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP 691 "and" PP2 "(Composition B1736);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP691 "and" PP3 "(Composition B1737);" Compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP691” and “PP1051” (composition B1738); “any one of Compound AA1-BA1 to AK2688-BK1287”, “PP691”, and “PP1054” (Composition B1739); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP691” and “PP1055” (Composition B1740); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP202” and “PP209” (composition B1741); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP202” and “PP256” (composition B1742) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP202 ”and“ PP257 ”(composition B 1743);“ compound AA1-BA1 to AK2688-BK1287 A combination of “PP202” and “PP258” (Composition B1744); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP202” and “PP366” (Composition B1745) "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP202" and "PP250" (Composition B1746); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP202". And “PP 251” (Composition B1747); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 202” and “PP 252” (Composition B1748); “Compound AA 1-BA 1 ~ A combination of “any one of AK2688-BK1287”, “PP202” and “PP363” (composition B1749); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP202” and “PP364” Combination (Composition B1750); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP202” and “PP2” (Composition B1751); “Compound Any one of AA1 -BA1 to AK2688-BK1287 "," PP202 "and" PP3 "(Composition B1752);" Any one of Compounds AA1 -BA1 to AK2688-BK1287 "," PP202 "and" PP2 " “Composition B1753);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP202 ”and“ PP1054 ”(Composition B1754);“ Compound AA1-BA1 to AK2688- Combination of “one of BK1287”, “PP202” and “PP1055” (composition
"Any one of Compounds AA1-BA1 to AK2688-BK1287" and a combination of "PP212" and "PP209" (Composition B1756); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP212” and “PP256” (Composition B1757); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP212” and “PP257” (Composition B1758); “Compound AA1 Any one of “-212 to 1-AK2688-BK1287”, “PP212” and “PP258” (composition B1759); “any one of compounds AA1-BA1-AK2688-BK1287”, “PP212” and “PP366” (Composition B1760); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP212” and “PP250” (Composition B1761); “Compound AA1-BA1 to AK2688-BK1287 “Any one”, a combination of “PP212” and “PP251” (composition B1762); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP212” and “P “Composition B1763);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP212 ”and“ PP363 ”(Composition B1764);“ Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP212” and “PP364” (Composition B1765); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP212” and “PP2” (Composition Substance B1766): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP212” and “PP3” (composition B1767); “any one of compounds AA1-BA1 to AK2688-BK1287” A combination of “PP 212” and “PP 1051” (Composition B 1768); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 212” and “PP 1054” (Composition B 1769); Any one of “-BA1 to AK2688-BK1287”, “PP212” and “PP1055” (Composition B1770); “Compound AA1-BA1 to AK2688-BK1287 “Combination of Tosu”, “PP263” and “PP209” (Composition B 1771); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP263” and “PP256” (Composition B1772) “Combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP263” and “PP257” (composition B1773); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP263” And “PP258” (Composition B1774); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP263” and “PP366” (Composition B1775); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP263” and “PP250” (composition B1776); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP263” and “PP251” (Composition B1777); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP263” and “PP252” (Composition B1778); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP263” and “PP363” (composition B1779); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP263” and “PP364” (Composition B1780); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP263” and “PP2” (Composition B1781); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1782);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP263 ”and“ PP1051 ”(composition B1783); “Any one of compounds AA1-BA1 to AK2688-BK1287”, “PP263” and “PP1054” (composition B1784); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP263” and “ “Composition B1785);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP203 ”and“ PP209 ”(Composition B1786); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP203” and “PP256” (Composition B1787); “Any one of Compounds AA1-BA1 to AK2688-BK1287” “Composition of PP203” and “PP257” (Composition B1788); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP203” and “PP258” (Composition B1789); “Compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP203” and “PP366” (composition B1790); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP203” and “PP250” (Composition B1791); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP203” and “PP251” (Composition B1792); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP203” and “PP252” (composition B1793); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP203” and “PP36” “Composition B1794);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP203 ”and“ PP364 ”(Composition B1795);“ Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP203” and “PP2” (composition B1796); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP203” and “PP3” (composition Substance B1797) “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP203” and “PP1051” (composition B1798); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP203” and “PP1054” (Composition B1799); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP203” and “PP1055” (Composition B1800); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP204” and “PP209” (composition B 1801); “any one of compounds AA1-BA1 to AK2688-BK1287” “Composition B1802);“ any one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP204 ”and“ PP257 ”(composition B1803); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP204” and “PP258” (Composition B1804); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP204” Combination with “PP 366” (Composition B1805); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 204” and “PP 250” (Composition B1806); “Compound AA1-BA1 to AK2688 -Any one of -BK1287, PP204 and PP251 (composition B1807); and any one of compounds AA1-BA1 to AK2688-BK1287 and PP204 and PP252 ( “Composition B1808);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP204 ”and“ PP363 ”(Composition B1809);“ Compound AA1-BA1 to A "Any one of K2688-BK1287", a combination of "PP204" and "PP364" (composition B1810); "a combination of any one of compounds AA1-BA1 to AK2688-BK1287", "PP204" and "PP2" (Composition B1811); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP204” and “PP3” (Composition B1812); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B 1813);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP 204 ”and“ PP1054 ”(composition B1814);“ composition B1814 ”; Any one of the compounds AA1-BA1 to AK2688-BK1287 and the combination of “PP204” and “PP1055” (composition B1815); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP201” and “PP201” “Composition B1816”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP201” and “PP256” (Composition B18 17) “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP201” and “PP257” (Composition B1818); “Any one of Compounds AA1-BA1 to AK2688-BK1287” A combination of PP201 "and" PP258 "(Composition B1819);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and a combination of" PP201 "and" PP366 "(Composition B1820);" Compound AA1- Any one of BA1 to AK2688-BK1287 and a combination of “PP201” and “PP250” (composition B1821); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP201”, and “PP251” Combination of “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP201” and “PP252” (composition B1823); any one of “compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP201” and “PP363” (composition B1824); “any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP201” and “PP364” (Composition B1825); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP201” and “PP2” (Composition B1826); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP201” and “PP3” (Composition B1827); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP201” and “PP1051” (Composition B1828 "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP201" and "PP1054" (Composition B1829); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP201" “Composition B1830”; “one of compounds AA1-BA1 to AK2688-BK1287” and “PP429” and “PP209” (composition B1831); “compound AA1-BA1” ~ A combination of one of “AK2688-BK1287”, “PP429” and “PP256” (Composition B1832); “Any one of Compounds AA1-BA1-AK2688-BK1287 “Composition B1833”; “one of compounds AA1-BA1 to AK2688-BK1287”, “PP429” and “PP258” (composition B1834); Any one of the compounds AA1-BA1 to AK2688-BK1287 and “PP429” and “PP366” (Composition B1835); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP429” and “Composition B1836);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP429 ”and“ PP251 ”(Composition B1837);“ Compound AA1-BA1 to AK2688- Any one of BK1287, a combination of “PP429” and “PP252” (Composition B1838); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP429” and “PP363” (Composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP429” and “PP364” (composition B1840); “compound AA1-BA1 to AK26”; "Any one of 88-BK1287", a combination of "PP429" and "PP2" (composition B 1841); "a combination of any one of compounds AA1-BA1 to AK2688-BK1287", "PP429" and "PP3" (Composition B1842); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP429” and “PP1051” (Composition B1843); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B 1844);“ one of compounds AA1-BA1 to AK2688-BK1287 ”and“ PP 429 ”and“ PP1055 ”(composition B1845);“ composition B1845 ”; Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP430” and “PP209” (composition B1846); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP430” and “Composition B 1847) with“ PP 256 ”;“ Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287 ”,“ PP 430 ”and“ PP 257 ”(Composition B 1848 “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP430” and “PP258” (Composition B1849); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP430” And “PP 366” (Composition B 1850); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 430” and “PP 250” (Composition B 1851); “Compound AA 1-BA 1 to “Any one of AK2688-BK1287”, a combination of “PP430” and “PP251” (composition B1852); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP430” and “PP252” (Composition B1853); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP430” and “PP363” in combination (Composition B1854); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “PP430” and “PP364” (composition B1855); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP430” and “PP2” Combination (Composition B1856); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP430” and “PP3” (Composition B1857); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP430” and “PP1051” (composition B1858); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP430” and “PP1054” (composition B1859); “Any one of the compounds AA1-BA1 to AK2688-BK1287
“Composition B1860”; “one of compounds AA1-BA1 to AK2688-BK1287” and “PP442” and “PP209” (composition B1861); “composition B1861”; Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP 442” and “PP 256” (Composition B 1862); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 442” and “PP “Composition B 1863);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 442 ”and“ PP258 ”(Composition B 1864);“ Compound AA 1-BA 1-AK 2688- A combination of “one of BK1287”, “PP 442” and “PP 366” (composition B 1865); “one of compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 442” and “PP 250” (composition A combination of “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP 442” and “PP 251” (composition B 1867); “compound AA 1-BA 1 to AK 26”; "Any one of 88-BK1287", a combination of "PP 442" and "PP 252" (composition B 1868); "a combination of any one of compounds AA1-BA1 to AK2688-BK1287", "PP 442" and "PP 363" (Composition B 1869); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP 442” and “PP 364” (Composition B1870); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “Composition B1871);“ one of compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 442 ”and“ PP3 ”(composition B1872); “Any one of compounds AA1-BA1 to AK2688-BK1287”, “PP 442” and “PP1051” (composition B1873); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP 442” and “PP4” Combination with PP 1054 (Composition B 1874); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 442” and “PP 1055” (Composition B 1875 "Any one of Compounds AA1-BA1 to AK2688-BK1287", and a combination of "PP701" and "PP209" (Composition B1876); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP701" And “PP256” (Composition B1877); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP701” and “PP257” (Composition B1878); “Compound AA1-BA1” “Any one of AK2688-BK1287”, a combination of “PP701” and “PP258” (composition B1879); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP701” and “PP366” (Composition B1880); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP701” and “PP250” (Composition B1881); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “The combination of“ PP 701 ”and“ PP 251 ”(composition B 1882);“ any one of compounds AA1-BA 1 to AK 2688-BK 1287 ”,“ PP 701 ”and“ PP 252 ” (Composition B 1883); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 701” and “PP 363” (Composition B1884); Any of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “K” one, “PP 701” and “PP 364” (composition B 1885); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 701” and “PP 2” (composition B 1886) "Any one of Compounds AA1-BA1 to AK2688-BK1287", a combination of "PP701" and "PP3" (Composition B 1887); "Any one of Compounds AA1-BA1 to AK2688-BK1287" and "PP701" And “PP1051” (Composition B1888); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP701” and “PP1054” (Composition B1889); “Compound AA1-BA1 “Any one of AK2688-BK1287”, a combination of “PP701” and “PP1055” (composition B1890); “any one of compounds AA1-BA1 to AK2688-BK1287 And “PP702” and “PP209” (Composition B1891); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP702” and “PP256” (Composition B1892); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP702” and “PP257” (composition B1893); “any one of compound AA1-BA1 to AK2688-BK1287”, “PP702” and “PP258” (Composition B1894); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP702” and “PP366” (Composition B1895); “Compound AA1-BA1 to AK2688-BK1287” Any one of “PP702” and “PP250” (composition B1896); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP702” and “PP251” (composition “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP702” and “PP252” (Composition B1898); “Compound AA1-BA1 to AK2688- A combination of “one of BK1287”, “PP702” and “PP363” (composition B1899); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287”, “PP702” and “PP364” (composition Substance B1900): “one of compounds AA1-BA1 to AK2688-BK1287” in combination with “PP702” and “PP2” (composition B1901); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP702” and “PP3” (Composition B1902); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP702” and “PP1051” (Composition B1903); “Compound AA1 Any one of “-BA1 to AK2688-BK1287”, “PP702” and “PP1054” (composition B1904); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP702” and “PP1055” (Composition B 1905); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287”, “PP 703” and “PP 209” (Composition B 1906) “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP703” and “PP256” (Composition B1907); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP703” Combination with “PP 257” (Composition B 1908); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 703” and “PP 258” (Composition B 1 909); “Compound AA 1-BA 1-AK 2688 Any one of “-BK1287”, “PP703” and “PP366” (composition B1910); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP703” and “PP250” “Composition B1911);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP703 ”and“ PP251 ”(Composition B1912);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP703” and “PP252” (Composition B1913); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP703” and “PP363” Combination (Composition B1914); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP703” and “PP364” (Composition B1915); Any one of “Compounds AA1-BA1 to AK2688-BK1287” A combination of “one”, “PP703” and “PP2” (composition B1916); “a combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP703” and “PP3” (composition B1917); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP703” and “PP1051” (Composition B1918); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP703” “Composition B1919) with“ PP1054 ”;“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP703 ”and“ PP1055 ”(Composition B1920);“ Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP277” and “PP209” (composition B1921); “any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 277” and “PP 256” (Composition B 1922); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 277” and “PP 257” (Composition B 1923); Any one of “-BA1 to AK2688-BK1287” and “PP277” and “PP258” (Composition B1924); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP277” and “PP366” (Composition B1925); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP277” and “PP250” (Composition B1926); “Compound AA1-BA1 to AK2688-BK1287 Any one of the combinations of “PP277” and “PP251” (Composition B1927); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP277” and “PP252” (Composition B1928 "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP 277" and "PP 363" (Composition B 1929); "Compounds AA 1-BA 1 to AK 2688-BK 1 Any one of 287, “PP 277” and “PP 364” (composition B 1930); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 277” and “PP 2” (composition “Any one of compounds AA1-BA1 to AK2688-BK1287” and “PP277” and “PP3” (composition B1932); “any one of compounds AA1-BA1 to AK2688-BK1287” Combination of “PP 277” and “PP 1051” (Composition B 1933); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 277” and “PP 1054” (Composition B 1 934); Any one of “-BA1 to AK2688-BK1287”, “PP277” and “PP1055” (composition B1935); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP277-1” and “PP277” “Composition B1936);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP277-1 ”and“ PP256 ”(Composition B1937); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP277-1” and “PP257” (Composition B1938); “Any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP 277-1” and “PP 258” (Composition B 1939); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 277-1” and “PP 366” (Composition B 1940) "Any one of Compounds AA1-BA1 to AK2688-BK1287" in combination with "PP277-1" and "PP250" (Composition B1941); "Any one of Compounds AA1-BA1 to AK2688-BK1287" Combination of “PP 277-1” and “PP 251” (Composition B 1942); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 277-1” and “PP 252” (Composition B 1943) “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 277-1” and “PP 363” (Composition B 1944); “Attachment of Compounds AA 1-BA 1 to AK 2688-BK 1287 Combination of “one piece”, “PP 277-1” and “PP 364” (composition B 1945); “one of compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 277-1” and “PP 2” (Composition B1946); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP277-1” and “PP3” (Composition B1947); Any one of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “one”, “PP277-1” and “PP1051” (composition B 1948); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP277-1” to “PP1054” Composition B1949): “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP277-1” and “PP1055” (Composition B1950);

“Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP209” and “PP250” (Composition B1951); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP209” Combination with “PP 251” (Composition B 1952); “Any one of Compounds AA 1-BA 1-AK 2688-BK 1287”, “PP 209” and “PP 252” (Composition B 1953); “Compound AA 1-BA 1-AK 2688 -Any one of -BK1287, a combination of "PP209" and "PP363" (composition B 1954); a combination of "any one of compounds AA1-BA1 to AK2688-BK1287", "PP209" and "PP364" “Composition B1955);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP209 ”and“ PP2 ”(Composition B1956);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP 209” and “PP 3” (Composition B 1957); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 209” and “PP 1051” “Composition B 1958);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 209 ”and“ PP 1054 ”(Composition B 1959);“ Compounds AA 1-BA 1 to AK 2688-BK 1287 A combination of “one”, “PP209” and “PP1055” (Composition B1960); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP256” and “PP250” (Composition B1961); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP256” and “PP251” (Composition B 1962); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP256” “Composition B 1963);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 256 ”and“ PP 363 ”(Composition B 1964);“ Compound AA 1-BA 1 to AK 2688 ” Any one of “-BK1287”, “combination of“ PP256 ”and“ PP364 ”(composition B1965);“ any one of compounds AA1-BA1 to AK2688-BK1287 ” “Combination of PP256” and “PP2” (composition B1966); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP256” and “PP3” (composition B1967); “compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP256” and “PP1051” (Composition B1968); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP256” and “PP1054” (Composition B1969); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP256” and “PP1055” (Composition B1970); Any one of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “K”, “PP 257” and “PP 250” (Composition B 1971); “Any one of Compounds AA 1-BA 1 to AK 2688-BK 1287” and “PP 257” and “PP 251” (Composition B 1972) “Combination of“ any one of compounds AA1-BA1 to AK2688-BK1287 ”with“ PP257 ”and“ PP252 ”(composition B1973);“ compound AA1-BA1 to AK2688-BK1287 Any one of “PP257” and “PP363” (Composition B1974); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP257” and “PP364” (Composition B1975); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP257” and “PP2” (Composition B1976); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “B. “A combination of PP257” and “PP3” (Composition B 1977); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 257” and “PP1051” (Composition B1978); “Compound AA1− Any one of BA1 to AK2688-BK1287 and a combination of “PP257” and “PP1054” (composition B 1979); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP257” and “PP1055” (Composition B1980); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP258” and “PP250” (Composition B1981); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP258” and “PP251” (Composition B 1982); “any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP258” “Composition B 1983”; “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 258” and “PP 363” (Composition B 1984); “Compound AA 1-BA 1 to AK 2688 Any one of “-BK1287”, “PP258” and “PP364” (composition B1985); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP258” and “PP2” Composition B 1986); "Any one of Compounds AA1-BA1 to AK2688-BK1287", "PP258" and "PP3" (Composition B1987); "Any one of Compounds AA1-BA1 to AK2688-BK1287" , “PP258” and “PP1051” (Composition B 1988); “One of Compounds AA1-BA1 to AK2688-BK1287”, “PP258” and “PP1054” (Composition B1989); “Any one of Compounds AA1-BA1 to AK2688-BK1287” in combination with “PP258” and “PP1055” (Composition B1990); “Any one of Compounds AA1-BA1 to AK2688-BK1287 “PP 366” and “PP 250” (Composition B 1991); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 366” and “PP 251” (Composition B 1992); Any one of the compounds AA1-BA1 to AK2688-BK1287 in combination with “PP366” and “PP252” (composition B1993); “any one of the compounds AA1-BA1 to AK2688-BK1287”, “PP366” and “PP268” “Composition B 1994);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP 366 ”and“ PP 364 ”(Composition B 1995);“ Compound AA 1-BA 1-AK 2688- Any one of BK1287, a combination of “PP 366” and “PP 2” (Composition B 1996); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 36 6 "and" PP3 "(Composition B 1997);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP 366 "and" PP1051 "(Composition B 1998);" Compound AA 1- " Any one of BA1 to AK2688-BK1287 and a combination of “PP366” and “PP1054” (composition B1999); “any one of compounds AA1-BA1 to AK2688-BK1287”, “PP366” and “PP1055” (Composition B2000); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP250” and “PP363” (Composition B2001); Any one of “Compounds AA1-BA1 to AK2688-BK1287” Combination of “Kanichi”, “PP250” and “PP364” (Composition B 2002); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP250” and “PP2” (Composition B 2003) “One of compounds AA1-BA1 to AK2688-BK1287” and “PP250” and “PP3” (composition B 2004); “compound AA1-BA1 to AK2688-BK1287” Combination of “one piece”, “PP250” and “PP1051” (composition B 2005); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP250” and “PP1054” (composition B2006) “Combination of any one of compounds AA1-BA1 to AK2688-BK1287” with “PP250” and “PP1055” (composition B2007); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP251” And “PP 363” (Composition B 2008); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP 251” and “PP 364” (Composition B 2009); “Compound AA 1-BA 1 ~ A combination of “one of AK2688-BK1287”, “PP251” and “PP2” (composition B 2010); “one of compounds AA1-BA1 to AK2688-BK1287”, “PP251” and “PP3” Combination (Composition B 2011); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP 251” and “PP 1051” (Composition B 2012); “Compound Any one of AA1-BA1 to AK2688-BK1287 and “PP251” and “PP1054” (Composition B 2013); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP251” and “PP1055” (Composition B2014); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP252” and “PP363” (Composition B2015); “Compound AA1-BA1 to AK2688-BK1287” Any one of “PP252” and “PP364” (Composition B 2016); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP252” and “PP2” (Composition B2017); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP252” and “PP3” (Composition B2018); “Any one of Compounds AA1-BA1 to AK2688-BK1287” Combination of PP252 "and" PP1051 "(Composition B2019);" Any one of Compounds AA1-BA1 to AK2688-BK1287 "and" PP252 "and" PP1054 " Composition B2020); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP252” and “PP1055” (Composition B2021); “Any one of Compounds AA1-BA1 to AK2688-BK1287” And “PP 363” and “PP 2” (Composition B 2022); “Any one of Compounds AA1-BA 1 to AK 2688-BK 1287” and “PP 363” and “PP 3” (Composition B 2023); Any one of AA1-BA1 to AK2688-BK1287 and “PP363” and “PP1051” (Composition B2024); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP363” and “PP1054” (Composition B2025); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP363” and “PP1055” (Composition B2026); “Compound AA1-BA1 to AK2688-BK1287” Any one of “PP364” and “PP2” (composition B2027); “any one of compounds AA1-BA1 to AK2688-BK1287” and “PP364” Combination with “PP3” (Composition B2028); “Any one of Compounds AA1-BA1 to AK2688-BK1287”, “PP364” and “PP1051” (Composition B2029); “Compound AA1-BA1 to AK2688 Any one of “-BK1287”, “PP364” and “PP1054” (composition B2030); “one of compounds AA1-BA1 to AK2688-BK1287” and “PP364” and “PP1055” “Composition B2031);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ”,“ PP2 ”and“ PP1054 ”(Composition B2032);“ Any one of Compounds AA1-BA1 to AK2688-BK1287 ” And “PP2” and “PP1055” (Composition B2033); “Any one of Compounds AA1-BA1 to AK2688-BK1287” and “PP3” and “PP1054” (Composition B2034); “Compound Any one of AA1-BA1 to AK2688-BK1287, a combination of “PP3” and “PP1055” (Composition B 2035); “Any of Compounds AA1-BA1 to AK2688-BK1287 Combination of one, "and" PP1051 "and" PP1054 "(composition B2036); the combination of the" any one of the compounds AA1-BA1~AK2688-BK1287 "and" PP1051 "and" PP1055 "(composition B2037).

  The composition of the present invention may further contain an inert carrier. The composition of the present invention is generally prepared by mixing the composition of the present invention with an inert carrier such as a solid carrier, a liquid carrier, a gaseous carrier and the like, and adding a surfactant and other pharmaceutical auxiliaries as required. Are formulated into emulsions, oils, powders, granules, wettable powders, flowables, microcapsules and the like.

  Examples of solid carriers used in formulation include clays (kaolin clay, diatomaceous earth, bentonite, fubasami clay, acid clay etc.), synthetic hydrous silicon oxide, talc, ceramics, and other inorganic minerals (sericite, quartz, sulfur) Fine powders and granules of activated carbon, calcium carbonate, hydrated silica etc., chemical fertilizers (ammonium sulfate, ammonium phosphate, ammonium nitrate, urea, sodium chloride etc.), etc., and synthetic resins (polypropylene, polyacrylonitrile, polymethyl methacrylate) And polyester resins such as polyethylene terephthalate, nylon resins such as nylon-6, nylon-11, and nylon-66, polyamide resins, polyvinyl chloride, polyvinylidene chloride, vinyl chloride-propylene copolymer, and the like.

  Examples of liquid carriers include water, alcohols (methanol, ethanol, isopropyl alcohol, butanol, hexanol, benzyl alcohol, ethylene glycol, propylene glycol, phenoxyethanol etc.), ketones (acetone, methyl ethyl ketone, cyclohexanone etc.), aromatic hydrocarbons (Toluene, xylene, ethylbenzene, dodecylbenzene, phenylxylylethane, methylnaphthalene etc.), aliphatic hydrocarbons (hexane, cyclohexane, kerosene, light oil etc.), esters (ethyl acetate, butyl acetate, isopropyl myristate, Ethyl oleate, diisopropyl adipate, diisobutyl adipate, propylene glycol monomethyl ether acetate, etc., nitriles (acetonitrile, isobutyro) Tolyl etc., ethers (diisopropyl ether, 1,4-dioxane, ethylene glycol dimethyl ether, diethylene glycol dimethyl ether, diethylene glycol monomethyl ether, propylene glycol monomethyl ether, dipropylene glycol monomethyl ether, 3-methoxy-3-methyl-1-butanol, etc. Acid amides (N, N-dimethylformamide, N, N-dimethylacetamide etc.), halogenated hydrocarbons (dichloromethane, trichloroethane, carbon tetrachloride etc.), sulfoxides (dimethyl sulfoxide etc.), propylene carbonate and vegetable oil (Soybean oil, cottonseed oil, etc.).

  Examples of the gaseous carrier include fluorocarbon, butane gas, LPG (liquefied petroleum gas), dimethyl ether and carbon dioxide gas.

  Examples of surfactants include nonionic surfactants such as polyoxyethylene alkyl ether, polyoxyethylene alkyl aryl ether, polyethylene glycol fatty acid ester, and anions such as alkyl sulfonate, alkyl benzene sulfonate, and alkyl sulfate. Surfactants may be mentioned.

  As other pharmaceutical adjuvants, fixing agents, dispersing agents, coloring agents, stabilizers and the like, specifically, casein, gelatin, saccharides (starch, gum arabic, cellulose derivative, alginic acid etc.), lignin derivative, bentonite, Synthetic water-soluble polymers (polyvinyl alcohol, polyvinyl pyrrolidone, polyacrylic acids, etc.), PAP (isopropyl acid phosphate), BHT (2,6-di-tert-butyl-4-methylphenol), BHA (2-tert- A mixture of butyl-4-methoxyphenol and 3-tert-butyl-4-methoxyphenol).

  In addition, the composition of the present invention may further contain a compound such as anthraquinone which is used as a bird repellent.

