JP2013503170A5 - - Google Patents

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Publication number
JP2013503170A5
JP2013503170A5 JP2012526933A JP2012526933A JP2013503170A5 JP 2013503170 A5 JP2013503170 A5 JP 2013503170A5 JP 2012526933 A JP2012526933 A JP 2012526933A JP 2012526933 A JP2012526933 A JP 2012526933A JP 2013503170 A5 JP2013503170 A5 JP 2013503170A5
Authority
JP
Japan
Prior art keywords
phenyl
oxy
trifluoromethyl
pyrimidinyl
methylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012526933A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013503170A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2010/046564 external-priority patent/WO2011025798A1/en
Publication of JP2013503170A publication Critical patent/JP2013503170A/ja
Publication of JP2013503170A5 publication Critical patent/JP2013503170A5/ja
Pending legal-status Critical Current

Links

JP2012526933A 2009-08-28 2010-08-25 化合物および方法 Pending JP2013503170A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23781509P 2009-08-28 2009-08-28
US61/237,815 2009-08-28
PCT/US2010/046564 WO2011025798A1 (en) 2009-08-28 2010-08-25 Compounds and methods

Publications (2)

Publication Number Publication Date
JP2013503170A JP2013503170A (ja) 2013-01-31
JP2013503170A5 true JP2013503170A5 (https=) 2013-10-10

Family

ID=43628352

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012526933A Pending JP2013503170A (ja) 2009-08-28 2010-08-25 化合物および方法

Country Status (4)

Country Link
US (1) US20120157482A1 (https=)
EP (1) EP2470022A4 (https=)
JP (1) JP2013503170A (https=)
WO (1) WO2011025798A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11602534B2 (en) 2017-12-21 2023-03-14 Hefei Institutes Of Physical Science, Chinese Academy Of Sciences Pyrimidine derivative kinase inhibitors
CN110698352B (zh) * 2019-10-29 2023-01-17 邢台学院 一种3-溴-5-氨基邻苯二酚二甲醚的合成方法
GB202006382D0 (en) 2020-04-30 2020-06-17 Spermatech As Use
US20250177391A1 (en) * 2022-02-23 2025-06-05 President And Fellows Of Harvard College Inhibitors of ddr1 and ddr2 for the treatment of arthritis

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1213022C (zh) * 1997-12-22 2005-08-03 拜尔有限公司 用对称和不对称的取代二苯脲抑制raf激酶
US7517880B2 (en) * 1997-12-22 2009-04-14 Bayer Pharmaceuticals Corporation Inhibition of p38 kinase using symmetrical and unsymmetrical diphenyl ureas
WO1999032463A1 (en) * 1997-12-22 1999-07-01 Bayer Corporation INHIBITION OF p38 KINASE USING SYMMETRICAL AND UNSYMMETRICAL DIPHENYL UREAS
PE20040522A1 (es) * 2002-05-29 2004-09-28 Novartis Ag Derivados de diarilurea dependientes de la cinasa de proteina
US7459562B2 (en) * 2004-04-23 2008-12-02 Bristol-Myers Squibb Company Monocyclic heterocycles as kinase inhibitors
JP5124812B2 (ja) * 2004-11-24 2013-01-23 国立大学法人 熊本大学 Mapキナーゼtnni3kを用いた心疾患治療剤
GB0500435D0 (en) * 2005-01-10 2005-02-16 Novartis Ag Organic compounds
DE602007010038D1 (de) * 2006-12-22 2010-12-02 Hoffmann La Roche Pyrimidylderivate als proteinkinaseinhibitoren

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