JP2014101357A5 - - Google Patents
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- JP2014101357A5 JP2014101357A5 JP2013220736A JP2013220736A JP2014101357A5 JP 2014101357 A5 JP2014101357 A5 JP 2014101357A5 JP 2013220736 A JP2013220736 A JP 2013220736A JP 2013220736 A JP2013220736 A JP 2013220736A JP 2014101357 A5 JP2014101357 A5 JP 2014101357A5
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- JP
- Japan
- Prior art keywords
- substituted
- pharmaceutical composition
- unsubstituted
- composition according
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 239000008194 pharmaceutical composition Substances 0.000 claims 10
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 150000001875 compounds Chemical class 0.000 claims 2
- 230000001629 suppression Effects 0.000 claims 2
- -1 Cyano, carboxy Chemical group 0.000 claims 1
- 208000008589 Obesity Diseases 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 claims 1
- 239000000883 anti-obesity agent Substances 0.000 claims 1
- 229940125710 antiobesity agent Drugs 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 1
- 125000000392 cycloalkenyl group Chemical group 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000004438 haloalkoxy group Chemical group 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 150000002367 halogens Chemical class 0.000 claims 1
- 125000001072 heteroaryl group Chemical group 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 1
- 230000002401 inhibitory effect Effects 0.000 claims 1
- 235000020824 obesity Nutrition 0.000 claims 1
- 125000001424 substituent group Chemical group 0.000 claims 1
- 125000000547 substituted alkyl group Chemical group 0.000 claims 1
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2013220736A JP5590587B2 (ja) | 2012-10-26 | 2013-10-24 | Npyy5受容体拮抗作用を有する医薬組成物 |
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2012236827 | 2012-10-26 | ||
JP2012236827 | 2012-10-26 | ||
JP2013220736A JP5590587B2 (ja) | 2012-10-26 | 2013-10-24 | Npyy5受容体拮抗作用を有する医薬組成物 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2014101357A JP2014101357A (ja) | 2014-06-05 |
JP2014101357A5 true JP2014101357A5 (enrdf_load_stackoverflow) | 2014-08-07 |
JP5590587B2 JP5590587B2 (ja) | 2014-09-17 |
Family
ID=51024205
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2013220736A Active JP5590587B2 (ja) | 2012-10-26 | 2013-10-24 | Npyy5受容体拮抗作用を有する医薬組成物 |
Country Status (1)
Country | Link |
---|---|
JP (1) | JP5590587B2 (enrdf_load_stackoverflow) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112023006710A2 (pt) * | 2020-10-14 | 2023-10-03 | George Mason Res Foundation Inc | Métodos de fabricação de nanopartícula lipídica e composições derivadas da mesma |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0710950A2 (pt) * | 2006-04-28 | 2012-06-26 | Shionogi & Co | derivado de amina tendo atividade antagonìstica de receptor y5 de npi 53 a61p 3/04 a61p 9/04 a61p 9/12 a61p 15/00 a61p 25/08 a61p 25/20 a61p 25/24 a61p 43/00 c07c 311/07 c07c 317/36 c07d 207/325 c07d 211/14 c07d 213/38 c07d 213/74 c07d 213/82 c07d 215/38 c07d 217/04 c07d 217/14 c07d 217/22 c07d 219/10 c07d 231/38 c07d 233/61 c07d 235/30 c07d 237/20 c07d 237/22 c07d 237/34 c07d 239/42 c07d 241/20 c07d 261/14 c07d 261/20 c07d 263/58 c07d 265/30 c07d 265/36 c07d 267/14 c07d 275/02 c07d 277/28 c07d 277/62 c07d 277/82 c07d 295/12 c07d 295/18 c07d 333/36 c07d 333/40 c07d 333/66 c07d 333/72 c07d 403/04 c07d 409/04 c07d 413/04 c07d 417/12 c07d 498/04 c07d 513/04 |
SA08290668B1 (ar) * | 2007-10-25 | 2012-02-12 | شيونوجي آند كو.، ليمتد | مشتقات أمين لها نشاط مضاد لمستقبل npy y5 واستخداماتها |
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2013
- 2013-10-24 JP JP2013220736A patent/JP5590587B2/ja active Active