JP2013532130A5 - - Google Patents
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- JP2013532130A5 JP2013532130A5 JP2013510364A JP2013510364A JP2013532130A5 JP 2013532130 A5 JP2013532130 A5 JP 2013532130A5 JP 2013510364 A JP2013510364 A JP 2013510364A JP 2013510364 A JP2013510364 A JP 2013510364A JP 2013532130 A5 JP2013532130 A5 JP 2013532130A5
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Applications Claiming Priority (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US33499110P | 2010-05-14 | 2010-05-14 | |
US61/334,991 | 2010-05-14 | ||
US37074510P | 2010-08-04 | 2010-08-04 | |
US61/370,745 | 2010-08-04 | ||
US37586310P | 2010-08-22 | 2010-08-22 | |
US61/375,863 | 2010-08-22 | ||
PCT/US2011/036701 WO2011143669A2 (en) | 2010-05-14 | 2011-05-16 | Compositions and methods for treating neoplasia, inflammatory disease and other disorders |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2015049960A Division JP5937247B2 (ja) | 2010-05-14 | 2015-03-12 | 新生物、炎症性疾患、およびその他の障害を治療するための組成物および方法 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2013532130A JP2013532130A (ja) | 2013-08-15 |
JP2013532130A5 true JP2013532130A5 (nl) | 2014-11-06 |
JP5715241B2 JP5715241B2 (ja) | 2015-05-07 |
Family
ID=49052897
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2013510364A Active JP5715241B2 (ja) | 2010-05-14 | 2011-05-16 | 新生物、炎症性疾患、およびその他の障害を治療するための組成物および方法 |
JP2015049960A Active JP5937247B2 (ja) | 2010-05-14 | 2015-03-12 | 新生物、炎症性疾患、およびその他の障害を治療するための組成物および方法 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2015049960A Active JP5937247B2 (ja) | 2010-05-14 | 2015-03-12 | 新生物、炎症性疾患、およびその他の障害を治療するための組成物および方法 |
Country Status (1)
Country | Link |
---|---|
JP (2) | JP5715241B2 (nl) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2011252808B2 (en) | 2010-05-14 | 2015-05-14 | Dana-Farber Cancer Institute, Inc. | Compositions and methods for treating neoplasia, inflammatory disease and other disorders |
EP2569429A4 (en) * | 2010-05-14 | 2013-09-25 | Dana Farber Cancer Inst Inc | COMPOSITIONS AND METHOD OF METABOLIC MODULATION |
MX2014015986A (es) * | 2012-06-25 | 2016-02-11 | Oncoethix Gmbh | Metodo para tratar linfoma utilizando compuestos de tienotriazolodiazepina. |
KR20160037201A (ko) * | 2013-08-06 | 2016-04-05 | 온코에틱스 게엠베하 | Bet-브로모도메인 억제제를 사용한 미만성 거대 b-세포 림프종 (dlbcl)의 치료 방법 |
US11446309B2 (en) | 2013-11-08 | 2022-09-20 | Dana-Farber Cancer Institute, Inc. | Combination therapy for cancer using bromodomain and extra-terminal (BET) protein inhibitors |
RU2722179C2 (ru) | 2014-02-28 | 2020-05-28 | Тэнша Терапеутикс, Инк. | Лечение состояний, ассоциированных с гиперинсулинемией |
JP2018520124A (ja) * | 2015-06-26 | 2018-07-26 | テンシャ セラピューティクス,インコーポレイテッド | Nut正中線癌の治療 |
UA123946C2 (uk) | 2015-09-11 | 2021-06-30 | Дана-Фарбер Кенсер Інстітьют, Інк. | Ацетамідтієнотриазолодіазепіни й шляхи їх застосування |
RU2750164C2 (ru) * | 2015-09-11 | 2021-06-22 | Дана-Фарбер Кэнсер Инститьют, Инк. | Цианотиенотриазолодиазепины и пути их применения |
CN108289957A (zh) * | 2015-10-02 | 2018-07-17 | 达纳-法伯癌症研究所股份有限公司 | 溴区结构域抑制剂和检查点阻断的组合疗法 |
ES2882066T3 (es) * | 2016-02-15 | 2021-12-01 | Univ Michigan Regents | 1,4-oxazepinas fusionadas y análogos relacionados como inhibidores de bromodominio BET |
WO2018109053A1 (en) * | 2016-12-16 | 2018-06-21 | F. Hoffmann-La Roche Ag | Process for the manufacture of diazepine derivatives |
CN109503618A (zh) * | 2017-09-14 | 2019-03-22 | 成都海创药业有限公司 | 一种brd4抑制剂 |
CN112312916A (zh) * | 2018-06-13 | 2021-02-02 | 戴布里股份公司 | 缩合三氮杂卓衍生物的制备及其作为bet抑制剂的用途 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL127516A0 (en) * | 1996-06-12 | 1999-10-28 | Japan Tobacco Inc | A cytokine production inhibitor |
US7589167B2 (en) * | 2000-02-22 | 2009-09-15 | J. David Gladstone Institutes | ZA loops of bromodomains |
MXPA05009151A (es) * | 2003-02-27 | 2005-10-20 | Abbott Lab | Inhibidores de cinasa heterociclica. |
CN101910182B (zh) * | 2007-12-28 | 2013-07-17 | 田边三菱制药株式会社 | 抗癌剂 |
CN102781943B (zh) * | 2009-11-05 | 2016-10-05 | 葛兰素史密丝克莱恩有限责任公司 | 苯并二氮杂*溴结构域抑制剂 |
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2011
- 2011-05-16 JP JP2013510364A patent/JP5715241B2/ja active Active
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2015
- 2015-03-12 JP JP2015049960A patent/JP5937247B2/ja active Active