AR064564A1 - Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea. - Google Patents

Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea.

Info

Publication number
AR064564A1
AR064564A1 ARP070105933A AR064564A1 AR 064564 A1 AR064564 A1 AR 064564A1 AR P070105933 A ARP070105933 A AR P070105933A AR 064564 A1 AR064564 A1 AR 064564A1
Authority
AR
Argentina
Prior art keywords
alkyl
sulfanyl
halogen atoms
alkenyl
halogen
Prior art date
Application number
Other languages
English (en)
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of AR064564A1 publication Critical patent/AR064564A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • C07D339/08—Six-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Un procedimiento para preparar este compuesto. Una composicion fungicida que comprende un compuesto de formula general (1). Un método para tratar plantas mediante la aplicacion de un compuesto de formula general (1) o una composicion que lo comprende. Reivindicacion 1: Un compuesto de formula general (1), en la que, R1 es un átomo de hidrogeno, un átomo de halogeno, un alquilo C1-6, un alquenilo C2-6, un alquinilo C2-6, un tri(alquilo C1-8)sililo, un cicloalquilo C3-6, un halogenocicloalquilo C3-6 que tiene 1 a 5 átomos de halogeno; R2 y R3 se seleccionan independientemente uno de otro para que sean un átomo de hidrogeno, un átomo de halogeno, un alquilo C1-6 , un alquenilo C2-6, un alquinilo C2-6, un tri(alquilo C1- 8)sililo, un cicloalquilo C3-6, un halogenocicloalquilo C3-6 que tiene 1 a 5 átomos de halogeno; R4 y R5 se seleccionan independientemente uno de otro para que sean un átomo de hidrogeno, un átomo de halogeno, un alquilo C1-6, un alquenilo C2-6, un alquinilo C2-6, un tri(alquilo C1-8)sililo, un cicloalquilo C3-6 un halogenocicloalquilo C3-6 que tiene 1 a 5 átomos de halogeno; o R2 o R3 pueden formar junto con R4 o R5 un cicloalquilo C3-7; R6 es un átomo de hidrogeno, un alquilo C1-6, o un cicloalquilo C3-7, y Het representa un heterociclo no condensado de 5, 6 o 7 elementos, opcionalmente sustituido con uno, dos o tres heteroátomos que pueden ser iguales o diferentes, estando Het unido por un átomo de C; estando sustituido Het en la porcion orto por un sustituyente seleccionado para que sea un átomo de halogeno, un grupo nitro, ciano, sulfanilo, pentafluoro-gamma6-sulfanilo, alquilo C1-8- halogenoalquilo C1-8 que tiene 1 a 5 átomos de halogeno, alquenilo C2-8, alquinilo C2-8, alcoxi C1-8, halogenoalcoxi C1-8 que tiene 1 a 5 átomos de halogeno, alcoxi C1-8-alquenilo C2-8, un alquil C1-8-sulfanilo, o un halogenoalquil C1-8-sulfanilo que tiene 1 a 5 átomos de halogeno, y opcionalmente sustituidos en cualquier otra posicion por uno o más sustituyentes seleccionados independientemente uno de otro de un átomo de halogeno, un grupo nitro, ciano, sulfanilo, pentafluoro-gamma6-sulfanilo, formilo, formiloxi, formilamino, carboxi, alquilo C1-8, halogenoalquilo C1-8 que tiene 1 a 5 átomos de halogeno, alquenilo C2-8, alquinilo C2-8, alcoxi C1-8, halogenoalcoxi C1-8 que tiene 1 a 5 átomos de halogeno, alcoxi C1-8alquenilo C2-8, alquil C1-8-sulfanilo o un halogenoalquil C1-8-sulfanilo con 1 a 5 átomos de halogeno; así como sus sales, N-oxidos, complejos metálicos, complejos metaloides e isomeros opticamente activos. Reivindicacion 10: Un procedimiento para la preparacion de un compuesto de formula general (1) como se define en la reivindicacion 1, que comprende hacer reaccionar un derivado de la N-alquinilcarboxamida de formula general (2) o una de sus sales: en la que R1, R2, R3, R4, R5 y R6 son como se definio en la reivindicacion 1; con un derivado de ácido carboxílico de formula general (3), en la que: Het es como se definio en la reivindicacion 1; y - L1 es un grupo saliente seleccionado para que sea un átomo de halogeno, un grupo hidroxilo, -ORa, -OCORa, siendo Ra un alquilo C1-6, un haloalquilo C1-6, un bencilo, 4-metoxibencilo, pentafluorofenilo o un grupo de formula (4) en presencia de un catalizador y, si L1 es un grupo hidroxilo, en presencia de un agente de condensacion.
ARP070105933 2007-01-03 2007-12-27 Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea. AR064564A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07100063 2007-01-03

Publications (1)

Publication Number Publication Date
AR064564A1 true AR064564A1 (es) 2009-04-08

Family

ID=37969863

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070105933 AR064564A1 (es) 2007-01-03 2007-12-27 Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea.

Country Status (3)

Country Link
AR (1) AR064564A1 (es)
CL (1) CL2008000005A1 (es)
WO (1) WO2008081017A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011151370A1 (en) * 2010-06-03 2011-12-08 Bayer Cropscience Ag N-[(het)arylalkyl)] pyrazole (thio)carboxamides and their heterosubstituted analogues
WO2012093100A1 (en) * 2011-01-05 2012-07-12 Syngenta Participations Ag Pyrazol-4-yl carboxamide derivatives as microbiocides
WO2020244970A1 (en) * 2019-06-06 2020-12-10 Basf Se New carbocyclic pyridine carboxamides

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4064135A (en) * 1976-07-19 1977-12-20 Syntex (U.S.A.) Inc. Certain thiazole-5-carboxamide compounds
DE4029654A1 (de) * 1990-09-19 1992-04-02 Hoechst Ag 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
DE10136065A1 (de) * 2001-07-25 2003-02-13 Bayer Cropscience Ag Pyrazolylcarboxanilide
JP4398866B2 (ja) * 2002-10-18 2010-01-13 ビーエーエスエフ ソシエタス・ヨーロピア １−フェニルピロリジン−２−オン−３−カルボキサミド
DE102004059725A1 (de) * 2004-12-11 2006-06-22 Bayer Cropscience Ag 2-Alkyl-cycloalk(en)yl-carboxamide
EP1885712B1 (en) * 2005-05-18 2011-02-23 Bayer CropScience AG New 2-pyridinylcycloalkylcarboxamide derivatives as fungicides.

Also Published As

Publication number Publication date
CL2008000005A1 (es) 2008-07-11
WO2008081017A1 (en) 2008-07-10

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