  The composition of the present invention may be used by mixing it with various oils such as mineral oil and vegetable oil, or surfactants. Oils which can be specifically mixed and used, and surfactants such as Nimbus (registered trademark), Assist (registered trademark), Aureo (registered trademark), Iharol (registered trademark), Silwet L-77 (registered trademark), BreakThru (R), Sundance II (R), Induce (R), Penetrator (R), AgriDex (R), Lutensol A8 (R), NP-7 (R), Triton (R) , Nufilm (registered trademark), Emulgator NP7 (registered trademark), Emulad (registered trademark), TRITON X 45 (registered trademark), AGRAL 90 (registered trademark), AGROTIN (registered trademark), ARPON (registered trademark), EnSpray N (registered trademark) Registration Target), and the like BANOLE (registered trademark)

  The compositions of the invention can be used to protect plants from plant diseases. Examples of plant diseases that can be controlled by the composition of the present invention include plant diseases caused by plant pathogens such as filamentous fungi and bacteria, and specific examples include, but are not limited to: It is not a thing.

Rice blast (Magnaporthe grisea), sesame leaf blight (Cochliobolus miyabeanus), sheath blight (Rhizoctonia solani), dreadling (Gibberella fujikuroi), yellow dwarf (Sclerophthora macrospora); wheat powdery mildew (Blumeria graminis) of wheat ), Fusarium head blight (Fusarium graminearum, Fusarium avenaceum, Fusarium culmorum, Microdochium nivale), yellow rust (Puccinia striiformis), black rust (Puccinia graminis), red rust (Puccinia recondita), red snowfever (Microdochium nivale) Microdochium majus), snow blight scleroderma (Typhula incarnata, Typhula ishikariensis), naked scab (Ustilago tritici), raccoon sclera (Tilletia caries, Tilletia controversa), scab (Pseudocercosporella herpotrichoides), leaf scab tritici), downy mildew (Stagonospora nodorum), yellow spot (Pyrenophora tritici-repentis), seedling blight (Rhizoctonia solani) caused by Rhizoctonia spp., blight (Gaeuma) nnomyces graminis); powdery mildew of barley (Blumeria graminis), red mold (Fusarium graminearum, Fusarium avenaceum, Fusarium culmorum, Microdochium nivale), yellow rust (Puccinia striiformis), black rust (Puccinia graminis) Puccinia hordei), small rust (Puccinia hordei), bare smut (Ustilago nuda), cloud disease (Rhynchosporium secalis), web blight (Pyrenophora teres), spotted disease (Cochliobolus sativus), leaf blight (Pyrenophora graminea), Ramularia leaf spot disease (Ramularia collo-cygni), Rhizoctonia spp. Seedling blight (Rhizoctonia solani); corn rust (Puccinia sorghi), southern rust (Puccinia polysora), soot disease (Setosphaeria turcica), tropical Rust (Physopella zeae), Sesame Leaf Blight (Cochliobolus heterostrophus), Anthracnose (Colletotrichum graminicola), Gray Leaf Spot (Cercospora zeae-maydis), Brown spot disease (Kabatiella zeae), Phaeosphaeria leaf spot disease (Phaeosphaeria maydis), Stenocarpella maydis, Stenocarpella macrospora, Stochlot's disease (Fusarium graminearum, Fusarium verticilioides, Colletotrichum graminicola), Spikelosis (Ustilago maydis) Downy mildew (Colletotrichum gossypii), mildew (Ramularia areola), black spot (Alternaria macrospora, Alternaria gossypii), Black root rot (Thielaviopsis basicola) by Thielaviopsis spp .; Hemorrhea of coffee (Hemileia vastatrix), leaf spot Disease (Cercospora coffeicola); Sclerotinia sclerotiorum of rapeseed (Sclerotinia sclerotiorum), black spot (Alternaria brassicae), root scab (Phoma lingam); rust of sugar cane (Puccinia melanocephala, Puccinia kuehnii), black scallop Sunflower rust (Puccinia helianthi), downy mildew (Plasmopara halstedii); citrus black spot (Diaporthe citri) Scab (Elsinoe fawcetti), fruit rot (Penicillium digitatum, Penicillium italicum), plague (Phytophthora parasitica, Phytophthora citrophthora); Monilia disease of the apple (Monilinia mali); leucotricha), spotted leaf rot (Alternaria alternata apple pathotype), scab (Venturia inaequalis), anthracnose (Glomerella cingulata), brown spot (Diplocon mali), ringworm (Botyosphaeria berengeriana), plague (Phytophtora cactorum); Pear scab disease (Venturia nashicola, Venturia pirina), black spot disease (Alternaria alternata Japanese pear pathology), red star disease (Gymnosporangium haraeanum); peach scab (Monilinia fructicola), scab disease (Cladosporium carpophilum), phophoposis (Phomopsis sp.); Grape scab (Elsinoe ampelina), late rot (Glomerella cingulata), powdery mildew (Uncinula necator), rust Phakopsora ampelopsidis), blacklot disease (Guignardia bidwellii), downy mildew (Plasmoparaviticola); anthracnose of oyster (Gloeosporium kaki), deciduous disease (Cercospora kaki, Mycosphaerella nawae); , Powdery mildew (Sphaerotheca fuliginea), scab (Didymella bryoniae), brown spot (Corynespora cassiicola), scab (Fusarium oxysporum), downy mildew (Pseudoperonospora cubensis), plague (Phytophthora sp.), Blight (Pythium sp.); Tomato blight (Alternaria solani), leaf blight (Cladosporium fulvum), cast mildew (Pseudocercospora fuligena), plague (Phytophthora infestans), powdery mildew (Leveillula taurica); eggplant Brown scab (Phomopsis vexans), powdery mildew (Erysiphe cichoracearum); black spot of cruciferous vegetables (Alternaria japonica), scab (Cercosporella brassicae), scab (Plasmodiophora brassicae), Disease (Peronospora parasitica); rust disease of green onion (Puccinia allii); purpuric disease of soybean (Cercospora kikuchii), mildew (Elsinoe glycines), black spot disease (Diaporthe phaseolorum var. Sojae), rust disease (Phakopsora pachyrhizi), Brown ring disease (Corynespora cassiicola), anthracnose (Colletotrichum glycines, Colletotrithum truncatum), leaf blight (Rhizoctonia solani), brown disease (Septoria glycines), spot disease (Cercospora sojina), sclerotiosis (Sclerotinia sclerotium) Powdery mildew (Microsphaera diffusa), downy mildew (Phytophthora sojae), downy mildew (Peronospora manshurica), sudden death (Fusarium virguliforme); sclerotinia sclerotiorum of green beans, rust (Uromyces appendiculatus) Plaque (Phaeoisariopsis griseola), Anthracnose (Colletotrichum lindemuthianum); Black-spot of peanut (Cercospora personata), Brown-spot (Cercospora arachidicola), White scab (Sclerotium rolfsii); Powdery mildew of wild boar (Erysiphe pisi); summer rot of potato (Alternaria solani), plague (Phytophthora infestans), rot of rot (Phytophthora erythroseptica), powdery mildew (Spongospora subterranean f. Sp. Subterranea), half body wilt Disease (Verticillium albo-atrum, Verticillium dahliae, Verticillium nigrescens); powdery mildew of strawberries (Sphaerotheca humuli); tea scab (Exobasidium reticulatum), scab (Elsinoe leucospila), rotational blight (Pestalotiopsis sp.) Anthracnose (Colletotrichum theae-sinensis); tobacco scab (Alternaria longipes), anthracnose (Colletotrichum tabacum), downy mildew (Peronospora tabacina), plague (Phytophthora nicotianae); sugar beet (Cercospora beticola) , Leaf rot (Thanatephorus cucumeris), root rot (Thanatephorus cucumeris), black root disease (Aphanomyces cochlioides), rust (Uromyces betae); rose scab (Diplocarpon rosae) Powdery mildew (Sphaerotheca pannosa); Chrysanthemum leaf blight (Septoria chrysanthemi-indici), white rust (Puccinia horiana); allii), Botrytis rot (Botrytis squamosa); Botrytis cinerea of various crops, Botrytis sclerotis (Sclerotinia sclerotiorum); Japanese black radish (Alternaria brassicicola); Dollar spot disease of the shiva (Sclerotinia) homoeocarpa), brown patch disease and large patch disease (Rhizoctonia solani) of Shiva; and Sigatoka disease of banana (Mycosphaerella fijiensis, Mycosphaerella musicola).
Seed disease or early growth of various crops caused by Aspergillus spp., Penicillium sp., Fusarium sp., Gibberella sp., Tricoderma sp., Thieloviopsis sp., Rhizopus sp., Rhizopus sp., Mucor sp., Corcium sp., Phoma, Rhizoctonia sp., Diplodia sp. Diseases of Virus diseases of various crops mediated by Polymixa genus or Olpidium genus etc.
Seedling blight of rice (Burkholderia plantarii); spotted blight of cucumber (Pseudomonas syringae pv. Lachrymans); blight of eggplant (Ralstonia solanacearum); carotovora) etc.

  The composition containing the present compound and one or more components selected from group B can be used to control pests such as harmful insects and harmful mites. Specific examples of such harmful animals include, but are not limited to, the following.

  Semi-lepidoptera (Hemiptera): Hemetobiunka (Laodelphax striatellus), Tobiirounka (Nilaparvata lugens), Sejirounka (Sogatella furcifera), Cornflower (Peregrinus maidis), Lobluntia (Javesella pellucida), Black-tailed Ubiclusi Leafhopper family (Delphacidae); green leafhopper (Nephotettix cincticeps), giant leafhopper green leafhopper (Nephotettix virescens), black leafhopper green leafhopper (Nephotettix nigropictus), green leafhopper leafworm (Recilia dorsalis), green leafhopper foliage ), Corn leaf hopper (Dalbulus maidis), white leafhopper (Cofana spectra), etc., leafhopper family (Cicadelidae); Mahanarva posticata, Mahanarva fimbriolata, etc. (Cercopidae); Brash beetle (Aphis fabae), soybean aphid (Aphis glycines), cotton aphid (Aphis gossypii), European apple aphid (Aphis pomi), black-and-white aphid (Aphis spiraecola), green-billed aphid (Myzus persicae), blue-toothed aphid , Radish aphids (brevicoryne brassicae), Rosy apple aphid (Dysaphis plantaginea), imago radish aphids (Lipaphis erysimi), tulip pokeweed aphids (Macrosiphum euphorbiae), potato pokeweed aphids (Macrosiphum euphorbiae), potato pokeweed aphid (Alacorth cichalis). Aphids (Rhopalosiphum padi), corn aphids (Rhopalosiphum maidis), red-handed aphids (Toxoptera citricidus), Peach coptis Aphid (Hyalopterus pruni), bryophytes (Melanaph) Aphididae (Aphididae), such as the black-tailed aphid (Tetranaura nigriabdominalis), the yellow-billed aphid (Ceratovacuna lanigera), and the like (Eriosoma lanigerum); Leaf phylloxera (Phylloxera notabilis), Southern pecan leaf phylloxera (Phylloxera russellae) and other nematode (Phylloxeridae); A rice black bug (Scotinophara lurida), a Malayan rice black bug (Scotinophara coarctata), a green bug (Nezara antennata), a goby bug (Eysarcoris aeneus), a goby bug (Eysarcoris lewisi), a goby beetle (Eysarcoris lewisi), village Blue-headed stink bug (Eysarcoris annamita), Gray-backed bug (Halyomorpha halys), South African stink bug (Nezara viridula), Brown stink bug (Euschistus heros), Red banded stink bug (Piezodorus guildinii), Oebalus pugnax, etc. Brentaridae (Cydnidae), such as Burrower brown bug (Scaptocoris castanea); ;; Helicidae (Coreidae), such as Cletus punctiger, Leptoglossus australis, etc .; Caverelius saccharivorus, Togo hemipterus, Bugs such as Blissus leucopterus) (Lygaeidae); Trichonotidae, such as Trigonotylus caelestialium, Red-handed Tortoise (Stenotus rubrovittatus), Green-winged Tufted Turtle (Stenodema calcarata), Lys-biosis (Lygus linealis) etc. , Bemisia tabaci (Bemisia tabaci), Orange leafworm (Dialeurodes citri), Red-winged leafhopper (Aleurocanthus spiniferus), White-tailed lice (Aleurocanthus camelliae), White-leafed leafworm (Pealius euryae), etc. (Abgrallaspis cyanophylli), Red-backed scale insect (Aonidiella aurantii), Yellow-backed scale insect (Diaspidiotus perniciosus), Red-tailed scale insect (Pseudaulacaspis pentagona), Red-winged scale insect (Unaspis yanonensis), Red-tailed mealybug (Unaspis citri), etc., Marukabidae (Diaspididae); ruby (Ceroplastes rubens), etc., cataclyssidae (Coccidae); Anemone mealworm (Margarodidae); Anemone mealworm (Phenacoccus solani), a mealworm mealworm (Phenacoccus sorenopsis), a mealworm mealworm (Planococcus kraunhiae), a mealworm mealworm (Planococcus comstocki), a mealworm mealworm (Planococcus gyrus) (Pseudococcus calceolariae), mealybug (Pseudococcus longispinus), tutormyri bug (Brevennia rehi), etc. Pseudococcidae (Pseudococcidae); ioza erytreae), nashi-kushi lice (Cacopsylla pyrisuga), psyllid lice (Cacopsylla chinensis), potato short-tailed lice (Bacterica cockerelli), pear psylla (Cacopsylla pyricola), etc. Glymbidae such as Corythucha marmorata), Stephanitis nashi, and Tsujigunbai (Stephanitis pyrioides); Cicidae (Cimicidae) such as the bedbug (Cimex lectularius) and the like (Cicadidae) such as Giant Cicada (Quesada gigas)

  Lepidoptera insects (Lepidoptera): Nymphs (Chilo suppressalis), Darkheaded stem borer (Chilo polychrysus), White stem borer (Scirpophaga innotata), Itten's tree magnolia (Scirpophaga incertulas), Rupela albina, Kobomeiga (Cinatalitraceitraceitracel Red clover (Marasmia exigua), cotton dwarf (Notarcha derogata), African dwarf (Ostrinia furnacalis), European corn borer (Ostrinia nubilalis), black-legged moth (Hellula undulis), Monquil chronogare (Herpetogramma luctigueta) Rice case worms (Nymphula depunctalis), Sugarcane borer (Diatraea saccharalis), etc. (Cambididae); , Roy Spurge (Spodoptera exigua), Sturgeon (Mythimna separata), Sparrow (Mamestra brassicae), Spurge (Sesamia inferens), Spodoptera mauritia, Phylum oryzae (Naranga aenescens), Spurges exempta), spiny moth (Agrotis ipsilon), spiny eel (Autographa nigrisigna), inykin owava (Plusia festucae), Soybean looper (Chrysodeixis includens), Trichoplusia spp. Helicoverpa armigera), Helicoverpa zea etc. Helicoverpa, Velvetbean caterpillar (Anticarsia gemmatalis), Cotton leafworm (Alabama argillacea), Hop vine borer (Hydraecia immanis) etc. Yagidae (Noctuiipalis); Pae) et al. (Pieridae); Anemonefish (Grapholita molesta), Anemonefish (Grapholita dimorpha), Leguminivora (Leguminivora glycinivorella), Azukisya Mushiga (Matsumuraeses azukivora), Anemone parrotfish (Adoxophycha or Hamaki (Adoxophyes honmai), Chahamaki (Homona magnanima), Midarekamonhamaki (Archips fuscocupreanus), codling moth (Cydia pomonella), Kanshashini Hamami (Tetramoera schistaceana), Bean Shoot Borer (Epinotia aporema) luciferitracit Etc.) (Corappilia theivora), Gypsophilidae (Gracillariidae) of the family of Phyllonorycter ringoniella; Lymanetiidae (Lyonetriidae): Lyonetidae (Lyonetia prunifolia), such as the leafminer (Lyonetia prunifoliella); Lymanetrid (Lyantria dispar), etc. Lymantriidae (Lymantriidae), such as the genus Lymantria, Euproctis pseudoconspersa, etc. Pluteliidae, such as Plutella xylostella); Anarchia lineatella; Archeidae (Arctiidae) such as Cunea et al .; Castniidae such as Giant Sugarcane borer (Telchin licus); ); Hero helicopter Anemoneidae (Limacadidae), such as Parasa lepida; Anemoneidae (Stathmopodidae), such as Stathumopoda masinissa, etc. (Sesiidae); Hesperiidae (Hesperiidae) such as the ladybug (Parnara guttata).

  Thysanoptera: Thripsidae (Frankliniella occidentalis), Thrips palmi (Thrips palmi), Chalyss occidentalis (Scirtothrips dorsalis), Locustoids (Thrips tabaci), Philosophis japonicus (Frankliniella intimasite) And Thripidae such as Echinothrips americanus); Thripidae (Phlaeothripidae) such as Haekohrrips aculeatus.

  Diptera: Insect fly (Delia platura), Onion fly (Delia antiqua), etc. Anthomyiidae; Sugar beet rooted magots (Tetanops myopaeformis), etc. A family of freshwater flies such as the tomato leafminer fly (Liriomyza sativae), a bean leafminer fly (Liliomyza trifolii), a leafminer fly (Chromatomyia horticola), and the like; Fruit fly (Bactrocera latifrons), olive fruit fly (Bactrocera oleae), quince fruit fly (Bactrocera tryoni), fruit fly (Ceratitis capitata) and other fruit flies (Tephritidae); A fly family (Ephydridae), such as Hydrellia philippina, a rice leafhopper (Hydrellia sasakii), a Drosophila family such as Drosophila melanogaster (Drosophila suzukii); Butterflies (Clogmia albipunctata), etc .; Brachysia fly (Sciaridae), such as fly (Bradysia difermis); Hessy fly (Mayetiola destructor), and Echinoidea (Orseolia oryzae) Macrophaga (Diopsidae) such as Macrophthalma et al .; Tipula aino, Common cranefly (Tipula oleracea), European cranefly (Tipula paludosa) etc.

  Coleoptera insect pest (Coleoptera): Western corn rootworm (Diabrotica virgifera virgifera), Southern corn rootworm (Diabrotica undecimpunctata howardi), Northern corn rootworm (Diabrotica barberi), Mexican corn rootworm (Diabrotica virgifera zeae), Banded Cucumber Beetle (Diabrotica virgifera zeae) Diabrotica balteata), Cucurbit Beetle (Diabrotica speciosa), Bean Leaf Beetle (Cerotoma trifurcata), Cubial Leaf Beetle (Oulema melanopus), Ground Leaf Beetle (Aulacophora femoralis), Sweet potato leaf beetle (Phyllo tta striola ate leaves) Oulema oryzae), grape colapice (Colaspis brunnea), corn flare beetle (Chaetocnema pulicaria), sweet potato beetle (Chaetocnema confi), potato flare beetle (Epitrix cucum) eris), green leaf beetle (Dicladispa armigera), grape Colaspis (Colaspis brunnea), southern corn leaf beetle (Myochrous denticollis), pokeweed leaf beetle (Laccoptera quadrimacu), tobacco leaf beetle (Epitrix hirtipennis), as a member of the family Carabidae (Carabidae), such as (Stenolophus lecontei), Slender seedcorn beetle (Clivina impressifrons); Scarabaeidae (Scarabaeidae) such as European Chafer (Rhizotrogus majalis), Black Marocigan (Tomarus gibbosus), Holotrichia spp., Phyllophaga crinita etc .; Phyllophaga spp. , Imo Weevils (Euscepes postfasciatus), alfalfa snails (Hypera postica), snails (Sitophilus zeamais), rice snails (Echinocnemus squameus), rice water stalks (Lissorhoptrus oryzophilus), ss. Weevil (Sphenophorus venatus), Southern Corn Billbug (Sphenophorus callosus), Soybean stalk weevil (Sternechus subsignatus), Sgarcane wiivil (Sphenophorus levis), Sabipotanus beetle (Scepticus griseus), Tobihiro leopardian beetle subfasciatus), spinach beetle (Tomicus piniperda), Coffee Berry Borer (Hypothenemus hampei), etc. Weevil family (Curculionidae); Kokunustododoki (Tribolium castaneum), Hiratakodonokidoki (Tribolium confusum) And the like (Coccinelidae) such as Trichorididae (Tenebrionidae) and Nito-ya-boushitoto (Epilachna vigintioctopunctata) etc .; (Malasiaca), Cerambycidae such as Migdolus fryanus (Cerambycidae); Okinawa dwarf beetle (Melanotus okinawensis), Tobiyromanabosochi (Agriotes fuscicollis), Combiidae (Melanotus legatus) etc. Anchastus sp., Melanotus sp., Limonius sp., Conoderus sp., Ctenicera sp.); Staphylinidae (Staphylinidae), such as Paederus fuscipes.

  Orthopteran pests (Orthoptera): Toocta grasshopper (Locusta migratoria), Toroca grasshopper (Dociostaurus maroccanus), Australian Tobibatata (Chortoicetes terminifera), Red-footed grasshopper (Nomadacris septemfasciata), Brown Locust (Locustana pallitalucilatio) Italian Locust (Calliptamus italicus), Differential grasshopper (Melanoplus differentialis), Two striped grasshopper (Melanoplus bivittatus), Migratory grasshopper (Melanoplus sanguinipelus), Red-Legged grasshopper (Melh gregaria), Yellow-winged locust (Gastrimargus musicus), Spur-throated locust (Austracris guttulosa), Kobayinago (Oxya yezoensis), Hanekinago (Oxya japonica), Trichoderma japonicus (Patanga succi nectiograms), etc. africana) and others (Gryllotalpidae); European crickets (Acheta domesticus), European crickets (Teleogrylus emma) such as crickets (Gryllidae); Mormon cricket (Anabrus simplex) and the like.

  Hymenoptera pest (Hymenoptera): Fire ant (Solenopsis spp.) Family, Brown leaf-cutting ant (Atta capiguara) and other ant family (Formicidae), etc.

  Cockroach second order (Blattodea): German cockroach (Blattella germanica) and other German cockroaches (Blattellidae); Family (Blattidae); Yamato termites (Reticulitermes speratus), house termites (Coptotermes formosanus), American termites (Incisitermes minor), Dicta termites (Cryptotermes domesticus), Taiwan termites (Odontotermes formosanus), White-spotted termites (Glyptotermes satsumensis), Chinese termite (Glyptotermes nakajimai), Catan termite (Glyptotermes fuscus), Oolongtermite (Hodotermopsis sjostedti), N. vulgaris (Coptotermes guangzhouensis), Amami Loari (Reticulitermes amamianus), Miyatake termite (Reticulitermes miyatakei), Cameroon termite (Reticulitermes kanmonensis), Takasago termite (Nasutitermes takasagoensis), Nitobe termite (Pericapritermes nitobei), Musashi termi (Sinocapritimates) ).

  Acarid pests (Acari): Two-spotted spider mite (Tetranychus urticae), Kanzawa spider mite (Tetranychus kanzawai), Mitobine spider mite (Tetranychus evansi), an orange spider mite (Panonychus citri), an apple spider mite (Panonychus ulmi), a genus of the genus Oligonica. (Aculops pelekassi), Trichoderma sativa (Phyllocoptruta citri), Tomato saprophysus (Aculops lycopersici), Trichoderma japonicus (Calacarus carinatus), Trichoderma japonicus (Acaphylla theavagrans), Verponica sativa mite (Eriophyes chibalis ichichalis) Eriophyidae (Eriophyidae) such as Aceria diospyri, Aceria tosichella, Shevtchenkella sp., Etc .; Psinocarididae (Tarsonemidae) such as Chanophocarpus (Polyphagotarsonemus latus), etc .; Red-tailed mite (Tenuipalpidae); Red-tailed mite (Tuckerellidae); Ixodes persulcatus), black legged ticks (Ixodes scapularis), American lice mite (Amblyomma americanum), red ticks (Boophilus microplus), red lice mite (Rhipicephalus sanguineus), etc., ticks (Ixodidae); Acaridae (Acaridae) such as Trichophagus similis; Acaridae (Pyroglyphidae) such as Dermatophagoides farinae, Dermatophagoides pteronyssinus, etc .; Cheyletus er uditus), Cheyletus malaccensis, Cheyletus moorei, Cheyletiella yasguri et al. (Cheyletidae); Omitectes cynotis, Trichoderma (Sarcoptes scabiei), etc. Antipodidae (Demodicidae), such as the deciduous dog mite (Demodex canis); Leptocarpus (Listrophoridae); And the like (Dermanyssidae); Leptotrombidium akamushi etc. and the like (Trombiculidae).

Arachnid pests (Araneae): Echinochidae (Eutichuridae) such as Cheiracanthium japonicum etc .; Hemimorphidae (Theridiidae) such as Latrodectus hasseltii etc.
Ovisyasdes pests (Polydesmida): Nepheta (Oxidus gracilis), Nematode (Nedyopus tambanus) and other nematode (Paradoxosomatidae), etc.
Isopoda pests (Isopoda): Lepidoptera (Armadillidiidae) such as Armadillidium vulgare etc.

Lipopod pests (Chilopoda): Scutigeridae such as Thereuonema hilgendorfi; Scolopendra subspinipes et al. (Scolopendridae);
Gastropoda pests (Gastropoda): Limax marginatus, Limax flavus and other family Limacidae (Limacidea); And the like (Ampullariidae); and the genus Allium (Lymnaeidae) and the like, such as the Arimopeplea ollula.

  Nematoda (Nematoda): Aphelenchoides sp. (Aphelenchoides besseyi) etc. Aphelenchoididae (Aphelenchoididae); similis) and the like (Pratylenchidae); Javanese Nematode (Meloidogyne javanica), Sweet potato Nematode (Meloidogyne incognita), Northern Nematode (Meloidogyne hapla), Soybean cyst nematode (Heterodera glycines), White-tailed nematode (Globodera pallida) heterodera (Heteroderidae); Rotylenchulus reniformis et al. Hoplolaimidae; strawberry mesenchu (Nothotylenchus acris), dichilenx Anguinaceae family (Anguinidae) such as gypsy (Ditylenchus dipsaci); Tyrenculus family (Tylenchulidae) such as Tyrenculus seminetrans (Tylenchulus seminetrans); A Parasitaphelenchidae such as Bursaphelenchus xylophilus etc.

  The harmful insects and harmful acarids of the subject may be insects and acarids which have reduced drug sensitivity to insecticidal and acaricidal agents, or drug resistant. However, when the drug sensitivity is significantly reduced or drug resistance is significantly developed, it is desirable to use the composition of the present invention containing an insecticide / acaricide other than the target insecticide / acaricide.

  The compounds of the present invention can also be used to protect plants from plant diseases caused by insect-borne viruses or insect-borne bacteria.

