JP2012149082A5 - - Google Patents
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- Publication number
- JP2012149082A5 JP2012149082A5 JP2012075641A JP2012075641A JP2012149082A5 JP 2012149082 A5 JP2012149082 A5 JP 2012149082A5 JP 2012075641 A JP2012075641 A JP 2012075641A JP 2012075641 A JP2012075641 A JP 2012075641A JP 2012149082 A5 JP2012149082 A5 JP 2012149082A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- halogen
- haloalkyl
- formula
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 229910052736 halogen Inorganic materials 0.000 claims 32
- 150000002367 halogens Chemical class 0.000 claims 32
- 125000005843 halogen group Chemical group 0.000 claims 30
- 229910052739 hydrogen Inorganic materials 0.000 claims 27
- 239000001257 hydrogen Substances 0.000 claims 27
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 25
- 150000002431 hydrogen Chemical class 0.000 claims 25
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims 22
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims 15
- 229910052801 chlorine Inorganic materials 0.000 claims 15
- 239000000460 chlorine Substances 0.000 claims 15
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims 14
- 229910052731 fluorine Inorganic materials 0.000 claims 14
- 239000011737 fluorine Substances 0.000 claims 14
- 125000001246 bromo group Chemical group Br* 0.000 claims 12
- 125000004093 cyano group Chemical group *C#N 0.000 claims 10
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 7
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 6
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 6
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims 5
- 125000000623 heterocyclic group Chemical group 0.000 claims 5
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 5
- 244000005700 microbiome Species 0.000 claims 5
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 claims 4
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 3
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 3
- 125000004429 atom Chemical group 0.000 claims 3
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 3
- 125000005347 halocycloalkyl group Chemical group 0.000 claims 3
- 238000000034 method Methods 0.000 claims 3
- 229910052760 oxygen Inorganic materials 0.000 claims 3
- 239000001301 oxygen Substances 0.000 claims 3
- 229910052717 sulfur Inorganic materials 0.000 claims 3
- 239000011593 sulfur Substances 0.000 claims 3
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims 2
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims 2
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 claims 2
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 claims 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 2
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 claims 2
- 239000004606 Fillers/Extenders Substances 0.000 claims 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 2
- 125000000217 alkyl group Chemical group 0.000 claims 2
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 claims 2
- 229910052794 bromium Inorganic materials 0.000 claims 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 2
- 239000003085 diluting agent Substances 0.000 claims 2
- 125000004438 haloalkoxy group Chemical group 0.000 claims 2
- 125000001188 haloalkyl group Chemical group 0.000 claims 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 2
- 229910052757 nitrogen Inorganic materials 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 2
