JP2015178456A - 高速メチル化法 - Google Patents

高速メチル化法 Download PDF

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Publication number
JP2015178456A
JP2015178456A JP2012159725A JP2012159725A JP2015178456A JP 2015178456 A JP2015178456 A JP 2015178456A JP 2012159725 A JP2012159725 A JP 2012159725A JP 2012159725 A JP2012159725 A JP 2012159725A JP 2015178456 A JP2015178456 A JP 2015178456A
Authority
JP
Japan
Prior art keywords
methylation
boronic acid
acid ester
reaction
carbon
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012159725A
Other languages
English (en)
Japanese (ja)
Inventor
正昭 鈴木
Masaaki Suzuki
正昭 鈴木
良祐 伊集院
Ryosuke IJUIN
良祐 伊集院
久志 土居
Hisashi Doi
久志 土居
浩子 古山
Hiroko Furuyama
浩子 古山
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gifu University NUC
RIKEN Institute of Physical and Chemical Research
Original Assignee
Gifu University NUC
RIKEN Institute of Physical and Chemical Research
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gifu University NUC, RIKEN Institute of Physical and Chemical Research filed Critical Gifu University NUC
Priority to JP2012159725A priority Critical patent/JP2015178456A/ja
Priority to PCT/JP2013/069548 priority patent/WO2014014067A1/fr
Publication of JP2015178456A publication Critical patent/JP2015178456A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
    • C07C217/14—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
    • C07C217/16—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring not being further substituted
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05—Isotopically modified compounds, e.g. labelled

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2012159725A 2012-07-18 2012-07-18 高速メチル化法 Pending JP2015178456A (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2012159725A JP2015178456A (ja) 2012-07-18 2012-07-18 高速メチル化法
PCT/JP2013/069548 WO2014014067A1 (fr) 2012-07-18 2013-07-18 PROCÉDÉ DE MÉTHYLATION DE CARBONE sp3

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2012159725A JP2015178456A (ja) 2012-07-18 2012-07-18 高速メチル化法

Publications (1)

Publication Number Publication Date
JP2015178456A true JP2015178456A (ja) 2015-10-08

Family

ID=49948889

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012159725A Pending JP2015178456A (ja) 2012-07-18 2012-07-18 高速メチル化法

Country Status (2)

Country Link
JP (1) JP2015178456A (fr)
WO (1) WO2014014067A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021199310A1 (fr) * 2020-03-31 2021-10-07 エヌ・イーケムキャット株式会社 Procédé de production d'un composé aromatique

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9845295B2 (en) * 2015-11-24 2017-12-19 Purdue Research Foundation Triphenylethylene compounds and uses thereof
CN114249625A (zh) * 2021-12-08 2022-03-29 江苏省中国科学院植物研究所 一种过渡金属催化(杂)芳基甲酸与三甲基环三氧硼烷脱羰偶联制备甲基(杂)芳烃的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8067631B2 (en) * 2005-10-21 2011-11-29 Gifu University Method of rapid methylation of alkene compound and kit for PET tracer preparation using the same
JP5279077B2 (ja) * 2006-08-25 2013-09-04 独立行政法人理化学研究所 高速メチル化法、ｐｅｔトレーサー調製用キット、及びｐｅｔ用トレーサーの製造方法

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021199310A1 (fr) * 2020-03-31 2021-10-07 エヌ・イーケムキャット株式会社 Procédé de production d'un composé aromatique

Also Published As

Publication number Publication date
WO2014014067A1 (fr) 2014-01-23

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