  Such insect-borne viruses include, for example, the following.

  Rice hatching virus (Rice tungro spherical virus), rice tungro bacillus virus (Rice tungro bacilliform virus), rice grassy stunt virus (Rice grassy stunt virus), rice ragged stunt virus (Rice ragged stunt virus), rice streak dead virus ( Rice stripe virus), Rice black streaked dwarf virus, Rice southern black streaked dwarf virus, Rice gall dwarf virus, Rice hoja disease (Rice hoja) blanca virus), rice yellow leaf virus (Rice yellow stunt virus), rice yellow mottle virus, rice dwarf virus, wheat cereals northern virus (Northern cereal mosaic virus) barley yellow dwarf virus (Barley yellow dwarf virus), Barley mild mosaic virus, Barley yellow dwarf virus (Barley yellow dwarf virus-PAV), Yellow Dwarf RPS virus (Cereal yellow dwarf virus-RPS), Wheat yellow leaf virus (Wheat yellow leaf virus), Oat sterile dwarf virus, Wheat streak mosaic virus, Maize dwarf mosaic virus, Maize stripe virus, Maize stripe virus Chlorotic mottle virus, Maize chlorotic dwarf virus, Maize rayado fino virus, Sugarcane mosaic virus (Sugarcane mosaic virus), Fiji disease virus, Sugarcane yellow leaf virus Soybean mild mosaic virus, Soybean mild mosaic virus, Blueberry virus (Cycasca virus) necrotic stunt), soybean dwarf virus, milk vetch dwarf virus, soybean mosaic virus, soybean mosaic virus, alfalfa mosaic virus, bean yellow mosaic virus (Bean yellow mosaic) virus), bean mosaic virus (Bean c) ommon mosaic virus), southern bean mosaic virus (Southern bean mosaic virus), peanut rooted virus (Peanut stunt virus), broad bean wilt virus 1 (Broad bean wilt virus 1), broad bean wilt virus 2 (Broad bean wilt virus 2) , Broad bean necrosis virus (Broad bean necrosis virus), Broad bean yellow vein virus (Broad bean yellow vein virus), Clover yellow vein virus (Clover yellow vein virus), Peony mottle virus (Peanut mottle virus), Tobacco strip Mottle virus (Tobacco streak virus), Bean pod mottle virus, Cowpea chlorotic mottle virus, Mung bean yellow mosaic virus, Soybean crinkle leaf virus, Tomato chlorosis virus (Tomato chlorosis virus), Tomato spotted wilt virus (Tomato spotted wilt virus) ), Tomato yellow leaf curl virus (Tomato yellow leaf curl virus), tomato aspermy virus (T omato aspermy virus), tomato infectious chlorosis virus, potato leafroll virus, potato virus Y, melon yellow spot virus, melon Necrotic spot virus (Melon necrotic spot virus), Watermelon mosaic virus (Watermelon mosaic virus), Cucumber mosaic virus (Cucumber mosaic virus), Zucchini yellow spot mosaic virus (Zucchini yellow mosaic virus), Cub mosaic virus (Turnip mosaic virus), Cub Yellowing mosaic virus (Turnip yellow mosaic virus), cauliflower mosaic virus (Cauliflower mosaic virus), Lettuce mosaic virus (Lettuce mosaic virus), celery mosaic virus (Celery mosaic virus), beet mosaic virus (Beet mosaic virus), foliars withdrawal Green yellowing (Cucurbit chlorotic yellows virus), Capsicum chlorosis virus (Capsicum chlorosis virus), Beet pseudo yellows virus (Beet pseudo yellows virus), Leek yellow stripe virus (Leak yellow stripe virus), Onion yellow dwarf virus (Onion yellow dwarf virus) ), Sweet potato feathery mottle virus, Sweet potato shukuyo mosaic virus, Strawberry mottle virus, Strawberry mild yellow edge virus (Strawberry mild yellow edge virus), Strawberry strawberry) Pseudomild yellow edge virus (Strawberry pseudomild yellow edge virus), Strawberry crinkle virus (Strawberry crinkle virus), Strawberry vein banding virus (Strawberry vein banding virus), Japanese plum ringprint virus (plum pox virus), Chrysanthemum spruce virus (Chrysanthemum stem necrosis virus), Impatiens necrotic spot virus, Iris yellow spot virus, Lily mottle cirus, Lily symptomless virus, tulip mosaic virus etc (Tulip mosaic virus) etc.

  Examples of insect-borne bacteria include the following.

  Rice chlorosis Phytoplasma (Candidatus Phytoplasma oryzae), Candidatus Phytoplasma asteris, Maize bushy stunt phytoplasma, Citrus Asiaticus (Candidatus Liberbacter asiaticus), Citrus Africania (Candidatus Liberbacter aficannus) (Candidatus Liberbacter americanus) etc.

  The pest control method of the present invention (hereinafter referred to as the present control method) comprises the present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E and Group F. Applying the amount to the plant or to the soil on which the plant is grown. Such plants include, for example, stems and leaves of plants, seeds of plants, bulbs of plants and seedlings of plants. Here, the bulbs mean bulbs, corms, rhizomes, tubers, tubers and rhizomes, and also include so-called seeds.

  In the control method of the present invention, the compound and one or more components selected from Group A, Group B, Group C, Group D, Group E, and Group F are soils for cultivating plants or plants separately at the same time, or harmful It may be applied to habitats of organisms or pests.

  In the present invention, habitats of harmful organisms include paddy fields, upland fields, tea gardens, orchards, non-agricultural lands, nursery trays and nursery boxes, nursery soils and nursery mats, and hydroponic fluid in hydroponic farms.

  In the control method of the present invention, it is also possible to use the present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E, and Group F as they are or as they are, or to use the present composition as they are. Usually, the compound of the present invention and one or more components selected from the group A, group B, group C, group D, group E and group F are formulated, or the composition of the present invention is formulated For example, the pest may be controlled by applying it to a plant or the soil where the plant is grown, and it may be applied to the pest or the habitat of the pest in the same manner as the known pest control agent. An organism may be contacted or ingested to control pests.

  Specifically, as the application method in the control method of the present invention, for example, application to foliage of plants such as foliage application, flower vase or panicle, soil before planting or after planting (cultivation site) Application, seed disinfection and soaking, application to seeds such as seed coat, application to seedlings, application to bulbs such as seed meal, and the like can be mentioned.

  When applied to a plant or plant cultivation site, the composition of the present invention is applied one or more times. The plant or plant cultivation site may already be inhabited by the pest or may be pre-emergence.

  When applied to the pest or the habitat of the pest, the composition of the present invention is applied one or more times. The plant or plant cultivation site may already be inhabited by the pest or may be pre-emergence.

  As a method of applying to the foliage, flower vase or ear of a plant in the control method of the present invention, a method of applying to the flower vase or whole plant at flowering time including flowering before flowering, during flowering, after flowering may be mentioned. There is a method of spraying the panicle at the heading time or the whole plant.

  Other application methods include, for example, hydroponic treatment.

  Specifically, the spraying treatment in the present invention includes, for example, the present compound and Groups A, Groups B, Groups D, Groups D, Groups E and Groups on the surface of plants such as foliage spraying, trunk spraying, etc. or on pests themselves. By applying one or more components selected from F, or the composition of the present invention, it is a method of expressing pest control efficacy.

  The soil treatment in the present invention is selected, for example, from the present compound and groups A, B, C, D, E and F in the root zone of a crop to be protected from damage such as feeding by pests. A method of controlling pests directly by applying one or more components thereof, or the composition of the present invention, or controlling the pests by permeating the active ingredient from the root or the like into the inside of a plant; Specifically, for example, planting hole processing (planting hole spraying, planting hole treated soil mixing), stock source processing (stock source spraying, stock source soil mixing, stock source irrigation, rearing seedling period second half stock source processing), planting groove processing (Planting groove spraying, mixed groove soiling), rowing treatment (rowing dispersion, rowing soil mixing, growth period rowing dispersion), rowing treatment at the time of sowing (rowing dispersion at the time of sowing, rowing soil mixing at the time of sowing) Surface treatment (whole soil dispersion, whole soil mixing), side treatment, water surface treatment (water surface application, water surface after springing) Other) soil dispersion treatment (growing stage granular material foliar spray, under crown or around main stem spray, soil surface spray, soil surface mix, seed hole spray, buttock land surface spray, inter-plant spray), other irrigation treatment (soil) Irrigation, nursery season irrigation, chemical solution injection process, underground irrigation, chemical solution drip irrigation, chemistry), nursery box treatment (seedling box dispersion, nursery box irrigation, seedling box medical treatment water), nursery tray treatment (seedling tray dispersion, Seedling tray irrigation, seedling tray medical solution watering, nursery treatment (seedling dispersion, nursery irrigation, aquaculture seedling dispersion, seedling immersion), mixed treatment with floor soil (bed soil mixing, mixed bed before seeding, soiling before seeding, during seeding, At the time of sowing, it can be applied after covered soil, sprayed into soil, mixed with soil (mixed with soil, mixed with soil, mixed with soil, mixed with soil, mixed with rain), treated with potting location, sprayed with flower bunches, mixed with paste fertilizer.

  The seed treatment in the present invention is, for example, a control effect against pests by applying the active ingredient directly to or in the vicinity of seeds, seeds or bulbs of a crop to be protected from damage such as feeding by pests. Specifically, for example, spray treatment, smearing treatment, immersion treatment, impregnation treatment, coating treatment, film coating treatment, pellet coating treatment may be mentioned.

  The hydroponic solution treatment in the present invention is, for example, applying an active ingredient to the hydroponic solution etc. in order to permeate and transfer from the root to the inside of the plant body of the crop to be protected from damage such as feeding by pests. It is a method of protecting the crop from damage by pests, and specific examples thereof include water culture solution mixing, water culture solution mixing, and the like.

  In addition, a preparation containing the composition of the present invention is dipped in a plant by dipping, impregnating, coating, kneading, etc. in a sheet-like, string-like, tape-like, network-like resin, paper, cloth, etc. carrier. It can also be applied by a method such as spreading in the vicinity, spreading on the soil of origin, or covering the cultivation area of the crop.

When the control method of the present invention is used for pest control, the application amount of the present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E and Group F is the application time, application place Depending on the method of application, etc., it can be widely varied, but in general, the application rate is usually 1 to 10000 g in total of the active ingredients contained in the composition of the present invention per 10000 m ² . When the composition of the present invention is formulated into an emulsion, a wettable powder, a flowable, etc., the concentration of the total of the active ingredients contained in the composition of the present invention is usually 0.01 to 10000 ppm. Diluted and applied, and granules, dusts, etc. are usually applied as they are.

  The preparation or preparation may be sprayed directly on plants such as pests or crops to be protected from pests, or to control pests that inhabit the soil of cultivated land. It may be applied to the soil.

  The composition of the present invention can effectively control a wide range of objects in cereal fields, vegetable fields, floriculture fields, orchards or non-agricultural lands where ordinary cultivation or no-tillage cultivation is performed.

  In addition, when the present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E, and Group F, or the composition of the present invention are applied to rice, they are used in the nursery box treatment In direct sowing culture, you may use immediately after sowing.

  The time when the present compound and one or more components selected from group A, group B, group C, group D, group E and group F, or the composition of the present invention, is used for direct sowing culture of paddy rice Before, after direct sowing of paddy rice, direct application after dry seeding or after transplanting rice, specifically, before sowing, at the time of sowing, immediately after sowing, 21 days after sowing, 3 days after sowing, 21 days after sowing, or sowing From 5 days to 21 days after sowing can be mentioned.

  The time to apply the present compound and one or more components selected from group A, group B, group C, group D, group E and group F, or the composition of the present invention to a nursery box, is at the time of sowing of rice, before transplanting. Immediately after transplantation, 21 days after seeding, the day of transplantation, 3 days after transplantation to 21 days after transplantation, or 5 days after transplantation to 21 days after transplantation.

  When using the present compound and one or more components selected from group A, group B, group C, group D, group E and group F, or the composition of the present invention, the soil surface of the paddy field is in a dry state The soil surface may be wet, but may be in a wet state (water depth 0 cm), or may be watered at a water level that does not affect the application. In addition, the composition of the present invention can also be used in System of Rice Intensification (SRI).

As a plant which can use this invention composition, the following is mentioned, for example.
Maize, rice, wheat, barley, rye, triticale, oats, sorghum, cotton, soybeans, peanuts, peanuts, green beans, lima beans, azuki beans, cowpeas, mung beans, safflower beans, safflower beans, bamboo azuki beans, moth beans, tepary beans, broad beans Agricultural products such as peas, chickpeas, lentils, lupine, pigeons, alfalfa, buckwheat, sugar beet, Brassica napus, sunflower, sugar cane, tobacco etc.
Solanaceous vegetables (eggplant, tomato, pepper, pepper, bell pepper, potato), cucurbitaceous vegetables (cucumber, pumpkin, zucchini, watermelon, melon, squash etc.), cruciferous vegetables (Japanese radish, turnip, horseradish, kohlrabi, Chinese cabbage, cabbage, mustard, broccoli, cauliflower, etc., Asteraceae vegetables (burdock, shung chrysanthemum, artichoke, lettuce, etc.), Liliaceae vegetables (such as green onion, onion, garlic, asparagus), Seriaceae vegetables (carrot, parsley, celery) , American buckwheat, etc.) Anthaceae vegetables (spinach, swiss chard, etc.), sorghums (sesame, mint, basil, lavender etc.), strawberries, sweet potatoes, yams, vegetables such as taro,
Fruits (apple, pear, Japanese pear, karin, quince etc.), kernel fruits (momo, plum, nectarine, plum, apricot, apricot, prune etc), citrus fruits (palms, orange, lemon, lime, grapefruit etc) , Nuts (chestnuts, walnuts, hazelnuts, almonds, pistachios, cashews, macadamias etc), berries (blueberries, cranberries, blackberries, raspberries etc), grapes, oysters, olives, loquats, bananas, coffee, date palms, Fruit trees such as coconut palm,
Tea, mulberry, flowering tree, street tree (ASB, birch, eucalyptus, eucalyptus, eucalyptus, ginkgo, lilac, maple, oak, poplar, persimmon, persimmon, futuristic, fussus, platanus, persimmon, persimmon, birch, birch, nematode, nezu, pine, spruce, yew) Flowers, houseplants, ferns, grasses.

  The above-mentioned plant is not limited as long as it is a variety generally cultivated.

The above-mentioned plant may be a plant bred by hybrid technology.
That is, a plant bred by hybrid technology is a first-generation hybrid obtained by crossing two different lines of breed, and in general, it is possible to use heterosis (generally, yield potential) having a trait superior to that of both parents. Plants that have the characteristics of increased, resulting in increased resistance to biotic and abiotic stress factors, and the like.

  The above-mentioned plant may be a plant modified using genetic recombination technology. For example, the registered database (GM APPROVAL DATABASE) of genetically modified crops in the electronic information site (http://www.isaaa.org/) of the International Agribio Agency (INTERNATINAL SERVICE for the ACQUISITION of AGRI-BIOTECH APPLICATIONS, ISAAA) Plants listed in). More specifically, a plant to which environmental stress resistance, disease resistance, herbicide resistance, insect resistance and the like have been imparted by genetic engineering, or traits related to growth and yield, quality of products, fertility traits and the like. It may be a modified plant.

Protophyllogenogen oxidase herbicides such as flumioxazin, 4-hydroxyphenylpyruvate dioxygenases such as mesotrione (hereinafter abbreviated as HPPD) to plants that have been rendered herbicide resistant by genetic engineering techniques ) Inhibitors, acetolactate synthetase (hereinafter abbreviated as ALS) inhibitors such as imazethapyr, thifensulfuron methyl, etc. 5-enolpyruvyl shikimate 3-phosphate synthase (hereinafter abbreviated as EPSPS) inhibitions such as glyphosate etc. Also included are plants to which resistance to herbicides such as agents, glutamine synthetase inhibitors such as glufosinate, auxin type herbicides such as 2,4-D, dicamba, and bromoxynil have been imparted by genetic engineering techniques.
Glyphosate resistant EPSPS gene (CP4 epsps) derived from Agrobacterium (Agrobacterium tumefaciens strain CP4) and glyphosate metabolizing enzyme derived from Bacillus licheniformis as an example of a plant to which herbicide resistance has been imparted by genetic recombination technology Glyphosate metabolizing enzyme genes (gat 4601, gat 6421) whose metabolic activity has been enhanced by shuffling (glyphosate N-acetyl transferase) gene, glyphosate metabolizing enzyme (glyphosate oxidase gene, goxv 247) from Ochrobacterum anthropi strain LBAA, Alternatively, there are glyphosate-resistant transgenic plants into which one or more EPSPS genes (mepsps, 2 mepsps) having a glyphosate-resistant mutation derived from maize have been introduced. Corn (Zea mays L.), soybean (Glycine max L.), cotton (Gossypium hirsutum L.), sugar beet (Beta vulgaris), canola (Brassica napus, Brassica rapa), alfalfa (Medicago sativa), potato (Solanum tuberrosum L.) Glyphosate resistant transgenic varieties of plants such as wheat) (Triticum aestivum), creeping bentgrass (Agrostis stolonifera) and the like.
Several glyphosate resistant transgenic plants are commercially available. For example, a transgenic plant expressing glyphosate-resistant EPSPS derived from Agrobacterium is a trade name including Roundup Ready (registered trademark), and expresses a glyphosate-metabolizing enzyme derived from Bacillus which has enhanced metabolic activity by shuffling technology. Genetically modified plants are trade names such as Optimum (registered trademark) GAT (registered trademark), Optimum (registered trademark) Gly canola etc., and genetically modified plants expressing EPSPS having a glyphosate resistant mutation derived from corn are GlyTol (registered trademark) It is already sold under the brand name).
Similarly, phosphinothricin N-acetyltransferase (Phosphinothricin N-acetyltransferase, PAT), which is a glufosinate-metabolizing enzyme derived from Streptomyces hygroscopicus, as an example of a plant to which herbicide resistance has been imparted by genetic engineering techniques. Glucosinate-resistant transgenic plant into which a gene (bar), a phosphinothricin N-acetyltransferase gene (pat) which is a glufosinate-metabolizing enzyme derived from Streptomyces viridochromogenes, or a synthesized pat gene etc. is introduced There is. There are glufosinate resistant transgenic varieties of plants such as corn, soybean, cotton, canola, rice (Oryza sativa L.), sugar beet, chicory (Cichorium intybus).
Several glufosinate resistant transgenic plants are commercially available. Transgenic plants expressing glufosinate metabolizing enzymes (bar, pat) from Streptomyces bacteria are already marketed under the tradenames containing LibertyLink®.
Similarly, as an example of a plant to which herbicide resistance has been imparted by genetic recombination technology, a genetic modification of bromoxynil resistance which has been introduced a nitrilase gene (bxn), which is a bromoxynil metabolism enzyme from Klebsiella pneumoniae subsp. Ozaenae There is a plant. Bromoxinyl-resistant transgenic varieties are produced in plants such as canola, cotton, tobacco (Nicotiana tabacum L.) and are already sold under the trade names including Navigator® canola or BXN® .
Similarly, as an example of a plant to which herbicide resistance has been imparted by genetic recombination technology, genetically modified carnation (Dianthus caryophyllus) in which a tobacco-derived ALS herbicide-resistant ALS gene (surB, S4-HrA) has been introduced as a selection marker. ). Also, a transgenic flax (Linum usitatissumum L.) into which an ALS herbicide resistant ALS gene derived from Arabidopsis thaliana (Arabidopsis thaliana) has been introduced has been developed under the trade name CDC Triffid Flax. Also, a genetically modified soybean into which an ALS herbicide-resistant ALS gene (csr1-2) derived from Arabidopsis thaliana has been introduced has been developed under the name of Culture®. Furthermore, genetically modified maize resistant to sulfonylurea type and imidazolinone type herbicides into which ALS herbicide resistant type ALS gene (zm-hra) derived from corn has been introduced, and ALS herbicide resistant type ALS gene derived from soybean (gm- There are genetically modified soybeans that are resistant to sulfonylurea herbicides into which hra) has been introduced.
Similarly, as an example of a plant to which herbicide resistance has been imparted by genetic engineering technology, isoxaflutole resistance gene combination introduced HPPD herbicide resistant HPPD gene (hppdPFW336) derived from Pseudomonas fluorescens strain A32 There are modified soybeans and mesotrione resistant transgenic soybeans into which the HPPD gene (avhppd-03) derived from oat (Avena sativa) has been introduced.
Similarly, as an example of a plant to which herbicide resistance has been imparted by genetic engineering technology, an aryloxyalkanoate dioxygenase, which is a 2,4-D metabolizing enzyme derived from Sphingobium herbicidovorans, is known. ), 2,4-D resistance into which the gene (aad-1) or the allyloxyalkanoate dioxigenase gene (aad-12), which is a 2,4-D metabolizing enzyme derived from Delftia acidovorans, is introduced The genetically modified maize, genetically modified soybean, genetically modified cotton and the like are some of which are developed under the trade names Enlist® Maize, Enlist® Soybean. In addition, dicamba-resistant genetically-modified soybean, genetically-modified cotton, etc. into which dicamba monooxygenase (Dicamba monooxygenase) gene (dmo), which is a dicamba metabolic enzyme derived from Stenotrophomonas maltophilia strain DI-6, has been introduced. is there.
Similarly, as an example of a plant that has been rendered tolerant to two or more herbicides by genetic engineering, a genetically modified cotton that is resistant to both glyphosate and glufosinate, a genetically modified maize is GlyTol® LibertyLink (R), which is already sold under the trade name Roundup Ready (R) LibertyLink (R) Maize. Also, a genetically modified soybean that is resistant to both glufosinate and 2,4-D is developed under the trade name Enlist® Soybean, and a genetically modified cotton that is resistant to both glufosinate and 2,4-D. There is also. A genetically modified soybean that is resistant to both glyphosate and dicamba is being developed under the trade name Genuity® Roundup Ready® 2 Xtend®. Genetically modified corn, soybean, which is resistant to both glyphosate and ALS inhibitors, is being developed under the trade name Optimum® GAT®. Besides, transgenic cotton resistant to both glufosinate and dicamba, genetically modified corn resistant to both glyphosate and 2,4-D, genetically modified soybean resistant to both glyphosate and HPPD herbicide Is also being developed. In addition, genetically modified soybeans that are resistant to glyphosate, glufosinate and three herbicides of 2,4-D have also been developed.

Examples of plants that have been imparted with insect resistance by genetic engineering techniques include plants that have been imparted with resistance to lepidopteran insects, coleopteran insects, insects of the order Two orders of order, and the like.
As an example of a plant that has been rendered resistant to lepidopteran insects by genetic engineering technology, a delta-endotoxin (δ-endotoxin), which is an insecticidal protein derived from soil bacteria Bacillus thuringiensis (hereinafter abbreviated as Bt bacteria), is encoded. And transgenic plants such as corn, soybean, cotton, rice, poplar (Populus sp.), Tomato (Lycopersicon esculentum), eggplant (Solanum melongena), etc. into which the gene for As a delta-endotoxin imparting resistance to lepidopteran insects, Cry1A, Cry1Ab, modified Cry1Ab (partially deleted Cry1Ab), Cry1Ac, Cry1Ab-Ac (hybrid protein in which Cry1Ab and Cry1Ac are fused), Cry1C, Cry1F , Cry1Fa2 (modified cry1F), moCry1F (modified Cry1F), Cry1A. 105 (a hybrid protein in which Cry1Ab, Cry1Ac, Cry1F is fused), Cry2Ab2, Cry2Ae, Cry9C, Vip3A, Vip3Aa20 and the like.
As an example of a plant which has been rendered resistant to a coleoptera by a genetic recombination technique, a transgenic plant such as maize or potato introduced with a gene encoding delta-endotoxin which is an insecticidal protein derived from soil bacterium Bt bacteria There is a plant. Examples of delta-endotoxin imparting resistance to coleopteran insects include Cry3A, mCry3A (modified Cry3A), Cry3Bb1, Cry34Ab1, Cry35Ab1 and the like.
As an example of a plant to which a resistance to Dipteran insects has been imparted by genetic recombination technology, a gene set in which a synthetic gene encoding a hybrid protein eCry3.1Ab is fused, which is a fusion of Cry3A derived from soil bacteria Bt bacteria and Cry1Ab. A transgenic maize, a transgenic cotton into which a gene encoding a trypsin inhibitor CpTI derived from cowpea (Vigna unguiculata) has been introduced, a gene combination into which a gene encoding an API which is a protease inhibitor protein A derived from Sagittaria sagittifolia is introduced There is a change poplar etc.
Insecticidal proteins that impart insect resistance to plants include hybrid proteins of the above insecticidal proteins, partially deficient proteins, and modified proteins. Hybrid proteins are produced by the combination of different domains of multiple insecticidal proteins using genetic engineering techniques, such as Cry1Ab-Ac or Cry1A. 105 mag is known. As proteins in which a part has been deleted, Cry1Ab or the like in which a part of the amino acid sequence has been deleted is known. As modified proteins, proteins in which one or more amino acids of natural delta-endotoxin are substituted, such as Cry1Fa2, moCry1F, mCry3A, etc. are known.
In addition, insecticidal proteins derived from Bacillus cereus and Bacillus popilliae (Bacillus popilliae), and insecticidal proteins derived from Bt bacteria Vip1 as insecticidal proteins that impart insect resistance to plants by genetic recombination techniques , Vip2, Vip3, insecticidal proteins from nematodes, scorpion toxins, spider toxins, spider toxins, toxins produced by animals such as bee toxins or insect specific neurotoxins, filamentous fungal toxins, plant lectins, agglutinin, trypsin inhibitors, serine Protease inhibitors, Protease inhibitors such as patatin, cystatin, papain inhibitors, Lysine, corn-RIP, abrin, luphin, saporin, ribosomal inactivated proteins (RIP) such as briosin, 3-hydroxysteroid oxidase, ecdysteroids -UDP-glucosyltrans Steroid metabolism enzymes such as cholesterol oxidase, ecdysone inhibitors, HMG-CoA reductase, ion channel inhibitors such as sodium channels, calcium channel inhibitors, juvenile hormone esterase, diuretic hormone receptor, stilbene synthase, bibenzyl synthase, Chitinase, glucanase and the like can be mentioned.

