JP2013501031A5 - - Google Patents
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- Publication number
- JP2013501031A5 JP2013501031A5 JP2012523342A JP2012523342A JP2013501031A5 JP 2013501031 A5 JP2013501031 A5 JP 2013501031A5 JP 2012523342 A JP2012523342 A JP 2012523342A JP 2012523342 A JP2012523342 A JP 2012523342A JP 2013501031 A5 JP2013501031 A5 JP 2013501031A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- oxo
- phenoxy
- pyridazin
- trifluoromethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0955504 | 2009-08-05 | ||
| FR0955504A FR2948939B1 (fr) | 2009-08-05 | 2009-08-05 | Derives de 2h pyridazin-3-ones, leur preparation et leur application en therapeutique humaine |
| PCT/EP2010/061426 WO2011015629A1 (en) | 2009-08-05 | 2010-08-05 | Derivatives of 2h pyridazin- 3 -ones, their preparation and their use as scd-1 inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013501031A JP2013501031A (ja) | 2013-01-10 |
| JP2013501031A5 true JP2013501031A5 (https=) | 2013-09-12 |
| JP5901520B2 JP5901520B2 (ja) | 2016-04-13 |
Family
ID=41582079
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012523342A Expired - Fee Related JP5901520B2 (ja) | 2009-08-05 | 2010-08-05 | ２ｈピリダジン−３−オン誘導体、その製造、およびそれらのｓｃｄ−１インヒビターとしての使用 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8946225B2 (https=) |
| EP (1) | EP2462121B1 (https=) |
| JP (1) | JP5901520B2 (https=) |
| AR (1) | AR077715A1 (https=) |
| ES (1) | ES2536841T3 (https=) |
| FR (1) | FR2948939B1 (https=) |
| HU (1) | HUE025513T2 (https=) |
| PL (1) | PL2462121T3 (https=) |
| TW (1) | TW201109313A (https=) |
| WO (1) | WO2011015629A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR086113A1 (es) | 2011-04-30 | 2013-11-20 | Abbott Lab | Isoxazolinas como agentes terapeuticos |
| WO2013056148A2 (en) * | 2011-10-15 | 2013-04-18 | Genentech, Inc. | Methods of using scd1 antagonists |
| WO2013085954A1 (en) | 2011-12-06 | 2013-06-13 | Janssen Pharmaceutica Nv | Substituted piperidinyl-carboxamide derivatives useful as scd 1 inhibitors |
| US9102669B2 (en) | 2011-12-06 | 2015-08-11 | Janssen Pharmaceutica Nv | Substituted piperidinyl-pyridazinyl derivatives useful as SCD 1 inhibitors |
| SG11201802180TA (en) | 2015-09-18 | 2018-04-27 | Univ Miyazaki | Long-acting adrenomedullin derivative |
| US11970486B2 (en) | 2016-10-24 | 2024-04-30 | Janssen Pharmaceutica Nv | Compounds and uses thereof |
| EA201991650A1 (ru) | 2017-01-06 | 2020-01-20 | Юманити Терапьютикс, Инк. | Способы лечения неврологических расстройств |
| CA3083000A1 (en) | 2017-10-24 | 2019-05-02 | Yumanity Therapeutics, Inc. | Compounds and uses thereof |
| BR112020019191A2 (pt) | 2018-03-23 | 2021-01-05 | Yumanity Therapeutics, Inc. | Compostos e seus usos |
| MX2021008903A (es) * | 2019-01-24 | 2021-11-04 | Yumanity Therapeutics Inc | Compuestos y usos de los mismos. |
| EA202192047A1 (ru) * | 2019-11-13 | 2021-12-08 | Юманити Терапьютикс, Инк. | Соединения и их применение |
| CN117164524B (zh) * | 2022-09-06 | 2026-02-03 | 杭州师范大学 | 具有parp7/hdac双靶点抑制活性的哒嗪酮衍生物及其制备方法和应用 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7759348B2 (en) | 2003-07-30 | 2010-07-20 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives and their use as therapeutic agents |
| CN101712653A (zh) * | 2003-07-30 | 2010-05-26 | 泽农医药公司 | 哒嗪衍生物和它们作为治疗剂的用途 |
| AU2005210326B2 (en) * | 2004-02-09 | 2009-10-22 | Nissan Chemical Industries, Ltd. | Drug for inhibiting vascular intimal hyperplasia |
| EP1966183A4 (en) * | 2005-12-20 | 2010-12-29 | Merck Frosst Canada Ltd | HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A-DELTA-9-DESATURASE |
| JP4984701B2 (ja) * | 2006-07-18 | 2012-07-25 | 富士ゼロックス株式会社 | Ｌｅｄプリントヘッドの製造方法 |
| JP4695565B2 (ja) * | 2006-08-21 | 2011-06-08 | 株式会社リコー | 画像形成装置 |
| US20110172230A1 (en) * | 2006-08-23 | 2011-07-14 | Takahiro Ishii | Urea compound or salt thereof |
| WO2008044767A1 (en) * | 2006-10-13 | 2008-04-17 | Takeda Pharmaceutical Company Limited | Aromatic amine derivative and use thereof |
| ATE488499T1 (de) | 2007-08-08 | 2010-12-15 | Graceway Pharmaceuticals Llc | Phenoxypyrrolidinderivat, seine verwendung sowie zusammensetzungen daraus |
-
2009
- 2009-08-05 FR FR0955504A patent/FR2948939B1/fr not_active Expired - Fee Related
-
2010
- 2010-07-28 TW TW099124897A patent/TW201109313A/zh unknown
- 2010-08-05 PL PL10742811T patent/PL2462121T3/pl unknown
- 2010-08-05 AR ARP100102874A patent/AR077715A1/es unknown
- 2010-08-05 US US13/388,884 patent/US8946225B2/en active Active
- 2010-08-05 HU HUE10742811A patent/HUE025513T2/hu unknown
- 2010-08-05 WO PCT/EP2010/061426 patent/WO2011015629A1/en not_active Ceased
- 2010-08-05 ES ES10742811.2T patent/ES2536841T3/es active Active
- 2010-08-05 EP EP10742811.2A patent/EP2462121B1/en active Active
- 2010-08-05 JP JP2012523342A patent/JP5901520B2/ja not_active Expired - Fee Related
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