JP2013520412A5 - - Google Patents

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Publication number
JP2013520412A5
JP2013520412A5 JP2012553848A JP2012553848A JP2013520412A5 JP 2013520412 A5 JP2013520412 A5 JP 2013520412A5 JP 2012553848 A JP2012553848 A JP 2012553848A JP 2012553848 A JP2012553848 A JP 2012553848A JP 2013520412 A5 JP2013520412 A5 JP 2013520412A5
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JP
Japan
Prior art keywords
solid form
schizophrenia
form according
cognitive deficits
xrpd pattern
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2012553848A
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English (en)
Japanese (ja)
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JP5746718B2 (ja
JP2013520412A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/SE2011/050170 external-priority patent/WO2011102793A1/en
Publication of JP2013520412A publication Critical patent/JP2013520412A/ja
Publication of JP2013520412A5 publication Critical patent/JP2013520412A5/ja
Application granted granted Critical
Publication of JP5746718B2 publication Critical patent/JP5746718B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012553848A 2010-02-18 2011-02-17 シクロプロピルアミド誘導体からなる固体形態 Expired - Fee Related JP5746718B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30558110P 2010-02-18 2010-02-18
US61/305,581 2010-02-18
PCT/SE2011/050170 WO2011102793A1 (en) 2010-02-18 2011-02-17 Solid forms comprising a cyclopropyl amide derivative

Publications (3)

Publication Number Publication Date
JP2013520412A JP2013520412A (ja) 2013-06-06
JP2013520412A5 true JP2013520412A5 (https=) 2014-03-20
JP5746718B2 JP5746718B2 (ja) 2015-07-08

Family

ID=44370079

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012553848A Expired - Fee Related JP5746718B2 (ja) 2010-02-18 2011-02-17 シクロプロピルアミド誘導体からなる固体形態

Country Status (17)

Country Link
US (1) US20110201622A1 (https=)
EP (1) EP2536701A4 (https=)
JP (1) JP5746718B2 (https=)
KR (1) KR20130034009A (https=)
CN (1) CN103140481A (https=)
AR (1) AR080203A1 (https=)
AU (1) AU2011218490B9 (https=)
BR (1) BR112012020780A2 (https=)
CA (1) CA2789884A1 (https=)
CL (1) CL2012002285A1 (https=)
IL (1) IL221430A0 (https=)
MX (1) MX2012009537A (https=)
NZ (1) NZ602108A (https=)
RU (1) RU2012136921A (https=)
SG (1) SG183231A1 (https=)
TW (1) TW201136898A (https=)
WO (1) WO2011102793A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SA08290520B1 (ar) 2007-08-22 2012-02-22 استرازينيكا ايه بي مشتقات سيكلو بروبيل أميد وتركيبات صيدلية تحتوي عليها لعلاج حالة مرضية سببها مستقبلات هيستامين h3
TW201039825A (en) * 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
RU2012139082A (ru) * 2010-02-18 2014-03-27 Астразенека Аб Способы получения производных циклопропиламида и связанных с ними промежуточных соединений
CN109438423A (zh) * 2018-09-12 2019-03-08 通化师范学院 一种肺癌靶向化合物azd-3759的合成工艺的新方法

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US5721359A (en) * 1993-03-12 1998-02-24 Pharmacia & Upjohn Company Crystalline ceftiofur free acid
US6383520B1 (en) * 1998-06-26 2002-05-07 Chugai Seiyaku Kabushiki Kaisha Fine powder of L-α-aminoadipic acid derivative, oral solid preparations containing the same, and method for treatment of bulk powders
US6284761B1 (en) * 1999-01-08 2001-09-04 Neurogen Corporation 1-phenyl-4-(1-[2-aryl]cyclopropyl)methylpiperazines: dopamine receptor ligands
WO2001051919A2 (en) * 2000-01-07 2001-07-19 Transform Pharmaceuticals, Inc. High-throughput formation, identification, and analysis of diverse solid-forms
US6521619B2 (en) * 2000-06-29 2003-02-18 Icos Corporation Aryl phenylcyclopropyl sulfide derivatives and their use as cell adhesion inhibiting anti-inflammatory and immune suppressive agents
PL364625A1 (en) * 2001-02-23 2004-12-13 Merck & Co, Inc. N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
US7145002B2 (en) * 2001-09-26 2006-12-05 Merck & Co. Inc. Crystalline forms of carbapenem antibiotics and methods of preparation
US6861432B2 (en) * 2001-11-23 2005-03-01 Schering Aktiengesellschaft Piperazine derivatives that destabilize androgen receptors
JP2005526800A (ja) * 2002-03-22 2005-09-08 エルジー・ライフ・サイエンシーズ・リミテッド (2S)−N−5−[アミノ(イミノ)メチル]−2−チエニルメチル−1−(2R)−2−[(カルボキシルメチル)アミノ]−3,3−ジフェニルプロパノイル−2−ピロリジンカルボキサミド・nH2Oの新しい結晶形
US20040077618A1 (en) * 2002-10-22 2004-04-22 Bennani Youssef L. Cycloalkylamides and their therapeutic applications
US20040209858A1 (en) * 2002-10-22 2004-10-21 Bennani Youssef L. Cycloalkylamides and their therapeutic applications
PL1615909T3 (pl) * 2003-04-23 2009-01-30 Glaxo Group Ltd Pochodne piperazyny i ich zastosowanie w leczeniu chorób neurologicznych i psychicznych
AR045595A1 (es) * 2003-09-04 2005-11-02 Vertex Pharma Composiciones utiles como inhibidores de proteinas quinasas
KR101336106B1 (ko) * 2005-09-16 2013-12-05 얀센 파마슈티카 엔.브이. 히스타민 h3 수용체의 조절제로서 사이클로프로필 아민
AU2007204426A1 (en) * 2006-01-13 2007-07-19 F. Hoffmann-La Roche Ag Cyclohexyl piperazinyl methanone derivatives and their use as histamine H3 receptor modulators
US9108948B2 (en) * 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
CN103382174A (zh) * 2006-06-23 2013-11-06 雅培制药有限公司 作为组胺h3受体调节物的环丙胺衍生物
TW200828371A (en) * 2006-09-21 2008-07-01 Matsushita Electric Industrial Co Ltd Chip-type filter
SA08290520B1 (ar) * 2007-08-22 2012-02-22 استرازينيكا ايه بي مشتقات سيكلو بروبيل أميد وتركيبات صيدلية تحتوي عليها لعلاج حالة مرضية سببها مستقبلات هيستامين h3
MX2010003155A (es) * 2007-10-04 2010-04-01 Hoffmann La Roche Derivados de ciclopropil aril amida y uso de los mismos.
PE20091313A1 (es) * 2008-01-15 2009-09-03 Lilly Co Eli (r)-2-(4-ciclopropansulfonil-fenil)-n-pirazin-2-il-3-(tetrahidropiran-4-il)-propionamida cristalina
TW201039825A (en) * 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
RU2012139082A (ru) * 2010-02-18 2014-03-27 Астразенека Аб Способы получения производных циклопропиламида и связанных с ними промежуточных соединений

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