JP2014501246A5 - - Google Patents

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Publication number
JP2014501246A5
JP2014501246A5 JP2013544634A JP2013544634A JP2014501246A5 JP 2014501246 A5 JP2014501246 A5 JP 2014501246A5 JP 2013544634 A JP2013544634 A JP 2013544634A JP 2013544634 A JP2013544634 A JP 2013544634A JP 2014501246 A5 JP2014501246 A5 JP 2014501246A5
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JP
Japan
Prior art keywords
alkyl
haloalkyl
ring
methyl
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2013544634A
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English (en)
Japanese (ja)
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JP2014501246A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/064324 external-priority patent/WO2012082580A2/en
Publication of JP2014501246A publication Critical patent/JP2014501246A/ja
Publication of JP2014501246A5 publication Critical patent/JP2014501246A5/ja
Pending legal-status Critical Current

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JP2013544634A 2010-12-17 2011-12-12 殺菌・殺カビ性アゾ環式アミド Pending JP2014501246A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201061424228P 2010-12-17 2010-12-17
US61/424,228 2010-12-17
PCT/US2011/064324 WO2012082580A2 (en) 2010-12-17 2011-12-12 Fungicidal azocyclic amides

Publications (2)

Publication Number Publication Date
JP2014501246A JP2014501246A (ja) 2014-01-20
JP2014501246A5 true JP2014501246A5 (enExample) 2015-01-15

Family

ID=45446208

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013544634A Pending JP2014501246A (ja) 2010-12-17 2011-12-12 殺菌・殺カビ性アゾ環式アミド

Country Status (10)

Country Link
US (1) US20130261154A1 (enExample)
EP (1) EP2651219A2 (enExample)
JP (1) JP2014501246A (enExample)
KR (1) KR20140017520A (enExample)
CN (1) CN103384470A (enExample)
AU (1) AU2011344161A1 (enExample)
BR (1) BR112013015166A2 (enExample)
CL (1) CL2013001722A1 (enExample)
MX (1) MX2013006936A (enExample)
WO (1) WO2012082580A2 (enExample)

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NZ612788A (en) 2010-12-17 2015-10-30 Reata Pharmaceuticals Inc Pyrazolyl and pyrimidinyl tricyclic enones as antioxidant inflammation modulators
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BR112013019667B1 (pt) 2011-02-01 2019-07-02 Bayer Intellectual Property Gmbh Compostos derivados de heteroaril-piperidina e -piperazina, seus usos, composição, processos de produção de compostos e de composições, método para o controle de fungos fitopatogênicos prejudiciais
ES2661849T3 (es) 2011-09-15 2018-04-04 Bayer Intellectual Property Gmbh Piperidinpirazoles como fungicidas
ES2647442T3 (es) 2011-12-27 2017-12-21 Bayer Intellectual Property Gmbh Compuestos intermedios para la preparación de derivados de heteroarilpiperidina y de heteroarilpiperazina como fungicidas
PL2809668T3 (pl) 2012-02-02 2018-02-28 Idorsia Pharmaceuticals Ltd Związki 4-(benzimidazol-2-ilo)tiazolowowe i pokrewne aza-pochodne
AU2013277673A1 (en) * 2012-06-22 2015-01-22 E. I. Du Pont De Nemours And Company Fungicidal heterocyclic compounds
EP2801575A1 (en) 2013-05-07 2014-11-12 Bayer CropScience AG Heteroaryldihydropyridine derivatives as fungicides
WO2014206896A1 (en) 2013-06-24 2014-12-31 Bayer Cropscience Ag Piperidinecarboxylic acid derivatives as fungicides
US9198898B2 (en) 2013-06-24 2015-12-01 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
US8906951B1 (en) 2013-06-24 2014-12-09 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
EA030067B1 (ru) 2013-07-22 2018-06-29 Идорсиа Фармасьютиклз Лтд Производные 1-(пиперазин-1-ил)-2-([1,2,4]триазол-1-ил)этанона
WO2015028457A1 (en) * 2013-08-28 2015-03-05 Bayer Cropscience Ag Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
PL3122746T3 (pl) * 2014-03-24 2018-11-30 Bayer Cropscience Aktiengesellschaft Pochodne fenylopiperydynokarboksyamidowe jako fungicydy
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AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
RS58349B1 (sr) 2015-01-15 2019-03-29 Idorsia Pharmaceuticals Ltd Hidroksialkil-piperazinski derivati kao modulatori cxcr3 receptora
WO2017138068A1 (ja) 2016-02-08 2017-08-17 株式会社エス・ディー・エス バイオテック 1,2-ベンゼンジメタノール化合物の製造方法
KR102605762B1 (ko) 2016-02-08 2023-11-27 고완 크롭 프로텍션 리미티드 살균성 조성물
EP3525590B1 (en) * 2016-10-14 2025-08-20 Boehringer Ingelheim Vetmedica GmbH Pesticidal and parasiticidal vinyl isoxazoline compounds
KR20200105652A (ko) 2017-09-08 2020-09-08 피아이 인더스트리스 엘티디. 새로운 살균성 헤테로시클릭 화합물
WO2019048988A1 (en) * 2017-09-08 2019-03-14 Pi Industries Ltd. Novel fungidal heterocyclic compounds
US11066404B2 (en) 2018-10-11 2021-07-20 Incyte Corporation Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors
US11384083B2 (en) 2019-02-15 2022-07-12 Incyte Corporation Substituted spiro[cyclopropane-1,5′-pyrrolo[2,3-d]pyrimidin]-6′(7′h)-ones as CDK2 inhibitors
US11472791B2 (en) 2019-03-05 2022-10-18 Incyte Corporation Pyrazolyl pyrimidinylamine compounds as CDK2 inhibitors
WO2020205560A1 (en) 2019-03-29 2020-10-08 Incyte Corporation Sulfonylamide compounds as cdk2 inhibitors
US11447494B2 (en) 2019-05-01 2022-09-20 Incyte Corporation Tricyclic amine compounds as CDK2 inhibitors
US11440914B2 (en) 2019-05-01 2022-09-13 Incyte Corporation Tricyclic amine compounds as CDK2 inhibitors
MX2022001940A (es) 2019-08-14 2022-05-10 Incyte Corp Compuestos de imidazolil pirimidinilamina como inhibidores de cdk2.
CN119930610A (zh) 2019-10-11 2025-05-06 因赛特公司 作为cdk2抑制剂的双环胺
CN116675704A (zh) * 2020-12-21 2023-09-01 深圳市祥根生物医药有限公司 一种吡咯衍生物及其制备方法和用途
US11981671B2 (en) 2021-06-21 2024-05-14 Incyte Corporation Bicyclic pyrazolyl amines as CDK2 inhibitors
US11976073B2 (en) 2021-12-10 2024-05-07 Incyte Corporation Bicyclic amines as CDK2 inhibitors

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