In addition, transgenic plants that have been rendered pest resistant by introducing one or more insecticidal protein genes are already known, and some transgenic plants are commercially available.
As an example of a genetically modified cotton which has been imparted with pest resistance, Bollgard (registered trademark) cotton which expresses the insecticidal protein Cry1Ac derived from Bt bacteria, Bollgard II (registered trademark) which expresses the insecticidal proteins Cry1 Ac and Cry2Ab derived from Bt bacteria ) Cotton, Bt bacteria-derived insecticidal protein Cry1Ac, Cry2Ab, Bollgard III (R) expressing Vip3A, Bt cell-derived insecticidal proteins Vip3A and Cry1Ac expressing VIPCOT (registered trademark), Bt cell-derived insecticidal A transgenic cotton having a trade name including WideStrike (registered trademark) that expresses the proteins Cry1Ac and Cry1F is commercially available.
As an example of genetically modified maize to which insect resistance has been imparted, YieldGard® Rootworm RW expressing the insecticidal protein Cry3Bb1 derived from Bt fungus, YieldGard Plus expressing the insecticidal proteins Cry1Ab and Cry3Bb1 derived from Bt bacterium (Trademark), an insecticidal protein Cry1A. YieldGard (registered trademark) VT Pro (registered trademark) and the like expressing 105 and Cry2Ab2 are commercially available. Agrisure® RW that expresses the insecticidal protein mCry3A derived from Bt fungus, Agrisure® Viptera which expresses the insecticidal protein Vip3Aa20 derived from Bt bacterium, Agrisure that expresses the insecticidal protein eCry3.1 Ab derived from Bt bacterium (Registered trademark) Duracade (registered trademark) and the like are also commercially available.
As an example of a genetically modified potato to which pest resistance has been imparted, Atlantic NewLeaf (registered trademark) potato, NewLeaf (registered trademark) Russell set Burbank potato, etc. expressing the insecticidal protein Cry3A derived from Bt bacteria are commercially available.

Plants that have been rendered disease resistant by genetic engineering techniques are beans (Phaseolus vulgaris), papaya (Carica papaya), plums (Prunus domestica), potatoes, squash (Cucurbita pepo) that have been rendered resistant to plant virus diseases. , Sweet pepper (Capsicum annuum), tomato and the like. Specifically, a transgenic plant that has been rendered resistant to plant virus disease, specifically, a gene set into which a gene that produces a double-stranded RNA of a bean golden mosaic virus replication protein is introduced. Replacement bean, Genetically modified papaya into which the coat protein gene of Papaya ringspot virus (Papaya ringspot virus) has been introduced, coat protein gene of potato virus Y (Potato virus Y), or potato leaf roll virus ( A transgenic potato in which a replicative enzyme domain gene of Potato leaf roll virus has been introduced, a coat protein gene of cucumber mosaic virus, a coat protein gene of watermelon mosaic virus, zucchini・ Yellow ・ Mosaic · Genetically engineered squash into which the coat protein gene of virus (Zucchini yellow mosaic virus) has been introduced, genetically modified sweet pepper into which the coat protein gene of cucumber mosaic virus (Cucumber mosaic virus) has been introduced, transgenic tomato etc. is there.
As an example of a genetically modified potato which has been rendered resistant to plant virus diseases, a genetically modified potato having a trade name including Newleaf (registered trademark) is commercially available.
Plants that have been given disease resistance also include plants that have been given the ability to produce anti-pathogenic substances that have selective effects using genetic engineering techniques. As an example of the antipathogenic substance, infection specific proteins (PR proteins) and the like are known (PRPs, EP392225). Such anti-pathogenic substances and transgenic plants producing them are described in EP392225, WO199533818, EP353191 and the like. Examples of anti-pathogenic substances include ion channel inhibitors such as sodium channel inhibitors, calcium channel inhibitors (virus-produced KP1, KP4 and KP6 toxins are known), stilbene synthase, biphenyl Produced by microorganisms such as benzyl synthase, chitinase, glucanase, peptide antibiotics, antibiotics having heterocycles, protein factors involved in plant disease resistance (called plant disease resistance genes and described in WO2003000906) Anti-pathogenic substances and the like.

For plants whose product quality has been modified by genetic engineering technology, modification of lignin production, modification of oil or fatty acid component, production of phytic acid degrading enzyme, modification of flower color, modification of alpha-amylase activity, modification of amino acid , Modification of starch or carbohydrate components, suppression of acrylamide formation, reduction of black spots due to mechanical damage, antiallergic properties, reduction of nicotine production, genetically modified plants with modified product quality such as aging or delayed ripening are mentioned Be
Alfalfa-derived S-adenosyl-L-methionine: trans-caffeoyl-CoA 3-methyltransferase (ccomt) gene involved in lignin production was introduced to generate double-stranded RNA and lignin content was reduced by RNA interference. There is a recombinant alfalfa.
Genetically modified canola with increased triacylglyceride content including lauric acid by introducing 12: 0 ACP thioesterase gene from laurier (Umbellularia californica) involved in fatty acid synthesis under the trade name Laurical® Canola It is being developed.
A recombinant canola that has enhanced the degradation of endogenous phytic acid by introducing the 3-phytase gene (phyA) from Aspergillus niger, which is a phytic acid degrading enzyme of plants, is Phytased ® Canola It has been developed under the trade name. Similarly, genetically modified maize has been developed, in which the degradation of endogenous phytic acid is enhanced by introducing the 3-phytase gene (phyA) from black mold.
A blue pigment delphinidin and an enzyme that produces the derivative thereof, a dihydroflavonol-4-reductase gene from petunia (Petunia hybrida) and a petunia, a pansy (Viola wittrockiana), a salvia (Salvia splendens), or a flavonoid derived from a carnation There is known a recombinant carnation whose flower color is controlled to blue by introducing a -3 ', 5'-hydroxylase gene. Genetically modified carnations in which the flower color is controlled to blue are: Moondust (registered trademark), Moonshadow (registered trademark), Moonshade (registered trademark), Moonlite (registered trademark), Moonaqua (registered trademark), Moonvista (registered trademark), Moonique (registered trademark) (Trademark), Moonpearl (trademark), Moonberry (trademark), Moonvelvet (trademark), etc. are developed by brand names. Also, by introducing anthocyanin-5-acyltransferase gene derived from torenia (Torenia sp.), Which is an enzyme that produces the blue pigment delphinidin and its derivative, and a flavonoid-3 ′, 5′-hydroxylase gene derived from pansy Genetically modified roses have also been developed in which the flower color is controlled to be blue.
Some genetically modified corns have enhanced bioethanol production by introducing the thermostable alpha-amylase gene (amy 797E) of Thermococcals sp. For starch degradation, under the trade name Enogen®. It is being developed.
Genetically modified maize containing Mavera® contains enhanced lysine production by introducing the dihydrodipicolinate synthetase gene (cordapA) from Corynebacterium glutamicum for the production of the amino acid lysine It has been developed under the trade name.
Genetically modified melon and transgenic tomato have been developed with improved shelf-life by introducing the S-adenosyl methione hydrolase gene (sam-K) from E. coli bacteriophage T3 for plant hormone ethylene production . In addition, a gene lacking a part of the tomato ACC-related enzyme gene involved in ethylene production of plant hormone, an ACC deaminase gene from Pseudomonas chlororaphis that decomposes ACC, which is an ethylene precursor, and a pectin in the cell wall are degraded We have also developed a transgenic tomato whose shelf life has been improved by introducing a double-stranded RNA gene of the tomato-derived polygalacturonase gene or a tomato-derived ACC oxidase gene involved in the production of ethylene. ing. A transgenic tomato whose shelf life has been improved by introducing a gene that produces double-stranded RNA of the tomato-derived polygalacturonase gene has been developed under the trade name of FLAVR SAVR®.
A gene producing a double-stranded RNA of a transcription factor gene promoting starch degradation from potato, a gene producing a double-stranded RNA of a polyphenol oxidase gene derived from potato, and a double-stranded RNA of a gene involved in asparagine production A product that includes Innate (R), a genetically modified potato in which the degradation of starch, the formation of black spots due to mechanical damage, and the possibility of carcinogenic substance (acrylamide) formation due to heating are reduced by introducing genes It is being developed by the name. In addition, a recombinant potato having a reduced amylose content by introducing an antisense gene of a potato synthase-derived starch synthetase has been developed under the trade name of Amflora (registered trademark).
By introducing a modified cedar pollen antigen protein gene (7 crp), a transgenic rice having an effect of alleviating hay fever in immune tolerance has been developed.
Genetically modified soybean in which the expression of the same gene is suppressed and oleic acid content is enhanced by introducing a partial gene (gm-fad2-1) of ω-6 desaturase derived from soybean that is a desaturase of fatty acid, Plenish ( It is developed under the trade name of registered trademark) or Treus (registered trademark). In addition, a gene for producing a double-stranded RNA of an acyl-acyl carrier protein protein thioesterase gene (fatb1-A) derived from soybean, and a double-stranded RNA of a δ-12 desaturase gene (fad2-1A) derived from soybean A genetically modified soybean whose saturated fatty acid content has been reduced by introducing the resulting gene has been developed under the trade name of Vistive Gold®. Also, a genetically modified soybean has been developed in which the content of ω3 fatty acid is enhanced by introducing the δ-6 desaturase gene (Pj. D6D) derived from primrose and the δ-12 desaturase gene (Nc. Fad3) derived from Neurospora crassa There is.
A transgenic tobacco has been developed in which the nicotine content is reduced by introducing an antisense gene of the quinolinate phosphoribosyltransferase gene (NtQPT1) derived from tobacco.
Endothelial tissue β is expressed specifically by introducing the phytoene synthase gene (psy) from trumpet spinach (Narcissus pseudonarciss) and the carotene desaturase gene (crt1) from the soil bacteria (Erwinia uredovora) that synthesizes carotenoids and expressing them specifically in the endosperm -Golden rice, a transgenic rice plant that can produce carotene and harvest rice containing vitamin A, has also been developed.

Examples of the plant whose fertility trait or the like has been modified by genetic recombination techniques include a plant having a male sterility and a fertility restoration trait imparted thereto. There are transgenic corn and transgenic chicory in which a male sterility trait has been imparted by expressing a ribonuclease gene (barnase) derived from Bacillus amyloliquefaciens in a tapetum cell of silkworm. In addition, there is also a transgenic corn which has been given a male sterility trait by introducing a DNA adenine methylase gene (dam) derived from E. coli. Furthermore, a gene combination in which the fertility trait is controlled by introducing a maize-derived alpha-amylase gene (zm-aa1) giving a male sterility trait and a maize-derived ms45 protein gene (ms45) giving a fertility recovery trait There is also a change corn.
There is a recombinant canola to which a fertility recovery function has been imparted by expressing a ribonuclease inhibitory protein gene (barstar) derived from Bacillus subtilis in silkworm tapetum cells. In addition, a gene set whose fertility trait has been controlled by expressing a ribonuclease gene (barnase) derived from Bacillus bacteria that gives a male sterility trait and a ribonuclease inhibitory protein gene (barstar) derived from Bacillus bacteria that gives a fertility recovery trait There is also a replacement canola.

  Plants to which environmental stress resistance has been imparted by genetic recombination techniques include transgenic plants to which drought tolerance has been imparted. A dry tolerant maize into which a low temperature shock protein gene (cspB) derived from Bacillus subtilis has been introduced has been developed under the brand name Genuity® DroughtGard®. Furthermore, a drought resistant sugar cane has been developed in which a choline dehydrogenase gene (RmBetA) derived from alfalfa rhizobium (Rhizobium meliloti) or E. coli (Esherichia coli) has been introduced.

  Examples of plants whose traits related to growth and yield have been modified by genetic recombination techniques include genetically modified plants having enhanced growth ability. For example, genetically modified soybeans and the like have been developed in which a gene (bbx32) encoding a transcription factor that controls diurnalities derived from Arabidopsis thaliana has been introduced.

The above-mentioned plant may be a plant modified using a technique other than genetic recombination technology. More specifically, it may be a plant to which environmental stress resistance, disease resistance, herbicide resistance, pest resistance or the like has been imparted by classical breeding technology, gene marker breeding technology, genome editing technology or the like.
Examples of plants that have been rendered herbicide-resistant by classical or genetic marker breeding techniques include corn, rice, wheat, sunflower (Helianthus annuus), canola, tolerant to imidazolinone-based ALS-inhibiting herbicides such as imazethapyr. Lentils (Lens culinaris) etc. are sold under the trade name Clearfield®. Moreover, STS soybean which is a sulfonylurea type herbicide resistant soybean etc. is mentioned as an example of the plant in which resistance with respect to sulfonyl type ALS inhibition type | mold herbicides, such as thifensulfuron methyl, etc. was provided by the classical or gene marker breeding technique. Similarly, SR corn and the like, which are cetoxidimium-resistant maize, are examples of plants which are tolerant to acetyl CoA carboxylase inhibitors such as trione oxime type and aryloxy phenoxy propionic acid type herbicides by classical or genetic marker breeding techniques. is there.
Examples of plants that have been given pest resistance by classical or genetic marker breeding techniques include soybeans that have the aphid resistance gene Rag1 (Resistance Aphid Gene 1) gene. In addition, examples of plants to which the resistance to nematode has been imparted by the classical breeding method include soybeans which have been imparted with resistance to cysto nematode, cotton which has been imparted with resistance to root knot nematode, and the like.
As a plant that has been rendered disease resistant by classical or genetic marker breeding techniques, it is conferred resistance to corn, Gray leaf spot, which is resistant to Anthracnose stalk rot. Maize, Maize resistant to Goss`s wilt, Maize resistant to Fusarium stalk rot, Maize resistant to Asian soybean rust Soybeans, peppers resistant to Phytophthora, lettuce resistant to powdery mildew, tomatoes resistant to Bacterial wilt, Geminivirus Examples include tomato which has been imparted with resistance, and lettuce which has been imparted with resistance to downy mildew.
As an example of a plant that has been rendered drought tolerant by classical or genetic marker breeding techniques, drought tolerant corn has been developed under the trade name Agrisure Artesian®, Optimum AQUAmax®.
Also, as an example of a plant to which herbicide resistance has been imparted by genome editing technology, the sulfonylurea type is a rapid variety development technology that introduces a sulfonylurea type herbicide resistance mutation into the ALS gene via a chimeric oligonucleotide of DNA and RNA. A herbicide tolerant canola has been developed under the tradename SU Canola®.

In the above-mentioned plants, environmental stress resistance, disease resistance, herbicide resistance, pest resistance, as described above, using genetic recombination technology, classical breeding technology, gene marker breeding, genome editing technology etc. Two or more types of properties possessed by the parent line by multiplying plants with two or more types of growth and yield traits, product quality, fertility traits, etc. and genetically modified plants having similar or different properties It also includes the strain given. An example of such a plant is a transgenic plant to which both herbicide resistance and pest resistance have been imparted.
For example, Roundup Ready (registered trademark) Bollgard (registered trademark) cotton, Roundup Ready (registered trademark) Bollgard II (registered trademark) cotton, Roundup Ready (registered trademark) as a Glyphosate-resistant and pest-resistant transgenic plant. Trade names such as Flex (registered trademark) Bollgard II (registered trademark) Cotton, Bollgard (registered trademark) III x Roundup Ready (registered trademark) Flex (registered trademark), and VIPCOT (registered trademark) Roundup Ready Flex (registered trademark) Cotton Genetically modified cotton has been developed. In addition, Agrisure (registered trademark) GT / RW, Roundup Ready (registered trademark) YieldGard (registered trademark) maize, Genuity (registered trademark) VT Double Pro (registered trademark), and Genuity (registered trademark) VT Triple Pro (registered trademark), YieldGard (R), YieldGard (R) CB + RW, YieldGard (R) VT (R) Rootworm (R) RR2, YieldGard (R) RW + RR, YieldGard (R) VT Triple, YieldGard (R) Genetically modified corn having a trade name such as Plus with RR has been developed. In addition, genetically modified soybeans such as Intacta (R) Roundup Ready (R) 2 Pro have also been developed.
For example, products such as Widestrike (registered trademark) Cotton, Twinlink (registered trademark) Cotton, Fibermax (registered trademark) LibertyLink (registered trademark) Bollgard II (registered trademark), and the like as a genetically modified plant that is given glufosinate resistance and pest resistance The name transgenic cotton has been developed. In addition, Agrisure (registered trademark) CB / LL, Agrisure (registered trademark) CB / LL / RW, Agrisure (registered trademark) Viptera (registered trademark) 2100, Agrisure (registered trademark) Viptera (registered trademark) 3100, Bt Xtra (registered trademark) Trademarks Maize, NaturGard Knockout (R), Herculex (R) RW, Herculex (R) CB, Herculex (R) XTRA, Starlink (R) Maize, Liberty Link (R) YieldGard (R) Genetically modified corn having a trade name such as Maize has been developed.
For example, Glyphosate-resistant, glufosinate-resistant, and pest-resistant genetically modified plants include Widestrike (R) Roundup Ready (R) Cotton, Widestrike (R) Roundup Ready Flex (R) Cotton, Widestrike A transgenic cotton having a trade name, such as Registered Trademark x Roundup Ready Flex (registered trademark) x VIPCOT (registered trademark) Cotton, Glytol (registered trademark) x Twinlink (registered trademark), has been developed. Also, Agrisure (registered trademark) GT / CB / LL, Agrisure (registered trademark) 3000 GT, Agrisure (registered trademark) 3122, Agrisure (registered trademark) Viptera (registered trademark) 3110, Agrisure (registered trademark) Viptera 3111, Agrisure (registered) Trademarks Viptera 3220, Agrisure (R) Duracade (R) 5122, Agrisure (R) Duracade (R) 5222, Optimum (R) Intrasect, Optimum (R) TRIsect, Optimum (R) Intrasect XTRA Optimum® Intrasect Xtreme, Genuity® SmartStax®, Power Core®, Herculex® I RR, Herculex® RW Roundup Ready® 2, Herculex Genetically modified corn having a trade name such as XTRA (registered trademark) RR has been developed.
For example, a transgenic cotton having a trade name such as BXN (registered trademark) Plus Bollgard (registered trademark) Cotton has been developed as a transgenic plant imparted with bromoxynil resistance and pest resistance.

An example of a line to which two or more of the above-mentioned plural traits are imparted is a transgenic plant to which disease resistance and pest resistance are imparted. For example, Hi-Lite NewLeaf (registered trademark) Y Potato, NewLeaf (registered trademark) Y Russet Burbank Potato, and Shepody NewLeaf (registered trademark) as a genetically modified plant that has been given potato virus Y (Potato virus Y) resistance and pest resistance. (Trademark) Y Potato, or a gene set having a trade name such as NewLeaf (registered trademark) Plus Russet Burbank Potato etc. as a transgenic plant that has been imparted with potato leaf roll virus resistance and pest resistance. Replacement potatoes have been developed.
An example of a line to which two or more of the above-mentioned plural traits are imparted is a transgenic plant to which a herbicide resistance and a modified product quality have been imparted. For example, genetically modified canola or genetically modified corn imparted with glufosinate resistance and dwarf character is being developed under the trade names InVigor® Canola, InVigor® Maize.
As an example of a line to which two or more of the above-mentioned plural traits are imparted, there is a transgenic plant to which pest resistance and modified product quality are imparted. For example, a genetically modified maize having a trait that enhances resistance to lepidopteran pests and lysine production has been developed under the trade name Mavera® YieldGard® Maize.
In addition, as an example of a line to which two or more kinds of multiple traits described above are given, a transgenic plant to which a herbicide tolerance and a modified fertility trait are given, a gene to which a herbicide tolerance and an environmental stress tolerance are given Recombinant plants, genetically modified plants having herbicide resistance and modified growth and yield traits, genetically modified plants having herbicide resistance, pest resistance and modified product quality, and herbicides Genetically modified plants and the like to which resistance, pest resistance and environmental stress resistance have been imparted have been developed.

  Furthermore, a plurality of useful traits such as the above-mentioned classical herbicide traits or herbicide resistance genes, insecticidal pest resistance genes, antipathogenic substance producing genes, oil component modification and amino acid content enhancement traits are listed. It also includes combined stack varieties. Also included are plants into which RNAi technology has been introduced.

  The present compound and one or more components selected from Group A, Group B, Group C, Group D, Group E and Group F, or the application of the composition of the present invention, plant species or plant varieties, their place of growth and growth Depending on the conditions (soil, climate, growing season, nutrients), the growth of plants is enhanced, the resistance to high or low temperature or tolerance is improved, the tolerance to drought in water or salt contained in the soil, the ability to flower Improve, improve harvestability, promote maturation, increase yield, increase fruit size, increase plant height, improve leaf green color, faster flowering, harvested product quality In some cases, it may be possible to improve and / or increase the nutritive value, increase sugar content in fruits, improve gluten strength, improve storage stability of harvested products, and / or improve processability.

  The compound and a specific herbicide, or the compound and a specific herbicide and one or more components selected from Group A, Group B, Group C, Group D, Group E, and Group F, by any method By applying it to a given crop, it is also possible to obtain a high "crop growth improvement effect" effectively and labor-saving. Here, the "crop growth improvement effect" means that the crop yield is increased as a result of controlling insect pests, diseases and weed pests of crops.

  Specifically, imidazolinone herbicides such as imidazolinone herbicides such as Clearfield® canola, imidazolinone herbicides such as the present compound and imazapyr, or imidazolinone herbicides such as the present compound, imazapyr and the like And one or more components selected from group A, group B, group C, group D, group E and group F can be applied at the same time or at different times to improve the growth of Clearfield canola.

  In addition, the present compound and glyphosate, or the present compound, glyphosate and Group A, Group B, Group C, Group D, Group D, to a glyphosate-tolerant crop, for example, RoundupReady (registered trademark) cotton or RoundupReady 2 soybean (registered trademark) One or more products selected from E and Group F can be applied at the same time or at different times to improve the growth of RoundupReady cotton and RoundupReady 2 soybean.

  In addition, the compound and glufosinate, or the compound, glufosinate and Group A, Group B, Group C, Group D, Group E, and Group F are selected from a glufosinate-resistant crop, for example, LibertyLink® corn. The growth of LibertyLink corn can be improved by applying one or more ingredients at the same time or at different times.

  In the control method of the present invention, the present compound, one or more components selected from group C, and one or more components selected from group E can also be applied in combination. The application method of one or more components selected from group E is not particularly limited, but it can be applied together with one or more components selected from group C, in which case one or more components selected from group C A preparation containing one ingredient and one or more ingredients selected from group E may be used alone, or a preparation containing one or more ingredients selected from group C and one or more ingredients selected from group E May be used in combination with a preparation containing Alternatively, plant seeds or bulbs can be used which carry one or more components selected from group E. Plant seeds or bulbs may be used after retaining one or more components selected from group E, or a commercially available seed retaining one or more components selected from group E may be purchased You may use it.

  In the control method of the present invention, when one or more components selected from group C are contained as an active ingredient, it is time to apply one or more components selected from group C before sowing or planting plant seeds, bulbs or seedlings For example, 50 days before sowing or planting to just before sowing or planting, 30 days before sowing or planting to just before sowing or planting, 20 days before sowing or planting to just before sowing or planting, or 10 days before sowing or planting Or just before planting can be mentioned.

  The time to apply one or more components selected from group C after sowing or planting of plant seeds, bulbs or seedlings is, for example, immediately after sowing or planting to 50 days after sowing or planting, or immediately after sowing to 3 days after sowing It can be mentioned.

  It is also possible to treat one or more components selected from group C simultaneously with planting, planting or planting seeds or bulbs.

  In the control method of the present invention, when one or more components selected from group C are contained as an active ingredient, as a specific application time when applying one or more components selected from group C after sowing of soybean seeds For example, it may be between the pre-emergence stage and the flowering stage of soybean. The period from before the emergence of soybean to the flowering stage is, for example, from the period before the emergence of soybean to the time of six double leaves, and the period before the emergence of soybean to the time of three double leaves.

  As a specific application time when applying one or more components selected from group C after sowing of corn seeds, for example, between the pre-emergence to 12-leaf stage and the pre-emergence to 8-leaf stage, The period from before budding to 6 leaf stage is mentioned. The leaf age of corn is determined by the leaf color method (Leaf Collar Method).

  As a time to apply one or more components selected from group C before sowing of cotton seeds, for example, 50 days before sowing-just before sowing, 30 days before sowing-just before sowing, 20 days before sowing-just before sowing are mentioned Be

  The herbicide is treated immediately after sowing-70 days after sowing, preferably 30 days after sowing-50 days after sowing of the seeds of cotton seed after sowing. As a specific treatment time in the case of treating a herbicide after sowing of cotton seeds, for example, between before the emergence of cotton and during the flowering stage, the larching stage of the stem base of cotton and the larch at 20 cm from the base The period is mentioned.

  The time to apply one or more components selected from Group C before planting sugar cane includes 40 days to immediately before planting, 30 days to immediately before planting, and 20 days to immediately before planting.

  As a time to apply one or more components selected from group C after planting sugar cane, immediately after planting-40 days after planting day, immediately after planting-20 days after planting day Immediately after wearing ~ 10 days after the planting day.

  Examples of the above-mentioned herbicides, safeners and plant growth regulators include those of the above-mentioned Group C, Group D and Group E.

  As one or more components selected from Group C above, flumioxazin, sulfentrazone, saflufenacil, oxyfluorfen, fomethafen, fomethafen sodium, glufosinate ammonium salt, chlorimuron ethyl, chloruramram methyl, piroqui Sasulfone, imazethapyr ammonium salt, metribuzin, 2,4-D, 2,4-D buttyl ester, 2,4-D dimethyl ammonium salt, 2,4-D diolamine salt, 2,4-D ethylhexyl Ester, 2,4-D isocutyl ester, 2,4-D isopropyl ammonium salt, 2,4-D sodium salt, 2,4-D triisopropanolamine salt, 2,4-D choline salt, dicamba, dicambadi Glycolamine salt, dicamba dimethyl ammonium salt, dicamba Isopropyl ammonium salt, dicamba potassium salt, dicamba sodium salt, Jikanbakorin salts, mesotrione, tembotrione, isoxaflutole and ametryn are preferred.

  Specific examples of the control target of the composition of the present invention include, but are not limited to, the following.

