JP2012180344A5 - - Google Patents
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- JP2012180344A5 JP2012180344A5 JP2012023811A JP2012023811A JP2012180344A5 JP 2012180344 A5 JP2012180344 A5 JP 2012180344A5 JP 2012023811 A JP2012023811 A JP 2012023811A JP 2012023811 A JP2012023811 A JP 2012023811A JP 2012180344 A5 JP2012180344 A5 JP 2012180344A5
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- JP
- Japan
- Prior art keywords
- alkyl
- membered
- haloalkyl
- membered heterocyclyl
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2012023811A JP5620417B2 (ja) | 2011-02-07 | 2012-02-07 | アミノピラゾール誘導体を含む医薬 |
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2011024078 | 2011-02-07 | ||
JP2011024078 | 2011-02-07 | ||
JP2012023811A JP5620417B2 (ja) | 2011-02-07 | 2012-02-07 | アミノピラゾール誘導体を含む医薬 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2012180344A JP2012180344A (ja) | 2012-09-20 |
JP2012180344A5 true JP2012180344A5 (hr) | 2014-10-02 |
JP5620417B2 JP5620417B2 (ja) | 2014-11-05 |
Family
ID=47011846
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2012023811A Active JP5620417B2 (ja) | 2011-02-07 | 2012-02-07 | アミノピラゾール誘導体を含む医薬 |
Country Status (1)
Country | Link |
---|---|
JP (1) | JP5620417B2 (hr) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2902489B9 (en) | 2012-09-27 | 2018-02-07 | Chugai Seiyaku Kabushiki Kaisha | Fgfr3 fusion gene and pharmaceutical drug targeting same |
CN103224479B (zh) * | 2013-04-26 | 2014-10-15 | 温州大学 | 一种2-芳基苯并呋喃类化合物的合成方法 |
KR20160035003A (ko) | 2013-07-31 | 2016-03-30 | 추가이 세이야쿠 가부시키가이샤 | 아미노피라졸 유도체 함유 의약품 제제 |
PE20160546A1 (es) | 2013-10-25 | 2016-05-26 | Novartis Ag | Compuestos derivados de piridilo biciclicos fusionados a anillo como inhibidores de fgfr4 |
MX2016006351A (es) * | 2013-12-13 | 2016-08-01 | Hoffmann La Roche | Inhibidores de tirosina cinasa de bruton. |
RU2648236C2 (ru) | 2013-12-13 | 2018-03-23 | Ф. Хоффманн-Ля Рош Аг | Ингибиторы тирозинкиназы брутона |
US10391081B2 (en) | 2013-12-27 | 2019-08-27 | Chugai Seiyaku Kabushiki Kaisha | FGFR gatekeeper mutant gene and drug targeting same |
CN106459993A (zh) | 2014-03-31 | 2017-02-22 | 德彪药业国际股份公司 | Fgfr融合体 |
ES2756748T3 (es) | 2014-10-03 | 2020-04-27 | Novartis Ag | Uso de derivados de piridilo bicíclicos de anillo fusionado como inhibidores de fgfr4 |
US9802917B2 (en) * | 2015-03-25 | 2017-10-31 | Novartis Ag | Particles of N-(5-cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-7-formyl-6-((4-methyl-2-oxopiperazin-1-yl)methyl)-3,4-dihydro-1,8-naphthyridine-1(2H)-carboxamide |
EP3312172B1 (en) | 2015-06-17 | 2020-05-06 | Chugai Seiyaku Kabushiki Kaisha | Aminopyrazole derivatives useful as src kinase inhibitors |
JP6549311B2 (ja) | 2015-08-20 | 2019-07-24 | 浙江海正薬業股▲ふん▼有限公司Zhejiang Hisun Pharmaceutical CO.,LTD. | インドール誘導体、その調製方法および医薬におけるその使用 |
CN110950848B (zh) * | 2018-09-27 | 2024-03-26 | 徐诺药业 | 新型氨基吡唑类衍生物的合成与应用 |
CN112358435B (zh) * | 2019-10-12 | 2023-01-10 | 中国医学科学院医药生物技术研究所 | 取代芳并杂环类化合物、制备方法和抑制ulk1及抗肿瘤用途 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP3590586B2 (ja) * | 1998-05-05 | 2004-11-17 | エフ.ホフマン−ラ ロシュ アーゲー | P−38mapキナーゼインヒビターとしてのピラゾール誘導体 |
US6316466B1 (en) * | 1998-05-05 | 2001-11-13 | Syntex (U.S.A.) Llc | Pyrazole derivatives P-38 MAP kinase inhibitors |
PT2298743E (pt) * | 2003-06-26 | 2012-12-04 | Novartis Ag | Inibidores de p38 quinase a base de heterociclo de 5 elementos |
AU2009273327A1 (en) * | 2008-07-23 | 2010-01-28 | F. Hoffmann-La Roche Ag | Heterocyclic antiviral compounds |
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2012
- 2012-02-07 JP JP2012023811A patent/JP5620417B2/ja active Active
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