JP2014509648A5 - - Google Patents

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Publication number
JP2014509648A5
JP2014509648A5 JP2014502672A JP2014502672A JP2014509648A5 JP 2014509648 A5 JP2014509648 A5 JP 2014509648A5 JP 2014502672 A JP2014502672 A JP 2014502672A JP 2014502672 A JP2014502672 A JP 2014502672A JP 2014509648 A5 JP2014509648 A5 JP 2014509648A5
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JP
Japan
Prior art keywords
alkyl
hydrogen
compound
heterocyclyl
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2014502672A
Other languages
English (en)
Japanese (ja)
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JP2014509648A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2012/030664 external-priority patent/WO2012135175A1/en
Publication of JP2014509648A publication Critical patent/JP2014509648A/ja
Publication of JP2014509648A5 publication Critical patent/JP2014509648A5/ja
Pending legal-status Critical Current

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JP2014502672A 2011-03-28 2012-03-27 (α−置換シクロアルキルアミノ及びヘテロシクリルアミノ)ピリミジニル及び1,3,5−トリアジニルベンズイミダゾール、その医薬組成物、並びに増殖性疾患の治療におけるそれらの使用 Pending JP2014509648A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161468506P 2011-03-28 2011-03-28
US61/468,506 2011-03-28
US201161530839P 2011-09-02 2011-09-02
US61/530,839 2011-09-02
PCT/US2012/030664 WO2012135175A1 (en) 2011-03-28 2012-03-27 (alpha-substituted cycloalkylamino and heterocyclylamino) pyrimidinyl and 1,3,5-triazinyl benzimidazoles, pharmaceutical compositions thereof, and their use in treating proliferative diseases

Publications (2)

Publication Number Publication Date
JP2014509648A JP2014509648A (ja) 2014-04-21
JP2014509648A5 true JP2014509648A5 (US07794700-20100914-C00152.png) 2015-05-14

Family

ID=45929632

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014502672A Pending JP2014509648A (ja) 2011-03-28 2012-03-27 (α−置換シクロアルキルアミノ及びヘテロシクリルアミノ)ピリミジニル及び1,3,5−トリアジニルベンズイミダゾール、その医薬組成物、並びに増殖性疾患の治療におけるそれらの使用

Country Status (8)

Country Link
US (1) US20140088102A1 (US07794700-20100914-C00152.png)
EP (1) EP2691389A1 (US07794700-20100914-C00152.png)
JP (1) JP2014509648A (US07794700-20100914-C00152.png)
AU (1) AU2012236722A1 (US07794700-20100914-C00152.png)
BR (1) BR112013024909A2 (US07794700-20100914-C00152.png)
CA (1) CA2831590A1 (US07794700-20100914-C00152.png)
SG (1) SG193984A1 (US07794700-20100914-C00152.png)
WO (1) WO2012135175A1 (US07794700-20100914-C00152.png)

Families Citing this family (6)

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Publication number Priority date Publication date Assignee Title
WO2012135160A1 (en) 2011-03-28 2012-10-04 Pathway Therapeutics Inc. (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases
BR112014014327A2 (pt) 2011-12-15 2017-06-13 Novartis Ag uso de inibidores da atividade ou função de pi3k
JP6434416B2 (ja) 2012-11-08 2018-12-05 ライゼン・ファーマシューティカルズ・エスアー PDE4阻害剤とPI3δ阻害剤または二重PI3δ−γキナーゼ阻害剤とを含有する薬学的組成物
AU2017326558B2 (en) 2016-09-19 2022-01-06 Mei Pharma, Inc. Combination therapy
CN117860758A (zh) 2017-05-23 2024-04-12 梅制药公司 联合疗法
AU2018318129A1 (en) 2017-08-14 2020-03-26 Mei Pharma, Inc. Combination therapy

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