Nettle weeds (Urticaceae): Hemerocallis (Urtica urens)
Scutellaris weed (Polygonaceae): Scutellaria vulgaris (Polygonum convolvulus), Sanaetade (Polygonum lapathifolium), American Scutellariae (Polygonum pensylvanicum), Harutade (Polygonum persicaria), Inutade (Polygonum longisetum), Psyllium (Polygonium) , Japanese gooseberry (Polygonum cuspidatum), sand snail (Rumex japonicus), longhorn snail (Rumex crispus), redwood snail (Rumex obtusifolius), sorrel (Rumex acetosa)
Prunusaceae weed (Portulacaceae): Prunella (Portulaca oleracea)
Horse mackerel weed (Caryophyllacea): chickweed (Stellaria media), calf commonwealth (Stellaria aquatica), minnow grass (Cerastium holosteoides), holly sand grass (Cerastium glomeratum), spiny grass (Spergula arvensis), mantemese
Pomegranate weed (Molluginaceae): Curcuma longiflorum (Mollugo verticillata)
Rhipicemum weeds (Chenopodiaceae): Scutellariae (Chenopodium album), Scutellariae (Chenopodium ambrosioides), Broomsticks (Kochia scoparia), Noharahijiki (Salsola kali), Atriplex spp.

Amaranthus weed (Amaranthaceae): Amaranthus (Amaranthus retroflexus), Amaryllis vulgaris (Amaranthus viridis), Cannilla (Amaranthus lividus), Hari-biru (Amaranthus spinosus), Horny Algaan Tow (Amaranthus hybridus), Amaranthus rudis, Amaranthus patulus, Amaranthus tuberculatos, Amaranthus blitoides, Amaranthus deflexus, Amaranthus quiititiveium, amelanthus ubiquitaci , Sanguinaria (Alternanthera tenella)
Poppyaceous weed (Papaveraceae): poplar (Papaver rhoeas), thistle (Argemone mexicana)
Brassicaceae weeds (Brassicaceae): Red nod (Raphanus raphanistrum), Noragarashi (Sinapis arvensis), Nazuna (Capsella bursa-pastoris), Amaranthus (Brassica juncea), Burrowing moth (Desculinia pinnata), Shrimp (Rorippa sylvestris), Gull Byasz (Thlaspi arvense), Porridge (Myagrum rugosum), Mamegun Byas (Lepidium virginicum), Orysia (Coronopus didymus)
Amaryllid weed (Capparaaceae): Cleome affinis

Leguminous weeds (Fabaceae): Kusanam (Aeschynomene indica), Zigzag jointed vetch (Aeschynomene rudis), American hornflower (Sesbania exaltata), Evisgusa (Cassia obtusifolia), Habasou (Cassia occidentalis), Jusuhagi (Desmodium timausium) adsendens), Illinois nuissimus (Desmodium illinoense), white clover (Trifolium repens), kudzu (Pueraria lobata), prickly pear (Vicia angustifolia), raccoon dog (Indigofera hirsuta), indigofera trulensis Vigna sinensis)
Anemoneid weed (Oxalidaceae): Anemonefish (Oxalis corniculata), Ottachi anemone (Oxalis strica), Oxalis oxidella (Oxalis oxyptera)
Freshwater weed (Geraniaceae): American Fuuro (Geranium carolinense), Dutch Fuuro (Erodium cicutarium)
Euphorbiaceae weed (Euphorbiaceae): Euphorbia helioscopia, Euphorbia maculata, Euphorbia humistrata, Euphorbia esula, Euphorbia hetraphylla, E. (Acalypha australis), Tropic croton (Croton glandulosus), Lobdo Croton (Croton lobatus), Brazil (Phyllanthus corcovadensis), Castor bean (Ricinus communis)

Malvaceous weeds (Malvaceae): Hevea (Abutilon theophrasti), Anemone deer (Sida rhombivoria), Maruba King deer (Sida cordifolia), American gore deer (Sida spinosa), fern Gurabiobi (Sida glaziovii), fern ), Ginseng (Hibiscus trionum), Amaryllis (Anoda cristata), Ekinoaki (Malvastrum coromandelianum)
Red-winged weeds (Onagraceae): Cleavage (Ludwigia epilobioides), red-winged lizard (Ludwigia octovalvis), soleid pokeweed (Ludwigia decurre)
Scutellaris Weed (Sterculiaceae): Prunus cypress (Waltheria indica)
Violet family weeds (Violaceae): persimmon (Viola arvensis), wild pansy (Viola tricolor)
Cucurbitaceae weed (Cucurbitaceae): Arecili (Sicyos angulatus), wild cucumber (Echinocystis lobata), wild bitter gourd (Momordica charantia)
Sprurgeon weeds (Lythraceae): Ammenia multiflora, Ammannia auriculata, Ammannia coccinea, Amitya (Lythrum salicaria), Orbita (Lythrum salicaria)
Shrimp Weed (Elatinaceae): Shrimp (Elatine triandra), California Waterwort (Elatine californica)

Seriaceae weeds (Apiaceae): Seri (Oenanthe javanica), Hemp ginseng (Conium maculatum)
Ucogillaceous weed (Araliaceae): Hydocotyle sibthorpioides, Brazil-dove Medusa (Hydrocotyle ranunculoides)
Amataceous weed (Ceratophyllaceae): A pine (Ceratophyllum demersum)
Hagoromomoaceae Weed (Cabombaceae): Hagoromomo (Cabomba caroliniana)
Allium spinosa weed (Haloragaceae): Blue-faced duck (Myriophyllum aquaticum), Fusamo (Myriophyllum verticillatum), water mill foils (Myriophyllum spicatum, Myriophyllum heterophyllum etc.)
Saturnia weed (Sapindaceae): Fusarium viper (Cardiospermum halicacabum)
Primrose weed (Primulaceae): Red-tailed riparian (Anagallis arvensis)
Sturgeon weed (Asclepiadaceae): Oorange cotton (Asclepias syriaca), honey wine milk weed (Ampelamus albidus)
Raccoon weeds (Rubiaceae): catch weed bed straws (Galium aparine), yam gras (Galium spurium var. Echinospermon), hirohafutabamugera (Spermacoce latifolia), brazil coriander (Richardia brasiliensis), winged falconite weed (Borrelia alata)

Convolvulus weed (Convolvulaceae): morning glory (Ipomoea nil), morning glory (Ipomoea hederacea), Marva morning glory (Ipomoea purpurea), Maruba american morning glory (Ipomoea hederacea var. , Noosaagaou (Ipomoea acuminata), Tsutano Haruko (Ipomoea hederifolia), Marubarukou (Ipomoea coccinea), Lepoucho (Ipomoea quamoclit), Ipomoea grandifolia (Ipomoea grandifolia), Ipomoea Aristolotiafolicotrithioliciol , Convolvulus arvensis, Calystegia hederacea, Convolvulus (Calystegia japonica), Eurasian Convolvulus (Merremia hedeacea), Hairy Wood Rose (Merremia aegyptia), Roadside Wood Rose (Merremi) a cissoides), asagao (Jacquemontia tamnifolia)
Purple family weed (Boraginaceae): Forget-me-not (Myosotis arvensis)
Lamiaceae weed (Lamiaceae): Lamium purpureum, Lamium amplexicaule, Leonotis nepetaefolia, Hyptis suaveolens, Hyptis lophanta (Hyptis lophatihichus)

Solanaceous weeds (Solanaceae): Datura stramonium, Solanum nigrum, Solanum americanum, American solanum pylanthum, Sornum sarachioides, Solanum thaliana , Squirrel eggplant (Solanum aculeatissimum), wild tomato (Solanum sisymbriifolium), warunaby (Solanum carolinense), physalis (Physalis angulata), smooth ground cherries (Physalis subglabrata), iosennari (Nicandra physaloides)
Scutellaria weed (Scrophulariaceae): Veronica hederaefolia, Veronica persica, Veronica arvensis, Azena (Lindernia ducuma), Azena (Lindernia dubia), Azetulifolius, as a extract (Dopatrium junceum), moth (Gratiola japonica),
Plantain weeds (Plantaginaceae): Planago asiatica, Planago lanceolata, Planago major, Planago major, Callitrice palustris

  Asteraceae weeds (Asteraceae): Monarch (Xanthium pensylvanicum), Monarch (Xanthium occidentale), Monarch (Xanthium italicum), Wild sunflower (Helianthus annuus), Chamomile (Matricaria chamomilla), Orysia camphor (Matricaria perforitum) ), Orso-Shak (Matricaria matricarioides), Mugwort (Artemisia princeps), Sesmus Artemisia vulgaris, Chinese Mugwort (Artemisia verlotorum), Scutellaria altissima (Solidago altissima), Daniocarpus (Taraxacum officigate), (Galinsoga parviflora), Novocython (Senecio vulgaris), Senecio braziliensis (Senecio brasiliensis), Senecio grisebachi (Senecio grisebachii), Arecynog (Conyza bonariensis), Himemushi Yomogi onyza canadensis), ragweed (Ambrosia artemisiaefolia), ambrosia tribe (Ambrosia trifida), taukogi (Bidens tripartita), kosendangusa (Bidens pilosa), American sentanosa (Bidens frondosa), bidense subalternate , American thistle (Cirsium vulgare), Maria thistle (Silybum marianum), musk thistle (Carduus nutans), Togechisha (Lactuca serriola), Nogeshi (Sonchus oleraceus), Onyokeshi (Sonchus asper), beach creeping ox eye (Wedelia glauca) Eto blackfoot (Melampodium perfoliatum), russius (Emilia sonchifolia), Shiozakiso (Tagetes minuta), Paracles (Blainvillea latifolia), Kotobikiiku (Tridax procumbens), Jerva porosa (Porophylllum rudeale), Paraguay Star bars (Acanthospermum australe), Bristley star bars (Acanthospermum hispidum), Fusuzaka (cardiospermum halicacabum), cuckoo thistle (Ageratum conyzoides), common bones set (Eupatorium perfoliatum), American Takasaburo (Eclipta altitratium) American Everlasting (Gamochaeta spicata), Gnaphalium spicatum, Jagelia japonica (Jaegeria hirta), Sesame (Parthenium hysterophorus), Mena Fami (Siegesbeckia orientalis), Meriken Tonso (Soliva sesive) Takasaburo (Eclipta alba), Persimmon (Centipeda minima),

Amaryllidaceae Weed (Alismataceae): Squid River (Sagittaria pygmaea), Omodaka (Sagittaria trifolia), P. edulis (Sagittaria sagittifolia), Tyrin Omodaka (Sagitaria montevidensis), Aeginashi (Sagittaria alitraceiium) aquatica)
Livulinaceae (Limnocharitaceae): Livularia (Limnocharis flava)
Tochikagami weed (Hydrocharitaceae): Frog bit (Limnobium spongia), Chromo (Hydrilla verticillata), common water nymph (Najas guadalupensis)
Araceae Weed (Araceae): Bianchi duckweed (Pistia stratiotes)
Duckweed weeds (Lemnaceae): Duckweed (Lemna aoukikusa), Duckweed (Spirodela polyrhiza), Geniaceae (Wolffia spp)
Phyllaceae weeds (Potamogetonaceae): Psyllium (Potamogeton distinctus), pond weeds (Potamogeton crispus, Potamogeton illinoensis, Stuckenia pectinata etc.)
Lilium weed (Liliaceae): Wild onion (Allium canadense), Wild garlic (Allium vineale), Nobil (Allium macrostemon)
Water weed: Water hyacinth (Eichhornia crassipes), Hemp helex (Heteranthera limosa), water hyacinth (Monochoria korsakowii), Allium (Monochoria vaginalis)
Achillea (Commelinaceae): Tussock (Commelina communis), Marubatu (Commela bengharensis), Electo dei Flower (Commelina erecta), Iboxa (Murdannia keisak)

  Grass weeds (Poaceae): Echinochloa crus-galli, Echinochloa oryzicola, Echinochloa crus-galli var formosensis, Late water glass (Echinochloa oryzoides), Echinochloa colona (Echinochloa colony) Echinochloa crus-pavonis), Enokologosa (Setaria viridis), Achinoenokologosa (Setaria faberi), Echinochloach (Setaria glauca), American Enokologa (Setaria geniculata), Redfinches (Digitaria ciliaris), Large Club Grass (Digitaria sanguignalis) Digitaria horizonis), Squidweed (Digitaria insularis), Echinode (Eleusine indica), Eurasian (Poa annua), Eurasian Mosquito (Poa trivialis), Eurasian Mosquito (Alospecurus aequalis), Blackgrass (Alopecurus myros) Barley (Avena fatua), Sorghum halepense, Shatha Cane (Sorghum vulgare), Agropyron repens, Barley (Lolium multiflorum), Boumy (Lolium rigidum), Barley (Bromus catharticus), Wild boar baboon (Bromus japonicus), common broom (Bromus secalinus), brown baboon (Bromus tectorum), hosonomemugi (Hordeum jubatum), goat's boar (Aegilops cylindrica), gospel bollworm (Phalaris arundinacea) spica-venti), oxabibi (Panicum dichotomiflorum), Texas panicum (Panicum texanum), Gineakibi (Panicum maximum), Meriken Nikkibi (Brachiaria platyphylla), Rujigrass (Brachiaria ruziziensis), Alexandergrass (Brachiaria plantaginea), Namgrass (Brachiaria decumbens), Parisade grass (Brachiaria brizantha), Colonybiia grass (Brachiaria humidicola), Shinrinioiga (Cenchrus echinatus), Himekuri noiga (Cenchrus pauciflorus), Narcobie (Eriochloa villosa), penicetium (Pellitimategium) ), Eragrostis pilosa, ruby gaya (Rhynchelitrum repens), Tatsunotsumegaya (Dactyloctenium aegyptium), Timothy grass (Ischaemum rugosum), Timotha (Isachne globosa), wild rice (Oryzas sativium), Parm (Paspalum maritimum), Prickly Pear Tree (Paspalum distichum), Chrysanthemum Grass (Pennisetum clandestinum), Sand Pricket (Pennisetum setosum), Hornbill (Rottboellia cochinchinensis), Azegaya (Leptochlolium (a a chinensis), Onia Zegaya (Leptochloa fascicularis), Itazegaya (Leptochloa filiformis), Amazon sprangle top (Leptochloa panicoides), Amazon sprangle top (Leptochloa panicoides), Amazonia sp (Glyceria acutiflora), Great Eel (Glyceria maxima)

Cactus weed (Cyperus microiria), Chypericus ciliatum (Cyperus microiria), Cyperus icri (Cyperus icri), Cyperus icri (Cyperus icri), Chyperus icri (Cyperus diffus.) (Cyperus odoratus), Cyperus cerotis, Chyperus rotundus, Cyperus esculentus, Kyllinga brevillima, Hidreich (Fimbristilitativeici), acicularis), Eleocharis kuroguwai, Schoenoplectus hotarui, Schoenoplectus juncoides, Schoenoplectus wallichii, Schoenoplectus mucronatus, Scutellariae (Schoenoplectus mucronatus) plectus triangulatus, Schoenoplectus nipponicus, Schoenoplectus triqueter, Squid (Bolboschoenus koshevnikovii), Squid (Bolboschoenus fluviatilis)
Horse mackerel weed (Equisetaceae): Japanese horsetail (Equisetum arvense), Inugina (Equisetum palustre)
Salamander weed (Salviniaceae): Salamander (Salvinia natans)
Amaryllidaceae weeds (Azollaaceae): Scutellaria japonicus (Azolla japonica), Scutellariae (Azolla imbricata)
Dendrobaceae (Marsileaceae): Dendless (Marsilea quadrifolia)
Others: filamentous algae (Pithophora, Cladophora), mosses, mosses, mosses, cyanobacteria, fern such as fern.

  The seeds used in the present invention are seeds of plants to which an effective amount of the present composition has been attached. The bulbs used in the present invention are bulbs of plants to which an effective amount of the composition of the present invention is attached. Also, for example, the composition of the present invention may be made into microcapsules and attached to seeds or bulbs. Also, in the attachment of the composition of the invention to the seeds or bulbs of a plant, the composition of the invention may completely or partially coat the seeds or bulbs, may be scattered on its surface, and / or Or it may exist in the inside.

  Hereinafter, the present invention will be described in more detail with formulation examples and test examples, but the present invention is not limited to the following examples. In the following examples, parts represent parts by weight unless otherwise specified.

  First, composition examples are shown.

  Specific compositions of the composition of the present invention are described in [Tables 1 to 31]. The composition of the present invention having the components described in [Tables 1-31] is described as “the composition of the present invention C1”, with the numbers described in [Tables 1-31]. In [Tables 1 to 31], * in the column of Component 1 represents any one kind of the compounds AA1-BA1 to AK2688-BK1287, and the numbers described in [] of the column of each component are each component Means parts by weight of

  Next, formulation examples are shown.

Formulation example 1
In the present invention, 50 parts of any one of the compositions A1 to A1626, B1 to B2096 or C1 to C604, 3 parts of calcium lignin sulfonate, 2 parts of magnesium lauryl sulfate and 45 parts of synthetic hydrous silicon oxide are thoroughly mixed and mixed. , Get the formulation.

Formulation example 2
In the invention, 20 parts of any one of the compositions A1 to A1626, B1 to B2096 or C1 to C604 and 1.5 parts of sorbitan trioleate are mixed with 28.5 parts of an aqueous solution containing 2 parts of polyvinyl alcohol After pulverizing by a grinding method, 40 parts of an aqueous solution containing 0.05 part of xanthan gum and 0.1 part of aluminum magnesium silicate is added to this, and 10 parts of propylene glycol is further added and mixed by stirring to obtain a preparation.

Formulation example 3
The preparation is obtained by thoroughly grinding and mixing 2 parts of any one of the compositions A1 to A1626, B1 to B2096 or C1 to C604, 88 parts of kaolin clay and 10 parts of talc according to the present invention.

Formulation example 4
By mixing 5 parts of any one composition according to the present invention A1 to A1626, B1 to B2096 or C1 to C604, 14 parts of polyoxyethylene styryl phenyl ether, 6 parts of calcium dodecylbenzene sulfonate and 75 parts of xylene , Get the formulation.

Formulation example 5
The present invention compositions A1 to A1626, B1 to B2096 or C1 to C604 2 parts, synthetic hydrolyzed silicon oxide 1 part, calcium lignin sulfonate 2 parts, bentonite 30 parts and kaolin clay 65 parts are well ground and mixed Then, water is added, the mixture is thoroughly mixed, granulated and dried to obtain a preparation.

Formulation Example 6
The composition of the present invention A1 to A1626, B1 to B2096 or C1 to C604 10 parts; 35 parts of white carbon containing 50 parts of polyoxyethylene alkyl ether sulfate ammonium salt; and 55 parts of water are mixed and pulverized. The formulation is obtained by processing using a machine.

  Next, test examples show that the composition of the present invention is useful for controlling pests.

Test Example 1 Control test against wheat leaf blight (Septoria tritici) A plastic pot is filled with soil, and wheat (variety; apodie) is sown and grown in a greenhouse for 10 days. A water dilution containing a surfactant or the like adjusted to contain any one of the compositions A1 to A1626, B1 to B2096 or C1 to C604 according to the present invention at a predetermined concentration (500 ppm) Spray the leaves and leaves to adhere well. After spraying, the plants are air-dried and 4 days later spray inoculated with an aqueous suspension of wheat spore (Septoria tritici) spores. After inoculation, the plants are placed under a humid atmosphere at 18 ° C. for 3 days, and then under illumination for 14 to 18 days, and then the lesion area is examined (this will be referred to as a treatment section).
On the other hand, wheat is grown in the same manner as in the treated area except that the diluted solution of the composition of the present invention is not sprayed with foliage (this is referred to as an untreated area). Investigate wheat leaf blight disease area as well as treated area.
From the lesion area of each of the treated area and the untreated area, the efficacy of the treated area is determined according to the following [Equation 1].
As a result, a high pest control effect is recognized.

Test Example 2 Control Test for Cucumber Powdery Mildew (Sphaerotheca fuliginea) The soil is packed in a plastic pot, and a cucumber (variety; Sagami Hankaku) is sown and grown in a greenhouse for 12 days. An aqueous dilution containing a surfactant or the like adjusted to contain any one of the compositions A1 to A1626, B1 to B2096 or C1 to C604 at a predetermined concentration (500 ppm) is sufficiently adhered to the cucumber leaf surface Spray the leaves and leaves as you like. After spraying, the plants were air-dried, and a QoI resistant strain in which the nucleotide sequence was mutated such that the amino acid residue at amino acid residue 143 of cytochrome b in the gene coding for cucumber powdery mildew (Sphaerotheca fuliginea, cytochrome b) ) Sprinkle spores and inoculate. After growing plants in a greenhouse at 24 ° C. in the daytime and at 20 ° C. in the night for 8 days, the lesion area is examined (this will be referred to as a treatment zone).
On the other hand, a cucumber is grown in the same manner as in the treated area except that the diluted solution of the composition of the present invention is not sprayed with foliage (this is referred to as an untreated area). Investigate the area of the disease spots of cucumber powdery mildew as well as the treated area.
From the lesion area of each of the treated area and the untreated area, the efficacy of the treated area is determined by [Equation 1].
As a result, a high pest control effect is recognized.

Test Example 3 Control test against tomato leaf mold (Cladosporium fulvum) A plastic pot is filled with soil, and a tomato (variety; patio) is sown and grown in a greenhouse for 3 weeks. The diluted aqueous solution containing a surfactant etc. adjusted to contain any one of the compositions A1 to A1626, B1 to B2096 or C1 to C604 according to the present invention to a predetermined concentration (500 ppm) is sufficient for the above-mentioned tomato leaf surface Spray foliage to adhere. After spraying, the plants were air-dried, and a QoI-resistant strain in which the nucleotide sequence was mutated such that the amino acid residue at position 129 of cytochrome b in the gene encoding tomato leaf mold fungus (Cladosporium fulvum, cytochrome b) was substituted from phenylalanine to leucine. 2.) Spray inoculate a water suspension of spores. After inoculation, the plants are placed in a greenhouse at 24 ° C. in the daytime at 20 ° C. in a humid atmosphere for 3 days, and then grown for 14 days in a greenhouse, and then the lesion area is examined. (This will be the treatment area.)
On the other hand, tomatoes are grown in the same manner as in the treated area except that the diluted solution of the composition of the present invention is not sprayed on foliage (this is referred to as an untreated area). Investigate the disease area of tomato leaf mold as well as the treated area.
From the lesion area of each of the treated area and the untreated area, the efficacy of the treated area is determined by [Equation 1].
As a result, a high pest control effect is recognized.

  According to the present invention, pests can be controlled.

Claims (6)

  Group (I), Group (II), Group (III), Group (IV), Group (V), Group (VI), Group (VII), Group (VIII), Group (IX), Group (X), Group (XI), Group (XII), Group (XIII), Group (XIV), Group (XV), Group (XVI), Group (XVII), Group (XVIII), Group (XVIII), Group (XIX), Group (XX), A pest comprising the compound according to any one selected from the group consisting of Group (XXI), Group (XXII) and Group (XXIII), and one or more components selected from the group consisting of Group A to Group F Control composition.
Group A; fungicide
Group B; Insecticide, acaricide
Group C; Herbicide
Group D; Safeners
Group E; plant growth regulator
Group F; Microbial material

Group (I): Formula (1)
[In the formula,
R¹Is the group P¹And C6-C16 aryl group optionally having one or more substituents selected from¹C7-C18 aralkyl group optionally having one or more substituents selected from¹C1-C12 alkyl group optionally having one or more substituents selected from¹C2-C12 alkenyl group optionally having one or more substituents selected from¹And C 2 -C 12 alkynyl group optionally having one or more substituents selected from¹C3-C12 cycloalkyl group optionally having one or more substituents selected from¹C2-C12 acyl group optionally having one or more substituents selected from¹Represents an adamantyl group optionally having one or more substituents, a C3-C12 trialkylsilyl group, a hydrogen atom, or a halogen atom (however, the C6-C16 aryl group, the C7-C18). The C1-C12 alkyl group, the C2-C12 alkenyl group, the C2-C12 alkynyl group, the C3-C12 cycloalkyl group, the C2-C12 acyl group, and the adamantyl group When they have two or more substituents, the substituents may be the same or different),
X¹Represents a sulfur atom or an oxygen atom,
R²Is a hydrogen atom, a C1-C12 alkyl group, a C1-C12 haloalkyl group, a C2-C12 alkenyl group, a C2-C12 haloalkenyl group, a C2-C12 alkynyl group, a C2-C12 haloalkynyl group, C2 -C12 represents an alkoxycarbonyl group, a hydroxycarbonyl group or a halogen atom,
R⁴And R⁵Each independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group, or
Or R⁴And R⁵And may form a C3-C6 cycloalkane ring together with the carbon atom to which they are attached,
R⁶, R⁷, R⁸, And R⁹And C1 to C12 alkyl group, halogen atom, C1 to C12 haloalkyl group, C3 to C12 cycloalkyl group, C3 to C12 halocycloalkyl group, C1 to C12 alkoxy group, C1 to C12 independently of each other. C.sub.1-C.sub.12 alkylthio group C.sub.1-C.sub.12 haloalkylthio group, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, C.sub.2-C.sub.12 alkenyl group, C.sub.2-C.sub.12 haloalkenyl Group, C2-C12 alkynyl group, C2-C12 haloalkynyl group, C3-C12 cycloalkyloxy group, C3-C12 halocycloalkyloxy group, C3-C12 cycloalkylthio group, C2-C12 alkenyloxy Group, C2-C12 alkynyloxy group, C2-C12 haloalkenyl Xy group, C2-C12 haloalkynyloxy group, C2-C12 alkynylthio group, C2-C12 alkenylthio group, C2-C12 haloalkenylthio group, C2-C12 haloalkynylthio group, C2-C12 Acyl group, C2-C12 haloacyl group, C2-C12 acyloxy group, C2-C12 acylthio group, C2-C12 alkoxycarbonyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group C1-C12 alkylsulfonyl group, C1-C12 haloalkylsulfonyl group, C1-C12 alkylsulfinyl group, C1-C12 haloalkylsulfinyl group, aminosulfonyl group optionally substituted with C1-C12 alkyl group, An amino group which may be substituted by a C1-C12 alkyl group, 1-C12 alkyl group optionally substituted aminocarbonyl group, a hydrogen atom, or represents a hydroxy group or a formyl group,
Or adjacent R⁶And R⁷, R⁷And R⁸, And R⁸And R⁹And may form a C4-C6 cycloalkene ring, a C5-C6 cycloalkyldiene ring, or a benzene ring together with the carbon atom to which they are attached,
R¹⁰Is a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkoxyalkyl group, a C3-C6 cycloalkyl group or a C3-C6 Represents a halocycloalkyl group of
Y¹Represents an oxygen atom or a sulfur atom,
Q¹Is an oxygen atom, a sulfur atom, or NR¹¹Represents a group,
R¹¹Represents a hydrogen atom, a C1-C6 alkyl group, or a C1-C6 haloalkyl group.
Group P¹: A halogen atom, C1-C12 alkyl group, C1-C12 haloalkyl group, C1-C12 alkoxy group, C1-C12 haloalkoxy group, C1-C12 alkylthio group, C1-C12 haloalkylthio group, hydroxycarbonyl Group, formyl group, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, C2-C12 alkenyl group, C2-C12 haloalkenyl group, C2-C12 alkynyl group, C2-C12 haloalkynyl Group, C3-C12 cycloalkyl group, C3-C12 halocycloalkyl group, C3-C12 cycloalkyloxy group, C3-C12 halocycloalkyloxy group, C3-C12 cycloalkylthio group, C2-C12 Alkenyloxy group, C2-C12 alkynyloxy group, C2-C 2 haloalkenyloxy group, C2-C12 haloalkynyloxy group, C2-C12 alkynylthio group, C2-C12 alkenylthio group, C2-C12 haloalkenylthio group, C2-C12 haloalkynylthio group, C2-C12 acyl group, C2-C12 haloacyl group, C2-C12 acyloxy group, C2-C12 acylthio group, C2-C12 alkoxycarbonyl group, C6-C16 aryl group, C6-C16 haloaryl group, C6-C16 aryloxy group, C6-C16 haloaryloxy group, C6-C16 arylthio group, C6-C16 haloarylthio group, C7-C18 aralkyl group, C7-C18 haloaralkyl group, C7- C18 arylalkoxy group, C7-C18 haloarylalkoxy group, C3-C12 tri Alkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C12 alkylsulfonyl group, C1-C12 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloarylsulfonyl group, C1-C12 Alkylsulfinyl group, C1-C12 haloalkylsulfinyl group, C6-C16 arylsulfinyl group, C6-C16 haloarylsulfinyl group, C2-C11 polyoxaalkyloxy group, C2-C5 oxacycloalkyloxy group, C1 An aminocarbonyl group which may be substituted with a -C12 alkyl group and / or a C6-C12 aryl group, an aminosulfonyl group which may be substituted with a C1-C12 alkyl group and / or a C6-C12 aryl group And C1-C12 The group consisting of even an amino group substituted with kill group. ]
A tetrazolinone compound represented by the formula:

Group (II): Formula (2)
[In the formula,
R²⁴And R²⁵Each represents a hydrogen atom or a C1-C3 alkyl group;
R²⁶Is a C1-C4 alkyl group, a C3-C6 cycloalkyl group, a C1-C4 haloalkyl group, a C3-C6 halocycloalkyl group, a halogen atom, a cyano group, a nitro group, a C2-C4 alkenyl group, a C2-C4 haloalkenyl group , A C 2 -C 4 alkynyl group, a C 2 -C 4 haloalkynyl group, a C 1 -C 4 alkoxy group, a C 1 -C 4 haloalkoxy group, a C 1 -C 4 alkylthio group or a C 1 -C 4 haloalkylthio group;
R²⁷, R²⁸And R²⁹Each represents a hydrogen atom or a halogen atom;
R³⁰Is a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C2-C3 alkynyl group, a C2-C3 haloalkynyl group, a C3-C5 cycloalkyl group or a C3-C5 Represents a halocycloalkyl group;
X²Represents an oxygen atom or a sulfur atom;
R³³Is a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a hydrogen atom, a C1 to C6 haloalkyl group, a C3 to C6 halocycloalkyl group, a C2 to C6 alkenyl group, a C2 to C6 haloalkenyl group, a C2 to C6 alkynyl group , A C 2 -C 6 haloalkynyl group, a C 1 -C 6 alkoxy group or a C 1 -C 6 alkylthio group;
Q²Is a phenyl group, a phenoxy group, a phenylthio group, a phenylamino group (however, the phenyl portion of the phenyl group, the phenoxy group, the phenylthio group and the phenylamino group together with the adjacent carbon atom is a four-membered ring, a five-membered ring, The ring may form one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom as a ring constituent atom, and the same carbon may be formed. The atom may have an oxo group, a thioxo group or a C1-C3 alkoxyimino group, may have one or two oxide groups on the same sulfur atom, and the phenyl moiety and the ring may be , Group P²¹And one or more atoms or groups selected from²¹When the atom or group selected from is 2 or more, the atom or group may be the same or different. ),
5- or 6-membered heterocyclyl group, 5- or 6-membered heterocyclyloxy group, 5- or 6-membered heterocyclylthio group, 5- or 6-membered heterocyclylamino group (provided that the 5- or 6-membered heterocyclyl group, 5- or 6-membered heterocyclyloxy group, 5 And the 5- or 6-membered heterocyclyl moiety of the 5- or 6-membered heterocyclylamino group and the 5- or 6-membered heterocyclylamino group together with the adjacent carbon atom form a 4-, 5-, 6- or 7-membered ring The ring may contain one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom as a ring member atom, and the 5- or 6-membered heterocyclyl moiety and the ring Are oxo, thioxo or C1-C3 alkoxyimino on the same carbon atom May also be, may have one or two oxide groups to the same sulfur atom, the group P²¹And one or more atoms or groups selected from²¹When the atom or group selected from is 2 or more, the atom or group may be the same or different. ),
A C3-C6 cycloalkyl group, a C3-C6 cycloalkenyl group, provided that the C3-C6 cycloalkyl group and the C3-C6 cycloalkenyl group, together with the adjacent carbon atom, are a 4-, 5-, or 6-membered ring Or a 7-membered ring may be formed, and the ring may contain one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom as a ring constituting atom, and the same sulfur atom may be used. The ring, the C3-C6 cycloalkyl group and the C3-C6 cycloalkenyl group may have an oxo group, a thioxo group or a C1-C3 alkoxyimino on the same carbon atom. Group may have a group P²¹And one or more atoms or groups selected from²¹When the atom or group selected from is 2 or more, the atom or group may be the same or different. ),
C 1 -C 4 alkyl group (provided that the C 1 -C 4 alkyl group may have an oxo group, a thioxo group or a C 1 -C 3 alkoxyimino group on the same carbon atom)²¹And one or more atoms or groups selected from²¹When the atom or group selected from is 2 or more, the atom or group may be the same or different. ),
C2-C4 alkenyl group or C2-C4 alkynyl group (provided that the C2-C4 alkenyl group and the C2-C4 alkynyl group are groups P)²¹And one or more atoms or groups selected from²¹When the atom or group selected from is 2 or more, the atom or group may be the same or different. Represents);
Or Q²Substituents and R³³And, together with the carbon atom or nitrogen atom to which they are attached, may form a 5-, 6- or 7-membered ring, and the ring is a group consisting of an oxygen atom, a sulfur atom and a nitrogen atom And one or more atoms selected from the group consisting of²⁴And one or more atoms or groups selected from²⁴When the atom or group selected from is 2 or more, the atom or group may be the same or different.
Group P²¹: Group P²³A C1-C6 alkyl group optionally having one or more atoms or groups selected from²³A C3-C6 cycloalkyl group which may have an atom or a group selected from
A phenyl group (however, the phenyl group may form a 4-, 5-, 6-, or 7-membered ring together with the adjacent carbon atom, and the ring includes an oxygen atom, a sulfur atom and a nitrogen atom; The ring may contain one or more atoms selected from the group consisting of atoms, and may have an oxo group, a thioxo group or a C1-C3 alkoxyimino group on the same carbon atom, and the same sulfur The phenyl group and the ring may have one or two oxide groups at one atom,²²And one or more atoms or groups selected from²²When the atom or group selected from is 2 or more, the atom or group may be the same or different. ),
5- or 6-membered heterocyclyl group (provided that the 5- or 6-membered heterocyclyl group may form a 4-, 5-, 6-, or 7-membered ring together with the adjacent carbon atom, and the ring is And one or more atoms selected from the group consisting of an oxygen atom, a sulfur atom and a nitrogen atom may be contained as a ring-constituting atom, and the 5- or 6-membered heterocyclyl group and the ring may have the same carbon atom And may have an oxo group, a thioxo group, or a C1-C3 alkoxyimino group, and may have one or two oxide groups on the same sulfur atom;²²And one or more atoms or groups selected from²²When the atom or group selected from is 2 or more, the atom or group may be the same or different. ),
C1-C6 haloalkoxy group, halogen atom, nitro group, C1-C6 alkoxy group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 alkenyloxy Group, C3-C6 haloalkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkynyloxy group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group Group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, cyano group, amino group, hydroxy group, mercapto group, pentafluorosulfanyl group, C3-C9 Trialkylsilyl group, C2-C6 alkyl Carbonyl group, C2-C6 alkoxycarbonyl group, C2-C8 alkylaminocarbonyl group and C2-C8 group consisting alkylcarbonylamino group.
Group P²²: Group P²³A C1-C6 alkyl group optionally having one or more atoms or groups selected from²³A C3-C6 cycloalkyl group which may have an atom or a group selected from
C1-C6 alkoxy group, C1-C6 haloalkoxy group, halogen atom, nitro group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 alkenyloxy Group, C3-C6 haloalkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkynyloxy group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group Group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, cyano group, amino group, hydroxy group, mercapto group, pentafluorosulfanyl group, C3-C9 Trialkylsilyl group, C2-C6 alkyl Carbonyl group, C2-C6 alkoxycarbonyl group, C2-C8 alkylaminocarbonyl group and C2-C8 group consisting alkylcarbonylamino group.
Group P²³A group consisting of a halogen atom, a C3 to C6 cycloalkyl group, a C3 to C6 halocycloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group and a C1 to C4 haloalkylthio group.
Group P²⁴: A halogen atom, a cyano group, a nitro group, a C1 to C4 alkyl group, a C3 to C6 cycloalkyl group, a C1 to C4 haloalkyl group, a C3 to C6 halocycloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, A group consisting of a C1-C4 alkylthio group and a C1-C4 haloalkylthio group. ]
A tetrazolinone compound represented by the formula:

Group (III): Formula (3)
[In the formula,
R⁴¹, R⁴², R⁴³And R⁵¹Each represents a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1-C6 alkylsulfinyl group, C1-C6 Haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, C2-C9 alkylamino Carbonyl group,
Group P³¹And a C1-C6 alkyl group optionally having a group selected from
Or group P³¹Represents a C3-C6 cycloalkyl group which may have a group selected from
R⁴⁴And R⁴⁵Each represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R⁴⁶Is a C1-C4 alkyl group which may have a halogen atom, a hydrogen atom, a halogen atom, a C1-C4 alkoxy group which may have a halogen atom, a C2-C4 alkenyl group, a C2-C4 haloalkenyl group , C2-C4 alkynyl group, C2-C4 haloalkynyl group, C1-C4 alkylthio group, C1-C4 haloalkylthio group, C3-C6 cycloalkyl group or C3-C6 halocycloalkyl group, cyano group, nitro group, C1- C4 alkylsulfinyl group, C1-C4 alkylsulfonyl group, C1-C4 haloalkylsulfinyl group, C1-C4 haloalkylsulfonyl group, C1-C6 alkylamino group or C1-C6 haloalkylamino group;
R⁴⁷, R⁴⁸And R⁴⁹Each represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C1-C3 alkoxy group, or a C1-C3 haloalkoxy group;
R⁵⁰Is a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C2-C3 alkynyl group, a C2-C3 haloalkynyl group, a C3-C5 cycloalkyl group, or a C3-C5 alkyl group. Represents a C5 halocycloalkyl group;
X³Represents an oxygen atom or a sulfur atom;
R⁵²Is
Group P³¹And a C1-C6 alkyl group optionally having a group selected from
Group P³¹And a C3-C6 cycloalkyl group optionally having a group selected from
Group P³²A phenyl group which may have a group selected from
Hydrogen atom, halogen atom, cyano group, nitro group, amino group, C2 to C6 alkenyl group, C2 to C6 haloalkenyl group, C1 to C6 haloalkyl group, C2 to C6 alkynyl group, C2 to C6 haloalkynyl group, C1 to C6 Alkoxy group, C1-C6 haloalkoxy group, C3-C6 cycloalkenyl group, C3-C6 halocycloalkenyl group, C1-C8 alkylamino group, C3-C12 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 Represents an alkoxycarbonyl group, or a C2-C9 alkylaminocarbonyl group;
R⁵³Are C1-C8 alkyl group, C1-C8 haloalkyl group, C2-C8 alkenyl group, C2-C8 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 cycloalkyl group, C3-C6 Halocycloalkyl group, C 3 -C 6 cycloalkenyl group, C 3 -C 6 halocycloalkenyl group,
Or group P³²And a benzyl group which may have a group selected from
Group P³¹: A group consisting of a halogen atom, a cyano group, a C3 to C6 cycloalkyl group, a C3 to C6 halocycloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group and a C1 to C4 haloalkylthio group .
Group P³²: Halogen atom, cyano group, amino group, hydroxy group, thiol group, C1-C6 alkyl group, C1-C6 haloalkyl group, C3-C6 cycloalkyl group, C3-C6 halocycloalkyl group, C2-C6 alkenyl group, C2 -C6 haloalkenyl group, C2-C6 alkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C8 alkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1-C6 alkylsulfinyl A group consisting of C1-C6 alkylsulfonyl group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, and C2-C9 alkylaminocarbonyl group. ]
A tetrazolinone compound represented by the formula:

Group (IV): Formula (4)
[In the formula,
R⁶¹And R⁶²Each independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R⁶³Is a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, a nitro group , Cyano group,
An aminocarbonyl group which may have a C1-C6 alkyl group,
C2-C6 haloalkenyl group, C2-C6 haloalkynyl group, C3-C6 halocycloalkyl group, C1-C6 haloalkoxy group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl group Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, C2-C6 alkoxycarbonyl group, hydroxyl group, thio Group, an amino group which may have a C1-C6 alkyl group, a pentafluorosulfanyl group, a C3-C9 trialkylsilyl group, a C5-C14 trialkylsilylethynyl group, a C1-C4 alkylsulfonyl group, a C1-C4 group. Represents a haloalkylsulfonyl group, a C1-C4 alkylsulfinyl group, a C1-C4 haloalkylsulfinyl group, a C2-C5 alkoxyalkyl group or a C2-C5 alkylthioalkyl group;
R⁶⁴, R⁶⁵And R⁶⁶Each independently represents a hydrogen atom, a halogen atom, a C1 to C4 alkyl group, a C1 to C4 haloalkyl group, a C3 to C5 cycloalkyl group, a C3 to C5 halocycloalkyl group, a C1 to C4 alkoxy group, or a C1 to C4 haloalkoxy Represents a group;
R⁶⁷Is a C1 to C6 alkyl group, a hydrogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C2 to C6 haloalkenyl group, a C2 to C6 alkoxyalkyl group, a C3 to C6 cycloalkyl group or a C3 to C6 halocycloalkyl Represents a group;
A⁴Is a halogen atom, group P⁴⁰C6-C16 aryl group optionally having one or more atoms or groups selected from⁴⁰Or a C3-C12 cycloalkyl group optionally having one or more atoms or groups selected from⁴⁰Or a C2-C9 heterocyclyl group optionally having one or more atoms or groups selected from (wherein the C2-C9 heterocyclyl group is selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom as a ring constituting atom) When containing one or more atoms and containing two or more atoms selected from the group consisting of nitrogen atoms, oxygen atoms and sulfur atoms, each of the atoms is identical to or different from at least one other atom of Furthermore, the carbon atom or nitrogen atom constituting the ring of the C2-C9 heterocyclyl group is⁴Combined with ) Or group P⁴⁰And the C3-C12 cycloalkenyl group optionally having one or more atoms or groups selected from (wherein the C6-C16 aryl group, the C3-C12 cycloalkyl group, the C2-C9 heterocyclyl group and the C3-C12 cycloalkenyl group is a group P⁴⁰When it has two or more atoms or groups selected from group P, each of the atoms or groups may be the same as at least one other atom or group. Or it may be different. );
Q⁴The following groups Q 41, Q 42, Q 43, Q 44, Q 46, Q 47, Q 48, Q 49, Q 50, Q 51 or Q 52 {# represents a binding site to A, and ● represents a binding site to an oxygen atom} Represents
R⁶⁸, R⁶⁹, R⁷⁰And R⁷¹Are each independently a hydrogen atom, a halogen atom, a group P⁴¹Or a C1-C6 alkyl group optionally having one or more atoms or groups selected from⁴¹Or C1-C6 cycloalkyl group optionally having one or more atoms or groups selected from C1-C6 alkoxy group, C1-C6 haloalkoxy group, cyano group, nitro group, amino group, hydroxy group, thiol group , C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group,
An amino group which may have a C1-C6 alkyl group,
An amino group which may have a C1-C6 haloalkyl group,
C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C9 tri An alkylsilyl group, a C2-C6 alkylcarbonyl group, a C2-C6 alkoxycarbonyl group or
Represents an aminocarbonyl group which may have a C1-C6 alkyl group;
X⁴Represents an oxygen atom or a sulfur atom.
Group P⁴⁰: Halogen atom, C1-C6 alkyl group, C1-C6 haloalkyl group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 cycloalkyl group, C3 -C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynylthio group , C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 Alkyl carbonyl group, C2 to C6 haloalkyl carbonyl group, C2 to C6 alkyl carbonyloxy group, C2 to C6 alkyl carbonyl thio group, hydroxycarbonyl group, formyl group, C2 to C6 alkoxycarbonyl group, nitro group, cyano group, hydroxyl group, C6-C16 aryl group, C6-C16 haloaryl group, C6-C16 aryloxy group, C6-C16 haloaryloxy group, C6-C16 arylthio group, C6-C16 haloarylthio group, C7-C18 aralkyl group, C7-C18 Haloaralkyl group, C7-C18 arylalkoxy group, C7-C18 haloarylalkoxy group, thiol group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C6 alkylsulfonyl group , C1-C6 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloaryl sulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C6-C16 arylsulfinyl group, C6-C16 haloarylsulfinyl group Group,
An amino group which may have a C1-C6 alkyl group,
An aminosulfonyl group optionally having a C1-C6 alkyl group and / or a C6-C12 aryl group
And a group consisting of an aminocarbonyl group which may have a C1-C6 alkyl group.
Group P⁴¹: A group consisting of a halogen atom, a cyano group, a C3 to C6 cycloalkyl group, a C3 to C6 halocycloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group and a C1 to C4 haloalkylthio group . ]
A tetrazolinone compound represented by the formula:

Group (V): Formula (5)
[In the formula,
Q⁵Represents the following groups Q53, Q54, Q55, Q56 or Q57;
R⁸¹, R⁸², R⁸³And R⁹¹Each represents a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1-C6 alkylsulfinyl group, C1-C6 Haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, C2-C8 alkylamino Carbonyl group, group P⁵¹Or a C1-C6 alkyl group optionally having a group selected from⁵¹Represents a C3-C6 cycloalkyl group which may have a group selected from
R⁸⁴And R⁸⁵Each represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R⁸⁶Is a C1-C4 alkyl group, a halogen atom, a C1-C4 alkoxy group, a cyano group, a nitro group, a C1-C4 haloalkyl group, a C2-C4 alkenyl group, a C2-C4 haloalkenyl group, a C3-C6 cycloalkyl group, a C2 -C4 alkynyl group, C2-C4 haloalkynyl group, C1-C4 haloalkoxy group, C1-C4 alkylthio group, C1-C4 alkylsulfinyl group, C1-C4 alkylsulfonyl group, C1-C4 haloalkylthio group, C1-C4 haloalkyl A sulfinyl group, a C1-C4 haloalkylsulfonyl group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C3-C6 halocycloalkyl group or a hydrogen atom;
R⁸⁷, R⁸⁸And R⁸⁹Each represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group or a C1-C3 alkoxy group;
R⁹⁰Is a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group, a C2-C3 alkynyl group, a C2-C3 haloalkynyl group, a C3-C5 cycloalkyl group or a C3-C5 group Represents a halocycloalkyl group;
X⁵Represents an oxygen atom or a sulfur atom;
A⁵¹And A⁵³Each represents a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C8 alkylamino group, C1-C8 dialkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C1-C6 Alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group Group, C2-C8 alkylamino carbonyl Group, group P⁵¹Or a C1-C6 alkyl group optionally having a group selected from⁵¹Represents a C3-C6 cycloalkyl group which may have a group selected from
A⁵², Z⁵¹And Z⁵⁴Each represents a hydrogen atom, an amino group, a C3-C6 alkenyl group, a C3-C6 haloalkenyl group, a C3-C6 alkynyl group, a C3-C6 haloalkynyl group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, C1 -C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C3-C6 cycloalkylsulfonyl group, C3-C6 halocycloalkylsulfonyl group, C2-C8 alkylaminosulfonyl group, C2-C8 haloalkylaminosulfonyl group, C3-C9 tri- Alkyl silyl group, C 2 -C 6 alkyl carbonyl group, C 2 -C 6 alkoxy carbonyl group, C 2 -C 8 alkyl amino carbonyl group, C 4-C 7 cycloalkyl methyl group, group P⁵¹Or a C1-C6 alkyl group optionally having a group selected from⁵¹Represents a C3-C6 cycloalkyl group which may have a group selected from
Z⁵⁵Represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C6 cycloalkyl group or a C1-C6 halocycloalkyl group;
Y⁵¹, Y⁵², Y⁵³, Z⁵²And Z⁵³Are each a hydrogen atom, a halogen atom, a cyano group, a nitro group, an amino group, a hydroxy group, a thiol group, an aldehyde group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 halo Alkynyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C3-C6 alkenyloxy group, C3-C6 haloalkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenyl Thio group, C3-C6 alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C1-C8 alkylamino group, C1-C8 haloalkylamino group, C1-C6 alkylthio group, C1-C6 halo Alkylthio group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C8 alkylaminosulfonyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, C2 -C8 alkylaminocarbonyl group, aminocarbonyl group, group P⁵¹Or a C1-C6 alkyl group optionally having a group selected from⁵¹Represents a C3-C6 cycloalkyl group which may have a group selected from
Or Y⁵¹And Y⁵²Together with the carbon atom to which they are attached, may form a 5-, 6-, or 7-membered saturated ring (provided that the saturated ring is an oxygen atom or a ring constituting atom thereof). May contain a sulfur atom, and the saturated ring is a group P⁵¹And may have a group selected from as a substituent);
Y⁵²And Y⁵³Together with the carbon atom to which they are attached, may form a 5-, 6-, or 7-membered saturated ring (provided that the saturated ring is an oxygen atom or a ring constituting atom thereof). May contain a sulfur atom, and the saturated ring is a group P⁵¹And may have a group selected from as a substituent);
Z⁵¹And Z⁵²And a carbon atom or nitrogen atom to which they are attached may form a 5-, 6-, or 7-membered saturated ring (provided that the saturated ring is a ring-constituting atom). The saturated ring may contain an oxygen atom, a nitrogen atom or a sulfur atom, and the saturated ring is a group P⁵¹And may have a group selected from as a substituent);
Z⁵²And Z⁵³And a carbon atom to which they are bound may form a 5-, 6-, or 7-membered saturated ring (provided that the saturated ring is an oxygen atom as a ring-constituting atom, The saturated ring may contain a nitrogen atom or a sulfur atom;⁵¹And may have a group selected from as a substituent).
Group P⁵¹: A group consisting of a halogen atom, a cyano group, a C3 to C6 cycloalkyl group, a C3 to C6 halocycloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group and a C1 to C4 haloalkylthio group . ]
A tetrazolinone compound represented by the formula:

Group (VI): Formula (6)
[In the formula, Q⁶Is the group P⁶¹And a 6-membered aromatic heterocyclic group which may have one or more atoms or groups selected from the following: provided that the hetero atom constituting the heterocyclic group is a nitrogen atom, and the number of nitrogen atoms is 1, 2 or 3);
R¹⁰¹, R¹⁰², R¹⁰³And R¹¹¹Are each independently, group P⁶²Or a C1-C6 alkyl group optionally having one or more atoms or groups selected from⁶²Or a C3-C6 cycloalkyl group optionally having one or more atoms or groups selected from H, a halogen atom, a hydrogen atom, a C1-C6 alkoxy group optionally having one or more halogen atoms, a cyano group, A nitro group, an amino group, a hydroxy group, a sulfanyl group, a C2 to C6 alkenyl group optionally having one or more halogen atoms, a C2 to C6 alkynyl group optionally having one or more halogen atoms, Amino group optionally having 2 C1-C8 alkyl groups (provided that it may have a halogen atom), C1-C6 alkylthio group optionally having one or more halogen atoms, one or more C1-C6 alkylsulfinyl group which may have one or more halogen atoms, C1-C6 alkylsulfonyl group which may have one or more halogen atoms, pentafluorosulfone Represents an aminocarbonyl group which may have one or more C2-C8 alkyl, C3-C9 trialkylsilyl group, C2-C6 alkylcarbonyl group, C2-C6 alkoxycarbonyl group, or one or more C2-C8 alkyl;
R¹⁰⁴And R¹⁰⁵Each independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R¹⁰⁶Is a C1-C6 alkyl group which may have one or more halogen atoms, a C3-C6 cycloalkyl group which may have one or more halogen atoms, a halogen atom, a hydrogen atom, one or more halogen atoms C2-C6 alkenyl group which may have, C1-C6 alkoxy group which may have one or more halogen atoms, C1-C6 alkylthio group which may have one or more halogen atoms, one or more C 2 -C 6 alkynyl group which may have one or more halogen atoms, a nitro group, a cyano group, an aminocarbonyl group which may have one or two C 1 -C 6 alkyl groups, one or more halogen atoms C3-C6 cycloalkoxy group which may be substituted, C3-C6 cycloalkylthio group which may contain one or more halogen atoms, C3-C6 which may contain one or more halogen atoms Alkenyloxy group, C3-C6 alkynyloxy group optionally having one or more halogen atoms, C3-C6 alkenylthio group optionally having one or more halogen atoms, one or more halogen atoms C3-C6 alkynylthio group, C2-C6 alkylcarbonyl group optionally having one or more halogen atoms, C2-C6 alkylcarbonyloxy group, C2-C6 alkylcarbonylthio group, C2-C6 alkoxy A carbonyl group, a hydroxy group, a sulfanyl group, an amino group which may have one or two C1-C6 alkyl groups, a pentafluorosulfanyl group, a C3-C9 trialkylsilyl group, a C5-C14 trialkylsilylethynyl group, C1-C4 alkylsulfonyl group optionally having one or more halogen atoms, one or more halogens Child C1-C4 alkyl sulfates may have a sulfinyl group, a C2-C5 alkoxyalkyl group, or C2-C5 alkylthioalkyl group;
R¹⁰⁷, R¹⁰⁸And R¹⁰⁹Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, a C2-C3 alkenyl group optionally having one or more halogen atoms, or one or more Represents a C1-C3 alkoxy group which may have a halogen atom of
R¹¹⁰Is a C1-C3 alkyl group optionally having one or more halogen atoms, a C2-C3 alkenyl group optionally having one or more halogen atoms, or one or more halogen atoms Represents a C2-C3 alkynyl group or a C3-C5 cycloalkyl group optionally having one or more halogen atoms;
X⁶Represents an oxygen atom or a sulfur atom.
Group P⁶¹C1 to C6 alkyl group optionally having one or more halogen atoms, halogen atom, C2 to C6 alkenyl group optionally having one or more halogen atoms, one or more halogen atoms C2-C6 alkynyl group, C3-C6 cycloalkyl group optionally having one or more halogen atoms, C1-C6 alkoxy group optionally having one or more halogen atoms, one or more halogen atoms C 1 -C 6 alkylthio group which may have one or more C 3 -C 6 cycloalkyloxy group which may have one or more halogen atoms, C 3-C 6 cycloalkylthio group which may have one or more halogen atoms Group, C3-C6 alkenyloxy group optionally having one or more halogen atoms, C3-C6 alkynyloxy group optionally having one or more halogen atoms, one or more groups C3-C6 alkenylthio group which may have a halogen atom, C3-C6 alkynylthio group which may have one or more halogen atoms, C2-C6 which may have one or more halogen atoms Alkyl carbonyl group, C2 to C6 alkyl carbonyloxy group, C2 to C6 alkyl carbonyl thio group, hydroxy carbonyl group, formyl group, C2 to C6 alkoxy carbonyl group, nitro group, cyano group, hydroxy group, one or more halogen atoms C6-C16 aryl group which may be substituted, C6-C16 aryloxy group which may have one or more halogen atoms, C6-C16 arylthio group which may have one or more halogen atoms, one or more C7-C18 aralkyl group optionally having one or more halogen atoms, C7-C18 optionally having one or more halogen atoms Reyl alkoxy group, sulfanyl group, pentafluorosulfanyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C6 alkylsulfonyl group optionally having one or more halogen atoms, one or more C6-C16 arylsulfonyl group which may have one or more halogen atoms, C1-C6 alkylsulfinyl group which may have one or more halogen atoms, C6-, which may have one or more halogen atoms An aminosulfonyl group which may have a C16 arylsulfinyl group, a C1-C6 alkyl group and / or a C6-C12 aryl group, an amino group, an amino group which may have one or two C1-C8 alkyl groups (But may have a halogen atom), and one or two C1-C6 alkyl groups A group consisting of optionally substituted aminocarbonyl groups.
Group P⁶²: A halogen atom, a cyano group, a C3-C6 cycloalkyl group optionally having one or more halogen atoms, a C1-C4 alkoxy group optionally having one or more halogen atoms, and one or more halogen atoms A group consisting of C1-C4 alkylthio group which may be possessed. ]
A tetrazolinone compound represented by the formula:

Group (VII): Formula (7)
[In the formula,
R¹²¹And R¹²²Each independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R¹²³Is a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, a nitro group , Cyano group, aminocarbonyl group optionally having C1 to C6 alkyl group, C2 to C6 haloalkenyl group, C2 to C6 haloalkynyl group, C3 to C6 halocycloalkyl group, C1 to C6 haloalkoxy group, C1 -C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group Group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynyl Thio group, C3 to C6 haloalkenylthio group, C3 to C6 haloalkynylthio group, C2 to C6 alkyl carbonyl group, C2 to C6 haloalkyl carbonyl group, C2 to C6 alkyl carbonyloxy group, C2 to C6 alkyl carbonyl thio group, C2 -C6 alkoxycarbonyl group, hydroxy group, sulfanyl group, amino group optionally having C1-C6 alkyl group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1 -C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C2-C5 alkoxyalkyl group, C2-C5 alkylthioalkyl group or hydrogen atom;
R¹²⁴, R¹²⁵And R¹²⁶Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group or a C1-C3 alkoxy group;
R¹²⁷Represents a C1-C3 alkyl group which may have one or more halogen atoms;
Q⁷Is the group P⁷²Or a divalent 5-membered aromatic heterocyclic group optionally having one or more atoms or groups selected from the following: provided that the heterocyclic group is one or more hetero atoms selected from a nitrogen atom, an oxygen atom and a sulfur atom And the number of nitrogen atoms is 0, 1, 2, 3 or 4 and the number of oxygen atoms and sulfur atoms is 0 or 1.
X⁷Represents an oxygen atom or a sulfur atom;
A⁷Is the group P⁷¹Or a 5- to 10-membered monocyclic or fused-ring heterocyclic group optionally having one or more atoms or groups selected from (wherein the heterocyclic group is a nitrogen atom, an oxygen atom or a sulfur atom) And one or more hetero atoms selected from the group consisting of, the number of nitrogen atoms is 0, 1, 2, 3 or 4 and the number of oxygen atoms and sulfur atoms is 0, 1, 2 or 3.
Group P⁷¹: Halogen atom, C1-C6 alkyl group, C1-C6 haloalkyl group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 cycloalkyl group, C3 -C6 halocycloalkyl group, C1-C6 alkoxy group, C1-C6 haloalkoxy group, C1-C6 alkylthio group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynylthio group , C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 Alkyl carbonyl group, C2 to C6 haloalkyl carbonyl group, C2 to C6 alkyl carbonyloxy group, C2 to C6 alkyl carbonyl thio group, hydroxycarbonyl group, formyl group, C2 to C6 alkoxycarbonyl group, nitro group, cyano group, hydroxy group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloarylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C1-C6 alkyl group A group consisting of an amino group which may be substituted, an aminosulfonyl group which may contain a C1-C6 alkyl group, and an aminocarbonyl group which may have a C1-C6 alkyl group.
Group P⁷²: Halogen atom, C1-C4 alkyl group, C1-C4 haloalkyl group, cyano group, C3-C6 cycloalkyl group, C3-C6 halocycloalkyl group, C1-C4 alkoxy group, C1-C4 haloalkoxy group, C1-C4 A group consisting of an alkylthio group and a C1-C4 haloalkylthio group. ]
And tetrazolinone compounds and salts thereof.

Group (VIII): Formula (8)
[In the formula,
R¹³¹Is the group P⁸¹Or a C6-C16 aryl group optionally having one or more atoms or groups selected from⁸¹Or a C1-C12 alkyl group optionally having one or more atoms or groups selected from⁸¹C3 to C12 cycloalkyl group optionally having one or more atoms or groups selected from⁸¹Or a C2-C12 alkenyl group optionally having one or more atoms or groups selected from⁸¹Or a C3-C12 cycloalkenyl group optionally having one or more atoms or groups selected from⁸¹C2 to C12 alkynyl group optionally having one or more atoms or groups selected from⁸¹Or a C2-C12 acyl group or a hydrogen atom optionally having one or more atoms or groups selected from (wherein the C6-C16 aryl group, the C1-C12 alkyl group, the C3-C12 cycloalkyl group , Said C2-C12 alkenyl group, said C3-C12 cycloalkenyl group, said C2-C12 alkynyl group and said C2-C12 acyl group are each a group P⁸¹When it has two or more atoms or groups selected from, the substituents may be the same or different. );
R¹³²And R¹³³Each represents a hydrogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C12 alkoxycarbonyl group, a hydroxycarbonyl group or a halogen atom;
R¹³⁴And R¹³⁵Each represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R¹³⁶Is a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, a nitro group , An aminocarbonyl group which may have a cyano group, a C 1 -C 6 alkyl group,
C2-C6 haloalkenyl group, C2-C6 haloalkynyl group, C3-C6 halocycloalkyl group, C1-C6 haloalkoxy group, C1-C6 haloalkylthio group, C3-C6 cycloalkyloxy group, C3-C6 halocycloalkyl group Oxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 Alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 acyl group, C2-C6 haloacyl group, C2-C6 acyloxy group, C2-C6 acylthio group, C2-C6 alkoxycarbonyl group , Hydroxyl group, thiol group, amino group, C -C6 alkylamino group, pentafluorosulfanyl group, C3-C9 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1-C4 alkylsulfonyl group, C1-C4 haloalkylsulfonyl group, C1-C4 alkylsulfinyl group , A C 1 -C 4 haloalkylsulfinyl group, a C 2 -C 5 alkoxyalkyl group or a C 2 -C 5 alkylthioalkyl group;
R¹³⁷, R¹³⁸And R¹³⁹Each represents a hydrogen atom, a halogen atom, a C1 to C4 alkyl group, a C1 to C4 haloalkyl group, a C3 to C5 cycloalkyl group, a C3 to C5 halocycloalkyl group, a C1 to C4 alkoxy group or a C1 to C4 haloalkoxy group;
R¹⁴⁰Represents a C1 to C6 alkyl group, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C2 to C6 haloalkenyl group, a C2 to C6 alkoxyalkyl group, a C3 to C6 cycloalkyl group or a C3 to C6 halocycloalkyl group ;
X⁸Represents an oxygen atom or a sulfur atom.
Group P⁸¹: Halogen atom, C1-C6 alkyl group, C1-C6 haloalkyl group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 cycloalkyl group, C3 -C6 halocycloalkyl group, C1 to C6 alkoxy group, C1 to C6 haloalkoxy group, C1 to C6 alkylthio group, C1 to C6 haloalkylthio group, C3 to C6 cycloalkyloxy group, C3 to C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynylthio group , C3-C6 haloalkenylthio group, C3-C6 Roalkynylthio group, C2-C6 acyl group, C2-C6 haloacyl group, C2-C6 acyloxy group, C2-C6 acylthio group, hydroxycarbonyl group, formyl group, C2-C6 alkoxycarbonyl group, nitro group, cyano group, hydroxyl Group, C6-C16 aryl group, C6-C16 haloaryl group, C6-C16 aryloxy group, C6-C16 haloaryloxy group, C6-C16 arylthio group, C6-C16 haloarylthio group, C7-C18 aralkyl group, C7 -C18 haloaralkyl group, C7-C18 arylalkoxy group, C7-C18 haloarylalkoxy group, thiol group, pentafluorosulfuranyl group, C3-C12 trialkylsilyl group, C5-C14 trialkylsilylethynyl group, C1- C6 alkylsul Group, C1-C6 haloalkylsulfonyl group, C6-C16 arylsulfonyl group, C6-C16 haloaryl sulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C6-C16 arylsulfinyl group, C6-C16 halo A group consisting of an aminosulfonyl group which may have an arylsulfinyl group, a C1-C6 alkyl group or a C6-C12 aryl group, and an aminocarbonyl group which may have a C1-C6 alkyl group. ]
A tetrazolinone compound represented by the formula:

Group (IX): Formula (9)
{In the ceremony,
A⁹Is group P⁹²Represents a 5-membered aromatic complex group selected from
R¹⁵⁴And R¹⁵⁵And each independently represents a hydrogen atom or an alkyl group having 1 to 3 carbon atoms, or
R¹⁵⁴When¹⁵⁵And may combine to form a C3-C6 cycloalkane ring together with the carbon atom to which they are attached;
R¹⁵⁶Is an alkyl group having 1 to 12 carbon atoms, a halogen atom, a haloalkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, a halocycloalkyl group having 3 to 12 carbon atoms, or 1 to 12 carbon atoms Alkoxy group, haloalkoxy group having 1 to 12 carbon atoms, alkylthio group having 1 to 12 carbon atoms, haloalkylthio group having 1 to 12 carbon atoms, nitro group, cyano group, hydroxyl group, thiol group, pentafluorosulfanyl group, carbon Alkenyl group having 2 to 12 carbon atoms, haloalkenyl group having 2 to 12 carbon atoms, alkynyl group having 2 to 12 carbon atoms, haloalkynyl group having 2 to 12 carbon atoms, cycloalkyloxy group having 3 to 12 carbon atoms, 3 to 12 halocycloalkyloxy group, C3 to C12 cycloalkylthio group, C2 to C12 alkenyloxy group, C2 to C12 aryl Nyloxy group, haloalkenyloxy group having 2 to 12 carbon atoms, haloalkynyloxy group having 2 to 12 carbon atoms, alkynylthio group having 2 to 12 carbon atoms, alkenylthio group having 2 to 12 carbon atoms, 2 to 12 carbon atoms Haloalkenylthio group, haloalkynylthio group having 2 to 12 carbon atoms, alkylcarbonyl group having 2 to 12 carbon atoms, haloalkylcarbonyl group having 2 to 12 carbon atoms, alkylcarbonyloxy group having 2 to 12 carbon atoms, 2 to 12 alkylcarbonylthio group, C2 to C12 alkoxycarbonyl group, C3 to C12 trialkylsilyl group, C5 to C14 trialkylsilylethynyl group, C1 to C12 alkylsulfonyl Group, haloalkylsulfonyl group having 1 to 12 carbon atoms, alkylsulfinyl group having 1 to 12 carbon atoms, and 1 to 12 carbon atoms Aroalkylsulfinyl group, an aminosulfonyl group optionally having an alkyl group having 1 to 12 carbon atoms, an amino group optionally having an alkyl group having 1 to 12 carbon atoms, an alkyl group having 1 to 12 carbon atoms Represents an aminocarbonyl group which may have a hydroxycarbonyl group or a formyl group;
R¹⁵⁷, R¹⁵⁸, And R¹⁵⁹Are, independently of each other, a hydrogen atom, an alkyl group having 1 to 12 carbon atoms, a halogen atom, a haloalkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, a halocycloalkyl group having 3 to 12 carbon atoms An alkoxy group having 1 to 12 carbon atoms, a haloalkoxy group having 1 to 12 carbon atoms, an alkylthio group having 1 to 12 carbon atoms, a haloalkylthio group having 1 to 12 carbon atoms, a nitro group, a cyano group, a hydroxyl group and a thiol group , Pentafluorosulfanyl group, alkenyl group having 2 to 12 carbon atoms, haloalkenyl group having 2 to 12 carbon atoms, alkynyl group having 2 to 12 carbon atoms, haloalkynyl group having 2 to 12 carbon atoms, or 3 to 12 carbon atoms Cycloalkyloxy group, halocycloalkyloxy group having 3 to 12 carbon atoms, cycloalkylthio group having 3 to 12 carbon atoms, alkenyloxy having 2 to 12 carbon atoms An alkynyloxy group having 2 to 12 carbon atoms, a haloalkenyloxy group having 2 to 12 carbon atoms, a haloalkynyloxy group having 2 to 12 carbon atoms, an alkynylthio group having 2 to 12 carbon atoms, an alkenyl having 2 to 12 carbon atoms Thio group, haloalkenylthio group having 2 to 12 carbon atoms, haloalkynylthio group having 2 to 12 carbon atoms, alkylcarbonyl group having 2 to 12 carbon atoms, haloalkylcarbonyl group having 2 to 12 carbon atoms, 2 to 12 carbon atoms Of alkylcarbonyloxy group, alkylcarbonylthio group having 2 to 12 carbon atoms, alkoxycarbonyl group having 2 to 12 carbon atoms, trialkylsilyl group having 3 to 12 carbon atoms, trialkylsilylethynyl group having 5 to 14 carbon atoms, Alkylsulfonyl having 1 to 12 carbons, haloalkylsulfonyl having 1 to 12 carbons, alkylsulfite having 1 to 12 carbons Group, a haloalkylsulfinyl group having 1 to 12 carbon atoms, an aminosulfonyl group which may have an alkyl group having 1 to 12 carbon atoms, an amino group which may have an alkyl group having 1 to 12 carbon atoms, Represents an aminocarbonyl group optionally having an alkyl group having 1 to 12 carbon atoms, a hydroxycarbonyl group, or a formyl group;
R¹⁶⁰Represents a C1-C3 alkyl group, or a C1-C3 haloalkyl group;
Y⁹Represents an oxygen atom or a sulfur atom;
Q⁹Is an oxygen atom, a sulfur atom, or NR¹⁷²Represents a group;
R¹⁷²Represents a hydrogen atom, an alkyl group having 1 to 6 carbon atoms, or a haloalkyl group having 1 to 6 carbon atoms.
Group P⁹²And a group consisting of the following structural formulas E1 to E36.
[Wherein, # is Q⁹Indicates the bonding position with
R¹⁶¹Is a hydrogen atom, an alkyl group having 1 to 6 carbon atoms, a haloalkyl group having 1 to 6 carbon atoms, an alkenyl group having 2 to 6 carbon atoms, a haloalkenyl group having 2 to 6 carbon atoms, an alkynyl group having 2 to 6 carbon atoms , Represents a haloalkynyl group having 2 to 6 carbon atoms;
R¹⁵⁰, R¹⁵², And R¹⁵³Are each a hydrogen atom, a halogen atom, an alkyl group having 1 to 6 carbon atoms, a haloalkyl group having 1 to 6 carbon atoms, an alkenyl group having 2 to 6 carbon atoms, a haloalkenyl group having 2 to 6 carbon atoms, 6 alkynyl group, haloalkynyl group having 2 to 6 carbon atoms, alkoxycarbonyl group having 2 to 6 carbon atoms, hydroxycarbonyl group or cyano group;
R¹⁵¹Is the group P⁹¹A C 6-16 aryl group optionally having one or more atoms or groups selected from⁹¹And an aralkyl group having 7 to 18 carbon atoms which may have one or more atoms or groups selected from⁹¹And C 3-12 cycloalkyl group optionally having one or more atoms or groups selected from⁹¹Represents an adamantyl group optionally having one or more atoms or a group selected from H, or a hydrogen atom (provided that the aryl group having 6 to 16 carbon atoms, the aralkyl group having 7 to 18 carbon atoms, the carbon atom And when the adamantyl group has two or more substituents, the substituents may be the same or different from each other).
Group P⁹¹: Halogen atom, alkyl group having 1 to 12 carbon atoms, haloalkyl group having 1 to 12 carbon atoms, alkoxy group having 1 to 12 carbon atoms, haloalkoxy group having 1 to 12 carbon atoms, alkylthio group having 1 to 12 carbon atoms, C1-12 haloalkylthio, hydroxycarbonyl, formyl, nitro, cyano, hydroxyl, thiol, pentafluorosulfanyl, alkenyl having 2 to 12 carbons, halo having 2 to 12 carbons Alkenyl group, alkynyl group having 2 to 12 carbon atoms, haloalkynyl group having 2 to 12 carbon atoms, cycloalkyl group having 3 to 12 carbon atoms, halocycloalkyl group having 3 to 12 carbon atoms, cyclo Alkyloxy group, C3-C12 halocycloalkyloxy group, C3-C12 cycloalkylthio group, C2-C12 alky Roxy group, alkynyloxy group having 2 to 12 carbon atoms, haloalkenyloxy group having 2 to 12 carbon atoms, haloalkynyloxy group having 2 to 12 carbon atoms, alkynylthio group having 2 to 12 carbon atoms, 2 to 12 carbon atoms Alkenylthio group, haloalkenylthio group having 2 to 12 carbon atoms, haloalkynylthio group having 2 to 12 carbon atoms, alkylcarbonyl group having 2 to 12 carbon atoms, haloalkylcarbonyl group having 2 to 12 carbon atoms, 2 carbon atoms An alkylcarbonyloxy group having 1 to 12 carbon atoms, an alkylcarbonylthio group having 2 to 12 carbon atoms, an alkoxycarbonyl group having 2 to 12 carbon atoms, an aryl group having 6 to 16 carbon atoms, a haloaryl group having 6 to 16 carbon atoms,ア リ ー ル 16 aryloxy group, C 6-16 haloaryloxy group, C 6-16 arylthio group, C 6-16 haloia Arylthio group, an aralkyl group having 7 to 18 carbon atoms, a haloaralkyl group having 7 to 18 carbon atoms, an arylalkoxy group having 7 to 18 carbon atoms, a haloarylalkoxy group having 7 to 18 carbon atoms, Alkylsilyl group, trialkylsilylethynyl group having 5 to 14 carbon atoms, alkylsulfonyl group having 1 to 12 carbon atoms, haloalkylsulfonyl group having 1 to 12 carbon atoms, arylsulfonyl group having 6 to 16 carbon atoms, 6 to 6 carbon atoms 16 haloarylsulfonyl group, alkylsulfinyl group having 1 to 12 carbon atoms, haloalkylsulfinyl group having 1 to 12 carbon atoms, arylsulfinyl group having 6 to 16 carbon atoms, haloarylsulfinyl group having 6 to 16 carbon atoms, carbon number 2-11 polyoxaalkyloxy group, C2-C5 oxacycloalkyloxy group, C1-C1 An aminocarbonyl group which may have 12 alkyl groups and / or an aryl group having 6 to 12 carbon atoms, an alkyl group having 1 to 12 carbon atoms and / or an aryl group having 6 to 12 carbon atoms A group consisting of an aminosulfonyl group which may be substituted and an amino group which may have an alkyl group having 1 to 12 carbon atoms. ]}
A tetrazolinone compound represented by the formula:

Group (X): Formula (10)
[In the formula,
R¹⁸¹And R¹⁸²Each independently represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group;
R¹⁸³And C 1 -C 6 alkyl group which may have one or more halogen atoms, C 1-C 6 alkoxy group which may have one or more halogen atoms, and one or more halogen atoms C3-C6 cycloalkyl group, halogen atom, C2-C6 alkenyl group optionally having one or more halogen atoms, cyano group, C1-C6 alkylthio group optionally having one or more halogen atoms, A C2-C6 alkynyl group which may have one or more halogen atoms, a nitro group, an aminocarbonyl group which may have one or more C1-C6 alkyl groups, or one or more halogen atoms Good C3-C6 cycloalkyloxy group, C3-C6 cycloalkylthio group optionally having one or more halogen atoms, C3-optionally having one or more halogen atoms 6 alkenyloxy group, C3-C6 alkynyloxy group optionally having one or more halogen atoms, C3-C6 alkenylthio group optionally having one or more halogen atoms, one or more halogen atoms C3-C6 alkynylthio group, C2-C6 alkoxycarbonyl group, hydroxy group, sulfanyl group, C1-C8 alkylamino group optionally having one or more halogen atoms, pentafluorosulfanyl group, C3 -C9 trialkylsilyl group, C1-C6 alkylsulfonyl group optionally having one or more halogen atoms, C1-C6 alkylsulfinyl group optionally having one or more halogen atoms, C2-C6 alkyl carbonyl Represents a group, a C2-C5 alkoxyalkyl group or a C2-C5 alkylthioalkyl group;
R¹⁸⁴, R¹⁸⁵And R¹⁸⁶Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or a C1-C3 alkoxy group optionally having one or more halogen atoms;
R¹⁸⁷Represents a C1-C3 alkyl group which may have one or more halogen atoms;
Q^TenIs group P¹⁰³Represents a divalent group selected from
A^TenIs the group P¹⁰²Or a C6-C16 aryloxy group optionally having one or more atoms or groups selected from¹⁰²C6-C16 arylthio group optionally having one or more atoms or groups selected from¹⁹⁵O-N = C (R¹⁹⁶)-, R¹⁹³R¹⁹⁴N-N = C (R¹⁹⁶)-, R¹⁹³R¹⁹⁴N-CH = N-, group P¹⁰²C7-C18 aralkyl group optionally having one or more atoms or groups selected from¹⁰²C7-C18 aralkyloxy group optionally having one or more atoms or groups selected from¹⁰²C7-C16 aryloxyalkyl group optionally having one or more atoms or groups selected from¹⁰²C7-C16 arylcarbonyl group optionally having one or more atoms or groups selected from¹⁰²Anilino group optionally having one or more atoms or groups selected from¹⁰²Or a C2-C9 heteroaryloxy group optionally having one or more atoms or groups selected from: wherein the heteroaryl moiety in the heteroaryloxy group is a 5-, 6-, 5-, or 5-membered ring; A fused ring with a member ring, a fused ring of a 5-membered ring and a 6-membered ring or a fused ring of a 6-membered ring and a 6-membered ring), a C3-C6 cycloalkyloxy group or a C4-C10 cycloalkylalkoxy group Representation
R¹⁹³And R¹⁹⁴Represents a C1-C3 alkyl group which may be the same or different and may have one or more halogen atoms;
R¹⁹⁵Is a C1-C6 alkyl group optionally having one or more halogen atoms, a C2-C6 alkenyl group optionally having one or more halogen atoms, C2 optionally having one or more halogen atoms -C6 alkynyl group, C3-C6 cycloalkyl group optionally having one or more halogen atoms, group P¹⁰¹Or a C7-C18 aralkyl group optionally having one or more atoms or groups selected from¹⁰¹Represents a phenyl group which may have one or more atoms or groups selected from
R¹⁹⁶Is a C1-C6 alkyl group which may have one or more halogen atoms, a hydrogen atom, a C3-C6 cycloalkyl group which may have one or more halogen atoms, or one or more halogen atoms Represents an optionally substituted phenyl group;
X^TenRepresents an oxygen atom or a sulfur atom.
Group P¹⁰¹: Halogen atom, cyano group, C1-C4 alkyl group optionally having one or more halogen atoms, C3-C6 cycloalkyl group optionally having one or more halogen atoms, one or more halogen atoms A group consisting of a C1-C4 alkoxy group which may have and a C1-C4 alkylthio group which may have one or more halogen atoms.
Group P¹⁰²C1 to C6 alkyl group optionally having one or more halogen atoms, halogen atom, cyano group, hydroxy group, C3 to C6 cycloalkyl group optionally having one or more halogen atoms, one or more C1-C6 alkoxy group which may have a halogen atom, C1-C6 alkylthio group which may have one or more halogen atoms, C2-C6 alkenyl group which may have one or more halogen atoms A C2 to C6 alkynyl group which may have one or more halogen atoms, a C1 to C8 alkylamino group which may have one or more halogen atoms, or one or more halogen atoms C1-C6 alkylsulfinyl group, C1-C6 alkylsulfonyl group optionally having one or more halogen atoms, pentafluorosulfanyl group, C2-C6 group Coxy carbonyl group, C2 to C6 alkyl carbonyl group, C2 to C6 alkyl carbonyloxy group, C2 to C6 alkyl carbonyl amino group, aminocarbonyl group optionally having one or more C1 to C6 alkyl groups, and C3 to C9 A group consisting of trialkylsilyl groups.
Group P¹⁰³: A group consisting of group Q11 and group Q12
(In the formula, R¹⁸⁸, R¹⁸⁹, R¹⁹⁰And R¹⁹¹Each independently represents a hydrogen atom, a halogen atom, or a C1-C4 alkyl group optionally having one or more halogen atoms;¹⁰Represents a binding site to, and ● represents a binding site to an oxygen atom. ). ]
A tetrazolinone compound represented by the formula:

Group (XI): Formula (11)
[In the formula,
R²⁰⁵Represents a C1-C3 alkyl group which may have one or more halogen atoms;
E⁴⁰Represents a divalent 5-membered heteroaryl group or a divalent 6-membered heteroaryl group;
Y¹¹Is-(CH₂)_n ¹¹-G-, -G- (CH₂)_n ¹¹-, -G- (CH₂)_n ¹¹-G-, -G-CH₂CH₂-G-CH₂CH₂-G-, -CH₂-G-CH₂CH₂-G-, -G-CH₂CH₂-G-CH₂-, -CH = CH-, -CH = CH-G-, -G-CH = CH-, -CH = CH-CH₂-G-, -G-CH₂-CH = CH-, -G-CH = CH-CH₂-, -CH₂-CH = CH-G-, -CH = CH-G-CH₂-, -CH₂-G-CH = CH-, -CH = CH-CH₂-G-CH₂-, -CH₂-G-CH₂-CH = CH-, -CH = CH-G-CH₂CH₂-, -CH₂CH₂-G-CH = CH-, -G-CH = CH-CH₂CH₂-, -CH₂CH₂-CH = CH-G-, -CH = CH-G-CH = CH-, -C≡C-, -C≡C-CH₂-G-, -G-CH₂-C≡C-, -C≡C-CH₂-G-CH₂-Or-CH₂-G-CH₂Represents -C≡C- (where Y is¹¹Is optionally substituted by one or more atoms or groups selected from the group consisting of halogen atoms and C1-C3 alkyl groups, and when substituted by two or more atoms or groups, the atoms and groups are G may be the same or different; G is an oxygen atom, a sulfur atom, or NR^BRepresents; R^BRepresents a hydrogen atom or a C1-C3 alkyl group, n¹¹Represents an integer of 1 to 10. Also, Y¹¹Q to the left of¹³Join and E on the right⁴⁰Joins. );
Q¹³Is a divalent C6-C10 aryl group, provided that the divalent C6-C10 aryl group is¹¹²And one or more atoms or groups selected from Or a divalent 5- to 10-membered heterocyclic group, provided that the divalent 5- to 10-membered heterocyclic group is a group P¹¹²And at least one atom selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom as a ring-constituting atom, and containing two or more atoms. If so, the atoms may be identical or different. Represents);
X¹¹Represents an oxygen atom or a sulfur atom;
A¹¹Is a C6-C10 aryl group, an adamantyl group, a C6-C10 aryloxy group, a C6-C10 arylthio group, a C6-C10 arylamino group, a C3-C10 cycloalkyl group, a 5-10-membered heterocyclic group (provided that the 5 The -10-membered heterocyclic group contains one or more atoms selected from the group consisting of nitrogen atom, oxygen atom and sulfur atom as ring constituent atoms, and in the case of containing two or more atoms, the atoms are the same or different And 5- to 10-membered heteroaryloxy group (wherein the 5- to 10-membered heteroaryloxy group is at least one member selected from the group consisting of nitrogen atom, oxygen atom and sulfur atom as a ring constituent atom). When the atoms contain two or more atoms, the atoms may be the same or different), a 5-10 membered heteroarylthio group (provided that the The -10-membered heteroarylthio group contains one or more atoms selected from the group consisting of nitrogen atoms, oxygen atoms and sulfur atoms as ring-constituting atoms, and in the case of containing two or more atoms, the atoms are identical or A 5- to 10-membered heteroarylamino group (wherein the 5- to 10-membered heteroarylamino group is selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom as a ring constituent atom) Containing one or more atoms, and when containing two or more atoms, the atoms may be the same or different), a C6-C10 arylsulfonyl group, a C6-C10 arylsulfinyl group, or a group P¹¹³Or —CH = NH optionally having one or two groups selected from¹¹³When having two groups selected from, the groups may be the same or different. Wherein the C6-C10 aryl group, the adamantyl group, the C6-C10 aryloxy group, the C6-C10 arylthio group, the C6-C10 arylamino group, the C3-C10 cycloalkyl group, and the 5- to 10-membered heterocyclic group , A 5- to 10-membered heteroaryloxy group, a 5- to 10-membered heteroarylthio group, a 5- to 10-membered heteroarylamino group, a C6-C10 arylsulfonyl group and a C6-C10 arylsulfinyl group¹¹¹And one or more atoms or groups selected from, and in the case of two or more atoms or groups, the atoms or groups may be the same or different. ).
Group P¹¹¹: Halogen atom, C1-C6 alkyl group, C1-C6 haloalkyl group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 cycloalkyl group, C3 -C6 halocycloalkyl group, C1 to C6 alkoxy group, C1 to C6 haloalkoxy group, C1 to C6 alkylthio group, C1 to C6 haloalkylthio group, C3 to C6 cycloalkyloxy group, C3 to C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynylthio group , C3-C6 haloalkenylthio group, C3-C6 halo Roalkynylthio group, C 2 -C 6 alkylcarbonyl group, C 2 -C 6 haloalkylcarbonyl group, C 2 -C 6 alkylcarbonyloxy group, C 2 -C 6 alkylcarbonylthio group, hydroxycarbonyl group, formyl group, C 2 -C 6 alkoxycarbonyl group, nitro Group, cyano group, hydroxyl group, C1 to C6 alkylsulfonyl group, C1 to C6 haloalkylsulfonyl group, C1 to C6 alkylsulfinyl group, C1 to C6 haloalkylsulfinyl group, amino optionally having C1 to C6 alkyl group A group, an aminosulfonyl group which may have a C1-C6 alkyl group, and an aminocarbonyl group which may have a C1-C6 alkyl group.
Group P¹¹²: A group consisting of a halogen atom, a cyano group, a C3 to C6 cycloalkyl group, a C3 to C6 halocycloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group and a C1 to C4 haloalkylthio group .
  Group P¹¹³A group consisting of a C1 to C6 alkyl group, a C1 to C6 haloalkyl group, a C3 to C6 cycloalkyl group, and a C3 to C6 halocycloalkyl group. ]
A tetrazolinone compound represented by the formula:

Group (XII): Formula (12)
[In the formula,
R²¹¹Is a C1 to C6 alkyl group, a C3 to C6 cycloalkyl group, a halogen atom, a C1 to C6 haloalkyl group, a C2 to C6 alkenyl group, a C1 to C6 alkoxy group, a C1 to C6 alkylthio group, a C2 to C6 alkynyl group, a nitro group , Cyano group, aminocarbonyl group optionally having C1 to C6 alkyl group, C2 to C6 haloalkenyl group, C2 to C6 haloalkynyl group, C3 to C6 halocycloalkyl group, C1 to C6 haloalkoxy group, C1 -C6 haloalkylthio group, C3 to C6 cycloalkyloxy group, C3 to C6 halocycloalkyloxy group, C3 to C6 cycloalkylthio group, C3 to C6 alkenyloxy group, C3 to C6 alkynyloxy group, C3 to C6 haloalkenyloxy Group, C 3 -C 6 haloalkynyloxy group, C 3 -C 6 alkeny Thio group, C3-C6 alkynylthio group, C3-C6 haloalkenylthio group, C3-C6 haloalkynylthio group, C2-C6 alkylcarbonyl group, C2-C6 haloalkylcarbonyl group, C2-C6 alkylcarbonyloxy group, C2-C6 C6 alkylcarbonylthio group, C2-C6 alkoxycarbonyl group, hydroxyl group, thiol group, amino group which may have C1-C6 alkyl group, pentafluorosulfuranyl group, C3-C9 trialkylsilyl group, C5 -C14 trialkylsilylethynyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, C2-C6 alkoxyalkyl group or C2-C6 alkylthioalkyl group It represents;
R²¹², R²¹³And R²¹⁴The same or different, each representing a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C2-C3 alkenyl group, a C2-C3 haloalkenyl group or a C1-C3 alkoxy group;
R²¹⁵Represents a C1-C3 alkyl group which may have one or more halogen atoms;
Y¹²Is -C (R^A1R^A2) -Z-, -C (R^A1R^A2) C (R^A3R^A4) -Z-, -C (R^A1R^A2) -Z-C (R^A3R^A4)-, -Z-C (R^A1R^A2) C (R^A3R^A4)-, -C (R^A1R^A2) C (R^A3R^A4) C (R^A5R^A6) -Z-, -C (R^A1R^A2) C (R^A3R^A4) -Z-C (R^A5R^A6)-, -C (R^A1R^A2) -Z-C (R^A3R^A4) C (R^A5R^A6)-, -Z-C (R^A1R^A2) C (R^A3R^A4) C (R^A5R^A6)-, -C (R^A1) = C (R^A2) C (R^A3R^A4) -Z-, -Z-C (R^A1R^A2) C (R^A3) = C (R^A4)-, -C≡C-C (R^A1R^A2) -Z-, -Z-C (R^A1R^A2) -C≡C-, -Z-C (R^A1R^A2) C (R^A3R^A4) -Z-, -C (R^A1) = C (R^A2)-, -C (R^A1) = C (R^A2) C (R^A3R^A4)-, -C (R^A1) = C (R^A2) C (R^A3R^A4) C (R^A5R^A6)-, -C (R^A1R^A2) C (R^A3) = C (R^A4) C (R^A5R^A6)-, -C (R^A1R^A2) C (R^A3R^A4) C (R^A5) = C (R^A6)-, -C (R^A1) = C (R^A2) C (R^A3) = C (R^A4)-, -C≡C-, -C≡C-C (R^A1R^A2)-, -C≡C-C (R^A1R^A2) C (R^A3R^A4)-, -C (R^A1R^A2) C (R^A3R^A4) -C≡C- or -C (R^A1R^A2) -C≡C-C (R^A3R^A4)-(But with each left edge and Q¹⁴And united, R^A1, R^A2, R^A3, R^A4, R^A5, And R^A6Each represents a hydrogen atom, a halogen atom or a C1-C3 alkyl group, and Z is an oxygen atom, a sulfur atom or NR^CRepresents R, R^CAnd each represents a C1 to C6 alkyl group, a C1 to C6 haloalkyl group, a C3 to C6 cycloalkyl group, or a C3 to C6 halocycloalkyl group. Represents);
Q¹⁴Is a divalent C3-C10 carbocyclic group or a divalent heterocyclic group (provided that the divalent heterocyclic group is at least one member selected from the group consisting of a nitrogen atom, an oxygen atom and a sulfur atom as a ring constituent atom) In the case of fused rings, 5-membered ring and 5-membered ring, 5-membered ring and 6-membered ring, and 6-membered ring in the case of fused rings And a 6-membered ring represent a fused ring));
X¹²Represents an oxygen atom or a sulfur atom;
A¹²Is a C6-C10 aryl group, a C6-C10 aryloxy group, a C6-C10 arylthio group, a C6-C10 arylsulfonyl group, a C6-C10 arylamino group, a hydrogen atom, a heterocyclic group (wherein the heterocyclic group is A ring-constituting atom containing one or more atoms selected from the group consisting of nitrogen atom, oxygen atom and sulfur atom, and containing two or more atoms selected from the group consisting of nitrogen atom, oxygen atom and sulfur atom; The atoms may be the same or different) or R^C2-O-N = C (R^C2)-(However, R^C2And each represents a C1 to C6 alkyl group, a C1 to C6 haloalkyl group, a C3 to C6 cycloalkyl group, or a C3 to C6 halocycloalkyl group. Represents. (Wherein, the divalent C3-C10 carbon group of Q, and the divalent heterocyclic group, and A¹²C6-C10 aryl group, C6-C10 aryloxy group, C6-C10 arylthio group, C6-C10 arylamino group and heterocyclic group are¹²¹And one or more atoms or groups selected from )
Group P¹²¹: Halogen atom, C1-C6 alkyl group, C1-C6 haloalkyl group, C2-C6 alkenyl group, C2-C6 haloalkenyl group, C2-C6 alkynyl group, C2-C6 haloalkynyl group, C3-C6 cycloalkyl group, C3 -C6 halocycloalkyl group, C1 to C6 alkoxy group, C1 to C6 haloalkoxy group, C1 to C6 alkylthio group, C1 to C6 haloalkylthio group, C3 to C6 cycloalkyloxy group, C3 to C6 halocycloalkyloxy group, C3-C6 cycloalkylthio group, C3-C6 alkenyloxy group, C3-C6 alkynyloxy group, C3-C6 haloalkenyloxy group, C3-C6 haloalkynyloxy group, C3-C6 alkenylthio group, C3-C6 alkynylthio group , C3-C6 haloalkenylthio group, C3-C6 Roalkynylthio group, C 2 -C 6 alkylcarbonyl group, C 2 -C 6 haloalkylcarbonyl group, C 2 -C 6 alkylcarbonyloxy group, C 2 -C 6 alkylcarbonylthio group, hydroxycarbonyl group, formyl group, C 2 -C 6 alkoxycarbonyl group, nitro Group, cyano group, hydroxyl group, C1-C6 alkylsulfonyl group, C1-C6 haloalkylsulfonyl group, C1-C6 alkylsulfinyl group, C1-C6 haloalkylsulfinyl group, amino group optionally having C1-C6 alkyl group And a group consisting of an aminosulfonyl group which may have a C1-C6 alkyl group and an aminocarbonyl group which may have a C1-C6 alkyl group. ]
A tetrazolinone compound represented by the formula:

Group (XIII): Formula (13)
[Wherein, X¹³Is CR²²⁶Or represents a nitrogen atom,
R²²¹, R²²², R²²³, R²²⁴And R²²⁶Each independently represents a halogen atom, a hydrogen atom, a cyano group, a C1 to C4 alkyl group optionally having one or more halogen atoms, or a C1 to C4 alkoxy optionally having one or more halogen atoms Represents a group,
R²²⁵Is a halogen atom, a C1-C4 alkyl group which may have one or more halogen atoms, a C3-C4 cycloalkyl group which may have one or more halogen atoms, or one or more halogen atoms. Represents a C1-C4 alkoxy group which may be substituted. ]
A tetrazolinone compound represented by the formula:

Group (XIV): Formula (14)
[In the formula, A¹⁴Represents a group A15, A16, A17 or A18 below;

R²³¹Is a hydrogen atom, a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or one or more halogens Represents a C1-C4 alkoxy group which may have an atom,
R²³²And R²³³Each represents a hydrogen atom, a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, or a C1-C4 alkoxy group optionally having one or more halogen atoms,
E⁵⁹And E⁶¹And each represents a hydrogen atom, a halogen atom, a C1-C4 alkoxy group optionally having one or more halogen atoms, or a C1-C4 alkyl group optionally having one or more halogen atoms,
E⁵³, E⁵⁸And E⁶⁰And each represents a hydrogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, or a C3-C4 cycloalkyl group optionally having one or more halogen atoms,
E⁵⁰, E⁵¹, E⁵², E⁵⁴, E⁵⁵, E⁵⁶And E⁵⁷Are each a hydrogen atom, a halogen atom, a cyano group, an aldehyde group, a C1-C4 alkoxy group optionally having one or more halogen atoms, a C1-C4 alkyl group optionally having one or more halogen atoms Or a C3-C4 cycloalkyl group optionally having one or more halogen atoms. ]
A tetrazolinone compound represented by the formula:

Group (XV): Formula (15)
[Wherein, R²⁴¹And R²⁴²Each independently represents a hydrogen atom, a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, or a C1-C4 alkoxy group optionally having one or more halogen atoms;
R²⁴³Is a hydrogen atom, a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or one or more halogen atoms Represents a C1-C4 alkoxy group which may have
R²⁴⁴Represents a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, a C1-C4 alkoxy group optionally having one or more halogen atoms, or a cyano group;
n¹⁵Represents an integer from 0 to 4 (provided that n is¹⁵When R is an integer of 2 or more, each R²⁴⁴Is at least one other R²⁴⁴It may be the same as or different from );
X¹⁵Is nitrogen or CR²⁴⁵Represents
R²⁴⁵Represents a hydrogen atom, a halogen atom, a C1 to C4 alkyl group optionally having one or more halogen atoms, a C1 to C4 alkoxy group optionally having one or more halogen atoms, or a cyano group. ]
A tetrazolinone compound represented by the formula:

Group (XVI): Formula (16)
[Wherein, R²⁵¹And R²⁵²Each independently represents a halogen atom, a C1-C4 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, one or more halogens A C2-C4 alkenyl group which may have an atom, a C2-C4 alkynyl group which may have one or more halogen atoms, a C1-C4 alkoxy group which may have one or more halogen atoms, Represents a C1-C4 alkylthio group which may have one or more halogen atoms, a cyano group or a nitro group, provided that m is¹⁶When is an integer of 2 or more, 2 or more of R²⁵¹May be the same or different, n¹⁶When is an integer of 2 or more, 2 or more of R²⁵²It may be the same or different. );
m¹⁶And n¹⁶Each independently represents an integer from 0 to 4;
R²⁵³And R²⁵⁴Each independently represents a hydrogen atom or a C1-C3 alkyl group optionally having one or more halogen atoms;
Y¹⁶Is the formula -OC (= X¹⁶) Z¹⁶R²⁵⁵Or-SC (= X¹⁶) Z¹⁶R²⁵⁵Represents
R²⁵⁵Represents a C1-C3 alkyl group which may have one or more halogen atoms;
Z¹⁶Is oxygen atom, sulfur atom, NR²⁵⁸Or direct binding;
R²⁵⁸Represents a C1-C3 alkyl group optionally having one or more halogen atoms or a hydrogen atom;
Q¹⁶Is group P¹³¹Represents a pyrazolyl group optionally having one or more atoms or groups selected from
W¹⁶And X¹⁶Each independently represents an oxygen atom or a sulfur atom.
Group P¹³¹: Having a halogen atom, a C1-C6 alkyl group which may have one or more halogen atoms, a C2-C6 alkenyl group which may have one or more halogen atoms, one or more halogen atoms C2-C6 alkynyl group, C3-C6 cycloalkyl group optionally having one or more halogen atoms, C1-C6 alkoxy group optionally having one or more halogen atoms, one or more halogen atoms C 1 -C 6 alkylthio group which may have one or more C 3 -C 6 cycloalkyloxy group which may have one or more halogen atoms, C 3-C 6 cycloalkylthio group which may have one or more halogen atoms Group, C3-C6 alkenyloxy group optionally having one or more halogen atoms, C3-C6 alkynyloxy optionally having one or more halogen atoms A C3-C6 alkenylthio group which may have one or more halogen atoms, a C3-C6 alkynylthio group which may have one or more halogen atoms, or one or more halogen atoms Good C2-C6 alkylcarbonyl group, C2-C6 alkylcarbonyloxy group optionally having one or more halogen atoms, C2-C6 alkylcarbonylthio group optionally having one or more halogen atoms, carboxy group An amino group optionally having a formyl group, a C2 to C6 alkoxycarbonyl group optionally having one or more halogen atoms, a nitro group, a cyano group, and a C1 to C6 alkyl group (however, the alkyl group) Is a group consisting of one or more halogen atoms). ]
An aromatic compound represented by

Group (XVII): Formula (17)
[Wherein, R²⁶¹Represents a halogen atom or a C1-C4 alkyl group optionally having one or more halogen atoms;
R²⁶³Represents a hydrogen atom or a C1-C4 alkyl group optionally having one or more halogen atoms;
R²⁶⁷Is a C1-C3 alkyl group which may have one or more halogen atoms, a hydrogen atom, a halogen atom, a C1-C3 alkoxy group which may have one or more halogen atoms, and one or more halogen atoms. A C3-C4 cycloalkyl group which may be substituted or a C2-C4 alkenyl group which may have one or more halogen atoms;
Z¹⁷Represents a halogen atom, a C1-C3 alkoxy group or a C1-C3 alkyl group;
Z¹⁸Represents a C1-C3 alkyl group optionally having one or more halogen atoms or a halogen atom;
Q¹⁷Represents the following groups Q18, Q19 or Q20;
R²⁶⁵Represents a C1-C3 alkyl group which may have one or more halogen atoms;
R²⁷⁰Represents a hydrogen atom, a hydroxyl group or a methyl group;
R²⁷¹Represents a hydrogen atom, a hydroxyl group, a methyl group or a methoxy group;
X¹⁷Represents an oxygen atom or a sulfur atom;
X¹⁸Is oxygen atom, sulfur atom, NR²⁷²Or direct binding;
R²⁷²Represents a C1-C3 alkyl group optionally having one or more halogen atoms, or a hydrogen atom. ]
An aromatic compound represented by

Group (XVIII): Formula (18)
[Wherein, R²⁸¹Represents a halogen atom or a C1-C4 alkyl group optionally having one or more halogen atoms;
R²⁸³Represents a hydrogen atom, a halogen atom or a C1-C4 alkyl group optionally having one or more halogen atoms;
R²⁸⁷Is a C1-C3 alkyl group which may have one or more halogen atoms, a hydrogen atom, a halogen atom, a C1-C3 alkoxy group which may have one or more halogen atoms, or one or more halogen atoms. Represents an optionally substituted C3-C4 cycloalkyl group;
A¹⁸Represents the following groups A19, A20 or A21;
Z¹⁹And Z²⁰Each independently represents a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, or a C1-C3 alkoxy group optionally having one or more halogen atoms;
Q^{twenty one}Represents the following groups Q22, Q23 or Q24;
R²⁸⁵Represents a C1-C3 alkyl group which may have one or more halogen atoms;
R²⁹⁰Represents a hydrogen atom, a hydroxyl group or a methyl group;
R²⁹¹Represents a hydrogen atom, a hydroxyl group, a methyl group or a methoxy group;
X¹⁹Represents an oxygen atom or a sulfur atom;
X²⁰Is oxygen atom, sulfur atom, NR²⁹²Or direct binding;
R²⁹²Represents a C1-C3 alkyl group optionally having one or more halogen atoms, or a hydrogen atom. ]
An aromatic compound represented by

Group (XIX): Formula (19)
[In the formula,
R³⁰¹Represents a hydrogen atom or a C1-C3 alkyl group;
R³⁰², R³⁰³, R³⁰⁴And R³⁰⁵Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or Represents a C1-C3 alkoxy group which may have one or more halogen atoms;
Z^{twenty one}Represents a C1-C3 alkyl group;
n¹⁹Represents an integer of 1 to 4; ]
The carbamate compound shown by these.

Group (XX): Formula (20)
[In the formula,
R³¹¹Represents a hydrogen atom or a C1-C3 alkyl group;
R³¹², R³¹³, R³¹⁴And R³¹⁵Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or Represents a C1-C3 alkoxy group which may have one or more halogen atoms;
Z^{twenty two}Represents a halogen atom;
Z^{twenty three}Represents a halogen atom or a C1-C3 alkyl group;
n²⁰Represents an integer of 0 to 3. ]
The carbamate compound shown by these.

Group (XXI): Formula (21)
[In the formula,
R³²¹Represents a hydrogen atom or a C1-C3 alkyl group;
R³²², R³²³, R³²⁴And R³²⁵Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or Represents a C1-C3 alkoxy group which may have one or more halogen atoms;
Z^{twenty four}Represents a C1-C3 alkyl group;
n^{twenty one}Represents an integer of 1 to 3. ]
The carbamate compound shown by these.

Group (XXII): Formula (22)
[In the formula,
R³³¹Represents a hydrogen atom or a C1-C3 alkyl group;
R³³², R³³³, R³³⁴And R³³⁵Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or Represents a C1-C3 alkoxy group which may have one or more halogen atoms;
Z^{twenty five}Represents a halogen atom;
Z²⁶Represents a halogen atom or a C1-C3 alkyl group;
n^{twenty two}Represents an integer of 0 to 2; ]
The carbamate compound shown by these.

Group (XXIII): Formula (23)
[Wherein, R³⁴¹Represents a hydrogen atom or a C1-C3 alkyl group;
R³⁴², R³⁴³, R³⁴⁴And R³⁴⁵Each independently represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group optionally having one or more halogen atoms, a C3-C4 cycloalkyl group optionally having one or more halogen atoms, or Represents a C1-C3 alkoxy group which may have one or more halogen atoms;
Z²⁷Represents a halogen atom, a C1-C3 alkyl group or a C1-C3 alkoxy group;
n^{twenty three}Represents an integer of 0 to 3. ]
The carbamate compound shown by these.   An effective amount of group (I), group (II), group (III), group (IV), group (V), group (VI), group (VII), group (VIII), group (group 1) according to claim 1 IX), group (X), group (XI), group (XII), group (XIII), group (XIV), group (XV), group (XVI), group (XVII), group (XVIII), group (XVIII), group (XVIII) A tetrazolinone compound according to any one selected from the group consisting of XIX), groups (XX), groups (XXI), groups (XXII) and groups (XXIII), and an effective amount of groups A to F according to claim 1 A pest control method comprising the step of applying a plant or a soil for cultivating a plant with one or more components selected from the group consisting of   The pest control method according to claim 2, wherein the plant is a seed, a bulb or a seedling.   The method for controlling pests according to claim 2, wherein the plant is corn, soybean, cotton, wheat, barley, sugar beet, Brassica napus or rice.   An effective amount of group (I), group (II), group (III), group (IV), group (V), group (VI), group (VII), group (VIII), group (group 1) according to claim 1 IX), group (X), group (XI), group (XII), group (XIII), group (XIV), group (XV), group (XVI), group (XVII), group (XVIII), group (XVIII), group (XVIII) A tetrazolinone compound according to any one selected from the group consisting of XIX), groups (XX), groups (XXI), groups (XXII) and groups (XXIII), and an effective amount of groups A to F according to claim 1 A pest control method comprising the step of applying one or more components selected from the group consisting of to a pest or a habitat of a pest.   A plant seed or bulb to which an effective amount of the pest control composition according to claim 1 is attached.