- 125000006413 ring segment Chemical group 0.000 claims 2
- 125000001424 substituent group Chemical group 0.000 claims 2
- 239000004094 surface-active agent Substances 0.000 claims 2
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 claims 1
- 125000004008 6 membered carbocyclic group Chemical group 0.000 claims 1
- ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical compound [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 claims 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 1
- PCPQWYHRMVULIX-UHFFFAOYSA-P [1-[2,3-dihydroxy-4-[4-(oxoazaniumylmethylidene)pyridin-1-yl]butyl]pyridin-4-ylidene]methyl-oxoazanium;dinitrate Chemical compound [O-][N+]([O-])=O.[O-][N+]([O-])=O.C1=CC(=C[NH+]=O)C=CN1CC(O)C(O)CN1C=CC(=C[NH+]=O)C=C1 PCPQWYHRMVULIX-UHFFFAOYSA-P 0.000 claims 1
- 239000002253 acid Substances 0.000 claims 1
- 125000003342 alkenyl group Chemical group 0.000 claims 1
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 claims 1
- 125000003236 benzoyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C(*)=O 0.000 claims 1
- 239000011230 binding agent Substances 0.000 claims 1
- 229910052799 carbon Inorganic materials 0.000 claims 1
- 125000004432 carbon atom Chemical group C* 0.000 claims 1
- 150000001732 carboxylic acid derivatives Chemical class 0.000 claims 1
- 239000003054 catalyst Substances 0.000 claims 1
- 239000003795 chemical substances by application Substances 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000002993 cycloalkylene group Chemical group 0.000 claims 1
- 125000001028 difluoromethyl group Chemical group [H]C(F)(F)* 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 150000004820 halides Chemical class 0.000 claims 1
- 125000004995 haloalkylthio group Chemical group 0.000 claims 1
- 125000001475 halogen functional group Chemical group 0.000 claims 1
- 239000011630 iodine Substances 0.000 claims 1
- 229910052740 iodine Inorganic materials 0.000 claims 1
- 125000000959 isobutyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])* 0.000 claims 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 125000004108 n-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 125000003170 phenylsulfonyl group Chemical group C1(=CC=CC=C1)S(=O)(=O)* 0.000 claims 1
- 229920006395 saturated elastomer Polymers 0.000 claims 1
- 125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 1
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 claims 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 1
- 0 Cc1c(*)[n]c(C)c1N Chemical compound Cc1c(*)[n]c(C)c1N 0.000 description 2
- HSQGRXTXMXMKPQ-UHFFFAOYSA-N Cc1c(C)[s]nn1 Chemical compound Cc1c(C)[s]nn1 HSQGRXTXMXMKPQ-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004059725.1 | 2004-12-11 | ||
| DE102004059725A DE102004059725A1 (de) | 2004-12-11 | 2004-12-11 | 2-Alkyl-cycloalk(en)yl-carboxamide |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007544812A Division JP5004804B2 (ja) | 2004-12-11 | 2005-12-08 | ２−アルキルシクロアルキル（又はアルケニル）カルボキサミド |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2012149082A JP2012149082A (ja) | 2012-08-09 |
| JP2012149082A5 true JP2012149082A5 (https=) | 2013-05-09 |
Family
ID=36390204
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007544812A Expired - Fee Related JP5004804B2 (ja) | 2004-12-11 | 2005-12-08 | ２−アルキルシクロアルキル（又はアルケニル）カルボキサミド |
| JP2012075642A Withdrawn JP2012176950A (ja) | 2004-12-11 | 2012-03-29 | ２−アルキルシクロアルキル（又はアルケニル）カルボキサミド |
