JP2014501246A5 - - Google Patents

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Publication number
JP2014501246A5
JP2014501246A5 JP2013544634A JP2013544634A JP2014501246A5 JP 2014501246 A5 JP2014501246 A5 JP 2014501246A5 JP 2013544634 A JP2013544634 A JP 2013544634A JP 2013544634 A JP2013544634 A JP 2013544634A JP 2014501246 A5 JP2014501246 A5 JP 2014501246A5
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JP
Japan
Prior art keywords
alkyl
haloalkyl
ring
methyl
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2013544634A
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English (en)
Japanese (ja)
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JP2014501246A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/064324 external-priority patent/WO2012082580A2/en
Publication of JP2014501246A publication Critical patent/JP2014501246A/ja
Publication of JP2014501246A5 publication Critical patent/JP2014501246A5/ja
Pending legal-status Critical Current

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JP2013544634A 2010-12-17 2011-12-12 殺菌・殺カビ性アゾ環式アミド Pending JP2014501246A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201061424228P 2010-12-17 2010-12-17
US61/424,228 2010-12-17
PCT/US2011/064324 WO2012082580A2 (en) 2010-12-17 2011-12-12 Fungicidal azocyclic amides

Publications (2)

Publication Number Publication Date
JP2014501246A JP2014501246A (ja) 2014-01-20
JP2014501246A5 true JP2014501246A5 (enExample) 2015-01-15

Family

ID=45446208

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013544634A Pending JP2014501246A (ja) 2010-12-17 2011-12-12 殺菌・殺カビ性アゾ環式アミド

Country Status (10)

Country Link
US (1) US20130261154A1 (enExample)
EP (1) EP2651219A2 (enExample)
JP (1) JP2014501246A (enExample)
KR (1) KR20140017520A (enExample)
CN (1) CN103384470A (enExample)
AU (1) AU2011344161A1 (enExample)
BR (1) BR112013015166A2 (enExample)
CL (1) CL2013001722A1 (enExample)
MX (1) MX2013006936A (enExample)
WO (1) WO2012082580A2 (enExample)

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BR112013015000A2 (pt) 2010-12-17 2016-08-09 Novartis Ag formas cristalinas de 5-cloron2-(2-isopropóxi-5-metil-4-piperidin-4-il-fenil)-n4-[2-(propano-2-sulfonil)-fenil]-pirimidina-2,4-diamina
CN103596929B (zh) 2010-12-17 2016-10-19 里亚塔医药公司 作为抗氧化发炎调节剂的吡唑及嘧啶三环烯酮
KR101848116B1 (ko) 2011-02-01 2018-04-11 바이엘 인텔렉쳐 프로퍼티 게엠베하 살진균제로서의 헤테로아릴 피페리딘 및 헤테로아릴 피페라진 유도체
ES2661849T3 (es) 2011-09-15 2018-04-04 Bayer Intellectual Property Gmbh Piperidinpirazoles como fungicidas
DK2921493T3 (da) 2011-12-27 2017-11-27 Bayer Ip Gmbh Heteroarylpiperidin og ¿piperazinderivater
AU2013216354B2 (en) 2012-02-02 2017-08-31 Idorsia Pharmaceuticals Ltd 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives
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EP2801575A1 (en) 2013-05-07 2014-11-12 Bayer CropScience AG Heteroaryldihydropyridine derivatives as fungicides
US9198898B2 (en) 2013-06-24 2015-12-01 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
US8906951B1 (en) 2013-06-24 2014-12-09 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
JP6430494B2 (ja) 2013-06-24 2018-11-28 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺真菌剤としてのピペリジンカルボン酸誘導体
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US9924721B2 (en) 2013-08-28 2018-03-27 Bayer Cropscience Aktiengesellschaft Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides
PE20161176A1 (es) * 2014-03-24 2016-11-19 Bayer Cropscience Ag Derivados de fenilpiperidincarboxamida como fungicidas
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
WO2016024350A1 (ja) 2014-08-13 2016-02-18 株式会社エス・ディー・エス バイオテック 縮合11員環化合物及びそれらを含有する農園芸用殺菌剤
AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
PL3245203T3 (pl) 2015-01-15 2019-05-31 Idorsia Pharmaceuticals Ltd Pochodne hydroksyalkilopiperazyny jako modulatory receptora cxcr3
WO2017138069A1 (ja) 2016-02-08 2017-08-17 株式会社エス・ディー・エス バイオテック 殺菌性組成物
JP6407457B2 (ja) 2016-02-08 2018-10-17 株式会社エス・ディー・エス バイオテック 1,2−ベンゼンジメタノール化合物の製造方法
AU2017344097A1 (en) * 2016-10-14 2019-05-02 Boehringer Ingelheim Animal Health USA Inc. Pesticidal and parasiticidal vinyl isoxazoline compounds
US20200281202A1 (en) 2017-09-08 2020-09-10 Pi Industries Ltd. Novel fungicidal heterocyclic compounds
WO2019048988A1 (en) 2017-09-08 2019-03-14 Pi Industries Ltd. Novel fungidal heterocyclic compounds
US11066404B2 (en) 2018-10-11 2021-07-20 Incyte Corporation Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors
US11384083B2 (en) 2019-02-15 2022-07-12 Incyte Corporation Substituted spiro[cyclopropane-1,5′-pyrrolo[2,3-d]pyrimidin]-6′(7′h)-ones as CDK2 inhibitors
TW202100520A (zh) 2019-03-05 2021-01-01 美商英塞特公司 作為cdk2 抑制劑之吡唑基嘧啶基胺化合物
WO2020205560A1 (en) 2019-03-29 2020-10-08 Incyte Corporation Sulfonylamide compounds as cdk2 inhibitors
US11447494B2 (en) 2019-05-01 2022-09-20 Incyte Corporation Tricyclic amine compounds as CDK2 inhibitors
WO2020223469A1 (en) 2019-05-01 2020-11-05 Incyte Corporation N-(1-(methylsulfonyl)piperidin-4-yl)-4,5-di hydro-1h-imidazo[4,5-h]quinazolin-8-amine derivatives and related compounds as cyclin-dependent kinase 2 (cdk2) inhibitors for treating cancer
CA3150681A1 (en) 2019-08-14 2021-02-18 Incyte Corporation Imidazolyl pyrimidinylamine compounds as cdk2 inhibitors
US11851426B2 (en) 2019-10-11 2023-12-26 Incyte Corporation Bicyclic amines as CDK2 inhibitors
CN114644634B (zh) * 2020-12-21 2023-06-20 深圳市祥根生物医药有限公司 一种吡咯衍生物及其制备方法和用途
US11981671B2 (en) 2021-06-21 2024-05-14 Incyte Corporation Bicyclic pyrazolyl amines as CDK2 inhibitors
US11976073B2 (en) 2021-12-10 2024-05-07 Incyte Corporation Bicyclic amines as CDK2 inhibitors

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