| JP2012075641A Withdrawn JP2012149082A (ja) | 2004-12-11 | 2012-03-29 | ２−アルキルシクロアルキル（又はアルケニル）カルボキサミド |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007544812A Expired - Fee Related JP5004804B2 (ja) | 2004-12-11 | 2005-12-08 | ２−アルキルシクロアルキル（又はアルケニル）カルボキサミド |
| JP2012075642A Withdrawn JP2012176950A (ja) | 2004-12-11 | 2012-03-29 | ２−アルキルシクロアルキル（又はアルケニル）カルボキサミド |
Country Status (15)
| Country | Link |
|---|---|
| US (3) | US8344015B2 (https=) |
| EP (4) | EP2216332B1 (https=) |
| JP (3) | JP5004804B2 (https=) |
| KR (1) | KR20070089940A (https=) |
| CN (1) | CN101072761A (https=) |
| AR (1) | AR054412A1 (https=) |
| AT (1) | ATE531259T1 (https=) |
| BR (1) | BRPI0515813A (https=) |
| CA (1) | CA2590220A1 (https=) |
| DE (1) | DE102004059725A1 (https=) |
| PL (2) | PL2215908T3 (https=) |
| RU (1) | RU2419607C9 (https=) |
| TW (1) | TW200637806A (https=) |
| WO (1) | WO2006061215A2 (https=) |
| ZA (1) | ZA200704636B (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102004059725A1 (de) | 2004-12-11 | 2006-06-22 | Bayer Cropscience Ag | 2-Alkyl-cycloalk(en)yl-carboxamide |
| ES2392104T3 (es) * | 2006-06-16 | 2012-12-04 | Syngenta Participations Ag | Derivados de carboxamida etenílica útiles como microbiocidas |
| AR064564A1 (es) * | 2007-01-03 | 2009-04-08 | Bayer Cropscience Ag | Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea. |
| JP2010270035A (ja) * | 2009-05-20 | 2010-12-02 | Sumitomo Chemical Co Ltd | アミド化合物ならびにその植物病害防除用途 |
| CN102858170B (zh) | 2010-04-28 | 2014-12-10 | 住友化学株式会社 | 杀虫组合物及其用途 |
| EP2576517B1 (en) | 2010-06-03 | 2014-12-17 | Bayer Intellectual Property GmbH | N-[(het)arylalkyl)]pyrazole (thio)carboxamides and their heterosubstituted analogues |
| CN103080091A (zh) * | 2010-06-03 | 2013-05-01 | 拜耳知识产权有限责任公司 | O-环丙基环己基-羧酰替苯胺类和它们用作杀真菌剂的用途 |
| WO2012065947A1 (en) | 2010-11-15 | 2012-05-24 | Bayer Cropscience Ag | 5-halogenopyrazolecarboxamides |
| US20130231303A1 (en) | 2010-11-15 | 2013-09-05 | Bayer Intellectual Property Gmbh | 5-halogenopyrazole(thio)carboxamides |
| ES2515042T3 (es) | 2011-01-05 | 2014-10-29 | Syngenta Participations Ag | Derivados de pirazol-4-il-carboxamida como microbiocidas |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3547917A (en) | 1966-12-07 | 1970-12-15 | Uniroyal Inc | 2-amino-4-methylthiazole-5-carboxamides |
| IL103614A (en) | 1991-11-22 | 1998-09-24 | Basf Ag | Carboxamides for controlling botrytis and certain novel such compounds |
| DE4231519A1 (de) * | 1992-09-21 | 1994-03-24 | Basf Ag | Cyclohex(en)ylcarbonsäureamide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| DE4231517A1 (de) * | 1992-09-21 | 1994-03-24 | Basf Ag | Carbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| JP3164762B2 (ja) * | 1995-04-11 | 2001-05-08 | 三井化学株式会社 | 置換チオフェン誘導体およびこれを有効成分とする農園芸用殺菌剤 |
| GB9510459D0 (en) * | 1995-05-24 | 1995-07-19 | Zeneca Ltd | Bicyclic amines |
| DE19629825A1 (de) * | 1996-07-24 | 1998-01-29 | Bayer Ag | Dihydrofuran-carboxamide |
| DE19629826A1 (de) | 1996-07-24 | 1998-01-29 | Bayer Ag | 1,3-Dimethyl-5-fluor-pyrazol-4-carboxamide |
| JP3982886B2 (ja) * | 1996-11-06 | 2007-09-26 | 三井化学株式会社 | 置換チオフェン誘導体およびこれを有効成分とする植物病害防除剤 |
| GB9624611D0 (en) | 1996-11-26 | 1997-01-15 | Zeneca Ltd | Bicyclic amine compounds |
| WO1998025924A1 (en) | 1996-11-26 | 1998-06-18 | Zeneca Limited | 8-azabicyclo[3.2.1]octane-, 8-azabicyclo[3.2.1]oct-6-ene-, 9-azabicyclo[3.3.1]nonane-, 9-aza-3-oxabicyclo[3.3.1]nonane- and 9-aza-3-thiabicyclo[3.3.1]nonane derivatives, their preparation and their use as insecticides |
| BR9813376A (pt) * | 1997-12-04 | 2001-06-19 | Dow Agrosciences Llc | Composição fungicidas e métodos e compostos para a preparação das mesmas |
| AU2931399A (en) * | 1998-03-06 | 1999-09-20 | F. Hoffmann-La Roche Ag | 3-(4-(4-cyanophenyl)thiazol-2-y))-1-(1h-1,2,4-triazol-1-yl) -butan-2-ol derivatives having antifungal activity |
| GB9817548D0 (en) * | 1998-08-12 | 1998-10-07 | Novartis Ag | Organic compounds |
| ES2271109T3 (es) * | 2000-11-08 | 2007-04-16 | Syngenta Participations Ag | Pirrocarboxamidas y pirrolcarbotioamidas y sus usos agroquimicos. |
| DE10136065A1 (de) * | 2001-07-25 | 2003-02-13 | Bayer Cropscience Ag | Pyrazolylcarboxanilide |
| DE10204391A1 (de) | 2002-02-04 | 2003-08-14 | Bayer Cropscience Ag | Difluormethylthiazolylcarboxanilide |
| DE10204390A1 (de) * | 2002-02-04 | 2003-08-14 | Bayer Cropscience Ag | Disubstituierte Thiazolylcarboxanilide |
| GB0207253D0 (en) * | 2002-03-27 | 2002-05-08 | Syngenta Participations Ag | Chemical compounds |
| JP4722829B2 (ja) * | 2003-02-14 | 2011-07-13 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | オキサチンカルボキサミド |
| DE102004041530A1 (de) * | 2004-08-27 | 2006-03-02 | Bayer Cropscience Ag | Biphenylthiazolcarboxamide |
| DE102004059725A1 (de) | 2004-12-11 | 2006-06-22 | Bayer Cropscience Ag | 2-Alkyl-cycloalk(en)yl-carboxamide |
| DE102005025989A1 (de) * | 2005-06-07 | 2007-01-11 | Bayer Cropscience Ag | Carboxamide |
| WO2009016222A1 (en) * | 2007-07-31 | 2009-02-05 | Bayer Cropscience Sa | Fungicide n-5-membered fused heteroaryl-methylene-n-cycloalkyl-carboxamide derivatives |
-
2004
- 2004-12-11 DE DE102004059725A patent/DE102004059725A1/de not_active Withdrawn
-
2005
- 2005-12-08 EP EP10156889.7A patent/EP2216332B1/de not_active Expired - Lifetime
- 2005-12-08 US US11/721,417 patent/US8344015B2/en not_active Expired - Fee Related
- 2005-12-08 WO PCT/EP2005/013140 patent/WO2006061215A2/de not_active Ceased
- 2005-12-08 CA CA002590220A patent/CA2590220A1/en not_active Abandoned
- 2005-12-08 EP EP09005139A patent/EP2098120A3/de not_active Ceased
- 2005-12-08 PL PL10156885T patent/PL2215908T3/pl unknown
- 2005-12-08 AT AT10156885T patent/ATE531259T1/de active
- 2005-12-08 CN CNA2005800421989A patent/CN101072761A/zh active Pending
- 2005-12-08 EP EP05819324A patent/EP1824836A2/de not_active Ceased
- 2005-12-08 RU RU2007125964/04A patent/RU2419607C9/ru not_active IP Right Cessation
- 2005-12-08 BR BRPI0515813-3A patent/BRPI0515813A/pt not_active IP Right Cessation
- 2005-12-08 KR KR1020077013727A patent/KR20070089940A/ko not_active Ceased
- 2005-12-08 JP JP2007544812A patent/JP5004804B2/ja not_active Expired - Fee Related
- 2005-12-08 EP EP10156885A patent/EP2215908B1/de not_active Expired - Lifetime
- 2005-12-08 PL PL10156889T patent/PL2216332T3/pl unknown
- 2005-12-09 TW TW094143525A patent/TW200637806A/zh unknown
- 2005-12-09 AR ARP050105162A patent/AR054412A1/es unknown
-
2007
- 2007-06-08 ZA ZA200704636A patent/ZA200704636B/xx unknown
-
2011
- 2011-06-30 US US13/173,723 patent/US8299047B2/en not_active Expired - Fee Related
-
2012
- 2012-03-29 JP JP2012075642A patent/JP2012176950A/ja not_active Withdrawn
- 2012-03-29 JP JP2012075641A patent/JP2012149082A/ja not_active Withdrawn
- 2012-11-27 US US13/686,557 patent/US8748471B2/en not_active Expired - Fee Related
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